| Aak1 (AAK1) | NAK | Other | 7lvh | A | | n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamide | Mouse | 13820 | |
| Aak1 (AAK1) | NAK | Other | 7lvi | A | A | (2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamide | Mouse | 13822 | |
| Aak1 (AAK1) | NAK | Other | 7lvi | A | B | (2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamide | Mouse | 13821 | |
| Aak1 (AAK1) | NAK | Other | 7rj6 | A | A | 5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Mouse | 14132 | |
| Aak1 (AAK1) | NAK | Other | 7rj6 | A | B | 5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Mouse | 14131 | |
| Aak1 (AAK1) | NAK | Other | 7rj7 | A | A | 2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrile | Mouse | 14128 | |
| Aak1 (AAK1) | NAK | Other | 7rj7 | A | B | 2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrile | Mouse | 14129 | |
| Aak1 (AAK1) | NAK | Other | 7rj8 | A | A | n-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamide | Mouse | 14130 | |
| Aak1 (AAK1) | NAK | Other | 7rj8 | A | B | n-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamide | Mouse | 14127 | |
| AAK1 | NAK | Other | 4wsq | A | A | k-252a | Human | 3834 | |
| AAK1 | NAK | Other | 4wsq | A | B | k-252a | Human | 3836 | |
| AAK1 | NAK | Other | 4wsq | B | A | k-252a | Human | 3833 | |
| AAK1 | NAK | Other | 4wsq | B | B | k-252a | Human | 3835 | |
| AAK1 | NAK | Other | 5l4q | A | A | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6679 | |
| AAK1 | NAK | Other | 5l4q | A | B | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6677 | |
| AAK1 | NAK | Other | 5l4q | B | A | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6680 | |
| AAK1 | NAK | Other | 5l4q | B | B | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6678 | |
| AAK1 | NAK | Other | 5te0 | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 7156 | |
| AAK1 | NAK | Other | 8gmc | A | | 5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 14843 | |
| AAK1 | NAK | Other | 8gmd | A | | (5p)-3-({(8r)-5-[(4-aminopiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-[2-(propan-2-yl)-2h-tetrazol-5-yl]phenol | Human | 14844 | |
| Abl1 (ABL1) | Abl | TK | 1fpu | A | | n-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamide | Mouse | 5728 | |
| Abl1 (ABL1) | Abl | TK | 1fpu | B | | n-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamide | Mouse | 5705 | |
| Abl1 (ABL1) | Abl | TK | 1iep | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5703 | |
| Abl1 (ABL1) | Abl | TK | 1iep | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5727 | |
| Abl1 (ABL1) | Abl | TK | 1m52 | A | | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Mouse | 5720 | |
| Abl1 (ABL1) | Abl | TK | 1m52 | B | | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Mouse | 5715 | |
| Abl1 (ABL1) | Abl | TK | 1opj | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5732 | |
| Abl1 (ABL1) | Abl | TK | 1opj | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5736 | |
| Abl1 (ABL1) | Abl | TK | 1opk | A | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Mouse | 5709 | |
| Abl1 (ABL1) | Abl | TK | 2hzn | A | | 1-[4-(pyridin-4-yloxy)phenyl]-3-[3-(trifluoromethyl)phenyl]urea | Mouse | 5701 | |
| Abl1 (ABL1) | Abl | TK | 2qoh | A | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5707 | |
| Abl1 (ABL1) | Abl | TK | 2qoh | B | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5716 | |
| Abl1 (ABL1) | Abl | TK | 2z60 | A | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5735 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | A | A | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5726 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | A | B | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5729 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | B | A | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5712 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | B | B | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5737 | |
| Abl1 (ABL1) | Abl | TK | 3dk6 | A | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5725 | |
| Abl1 (ABL1) | Abl | TK | 3dk6 | B | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5718 | |
| Abl1 (ABL1) | Abl | TK | 3dk7 | A | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5704 | |
| Abl1 (ABL1) | Abl | TK | 3dk7 | B | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5714 | |
| Abl1 (ABL1) | Abl | TK | 3ik3 | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Mouse | 5731 | |
| Abl1 (ABL1) | Abl | TK | 3ik3 | B | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Mouse | 5739 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5734 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5723 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5710 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5722 | |
| Abl1 (ABL1) | Abl | TK | 3kf4 | A | | n-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amine | Mouse | 5717 | |
| Abl1 (ABL1) | Abl | TK | 3kf4 | B | | n-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amine | Mouse | 5741 | |
| Abl1 (ABL1) | Abl | TK | 3kfa | A | | 3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamide | Mouse | 5742 | |
| Abl1 (ABL1) | Abl | TK | 3kfa | B | | 3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamide | Mouse | 5740 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5733 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5708 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5713 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5706 | |
| Abl1 (ABL1) | Abl | TK | 3mss | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5724 | |
| Abl1 (ABL1) | Abl | TK | 3mss | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5730 | |
| Abl1 (ABL1) | Abl | TK | 3mss | C | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5719 | |
| Abl1 (ABL1) | Abl | TK | 3mss | D | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5702 | |
| Abl1 (ABL1) | Abl | TK | 3oxz | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Mouse | 5721 | |
| Abl1 (ABL1) | Abl | TK | 3oy3 | A | | 5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamide | Mouse | 5711 | |
| Abl1 (ABL1) | Abl | TK | 3oy3 | B | | 5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamide | Mouse | 5738 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10645 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10647 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10648 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10646 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10609 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10608 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10611 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10610 | |
| ABL1 | Abl | TK | 1opl | A | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1104 | |
| ABL1 | Abl | TK | 1opl | B | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1086 | |
| ABL1 | Abl | TK | 2e2b | A | | n-[3-(4,5'-bipyrimidin-2-ylamino)-4-methylphenyl]-4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-3-(trifluoromethyl)benzamide | Human | 1054 | |
| ABL1 | Abl | TK | 2e2b | B | | n-[3-(4,5'-bipyrimidin-2-ylamino)-4-methylphenyl]-4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-3-(trifluoromethyl)benzamide | Human | 1065 | |
| ABL1 | Abl | TK | 2f4j | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 1090 | |
| ABL1 | Abl | TK | 2fo0 | A | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1073 | |
| ABL1 | Abl | TK | 2g1t | A | | - | Human | 1045 | |
| ABL1 | Abl | TK | 2g1t | B | | - | Human | 1105 | |
| ABL1 | Abl | TK | 2g1t | C | | - | Human | 1064 | |
| ABL1 | Abl | TK | 2g1t | D | | - | Human | 1096 | |
| ABL1 | Abl | TK | 2g2f | A | | - | Human | 1097 | |
| ABL1 | Abl | TK | 2g2f | B | | phosphothiophosphoric acid-adenylate ester | Human | 1079 | |
| ABL1 | Abl | TK | 2g2h | A | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1106 | |
| ABL1 | Abl | TK | 2g2h | B | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1089 | |
| ABL1 | Abl | TK | 2g2i | A | | adenosine-5'-diphosphate | Human | 1111 | |
| ABL1 | Abl | TK | 2g2i | B | | adenosine-5'-diphosphate | Human | 1075 | |
| ABL1 | Abl | TK | 2gqg | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1060 | |
| ABL1 | Abl | TK | 2gqg | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1053 | |
| ABL1 | Abl | TK | 2gqg | B | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1084 | |
| ABL1 | Abl | TK | 2gqg | B | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1082 | |
| ABL1 | Abl | TK | 2hiw | A | | 7-amino-1-methyl-3-(2-methyl-5-{[3-(trifluoromethyl)benzoyl]amino}phenyl)-2-oxo-2,3-dihydropyrimido[4,5-d]pyrimidin-1-ium | Human | 1069 | |
| ABL1 | Abl | TK | 2hiw | B | | 7-amino-1-methyl-3-(2-methyl-5-{[3-(trifluoromethyl)benzoyl]amino}phenyl)-2-oxo-2,3-dihydropyrimido[4,5-d]pyrimidin-1-ium | Human | 1110 | |
| ABL1 | Abl | TK | 2hyy | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1092 | |
| ABL1 | Abl | TK | 2hyy | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1078 | |
| ABL1 | Abl | TK | 2hyy | C | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1048 | |
| ABL1 | Abl | TK | 2hyy | D | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1068 | |
| ABL1 | Abl | TK | 2hz0 | A | A | 2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamide | Human | 1052 | |
| ABL1 | Abl | TK | 2hz0 | A | B | 2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamide | Human | 1083 | |
| ABL1 | Abl | TK | 2hz0 | B | A | 2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamide | Human | 1095 | |
| ABL1 | Abl | TK | 2hz0 | B | B | 2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamide | Human | 1109 | |
| ABL1 | Abl | TK | 2hz4 | A | | - | Human | 1059 | |
| ABL1 | Abl | TK | 2hz4 | B | | 1,2,3,4-tetrahydrogen-staurosporine | Human | 1058 | |
| ABL1 | Abl | TK | 2hz4 | C | | - | Human | 1067 | |
| ABL1 | Abl | TK | 2hzi | A | A | 6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1102 | |
| ABL1 | Abl | TK | 2hzi | A | B | 6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1087 | |
| ABL1 | Abl | TK | 2hzi | B | A | 6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1108 | |
| ABL1 | Abl | TK | 2hzi | B | B | 6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1055 | |
| ABL1 | Abl | TK | 2v7a | A | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 1088 | |
| ABL1 | Abl | TK | 2v7a | B | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 1072 | |
| ABL1 | Abl | TK | 3cs9 | A | A | nilotinib | Human | 1080 | |
| ABL1 | Abl | TK | 3cs9 | A | B | nilotinib | Human | 1107 | |
| ABL1 | Abl | TK | 3cs9 | B | A | nilotinib | Human | 1050 | |
| ABL1 | Abl | TK | 3cs9 | B | B | nilotinib | Human | 1112 | |
| ABL1 | Abl | TK | 3cs9 | C | A | nilotinib | Human | 1046 | |
| ABL1 | Abl | TK | 3cs9 | C | B | nilotinib | Human | 1093 | |
| ABL1 | Abl | TK | 3cs9 | D | A | nilotinib | Human | 1077 | |
| ABL1 | Abl | TK | 3cs9 | D | B | nilotinib | Human | 1066 | |
| ABL1 | Abl | TK | 3pyy | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1049 | |
| ABL1 | Abl | TK | 3pyy | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1071 | |
| ABL1 | Abl | TK | 3pyy | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1062 | |
| ABL1 | Abl | TK | 3pyy | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1098 | |
| ABL1 | Abl | TK | 3qri | A | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1051 | |
| ABL1 | Abl | TK | 3qri | A | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1047 | |
| ABL1 | Abl | TK | 3qri | B | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1103 | |
| ABL1 | Abl | TK | 3qri | B | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1076 | |
| ABL1 | Abl | TK | 3qrj | A | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1085 | |
| ABL1 | Abl | TK | 3qrj | A | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1099 | |
| ABL1 | Abl | TK | 3qrj | B | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1101 | |
| ABL1 | Abl | TK | 3qrj | B | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1070 | |
| ABL1 | Abl | TK | 3qrk | A | | (3s)-6-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid | Human | 1056 | |
| ABL1 | Abl | TK | 3ue4 | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 1057 | |
| ABL1 | Abl | TK | 3ue4 | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 1074 | |
| ABL1 | Abl | TK | 4twp | A | | axitinib | Human | 1091 | |
| ABL1 | Abl | TK | 4twp | B | | axitinib | Human | 1081 | |
| ABL1 | Abl | TK | 4wa9 | A | | axitinib | Human | 1061 | |
| ABL1 | Abl | TK | 4wa9 | B | | axitinib | Human | 1063 | |
| ABL1 | Abl | TK | 4xey | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1094 | |
| ABL1 | Abl | TK | 4xey | B | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1100 | |
| ABL1 | Abl | TK | 4yc8 | A | | 2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-n-(4-phenoxyphenyl)-1,3-thiazole-5-carboxamide | Human | 6419 | |
| ABL1 | Abl | TK | 4yc8 | B | | 2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-n-(4-phenoxyphenyl)-1,3-thiazole-5-carboxamide | Human | 6420 | |
| ABL1 | Abl | TK | 4zog | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 7043 | |
| ABL1 | Abl | TK | 4zog | B | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 7042 | |
| ABL1 | Abl | TK | 5hu9 | A | A | 4-[(4-methylpiperazin-1-yl)methyl]-n-(4-methyl-3-{[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]oxy}phenyl)-3-(trifluoromethyl)benzamide | Human | 6754 | |
| ABL1 | Abl | TK | 5hu9 | A | B | 4-[(4-methylpiperazin-1-yl)methyl]-n-(4-methyl-3-{[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]oxy}phenyl)-3-(trifluoromethyl)benzamide | Human | 6755 | |
| ABL1 | Abl | TK | 5mo4 | A | A | nilotinib | Human | 7527 | |
| ABL1 | Abl | TK | 5mo4 | A | B | nilotinib | Human | 7526 | |
| ABL1 | Abl | TK | 6bl8 | A | A | purvalanol b | Human | 9699 | |
| ABL1 | Abl | TK | 6bl8 | A | B | purvalanol b | Human | 9698 | |
| ABL1 | Abl | TK | 6bl8 | B | A | purvalanol b | Human | 9701 | |
| ABL1 | Abl | TK | 6bl8 | B | B | purvalanol b | Human | 9700 | |
| ABL1 | Abl | TK | 6npe | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10946 | |
| ABL1 | Abl | TK | 6npe | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10943 | |
| ABL1 | Abl | TK | 6npe | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10947 | |
| ABL1 | Abl | TK | 6npe | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10945 | |
| ABL1 | Abl | TK | 6npu | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10942 | |
| ABL1 | Abl | TK | 6npu | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10944 | |
| ABL1 | Abl | TK | 6npv | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10948 | |
| ABL1 | Abl | TK | 6npv | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10951 | |
| ABL1 | Abl | TK | 6npv | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10949 | |
| ABL1 | Abl | TK | 6npv | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10950 | |
| ABL1 | Abl | TK | 6xr6 | A | 1 | - | Human | 12905 | |
| ABL1 | Abl | TK | 6xr6 | A | 10 | - | Human | 12901 | |
| ABL1 | Abl | TK | 6xr6 | A | 11 | - | Human | 12872 | |
| ABL1 | Abl | TK | 6xr6 | A | 12 | - | Human | 12871 | |
| ABL1 | Abl | TK | 6xr6 | A | 13 | - | Human | 12869 | |
| ABL1 | Abl | TK | 6xr6 | A | 14 | - | Human | 12873 | |
| ABL1 | Abl | TK | 6xr6 | A | 15 | - | Human | 12862 | |
| ABL1 | Abl | TK | 6xr6 | A | 16 | - | Human | 12902 | |
| ABL1 | Abl | TK | 6xr6 | A | 17 | - | Human | 12874 | |
| ABL1 | Abl | TK | 6xr6 | A | 18 | - | Human | 12912 | |
| ABL1 | Abl | TK | 6xr6 | A | 19 | - | Human | 12892 | |
| ABL1 | Abl | TK | 6xr6 | A | 2 | - | Human | 12878 | |
| ABL1 | Abl | TK | 6xr6 | A | 20 | - | Human | 12861 | |
| ABL1 | Abl | TK | 6xr6 | A | 3 | - | Human | 12908 | |
| ABL1 | Abl | TK | 6xr6 | A | 4 | - | Human | 12898 | |
| ABL1 | Abl | TK | 6xr6 | A | 5 | - | Human | 12858 | |
| ABL1 | Abl | TK | 6xr6 | A | 6 | - | Human | 12896 | |
| ABL1 | Abl | TK | 6xr6 | A | 7 | - | Human | 12881 | |
| ABL1 | Abl | TK | 6xr6 | A | 8 | - | Human | 12906 | |
| ABL1 | Abl | TK | 6xr6 | A | 9 | - | Human | 12885 | |
| ABL1 | Abl | TK | 6xr7 | A | 1 | - | Human | 12867 | |
| ABL1 | Abl | TK | 6xr7 | A | 10 | - | Human | 12903 | |
| ABL1 | Abl | TK | 6xr7 | A | 11 | - | Human | 12866 | |
| ABL1 | Abl | TK | 6xr7 | A | 12 | - | Human | 12860 | |
| ABL1 | Abl | TK | 6xr7 | A | 13 | - | Human | 12910 | |
| ABL1 | Abl | TK | 6xr7 | A | 14 | - | Human | 12865 | |
| ABL1 | Abl | TK | 6xr7 | A | 15 | - | Human | 12913 | |
| ABL1 | Abl | TK | 6xr7 | A | 16 | - | Human | 12859 | |
| ABL1 | Abl | TK | 6xr7 | A | 17 | - | Human | 12870 | |
| ABL1 | Abl | TK | 6xr7 | A | 18 | - | Human | 12909 | |
| ABL1 | Abl | TK | 6xr7 | A | 19 | - | Human | 12879 | |
| ABL1 | Abl | TK | 6xr7 | A | 2 | - | Human | 12883 | |
| ABL1 | Abl | TK | 6xr7 | A | 20 | - | Human | 12914 | |
| ABL1 | Abl | TK | 6xr7 | A | 3 | - | Human | 12900 | |
| ABL1 | Abl | TK | 6xr7 | A | 4 | - | Human | 12894 | |
| ABL1 | Abl | TK | 6xr7 | A | 5 | - | Human | 12857 | |
| ABL1 | Abl | TK | 6xr7 | A | 6 | - | Human | 12897 | |
| ABL1 | Abl | TK | 6xr7 | A | 7 | - | Human | 12907 | |
| ABL1 | Abl | TK | 6xr7 | A | 8 | - | Human | 12863 | |
| ABL1 | Abl | TK | 6xr7 | A | 9 | - | Human | 12915 | |
| ABL1 | Abl | TK | 6xrg | A | 1 | - | Human | 12890 | |
| ABL1 | Abl | TK | 6xrg | A | 10 | - | Human | 12889 | |
| ABL1 | Abl | TK | 6xrg | A | 11 | - | Human | 12877 | |
| ABL1 | Abl | TK | 6xrg | A | 12 | - | Human | 12882 | |
| ABL1 | Abl | TK | 6xrg | A | 13 | - | Human | 12904 | |
| ABL1 | Abl | TK | 6xrg | A | 14 | - | Human | 12875 | |
| ABL1 | Abl | TK | 6xrg | A | 15 | - | Human | 12911 | |
| ABL1 | Abl | TK | 6xrg | A | 16 | - | Human | 12887 | |
| ABL1 | Abl | TK | 6xrg | A | 17 | - | Human | 12916 | |
| ABL1 | Abl | TK | 6xrg | A | 18 | - | Human | 12880 | |
| ABL1 | Abl | TK | 6xrg | A | 19 | - | Human | 12886 | |
| ABL1 | Abl | TK | 6xrg | A | 2 | - | Human | 12895 | |
| ABL1 | Abl | TK | 6xrg | A | 20 | - | Human | 12888 | |
| ABL1 | Abl | TK | 6xrg | A | 3 | - | Human | 12893 | |
| ABL1 | Abl | TK | 6xrg | A | 4 | - | Human | 12899 | |
| ABL1 | Abl | TK | 6xrg | A | 5 | - | Human | 12884 | |
| ABL1 | Abl | TK | 6xrg | A | 6 | - | Human | 12876 | |
| ABL1 | Abl | TK | 6xrg | A | 7 | - | Human | 12868 | |
| ABL1 | Abl | TK | 6xrg | A | 8 | - | Human | 12864 | |
| ABL1 | Abl | TK | 6xrg | A | 9 | - | Human | 12891 | |
| ABL1 | Abl | TK | 7cc2 | A | | [4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methyl-phenyl]boronic acid | Human | 13620 | |
| ABL1 | Abl | TK | 7dt2 | A | | [4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methanoyl-5-methoxy-phenyl]boronic acid | Human | 13621 | |
| ABL1 | Abl | TK | 7n9g | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 14197 | |
| ABL1 | Abl | TK | 7w7x | A | | 5-[5-(dimethylcarbamoyl)pyridin-3-yl]-3-(5-fluorosulfonyloxy-2-methoxy-phenyl)-1h-pyrrolo[2,3-b]pyridine | Human | 14196 | |
| ABL1 | Abl | TK | 7w7y | A | | 5-[3-(5-methanoyl-2-methoxy-4-oxidanyl-phenyl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-~{n},~{n}-dimethyl-pyridine-3-carboxamide | Human | 14195 | |
| ABL1 | Abl | TK | 8h7f | A | | 1-[6-(6-methoxyisoquinolin-7-yl)-1,3-benzothiazol-2-yl]-3-(2-oxidanylideneethyl)urea | Human | 14632 | |
| ABL1 | Abl | TK | 8h7h | A | | 5-[3-(6-methoxyisoquinolin-7-yl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-~{n}-methyl-~{n}-prop-2-ynyl-pyridine-3-carboxamide | Human | 14666 | |
| ABL1 | Abl | TK | 8ssn | A | | 6,7-dimethoxy-n-(4-phenoxyphenyl)quinazolin-4-amine | Human | 14878 | |
| Abl2 (ABL2) | Abl | TK | 4xli | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5689 | |
| Abl2 (ABL2) | Abl | TK | 4xli | B | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5690 | |
| ABL2 | Abl | TK | 2xyn | A | A | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 110 | |
| ABL2 | Abl | TK | 2xyn | A | B | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 112 | |
| ABL2 | Abl | TK | 2xyn | B | A | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 111 | |
| ABL2 | Abl | TK | 2xyn | B | B | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 113 | |
| ABL2 | Abl | TK | 2xyn | C | A | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 116 | |
| ABL2 | Abl | TK | 2xyn | C | B | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 114 | |
| ABL2 | Abl | TK | 3gvu | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 117 | |
| ABL2 | Abl | TK | 3gvu | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 109 | |
| ABL2 | Abl | TK | 3hmi | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 115 | |
| ABL2 | Abl | TK | 3hmi | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 118 | |
| ACVR1 (ALK2) | STKR | TKL | 3h9r | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 1531 | |
| ACVR1 (ALK2) | STKR | TKL | 3mtf | A | A | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 1513 | |
| ACVR1 (ALK2) | STKR | TKL | 3mtf | A | B | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 1521 | |
| ACVR1 (ALK2) | STKR | TKL | 3mtf | B | A | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 1515 | |
| ACVR1 (ALK2) | STKR | TKL | 3mtf | B | B | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 1530 | |
| ACVR1 (ALK2) | STKR | TKL | 3oom | A | A | 1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanone | Human | 1517 | |
| ACVR1 (ALK2) | STKR | TKL | 3oom | A | B | 1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanone | Human | 1518 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | A | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1527 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | A | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1524 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | B | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1510 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | B | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1523 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | C | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1516 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | C | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1533 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | D | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1520 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | D | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1529 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | A | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1528 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | A | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1508 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | B | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1514 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | B | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1526 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | C | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1511 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | C | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1522 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | D | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1519 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | D | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1512 | |
| ACVR1 (ALK2) | STKR | TKL | 4c02 | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 1525 | |
| ACVR1 (ALK2) | STKR | TKL | 4c02 | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 1532 | |
| ACVR1 (ALK2) | STKR | TKL | 4dym | A | | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 1509 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | A | A | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8514 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | A | B | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8518 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | B | A | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8516 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | B | B | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8519 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | C | A | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8517 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | C | B | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8513 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | D | A | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8520 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | D | B | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8515 | |
| ACVR1 (ALK2) | STKR | TKL | 5oy6 | A | | cyclical inhibitor od36 | Human | 8532 | |
| ACVR1 (ALK2) | STKR | TKL | 5oy6 | B | | cyclical inhibitor od36 | Human | 8531 | |
| ACVR1 (ALK2) | STKR | TKL | 5oy6 | C | | cyclical inhibitor od36 | Human | 8529 | |
| ACVR1 (ALK2) | STKR | TKL | 5oy6 | D | | cyclical inhibitor od36 | Human | 8534 | |
| ACVR1 (ALK2) | STKR | TKL | 5s75 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13714 | |
| ACVR1 (ALK2) | STKR | TKL | 5s75 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13718 | |
| ACVR1 (ALK2) | STKR | TKL | 5s76 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13691 | |
| ACVR1 (ALK2) | STKR | TKL | 5s76 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13672 | |
| ACVR1 (ALK2) | STKR | TKL | 5s77 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13694 | |
| ACVR1 (ALK2) | STKR | TKL | 5s77 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13698 | |
| ACVR1 (ALK2) | STKR | TKL | 5s78 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13716 | |
| ACVR1 (ALK2) | STKR | TKL | 5s78 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13686 | |
| ACVR1 (ALK2) | STKR | TKL | 5s79 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13704 | |
| ACVR1 (ALK2) | STKR | TKL | 5s79 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13708 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7a | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13683 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7a | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13644 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7b | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13650 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7b | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13719 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7c | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13689 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7c | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13690 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7c | A | C | - | Human | 13702 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7c | A | D | - | Human | 13680 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7d | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13730 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7d | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13668 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7e | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13715 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7e | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13643 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7f | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13671 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7f | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13737 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7g | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13713 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7g | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13717 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7h | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13682 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7h | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13660 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7i | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13699 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7i | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13663 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7i | A | C | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13653 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7j | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13712 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7j | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13648 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7k | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13649 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7k | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13732 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7l | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13676 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7l | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13736 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7l | A | C | - | Human | 13665 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7m | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13666 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7m | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13739 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7m | A | C | - | Human | 13705 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7n | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13655 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7n | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13659 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7o | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13733 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7o | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13664 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7o | A | C | - | Human | 13647 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7p | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13695 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7p | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13687 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7q | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13670 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7q | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13678 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7r | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13731 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7r | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13654 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7s | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13667 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7s | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13677 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7s | A | C | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13651 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7t | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13723 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7t | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13709 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7u | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13675 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7u | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13696 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7v | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13707 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7v | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13711 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7w | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13700 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7w | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13662 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7x | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13646 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7x | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13692 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7y | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13727 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7y | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13684 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7z | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13652 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7z | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13674 | |
| ACVR1 (ALK2) | STKR | TKL | 5s80 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13728 | |
| ACVR1 (ALK2) | STKR | TKL | 5s80 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13669 | |
| ACVR1 (ALK2) | STKR | TKL | 5s81 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13661 | |
| ACVR1 (ALK2) | STKR | TKL | 5s81 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13697 | |
| ACVR1 (ALK2) | STKR | TKL | 5s82 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13681 | |
| ACVR1 (ALK2) | STKR | TKL | 5s82 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13701 | |
| ACVR1 (ALK2) | STKR | TKL | 5s83 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13706 | |
| ACVR1 (ALK2) | STKR | TKL | 5s83 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13685 | |
| ACVR1 (ALK2) | STKR | TKL | 5s84 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13734 | |
| ACVR1 (ALK2) | STKR | TKL | 5s84 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13656 | |
| ACVR1 (ALK2) | STKR | TKL | 5s84 | A | C | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13722 | |
| ACVR1 (ALK2) | STKR | TKL | 5s85 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13710 | |
| ACVR1 (ALK2) | STKR | TKL | 5s85 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13720 | |
| ACVR1 (ALK2) | STKR | TKL | 5s85 | A | C | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13679 | |
| ACVR1 (ALK2) | STKR | TKL | 5s86 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13724 | |
| ACVR1 (ALK2) | STKR | TKL | 5s86 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13729 | |
| ACVR1 (ALK2) | STKR | TKL | 5s87 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13738 | |
| ACVR1 (ALK2) | STKR | TKL | 5s87 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13735 | |
| ACVR1 (ALK2) | STKR | TKL | 5s88 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13657 | |
| ACVR1 (ALK2) | STKR | TKL | 5s88 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13703 | |
| ACVR1 (ALK2) | STKR | TKL | 5s89 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13673 | |
| ACVR1 (ALK2) | STKR | TKL | 5s89 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13688 | |
| ACVR1 (ALK2) | STKR | TKL | 5s8a | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13725 | |
| ACVR1 (ALK2) | STKR | TKL | 5s8a | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13693 | |
| ACVR1 (ALK2) | STKR | TKL | 5s8b | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13726 | |
| ACVR1 (ALK2) | STKR | TKL | 5s8b | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13721 | |
| ACVR1 (ALK2) | STKR | TKL | 5s9k | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13645 | |
| ACVR1 (ALK2) | STKR | TKL | 5s9k | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13658 | |
| ACVR1 (ALK2) | STKR | TKL | 6acr | A | | n-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amine | Human | 10969 | |
| ACVR1 (ALK2) | STKR | TKL | 6acr | B | | n-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amine | Human | 10968 | |
| ACVR1 (ALK2) | STKR | TKL | 6eix | A | A | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 8530 | |
| ACVR1 (ALK2) | STKR | TKL | 6eix | A | B | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 8533 | |
| ACVR1 (ALK2) | STKR | TKL | 6gi6 | A | | 5-methyl-6-quinolin-5-yl-3~{h}-quinazolin-4-one | Human | 9919 | |
| ACVR1 (ALK2) | STKR | TKL | 6gin | A | A | 3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-one | Human | 9914 | |
| ACVR1 (ALK2) | STKR | TKL | 6gin | A | B | 3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-one | Human | 9918 | |
| ACVR1 (ALK2) | STKR | TKL | 6gin | B | A | 3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-one | Human | 9920 | |
| ACVR1 (ALK2) | STKR | TKL | 6gin | B | B | 3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-one | Human | 9916 | |
| ACVR1 (ALK2) | STKR | TKL | 6gip | A | A | 2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-one | Human | 9915 | |
| ACVR1 (ALK2) | STKR | TKL | 6gip | A | B | 2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-one | Human | 9917 | |
| ACVR1 (ALK2) | STKR | TKL | 6i1s | A | A | (4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione | Human | 11603 | |
| ACVR1 (ALK2) | STKR | TKL | 6i1s | A | B | (4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione | Human | 11604 | |
| ACVR1 (ALK2) | STKR | TKL | 6jux | A | A | 4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amine | Human | 12161 | |
| ACVR1 (ALK2) | STKR | TKL | 6jux | A | B | 4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amine | Human | 12160 | |
| ACVR1 (ALK2) | STKR | TKL | 6srh | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 11632 | |
| ACVR1 (ALK2) | STKR | TKL | 6srh | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 11630 | |
| ACVR1 (ALK2) | STKR | TKL | 6srh | B | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 11631 | |
| ACVR1 (ALK2) | STKR | TKL | 6srh | B | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 11633 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | A | A | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11735 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | A | B | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11737 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | B | A | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11734 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | B | B | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11736 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | A | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11779 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | A | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11784 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | B | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11781 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | B | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11782 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | C | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11778 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | C | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11780 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | D | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11783 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | D | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11785 | |
| ACVR1 (ALK2) | STKR | TKL | 6t8n | A | A | cyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanone | Human | 11831 | |
| ACVR1 (ALK2) | STKR | TKL | 6t8n | A | B | cyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanone | Human | 11830 | |
| ACVR1 (ALK2) | STKR | TKL | 6t8n | B | A | cyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanone | Human | 11828 | |
| ACVR1 (ALK2) | STKR | TKL | 6t8n | B | B | cyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanone | Human | 11829 | |
| ACVR1 (ALK2) | STKR | TKL | 6tn8 | A | A | 4-[4-[(dimethylamino)methyl]-2,5-dimethoxy-phenyl]-2-methyl-2,7-naphthyridin-1-one | Human | 11888 | |
| ACVR1 (ALK2) | STKR | TKL | 6tn8 | A | B | 4-[4-[(dimethylamino)methyl]-2,5-dimethoxy-phenyl]-2-methyl-2,7-naphthyridin-1-one | Human | 11887 | |
| ACVR1 (ALK2) | STKR | TKL | 6unq | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 13783 | |
| ACVR1 (ALK2) | STKR | TKL | 6unq | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 13784 | |
| ACVR1 (ALK2) | STKR | TKL | 6unr | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13785 | |
| ACVR1 (ALK2) | STKR | TKL | 6uns | A | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 13782 | |
| ACVR1 (ALK2) | STKR | TKL | 6uns | A | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 13781 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | A | A | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12277 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | A | B | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12278 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | B | A | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12276 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | B | B | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12275 | |
| ACVR1 (ALK2) | STKR | TKL | 6zgc | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 12638 | |
| ACVR1 (ALK2) | STKR | TKL | 6zgc | B | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 12641 | |
| ACVR1 (ALK2) | STKR | TKL | 6zgc | C | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 12640 | |
| ACVR1 (ALK2) | STKR | TKL | 6zgc | D | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 12639 | |
| ACVR1 (ALK2) | STKR | TKL | 7a21 | A | A | 4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12777 | |
| ACVR1 (ALK2) | STKR | TKL | 7a21 | A | B | 4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12779 | |
| ACVR1 (ALK2) | STKR | TKL | 7a21 | B | A | 4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12776 | |
| ACVR1 (ALK2) | STKR | TKL | 7a21 | B | B | 4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12778 | |
| ACVR1 (ALK2) | STKR | TKL | 7c3g | A | A | ~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amine | Human | 13389 | |
| ACVR1 (ALK2) | STKR | TKL | 7c3g | A | B | ~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amine | Human | 13390 | |
| ACVR1 (ALK2) | STKR | TKL | 7c3g | B | A | ~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amine | Human | 13392 | |
| ACVR1 (ALK2) | STKR | TKL | 7c3g | B | B | ~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amine | Human | 13391 | |
| ACVR1 (ALK2) | STKR | TKL | 7nns | B | A | momelotinib | Human | 13465 | |
| ACVR1 (ALK2) | STKR | TKL | 7nns | B | B | momelotinib | Human | 13464 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7w | A | A | 6-methyl-9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,7-dihydropyrido[4,3-d][2]benzazepine | Human | 14608 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7w | A | B | 6-methyl-9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,7-dihydropyrido[4,3-d][2]benzazepine | Human | 14609 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7z | A | A | 9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1]benzoxepino[5,4-c]pyridine | Human | 14605 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7z | A | B | 9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1]benzoxepino[5,4-c]pyridine | Human | 14604 | |
| ACVR1 (ALK2) | STKR | TKL | 8pod | A | | 6-(4-piperazin-1-ylphenyl)-3-quinolin-4-yl-furo[3,2-b]pyridine | Human | 15314 | |
| ACVR1 (ALK2) | STKR | TKL | 8r7g | A | A | 2-fluoranyl-6-methoxy-4-[4-methyl-5-[4-(4-propan-2-ylpiperazin-1-yl)phenyl]pyridin-3-yl]benzamide | Human | 15267 | |
| ACVR1 (ALK2) | STKR | TKL | 8r7g | A | B | 2-fluoranyl-6-methoxy-4-[4-methyl-5-[4-(4-propan-2-ylpiperazin-1-yl)phenyl]pyridin-3-yl]benzamide | Human | 15266 | |
| ACVR2A (ACTR2) | STKR | TKL | 3q4t | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 2682 | |
| ACVR2A (ACTR2) | STKR | TKL | 3q4t | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 2686 | |
| ACVR2A (ACTR2) | STKR | TKL | 3q4t | B | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 2680 | |
| ACVR2A (ACTR2) | STKR | TKL | 3q4t | B | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 2684 | |
| ACVR2A (ACTR2) | STKR | TKL | 3soc | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2675 | |
| ACVR2A (ACTR2) | STKR | TKL | 3soc | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2676 | |
| ACVR2A (ACTR2) | STKR | TKL | 3soc | B | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2677 | |
| ACVR2A (ACTR2) | STKR | TKL | 3soc | B | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2685 | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | A | A | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | 2678 | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | A | B | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | 2681 | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | B | A | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | 2683 | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | B | B | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | 2679 | |
| ACVR2B (ACTR2B) | STKR | TKL | 2qlu | A | | adenine | Human | 2940 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | A | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1266 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | B | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1273 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | C | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1269 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | D | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1258 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | E | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1263 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | F | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1276 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | G | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1272 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | H | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1260 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | I | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1261 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | J | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1277 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | K | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1267 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | L | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1265 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | M | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1268 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | N | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1257 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | O | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1262 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | P | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1270 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | Q | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1274 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | R | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1256 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | S | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1259 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | T | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1264 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | U | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1278 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | V | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1271 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | W | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1255 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | X | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1275 | |
| AKT1 | Akt | AGC | 3cqu | A | A | n-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6764 | |
| AKT1 | Akt | AGC | 3cqu | A | B | n-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6762 | |
| AKT1 | Akt | AGC | 3cqw | A | A | 5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine | Human | 6763 | |
| AKT1 | Akt | AGC | 3cqw | A | B | 5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine | Human | 6765 | |
| AKT1 | Akt | AGC | 3mv5 | A | A | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 2537 | |
| AKT1 | Akt | AGC | 3mv5 | A | B | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 2532 | |
| AKT1 | Akt | AGC | 3mvh | A | A | n-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamide | Human | 2538 | |
| AKT1 | Akt | AGC | 3mvh | A | B | n-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamide | Human | 2531 | |
| AKT1 | Akt | AGC | 3o96 | A | | - | Human | 2545 | |
| AKT1 | Akt | AGC | 3ocb | A | | (2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amine | Human | 2548 | |
| AKT1 | Akt | AGC | 3ocb | B | | (2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amine | Human | 2534 | |
| AKT1 | Akt | AGC | 3ow4 | A | | (2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amine | Human | 2547 | |
| AKT1 | Akt | AGC | 3ow4 | B | | (2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amine | Human | 2533 | |
| AKT1 | Akt | AGC | 3qkk | A | | n-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(2r)-6-hydroxy-4-oxo-3,4-dihydro-1'h-spiro[chromene-2,3'-piperidin]-1'-yl]propyl}-2,6-dimethylbenzenesulfonamide | Human | 2535 | |
| AKT1 | Akt | AGC | 3qkl | A | | n-{(2s)-3-[(3s)-8',9'-dihydro-1h,3'h-spiro[piperidine-3,7'-pyrano[3,2-e]indazol]-1-yl]-2-hydroxypropyl}-n-(2-ethoxyethyl)-2,6-dimethylbenzenesulfonamide | Human | 2544 | |
| AKT1 | Akt | AGC | 3qkm | A | | n-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(5r)-2-(quinazolin-4-yl)-2,7-diazaspiro[4.5]dec-7-yl]propyl}-2,6-dimethylbenzenesulfonamide | Human | 2546 | |
| AKT1 | Akt | AGC | 4ejn | A | | - | Human | 2542 | |
| AKT1 | Akt | AGC | 4ekk | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2541 | |
| AKT1 | Akt | AGC | 4ekk | B | | phosphoaminophosphonic acid-adenylate ester | Human | 2539 | |
| AKT1 | Akt | AGC | 4ekl | A | | (2s)-2-(4-chlorophenyl)-1-{4-[(5r,7r)-7-hydroxy-5-methyl-6,7-dihydro-5h-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl}-3-(propan-2-ylamino)propan-1-one | Human | 2540 | |
| AKT1 | Akt | AGC | 4gv1 | A | A | 4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | 2543 | |
| AKT1 | Akt | AGC | 4gv1 | A | B | 4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | 2536 | |
| AKT1 | Akt | AGC | 5kcv | A | | 3-[3-[4-(1-azanylcyclobutyl)phenyl]-5-phenyl-imidazo[4,5-b]pyridin-2-yl]pyridin-2-amine | Human | 6708 | |
| AKT1 | Akt | AGC | 6buu | A | A | - | Human | 10432 | |
| AKT1 | Akt | AGC | 6buu | A | B | - | Human | 10433 | |
| AKT1 | Akt | AGC | 6buu | A | C | - | Human | 10438 | |
| AKT1 | Akt | AGC | 6buu | B | A | - | Human | 10430 | |
| AKT1 | Akt | AGC | 6buu | B | B | - | Human | 10439 | |
| AKT1 | Akt | AGC | 6buu | B | C | - | Human | 10428 | |
| AKT1 | Akt | AGC | 6ccy | A | A | (5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-one | Human | 9868 | |
| AKT1 | Akt | AGC | 6ccy | A | B | (5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-one | Human | 9869 | |
| AKT1 | Akt | AGC | 6hhf | A | | borussertib | Human | 10970 | |
| AKT1 | Akt | AGC | 6hhg | A | | ~{n}-[2-chloranyl-5-[[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]carbamoylamino]phenyl]propanamide | Human | 10916 | |
| AKT1 | Akt | AGC | 6hhh | A | | ~{n}-[4-[4-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperazin-1-yl]phenyl]propanamide | Human | 10915 | |
| AKT1 | Akt | AGC | 6hhi | A | | ~{n}-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]-3-(propanoylamino)benzamide | Human | 10913 | |
| AKT1 | Akt | AGC | 6hhj | A | | ~{n}-[1-methyl-2-oxidanylidene-3-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]benzimidazol-5-yl]propanamide | Human | 10914 | |
| AKT1 | Akt | AGC | 6npz | A | A | - | Human | 10880 | |
| AKT1 | Akt | AGC | 6npz | A | B | - | Human | 10882 | |
| AKT1 | Akt | AGC | 6npz | B | A | - | Human | 10881 | |
| AKT1 | Akt | AGC | 6npz | B | B | - | Human | 10879 | |
| AKT1 | Akt | AGC | 6s9w | A | A | ~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 11748 | |
| AKT1 | Akt | AGC | 6s9w | A | B | ~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 11747 | |
| AKT1 | Akt | AGC | 6s9x | A | | ~{n}-[3-[1-[[4-[5-[(4-hydroxyphenyl)methyl]-6-oxidanylidene-2-phenyl-1~{h}-pyrazin-3-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 11746 | |
| AKT1 | Akt | AGC | 7apj | A | | - | Human | 13854 | |
| AKT1 | Akt | AGC | 7nh4 | A | A | ~{n}-[3-[1-[[4-[5-(hydroxymethyl)-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 13865 | |
| AKT1 | Akt | AGC | 7nh4 | A | B | ~{n}-[3-[1-[[4-[5-(hydroxymethyl)-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 13866 | |
| AKT1 | Akt | AGC | 7nh5 | A | A | ~{n}-methyl-6-[4-[[4-[2-oxidanylidene-6-(propanoylamino)-3~{h}-benzimidazol-1-yl]piperidin-1-yl]methyl]phenyl]-5-phenyl-pyridine-3-carboxamide | Human | 13867 | |
| AKT1 | Akt | AGC | 7nh5 | A | B | ~{n}-methyl-6-[4-[[4-[2-oxidanylidene-6-(propanoylamino)-3~{h}-benzimidazol-1-yl]piperidin-1-yl]methyl]phenyl]-5-phenyl-pyridine-3-carboxamide | Human | 13868 | |
| AKT1 | Akt | AGC | 8uvy | A | A | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15378 | |
| AKT1 | Akt | AGC | 8uvy | A | B | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15381 | |
| AKT1 | Akt | AGC | 8uw2 | A | A | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15379 | |
| AKT1 | Akt | AGC | 8uw2 | A | B | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15380 | |
| AKT1 | Akt | AGC | 8uw7 | A | A | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15385 | |
| AKT1 | Akt | AGC | 8uw7 | A | B | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15382 | |
| AKT1 | Akt | AGC | 8uw9 | A | A | n-({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)-2-(2-fluoro-4-formyl-3-hydroxyphenyl)acetamide | Human | 15383 | |
| AKT1 | Akt | AGC | 8uw9 | A | B | n-({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)-2-(2-fluoro-4-formyl-3-hydroxyphenyl)acetamide | Human | 15384 | |
| AKT2 | Akt | AGC | 1gzk | A | | - | Human | 1916 | |
| AKT2 | Akt | AGC | 1gzn | A | | - | Human | 1915 | |
| AKT2 | Akt | AGC | 1gzo | A | | - | Human | 1914 | |
| AKT2 | Akt | AGC | 1mrv | A | | - | Human | 1917 | |
| AKT2 | Akt | AGC | 1mry | A | | - | Human | 1907 | |
| AKT2 | Akt | AGC | 1o6k | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1923 | |
| AKT2 | Akt | AGC | 1o6l | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1906 | |
| AKT2 | Akt | AGC | 2jdo | A | | isoquinoline-5-sulfonic acid (2-(2-(4-chlorobenzyloxy)ethylamino)ethyl)amide | Human | 1922 | |
| AKT2 | Akt | AGC | 2jdr | A | | (2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amine | Human | 1918 | |
| AKT2 | Akt | AGC | 2uw9 | A | | 4-(4-chlorophenyl)-4-[4-(1h-pyrazol-4-yl)phenyl]piperidine | Human | 1919 | |
| AKT2 | Akt | AGC | 2x39 | A | | 4-amino-n-(4-chlorobenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | 1913 | |
| AKT2 | Akt | AGC | 2xh5 | A | | 4-(4-tert-butylbenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-aminium | Human | 1924 | |
| AKT2 | Akt | AGC | 3d0e | A | | 4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-ol | Human | 1912 | |
| AKT2 | Akt | AGC | 3d0e | B | | 4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-ol | Human | 1920 | |
| AKT2 | Akt | AGC | 3e87 | A | A | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | 1910 | |
| AKT2 | Akt | AGC | 3e87 | A | B | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | 1911 | |
| AKT2 | Akt | AGC | 3e87 | B | A | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | 1909 | |
| AKT2 | Akt | AGC | 3e87 | B | B | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | 1903 | |
| AKT2 | Akt | AGC | 3e88 | A | | 4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1908 | |
| AKT2 | Akt | AGC | 3e88 | B | | 4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1905 | |
| AKT2 | Akt | AGC | 3e8d | A | A | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1921 | |
| AKT2 | Akt | AGC | 3e8d | A | B | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1926 | |
| AKT2 | Akt | AGC | 3e8d | B | A | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1925 | |
| AKT2 | Akt | AGC | 3e8d | B | B | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1904 | |
| AKT2 | Akt | AGC | 8q61 | A | A | 6-[4-(1-azanyl-3-methyl-3-oxidanyl-cyclobutyl)phenyl]-7-phenyl-1-propyl-pyrido[2,3-b][1,4]oxazin-2-one | Human | 14978 | |
| AKT2 | Akt | AGC | 8q61 | A | B | 6-[4-(1-azanyl-3-methyl-3-oxidanyl-cyclobutyl)phenyl]-7-phenyl-1-propyl-pyrido[2,3-b][1,4]oxazin-2-one | Human | 14979 | |
| AKT2 | Akt | AGC | 9c1w | A | | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15393 | |
| ALK | ALK | TK | 2xb7 | A | | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 5365 | |
| ALK | ALK | TK | 2xba | A | | 5-[(2r)-2-hydroxy-2-phenylacetyl]-3-({[4-(4-methylpiperazin-1-yl)phenyl]carbonyl}amino)-1,6-dihydropyrrolo[3,4-c]pyrazol-5-ium | Human | 5408 | |
| ALK | ALK | TK | 2xp2 | A | | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 5394 | |
| ALK | ALK | TK | 2yfx | A | | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 5402 | |
| ALK | ALK | TK | 2yhv | A | | - | Human | 5384 | |
| ALK | ALK | TK | 2yjr | A | A | - | Human | 5399 | |
| ALK | ALK | TK | 2yjr | A | B | - | Human | 5380 | |
| ALK | ALK | TK | 2yjs | A | | - | Human | 5373 | |
| ALK | ALK | TK | 3aox | A | A | 9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrile | Human | 5387 | |
| ALK | ALK | TK | 3aox | A | B | 9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrile | Human | 5370 | |
| ALK | ALK | TK | 3l9p | A | A | - | Human | 5363 | |
| ALK | ALK | TK | 3l9p | A | B | - | Human | 5375 | |
| ALK | ALK | TK | 3lcs | A | A | staurosporine | Human | 5381 | |
| ALK | ALK | TK | 3lcs | A | B | staurosporine | Human | 5376 | |
| ALK | ALK | TK | 3lct | A | A | adenosine-5'-diphosphate | Human | 5393 | |
| ALK | ALK | TK | 3lct | A | B | adenosine-5'-diphosphate | Human | 5400 | |
| ALK | ALK | TK | 4anl | A | | - | Human | 5385 | |
| ALK | ALK | TK | 4anq | A | | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 5368 | |
| ALK | ALK | TK | 4ans | A | | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 5374 | |
| ALK | ALK | TK | 4ccb | A | | 3-[(1r)-1-[5-fluoranyl-2-(1,2,3-triazol-2-yl)phenyl]ethoxy]-5-(3-methyl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 5390 | |
| ALK | ALK | TK | 4ccu | A | | 2-(5-(6-amino-5-((r)-1-(5-fluoro-2-(2h-1,2,3-triazol-2-yl)phenyl)ethoxy)pyridin-3-yl)-4-methylthiazol-2-yl)propan-2-ol | Human | 5396 | |
| ALK | ALK | TK | 4cd0 | A | | (2r)-2-[5-(6-amino-5-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diol | Human | 5407 | |
| ALK | ALK | TK | 4cli | A | | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | 5405 | |
| ALK | ALK | TK | 4clj | A | | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | 5369 | |
| ALK | ALK | TK | 4cmo | A | | 2-[(1r)-1-{[3-amino-6-(2-methoxypyridin-3-yl)pyrazin-2-yl]oxy}ethyl]-4-fluoro-n-methylbenzamide | Human | 5391 | |
| ALK | ALK | TK | 4cmt | A | | 3-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}-5-[3-(methylsulfonyl)phenyl]pyridin-2-amine | Human | 5371 | |
| ALK | ALK | TK | 4cmu | A | | (10r)-7-amino-12-fluoro-1,3,10,16-tetramethyl-16,17-dihydro-1h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 5398 | |
| ALK | ALK | TK | 4cnh | A | | 3-[(1r)-1-(5-fluoro-2-methoxyphenyl)ethoxy]-5-(1-methyl-1h-1,2,3-triazol-5-yl)pyridin-2-amine | Human | 5388 | |
| ALK | ALK | TK | 4cnh | B | | 3-[(1r)-1-(5-fluoro-2-methoxyphenyl)ethoxy]-5-(1-methyl-1h-1,2,3-triazol-5-yl)pyridin-2-amine | Human | 5378 | |
| ALK | ALK | TK | 4ctb | A | | (5r)-8-amino-3-fluoro-5,19-dimethyl-20-oxo-5,18,19,20-tetrahydro-11,7-(azeno)pyrido[2',1':2,3]imidazo[4,5-h][2,5,11]benzoxadiazacyclotetradecine-14-carbonitrile | Human | 5395 | |
| ALK | ALK | TK | 4ctc | A | | (10r)-7-amino-3-cyclopropyl-12-fluoro-1,10,16-trimethyl-16,17-dihydro-1h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 5364 | |
| ALK | ALK | TK | 4dce | A | | (3s)-n-(4-methylbenzyl)-1-{2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}piperidine-3-carboxamide | Human | 5379 | |
| ALK | ALK | TK | 4dce | B | | (3s)-n-(4-methylbenzyl)-1-{2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}piperidine-3-carboxamide | Human | 5372 | |
| ALK | ALK | TK | 4fnw | A | | - | Human | 5403 | |
| ALK | ALK | TK | 4fnx | A | | - | Human | 5366 | |
| ALK | ALK | TK | 4fny | A | | n-(4-chlorophenyl)-5-[(6,7-dimethoxyquinolin-4-yl)oxy]-1,3-benzoxazol-2-amine | Human | 5367 | |
| ALK | ALK | TK | 4fnz | A | | (3s)-n-[3-(trifluoromethoxy)benzyl]-1-{2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}piperidine-3-carboxamide | Human | 5397 | |
| ALK | ALK | TK | 4fob | A | | n-{1-[cis-4-(hydroxymethyl)cyclohexyl]-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl}-3-(prop-2-en-1-ylsulfamoyl)benzamide | Human | 5377 | |
| ALK | ALK | TK | 4foc | A | | methyl cis-4-[2-(benzoylamino)-6-(piperidin-1-ylmethyl)-1h-benzimidazol-1-yl]cyclohexanecarboxylate | Human | 5392 | |
| ALK | ALK | TK | 4fod | A | A | 4-fluoro-n-{(2e)-6-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-1-[cis-4-(propan-2-ylcarbamoyl)cyclohexyl]-1,3-dihydro-2h-benzimidazol-2-ylidene}benzamide | Human | 5383 | |
| ALK | ALK | TK | 4fod | A | B | 4-fluoro-n-{(2e)-6-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-1-[cis-4-(propan-2-ylcarbamoyl)cyclohexyl]-1,3-dihydro-2h-benzimidazol-2-ylidene}benzamide | Human | 5404 | |
| ALK | ALK | TK | 4joa | A | A | 3-[1-(2,5-difluorobenzyl)-1h-pyrazol-4-yl]-5-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 5389 | |
| ALK | ALK | TK | 4mkc | A | A | 5-chloro-n~2~-[5-methyl-4-(piperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]pyrimidine-2,4-diamine | Human | 5401 | |
| ALK | ALK | TK | 4mkc | A | B | 5-chloro-n~2~-[5-methyl-4-(piperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]pyrimidine-2,4-diamine | Human | 5386 | |
| ALK | ALK | TK | 4tt7 | A | A | - | Human | 5406 | |
| ALK | ALK | TK | 4tt7 | A | B | - | Human | 5382 | |
| ALK | ALK | TK | 4z55 | A | A | n~6~-[5-methyl-4-(1-methylpiperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]-2h-pyrazolo[3,4-d]pyrimidine-4,6-diamine | Human | 6393 | |
| ALK | ALK | TK | 4z55 | A | B | n~6~-[5-methyl-4-(1-methylpiperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]-2h-pyrazolo[3,4-d]pyrimidine-4,6-diamine | Human | 6392 | |
| ALK | ALK | TK | 5a9u | A | A | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | 6692 | |
| ALK | ALK | TK | 5a9u | A | B | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | 6685 | |
| ALK | ALK | TK | 5aa8 | A | A | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | 6688 | |
| ALK | ALK | TK | 5aa8 | A | B | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | 6684 | |
| ALK | ALK | TK | 5aa9 | A | A | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | 6682 | |
| ALK | ALK | TK | 5aa9 | A | B | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | 6687 | |
| ALK | ALK | TK | 5aaa | A | A | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 6691 | |
| ALK | ALK | TK | 5aaa | A | B | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 6683 | |
| ALK | ALK | TK | 5aab | A | A | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 6689 | |
| ALK | ALK | TK | 5aab | A | B | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 6681 | |
| ALK | ALK | TK | 5aac | A | A | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 6690 | |
| ALK | ALK | TK | 5aac | A | B | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 6686 | |
| ALK | ALK | TK | 5fto | A | A | entrectinib | Human | 6520 | |
| ALK | ALK | TK | 5fto | A | B | entrectinib | Human | 6521 | |
| ALK | ALK | TK | 5ftq | A | A | n-[5-(3,5-difluorobenzyl)-1h-indazol-3-yl]-2-[(4-hydroxycyclohexyl)amino]-4-(4-methylpiperazin-1-yl) benzamide | Human | 6519 | |
| ALK | ALK | TK | 5ftq | A | B | n-[5-(3,5-difluorobenzyl)-1h-indazol-3-yl]-2-[(4-hydroxycyclohexyl)amino]-4-(4-methylpiperazin-1-yl) benzamide | Human | 6518 | |
| ALK | ALK | TK | 5imx | A | | 5-chloro-n~2~-{5-methyl-4-(1-methylpiperidin-4-yl)-2-[(propan-2-yl)oxy]phenyl}-n~4~-{1-methyl-3-[(propan-2-yl)sulfonyl]-1h-pyrazol-4-yl}pyrimidine-2,4-diamine | Human | 6604 | |
| ALK | ALK | TK | 5iug | A | A | n-[3-(4-{[(5-tert-butyl-1,2-oxazol-3-yl)carbamoyl]amino}-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamide | Human | 6640 | |
| ALK | ALK | TK | 5iug | A | B | n-[3-(4-{[(5-tert-butyl-1,2-oxazol-3-yl)carbamoyl]amino}-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamide | Human | 6639 | |
| ALK | ALK | TK | 5iuh | A | | 4-[(4-methylpiperazin-1-yl)methyl]-n-{3-[3-methyl-4-({[5-(propan-2-yl)-1,2-oxazol-3-yl]carbamoyl}amino)phenyl]-1h-pyrazol-5-yl}benzamide | Human | 6638 | |
| ALK | ALK | TK | 5iui | A | A | n-[3-(4-amino-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamide | Human | 6641 | |
| ALK | ALK | TK | 5iui | A | B | n-[3-(4-amino-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamide | Human | 6642 | |
| ALK | ALK | TK | 5kz0 | A | | 2-[(1~{r})-1-[2-azanyl-5-(1,3-dimethylpyrazol-4-yl)pyridin-3-yl]oxyethyl]-4-fluoranyl-~{n},~{n}-dimethyl-benzamide | Human | 6970 | |
| ALK | ALK | TK | 6cdt | A | | - | Human | 11263 | |
| ALK | ALK | TK | 6e0r | A | A | n-[(1s)-1-(5-fluoropyridin-2-yl)ethyl]-1-(5-methyl-1h-pyrazol-3-yl)-3-[(oxetan-3-yl)sulfonyl]-1h-pyrrolo[2,3-b]pyridin-6-amine | Human | 11268 | |
| ALK | ALK | TK | 6e0r | A | B | n-[(1s)-1-(5-fluoropyridin-2-yl)ethyl]-1-(5-methyl-1h-pyrazol-3-yl)-3-[(oxetan-3-yl)sulfonyl]-1h-pyrrolo[2,3-b]pyridin-6-amine | Human | 11266 | |
| ALK | ALK | TK | 6ebw | A | A | [6-{[(1s)-1-(5-fluoropyridin-2-yl)ethyl]amino}-1-(5-methyl-1h-pyrazol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl](morpholin-4-yl)methanone | Human | 11269 | |
| ALK | ALK | TK | 6ebw | A | B | [6-{[(1s)-1-(5-fluoropyridin-2-yl)ethyl]amino}-1-(5-methyl-1h-pyrazol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl](morpholin-4-yl)methanone | Human | 11264 | |
| ALK | ALK | TK | 6edl | A | A | n-[(1s)-1-(2,4-difluorophenyl)ethyl]-3-(5-methyl-1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-6-amine | Human | 11267 | |
| ALK | ALK | TK | 6edl | A | B | n-[(1s)-1-(2,4-difluorophenyl)ethyl]-3-(5-methyl-1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-6-amine | Human | 11265 | |
| ALK | ALK | TK | 6mx8 | A | A | 5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamine | Human | 10798 | |
| ALK | ALK | TK | 6mx8 | A | B | 5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamine | Human | 10799 | |
| ALK | ALK | TK | 7btt | A | A | 2-(dimethylamino)-1-[5-methoxy-6-[[4-[(2-propan-2-ylsulfonylphenyl)amino]-5h-pyrrolo[3,2-d]pyrimidin-2-yl]amino]-2,3-dihydroindol-1-yl]ethanone | Human | 13484 | |
| ALK | ALK | TK | 7btt | A | B | 2-(dimethylamino)-1-[5-methoxy-6-[[4-[(2-propan-2-ylsulfonylphenyl)amino]-5h-pyrrolo[3,2-d]pyrimidin-2-yl]amino]-2,3-dihydroindol-1-yl]ethanone | Human | 13483 | |
| ALK | ALK | TK | 7jy4 | A | | 1-{(1s,2s)-1-(2,4-difluorophenyl)-2-[2-(3-methyl-1h-pyrazol-5-yl)-4-(trifluoromethyl)phenoxy]cyclopropyl}methanamine | Human | 13240 | |
| ALK | ALK | TK | 7jyr | A | A | 4-{[(1r,2r)-2-(2,4-difluorophenyl)cyclopropyl]oxy}-3-(5-methyl-1h-pyrazol-3-yl)benzonitrile | Human | 13243 | |
| ALK | ALK | TK | 7jyr | A | B | 4-{[(1r,2r)-2-(2,4-difluorophenyl)cyclopropyl]oxy}-3-(5-methyl-1h-pyrazol-3-yl)benzonitrile | Human | 13241 | |
| ALK | ALK | TK | 7jys | A | A | 3-(3-chlorophenyl)-5-methyl-1h-pyrazole | Human | 13244 | |
| ALK | ALK | TK | 7jys | A | B | 3-(3-chlorophenyl)-5-methyl-1h-pyrazole | Human | 13239 | |
| ALK | ALK | TK | 7jyt | A | A | 3-(3-methyl-1h-pyrazol-5-yl)pyridine | Human | 13238 | |
| ALK | ALK | TK | 7jyt | A | B | 3-(3-methyl-1h-pyrazol-5-yl)pyridine | Human | 13242 | |
| ALK | ALK | TK | 7r7k | A | | 4-(6-amino-5-{(1r)-1-[5-fluoro-2-(2h-1,2,3-triazol-2-yl)phenyl]ethoxy}pyridin-3-yl)-2,3-dihydro-1h-isoindol-1-one | Human | 14267 | |
| ALK | ALK | TK | 7r7r | A | | (2r)-2-[5-(6-amino-5-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diol | Human | 14266 | |
| ALK | ALK | TK | 8arj | A | A | 3-(dimethylamino)-1-[3-[4-(4-methylpiperazin-1-yl)phenyl]-9~{h}-pyrido[2,3-b]indol-6-yl]prop-2-en-1-one | Human | 14366 | |
| ALK | ALK | TK | 8arj | A | B | 3-(dimethylamino)-1-[3-[4-(4-methylpiperazin-1-yl)phenyl]-9~{h}-pyrido[2,3-b]indol-6-yl]prop-2-en-1-one | Human | 14367 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 5luq | A | | - | Human | 9321 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 5luq | B | | - | Human | 9319 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 5w1r | A | | - | Human | 9320 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 5y3r | C | | - | Human | 9318 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zfp | A | | - | Human | 12926 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zh2 | A | | - | Human | 12927 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zh4 | A | | - | Human | 12930 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zh6 | A | | - | Human | 12929 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zh8 | A | | - | Human | 12925 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zha | A | | - | Human | 12931 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zhe | A | | - | Human | 12928 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zhe | F | | - | Human | 12932 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k0y | A | A | - | Human | 13213 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k0y | A | B | - | Human | 13214 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k10 | A | | - | Human | 13217 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k11 | A | | - | Human | 13208 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k17 | A | | - | Human | 13215 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k17 | B | | - | Human | 13212 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k19 | A | | - | Human | 13216 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k1b | A | | - | Human | 13218 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k1j | A | | - | Human | 13209 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k1k | A | | - | Human | 13211 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k1n | A | | - | Human | 13210 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7lt3 | C | | adenosine-5'-diphosphate | Human | 13500 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7lt3 | L | | adenosine-5'-diphosphate | Human | 13501 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7nfc | A | | - | Human | 13852 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7nfe | A | | - | Human | 13851 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7otm | A | | 8-(dibenzo[b,d]thiophen-4-yl)-2-(morpholin-4-yl)-4h-chromen-4-one | Human | 14061 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7otp | A | | phosphothiophosphoric acid-adenylate ester | Human | 14054 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7otv | A | | (1s,6br,9as,11r,11br)-9a,11b-dimethyl-1-[(methyloxy)methyl]-3,6,9-trioxo-1,6,6b,7,8,9,9a,10,11,11b-decahydro-3h-furo[4,3,2-de]indeno[4,5-h][2]benzopyran-11-yl acetate | Human | 14063 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7otw | A | | 7-methyl-2-[(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(oxan-4-yl)purin-8-one | Human | 14056 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7oty | A | | (~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanol | Human | 14057 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7sgl | A | A | adenosine-5'-triphosphate | Human | 14059 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7sgl | A | B | adenosine-5'-triphosphate | Human | 14062 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7su3 | A | A | adenosine-5'-triphosphate | Human | 14058 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7su3 | A | B | adenosine-5'-triphosphate | Human | 14053 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7sud | A | A | adenosine-5'-triphosphate | Human | 14055 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7sud | A | B | adenosine-5'-triphosphate | Human | 14060 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7tyr | A | A | - | Human | 14322 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7tyr | A | B | - | Human | 14321 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7z87 | A | A | (~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanol | Human | 14592 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7z87 | A | B | (~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanol | Human | 14593 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7z88 | A | | (~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanol | Human | 14594 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 8bh3 | A | | - | Human | 14768 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 8bhv | A | | - | Human | 14769 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 8bhy | A | | - | Human | 14770 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 8ezb | C | | adenosine-5'-triphosphate | Human | 14798 | |
| ATM | PIKK | Atypical | 5np0 | A | | - | Human | 9267 | |
| ATM | PIKK | Atypical | 5np0 | B | | - | Human | 9266 | |
| ATM | PIKK | Atypical | 5np1 | A | | - | Human | 9268 | |
| ATM | PIKK | Atypical | 6k9k | A | | - | Human | 11897 | |
| ATM | PIKK | Atypical | 6k9l | A | | - | Human | 11896 | |
| ATM | PIKK | Atypical | 6k9l | B | | - | Human | 11895 | |
| ATM | PIKK | Atypical | 7ni4 | A | | 8-(1,3-dimethylpyrazol-4-yl)-1-(3-fluoranyl-5-methoxy-pyridin-4-yl)-7-methoxy-3-methyl-imidazo[4,5-c]quinolin-2-one | Human | 13864 | |
| ATM | PIKK | Atypical | 7ni5 | A | | 2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-one | Human | 13863 | |
| ATM | PIKK | Atypical | 7ni6 | A | | phosphothiophosphoric acid-adenylate ester | Human | 13862 | |
| ATM | PIKK | Atypical | 7sic | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14101 | |
| ATM | PIKK | Atypical | 7sid | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14102 | |
| ATM | PIKK | Atypical | 8oxm | B | | phosphoaminophosphonic acid-adenylate ester | Human | 14992 | |
| ATM | PIKK | Atypical | 8oxo | B | | phosphoaminophosphonic acid-adenylate ester | Human | 14993 | |
| ATM | PIKK | Atypical | 8oxp | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14991 | |
| ATM | PIKK | Atypical | 8oxq | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14990 | |
| ATR | PIKK | Atypical | 5yz0 | A | | - | Human | 9523 | |
| ATR | PIKK | Atypical | 5yz0 | B | | - | Human | 9524 | |
| Aurka (AurA) | AUR | Other | 3d14 | A | A | 1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]urea | Mouse | 5781 | |
| Aurka (AurA) | AUR | Other | 3d14 | A | B | 1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]urea | Mouse | 5775 | |
| Aurka (AurA) | AUR | Other | 3d15 | A | A | 1-(3-chlorophenyl)-3-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}urea | Mouse | 5777 | |
| Aurka (AurA) | AUR | Other | 3d2i | A | | 1-(5-{2-[(1-methyl-1h-pyrazolo[4,3-d]pyrimidin-7-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]urea | Mouse | 5782 | |
| Aurka (AurA) | AUR | Other | 3d2k | A | | (7-{[2-(2-{[(3-chlorophenyl)carbamoyl]amino}-1,3-thiazol-5-yl)ethyl]amino}-1h-pyrazolo[4,3-d]pyrimidin-1-yl)acetic acid | Mouse | 5776 | |
| Aurka (AurA) | AUR | Other | 3daj | A | | n-butyl-3-{[6-(9h-purin-6-ylamino)hexanoyl]amino}benzamide | Mouse | 5779 | |
| Aurka (AurA) | AUR | Other | 3dj5 | A | | 3-({3-[(6-amino-5-bromopyrimidin-4-yl)sulfanyl]propanoyl}amino)-4-methoxy-n-phenylbenzamide | Mouse | 5783 | |
| Aurka (AurA) | AUR | Other | 3dj6 | A | | 4-methoxy-n-phenyl-3-({3-[(1h-pyrrolo[2,3-b]pyridin-5-ylmethyl)sulfanyl]propanoyl}amino)benzamide | Mouse | 5778 | |
| Aurka (AurA) | AUR | Other | 3dj7 | A | A | 1-(5-{2-[(6-amino-5-bromopyrimidin-4-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]urea | Mouse | 5780 | |
| AURKA (AurA) | Aur | Other | 1mq4 | A | | adenosine-5'-diphosphate | Human | 1977 | |
| AURKA (AurA) | Aur | Other | 1muo | A | | adenosine | Human | 2062 | |
| AURKA (AurA) | Aur | Other | 1ol5 | A | | adenosine-5'-diphosphate | Human | 2080 | |
| AURKA (AurA) | Aur | Other | 1ol6 | A | | adenosine-5'-triphosphate | Human | 2081 | |
| AURKA (AurA) | Aur | Other | 1ol7 | A | | adenosine-5'-diphosphate | Human | 2014 | |
| AURKA (AurA) | Aur | Other | 2bmc | A | | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | 2015 | |
| AURKA (AurA) | Aur | Other | 2bmc | B | | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | 2008 | |
| AURKA (AurA) | Aur | Other | 2bmc | C | | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | 2060 | |
| AURKA (AurA) | Aur | Other | 2bmc | D | | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | 1984 | |
| AURKA (AurA) | Aur | Other | 2bmc | E | | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | 2069 | |
| AURKA (AurA) | Aur | Other | 2bmc | F | | (3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamide | Human | 1993 | |
| AURKA (AurA) | Aur | Other | 2c6d | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2019 | |
| AURKA (AurA) | Aur | Other | 2c6d | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 1981 | |
| AURKA (AurA) | Aur | Other | 2c6e | A | | n-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamide | Human | 1989 | |
| AURKA (AurA) | Aur | Other | 2c6e | B | | n-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamide | Human | 2046 | |
| AURKA (AurA) | Aur | Other | 2dwb | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2035 | |
| AURKA (AurA) | Aur | Other | 2j4z | A | | 4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamide | Human | 2053 | |
| AURKA (AurA) | Aur | Other | 2j4z | B | | 4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamide | Human | 1990 | |
| AURKA (AurA) | Aur | Other | 2j50 | A | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 2001 | |
| AURKA (AurA) | Aur | Other | 2j50 | B | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 2050 | |
| AURKA (AurA) | Aur | Other | 2np8 | A | | n-{3-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]phenyl}cyclopropanecarboxamide | Human | 2075 | |
| AURKA (AurA) | Aur | Other | 2w1c | A | | 4-{[2-(4-{[(4-fluorophenyl)carbonyl]amino}-1h-pyrazol-3-yl)-1h-benzimidazol-6-yl]methyl}morpholin-4-ium | Human | 2027 | |
| AURKA (AurA) | Aur | Other | 2w1d | A | | 2-(1h-pyrazol-3-yl)-1h-benzimidazole | Human | 2011 | |
| AURKA (AurA) | Aur | Other | 2w1e | A | | 4-[(2-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-3-yl}-1h-benzimidazol-5-yl)methyl]morpholin-4-ium | Human | 2038 | |
| AURKA (AurA) | Aur | Other | 2w1f | A | | n-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamide | Human | 2055 | |
| AURKA (AurA) | Aur | Other | 2w1g | A | | 2-{4-[(cyclopropylcarbamoyl)amino]-1h-pyrazol-3-yl}-6-(morpholin-4-ium-4-ylmethyl)-1h-3,1-benzimidazol-3-ium | Human | 1962 | |
| AURKA (AurA) | Aur | Other | 2wqe | A | | adenosine-5'-diphosphate | Human | 2071 | |
| AURKA (AurA) | Aur | Other | 2wtv | A | A | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2056 | |
| AURKA (AurA) | Aur | Other | 2wtv | A | B | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 1997 | |
| AURKA (AurA) | Aur | Other | 2wtv | B | A | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2037 | |
| AURKA (AurA) | Aur | Other | 2wtv | B | B | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2057 | |
| AURKA (AurA) | Aur | Other | 2wtv | C | A | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2017 | |
| AURKA (AurA) | Aur | Other | 2wtv | C | B | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2016 | |
| AURKA (AurA) | Aur | Other | 2wtv | D | A | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2078 | |
| AURKA (AurA) | Aur | Other | 2wtv | D | B | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2076 | |
| AURKA (AurA) | Aur | Other | 2wtw | A | | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 1956 | |
| AURKA (AurA) | Aur | Other | 2x6d | A | A | 6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridine | Human | 1978 | |
| AURKA (AurA) | Aur | Other | 2x6d | A | B | 6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridine | Human | 1975 | |
| AURKA (AurA) | Aur | Other | 2x6e | A | | 6-bromo-7-{4-[(5-methylisoxazol-3-yl)methyl]piperazin-1-yl}-2-[4-(4-methylpiperazin-1-yl)phenyl]-1h-imidazo[4,5-b]pyridine | Human | 2079 | |
| AURKA (AurA) | Aur | Other | 2x81 | A | | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 1966 | |
| AURKA (AurA) | Aur | Other | 2xne | A | | 3-chloro-n-(4-morpholin-4-ylphenyl)-6-pyridin-3-ylimidazo[1,2-a]pyrazin-8-amine | Human | 7221 | |
| AURKA (AurA) | Aur | Other | 2xng | A | A | n-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamide | Human | 1994 | |
| AURKA (AurA) | Aur | Other | 2xng | A | B | n-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamide | Human | 2083 | |
| AURKA (AurA) | Aur | Other | 2xru | A | | 3-({[4-(4-methylpiperazin-1-yl)phenyl]carbonyl}amino)-n-[(1r)-1-phenylpropyl]-1h-thieno[3,2-c]pyrazole-5-carboxamide | Human | 1954 | |
| AURKA (AurA) | Aur | Other | 3coh | A | | 8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-one | Human | 1963 | |
| AURKA (AurA) | Aur | Other | 3coh | B | | 8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-one | Human | 2024 | |
| AURKA (AurA) | Aur | Other | 3e5a | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 2006 | |
| AURKA (AurA) | Aur | Other | 3efw | A | | 1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]urea | Human | 2010 | |
| AURKA (AurA) | Aur | Other | 3efw | B | | 1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]urea | Human | 2074 | |
| AURKA (AurA) | Aur | Other | 3fdn | A | | n-[3-(acetylamino)phenyl]-5-{(2e)-2-[(4-methoxyphenyl)methylidene]hydrazino}-3-methyl-1h-pyrazole-4-carboxamide | Human | 1973 | |
| AURKA (AurA) | Aur | Other | 3h0y | A | | 2-chloro-n-[4-({5-fluoro-2-[(4-hydroxyphenyl)amino]pyrimidin-4-yl}amino)phenyl]benzamide | Human | 1965 | |
| AURKA (AurA) | Aur | Other | 3h0z | A | | 4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamide | Human | 1970 | |
| AURKA (AurA) | Aur | Other | 3h0z | B | | 4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamide | Human | 1986 | |
| AURKA (AurA) | Aur | Other | 3h0z | C | | 4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamide | Human | 2063 | |
| AURKA (AurA) | Aur | Other | 3h10 | A | | 9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amine | Human | 2009 | |
| AURKA (AurA) | Aur | Other | 3h10 | B | | 9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amine | Human | 1988 | |
| AURKA (AurA) | Aur | Other | 3h10 | D | | 9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amine | Human | 2059 | |
| AURKA (AurA) | Aur | Other | 3ha6 | A | | n~2~-(3,4-dimethoxyphenyl)-n~4~-[2-(2-fluorophenyl)ethyl]-n~6~-quinolin-6-yl-1,3,5-triazine-2,4,6-triamine | Human | 2048 | |
| AURKA (AurA) | Aur | Other | 3k5u | A | | 2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanol | Human | 2031 | |
| AURKA (AurA) | Aur | Other | 3lau | A | | n-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]butanamide | Human | 1971 | |
| AURKA (AurA) | Aur | Other | 3m11 | A | | 1-(4-{2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylurea | Human | 2036 | |
| AURKA (AurA) | Aur | Other | 3myg | A | | 2-{ethyl[(5-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}isothiazol-3-yl)methyl]amino}-2-methylpropan-1-ol | Human | 2065 | |
| AURKA (AurA) | Aur | Other | 3nrm | A | | n-(3-methylisothiazol-5-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-amine | Human | 2052 | |
| AURKA (AurA) | Aur | Other | 3o50 | A | | n-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamide | Human | 1958 | |
| AURKA (AurA) | Aur | Other | 3o50 | B | | n-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamide | Human | 2067 | |
| AURKA (AurA) | Aur | Other | 3o51 | A | | n-[4-({3-[5-fluoro-2-(methylideneamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-2-(phenylamino)benzamide | Human | 1974 | |
| AURKA (AurA) | Aur | Other | 3p9j | A | | 4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-one | Human | 2003 | |
| AURKA (AurA) | Aur | Other | 3qbn | A | | 5-chloro-n~4~-cyclopropyl-n~2~-[4-(2-methoxyethoxy)phenyl]pyrimidine-2,4-diamine | Human | 2032 | |
| AURKA (AurA) | Aur | Other | 3r21 | A | A | n-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamide | Human | 1991 | |
| AURKA (AurA) | Aur | Other | 3r21 | A | B | n-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamide | Human | 2033 | |
| AURKA (AurA) | Aur | Other | 3r22 | A | | n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamide | Human | 2034 | |
| AURKA (AurA) | Aur | Other | 3unz | A | | 4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 1972 | |
| AURKA (AurA) | Aur | Other | 3unz | B | | 4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 2049 | |
| AURKA (AurA) | Aur | Other | 3uo4 | A | | 4-{[4-(biphenyl-2-ylamino)pyrimidin-2-yl]amino}benzoic acid | Human | 1976 | |
| AURKA (AurA) | Aur | Other | 3uo5 | A | | 4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acid | Human | 2045 | |
| AURKA (AurA) | Aur | Other | 3uo6 | A | | 4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 1985 | |
| AURKA (AurA) | Aur | Other | 3uo6 | B | | 4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 1960 | |
| AURKA (AurA) | Aur | Other | 3uod | A | | 4-[(4-{[2-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzoic acid | Human | 1980 | |
| AURKA (AurA) | Aur | Other | 3uoh | A | | 4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 2077 | |
| AURKA (AurA) | Aur | Other | 3uoh | B | | 4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 2000 | |
| AURKA (AurA) | Aur | Other | 3uoj | A | | 4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 2042 | |
| AURKA (AurA) | Aur | Other | 3uoj | B | | 4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 1979 | |
| AURKA (AurA) | Aur | Other | 3uok | A | | 4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acid | Human | 2054 | |
| AURKA (AurA) | Aur | Other | 3uok | B | | 4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acid | Human | 2047 | |
| AURKA (AurA) | Aur | Other | 3uol | A | | n~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamine | Human | 2004 | |
| AURKA (AurA) | Aur | Other | 3uol | B | | n~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamine | Human | 2051 | |
| AURKA (AurA) | Aur | Other | 3up2 | A | | 4-[(4-{[2-(trifluoromethoxy)phenyl]amino}pyrimidin-2-yl)amino]benzoic acid | Human | 2005 | |
| AURKA (AurA) | Aur | Other | 3up7 | A | | 2-({2-[(4-carboxyphenyl)amino]pyrimidin-4-yl}amino)benzoic acid | Human | 2025 | |
| AURKA (AurA) | Aur | Other | 3vap | A | | 3-(1-{2-[(3-fluoropyridinium-4-yl)amino]-2-oxoethyl}-1h-pyrazol-4-yl)-6-methyl-8-[(3-{[(1r,3r)-3-methylpiperidinium-1-yl]methyl}-1,2-thiazol-5-yl)amino]imidazo[1,2-a]pyrazin-1-ium | Human | 2029 | |
| AURKA (AurA) | Aur | Other | 3w10 | A | | 1-(3-methoxyphenyl)-n-(5-methyl-1h-pyrazol-3-yl)isoquinolin-3-amine | Human | 2068 | |
| AURKA (AurA) | Aur | Other | 3w16 | A | | 4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-one | Human | 2012 | |
| AURKA (AurA) | Aur | Other | 3w18 | A | | 2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamide | Human | 1961 | |
| AURKA (AurA) | Aur | Other | 3w18 | B | | 2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamide | Human | 1967 | |
| AURKA (AurA) | Aur | Other | 3w2c | A | | 2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamide | Human | 2066 | |
| AURKA (AurA) | Aur | Other | 3w2c | C | | 2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamide | Human | 2021 | |
| AURKA (AurA) | Aur | Other | 3w2c | E | | 2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamide | Human | 1953 | |
| AURKA (AurA) | Aur | Other | 3w2c | G | | 2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamide | Human | 2026 | |
| AURKA (AurA) | Aur | Other | 4b0g | A | A | 6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridine | Human | 2082 | |
| AURKA (AurA) | Aur | Other | 4b0g | A | B | 6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridine | Human | 2070 | |
| AURKA (AurA) | Aur | Other | 4bn1 | A | A | adenosine-5'-diphosphate | Human | 1955 | |
| AURKA (AurA) | Aur | Other | 4bn1 | A | B | adenosine-5'-diphosphate | Human | 1983 | |
| AURKA (AurA) | Aur | Other | 4byi | A | | (s)-n-((1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)methyl)acetamide | Human | 1992 | |
| AURKA (AurA) | Aur | Other | 4byj | A | | (s)-n-(1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)acetamide | Human | 1969 | |
| AURKA (AurA) | Aur | Other | 4c3p | A | | phosphomethylphosphonic acid adenylate ester | Human | 2018 | |
| AURKA (AurA) | Aur | Other | 4c3p | D | | phosphomethylphosphonic acid adenylate ester | Human | 2030 | |
| AURKA (AurA) | Aur | Other | 4c3r | A | | phosphomethylphosphonic acid adenylate ester | Human | 2058 | |
| AURKA (AurA) | Aur | Other | 4ceg | A | | adenosine-5'-diphosphate | Human | 2073 | |
| AURKA (AurA) | Aur | Other | 4dea | A | | 4,4'-(pyrimidine-2,4-diyldiimino)dibenzoic acid | Human | 2064 | |
| AURKA (AurA) | Aur | Other | 4deb | A | | 4-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzamide | Human | 1996 | |
| AURKA (AurA) | Aur | Other | 4ded | A | | 2-({2-[(4-carbamoylphenyl)amino]pyrimidin-4-yl}amino)benzamide | Human | 2043 | |
| AURKA (AurA) | Aur | Other | 4dee | A | | adenosine-5'-diphosphate | Human | 1952 | |
| AURKA (AurA) | Aur | Other | 4dhf | A | | 7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 1964 | |
| AURKA (AurA) | Aur | Other | 4dhf | B | | 7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 1982 | |
| AURKA (AurA) | Aur | Other | 4j8m | A | | 1-[4-[[4-[(5-cyclopentyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]-3-[3-(trifluoromethyl)phenyl]urea | Human | 2020 | |
| AURKA (AurA) | Aur | Other | 4j8n | A | | - | Human | 2028 | |
| AURKA (AurA) | Aur | Other | 4j8n | B | | - | Human | 2061 | |
| AURKA (AurA) | Aur | Other | 4j8n | C | | - | Human | 2007 | |
| AURKA (AurA) | Aur | Other | 4j8n | D | | - | Human | 1995 | |
| AURKA (AurA) | Aur | Other | 4jai | A | | n-{4-[(6-oxo-5,6-dihydrobenzo[c][1,8]naphthyridin-1-yl)amino]phenyl}benzamide | Human | 1999 | |
| AURKA (AurA) | Aur | Other | 4jaj | A | | benzo[c][1,8]naphthyridin-6(5h)-one | Human | 2040 | |
| AURKA (AurA) | Aur | Other | 4jbo | A | | 1-(4-{2-[(6-{4-[2-(dimethylamino)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylurea | Human | 2072 | |
| AURKA (AurA) | Aur | Other | 4jbp | A | | 1-(4-{2-[(6-{4-[2-(4-hydroxypiperidin-1-yl)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylurea | Human | 2041 | |
| AURKA (AurA) | Aur | Other | 4jbq | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 1957 | |
| AURKA (AurA) | Aur | Other | 4o0s | A | | adenosine | Human | 2039 | |
| AURKA (AurA) | Aur | Other | 4o0u | A | | adenosine | Human | 2022 | |
| AURKA (AurA) | Aur | Other | 4o0w | A | | adenosine | Human | 1959 | |
| AURKA (AurA) | Aur | Other | 4prj | A | | n-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamide | Human | 2023 | |
| AURKA (AurA) | Aur | Other | 4uyn | A | | ethyl (9s)-9-[5-(1h-benzimidazol-2-ylsulfanyl)furan-2-yl]-8-hydroxy-5,6,7,9-tetrahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylate | Human | 2002 | |
| AURKA (AurA) | Aur | Other | 4uzd | A | | ethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylate | Human | 2013 | |
| AURKA (AurA) | Aur | Other | 4uzd | B | | ethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylate | Human | 1968 | |
| AURKA (AurA) | Aur | Other | 4uzh | A | | (4s)-4-(2-fluorophenyl)-2,4,6,7,8,9-hexahydro-5h-pyrazolo[3,4-b][1,7]naphthyridin-5-one | Human | 1998 | |
| AURKA (AurA) | Aur | Other | 4zs0 | A | | 5-hydroxy-1'h-1,2'-bibenzimidazol-2(3h)-one | Human | 6801 | |
| AURKA (AurA) | Aur | Other | 4ztq | A | | (2z,5z)-2-[(4-ethylphenyl)imino]-3-(2-methoxyethyl)-5-(pyridin-4-ylmethylidene)-1,3-thiazolidin-4-one | Human | 6804 | |
| AURKA (AurA) | Aur | Other | 4ztr | A | | 6-({4-[(z)-{(2z)-2-[(4-ethylphenyl)imino]-3-methyl-4-oxo-1,3-thiazolidin-5-ylidene}methyl]pyridin-2-yl}amino)pyridine-3-carboxylic acid | Human | 6817 | |
| AURKA (AurA) | Aur | Other | 4zts | A | | (2z,5z)-2-[(4-ethylphenyl)imino]-3-methyl-5-[(2-{[4-(1h-tetrazol-5-yl)phenyl]amino}pyridin-4-yl)methylidene]-1,3-thiazolidin-4-one | Human | 6814 | |
| AURKA (AurA) | Aur | Other | 5aad | A | | 7-(1-benzyl-1h-pyrazol-4-yl)-6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridine | Human | 6011 | |
| AURKA (AurA) | Aur | Other | 5aae | A | | 3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-5-methylisoxazole | Human | 6012 | |
| AURKA (AurA) | Aur | Other | 5aaf | A | | 3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-n,n-dimethylbenzamide | Human | 6013 | |
| AURKA (AurA) | Aur | Other | 5aag | A | | [3-[[4-[6-chloranyl-2-(1,3-dimethylpyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl]pyrazol-1-yl]methyl]phenyl]-(4-methylpiperazin-1-yl)methanone | Human | 6010 | |
| AURKA (AurA) | Aur | Other | 5dn3 | A | A | adenosine-5'-triphosphate | Human | 6802 | |
| AURKA (AurA) | Aur | Other | 5dn3 | A | B | adenosine-5'-triphosphate | Human | 6818 | |
| AURKA (AurA) | Aur | Other | 5dnr | A | A | adenosine-5'-triphosphate | Human | 6810 | |
| AURKA (AurA) | Aur | Other | 5dnr | A | B | adenosine-5'-triphosphate | Human | 6809 | |
| AURKA (AurA) | Aur | Other | 5dos | A | | adenosine-5'-triphosphate | Human | 6807 | |
| AURKA (AurA) | Aur | Other | 5dpv | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6808 | |
| AURKA (AurA) | Aur | Other | 5dpv | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6826 | |
| AURKA (AurA) | Aur | Other | 5dr2 | A | | adenosine-5'-triphosphate | Human | 6825 | |
| AURKA (AurA) | Aur | Other | 5dr6 | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6811 | |
| AURKA (AurA) | Aur | Other | 5dr6 | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6805 | |
| AURKA (AurA) | Aur | Other | 5dr9 | A | | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6821 | |
| AURKA (AurA) | Aur | Other | 5drd | A | | adenosine-5'-triphosphate | Human | 6823 | |
| AURKA (AurA) | Aur | Other | 5dt0 | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6806 | |
| AURKA (AurA) | Aur | Other | 5dt0 | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 6803 | |
| AURKA (AurA) | Aur | Other | 5dt3 | A | | adenosine-5'-triphosphate | Human | 6816 | |
| AURKA (AurA) | Aur | Other | 5dt4 | A | | adenosine-5'-triphosphate | Human | 6815 | |
| AURKA (AurA) | Aur | Other | 5ew9 | A | A | 4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acid | Human | 6359 | |
| AURKA (AurA) | Aur | Other | 5ew9 | A | B | 4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acid | Human | 6360 | |
| AURKA (AurA) | Aur | Other | 5g15 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 9737 | |
| AURKA (AurA) | Aur | Other | 5g15 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 9739 | |
| AURKA (AurA) | Aur | Other | 5g1x | A | A | adenosine-5'-diphosphate | Human | 7267 | |
| AURKA (AurA) | Aur | Other | 5g1x | A | B | adenosine-5'-diphosphate | Human | 7266 | |
| AURKA (AurA) | Aur | Other | 5l8j | A | A | adenosine-5'-diphosphate | Human | 6820 | |
| AURKA (AurA) | Aur | Other | 5l8j | A | B | adenosine-5'-diphosphate | Human | 6812 | |
| AURKA (AurA) | Aur | Other | 5l8k | A | A | adenosine-5'-diphosphate | Human | 6819 | |
| AURKA (AurA) | Aur | Other | 5l8k | A | B | adenosine-5'-diphosphate | Human | 6813 | |
| AURKA (AurA) | Aur | Other | 5l8l | A | A | adenosine-5'-diphosphate | Human | 6822 | |
| AURKA (AurA) | Aur | Other | 5l8l | A | B | adenosine-5'-diphosphate | Human | 6824 | |
| AURKA (AurA) | Aur | Other | 5lxm | A | A | adenosine-5'-diphosphate | Human | 7142 | |
| AURKA (AurA) | Aur | Other | 5lxm | A | B | adenosine-5'-diphosphate | Human | 7141 | |
| AURKA (AurA) | Aur | Other | 5obj | A | | adenosine-5'-triphosphate | Human | 8305 | |
| AURKA (AurA) | Aur | Other | 5obr | A | | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8304 | |
| AURKA (AurA) | Aur | Other | 5odt | A | A | adenosine-5'-diphosphate | Human | 9738 | |
| AURKA (AurA) | Aur | Other | 5odt | A | B | adenosine-5'-diphosphate | Human | 9736 | |
| AURKA (AurA) | Aur | Other | 5one | A | A | 4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamide | Human | 8371 | |
| AURKA (AurA) | Aur | Other | 5one | A | B | 4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamide | Human | 8370 | |
| AURKA (AurA) | Aur | Other | 5orl | A | | adenosine-5'-diphosphate | Human | 8642 | |
| AURKA (AurA) | Aur | Other | 5orn | A | | adenosine-5'-diphosphate | Human | 8649 | |
| AURKA (AurA) | Aur | Other | 5oro | A | | adenosine-5'-diphosphate | Human | 8641 | |
| AURKA (AurA) | Aur | Other | 5orp | A | | adenosine-5'-diphosphate | Human | 8648 | |
| AURKA (AurA) | Aur | Other | 5orr | A | | adenosine-5'-diphosphate | Human | 8636 | |
| AURKA (AurA) | Aur | Other | 5ors | A | | adenosine-5'-diphosphate | Human | 8646 | |
| AURKA (AurA) | Aur | Other | 5ort | A | | adenosine-5'-diphosphate | Human | 8638 | |
| AURKA (AurA) | Aur | Other | 5orv | A | | adenosine-5'-diphosphate | Human | 8643 | |
| AURKA (AurA) | Aur | Other | 5orw | A | | adenosine-5'-diphosphate | Human | 8631 | |
| AURKA (AurA) | Aur | Other | 5orx | A | | adenosine-5'-diphosphate | Human | 8644 | |
| AURKA (AurA) | Aur | Other | 5ory | A | | adenosine-5'-diphosphate | Human | 8627 | |
| AURKA (AurA) | Aur | Other | 5orz | A | A | adenosine-5'-diphosphate | Human | 8639 | |
| AURKA (AurA) | Aur | Other | 5orz | A | B | adenosine-5'-diphosphate | Human | 8650 | |
| AURKA (AurA) | Aur | Other | 5os0 | A | | adenosine-5'-diphosphate | Human | 8632 | |
| AURKA (AurA) | Aur | Other | 5os1 | A | A | adenosine-5'-diphosphate | Human | 8628 | |
| AURKA (AurA) | Aur | Other | 5os1 | A | B | adenosine-5'-diphosphate | Human | 8630 | |
| AURKA (AurA) | Aur | Other | 5os2 | A | A | adenosine-5'-diphosphate | Human | 8635 | |
| AURKA (AurA) | Aur | Other | 5os2 | A | B | adenosine-5'-diphosphate | Human | 8633 | |
| AURKA (AurA) | Aur | Other | 5os3 | A | | adenosine-5'-diphosphate | Human | 8637 | |
| AURKA (AurA) | Aur | Other | 5os4 | A | | adenosine-5'-diphosphate | Human | 8652 | |
| AURKA (AurA) | Aur | Other | 5os5 | A | A | adenosine-5'-diphosphate | Human | 8647 | |
| AURKA (AurA) | Aur | Other | 5os5 | A | B | adenosine-5'-diphosphate | Human | 8629 | |
| AURKA (AurA) | Aur | Other | 5os6 | A | | adenosine-5'-diphosphate | Human | 8651 | |
| AURKA (AurA) | Aur | Other | 5osd | A | | adenosine-5'-diphosphate | Human | 8634 | |
| AURKA (AurA) | Aur | Other | 5ose | A | | adenosine-5'-diphosphate | Human | 8645 | |
| AURKA (AurA) | Aur | Other | 5osf | A | | adenosine-5'-diphosphate | Human | 8640 | |
| AURKA (AurA) | Aur | Other | 5zan | A | | 7-(4-methylpiperazin-1-yl)-n-(5-methyl-1h-pyrazol-3-yl)-2-[(e)-2-phenylethenyl]quinazolin-4-amine | Human | 10898 | |
| AURKA (AurA) | Aur | Other | 6c2r | A | A | (2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acid | Human | 10864 | |
| AURKA (AurA) | Aur | Other | 6c2r | A | B | (2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acid | Human | 10865 | |
| AURKA (AurA) | Aur | Other | 6c2t | A | A | (2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acid | Human | 10866 | |
| AURKA (AurA) | Aur | Other | 6c2t | A | B | (2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acid | Human | 10863 | |
| AURKA (AurA) | Aur | Other | 6c83 | A | | phosphomethylphosphonic acid adenylate ester | Human | 10934 | |
| AURKA (AurA) | Aur | Other | 6c83 | B | | phosphomethylphosphonic acid adenylate ester | Human | 10935 | |
| AURKA (AurA) | Aur | Other | 6cpe | A | A | - | Human | 10036 | |
| AURKA (AurA) | Aur | Other | 6cpe | A | B | - | Human | 10035 | |
| AURKA (AurA) | Aur | Other | 6cpf | A | | phosphomethylphosphonic acid adenylate ester | Human | 10033 | |
| AURKA (AurA) | Aur | Other | 6cpg | A | | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 10032 | |
| AURKA (AurA) | Aur | Other | 6cpg | D | | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 10034 | |
| AURKA (AurA) | Aur | Other | 6gra | A | | 1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)urea | Human | 11130 | |
| AURKA (AurA) | Aur | Other | 6hjj | A | A | ~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamide | Human | 10410 | |
| AURKA (AurA) | Aur | Other | 6hjj | A | B | ~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamide | Human | 10412 | |
| AURKA (AurA) | Aur | Other | 6hjk | A | | (~{e})-~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-but-2-enamide | Human | 10411 | |
| AURKA (AurA) | Aur | Other | 6i2u | A | | - | Human | 11652 | |
| AURKA (AurA) | Aur | Other | 6r49 | A | | adenosine-5'-diphosphate | Human | 11131 | |
| AURKA (AurA) | Aur | Other | 6r4a | A | | adenosine-5'-diphosphate | Human | 11134 | |
| AURKA (AurA) | Aur | Other | 6r4b | A | B | adenosine-5'-diphosphate | Human | 11133 | |
| AURKA (AurA) | Aur | Other | 6r4c | A | | adenosine-5'-diphosphate | Human | 11135 | |
| AURKA (AurA) | Aur | Other | 6r4d | A | | adenosine-5'-diphosphate | Human | 11132 | |
| AURKA (AurA) | Aur | Other | 6vpg | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 12659 | |
| AURKA (AurA) | Aur | Other | 6vpg | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 12667 | |
| AURKA (AurA) | Aur | Other | 6vph | A | A | dithiane diol | Human | 12666 | |
| AURKA (AurA) | Aur | Other | 6vph | A | B | dithiane diol | Human | 12655 | |
| AURKA (AurA) | Aur | Other | 6vpi | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 12656 | |
| AURKA (AurA) | Aur | Other | 6vpi | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 12669 | |
| AURKA (AurA) | Aur | Other | 6vpj | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 12657 | |
| AURKA (AurA) | Aur | Other | 6vpj | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 12654 | |
| AURKA (AurA) | Aur | Other | 6vpl | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 12662 | |
| AURKA (AurA) | Aur | Other | 6vpl | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 12670 | |
| AURKA (AurA) | Aur | Other | 6vpl | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 12664 | |
| AURKA (AurA) | Aur | Other | 6vpl | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 12668 | |
| AURKA (AurA) | Aur | Other | 6vpm | A | A | adenosine monophosphate | Human | 12661 | |
| AURKA (AurA) | Aur | Other | 6vpm | A | B | adenosine monophosphate | Human | 12658 | |
| AURKA (AurA) | Aur | Other | 6vpm | B | A | adenosine monophosphate | Human | 12660 | |
| AURKA (AurA) | Aur | Other | 6vpm | B | B | adenosine monophosphate | Human | 12663 | |
| AURKA (AurA) | Aur | Other | 6xka | A | | - | Human | 12665 | |
| AURKA (AurA) | Aur | Other | 6z4y | A | A | 6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12306 | |
| AURKA (AurA) | Aur | Other | 6z4y | A | B | 6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12307 | |
| AURKA (AurA) | Aur | Other | 7ayh | A | | 7-[2-[(4-methoxyphenyl)amino]pyrimidin-4-yl]-1,3,4,5-tetrahydro-1-benzazepin-2-one | Human | 13228 | |
| AURKA (AurA) | Aur | Other | 7ayi | A | | 7-(2-phenylazanylpyrimidin-4-yl)-1,3,4,5-tetrahydro-1-benzazepin-2-one | Human | 13229 | |
| AURKA (AurA) | Aur | Other | 7fic | A | A | 6-[(5-cyclopropyl-1~{h}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{n}-prop-2-ynyl-pyrimidine-4-carboxamide | Human | 14234 | |
| AURKA (AurA) | Aur | Other | 7fic | A | B | 6-[(5-cyclopropyl-1~{h}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{n}-prop-2-ynyl-pyrimidine-4-carboxamide | Human | 14233 | |
| AURKA (AurA) | Aur | Other | 7o2v | A | | 1-[[3,4-bis(fluoranyl)phenyl]methyl]-~{n}-[(1~{r})-2-[[(3~{e})-3-(1~{h}-imidazol-5-ylmethylidene)-2-oxidanylidene-1~{h}-indol-5-yl]amino]-2-oxidanylidene-1-phenyl-ethyl]-6-methyl-2-oxidanylidene-pyridine-3-carboxamide | Human | 13947 | |
| AURKA (AurA) | Aur | Other | 7ztl | A | A | adenosine-5'-diphosphate | Human | 14582 | |
| AURKA (AurA) | Aur | Other | 7ztl | A | B | adenosine-5'-diphosphate | Human | 14581 | |
| AURKA (AurA) | Aur | Other | 8c14 | A | A | adenosine-5'-diphosphate | Human | 15143 | |
| AURKA (AurA) | Aur | Other | 8c14 | A | B | adenosine-5'-diphosphate | Human | 15150 | |
| AURKA (AurA) | Aur | Other | 8c15 | A | A | adenosine-5'-diphosphate | Human | 15141 | |
| AURKA (AurA) | Aur | Other | 8c15 | A | B | adenosine-5'-diphosphate | Human | 15151 | |
| AURKA (AurA) | Aur | Other | 8c1d | A | A | adenosine-5'-diphosphate | Human | 15152 | |
| AURKA (AurA) | Aur | Other | 8c1d | A | B | adenosine-5'-diphosphate | Human | 15138 | |
| AURKA (AurA) | Aur | Other | 8c1e | A | | adenosine-5'-triphosphate | Human | 15145 | |
| AURKA (AurA) | Aur | Other | 8c1f | A | A | adenosine-5'-diphosphate | Human | 15140 | |
| AURKA (AurA) | Aur | Other | 8c1f | A | B | adenosine-5'-diphosphate | Human | 15149 | |
| AURKA (AurA) | Aur | Other | 8c1g | A | | adenosine-5'-diphosphate | Human | 15148 | |
| AURKA (AurA) | Aur | Other | 8c1h | A | A | adenosine-5'-diphosphate | Human | 15147 | |
| AURKA (AurA) | Aur | Other | 8c1h | A | B | adenosine-5'-diphosphate | Human | 15142 | |
| AURKA (AurA) | Aur | Other | 8c1i | A | A | adenosine-5'-diphosphate | Human | 15144 | |
| AURKA (AurA) | Aur | Other | 8c1i | A | B | adenosine-5'-diphosphate | Human | 15139 | |
| AURKA (AurA) | Aur | Other | 8c1k | A | | adenosine-5'-diphosphate | Human | 15146 | |
| AURKA (AurA) | Aur | Other | 8c1m | A | | adenosine-5'-diphosphate | Human | 15137 | |
| AURKA (AurA) | Aur | Other | 8guw | A | | adenosine-5'-diphosphate | Human | 14753 | |
| AURKA (AurA) | Aur | Other | 8jf4 | A | | 2-[4-[4-[bis(oxidanylidene)-$l^5-sulfanyl]oxyphenyl]carbonylpiperazin-1-yl]-6-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-n-prop-2-ynyl-pyrimidine-4-carboxamide | Human | 15217 | |
| AURKA (AurA) | Aur | Other | 8jg8 | A | | 4-[5-[3-[bis(oxidanylidene)-$l^5-sulfanyl]oxyphenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-yl]morpholine | Human | 15272 | |
| AURKA (AurA) | Aur | Other | 8jmx | A | | 5-(4-morpholin-4-yl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2-oxidanyl-benzaldehyde | Human | 14864 | |
| AURKA (AurA) | Aur | Other | 8of5 | A | | adenosine-5'-diphosphate | Human | 15218 | |
| AURKA (AurA) | Aur | Other | 8pr7 | A | | adenosine-5'-diphosphate | Human | 15292 | |
| AURKA (AurA) | Aur | Other | 8sso | A | A | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 14866 | |
| AURKA (AurA) | Aur | Other | 8sso | A | B | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 14867 | |
| AURKA (AurA) | Aur | Other | 8sso | A | C | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 14863 | |
| AURKA (AurA) | Aur | Other | 8ssp | A | A | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 14868 | |
| AURKA (AurA) | Aur | Other | 8ssp | A | B | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 14865 | |
| AURKB (AurB) | Aur | Other | 4af3 | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 407 | |
| AURKC (AurC) | Aur | Other | 6gr8 | A | A | 1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)urea | Human | 11122 | |
| AURKC (AurC) | Aur | Other | 6gr8 | A | B | 1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)urea | Human | 11125 | |
| AURKC (AurC) | Aur | Other | 6gr9 | A | A | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 11123 | |
| AURKC (AurC) | Aur | Other | 6gr9 | A | B | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 11124 | |
| AXL | Axl | TK | 5u6b | A | | (10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 8258 | |
| AXL | Axl | TK | 5u6b | B | | (10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 8260 | |
| AXL | Axl | TK | 5u6b | C | | (10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 8257 | |
| AXL | Axl | TK | 5u6b | D | | (10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 8259 | |
| BMP2K (BIKE) | NAK | Other | 4w9w | A | A | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 3274 | |
| BMP2K (BIKE) | NAK | Other | 4w9w | A | B | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 3272 | |
| BMP2K (BIKE) | NAK | Other | 4w9x | A | | baricitinib | Human | 3273 | |
| BMP2K (BIKE) | NAK | Other | 5i3o | A | | n-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamide | Human | 6437 | |
| BMP2K (BIKE) | NAK | Other | 5i3o | B | | n-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamide | Human | 6434 | |
| BMP2K (BIKE) | NAK | Other | 5i3r | A | | n-[6-(3-{[(cyclopropylmethyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]cyclopropanecarboxamide | Human | 6435 | |
| BMP2K (BIKE) | NAK | Other | 5i3r | B | | n-[6-(3-{[(cyclopropylmethyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]cyclopropanecarboxamide | Human | 6436 | |
| BMP2K (BIKE) | NAK | Other | 5ikw | A | | n-(6-{3-[(cyclopropylsulfonyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamide | Human | 6709 | |
| BMPR1B | STKR | TKL | 3mdy | A | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1502 | |
| BMPR1B | STKR | TKL | 3mdy | A | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1501 | |
| BMPR1B | STKR | TKL | 3mdy | C | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1503 | |
| BMPR1B | STKR | TKL | 3mdy | C | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1500 | |
| BMPR2 | STKR | TKL | 3g2f | A | A | adenosine-5'-diphosphate | Human | 6870 | |
| BMPR2 | STKR | TKL | 3g2f | A | B | adenosine-5'-diphosphate | Human | 6868 | |
| BMPR2 | STKR | TKL | 3g2f | B | A | adenosine-5'-diphosphate | Human | 6867 | |
| BMPR2 | STKR | TKL | 3g2f | B | B | adenosine-5'-diphosphate | Human | 6869 | |
| BMPR2 | STKR | TKL | 6unp | A | A | adenosine-5'-diphosphate | Human | 13795 | |
| BMPR2 | STKR | TKL | 6unp | A | B | adenosine-5'-diphosphate | Human | 13794 | |
| BMX | Tec | TK | 3sxr | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 3482 | |
| BMX | Tec | TK | 3sxr | B | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 3481 | |
| BMX | Tec | TK | 3sxs | A | | 1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 3483 | |
| BMX | Tec | TK | 6i99 | A | | ~{n}-[2-methyl-5-[8-[4-(methylsulfonylamino)phenyl]-2-oxidanylidene-benzo[h][1,6]naphthyridin-1-yl]phenyl]-3-oxidanyl-propanamide | Human | 12348 | |
| BMX | Tec | TK | 6i99 | B | | ~{n}-[2-methyl-5-[8-[4-(methylsulfonylamino)phenyl]-2-oxidanylidene-benzo[h][1,6]naphthyridin-1-yl]phenyl]-3-oxidanyl-propanamide | Human | 12349 | |
| BMX | Tec | TK | 8x2a | A | A | 4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamide | Human | 15131 | |
| BMX | Tec | TK | 8x2a | A | B | 4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamide | Human | 15130 | |
| BRAF | RAF | TKL | 1uwh | A | | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 3127 | |
| BRAF | RAF | TKL | 1uwh | B | | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 3109 | |
| BRAF | RAF | TKL | 1uwj | A | | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 3135 | |
| BRAF | RAF | TKL | 1uwj | B | | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 3105 | |
| BRAF | RAF | TKL | 2fb8 | A | | (1z)-5-(2-{4-[2-(dimethylamino)ethoxy]phenyl}-5-pyridin-4-yl-1h-imidazol-4-yl)indan-1-one oxime | Human | 3062 | |
| BRAF | RAF | TKL | 2fb8 | B | | (1z)-5-(2-{4-[2-(dimethylamino)ethoxy]phenyl}-5-pyridin-4-yl-1h-imidazol-4-yl)indan-1-one oxime | Human | 3086 | |
| BRAF | RAF | TKL | 3c4c | A | | n-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamide | Human | 3115 | |
| BRAF | RAF | TKL | 3c4c | B | | n-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamide | Human | 3063 | |
| BRAF | RAF | TKL | 3d4q | A | | (1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oxime | Human | 3095 | |
| BRAF | RAF | TKL | 3d4q | B | | (1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oxime | Human | 3060 | |
| BRAF | RAF | TKL | 3idp | A | | n~1~-(4-chlorophenyl)-6-methyl-n~5~-[3-(7h-purin-6-yl)pyridin-2-yl]isoquinoline-1,5-diamine | Human | 3077 | |
| BRAF | RAF | TKL | 3idp | B | | n~1~-(4-chlorophenyl)-6-methyl-n~5~-[3-(7h-purin-6-yl)pyridin-2-yl]isoquinoline-1,5-diamine | Human | 3121 | |
| BRAF | RAF | TKL | 3ii5 | A | | n-[3-(3-{4-[(dimethylamino)methyl]phenyl}pyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-3-(trifluoromethyl)benzamide | Human | 3116 | |
| BRAF | RAF | TKL | 3ii5 | B | | n-[3-(3-{4-[(dimethylamino)methyl]phenyl}pyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-3-(trifluoromethyl)benzamide | Human | 3076 | |
| BRAF | RAF | TKL | 3og7 | A | | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 3113 | |
| BRAF | RAF | TKL | 3og7 | B | | - | Human | 3140 | |
| BRAF | RAF | TKL | 3ppj | A | | methyl 3-{[(5s)-1-(hydroxyamino)-5h-inden-5-yl]amino}furo[2,3-c]pyridine-2-carboxylate | Human | 3091 | |
| BRAF | RAF | TKL | 3ppj | B | | methyl 3-{[(5s)-1-(hydroxyamino)-5h-inden-5-yl]amino}furo[2,3-c]pyridine-2-carboxylate | Human | 3087 | |
| BRAF | RAF | TKL | 3ppk | A | | 3-[(5-hydroxynaphthalen-2-yl)amino]-n-(pyrimidin-4-yl)furo[2,3-c]pyridine-2-carboxamide | Human | 3106 | |
| BRAF | RAF | TKL | 3ppk | B | | 3-[(5-hydroxynaphthalen-2-yl)amino]-n-(pyrimidin-4-yl)furo[2,3-c]pyridine-2-carboxamide | Human | 3092 | |
| BRAF | RAF | TKL | 3prf | A | | 2-chloro-5-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}phenol | Human | 3129 | |
| BRAF | RAF | TKL | 3prf | B | | 2-chloro-5-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}phenol | Human | 3139 | |
| BRAF | RAF | TKL | 3pri | A | | 3-(4-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}-1h-indazol-3-yl)propan-1-ol | Human | 3093 | |
| BRAF | RAF | TKL | 3pri | B | | 3-(4-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}-1h-indazol-3-yl)propan-1-ol | Human | 3103 | |
| BRAF | RAF | TKL | 3psb | A | | ethyl 3-{[1-(hydroxyamino)-2h-inden-5-yl]amino}thieno[2,3-c]pyridine-2-carboxylate | Human | 3111 | |
| BRAF | RAF | TKL | 3psb | B | | ethyl 3-{[1-(hydroxyamino)-2h-inden-5-yl]amino}thieno[2,3-c]pyridine-2-carboxylate | Human | 3125 | |
| BRAF | RAF | TKL | 3psd | A | | 6-[1-(piperidin-4-yl)-3-(pyridin-4-yl)-1h-pyrazol-4-yl]indeno[1,2-c]pyrazole | Human | 3142 | |
| BRAF | RAF | TKL | 3psd | B | | 6-[1-(piperidin-4-yl)-3-(pyridin-4-yl)-1h-pyrazol-4-yl]indeno[1,2-c]pyrazole | Human | 3083 | |
| BRAF | RAF | TKL | 3q4c | A | | [(1,2,3,4,5,6-eta)-(1s,2r,3r,4r,5s,6s)-1-carboxycyclohexane-1,2,3,4,5,6-hexayl](chloro)(3-methyl-5,7-dioxo-6,7-dihydro-5h-pyrido[2,3-a]pyrrolo[3,4-c]carbazol-12-ide-kappa~2~n~1~,n~12~)ruthenium(1+) | Human | 7251 | |
| BRAF | RAF | TKL | 3q4c | B | | - | Human | 7250 | |
| BRAF | RAF | TKL | 3q96 | A | | (2s)-n-[3-(2-aminopropan-2-yl)-5-(trifluoromethyl)phenyl]-7-[(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-4-yl)oxy]-1,2,3,4-tetrahydronaphthalene-2-carboxamide | Human | 3072 | |
| BRAF | RAF | TKL | 3q96 | B | | (2s)-n-[3-(2-aminopropan-2-yl)-5-(trifluoromethyl)phenyl]-7-[(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-4-yl)oxy]-1,2,3,4-tetrahydronaphthalene-2-carboxamide | Human | 3089 | |
| BRAF | RAF | TKL | 3skc | A | | 2,6-difluoro-n-[(5s)-3-methoxy-5h-pyrazolo[3,4-b]pyridin-5-yl]-3-[(phenylsulfonyl)amino]benzamide | Human | 3100 | |
| BRAF | RAF | TKL | 3skc | B | | 2,6-difluoro-n-[(5s)-3-methoxy-5h-pyrazolo[3,4-b]pyridin-5-yl]-3-[(phenylsulfonyl)amino]benzamide | Human | 3128 | |
| BRAF | RAF | TKL | 3tv4 | A | | n-(6-amino-5-bromopyridin-3-yl)-2,6-difluoro-3-[(propylsulfonyl)amino]benzamide | Human | 3054 | |
| BRAF | RAF | TKL | 3tv4 | B | | n-(6-amino-5-bromopyridin-3-yl)-2,6-difluoro-3-[(propylsulfonyl)amino]benzamide | Human | 3133 | |
| BRAF | RAF | TKL | 3tv6 | A | | 2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)-3-[(propylsulfonyl)amino]benzamide | Human | 3080 | |
| BRAF | RAF | TKL | 3tv6 | B | | 2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)-3-[(propylsulfonyl)amino]benzamide | Human | 3136 | |
| BRAF | RAF | TKL | 4cqe | A | | n-{4-[2-(1-cyclopropylpiperidin-4-yl)-4-(3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)-1,3-thiazol-5-yl]pyridin-2-yl}acetamide | Human | 3088 | |
| BRAF | RAF | TKL | 4cqe | B | | n-{4-[2-(1-cyclopropylpiperidin-4-yl)-4-(3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)-1,3-thiazol-5-yl]pyridin-2-yl}acetamide | Human | 3107 | |
| BRAF | RAF | TKL | 4dbn | A | | 2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamide | Human | 3052 | |
| BRAF | RAF | TKL | 4dbn | B | | 2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamide | Human | 3070 | |
| BRAF | RAF | TKL | 4e26 | A | | 5-chloro-7-[(r)-furan-2-yl(pyridin-2-ylamino)methyl]quinolin-8-ol | Human | 3108 | |
| BRAF | RAF | TKL | 4e26 | B | | 5-chloro-7-[(r)-furan-2-yl(pyridin-2-ylamino)methyl]quinolin-8-ol | Human | 3102 | |
| BRAF | RAF | TKL | 4e4x | A | | n-(2,4-difluoro-3-{2-[(3-hydroxypropyl)amino]-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl}phenyl)propane-1-sulfonamide | Human | 3051 | |
| BRAF | RAF | TKL | 4e4x | B | | n-(2,4-difluoro-3-{2-[(3-hydroxypropyl)amino]-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl}phenyl)propane-1-sulfonamide | Human | 3104 | |
| BRAF | RAF | TKL | 4ehe | A | | 4-amino-n-{2,6-difluoro-3-[(propylsulfonyl)amino]phenyl}thieno[3,2-d]pyrimidine-7-carboxamide | Human | 3112 | |
| BRAF | RAF | TKL | 4ehe | B | | 4-amino-n-{2,6-difluoro-3-[(propylsulfonyl)amino]phenyl}thieno[3,2-d]pyrimidine-7-carboxamide | Human | 3082 | |
| BRAF | RAF | TKL | 4ehg | A | | n-{2,4-difluoro-3-[({6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}carbamoyl)amino]phenyl}propane-1-sulfonamide | Human | 3064 | |
| BRAF | RAF | TKL | 4ehg | B | | n-{2,4-difluoro-3-[({6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}carbamoyl)amino]phenyl}propane-1-sulfonamide | Human | 3078 | |
| BRAF | RAF | TKL | 4fc0 | A | | 2-chloro-3-[(2-cyanopropan-2-yl)oxy]-n-{5-[{2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}(methyl)amino]-2-fluorophenyl}benzamide | Human | 3131 | |
| BRAF | RAF | TKL | 4fc0 | B | | 2-chloro-3-[(2-cyanopropan-2-yl)oxy]-n-{5-[{2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}(methyl)amino]-2-fluorophenyl}benzamide | Human | 3069 | |
| BRAF | RAF | TKL | 4fk3 | A | | n-{2,4-difluoro-3-[(5-pyridin-3-yl-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]phenyl}ethanesulfonamide | Human | 3118 | |
| BRAF | RAF | TKL | 4fk3 | B | | - | Human | 3068 | |
| BRAF | RAF | TKL | 4g9c | A | | 3-{[3-(2-cyanopropan-2-yl)benzoyl]amino}-2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)benzamide | Human | 3084 | |
| BRAF | RAF | TKL | 4g9c | B | | 3-{[3-(2-cyanopropan-2-yl)benzoyl]amino}-2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)benzamide | Human | 3067 | |
| BRAF | RAF | TKL | 4g9r | A | | 3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamide | Human | 3130 | |
| BRAF | RAF | TKL | 4g9r | B | | 3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamide | Human | 3101 | |
| BRAF | RAF | TKL | 4h58 | A | A | n-(4-{[(2-methoxyethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)quinazolin-2-amine | Human | 3137 | |
| BRAF | RAF | TKL | 4h58 | A | B | n-(4-{[(2-methoxyethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)quinazolin-2-amine | Human | 3110 | |
| BRAF | RAF | TKL | 4h58 | B | A | - | Human | 3097 | |
| BRAF | RAF | TKL | 4h58 | B | B | - | Human | 3120 | |
| BRAF | RAF | TKL | 4h58 | C | A | - | Human | 3056 | |
| BRAF | RAF | TKL | 4h58 | C | B | - | Human | 3114 | |
| BRAF | RAF | TKL | 4jvg | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 3134 | |
| BRAF | RAF | TKL | 4jvg | B | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 3085 | |
| BRAF | RAF | TKL | 4jvg | C | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 3050 | |
| BRAF | RAF | TKL | 4jvg | D | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 3059 | |
| BRAF | RAF | TKL | 4ksp | A | | n-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]acetyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide | Human | 3081 | |
| BRAF | RAF | TKL | 4ksp | B | | n-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]acetyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide | Human | 3066 | |
| BRAF | RAF | TKL | 4ksq | A | | n-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide | Human | 3065 | |
| BRAF | RAF | TKL | 4ksq | B | | n-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamide | Human | 3055 | |
| BRAF | RAF | TKL | 4mbj | A | | 2,6-difluoro-n-(1h-imidazo[4,5-b]pyridin-6-yl)-3-[(propylsulfonyl)amino]benzamide | Human | 3090 | |
| BRAF | RAF | TKL | 4mbj | B | | 2,6-difluoro-n-(1h-imidazo[4,5-b]pyridin-6-yl)-3-[(propylsulfonyl)amino]benzamide | Human | 3057 | |
| BRAF | RAF | TKL | 4mne | B | A | - | Human | 3075 | |
| BRAF | RAF | TKL | 4mne | B | B | - | Human | 3061 | |
| BRAF | RAF | TKL | 4mne | C | A | - | Human | 3122 | |
| BRAF | RAF | TKL | 4mne | C | B | - | Human | 3058 | |
| BRAF | RAF | TKL | 4mne | F | A | - | Human | 3099 | |
| BRAF | RAF | TKL | 4mne | F | B | - | Human | 3117 | |
| BRAF | RAF | TKL | 4mne | G | A | - | Human | 3071 | |
| BRAF | RAF | TKL | 4mne | G | B | - | Human | 3073 | |
| BRAF | RAF | TKL | 4mnf | A | A | 2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanol | Human | 3096 | |
| BRAF | RAF | TKL | 4mnf | A | B | 2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanol | Human | 3141 | |
| BRAF | RAF | TKL | 4mnf | B | A | 2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanol | Human | 3124 | |
| BRAF | RAF | TKL | 4mnf | B | B | 2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanol | Human | 3098 | |
| BRAF | RAF | TKL | 4pp7 | A | | n-{2,4-difluoro-3-[methyl(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamide | Human | 3094 | |
| BRAF | RAF | TKL | 4pp7 | B | | n-{2,4-difluoro-3-[methyl(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamide | Human | 3126 | |
| BRAF | RAF | TKL | 4r5y | A | | 5-({(1r,1as,6br)-1-[5-(trifluoromethyl)-1h-benzimidazol-2-yl]-1a,6b-dihydro-1h-cyclopropa[b][1]benzofuran-5-yl}oxy)-3,4-dihydro-1,8-naphthyridin-2(1h)-one | Human | 6414 | |
| BRAF | RAF | TKL | 4r5y | B | | 5-({(1r,1as,6br)-1-[5-(trifluoromethyl)-1h-benzimidazol-2-yl]-1a,6b-dihydro-1h-cyclopropa[b][1]benzofuran-5-yl}oxy)-3,4-dihydro-1,8-naphthyridin-2(1h)-one | Human | 6413 | |
| BRAF | RAF | TKL | 4rzv | A | | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6944 | |
| BRAF | RAF | TKL | 4rzv | B | | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6941 | |
| BRAF | RAF | TKL | 4rzw | A | | 3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamide | Human | 6939 | |
| BRAF | RAF | TKL | 4rzw | B | | 3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamide | Human | 6942 | |
| BRAF | RAF | TKL | 4wo5 | A | | n-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamide | Human | 3079 | |
| BRAF | RAF | TKL | 4wo5 | B | | n-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamide | Human | 3143 | |
| BRAF | RAF | TKL | 4xv1 | A | | n'-(3-{[5-(2-cyclopropylpyrimidin-5-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)-n-ethyl-n-methylsulfuric diamide | Human | 6214 | |
| BRAF | RAF | TKL | 4xv1 | B | | - | Human | 6216 | |
| BRAF | RAF | TKL | 4xv2 | A | | dabrafenib | Human | 6213 | |
| BRAF | RAF | TKL | 4xv2 | B | | dabrafenib | Human | 6219 | |
| BRAF | RAF | TKL | 4xv3 | A | | n'-{3-[5-(2-aminopyrimidin-4-yl)-2-tert-butyl-1,3-thiazol-4-yl]-2-fluorophenyl}-n-ethyl-n-methylsulfuric diamide | Human | 6217 | |
| BRAF | RAF | TKL | 4xv3 | B | | - | Human | 6218 | |
| BRAF | RAF | TKL | 4xv9 | A | A | n-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}-4-(trifluoromethyl)benzenesulfonamide | Human | 6220 | |
| BRAF | RAF | TKL | 4xv9 | A | B | n-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}-4-(trifluoromethyl)benzenesulfonamide | Human | 6215 | |
| BRAF | RAF | TKL | 4yht | A | | 3-[(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6442 | |
| BRAF | RAF | TKL | 4yht | B | | 3-[(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6443 | |
| BRAF | RAF | TKL | 5c9c | A | A | 1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}urea | Human | 3123 | |
| BRAF | RAF | TKL | 5c9c | A | B | 1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}urea | Human | 3074 | |
| BRAF | RAF | TKL | 5c9c | B | A | 1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}urea | Human | 3138 | |
| BRAF | RAF | TKL | 5c9c | B | B | 1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}urea | Human | 3119 | |
| BRAF | RAF | TKL | 5csw | A | | dabrafenib | Human | 6433 | |
| BRAF | RAF | TKL | 5csw | B | | dabrafenib | Human | 6431 | |
| BRAF | RAF | TKL | 5csx | A | | n-(3-{5-[(1-ethylpiperidin-4-yl)(methyl)amino]-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-1-yl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6432 | |
| BRAF | RAF | TKL | 5ct7 | A | | 1-methyl-5-({2-[5-(trifluoromethyl)-1h-imidazol-2-yl]pyridin-4-yl}oxy)-n-[4-(trifluoromethyl)phenyl]-1h-benzimidazol-2-amine | Human | 6032 | |
| BRAF | RAF | TKL | 5ct7 | B | | 1-methyl-5-({2-[5-(trifluoromethyl)-1h-imidazol-2-yl]pyridin-4-yl}oxy)-n-[4-(trifluoromethyl)phenyl]-1h-benzimidazol-2-amine | Human | 6033 | |
| BRAF | RAF | TKL | 5fd2 | A | | 6-[2-[[3-(dimethylsulfamoylamino)-2,6-bis(fluoranyl)phenyl]amino]pyridin-3-yl]-7~{h}-purine | Human | 6603 | |
| BRAF | RAF | TKL | 5fd2 | B | | 6-[2-[[3-(dimethylsulfamoylamino)-2,6-bis(fluoranyl)phenyl]amino]pyridin-3-yl]-7~{h}-purine | Human | 6602 | |
| BRAF | RAF | TKL | 5hi2 | A | | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 6515 | |
| BRAF | RAF | TKL | 5hid | A | A | 3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamide | Human | 6506 | |
| BRAF | RAF | TKL | 5hid | A | B | 3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamide | Human | 6512 | |
| BRAF | RAF | TKL | 5hid | B | A | 3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamide | Human | 6511 | |
| BRAF | RAF | TKL | 5hid | B | B | 3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamide | Human | 6517 | |
| BRAF | RAF | TKL | 5hie | A | A | dabrafenib | Human | 6516 | |
| BRAF | RAF | TKL | 5hie | A | B | dabrafenib | Human | 6508 | |
| BRAF | RAF | TKL | 5hie | B | A | dabrafenib | Human | 6509 | |
| BRAF | RAF | TKL | 5hie | B | B | dabrafenib | Human | 6505 | |
| BRAF | RAF | TKL | 5hie | C | A | dabrafenib | Human | 6513 | |
| BRAF | RAF | TKL | 5hie | C | B | dabrafenib | Human | 6507 | |
| BRAF | RAF | TKL | 5hie | D | A | dabrafenib | Human | 6510 | |
| BRAF | RAF | TKL | 5hie | D | B | dabrafenib | Human | 6514 | |
| BRAF | RAF | TKL | 5ita | A | | n-{2-cyano-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamide | Human | 6940 | |
| BRAF | RAF | TKL | 5ita | B | | n-{2-cyano-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamide | Human | 6943 | |
| BRAF | RAF | TKL | 5jrq | A | | (3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)[5-(4-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methanone | Human | 7061 | |
| BRAF | RAF | TKL | 5jrq | B | | (3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)[5-(4-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methanone | Human | 7054 | |
| BRAF | RAF | TKL | 5jsm | A | A | - | Human | 7056 | |
| BRAF | RAF | TKL | 5jsm | A | B | - | Human | 7058 | |
| BRAF | RAF | TKL | 5jsm | B | A | n,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide) | Human | 7060 | |
| BRAF | RAF | TKL | 5jsm | B | B | n,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide) | Human | 7062 | |
| BRAF | RAF | TKL | 5jsm | C | A | n,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide) | Human | 7059 | |
| BRAF | RAF | TKL | 5jsm | C | B | n,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide) | Human | 7063 | |
| BRAF | RAF | TKL | 5jsm | D | A | - | Human | 7055 | |
| BRAF | RAF | TKL | 5jsm | D | B | - | Human | 7053 | |
| BRAF | RAF | TKL | 5jt2 | A | | 2,2'-oxybis[n-({4-[3-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorobenzene-1-carbonyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]phenyl}methyl)acetamide] | Human | 7065 | |
| BRAF | RAF | TKL | 5jt2 | B | | - | Human | 7057 | |
| BRAF | RAF | TKL | 5jt2 | C | | 2,2'-oxybis[n-({4-[3-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorobenzene-1-carbonyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]phenyl}methyl)acetamide] | Human | 7064 | |
| BRAF | RAF | TKL | 5jt2 | D | | - | Human | 7066 | |
| BRAF | RAF | TKL | 5val | A | | n-(3-tert-butylphenyl)-4-methyl-3-[6-(morpholin-4-yl)pyrimidin-4-yl]benzamide | Human | 8190 | |
| BRAF | RAF | TKL | 5val | B | | n-(3-tert-butylphenyl)-4-methyl-3-[6-(morpholin-4-yl)pyrimidin-4-yl]benzamide | Human | 8188 | |
| BRAF | RAF | TKL | 5vam | A | A | n-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamide | Human | 8185 | |
| BRAF | RAF | TKL | 5vam | A | B | n-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamide | Human | 8189 | |
| BRAF | RAF | TKL | 5vam | B | A | n-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamide | Human | 8186 | |
| BRAF | RAF | TKL | 5vam | B | B | n-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamide | Human | 8187 | |
| BRAF | RAF | TKL | 6b8u | A | | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | 8679 | |
| BRAF | RAF | TKL | 6b8u | B | | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | 8678 | |
| BRAF | RAF | TKL | 6cad | A | | 1-(propan-2-yl)-3-({3-[3-(trifluoromethyl)phenyl]isoquinolin-8-yl}ethynyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 9576 | |
| BRAF | RAF | TKL | 6cad | B | | 1-(propan-2-yl)-3-({3-[3-(trifluoromethyl)phenyl]isoquinolin-8-yl}ethynyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 9575 | |
| BRAF | RAF | TKL | 6n0p | A | A | n-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamide | Human | 11597 | |
| BRAF | RAF | TKL | 6n0p | A | B | n-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamide | Human | 11596 | |
| BRAF | RAF | TKL | 6n0p | B | A | n-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamide | Human | 11594 | |
| BRAF | RAF | TKL | 6n0p | B | B | n-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamide | Human | 11595 | |
| BRAF | RAF | TKL | 6n0q | A | A | n-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamide | Human | 11771 | |
| BRAF | RAF | TKL | 6n0q | A | B | n-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamide | Human | 11768 | |
| BRAF | RAF | TKL | 6n0q | B | A | n-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamide | Human | 11770 | |
| BRAF | RAF | TKL | 6n0q | B | B | n-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamide | Human | 11769 | |
| BRAF | RAF | TKL | 6nsq | A | | 5-[(4-amino-1-ethyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-n-(4-chlorophenyl)-6-methylisoquinolin-1-amine | Human | 11328 | |
| BRAF | RAF | TKL | 6nsq | B | | 5-[(4-amino-1-ethyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-n-(4-chlorophenyl)-6-methylisoquinolin-1-amine | Human | 11329 | |
| BRAF | RAF | TKL | 6nyb | A | | phosphothiophosphoric acid-adenylate ester | Human | 11708 | |
| BRAF | RAF | TKL | 6p3d | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 12809 | |
| BRAF | RAF | TKL | 6p7g | A | | 3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamide | Human | 12810 | |
| BRAF | RAF | TKL | 6p7g | B | | 3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamide | Human | 12806 | |
| BRAF | RAF | TKL | 6p7g | C | | 3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamide | Human | 12807 | |
| BRAF | RAF | TKL | 6p7g | D | | 3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamide | Human | 12808 | |
| BRAF | RAF | TKL | 6pp9 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 11711 | |
| BRAF | RAF | TKL | 6pp9 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 11709 | |
| BRAF | RAF | TKL | 6q0j | A | A | - | Human | 11704 | |
| BRAF | RAF | TKL | 6q0j | A | B | - | Human | 11701 | |
| BRAF | RAF | TKL | 6q0j | B | A | - | Human | 11703 | |
| BRAF | RAF | TKL | 6q0j | B | B | - | Human | 11712 | |
| BRAF | RAF | TKL | 6q0k | A | | - | Human | 11706 | |
| BRAF | RAF | TKL | 6q0k | B | | - | Human | 11710 | |
| BRAF | RAF | TKL | 6q0t | A | A | - | Human | 11705 | |
| BRAF | RAF | TKL | 6q0t | A | B | - | Human | 11707 | |
| BRAF | RAF | TKL | 6q0t | B | A | - | Human | 11702 | |
| BRAF | RAF | TKL | 6q0t | B | B | - | Human | 11700 | |
| BRAF | RAF | TKL | 6u2g | B | | phosphomethylphosphonic acid adenylate ester | Human | 11567 | |
| BRAF | RAF | TKL | 6u2h | C | A | 2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanol | Human | 11568 | |
| BRAF | RAF | TKL | 6u2h | D | A | 2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanol | Human | 11569 | |
| BRAF | RAF | TKL | 6uan | B | | - | Human | 11641 | |
| BRAF | RAF | TKL | 6uan | C | | - | Human | 11642 | |
| BRAF | RAF | TKL | 6uuo | A | | 1-[4-{[1-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-5-yl](methyl)amino}pyridin-1(4h)-yl]ethan-1-one | Human | 12347 | |
| BRAF | RAF | TKL | 6uuo | B | | 1-[4-{[1-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-5-yl](methyl)amino}pyridin-1(4h)-yl]ethan-1-one | Human | 12346 | |
| BRAF | RAF | TKL | 6v2u | A | | dabrafenib | Human | 13034 | |
| BRAF | RAF | TKL | 6v2u | B | | dabrafenib | Human | 13031 | |
| BRAF | RAF | TKL | 6v2w | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 13026 | |
| BRAF | RAF | TKL | 6v2w | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 13032 | |
| BRAF | RAF | TKL | 6v34 | A | | 6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide | Human | 13200 | |
| BRAF | RAF | TKL | 6v34 | B | | 6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide | Human | 13199 | |
| BRAF | RAF | TKL | 6xag | C | A | - | Human | 12922 | |
| BRAF | RAF | TKL | 6xag | D | A | - | Human | 12921 | |
| BRAF | RAF | TKL | 6xfp | A | A | 4-amino-n-{1-[(3-chloro-2-fluorophenyl)amino]-6-methylisoquinolin-5-yl}thieno[3,2-d]pyrimidine-7-carboxamide | Human | 13403 | |
| BRAF | RAF | TKL | 6xfp | A | B | 4-amino-n-{1-[(3-chloro-2-fluorophenyl)amino]-6-methylisoquinolin-5-yl}thieno[3,2-d]pyrimidine-7-carboxamide | Human | 13404 | |
| BRAF | RAF | TKL | 6xlo | A | | 3-(2-cyanopropan-2-yl)-n-[2-fluoro-4-methyl-5-(7-methyl-8-oxo-7,8-dihydropyrido[2,3-d]pyridazin-3-yl)phenyl]benzamide | Human | 13618 | |
| BRAF | RAF | TKL | 7k0v | A | A | n-(3,3-dimethylbutyl)-n'-{2-fluoro-5-[(5-fluoro-3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]-4-methylphenyl}urea | Human | 13617 | |
| BRAF | RAF | TKL | 7k0v | A | B | n-(3,3-dimethylbutyl)-n'-{2-fluoro-5-[(5-fluoro-3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]-4-methylphenyl}urea | Human | 13616 | |
| BRAF | RAF | TKL | 7m0t | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13525 | |
| BRAF | RAF | TKL | 7m0u | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13527 | |
| BRAF | RAF | TKL | 7m0v | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 13526 | |
| BRAF | RAF | TKL | 7m0v | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 13522 | |
| BRAF | RAF | TKL | 7m0w | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13528 | |
| BRAF | RAF | TKL | 7m0x | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 13524 | |
| BRAF | RAF | TKL | 7m0x | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 13523 | |
| BRAF | RAF | TKL | 7m0y | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13520 | |
| BRAF | RAF | TKL | 7m0z | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13521 | |
| BRAF | RAF | TKL | 7mfd | A | | - | Human | 14077 | |
| BRAF | RAF | TKL | 7mfe | A | | - | Human | 14078 | |
| BRAF | RAF | TKL | 7p3v | A | | ~{n}-[3-[5-(2-azanylpyrimidin-4-yl)-2-[(3~{s})-morpholin-3-yl]-1,3-thiazol-4-yl]-2-fluoranyl-phenyl]-2,5-bis(fluoranyl)benzenesulfonamide | Human | 13961 | |
| BRAF | RAF | TKL | 7shv | A | A | 2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanol | Human | 14482 | |
| BRAF | RAF | TKL | 7shv | A | B | 2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanol | Human | 14481 | |
| BRAF | RAF | TKL | 8c7x | A | A | ~{n}-[3-[(5-chloranyl-1~{h}-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-bis(fluoranyl)phenyl]-3-(2-cyanopropan-2-yl)benzamide | Human | 14630 | |
| BRAF | RAF | TKL | 8c7x | A | B | ~{n}-[3-[(5-chloranyl-1~{h}-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-bis(fluoranyl)phenyl]-3-(2-cyanopropan-2-yl)benzamide | Human | 14627 | |
| BRAF | RAF | TKL | 8c7y | A | A | ~{n}-[3-[(5-chloranyl-1~{h}-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-bis(fluoranyl)phenyl]-3-(2-cyanopropan-2-yl)benzamide | Human | 14629 | |
| BRAF | RAF | TKL | 8c7y | A | B | ~{n}-[3-[(5-chloranyl-1~{h}-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-bis(fluoranyl)phenyl]-3-(2-cyanopropan-2-yl)benzamide | Human | 14628 | |
| BRAF | RAF | TKL | 8dgs | A | A | phosphothiophosphoric acid-adenylate ester | Human | 14831 | |
| BRAF | RAF | TKL | 8dgs | A | B | phosphothiophosphoric acid-adenylate ester | Human | 14829 | |
| BRAF | RAF | TKL | 8dgt | A | A | phosphothiophosphoric acid-adenylate ester | Human | 14832 | |
| BRAF | RAF | TKL | 8dgt | A | B | phosphothiophosphoric acid-adenylate ester | Human | 14830 | |
| BRAF | RAF | TKL | 8f7o | A | A | 6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide | Human | 14704 | |
| BRAF | RAF | TKL | 8f7o | A | B | 6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamide | Human | 14703 | |
| BRAF | RAF | TKL | 8f7p | A | A | n-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamide | Human | 14705 | |
| BRAF | RAF | TKL | 8f7p | A | B | n-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamide | Human | 14702 | |
| BRAF | RAF | TKL | 8qqg | A | A | (3~{s})-~{n}-[4-methyl-3-[2-morpholin-4-yl-6-[[(2~{r})-1-oxidanylpropan-2-yl]amino]pyridin-4-yl]phenyl]-3-[2,2,2-tris(fluoranyl)ethyl]pyrrolidine-1-carboxamide | Human | 15178 | |
| BRAF | RAF | TKL | 8qqg | A | B | (3~{s})-~{n}-[4-methyl-3-[2-morpholin-4-yl-6-[[(2~{r})-1-oxidanylpropan-2-yl]amino]pyridin-4-yl]phenyl]-3-[2,2,2-tris(fluoranyl)ethyl]pyrrolidine-1-carboxamide | Human | 15179 | |
| BRAF | RAF | TKL | 9bfb | A | A | n-{2-chloro-3-[(3,5-dimethyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]-4-fluorophenyl}-3-fluoropropane-1-sulfonamide | Human | 15365 | |
| BRAF | RAF | TKL | 9bfb | A | B | n-{2-chloro-3-[(3,5-dimethyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]-4-fluorophenyl}-3-fluoropropane-1-sulfonamide | Human | 15366 | |
| Brsk2 (BRSK2) | CAMKL | CAMK | 4ynz | A | | - | Mouse | 6293 | |
| Brsk2 (BRSK2) | CAMKL | CAMK | 4ynz | B | | - | Mouse | 6291 | |
| Brsk2 (BRSK2) | CAMKL | CAMK | 4yom | B | | - | Mouse | 6292 | |
| Btk (BTK) | Tec | TK | 4xi2 | A | | - | Mouse | 5815 | |
| Btk (BTK) | Tec | TK | 6mny | A | A | 5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamide | Mouse | 11307 | |
| Btk (BTK) | Tec | TK | 6mny | A | B | 5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamide | Mouse | 11308 | |
| Btk (BTK) | Tec | TK | 6mny | B | A | - | Mouse | 11306 | |
| Btk (BTK) | Tec | TK | 6mny | B | B | - | Mouse | 11309 | |
| Btk (BTK) | Tec | TK | 8fd9 | A | A | acalabrutinib | Mouse | 14836 | |
| Btk (BTK) | Tec | TK | 8fd9 | A | B | acalabrutinib | Mouse | 14835 | |
| Btk (BTK) | Tec | TK | 8ff0 | A | | 6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-one | Mouse | 14834 | |
| Btk (BTK) | Tec | TK | 8gmb | A | | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | 14999 | |
| Btk (BTK) | Tec | TK | 8s93 | A | A | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | 14997 | |
| Btk (BTK) | Tec | TK | 8s93 | A | B | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | 14996 | |
| Btk (BTK) | Tec | TK | 8s9f | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 14998 | |
| BTK | Tec | TK | 1k2p | A | | - | Human | 2918 | |
| BTK | Tec | TK | 1k2p | B | | - | Human | 2919 | |
| BTK | Tec | TK | 3gen | A | A | 4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentane | Human | 2928 | |
| BTK | Tec | TK | 3gen | A | B | 4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentane | Human | 2900 | |
| BTK | Tec | TK | 3k54 | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 2932 | |
| BTK | Tec | TK | 3k54 | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 2906 | |
| BTK | Tec | TK | 3ocs | A | | 4-tert-butyl-n-[2-methyl-3-(4-methyl-6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-5-oxo-4,5-dihydropyrazin-2-yl)phenyl]benzamide | Human | 2907 | |
| BTK | Tec | TK | 3oct | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 2899 | |
| BTK | Tec | TK | 3oct | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 2908 | |
| BTK | Tec | TK | 3p08 | A | | - | Human | 2905 | |
| BTK | Tec | TK | 3p08 | B | | - | Human | 2894 | |
| BTK | Tec | TK | 3pix | A | | 7-(4-methylpiperazin-1-yl)-4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-(propan-2-yl)phthalazin-1(2h)-one | Human | 2927 | |
| BTK | Tec | TK | 3piy | A | | 6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-one | Human | 2909 | |
| BTK | Tec | TK | 3piz | A | | [5-amino-1-(2-methylphenyl)-1h-pyrazol-4-yl]{3-[1-(methylsulfonyl)piperidin-4-yl]phenyl}methanone | Human | 2922 | |
| BTK | Tec | TK | 3pj1 | A | | 3-(2,6-dichlorophenyl)-7-({4-[2-(diethylamino)ethoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 2904 | |
| BTK | Tec | TK | 3pj2 | A | | 2-({4-[2-(diethylamino)ethoxy]phenyl}amino)-6-(4-fluorophenoxy)-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 2911 | |
| BTK | Tec | TK | 3pj3 | A | | 2-methyl-n-(2-phenyl-3h-imidazo[4,5-b]pyridin-6-yl)-5-{[(2e)-3-phenylprop-2-enoyl]amino}benzamide | Human | 2910 | |
| BTK | Tec | TK | 4nwm | A | A | 4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamide | Human | 2930 | |
| BTK | Tec | TK | 4nwm | A | B | 4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamide | Human | 2917 | |
| BTK | Tec | TK | 4nwm | B | A | 4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamide | Human | 2898 | |
| BTK | Tec | TK | 4nwm | B | B | 4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamide | Human | 2903 | |
| BTK | Tec | TK | 4ot5 | A | | 4-tert-butyl-n-{3-[8-({4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}amino)imidazo[1,2-a]pyrazin-6-yl]phenyl}benzamide | Human | 2913 | |
| BTK | Tec | TK | 4ot6 | A | | 4-(methylsulfonyl)-n-[3-(8-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}imidazo[1,2-a]pyrazin-6-yl)phenyl]benzamide | Human | 2931 | |
| BTK | Tec | TK | 4otf | A | A | n-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | Human | 2901 | |
| BTK | Tec | TK | 4otf | A | B | n-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | Human | 2921 | |
| BTK | Tec | TK | 4otq | A | | 1-{5-[3-(7-tert-butyl-4-oxoquinazolin-3(4h)-yl)-2-methylphenyl]-1-methyl-2-oxo-1,2-dihydropyridin-3-yl}-3-methylurea | Human | 2895 | |
| BTK | Tec | TK | 4otr | A | | 6-cyclopropyl-2-[3-(5-{[5-(4-ethylpiperazin-1-yl)pyridin-2-yl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-(hydroxymethyl)phenyl]-8-fluoroisoquinolin-1(2h)-one | Human | 2896 | |
| BTK | Tec | TK | 4rfy | A | A | 6-(dimethylamino)-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]-3,4-dihydroisoquinolin-1(2h)-one | Human | 2935 | |
| BTK | Tec | TK | 4rfy | A | B | 6-(dimethylamino)-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]-3,4-dihydroisoquinolin-1(2h)-one | Human | 2933 | |
| BTK | Tec | TK | 4rfz | A | | 6-(dimethylamino)-8-fluoro-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]isoquinolin-1(2h)-one | Human | 2925 | |
| BTK | Tec | TK | 4rg0 | A | | 2-{8-fluoro-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]-1-oxo-1,2,3,4-tetrahydroisoquinolin-6-yl}-2-methylpropanenitrile | Human | 2929 | |
| BTK | Tec | TK | 4rx5 | A | A | n-(6-fluoro-2-methyl-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl)-1-benzothiophene-2-carboxamide | Human | 6259 | |
| BTK | Tec | TK | 4rx5 | A | B | n-(6-fluoro-2-methyl-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl)-1-benzothiophene-2-carboxamide | Human | 6258 | |
| BTK | Tec | TK | 4yhf | A | A | (2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrile | Human | 2916 | |
| BTK | Tec | TK | 4yhf | A | B | (2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrile | Human | 2902 | |
| BTK | Tec | TK | 4yhf | B | A | (2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrile | Human | 2897 | |
| BTK | Tec | TK | 4yhf | B | B | (2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrile | Human | 2912 | |
| BTK | Tec | TK | 4z3v | A | A | 4-amino-8-(5-methyl-1h-indazol-6-yl)cinnoline-3-carboxamide | Human | 2934 | |
| BTK | Tec | TK | 4z3v | A | B | 4-amino-8-(5-methyl-1h-indazol-6-yl)cinnoline-3-carboxamide | Human | 2914 | |
| BTK | Tec | TK | 4zly | A | A | 4-aminocinnoline-3-carboxamide | Human | 2926 | |
| BTK | Tec | TK | 4zly | A | B | 4-aminocinnoline-3-carboxamide | Human | 2920 | |
| BTK | Tec | TK | 4zly | A | C | 4-aminocinnoline-3-carboxamide | Human | 2915 | |
| BTK | Tec | TK | 4zlz | A | A | 4-amino-8-(4-methylpyridin-3-yl)cinnoline-3-carboxamide | Human | 2923 | |
| BTK | Tec | TK | 4zlz | A | B | 4-amino-8-(4-methylpyridin-3-yl)cinnoline-3-carboxamide | Human | 2924 | |
| BTK | Tec | TK | 5bpy | A | | 6-{(3r)-3-[(4-tert-butylbenzoyl)amino]piperidin-1-yl}-2-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}pyridine-3-carboxamide | Human | 6095 | |
| BTK | Tec | TK | 5bpy | B | | 6-{(3r)-3-[(4-tert-butylbenzoyl)amino]piperidin-1-yl}-2-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}pyridine-3-carboxamide | Human | 6094 | |
| BTK | Tec | TK | 5bq0 | A | A | 4-(2-chlorophenyl)-7-[(4-methylpiperazin-1-yl)carbonyl]-9h-carbazole-1-carboxamide | Human | 6871 | |
| BTK | Tec | TK | 5bq0 | A | B | 4-(2-chlorophenyl)-7-[(4-methylpiperazin-1-yl)carbonyl]-9h-carbazole-1-carboxamide | Human | 6872 | |
| BTK | Tec | TK | 5fbn | C | A | 4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 6381 | |
| BTK | Tec | TK | 5fbn | C | B | 4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 6382 | |
| BTK | Tec | TK | 5fbn | D | A | 4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 6384 | |
| BTK | Tec | TK | 5fbn | D | B | 4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 6383 | |
| BTK | Tec | TK | 5fbo | A | A | 4-[8-azanyl-3-[(3~{r},6~{s})-1-cyclopropylcarbonyl-6-methyl-piperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoranyl-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 6455 | |
| BTK | Tec | TK | 5fbo | A | B | 4-[8-azanyl-3-[(3~{r},6~{s})-1-cyclopropylcarbonyl-6-methyl-piperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoranyl-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 6456 | |
| BTK | Tec | TK | 5j87 | A | A | n-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 8002 | |
| BTK | Tec | TK | 5j87 | A | B | n-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 8003 | |
| BTK | Tec | TK | 5j87 | B | A | n-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 8005 | |
| BTK | Tec | TK | 5j87 | B | B | n-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 8007 | |
| BTK | Tec | TK | 5j87 | C | A | n-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 8004 | |
| BTK | Tec | TK | 5j87 | C | B | n-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 8006 | |
| BTK | Tec | TK | 5j87 | D | A | n-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 8008 | |
| BTK | Tec | TK | 5j87 | D | B | n-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 8001 | |
| BTK | Tec | TK | 5jrs | A | | 4-[2-fluoro-3-(4-oxoquinazolin-3(4h)-yl)phenyl]-7-(2-hydroxypropan-2-yl)-9h-carbazole-1-carboxamide | Human | 7032 | |
| BTK | Tec | TK | 5jrs | B | | 4-[2-fluoro-3-(4-oxoquinazolin-3(4h)-yl)phenyl]-7-(2-hydroxypropan-2-yl)-9h-carbazole-1-carboxamide | Human | 7033 | |
| BTK | Tec | TK | 5kup | A | A | 6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-6-oxidanylidene-5-(pyrimidin-4-ylamino)pyridin-3-yl]pyridin-2-yl]phthalazin-1-one | Human | 7051 | |
| BTK | Tec | TK | 5kup | A | B | 6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-6-oxidanylidene-5-(pyrimidin-4-ylamino)pyridin-3-yl]pyridin-2-yl]phthalazin-1-one | Human | 7052 | |
| BTK | Tec | TK | 5p9f | A | A | n-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | Human | 7632 | |
| BTK | Tec | TK | 5p9f | A | B | n-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | Human | 7629 | |
| BTK | Tec | TK | 5p9g | A | A | 6-cyclopropyl-8-fluoranyl-2-[2-(hydroxymethyl)-3-[1-methyl-5-[[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridin-3-yl]phenyl]isoquinolin-1-one | Human | 7635 | |
| BTK | Tec | TK | 5p9g | A | B | 6-cyclopropyl-8-fluoranyl-2-[2-(hydroxymethyl)-3-[1-methyl-5-[[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridin-3-yl]phenyl]isoquinolin-1-one | Human | 7644 | |
| BTK | Tec | TK | 5p9h | A | A | 6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-5-[[5-(1-methylpiperidin-4-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridazin-3-yl]pyridin-2-yl]phthalazin-1-one | Human | 7631 | |
| BTK | Tec | TK | 5p9h | A | B | 6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-5-[[5-(1-methylpiperidin-4-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridazin-3-yl]pyridin-2-yl]phthalazin-1-one | Human | 7643 | |
| BTK | Tec | TK | 5p9i | A | A | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 7627 | |
| BTK | Tec | TK | 5p9i | A | B | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 7642 | |
| BTK | Tec | TK | 5p9i | A | C | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 7638 | |
| BTK | Tec | TK | 5p9j | A | A | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 7637 | |
| BTK | Tec | TK | 5p9j | A | B | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 7628 | |
| BTK | Tec | TK | 5p9j | A | C | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 7640 | |
| BTK | Tec | TK | 5p9k | A | A | 4-[4-[[5-fluoranyl-4-[[3-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]phenoxy]-~{n}-methyl-pyridine-2-carboxamide | Human | 7633 | |
| BTK | Tec | TK | 5p9k | A | B | 4-[4-[[5-fluoranyl-4-[[3-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]phenoxy]-~{n}-methyl-pyridine-2-carboxamide | Human | 7636 | |
| BTK | Tec | TK | 5p9k | A | C | 4-[4-[[5-fluoranyl-4-[[3-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]phenoxy]-~{n}-methyl-pyridine-2-carboxamide | Human | 7626 | |
| BTK | Tec | TK | 5p9l | A | A | ~{n}-[3-[[5-fluoranyl-2-[[4-(2-methoxyethoxy)phenyl]amino]pyrimidin-4-yl]amino]phenyl]propanamide | Human | 7625 | |
| BTK | Tec | TK | 5p9l | A | B | ~{n}-[3-[[5-fluoranyl-2-[[4-(2-methoxyethoxy)phenyl]amino]pyrimidin-4-yl]amino]phenyl]propanamide | Human | 7630 | |
| BTK | Tec | TK | 5p9m | A | A | 6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-one | Human | 7634 | |
| BTK | Tec | TK | 5p9m | A | B | 6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-one | Human | 7639 | |
| BTK | Tec | TK | 5p9m | A | C | 6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-one | Human | 7641 | |
| BTK | Tec | TK | 5t18 | A | A | 6-fluoro-5-(r)-(3-(s)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4h)-yl)-2-methylphenyl)-2-(s)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamide | Human | 7508 | |
| BTK | Tec | TK | 5t18 | A | B | 6-fluoro-5-(r)-(3-(s)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4h)-yl)-2-methylphenyl)-2-(s)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamide | Human | 7507 | |
| BTK | Tec | TK | 5u9d | A | A | (r)-n-methyl-2-(3-((quinoxalin-6-ylamino)methyl)furan-2-carbonyl)-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamide | Human | 7393 | |
| BTK | Tec | TK | 5u9d | A | B | (r)-n-methyl-2-(3-((quinoxalin-6-ylamino)methyl)furan-2-carbonyl)-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamide | Human | 7392 | |
| BTK | Tec | TK | 5vfi | A | A | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Human | 9602 | |
| BTK | Tec | TK | 5vfi | A | B | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Human | 9601 | |
| BTK | Tec | TK | 5vgo | A | A | 2-(2-methoxyethoxy)ethanol | Human | 8218 | |
| BTK | Tec | TK | 5vgo | A | B | 2-(2-methoxyethoxy)ethanol | Human | 8219 | |
| BTK | Tec | TK | 5xyz | A | A | n-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamide | Human | 9929 | |
| BTK | Tec | TK | 5xyz | A | B | n-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamide | Human | 9932 | |
| BTK | Tec | TK | 5xyz | B | A | n-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamide | Human | 9931 | |
| BTK | Tec | TK | 5xyz | B | B | n-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamide | Human | 9930 | |
| BTK | Tec | TK | 5zz4 | A | | n-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 10479 | |
| BTK | Tec | TK | 5zz4 | B | | n-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 10468 | |
| BTK | Tec | TK | 5zz4 | C | | n-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 10464 | |
| BTK | Tec | TK | 5zz4 | D | | n-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 10478 | |
| BTK | Tec | TK | 5zz4 | E | | n-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 10470 | |
| BTK | Tec | TK | 5zz4 | F | | n-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamide | Human | 10469 | |
| BTK | Tec | TK | 6aua | A | A | n-{3-[(2r)-6-{[3-amino-4-(morpholine-4-carbonyl)phenyl]amino}-5-oxo-2,5-dihydropyrazin-2-yl]-2-methylphenyl}-4-(piperidin-1-yl)benzamide | Human | 10472 | |
| BTK | Tec | TK | 6aua | A | B | n-{3-[(2r)-6-{[3-amino-4-(morpholine-4-carbonyl)phenyl]amino}-5-oxo-2,5-dihydropyrazin-2-yl]-2-methylphenyl}-4-(piperidin-1-yl)benzamide | Human | 10473 | |
| BTK | Tec | TK | 6aub | A | A | 4-tert-butyl-n-[2-methyl-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]benzamide | Human | 10466 | |
| BTK | Tec | TK | 6aub | A | B | 4-tert-butyl-n-[2-methyl-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]benzamide | Human | 10475 | |
| BTK | Tec | TK | 6bik | A | A | 4-tert-butyl-n-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridazin-3-yl)phenyl]benzamide | Human | 10680 | |
| BTK | Tec | TK | 6bik | A | B | 4-tert-butyl-n-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridazin-3-yl)phenyl]benzamide | Human | 10678 | |
| BTK | Tec | TK | 6bke | A | A | n-[2-(2-hydroxyethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamide | Human | 10681 | |
| BTK | Tec | TK | 6bke | A | B | n-[2-(2-hydroxyethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamide | Human | 10683 | |
| BTK | Tec | TK | 6bkh | A | A | n-[2-(hydroxymethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamide | Human | 10682 | |
| BTK | Tec | TK | 6bkh | A | B | n-[2-(hydroxymethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamide | Human | 10677 | |
| BTK | Tec | TK | 6bkw | A | A | n-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-1-methyl-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | Human | 10686 | |
| BTK | Tec | TK | 6bkw | A | B | n-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-1-methyl-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | Human | 10679 | |
| BTK | Tec | TK | 6bln | A | A | n-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | Human | 10685 | |
| BTK | Tec | TK | 6bln | A | B | n-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide | Human | 10684 | |
| BTK | Tec | TK | 6di0 | A | A | 6-(cyclohexylamino)pyridine-3-carboxamide | Human | 10629 | |
| BTK | Tec | TK | 6di0 | A | B | 6-(cyclohexylamino)pyridine-3-carboxamide | Human | 10626 | |
| BTK | Tec | TK | 6di0 | A | C | 6-(cyclohexylamino)pyridine-3-carboxamide | Human | 10628 | |
| BTK | Tec | TK | 6di1 | A | A | 4-amino-2-[(3s)-3-(propanoylamino)pyrrolidin-1-yl]pyrimidine-5-carboxamide | Human | 10630 | |
| BTK | Tec | TK | 6di1 | A | B | 4-amino-2-[(3s)-3-(propanoylamino)pyrrolidin-1-yl]pyrimidine-5-carboxamide | Human | 10627 | |
| BTK | Tec | TK | 6di3 | A | | 6-[(3s)-3-(acryloylamino)pyrrolidin-1-yl]-2-(4-phenoxyphenoxy)pyridine-3-carboxamide | Human | 10474 | |
| BTK | Tec | TK | 6di5 | A | A | 2-(4-phenoxyphenoxy)-6-[(1s,4s)-5-propanoyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyridine-3-carboxamide | Human | 10471 | |
| BTK | Tec | TK | 6di5 | A | B | 2-(4-phenoxyphenoxy)-6-[(1s,4s)-5-propanoyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyridine-3-carboxamide | Human | 10481 | |
| BTK | Tec | TK | 6di9 | A | A | 6-[(3s)-3-(acryloylamino)pyrrolidin-1-yl]-2-{[4-(tert-butylcarbamoyl)phenyl]amino}pyridine-3-carboxamide | Human | 10465 | |
| BTK | Tec | TK | 6di9 | A | B | 6-[(3s)-3-(acryloylamino)pyrrolidin-1-yl]-2-{[4-(tert-butylcarbamoyl)phenyl]amino}pyridine-3-carboxamide | Human | 10476 | |
| BTK | Tec | TK | 6e4f | A | A | 1,5-anhydro-2-{[5-(2-chloro-4-phenoxybenzene-1-carbonyl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-2,3,4-trideoxy-d-erythro-hexitol | Human | 10477 | |
| BTK | Tec | TK | 6e4f | A | B | 1,5-anhydro-2-{[5-(2-chloro-4-phenoxybenzene-1-carbonyl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-2,3,4-trideoxy-d-erythro-hexitol | Human | 10480 | |
| BTK | Tec | TK | 6ep9 | A | | n-[2-methyl-3-[4-methyl-6-[4-(4-methylpiperazine-1-carbonyl)anilino]-5-oxo-pyrazin-2-yl]phenyl]-4-(1-piperidyl)benzamide | Human | 10467 | |
| BTK | Tec | TK | 6hrp | A | | 6-~{tert}-butyl-8-fluoranyl-2-[2-(hydroxymethyl)-3-[1-methyl-5-[(5-morpholin-4-ylcarbonylpyridin-2-yl)amino]-6-oxidanylidene-pyridazin-3-yl]phenyl]phthalazin-1-one | Human | 10971 | |
| BTK | Tec | TK | 6hrt | A | | (9~{s})-12-(6-~{tert}-butyl-8-fluoranyl-1-oxidanylidene-phthalazin-2-yl)-6-methyl-4-[(5-morpholin-4-ylcarbonylpyridin-2-yl)amino]-9-oxidanyl-6-azatricyclo[9.4.0.0^{2,7}]pentadeca-1(15),2(7),3,11,13-pentaen-5-one | Human | 10972 | |
| BTK | Tec | TK | 6j6m | A | A | (7s)-2-(4-phenoxyphenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11767 | |
| BTK | Tec | TK | 6j6m | A | B | (7s)-2-(4-phenoxyphenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11766 | |
| BTK | Tec | TK | 6n9p | A | A | n-(3-{[2-amino-3-(4-phenoxyphenyl)pyridin-4-yl]oxy}phenyl)propanamide | Human | 10886 | |
| BTK | Tec | TK | 6n9p | A | B | n-(3-{[2-amino-3-(4-phenoxyphenyl)pyridin-4-yl]oxy}phenyl)propanamide | Human | 10887 | |
| BTK | Tec | TK | 6n9p | A | C | n-(3-{[2-amino-3-(4-phenoxyphenyl)pyridin-4-yl]oxy}phenyl)propanamide | Human | 10888 | |
| BTK | Tec | TK | 6nfh | A | A | 8-(2,3-dihydro-1h-inden-5-yl)-2-({4-[(2s)-3-(dimethylamino)-2-hydroxypropoxy]phenyl}amino)-5,8-dihydropteridine-6,7-dione | Human | 10964 | |
| BTK | Tec | TK | 6nfh | A | B | 8-(2,3-dihydro-1h-inden-5-yl)-2-({4-[(2s)-3-(dimethylamino)-2-hydroxypropoxy]phenyl}amino)-5,8-dihydropteridine-6,7-dione | Human | 10965 | |
| BTK | Tec | TK | 6nfi | A | A | n-(3-{[(2,6-dimethylphenyl)methyl]amino}-7-methoxyindeno[1,2-c]pyrazol-6-yl)methanesulfonamide | Human | 10962 | |
| BTK | Tec | TK | 6nfi | A | B | n-(3-{[(2,6-dimethylphenyl)methyl]amino}-7-methoxyindeno[1,2-c]pyrazol-6-yl)methanesulfonamide | Human | 10963 | |
| BTK | Tec | TK | 6nzm | A | A | n-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}urea | Human | 11144 | |
| BTK | Tec | TK | 6nzm | A | B | n-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}urea | Human | 11143 | |
| BTK | Tec | TK | 6nzm | D | A | n-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}urea | Human | 11141 | |
| BTK | Tec | TK | 6nzm | D | B | n-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}urea | Human | 11142 | |
| BTK | Tec | TK | 6o8i | A | A | 4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamide | Human | 11002 | |
| BTK | Tec | TK | 6o8i | A | B | 4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamide | Human | 11001 | |
| BTK | Tec | TK | 6omu | A | A | 1-[4-({[6-amino-5-(4-phenoxyphenyl)pyrimidin-4-yl]amino}methyl)piperidin-1-yl]prop-2-en-1-one | Human | 11529 | |
| BTK | Tec | TK | 6omu | A | B | 1-[4-({[6-amino-5-(4-phenoxyphenyl)pyrimidin-4-yl]amino}methyl)piperidin-1-yl]prop-2-en-1-one | Human | 11530 | |
| BTK | Tec | TK | 6omu | A | C | - | Human | 11528 | |
| BTK | Tec | TK | 6s90 | A | | 4-~{tert}-butyl-~{n}-[2-methyl-3-[6-[4-(4-methylpiperazin-1-yl)carbonylphenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]benzamide | Human | 11636 | |
| BTK | Tec | TK | 6s90 | B | | 4-~{tert}-butyl-~{n}-[2-methyl-3-[6-[4-(4-methylpiperazin-1-yl)carbonylphenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]benzamide | Human | 11635 | |
| BTK | Tec | TK | 6tfp | A | | ~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamide | Human | 12024 | |
| BTK | Tec | TK | 6tfp | B | | ~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamide | Human | 12020 | |
| BTK | Tec | TK | 6tfp | C | | ~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamide | Human | 12023 | |
| BTK | Tec | TK | 6tfp | D | | ~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamide | Human | 12021 | |
| BTK | Tec | TK | 6tfp | E | | ~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamide | Human | 12022 | |
| BTK | Tec | TK | 6vxq | A | A | n-{[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]methyl}benzamide | Human | 13100 | |
| BTK | Tec | TK | 6vxq | A | B | n-{[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]methyl}benzamide | Human | 13101 | |
| BTK | Tec | TK | 6w06 | A | A | 4-~{tert}-butyl-~{n}-[[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]methyl]benzamide | Human | 13099 | |
| BTK | Tec | TK | 6w06 | A | B | 4-~{tert}-butyl-~{n}-[[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]methyl]benzamide | Human | 13098 | |
| BTK | Tec | TK | 6w07 | A | A | ~{n}-[[2-methyl-4-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]phenyl]methyl]-3-propan-2-yloxy-azetidine-1-carboxamide | Human | 13096 | |
| BTK | Tec | TK | 6w07 | A | B | ~{n}-[[2-methyl-4-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]phenyl]methyl]-3-propan-2-yloxy-azetidine-1-carboxamide | Human | 13102 | |
| BTK | Tec | TK | 6w07 | A | C | ~{n}-[[2-methyl-4-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]phenyl]methyl]-3-propan-2-yloxy-azetidine-1-carboxamide | Human | 13097 | |
| BTK | Tec | TK | 6w7o | A | | [5-({[(3s)-2-(n-methyl-l-alanyl-3-methyl-l-valyl)-3-{[(1r)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl}-1,2,3,4-tetrahydroisoquinolin-7-yl]oxy}methyl)pyrazin-2-yl]methyl (3r)-3-{5-amino-4-carbamoyl-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazol-1-yl}piperidine-1-carboxylate | Human | 13195 | |
| BTK | Tec | TK | 6w7o | B | | [5-({[(3s)-2-(n-methyl-l-alanyl-3-methyl-l-valyl)-3-{[(1r)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl}-1,2,3,4-tetrahydroisoquinolin-7-yl]oxy}methyl)pyrazin-2-yl]methyl (3r)-3-{5-amino-4-carbamoyl-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazol-1-yl}piperidine-1-carboxylate | Human | 13196 | |
| BTK | Tec | TK | 6w8i | A | | - | Human | 12990 | |
| BTK | Tec | TK | 6w8i | B | | - | Human | 12991 | |
| BTK | Tec | TK | 6x3n | A | A | 4-{8-amino-3-[(6r,8as)-3-oxohexahydro-3h-[1,3]oxazolo[3,4-a]pyridin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-n-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 12514 | |
| BTK | Tec | TK | 6x3n | A | B | 4-{8-amino-3-[(6r,8as)-3-oxohexahydro-3h-[1,3]oxazolo[3,4-a]pyridin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-n-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 12510 | |
| BTK | Tec | TK | 6x3o | A | A | 4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 12513 | |
| BTK | Tec | TK | 6x3o | A | B | 4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 12512 | |
| BTK | Tec | TK | 6x3o | B | A | 4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 12508 | |
| BTK | Tec | TK | 6x3o | B | B | 4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 12511 | |
| BTK | Tec | TK | 6x3p | A | A | 4-{8-amino-3-[(6r,8as)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(cyclopropyloxy)-n-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 12516 | |
| BTK | Tec | TK | 6x3p | A | B | 4-{8-amino-3-[(6r,8as)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(cyclopropyloxy)-n-[4-(trifluoromethyl)pyridin-2-yl]benzamide | Human | 12517 | |
| BTK | Tec | TK | 6xe4 | A | A | (1s,2s)-n-[2'-(6-tert-butyl-8-fluoro-1-oxophthalazin-2(1h)-yl)-3'-(hydroxymethyl)-1-methyl-6-oxo[1,6-dihydro[3,4'-bipyridine]]-5-yl]-2-fluorocyclopropane-1-carboxamide | Human | 12515 | |
| BTK | Tec | TK | 6xe4 | A | B | (1s,2s)-n-[2'-(6-tert-butyl-8-fluoro-1-oxophthalazin-2(1h)-yl)-3'-(hydroxymethyl)-1-methyl-6-oxo[1,6-dihydro[3,4'-bipyridine]]-5-yl]-2-fluorocyclopropane-1-carboxamide | Human | 12509 | |
| BTK | Tec | TK | 7kxl | A | A | 3-tert-butyl-n-({2-fluoro-4-[2-(1-methyl-1h-pyrazol-4-yl)-1h-imidazo[4,5-b]pyridin-7-yl]phenyl}methyl)-1,2,4-oxadiazole-5-carboxamide | Human | 13563 | |
| BTK | Tec | TK | 7kxl | A | B | 3-tert-butyl-n-({2-fluoro-4-[2-(1-methyl-1h-pyrazol-4-yl)-1h-imidazo[4,5-b]pyridin-7-yl]phenyl}methyl)-1,2,4-oxadiazole-5-carboxamide | Human | 13561 | |
| BTK | Tec | TK | 7kxl | A | C | 3-tert-butyl-n-({2-fluoro-4-[2-(1-methyl-1h-pyrazol-4-yl)-1h-imidazo[4,5-b]pyridin-7-yl]phenyl}methyl)-1,2,4-oxadiazole-5-carboxamide | Human | 13576 | |
| BTK | Tec | TK | 7kxm | A | A | 4-tert-butyl-n-(2-methyl-3-{2-[4-(morpholine-4-carbonyl)phenyl]-1h-imidazo[4,5-b]pyridin-7-yl}phenyl)benzamide | Human | 13569 | |
| BTK | Tec | TK | 7kxm | A | B | 4-tert-butyl-n-(2-methyl-3-{2-[4-(morpholine-4-carbonyl)phenyl]-1h-imidazo[4,5-b]pyridin-7-yl}phenyl)benzamide | Human | 13564 | |
| BTK | Tec | TK | 7kxm | A | C | 4-tert-butyl-n-(2-methyl-3-{2-[4-(morpholine-4-carbonyl)phenyl]-1h-imidazo[4,5-b]pyridin-7-yl}phenyl)benzamide | Human | 13567 | |
| BTK | Tec | TK | 7kxn | A | A | 3-tert-butyl-n-[(1s)-6-{2-[5-methyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13574 | |
| BTK | Tec | TK | 7kxn | A | B | 3-tert-butyl-n-[(1s)-6-{2-[5-methyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13571 | |
| BTK | Tec | TK | 7kxn | A | C | 3-tert-butyl-n-[(1s)-6-{2-[5-methyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13570 | |
| BTK | Tec | TK | 7kxo | A | A | 3-tert-butyl-n-[(1r)-6-{2-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13573 | |
| BTK | Tec | TK | 7kxo | A | B | 3-tert-butyl-n-[(1r)-6-{2-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13568 | |
| BTK | Tec | TK | 7kxo | A | C | 3-tert-butyl-n-[(1r)-6-{2-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13572 | |
| BTK | Tec | TK | 7kxp | A | A | 3-tert-butyl-n-[(1s)-6-{2-[3-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13575 | |
| BTK | Tec | TK | 7kxp | A | B | 3-tert-butyl-n-[(1s)-6-{2-[3-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13566 | |
| BTK | Tec | TK | 7kxq | A | A | 3-tert-butyl-n-[(5r)-2-{2-[3,5-dimethyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-6,7,8,9-tetrahydro-5h-benzo[7]annulen-5-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13562 | |
| BTK | Tec | TK | 7kxq | A | B | 3-tert-butyl-n-[(5r)-2-{2-[3,5-dimethyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-6,7,8,9-tetrahydro-5h-benzo[7]annulen-5-yl]-1,2,4-oxadiazole-5-carboxamide | Human | 13565 | |
| BTK | Tec | TK | 7l5o | A | A | (2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile | Human | 14272 | |
| BTK | Tec | TK | 7l5o | A | B | (2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile | Human | 14271 | |
| BTK | Tec | TK | 7l5o | A | C | (2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile | Human | 14268 | |
| BTK | Tec | TK | 7l5p | A | A | (2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile | Human | 14269 | |
| BTK | Tec | TK | 7l5p | A | B | (2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrile | Human | 14270 | |
| BTK | Tec | TK | 7lty | A | A | ~{n}-[(5~{r})-2-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-6,7,8,9-tetrahydro-5~{h}-benzo[7]annulen-5-yl]-3-propan-2-yloxy-azetidine-1-carboxamide | Human | 14065 | |
| BTK | Tec | TK | 7lty | A | B | ~{n}-[(5~{r})-2-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-6,7,8,9-tetrahydro-5~{h}-benzo[7]annulen-5-yl]-3-propan-2-yloxy-azetidine-1-carboxamide | Human | 14069 | |
| BTK | Tec | TK | 7lty | A | C | ~{n}-[(5~{r})-2-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-6,7,8,9-tetrahydro-5~{h}-benzo[7]annulen-5-yl]-3-propan-2-yloxy-azetidine-1-carboxamide | Human | 14068 | |
| BTK | Tec | TK | 7lty | A | D | ~{n}-[(5~{r})-2-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-6,7,8,9-tetrahydro-5~{h}-benzo[7]annulen-5-yl]-3-propan-2-yloxy-azetidine-1-carboxamide | Human | 14064 | |
| BTK | Tec | TK | 7ltz | A | A | 1-~{tert}-butyl-~{n}-[(5~{r})-8-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-2-(oxetan-3-yl)-1,3,4,5-tetrahydro-2-benzazepin-5-yl]-1,2,3-triazole-4-carboxamide | Human | 14067 | |
| BTK | Tec | TK | 7ltz | A | B | 1-~{tert}-butyl-~{n}-[(5~{r})-8-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-2-(oxetan-3-yl)-1,3,4,5-tetrahydro-2-benzazepin-5-yl]-1,2,3-triazole-4-carboxamide | Human | 14066 | |
| BTK | Tec | TK | 7n4q | A | A | (2r)-2-(3-chloro-5-fluoroanilino)-2-cyclopropyl-n-[(3r)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]acetamide | Human | 14227 | |
| BTK | Tec | TK | 7n4q | A | B | (2r)-2-(3-chloro-5-fluoroanilino)-2-cyclopropyl-n-[(3r)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]acetamide | Human | 14224 | |
| BTK | Tec | TK | 7n4r | A | A | n-{2-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]ethyl}-n~2~-phenylglycinamide | Human | 14226 | |
| BTK | Tec | TK | 7n4r | A | B | n-{2-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]ethyl}-n~2~-phenylglycinamide | Human | 14228 | |
| BTK | Tec | TK | 7n4r | A | C | n-{2-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]ethyl}-n~2~-phenylglycinamide | Human | 14225 | |
| BTK | Tec | TK | 7n4s | A | | (3r,3'r)-3-anilino-1'-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)[1,3'-bipiperidin]-2-one | Human | 14229 | |
| BTK | Tec | TK | 7n5o | A | A | 5-(1h-benzimidazol-2-yl)-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 13896 | |
| BTK | Tec | TK | 7n5o | A | B | 5-(1h-benzimidazol-2-yl)-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 13891 | |
| BTK | Tec | TK | 7n5r | A | A | 5-phenyl-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 13895 | |
| BTK | Tec | TK | 7n5r | A | B | 5-phenyl-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 13890 | |
| BTK | Tec | TK | 7n5x | A | A | 5-(1-ethoxyisoquinolin-3-yl)-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 13893 | |
| BTK | Tec | TK | 7n5x | A | B | 5-(1-ethoxyisoquinolin-3-yl)-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 13889 | |
| BTK | Tec | TK | 7n5y | A | A | 5-(1-{[(3s)-1-propanoylpyrrolidin-3-yl]oxy}isoquinolin-3-yl)-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 13894 | |
| BTK | Tec | TK | 7n5y | A | B | 5-(1-{[(3s)-1-propanoylpyrrolidin-3-yl]oxy}isoquinolin-3-yl)-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 13892 | |
| BTK | Tec | TK | 7r60 | A | A | 2-(4-phenoxyphenoxy)-5-[(3r)-1-(prop-2-enoyl)piperidin-3-yl]pyridine-3-carboxamide | Human | 13937 | |
| BTK | Tec | TK | 7r60 | A | B | 2-(4-phenoxyphenoxy)-5-[(3r)-1-(prop-2-enoyl)piperidin-3-yl]pyridine-3-carboxamide | Human | 13939 | |
| BTK | Tec | TK | 7r61 | A | A | 5-{(3s)-1-[(z)-iminomethyl]piperidin-3-yl}-2-(4-phenoxyphenoxy)pyridine-3-carboxamide | Human | 13938 | |
| BTK | Tec | TK | 7r61 | A | B | 5-{(3s)-1-[(z)-iminomethyl]piperidin-3-yl}-2-(4-phenoxyphenoxy)pyridine-3-carboxamide | Human | 13936 | |
| BTK | Tec | TK | 7r61 | A | C | 5-{(3s)-1-[(z)-iminomethyl]piperidin-3-yl}-2-(4-phenoxyphenoxy)pyridine-3-carboxamide | Human | 13940 | |
| BTK | Tec | TK | 7yc9 | A | A | (7~{s})-2-(4-bromanyl-3,5-dimethoxy-phenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 14746 | |
| BTK | Tec | TK | 7yc9 | A | B | (7~{s})-2-(4-bromanyl-3,5-dimethoxy-phenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 14745 | |
| BTK | Tec | TK | 8e2m | A | A | (5p)-5-[4-methyl-6-(2-methylpropyl)pyridin-3-yl]-4-oxo-n-[(1r,2s)-2-propanamidocyclopentyl]-4,5-dihydro-3h-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide | Human | 14552 | |
| BTK | Tec | TK | 8e2m | A | B | (5p)-5-[4-methyl-6-(2-methylpropyl)pyridin-3-yl]-4-oxo-n-[(1r,2s)-2-propanamidocyclopentyl]-4,5-dihydro-3h-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide | Human | 14553 | |
| BTK | Tec | TK | 8e2m | A | C | (5p)-5-[4-methyl-6-(2-methylpropyl)pyridin-3-yl]-4-oxo-n-[(1r,2s)-2-propanamidocyclopentyl]-4,5-dihydro-3h-1-thia-3,5,8-triazaacenaphthylene-2-carboxamide | Human | 14551 | |
| BTK | Tec | TK | 8ejb | A | A | 5-[(3r)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamide | Human | 14614 | |
| BTK | Tec | TK | 8ejb | A | B | 5-[(3r)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamide | Human | 14615 | |
| BTK | Tec | TK | 8flg | A | A | n~2~-(3-chlorophenyl)-n-[(3r)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]glycinamide | Human | 14641 | |
| BTK | Tec | TK | 8flg | A | B | n~2~-(3-chlorophenyl)-n-[(3r)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]glycinamide | Human | 14634 | |
| BTK | Tec | TK | 8flh | A | A | 2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]azepan-1-yl}ethan-1-one | Human | 14637 | |
| BTK | Tec | TK | 8flh | A | B | 2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]azepan-1-yl}ethan-1-one | Human | 14638 | |
| BTK | Tec | TK | 8flh | A | C | 2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]azepan-1-yl}ethan-1-one | Human | 14639 | |
| BTK | Tec | TK | 8fll | A | A | pirtobrutinib | Human | 14636 | |
| BTK | Tec | TK | 8fll | A | B | pirtobrutinib | Human | 14640 | |
| BTK | Tec | TK | 8fln | A | A | pirtobrutinib | Human | 14642 | |
| BTK | Tec | TK | 8fln | A | B | pirtobrutinib | Human | 14635 | |
| BTK | Tec | TK | 8fln | A | C | pirtobrutinib | Human | 14633 | |
| BTK | Tec | TK | 8flv | A | A | 2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}ethan-1-one | Human | 14698 | |
| BTK | Tec | TK | 8flv | A | B | 2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}ethan-1-one | Human | 14699 | |
| BTK | Tec | TK | 8flv | A | C | 2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}ethan-1-one | Human | 14697 | |
| BTK | Tec | TK | 8gc7 | A | A | 5-(piperidin-1-yl)-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamide | Human | 15196 | |
| BTK | Tec | TK | 8gc7 | A | B | 5-(piperidin-1-yl)-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamide | Human | 15197 | |
| BTK | Tec | TK | 8gc8 | A | A | 5-(piperidin-1-yl)-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamide | Human | 15195 | |
| BTK | Tec | TK | 8gc8 | A | B | 5-(piperidin-1-yl)-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamide | Human | 15192 | |
| BTK | Tec | TK | 8tu3 | A | A | 1-[(4r)-4-{[(6p,8s)-6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}azepan-1-yl]propan-1-one | Human | 15362 | |
| BTK | Tec | TK | 8tu3 | A | B | 1-[(4r)-4-{[(6p,8s)-6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}azepan-1-yl]propan-1-one | Human | 15354 | |
| BTK | Tec | TK | 8tu3 | A | C | 1-[(4r)-4-{[(6p,8s)-6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}azepan-1-yl]propan-1-one | Human | 15359 | |
| BTK | Tec | TK | 8tu4 | A | A | n-methyl-n-[(1s,3r)-3-methyl-3-{[(6m,8s)-6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}cyclobutyl]propanamide | Human | 15360 | |
| BTK | Tec | TK | 8tu4 | A | B | n-methyl-n-[(1s,3r)-3-methyl-3-{[(6m,8s)-6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}cyclobutyl]propanamide | Human | 15357 | |
| BTK | Tec | TK | 8tu4 | A | C | n-methyl-n-[(1s,3r)-3-methyl-3-{[(6m,8s)-6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}cyclobutyl]propanamide | Human | 15355 | |
| BTK | Tec | TK | 8tu5 | A | A | 1-[(1s,5s,6s)-6-methyl-6-{[(6m,8r)-6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}-2-azabicyclo[3.2.0]heptan-2-yl]propan-1-one | Human | 15363 | |
| BTK | Tec | TK | 8tu5 | A | B | 1-[(1s,5s,6s)-6-methyl-6-{[(6m,8r)-6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}-2-azabicyclo[3.2.0]heptan-2-yl]propan-1-one | Human | 15358 | |
| BTK | Tec | TK | 8tu5 | A | C | 1-[(1s,5s,6s)-6-methyl-6-{[(6m,8r)-6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}-2-azabicyclo[3.2.0]heptan-2-yl]propan-1-one | Human | 15356 | |
| BTK | Tec | TK | 8u2d | A | A | (3r)-2-[n-(1h-indazole-5-carbonyl)-3-methyl-d-phenylalanyl]-n-methyl-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamide | Human | 15199 | |
| BTK | Tec | TK | 8u2d | A | B | (3r)-2-[n-(1h-indazole-5-carbonyl)-3-methyl-d-phenylalanyl]-n-methyl-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamide | Human | 15193 | |
| BTK | Tec | TK | 8u2e | A | A | (2s)-6-fluoro-5-[(3s)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-2-(4-methylpiperazine-1-carbonyl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamide | Human | 15198 | |
| BTK | Tec | TK | 8u2e | A | B | (2s)-6-fluoro-5-[(3s)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-2-(4-methylpiperazine-1-carbonyl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamide | Human | 15194 | |
| BTK | Tec | TK | 8yvv | A | A | - | Human | 15353 | |
| BTK | Tec | TK | 8yvv | A | B | - | Human | 15361 | |
| BUB1 | BUB | Other | 4qpm | A | | adenosine-5'-diphosphate | Human | 1843 | |
| BUB1 | BUB | Other | 4qpm | B | | adenosine-5'-diphosphate | Human | 1844 | |
| BUB1 | BUB | Other | 4r8q | A | | adenosine-5'-diphosphate | Human | 1842 | |
| BUB1 | BUB | Other | 5dmz | A | | adenosine-5'-diphosphate | Human | 6287 | |
| BUB1 | BUB | Other | 5dmz | B | | adenosine-5'-diphosphate | Human | 6286 | |
| BUB1 | BUB | Other | 6f7b | A | A | 2-[3,5-bis(fluoranyl)-4-[[3-[5-methoxy-4-[(3-methoxypyridin-4-yl)amino]pyrimidin-2-yl]indazol-1-yl]methyl]phenoxy]ethanol | Human | 10808 | |
| BUB1 | BUB | Other | 6f7b | A | B | 2-[3,5-bis(fluoranyl)-4-[[3-[5-methoxy-4-[(3-methoxypyridin-4-yl)amino]pyrimidin-2-yl]indazol-1-yl]methyl]phenoxy]ethanol | Human | 10807 | |
| BUB1B (BUBR1) | BUB | Other | 6tlj | S | | - | Human | 11992 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg7 | A | | adenosine-5'-triphosphate | Human | 4848 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg8 | A | | adenosine-5'-triphosphate | Human | 4850 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg8 | B | | adenosine-5'-triphosphate | Human | 4849 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg9 | A | | adenosine-5'-triphosphate | Human | 4846 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg9 | B | | adenosine-5'-triphosphate | Human | 4845 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fgb | A | | - | Human | 4847 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | A | A | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4829 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | A | B | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4830 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | C | A | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4832 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | C | B | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4831 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6qp5 | A | A | - | Human | 12028 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6qp5 | A | B | - | Human | 12029 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t28 | A | A | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamide | Human | 13202 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t28 | A | B | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamide | Human | 13205 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t29 | A | A | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamide | Human | 13204 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t29 | A | B | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamide | Human | 13203 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t6f | A | A | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamide | Human | 11939 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t6f | A | B | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamide | Human | 11940 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t6f | B | A | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamide | Human | 11941 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t6f | B | B | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamide | Human | 11942 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 8bfm | A | | pyrazolo[5,1-a]phthalazin-6-amine | Human | 14516 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 8bfs | A | A | 3~{h}-pyrrolo[2,3-c]isoquinolin-5-amine | Human | 14506 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 8bfs | A | B | 3~{h}-pyrrolo[2,3-c]isoquinolin-5-amine | Human | 14505 | |
| CAMK1G (CaMK1g) | CAMK1 | CAMK | 2jam | A | A | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1218 | |
| CAMK1G (CaMK1g) | CAMK1 | CAMK | 2jam | A | B | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1221 | |
| CAMK1G (CaMK1g) | CAMK1 | CAMK | 2jam | B | A | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1220 | |
| CAMK1G (CaMK1g) | CAMK1 | CAMK | 2jam | B | B | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1219 | |
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b55 | A | A | - | Mouse | 14244 | |
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b55 | A | B | - | Mouse | 14247 | |
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b56 | A | A | - | Mouse | 14245 | |
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b56 | A | B | - | Mouse | 14249 | |
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b57 | A | A | - | Mouse | 14246 | |
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b57 | A | B | - | Mouse | 14248 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 2vz6 | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 2472 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 2vz6 | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 2471 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 2vz6 | B | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 2474 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 2vz6 | B | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 2470 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 3soa | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 2473 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6vzk | A | | 4'-hydroxycinnamic acid | Human | 12165 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6w4o | O | | - | Human | 12485 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6w4p | H | | - | Human | 12484 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6x5g | A | A | - | Human | 13061 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6x5g | A | B | - | Human | 13068 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6x5q | A | | - | Human | 13056 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl0 | A | | methyl 6-o-(heptylcarbamoyl)-beta-l-altropyranoside | Human | 13111 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl0 | B | | methyl 6-o-(heptylcarbamoyl)-beta-l-altropyranoside | Human | 13114 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl1 | A | | adenosine-5'-triphosphate | Human | 13059 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl1 | B | | adenosine-5'-triphosphate | Human | 13062 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl2 | A | | - | Human | 13064 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7uiq | A | | - | Human | 14175 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7uir | A | | adenosine-5'-triphosphate | Human | 14173 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7uis | A | | - | Human | 14174 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujp | A | | adenosine-5'-diphosphate | Human | 14193 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujq | A | | methyl 6-o-(heptylcarbamoyl)-beta-l-altropyranoside | Human | 14189 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujr | A | | - | Human | 14191 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujs | A | | adenosine-5'-diphosphate | Human | 14190 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujt | A | | adenosine-5'-triphosphate | Human | 14192 | |
| CAMK2B (CaMK2b) | CAMK2 | CAMK | 3bhh | A | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 1507 | |
| CAMK2B (CaMK2b) | CAMK2 | CAMK | 3bhh | B | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 1506 | |
| CAMK2B (CaMK2b) | CAMK2 | CAMK | 3bhh | C | | - | Human | 1505 | |
| CAMK2B (CaMK2b) | CAMK2 | CAMK | 3bhh | D | | - | Human | 1504 | |
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | A | A | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8694 | |
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | A | B | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8691 | |
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | B | A | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8690 | |
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | B | B | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8693 | |
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | C | A | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8697 | |
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | C | B | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8692 | |
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | D | A | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8695 | |
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | D | B | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8696 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2vn9 | A | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2140 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2vn9 | B | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2139 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2wel | A | A | (3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamide | Human | 2138 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2wel | A | B | (3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamide | Human | 2137 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2wel | A | C | (3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamide | Human | 2136 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 5vlo | A | | n-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Human | 8348 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 5vlo | B | | n-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Human | 8347 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 6ayw | A | | n-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 8666 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 6ayw | B | | n-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 8665 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 8uso | A | | - | Human | 15247 | |
| CAMK2G (CaMK2g) | CAMK2 | CAMK | 2v7o | A | A | - | Human | 7239 | |
| CAMK2G (CaMK2g) | CAMK2 | CAMK | 2v7o | A | B | - | Human | 7238 | |
| CAMK4 (CaMK4) | CAMK1 | CAMK | 2w4o | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 2687 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6ccf | A | | n-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamide | Human | 9712 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6ccf | B | | n-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamide | Human | 9717 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | A | A | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9716 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | A | B | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9714 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | B | A | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9709 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | B | B | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9713 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | C | A | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9711 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | C | B | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9715 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | D | A | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9710 | |
| CAMKK1 (CaMKK1) | CAMKK | Other | 6cd6 | D | B | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9708 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 2zv2 | A | | 7-oxo-7h-benzimidazo[2,1-a]benz[de]isoquinoline-3-carboxylic acid | Human | 406 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5uy6 | A | | 2-cyclopentyl-4-(5-phenylfuro[2,3-b]pyridin-3-yl)benzoic acid | Human | 7982 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5uyj | A | A | 2-cyclopentyl-4-(7-methoxyquinolin-4-yl)benzoic acid | Human | 7560 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5uyj | A | B | 2-cyclopentyl-4-(7-methoxyquinolin-4-yl)benzoic acid | Human | 7559 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5vt1 | A | | 4-({5-[(3-hydroxy-4-methylphenyl)amino]-4-oxo-4h-1,2,6-thiadiazin-3-yl}amino)benzamide | Human | 7591 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5yv8 | A | A | 1-amino-4-hydroxy-9,10-dioxo-9,10-dihydroanthracene-2-carboxylic acid | Human | 10753 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5yv8 | A | B | 1-amino-4-hydroxy-9,10-dioxo-9,10-dihydroanthracene-2-carboxylic acid | Human | 10755 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5yv9 | A | | 5-chloro-2-methoxy-4[(1z)-3-(4-methoxyphenyl)-3-oxoprop-1-en-1-yl]aminobenzoic acid | Human | 10752 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5yva | A | | 3-(1h-tetrazol-5-yl)-10lambda~6~-thioxanthene-9,10,10-trione | Human | 10750 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5yvb | A | | (3z)-5-chloro-3-[(1-methyl-1h-pyrazol-4-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 10751 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 5yvc | A | | 3-{2,4-dimethyl-5-[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-1h-pyrrol-3-yl}propanoic acid | Human | 10754 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6bku | A | | 2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 8687 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6ble | A | A | 1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amine | Human | 8688 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6ble | A | B | 1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amine | Human | 8689 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6bql | A | | 2-({5-chloro-2-[(2-methoxy-4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}amino)-n-methylbenzamide | Human | 9061 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6bqp | A | | 1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amine | Human | 9064 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6bqq | A | | 4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 9063 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6brc | A | | 5-chloro-n~2~-{4-[4-(dimethylamino)piperidin-1-yl]-2-methoxyphenyl}-n~4~-[2-(dimethylphosphoryl)phenyl]pyrimidine-2,4-diamine | Human | 9062 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6brc | B | | 5-chloro-n~2~-{4-[4-(dimethylamino)piperidin-1-yl]-2-methoxyphenyl}-n~4~-[2-(dimethylphosphoryl)phenyl]pyrimidine-2,4-diamine | Human | 9060 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6cmj | A | A | 2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9784 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6cmj | A | B | 2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9783 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6cmj | B | A | 2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9786 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 6cmj | B | B | 2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 9785 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 8tuc | A | A | (4m)-2-cyclopentyl-4-(7-ethoxyquinazolin-4-yl)benzoic acid | Human | 15005 | |
| CAMKK2 (CaMKK2) | CAMKK | Other | 8tuc | A | B | (4m)-2-cyclopentyl-4-(7-ethoxyquinazolin-4-yl)benzoic acid | Human | 15004 | |
| CASK | CASK | CAMK | 3c0g | A | A | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3828 | |
| CASK | CASK | CAMK | 3c0g | A | B | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3827 | |
| CASK | CASK | CAMK | 3c0g | B | A | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3824 | |
| CASK | CASK | CAMK | 3c0g | B | B | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3826 | |
| CASK | CASK | CAMK | 3c0h | A | | adenosine monophosphate | Human | 3825 | |
| CASK | CASK | CAMK | 3c0h | B | | adenosine monophosphate | Human | 3817 | |
| CASK | CASK | CAMK | 3c0i | A | A | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3830 | |
| CASK | CASK | CAMK | 3c0i | A | B | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3819 | |
| CASK | CASK | CAMK | 3mfr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 3822 | |
| CASK | CASK | CAMK | 3mfr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 3831 | |
| CASK | CASK | CAMK | 3mfs | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 3818 | |
| CASK | CASK | CAMK | 3mfs | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 3829 | |
| CASK | CASK | CAMK | 3mft | A | A | - | Human | 3823 | |
| CASK | CASK | CAMK | 3mft | A | B | - | Human | 3821 | |
| CASK | CASK | CAMK | 3mfu | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 3816 | |
| CASK | CASK | CAMK | 3mfu | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 3832 | |
| CASK | CASK | CAMK | 3tac | A | | - | Human | 3820 | |
| CASK | CASK | CAMK | 6kmh | A | | - | Human | 12672 | |
| CASK | CASK | CAMK | 6kmh | B | | - | Human | 12671 | |
| CASK | CASK | CAMK | 7oai | A | A | 4-(cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-n-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | Human | 13584 | |
| CASK | CASK | CAMK | 7oai | A | B | 4-(cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-n-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | Human | 13583 | |
| CASK | CASK | CAMK | 7oaj | A | A | 4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-n-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | Human | 13582 | |
| CASK | CASK | CAMK | 7oaj | A | B | 4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-n-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | Human | 13581 | |
| CASK | CASK | CAMK | 7oak | A | | 2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclopentylamino)-n-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | Human | 13585 | |
| CASK | CASK | CAMK | 7oal | A | | 2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclohexylamino)-n-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | Human | 13586 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 3qfv | A | | 2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide | Human | 4860 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 3qfv | B | | 2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide | Human | 4857 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 3tku | A | | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 4862 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 3tku | B | | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 4859 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 4uak | A | A | adenosine-5'-diphosphate | Human | 4864 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 4uak | A | B | adenosine-5'-diphosphate | Human | 4863 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 4ual | A | A | 4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamide | Human | 4861 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 4ual | A | B | 4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamide | Human | 4858 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 5ote | A | | 2-[4-[(6~{s})-1,8-diazaspiro[5.5]undecan-8-yl]-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]-1,3-thiazole | Human | 9578 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 5otf | A | | (6~{s})-8-(3-pyrimidin-4-yl-1~{h}-pyrrolo[2,3-b]pyridin-4-yl)-1,8-diazaspiro[5.5]undecane | Human | 9577 | |
| CDC7 | CDC7 | Other | 4f99 | A | | adenosine-5'-diphosphate | Human | 4824 | |
| CDC7 | CDC7 | Other | 4f9a | A | | adenosine-5'-diphosphate | Human | 4825 | |
| CDC7 | CDC7 | Other | 4f9a | C | | adenosine-5'-diphosphate | Human | 4826 | |
| CDC7 | CDC7 | Other | 4f9b | A | | 2-(pyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4828 | |
| CDC7 | CDC7 | Other | 4f9b | C | | 2-(pyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4827 | |
| CDC7 | CDC7 | Other | 4f9c | A | | 8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 4823 | |
| CDC7 | CDC7 | Other | 6ya6 | A | A | 8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 13844 | |
| CDC7 | CDC7 | Other | 6ya6 | A | B | 8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 13841 | |
| CDC7 | CDC7 | Other | 6ya7 | A | A | adenosine-5'-diphosphate | Human | 13845 | |
| CDC7 | CDC7 | Other | 6ya7 | A | B | adenosine-5'-diphosphate | Human | 13842 | |
| CDC7 | CDC7 | Other | 6ya8 | A | A | adenosine-5'-diphosphate | Human | 13846 | |
| CDC7 | CDC7 | Other | 6ya8 | A | B | adenosine-5'-diphosphate | Human | 13843 | |
| CDK1 (CDC2) | CDK | CMGC | 4y72 | A | A | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4610 | |
| CDK1 (CDC2) | CDK | CMGC | 4y72 | A | B | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4609 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc3 | A | A | - | Human | 6555 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc3 | A | B | - | Human | 6554 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | A | A | - | Human | 4607 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | A | B | - | Human | 4616 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | C | A | - | Human | 4608 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | C | B | - | Human | 4611 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | E | A | - | Human | 4612 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | E | B | - | Human | 4614 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | G | A | - | Human | 4613 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | G | B | - | Human | 4615 | |
| CDK1 (CDC2) | CDK | CMGC | 5hq0 | A | A | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 6422 | |
| CDK1 (CDC2) | CDK | CMGC | 5hq0 | A | B | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 6421 | |
| CDK1 (CDC2) | CDK | CMGC | 5lqf | A | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 7364 | |
| CDK1 (CDC2) | CDK | CMGC | 5lqf | A | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 7366 | |
| CDK1 (CDC2) | CDK | CMGC | 5lqf | D | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 7365 | |
| CDK1 (CDC2) | CDK | CMGC | 5lqf | D | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 7367 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu2 | A | A | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | 10780 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu2 | A | B | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | 10776 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu3 | A | | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10778 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu4 | A | | ~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamine | Human | 10777 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu6 | A | | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 10774 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu7 | A | | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10781 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu7 | C | | - | Human | 10775 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu7 | E | | - | Human | 10782 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu7 | G | | - | Human | 10779 | |
| CDK1 (CDC2) | CDK | CMGC | 7nj0 | B | | - | Human | 13827 | |
| CDK12 (CRK7) | CDK | CMGC | 4cxa | A | | phosphoaminophosphonic acid-adenylate ester | Human | 4856 | |
| CDK12 (CRK7) | CDK | CMGC | 4cxa | C | | - | Human | 4853 | |
| CDK12 (CRK7) | CDK | CMGC | 4nst | A | | adenosine-5'-diphosphate | Human | 4852 | |
| CDK12 (CRK7) | CDK | CMGC | 4nst | C | | adenosine-5'-diphosphate | Human | 4851 | |
| CDK12 (CRK7) | CDK | CMGC | 4un0 | C | | - | Human | 4854 | |
| CDK12 (CRK7) | CDK | CMGC | 4un0 | D | | - | Human | 4855 | |
| CDK12 (CRK7) | CDK | CMGC | 5acb | C | | n-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamide | Human | 6701 | |
| CDK12 (CRK7) | CDK | CMGC | 5acb | D | | n-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamide | Human | 6702 | |
| CDK12 (CRK7) | CDK | CMGC | 6b3e | A | | 2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-ol | Human | 9452 | |
| CDK12 (CRK7) | CDK | CMGC | 6b3e | C | | 2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-ol | Human | 9453 | |
| CDK12 (CRK7) | CDK | CMGC | 6ckx | A | | n-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamide | Human | 10578 | |
| CDK12 (CRK7) | CDK | CMGC | 6ckx | C | | n-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamide | Human | 10579 | |
| CDK12 (CRK7) | CDK | CMGC | 6td3 | B | | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 12371 | |
| CDK12 (CRK7) | CDK | CMGC | 6td3 | E | | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 12369 | |
| CDK12 (CRK7) | CDK | CMGC | 6td3 | H | | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 12370 | |
| CDK12 (CRK7) | CDK | CMGC | 7nxk | A | | (e)-n-[4-[(1r,3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]cyclohexyl]oxyphenyl]-4-(dimethylamino)but-2-enamide | Human | 13547 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu1 | B | | (2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-ol | Human | 14930 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu2 | B | | ~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-propan-2-yl-purin-6-amine | Human | 14918 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu3 | B | | 2-morpholin-4-yl-9-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]purin-6-amine | Human | 14931 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu4 | B | | (2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-ol | Human | 14910 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu5 | B | | ~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amine | Human | 14926 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu6 | B | | ~{n}-(1~{h}-benzimidazol-2-ylmethyl)-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amine | Human | 14921 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu7 | B | | - | Human | 14913 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu9 | B | | r-roscovitine | Human | 14914 | |
| CDK12 (CRK7) | CDK | CMGC | 8bua | B | | (2~{r})-~{n}-(1~{h}-benzimidazol-2-yl)-2-(3-oxidanylidene-1~{h}-isoindol-2-yl)propanamide | Human | 14932 | |
| CDK12 (CRK7) | CDK | CMGC | 8bub | B | | ~{n}-(5-methyl-2,3-dihydro-1,3-thiazol-2-yl)-3-(5-methylfuran-2-yl)carbonyl-1,3-thiazolidine-4-carboxamide | Human | 14928 | |
| CDK12 (CRK7) | CDK | CMGC | 8buc | B | | 2-(1~{h}-benzimidazol-2-ylsulfanyl)-~{n}-(5-chloranylpyridin-2-yl)ethanamide | Human | 14909 | |
| CDK12 (CRK7) | CDK | CMGC | 8bud | B | | ~{n}-(5-bromanylpyridin-2-yl)-3-(4-oxidanylidenequinazolin-3-yl)propanamide | Human | 14929 | |
| CDK12 (CRK7) | CDK | CMGC | 8bue | B | | ~{n}-(1~{h}-benzimidazol-2-yl)-1-(2-methoxy-5-methyl-phenyl)-5-oxidanylidene-pyrrolidine-3-carboxamide | Human | 14912 | |
| CDK12 (CRK7) | CDK | CMGC | 8buf | B | | 2-(6,7-dihydro-4~{h}-thieno[3,2-c]pyridin-5-ylmethyl)-6,7-dimethoxy-3~{h}-quinazolin-4-one | Human | 14919 | |
| CDK12 (CRK7) | CDK | CMGC | 8bug | B | | 2-[2-[(6-methylpyridin-2-yl)amino]-1,3-thiazol-4-yl]-~{n}-(5-methyl-1,3-thiazol-2-yl)ethanamide | Human | 14935 | |
| CDK12 (CRK7) | CDK | CMGC | 8buh | B | | 6-[[[2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-9-propan-2-yl-purin-6-yl]amino]methyl]-3-pyridin-2-yl-1~{h}-pyridin-2-one | Human | 14922 | |
| CDK12 (CRK7) | CDK | CMGC | 8bui | B | | (2~{r})-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)amino]purin-2-yl]amino]butan-1-ol | Human | 14925 | |
| CDK12 (CRK7) | CDK | CMGC | 8buj | B | | (2~{r})-2-[[6-(octylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14933 | |
| CDK12 (CRK7) | CDK | CMGC | 8buk | B | | (2~{r})-2-[[6-(naphthalen-2-ylmethylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14927 | |
| CDK12 (CRK7) | CDK | CMGC | 8bul | B | | (2~{r})-2-[[6-(3-phenylpropylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14911 | |
| CDK12 (CRK7) | CDK | CMGC | 8bum | B | | (2r)-2-[[6-(5-naphthalen-1-ylpentylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14924 | |
| CDK12 (CRK7) | CDK | CMGC | 8bun | B | | (2~{r})-2-[[6-[(4-phenylphenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14916 | |
| CDK12 (CRK7) | CDK | CMGC | 8buo | B | | (2~{r})-2-[[6-[(3-fluoranyl-4-pyridin-2-yl-phenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14934 | |
| CDK12 (CRK7) | CDK | CMGC | 8bup | B | | (2~{r})-2-[[6-[3-(3-methylphenyl)propylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14923 | |
| CDK12 (CRK7) | CDK | CMGC | 8buq | B | | (2~{r})-2-[[6-[[1-(3-chlorophenyl)pyrazol-3-yl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14917 | |
| CDK12 (CRK7) | CDK | CMGC | 8bur | B | A | ~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamide | Human | 14915 | |
| CDK12 (CRK7) | CDK | CMGC | 8bur | B | B | ~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamide | Human | 14920 | |
| CDK12 (CRK7) | CDK | CMGC | 8bus | B | | 1,3-dimethyl-5-[[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]methyl]pyrazole-4-sulfonamide | Human | 14908 | |
| CDK12 (CRK7) | CDK | CMGC | 8but | B | | 2-[[6-[[4-(2-hydroxyethyloxy)phenyl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14936 | |
| CDK12 (CRK7) | CDK | CMGC | 8p81 | A | A | ~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amine | Human | 15062 | |
| CDK12 (CRK7) | CDK | CMGC | 8p81 | A | B | ~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amine | Human | 15061 | |
| CDK13 (CHED) | CDK | CMGC | 5efq | A | | adenosine-5'-diphosphate | Human | 6323 | |
| CDK13 (CHED) | CDK | CMGC | 5efq | C | | adenosine-5'-diphosphate | Human | 6324 | |
| CDK13 (CHED) | CDK | CMGC | 7nxj | A | | n-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamide | Human | 13544 | |
| CDK16 (PCTAIRE1) | CDK | CMGC | 3mtl | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 1701 | |
| CDK16 (PCTAIRE1) | CDK | CMGC | 3mtl | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 1702 | |
| CDK16 (PCTAIRE1) | CDK | CMGC | 5g6v | A | | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 7273 | |
| CDK16 (PCTAIRE1) | CDK | CMGC | 5g6v | B | | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 7274 | |
| CDK2 | CDK | CMGC | 1aq1 | A | | staurosporine | Human | 4267 | |
| CDK2 | CDK | CMGC | 1b38 | A | | adenosine-5'-triphosphate | Human | 4483 | |
| CDK2 | CDK | CMGC | 1b39 | A | | adenosine-5'-triphosphate | Human | 4407 | |
| CDK2 | CDK | CMGC | 1buh | A | | - | Human | 4178 | |
| CDK2 | CDK | CMGC | 1ckp | A | A | purvalanol b | Human | 4066 | |
| CDK2 | CDK | CMGC | 1ckp | A | B | purvalanol b | Human | 4214 | |
| CDK2 | CDK | CMGC | 1di8 | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 4577 | |
| CDK2 | CDK | CMGC | 1dm2 | A | A | 4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-one | Human | 4104 | |
| CDK2 | CDK | CMGC | 1dm2 | A | B | 4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-one | Human | 4024 | |
| CDK2 | CDK | CMGC | 1e1v | A | | 6-o-cyclohexylmethyl guanine | Human | 3886 | |
| CDK2 | CDK | CMGC | 1e1x | A | | 6-cyclohexylmethyloxy-5-nitroso-pyrimidine-2,4-diamine | Human | 4114 | |
| CDK2 | CDK | CMGC | 1e9h | A | | 2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acid | Human | 4302 | |
| CDK2 | CDK | CMGC | 1e9h | C | | 2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acid | Human | 4570 | |
| CDK2 | CDK | CMGC | 1f5q | A | A | - | Human | 4194 | |
| CDK2 | CDK | CMGC | 1f5q | A | B | - | Human | 4517 | |
| CDK2 | CDK | CMGC | 1f5q | C | A | - | Human | 4281 | |
| CDK2 | CDK | CMGC | 1f5q | C | B | - | Human | 3952 | |
| CDK2 | CDK | CMGC | 1fin | A | | adenosine-5'-triphosphate | Human | 4367 | |
| CDK2 | CDK | CMGC | 1fin | C | | adenosine-5'-triphosphate | Human | 4479 | |
| CDK2 | CDK | CMGC | 1fq1 | B | | adenosine-5'-triphosphate | Human | 4266 | |
| CDK2 | CDK | CMGC | 1fvt | A | | 4-(5-bromo-2-oxo-2h-indol-3-ylazo)-benzenesulfonamide | Human | 4480 | |
| CDK2 | CDK | CMGC | 1fvv | A | | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 4065 | |
| CDK2 | CDK | CMGC | 1fvv | C | | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 4461 | |
| CDK2 | CDK | CMGC | 1g5s | A | | 2-[trans-(4-aminocyclohexyl)amino]-6-(benzyl-amino)-9-cyclopentylpurine | Human | 3888 | |
| CDK2 | CDK | CMGC | 1gih | A | | 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-urea | Human | 3922 | |
| CDK2 | CDK | CMGC | 1gii | A | | 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-urea | Human | 4448 | |
| CDK2 | CDK | CMGC | 1gij | A | | 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-(5-pyrrolidin-2-yl-1h-pyrazol-3-yl)-urea | Human | 4542 | |
| CDK2 | CDK | CMGC | 1gy3 | A | | adenosine-5'-triphosphate | Human | 3978 | |
| CDK2 | CDK | CMGC | 1gy3 | C | | adenosine-5'-triphosphate | Human | 4445 | |
| CDK2 | CDK | CMGC | 1gz8 | A | A | 1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanol | Human | 3981 | |
| CDK2 | CDK | CMGC | 1gz8 | A | B | 1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanol | Human | 3956 | |
| CDK2 | CDK | CMGC | 1h00 | A | A | (2s)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | 4484 | |
| CDK2 | CDK | CMGC | 1h00 | A | B | (2r)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | 4428 | |
| CDK2 | CDK | CMGC | 1h01 | A | A | (2r)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | 3974 | |
| CDK2 | CDK | CMGC | 1h01 | A | B | (2s)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | 4561 | |
| CDK2 | CDK | CMGC | 1h07 | A | A | ((2-bromo-4-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrile | Human | 3918 | |
| CDK2 | CDK | CMGC | 1h07 | A | B | ((2-bromo-4-methylphenyl){6-[(4-{[(2s)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrile | Human | 3908 | |
| CDK2 | CDK | CMGC | 1h08 | A | A | (2r)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-ol | Human | 4220 | |
| CDK2 | CDK | CMGC | 1h08 | A | B | (2s)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-ol | Human | 4411 | |
| CDK2 | CDK | CMGC | 1h0v | A | A | 5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinone | Human | 4368 | |
| CDK2 | CDK | CMGC | 1h0v | A | B | 5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinone | Human | 3933 | |
| CDK2 | CDK | CMGC | 1h0w | A | A | 1-amino-6-cyclohex-3-enylmethyloxypurine | Human | 3987 | |
| CDK2 | CDK | CMGC | 1h0w | A | B | 1-amino-6-cyclohex-3-enylmethyloxypurine | Human | 4016 | |
| CDK2 | CDK | CMGC | 1h1p | A | | 6-o-cyclohexylmethyl guanine | Human | 4309 | |
| CDK2 | CDK | CMGC | 1h1p | C | | 6-o-cyclohexylmethyl guanine | Human | 4581 | |
| CDK2 | CDK | CMGC | 1h1q | A | | 2-anilino-6-cyclohexylmethoxypurine | Human | 4195 | |
| CDK2 | CDK | CMGC | 1h1q | C | | 2-anilino-6-cyclohexylmethoxypurine | Human | 4053 | |
| CDK2 | CDK | CMGC | 1h1r | A | A | 6-cyclohexylmethoxy-2-(3'-chloroanilino) purine | Human | 3906 | |
| CDK2 | CDK | CMGC | 1h1r | A | B | 6-cyclohexylmethoxy-2-(3'-chloroanilino) purine | Human | 4494 | |
| CDK2 | CDK | CMGC | 1h1r | C | A | 6-cyclohexylmethoxy-2-(3'-chloroanilino) purine | Human | 3920 | |
| CDK2 | CDK | CMGC | 1h1r | C | B | 6-cyclohexylmethoxy-2-(3'-chloroanilino) purine | Human | 4081 | |
| CDK2 | CDK | CMGC | 1h1s | A | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4400 | |
| CDK2 | CDK | CMGC | 1h1s | C | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4572 | |
| CDK2 | CDK | CMGC | 1h24 | A | | - | Human | 4199 | |
| CDK2 | CDK | CMGC | 1h24 | C | | - | Human | 4296 | |
| CDK2 | CDK | CMGC | 1h25 | A | | - | Human | 4273 | |
| CDK2 | CDK | CMGC | 1h25 | C | | - | Human | 4112 | |
| CDK2 | CDK | CMGC | 1h26 | A | | - | Human | 4122 | |
| CDK2 | CDK | CMGC | 1h26 | C | | - | Human | 4179 | |
| CDK2 | CDK | CMGC | 1h27 | A | | - | Human | 4116 | |
| CDK2 | CDK | CMGC | 1h27 | C | | - | Human | 4030 | |
| CDK2 | CDK | CMGC | 1h28 | A | | - | Human | 4169 | |
| CDK2 | CDK | CMGC | 1h28 | C | | - | Human | 4351 | |
| CDK2 | CDK | CMGC | 1hck | A | A | adenosine-5'-triphosphate | Human | 3878 | |
| CDK2 | CDK | CMGC | 1hck | A | B | adenosine-5'-triphosphate | Human | 4416 | |
| CDK2 | CDK | CMGC | 1hcl | A | A | - | Human | 4545 | |
| CDK2 | CDK | CMGC | 1hcl | A | B | - | Human | 4540 | |
| CDK2 | CDK | CMGC | 1jst | A | | adenosine-5'-triphosphate | Human | 4455 | |
| CDK2 | CDK | CMGC | 1jst | C | | adenosine-5'-triphosphate | Human | 4356 | |
| CDK2 | CDK | CMGC | 1jsu | A | | - | Human | 4146 | |
| CDK2 | CDK | CMGC | 1jsv | A | | 4-[(6-amino-4-pyrimidinyl)amino]benzenesulfonamide | Human | 4171 | |
| CDK2 | CDK | CMGC | 1jvp | P | 1 | 3-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazole | Human | 3919 | |
| CDK2 | CDK | CMGC | 1jvp | P | 2 | 3-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazole | Human | 4097 | |
| CDK2 | CDK | CMGC | 1ke5 | A | | n-methyl-4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamide | Human | 4376 | |
| CDK2 | CDK | CMGC | 1ke6 | A | | n-methyl-{4-[2-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)hydrazino]phenyl}methanesulfonamide | Human | 4219 | |
| CDK2 | CDK | CMGC | 1ke7 | A | | 3-{[(2,2-dioxido-1,3-dihydro-2-benzothien-5-yl)amino]methylene}-5-(1,3-oxazol-5-yl)-1,3-dihydro-2h-indol-2-one | Human | 4295 | |
| CDK2 | CDK | CMGC | 1ke8 | A | | 4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}-n-(1,3-thiazol-2-yl)benzenesulfonamide | Human | 4048 | |
| CDK2 | CDK | CMGC | 1ke9 | A | | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4250 | |
| CDK2 | CDK | CMGC | 1ogu | A | A | 4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamide | Human | 3965 | |
| CDK2 | CDK | CMGC | 1ogu | A | B | 4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamide | Human | 3935 | |
| CDK2 | CDK | CMGC | 1ogu | C | A | 4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamide | Human | 3964 | |
| CDK2 | CDK | CMGC | 1ogu | C | B | 4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamide | Human | 4560 | |
| CDK2 | CDK | CMGC | 1oi9 | A | A | 6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purine | Human | 4033 | |
| CDK2 | CDK | CMGC | 1oi9 | A | B | 6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purine | Human | 4492 | |
| CDK2 | CDK | CMGC | 1oi9 | C | A | 6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purine | Human | 4571 | |
| CDK2 | CDK | CMGC | 1oi9 | C | B | 6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purine | Human | 4036 | |
| CDK2 | CDK | CMGC | 1oiq | A | | n-[4-(2-methylimidazo[1,2-a]pyridin-3-yl)-2-pyrimidinyl]acetamide | Human | 4379 | |
| CDK2 | CDK | CMGC | 1oir | A | | 1-(dimethylamino)-3-(4-{{4-(2-methylimidazo[1,2-a]pyridin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-ol | Human | 4389 | |
| CDK2 | CDK | CMGC | 1oit | A | | 4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]benzenesulfonamide | Human | 4025 | |
| CDK2 | CDK | CMGC | 1oiu | A | A | 3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamide | Human | 4110 | |
| CDK2 | CDK | CMGC | 1oiu | A | B | 3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamide | Human | 4556 | |
| CDK2 | CDK | CMGC | 1oiu | C | A | 3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamide | Human | 4524 | |
| CDK2 | CDK | CMGC | 1oiu | C | B | 3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamide | Human | 4049 | |
| CDK2 | CDK | CMGC | 1oiy | A | A | 4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamide | Human | 4225 | |
| CDK2 | CDK | CMGC | 1oiy | A | B | 4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamide | Human | 3945 | |
| CDK2 | CDK | CMGC | 1oiy | C | A | 4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamide | Human | 4465 | |
| CDK2 | CDK | CMGC | 1oiy | C | B | 4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamide | Human | 4245 | |
| CDK2 | CDK | CMGC | 1okv | A | | - | Human | 3921 | |
| CDK2 | CDK | CMGC | 1okv | C | | - | Human | 4093 | |
| CDK2 | CDK | CMGC | 1okw | A | | - | Human | 4314 | |
| CDK2 | CDK | CMGC | 1okw | C | | - | Human | 3896 | |
| CDK2 | CDK | CMGC | 1ol1 | A | | - | Human | 4429 | |
| CDK2 | CDK | CMGC | 1ol1 | C | | - | Human | 3951 | |
| CDK2 | CDK | CMGC | 1ol2 | A | | - | Human | 4305 | |
| CDK2 | CDK | CMGC | 1ol2 | C | | - | Human | 4497 | |
| CDK2 | CDK | CMGC | 1p2a | A | | 5-[(2-aminoethyl)amino]-6-fluoro-3-(1h-pyrrol-2-yl)benzo[cd]indol-2(1h)-one | Human | 4422 | |
| CDK2 | CDK | CMGC | 1p5e | A | | 4,5,6,7-tetrabromobenzotriazole | Human | 4090 | |
| CDK2 | CDK | CMGC | 1p5e | C | | 4,5,6,7-tetrabromobenzotriazole | Human | 4434 | |
| CDK2 | CDK | CMGC | 1pf8 | A | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 3861 | |
| CDK2 | CDK | CMGC | 1pkd | A | | 7-hydroxystaurosporine | Human | 4170 | |
| CDK2 | CDK | CMGC | 1pkd | C | | 7-hydroxystaurosporine | Human | 3973 | |
| CDK2 | CDK | CMGC | 1pw2 | A | | - | Human | 4432 | |
| CDK2 | CDK | CMGC | 1pxi | A | A | 4-(2,5-dichlorothien-3-yl)pyrimidin-2-amine | Human | 4381 | |
| CDK2 | CDK | CMGC | 1pxi | A | B | - | Human | 3924 | |
| CDK2 | CDK | CMGC | 1pxj | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 3927 | |
| CDK2 | CDK | CMGC | 1pxj | A | B | - | Human | 3911 | |
| CDK2 | CDK | CMGC | 1pxk | A | A | n-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n'-hydroxyimidoformamide | Human | 3915 | |
| CDK2 | CDK | CMGC | 1pxk | A | B | - | Human | 3980 | |
| CDK2 | CDK | CMGC | 1pxl | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4233 | |
| CDK2 | CDK | CMGC | 1pxl | A | B | - | Human | 4074 | |
| CDK2 | CDK | CMGC | 1pxm | A | A | 3-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-ylamino]-phenol | Human | 3944 | |
| CDK2 | CDK | CMGC | 1pxm | A | B | - | Human | 3936 | |
| CDK2 | CDK | CMGC | 1pxn | A | A | 4-[4-(4-methyl-2-methylamino-thiazol-5-yl)-pyrimidin-2-ylamino]-phenol | Human | 4383 | |
| CDK2 | CDK | CMGC | 1pxn | A | B | - | Human | 4172 | |
| CDK2 | CDK | CMGC | 1pxo | A | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4512 | |
| CDK2 | CDK | CMGC | 1pxo | A | B | - | Human | 3860 | |
| CDK2 | CDK | CMGC | 1pxo | A | C | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4546 | |
| CDK2 | CDK | CMGC | 1pxo | A | D | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4167 | |
| CDK2 | CDK | CMGC | 1pxp | A | A | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 4316 | |
| CDK2 | CDK | CMGC | 1pxp | A | B | - | Human | 3943 | |
| CDK2 | CDK | CMGC | 1pye | A | | [2-amino-6-(2,6-difluoro-benzoyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl-methanone | Human | 4284 | |
| CDK2 | CDK | CMGC | 1qmz | A | | adenosine-5'-triphosphate | Human | 4242 | |
| CDK2 | CDK | CMGC | 1qmz | C | | adenosine-5'-triphosphate | Human | 4527 | |
| CDK2 | CDK | CMGC | 1r78 | A | A | 4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one | Human | 4253 | |
| CDK2 | CDK | CMGC | 1r78 | A | B | 4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one | Human | 4249 | |
| CDK2 | CDK | CMGC | 1urc | A | A | - | Human | 4334 | |
| CDK2 | CDK | CMGC | 1urc | A | B | - | Human | 4010 | |
| CDK2 | CDK | CMGC | 1urc | C | A | - | Human | 4006 | |
| CDK2 | CDK | CMGC | 1urc | C | B | - | Human | 3937 | |
| CDK2 | CDK | CMGC | 1urw | A | A | 2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]- | Human | 4054 | |
| CDK2 | CDK | CMGC | 1urw | A | B | 2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]- | Human | 4196 | |
| CDK2 | CDK | CMGC | 1v1k | A | A | (2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-ol | Human | 4189 | |
| CDK2 | CDK | CMGC | 1v1k | A | B | (2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-ol | Human | 3928 | |
| CDK2 | CDK | CMGC | 1vyw | A | | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamide | Human | 3992 | |
| CDK2 | CDK | CMGC | 1vyw | C | | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamide | Human | 4133 | |
| CDK2 | CDK | CMGC | 1vyz | A | | n-(5-cyclopropyl-1h-pyrazol-3-yl)benzamide | Human | 4325 | |
| CDK2 | CDK | CMGC | 1w0x | C | A | olomoucine | Human | 4537 | |
| CDK2 | CDK | CMGC | 1w0x | C | B | olomoucine | Human | 4478 | |
| CDK2 | CDK | CMGC | 1w8c | A | A | 6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amine | Human | 4332 | |
| CDK2 | CDK | CMGC | 1w8c | A | B | 6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amine | Human | 4197 | |
| CDK2 | CDK | CMGC | 1w98 | A | | - | Human | 4013 | |
| CDK2 | CDK | CMGC | 1wcc | A | A | 2-amino-6-chloropyrazine | Human | 4394 | |
| CDK2 | CDK | CMGC | 1wcc | A | B | 2-amino-6-chloropyrazine | Human | 3897 | |
| CDK2 | CDK | CMGC | 1y8y | A | | (5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-(4-methanesulfonylphenyl)amine | Human | 3914 | |
| CDK2 | CDK | CMGC | 1y91 | A | | 4-[5-(trans-4-aminocyclohexylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-7-ylamino]-n,n-dimethylbenzenesulfonamide | Human | 4505 | |
| CDK2 | CDK | CMGC | 1ykr | A | | 4-{[6-(2,6-dichlorobenzoyl)imidazo[1,2-a]pyridin-2-yl]amino}benzenesulfonamide | Human | 4578 | |
| CDK2 | CDK | CMGC | 2a0c | X | A | 2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenol | Human | 4157 | |
| CDK2 | CDK | CMGC | 2a0c | X | B | 2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenol | Human | 3868 | |
| CDK2 | CDK | CMGC | 2a4l | A | | r-roscovitine | Human | 4238 | |
| CDK2 | CDK | CMGC | 2b52 | A | | 1-(3-(2,4-dimethylthiazol-5-yl)-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)-3-(4-methylpiperazin-1-yl)urea | Human | 3997 | |
| CDK2 | CDK | CMGC | 2b53 | A | | 6-(3-aminophenyl)-n-(tert-butyl)-2-(trifluoromethyl)quinazolin-4-amine | Human | 3875 | |
| CDK2 | CDK | CMGC | 2b54 | A | | 6-(3,4-dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4(5h)-one | Human | 4292 | |
| CDK2 | CDK | CMGC | 2b55 | A | | 2-(4-(aminomethyl)piperidin-1-yl)-n-(3_cyclohexyl-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)acetamide | Human | 4216 | |
| CDK2 | CDK | CMGC | 2bhe | A | | (2z)-5'-bromo-2,3'-biindole-2',3(1h,1'h)-dione ammoniate | Human | 4184 | |
| CDK2 | CDK | CMGC | 2bhh | A | | (2e,3s)-3-hydroxy-5'-[(4-hydroxypiperidin-1-yl)sulfonyl]-3-methyl-1,3-dihydro-2,3'-biindol-2'(1'h)-one | Human | 4417 | |
| CDK2 | CDK | CMGC | 2bkz | A | | 1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 3942 | |
| CDK2 | CDK | CMGC | 2bkz | C | | 1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 4555 | |
| CDK2 | CDK | CMGC | 2bpm | A | | (2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamide | Human | 4042 | |
| CDK2 | CDK | CMGC | 2bpm | C | | (2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamide | Human | 4128 | |
| CDK2 | CDK | CMGC | 2btr | A | | n-(5-isopropyl-thiazol-2-yl)-2-pyridin-3-yl-acetamide | Human | 3998 | |
| CDK2 | CDK | CMGC | 2bts | A | | 4-[(5-isopropyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 4443 | |
| CDK2 | CDK | CMGC | 2c4g | A | | (3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-ium | Human | 4088 | |
| CDK2 | CDK | CMGC | 2c4g | C | | (3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-ium | Human | 4453 | |
| CDK2 | CDK | CMGC | 2c5n | A | A | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 4063 | |
| CDK2 | CDK | CMGC | 2c5n | A | B | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 4223 | |
| CDK2 | CDK | CMGC | 2c5n | C | A | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 4161 | |
| CDK2 | CDK | CMGC | 2c5n | C | B | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 3903 | |
| CDK2 | CDK | CMGC | 2c5o | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4388 | |
| CDK2 | CDK | CMGC | 2c5o | A | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4440 | |
| CDK2 | CDK | CMGC | 2c5o | C | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4414 | |
| CDK2 | CDK | CMGC | 2c5o | C | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4050 | |
| CDK2 | CDK | CMGC | 2c5v | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4012 | |
| CDK2 | CDK | CMGC | 2c5v | A | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4338 | |
| CDK2 | CDK | CMGC | 2c5v | C | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4384 | |
| CDK2 | CDK | CMGC | 2c5v | C | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4209 | |
| CDK2 | CDK | CMGC | 2c5x | A | A | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 4312 | |
| CDK2 | CDK | CMGC | 2c5x | A | B | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 3892 | |
| CDK2 | CDK | CMGC | 2c5x | C | A | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 4466 | |
| CDK2 | CDK | CMGC | 2c5x | C | B | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 4418 | |
| CDK2 | CDK | CMGC | 2c5y | A | A | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 6785 | |
| CDK2 | CDK | CMGC | 2c5y | A | B | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 6777 | |
| CDK2 | CDK | CMGC | 2c68 | A | | (5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydropyrazolo[1,5-a]pyrimidin-7-amine | Human | 6776 | |
| CDK2 | CDK | CMGC | 2c69 | A | | (5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-7-amine | Human | 6775 | |
| CDK2 | CDK | CMGC | 2c6i | A | | 4-{[5-(cyclohexylmethoxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 6774 | |
| CDK2 | CDK | CMGC | 2c6k | A | | 4-{[5-(cyclohexylamino)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 6773 | |
| CDK2 | CDK | CMGC | 2c6l | A | | 4-({5-[(4-aminocyclohexyl)amino][1,2,4]triazolo[1,5-a]pyrimidin-7-yl}amino)benzenesulfonamide | Human | 6779 | |
| CDK2 | CDK | CMGC | 2c6m | A | | 4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 6782 | |
| CDK2 | CDK | CMGC | 2c6o | A | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 6783 | |
| CDK2 | CDK | CMGC | 2c6t | A | | 4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 4371 | |
| CDK2 | CDK | CMGC | 2c6t | C | | 4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 3994 | |
| CDK2 | CDK | CMGC | 2cch | A | A | adenosine-5'-triphosphate | Human | 4303 | |
| CDK2 | CDK | CMGC | 2cch | A | B | adenosine-5'-triphosphate | Human | 4553 | |
| CDK2 | CDK | CMGC | 2cch | A | C | - | Human | 4566 | |
| CDK2 | CDK | CMGC | 2cch | C | A | adenosine-5'-triphosphate | Human | 3932 | |
| CDK2 | CDK | CMGC | 2cch | C | B | adenosine-5'-triphosphate | Human | 4000 | |
| CDK2 | CDK | CMGC | 2cch | C | C | - | Human | 4431 | |
| CDK2 | CDK | CMGC | 2cci | A | | adenosine-5'-triphosphate | Human | 4373 | |
| CDK2 | CDK | CMGC | 2cci | C | | adenosine-5'-triphosphate | Human | 4532 | |
| CDK2 | CDK | CMGC | 2cjm | A | | adenosine-5'-triphosphate | Human | 4406 | |
| CDK2 | CDK | CMGC | 2cjm | C | | adenosine-5'-triphosphate | Human | 4126 | |
| CDK2 | CDK | CMGC | 2clx | A | A | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 3909 | |
| CDK2 | CDK | CMGC | 2clx | A | B | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 3880 | |
| CDK2 | CDK | CMGC | 2ds1 | A | | (13r,15s)-13-methyl-16-oxa-8,9,12,22,24-pentaazahexacyclo[15.6.2.16,9.1,12,15.0,2,7.0,21,25]heptacosa-1(24),2,4,6,17(25),18,20-heptaene-23,26-dione | Human | 4513 | |
| CDK2 | CDK | CMGC | 2duv | A | | 2-(3,4-dihydroxyphenyl)-8-(1,1-dioxidoisothiazolidin-2-yl)-3-hydroxy-6-methyl-4h-chromen-4-one | Human | 4193 | |
| CDK2 | CDK | CMGC | 2exm | A | | n-(3-methylbut-2-en-1-yl)-9h-purin-6-amine | Human | 4055 | |
| CDK2 | CDK | CMGC | 2fvd | A | | (4-amino-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrimidin-5-yl)(2,3-difluoro-6-methoxyphenyl)methanone | Human | 4408 | |
| CDK2 | CDK | CMGC | 2g9x | A | | 3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-ol | Human | 3883 | |
| CDK2 | CDK | CMGC | 2g9x | C | | 3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-ol | Human | 4082 | |
| CDK2 | CDK | CMGC | 2i40 | A | A | 5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamide | Human | 4363 | |
| CDK2 | CDK | CMGC | 2i40 | A | B | 5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamide | Human | 4470 | |
| CDK2 | CDK | CMGC | 2i40 | C | A | 5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamide | Human | 4222 | |
| CDK2 | CDK | CMGC | 2i40 | C | B | 5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamide | Human | 4043 | |
| CDK2 | CDK | CMGC | 2iw6 | A | | [(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrile | Human | 4019 | |
| CDK2 | CDK | CMGC | 2iw6 | C | | [(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrile | Human | 4108 | |
| CDK2 | CDK | CMGC | 2iw8 | A | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4142 | |
| CDK2 | CDK | CMGC | 2iw8 | A | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4377 | |
| CDK2 | CDK | CMGC | 2iw8 | C | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4294 | |
| CDK2 | CDK | CMGC | 2iw8 | C | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4350 | |
| CDK2 | CDK | CMGC | 2iw9 | A | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4174 | |
| CDK2 | CDK | CMGC | 2iw9 | A | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 3955 | |
| CDK2 | CDK | CMGC | 2iw9 | C | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4218 | |
| CDK2 | CDK | CMGC | 2iw9 | C | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 3858 | |
| CDK2 | CDK | CMGC | 2j9m | A | A | 6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxide | Human | 4154 | |
| CDK2 | CDK | CMGC | 2j9m | A | B | 6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxide | Human | 4246 | |
| CDK2 | CDK | CMGC | 2jgz | A | | - | Human | 4117 | |
| CDK2 | CDK | CMGC | 2r3f | A | A | 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4175 | |
| CDK2 | CDK | CMGC | 2r3f | A | B | 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4291 | |
| CDK2 | CDK | CMGC | 2r3g | A | A | 6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amine | Human | 4276 | |
| CDK2 | CDK | CMGC | 2r3g | A | B | 6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amine | Human | 3923 | |
| CDK2 | CDK | CMGC | 2r3h | A | A | 3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amine | Human | 4152 | |
| CDK2 | CDK | CMGC | 2r3h | A | B | 3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amine | Human | 3970 | |
| CDK2 | CDK | CMGC | 2r3i | A | A | 5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4135 | |
| CDK2 | CDK | CMGC | 2r3i | A | B | 5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4059 | |
| CDK2 | CDK | CMGC | 2r3i | A | C | - | Human | 4317 | |
| CDK2 | CDK | CMGC | 2r3j | A | A | 3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4185 | |
| CDK2 | CDK | CMGC | 2r3j | A | B | 3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4544 | |
| CDK2 | CDK | CMGC | 2r3k | A | A | 3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amine | Human | 3953 | |
| CDK2 | CDK | CMGC | 2r3k | A | B | 3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amine | Human | 3876 | |
| CDK2 | CDK | CMGC | 2r3k | A | C | 3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amine | Human | 4022 | |
| CDK2 | CDK | CMGC | 2r3l | A | A | 3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amine | Human | 4200 | |
| CDK2 | CDK | CMGC | 2r3l | A | B | 3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amine | Human | 4085 | |
| CDK2 | CDK | CMGC | 2r3l | A | C | 3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amine | Human | 4496 | |
| CDK2 | CDK | CMGC | 2r3m | A | A | n-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amine | Human | 4286 | |
| CDK2 | CDK | CMGC | 2r3m | A | B | n-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amine | Human | 4576 | |
| CDK2 | CDK | CMGC | 2r3n | A | A | 3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4101 | |
| CDK2 | CDK | CMGC | 2r3n | A | B | 3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4046 | |
| CDK2 | CDK | CMGC | 2r3o | A | A | (5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanol | Human | 4147 | |
| CDK2 | CDK | CMGC | 2r3o | A | B | (5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanol | Human | 4354 | |
| CDK2 | CDK | CMGC | 2r3o | A | C | (5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanol | Human | 4229 | |
| CDK2 | CDK | CMGC | 2r3p | A | A | 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amine | Human | 4176 | |
| CDK2 | CDK | CMGC | 2r3p | A | B | 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amine | Human | 4392 | |
| CDK2 | CDK | CMGC | 2r3q | A | A | 3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxide | Human | 4038 | |
| CDK2 | CDK | CMGC | 2r3q | A | B | 3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxide | Human | 4459 | |
| CDK2 | CDK | CMGC | 2r3q | A | C | 3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxide | Human | 3976 | |
| CDK2 | CDK | CMGC | 2r3r | A | A | 3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4040 | |
| CDK2 | CDK | CMGC | 2r3r | A | B | 3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4215 | |
| CDK2 | CDK | CMGC | 2r64 | A | | n-[5-(1,1-dioxidoisothiazolidin-2-yl)-1h-indazol-3-yl]-2-(4-piperidin-1-ylphenyl)acetamide | Human | 4425 | |
| CDK2 | CDK | CMGC | 2uue | A | | 4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amine | Human | 4515 | |
| CDK2 | CDK | CMGC | 2uue | C | | 4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amine | Human | 4321 | |
| CDK2 | CDK | CMGC | 2uzb | A | C | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamide | Human | 4099 | |
| CDK2 | CDK | CMGC | 2uzb | A | D | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamide | Human | 3866 | |
| CDK2 | CDK | CMGC | 2uzb | C | C | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamide | Human | 4045 | |
| CDK2 | CDK | CMGC | 2uzb | C | D | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamide | Human | 4502 | |
| CDK2 | CDK | CMGC | 2uzd | A | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamide | Human | 3877 | |
| CDK2 | CDK | CMGC | 2uzd | C | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamide | Human | 3900 | |
| CDK2 | CDK | CMGC | 2uze | A | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acid | Human | 3949 | |
| CDK2 | CDK | CMGC | 2uze | C | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acid | Human | 4071 | |
| CDK2 | CDK | CMGC | 2uzl | A | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamide | Human | 3917 | |
| CDK2 | CDK | CMGC | 2uzl | C | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamide | Human | 4106 | |
| CDK2 | CDK | CMGC | 2uzn | A | | 4-{5-[(1z)-1-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)ethyl]-2-furyl}benzenesulfonamide | Human | 4064 | |
| CDK2 | CDK | CMGC | 2uzo | A | | 4-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamide | Human | 3862 | |
| CDK2 | CDK | CMGC | 2v0d | A | | 2-imino-5-(1-pyridin-2-yl-meth-(e)-ylidene)-1,3-thiazolidin-4-one | Human | 4327 | |
| CDK2 | CDK | CMGC | 2v22 | A | | - | Human | 4077 | |
| CDK2 | CDK | CMGC | 2v22 | C | | - | Human | 4255 | |
| CDK2 | CDK | CMGC | 2vta | A | | 1h-indazole | Human | 4118 | |
| CDK2 | CDK | CMGC | 2vth | A | | 5-hydroxynaphthalene-1-sulfonamide | Human | 4274 | |
| CDK2 | CDK | CMGC | 2vti | A | | n-(4-sulfamoylphenyl)-1h-indazole-3-carboxamide | Human | 4177 | |
| CDK2 | CDK | CMGC | 2vtj | A | | 4-[(6-chloropyrazin-2-yl)amino]benzenesulfonamide | Human | 3959 | |
| CDK2 | CDK | CMGC | 2vtl | A | | n-phenyl-1h-pyrazole-3-carboxamide | Human | 3870 | |
| CDK2 | CDK | CMGC | 2vtm | A | | pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 4283 | |
| CDK2 | CDK | CMGC | 2vtn | A | | 4-(acetylamino)-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4027 | |
| CDK2 | CDK | CMGC | 2vto | A | A | n-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamide | Human | 4421 | |
| CDK2 | CDK | CMGC | 2vto | A | B | n-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamide | Human | 3946 | |
| CDK2 | CDK | CMGC | 2vtp | A | A | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4511 | |
| CDK2 | CDK | CMGC | 2vtp | A | B | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4401 | |
| CDK2 | CDK | CMGC | 2vtq | A | | {[(2,6-difluorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamide | Human | 3891 | |
| CDK2 | CDK | CMGC | 2vtr | A | A | 5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 4391 | |
| CDK2 | CDK | CMGC | 2vtr | A | B | 5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 3907 | |
| CDK2 | CDK | CMGC | 2vts | A | | 5-[(4-aminocyclohexyl)amino]-7-(propan-2-ylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 4300 | |
| CDK2 | CDK | CMGC | 2vtt | A | | 4-{[(2,6-difluorophenyl)carbonyl]amino}-n-[(3s)-piperidin-3-yl]-1h-pyrazole-3-carboxamide | Human | 4100 | |
| CDK2 | CDK | CMGC | 2vu3 | A | A | 4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamide | Human | 4582 | |
| CDK2 | CDK | CMGC | 2vu3 | A | B | 4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamide | Human | 3884 | |
| CDK2 | CDK | CMGC | 2vv9 | A | A | 2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanol | Human | 3989 | |
| CDK2 | CDK | CMGC | 2vv9 | A | B | 2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanol | Human | 3881 | |
| CDK2 | CDK | CMGC | 2w05 | A | A | n-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 4547 | |
| CDK2 | CDK | CMGC | 2w05 | A | B | n-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 4256 | |
| CDK2 | CDK | CMGC | 2w06 | A | | 4-{[4-(1-cyclopropyl-2-methyl-1h-imidazol-5-yl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 3982 | |
| CDK2 | CDK | CMGC | 2w17 | A | A | n-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 3968 | |
| CDK2 | CDK | CMGC | 2w17 | A | B | n-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 4165 | |
| CDK2 | CDK | CMGC | 2w1h | A | | n-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamide | Human | 4228 | |
| CDK2 | CDK | CMGC | 2wev | A | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4067 | |
| CDK2 | CDK | CMGC | 2wev | A | B | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4580 | |
| CDK2 | CDK | CMGC | 2wev | A | C | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4007 | |
| CDK2 | CDK | CMGC | 2wev | C | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4503 | |
| CDK2 | CDK | CMGC | 2wev | C | B | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 3859 | |
| CDK2 | CDK | CMGC | 2wev | C | C | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4288 | |
| CDK2 | CDK | CMGC | 2wfy | A | A | - | Human | 4324 | |
| CDK2 | CDK | CMGC | 2wfy | A | B | - | Human | 4426 | |
| CDK2 | CDK | CMGC | 2wfy | C | A | - | Human | 4329 | |
| CDK2 | CDK | CMGC | 2wfy | C | B | - | Human | 4096 | |
| CDK2 | CDK | CMGC | 2whb | A | A | - | Human | 4471 | |
| CDK2 | CDK | CMGC | 2whb | A | B | - | Human | 4457 | |
| CDK2 | CDK | CMGC | 2whb | C | A | - | Human | 4132 | |
| CDK2 | CDK | CMGC | 2whb | C | B | - | Human | 4352 | |
| CDK2 | CDK | CMGC | 2wih | A | | n,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4163 | |
| CDK2 | CDK | CMGC | 2wih | C | | n,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4119 | |
| CDK2 | CDK | CMGC | 2wip | A | | 1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acid | Human | 4520 | |
| CDK2 | CDK | CMGC | 2wip | C | | 1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acid | Human | 4190 | |
| CDK2 | CDK | CMGC | 2wma | A | | - | Human | 4435 | |
| CDK2 | CDK | CMGC | 2wma | C | | - | Human | 4410 | |
| CDK2 | CDK | CMGC | 2wmb | A | | - | Human | 4060 | |
| CDK2 | CDK | CMGC | 2wmb | C | | - | Human | 4474 | |
| CDK2 | CDK | CMGC | 2wpa | A | | n-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamide | Human | 4399 | |
| CDK2 | CDK | CMGC | 2wpa | C | | n-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamide | Human | 4162 | |
| CDK2 | CDK | CMGC | 2wxv | A | | n,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4318 | |
| CDK2 | CDK | CMGC | 2wxv | C | | n,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4504 | |
| CDK2 | CDK | CMGC | 2x1n | A | A | 2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amine | Human | 4579 | |
| CDK2 | CDK | CMGC | 2x1n | A | B | 2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amine | Human | 4078 | |
| CDK2 | CDK | CMGC | 2x1n | C | A | 2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amine | Human | 3991 | |
| CDK2 | CDK | CMGC | 2x1n | C | B | 2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amine | Human | 4062 | |
| CDK2 | CDK | CMGC | 2xmy | A | A | 4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamide | Human | 4526 | |
| CDK2 | CDK | CMGC | 2xmy | A | B | 4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamide | Human | 3985 | |
| CDK2 | CDK | CMGC | 2xnb | A | A | 3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-one | Human | 4217 | |
| CDK2 | CDK | CMGC | 2xnb | A | B | 3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-one | Human | 4034 | |
| CDK2 | CDK | CMGC | 3bht | A | A | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 3950 | |
| CDK2 | CDK | CMGC | 3bht | A | B | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4491 | |
| CDK2 | CDK | CMGC | 3bht | C | A | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4151 | |
| CDK2 | CDK | CMGC | 3bht | C | B | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 3889 | |
| CDK2 | CDK | CMGC | 3bhu | A | A | 4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4105 | |
| CDK2 | CDK | CMGC | 3bhu | A | B | 4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4446 | |
| CDK2 | CDK | CMGC | 3bhu | C | A | 4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4087 | |
| CDK2 | CDK | CMGC | 3bhu | C | B | 4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4464 | |
| CDK2 | CDK | CMGC | 3bhv | A | A | 9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-ol | Human | 4531 | |
| CDK2 | CDK | CMGC | 3bhv | A | B | 9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-ol | Human | 4001 | |
| CDK2 | CDK | CMGC | 3bhv | C | A | 9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-ol | Human | 4353 | |
| CDK2 | CDK | CMGC | 3bhv | C | B | 9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-ol | Human | 4529 | |
| CDK2 | CDK | CMGC | 3ddp | A | A | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 6781 | |
| CDK2 | CDK | CMGC | 3ddp | A | B | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 6780 | |
| CDK2 | CDK | CMGC | 3ddp | C | A | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 6784 | |
| CDK2 | CDK | CMGC | 3ddp | C | B | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 6778 | |
| CDK2 | CDK | CMGC | 3ddq | A | A | r-roscovitine | Human | 4477 | |
| CDK2 | CDK | CMGC | 3ddq | A | B | r-roscovitine | Human | 4269 | |
| CDK2 | CDK | CMGC | 3ddq | C | A | r-roscovitine | Human | 4364 | |
| CDK2 | CDK | CMGC | 3ddq | C | B | r-roscovitine | Human | 4289 | |
| CDK2 | CDK | CMGC | 3dog | A | A | (2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol | Human | 4541 | |
| CDK2 | CDK | CMGC | 3dog | A | B | (2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol | Human | 4365 | |
| CDK2 | CDK | CMGC | 3dog | C | A | (2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol | Human | 4382 | |
| CDK2 | CDK | CMGC | 3dog | C | B | (2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol | Human | 4121 | |
| CDK2 | CDK | CMGC | 3eid | A | A | (2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-ol | Human | 4386 | |
| CDK2 | CDK | CMGC | 3eid | A | B | (2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-ol | Human | 4424 | |
| CDK2 | CDK | CMGC | 3eid | C | A | - | Human | 4072 | |
| CDK2 | CDK | CMGC | 3eid | C | B | - | Human | 4467 | |
| CDK2 | CDK | CMGC | 3ej1 | A | | n-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amine | Human | 4168 | |
| CDK2 | CDK | CMGC | 3ej1 | C | | n-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amine | Human | 4092 | |
| CDK2 | CDK | CMGC | 3eoc | A | | 5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine | Human | 4390 | |
| CDK2 | CDK | CMGC | 3eoc | C | | 5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine | Human | 3969 | |
| CDK2 | CDK | CMGC | 3ezr | A | | 3-methoxy-4-{3-[4-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}aniline | Human | 4475 | |
| CDK2 | CDK | CMGC | 3ezv | A | | 4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}aniline | Human | 4083 | |
| CDK2 | CDK | CMGC | 3f5x | A | | 4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}aniline | Human | 3882 | |
| CDK2 | CDK | CMGC | 3f5x | C | | 4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}aniline | Human | 3894 | |
| CDK2 | CDK | CMGC | 3fz1 | A | | (3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-one | Human | 4335 | |
| CDK2 | CDK | CMGC | 3ig7 | A | | n-{1-[cis-3-(acetylamino)cyclobutyl]-1h-imidazol-4-yl}-2-(4-methoxyphenyl)acetamide | Human | 4021 | |
| CDK2 | CDK | CMGC | 3igg | A | | n-[1-(cis-3-hydroxycyclobutyl)-1h-imidazol-4-yl]-2-(4-methoxyphenyl)acetamide | Human | 4360 | |
| CDK2 | CDK | CMGC | 3le6 | A | | 5-(2-chlorophenyl)-3-methyl-7-nitropyrazolo[3,4-b][1,4]benzodiazepine | Human | 4125 | |
| CDK2 | CDK | CMGC | 3lfn | A | | n-[6-(4-hydroxyphenyl)-5-phenyl-1h-indazol-3-yl]butanamide | Human | 4330 | |
| CDK2 | CDK | CMGC | 3lfq | A | | n-(6,7-difluoro-5-phenyl-1h-indazol-3-yl)butanamide | Human | 4320 | |
| CDK2 | CDK | CMGC | 3lfs | A | | n-(6-chloro-5-phenyl-1h-indazol-3-yl)butanamide | Human | 4069 | |
| CDK2 | CDK | CMGC | 3my5 | A | A | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 4554 | |
| CDK2 | CDK | CMGC | 3my5 | A | B | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 3887 | |
| CDK2 | CDK | CMGC | 3my5 | A | C | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 3910 | |
| CDK2 | CDK | CMGC | 3my5 | C | A | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 4473 | |
| CDK2 | CDK | CMGC | 3my5 | C | B | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 4003 | |
| CDK2 | CDK | CMGC | 3my5 | C | C | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 3929 | |
| CDK2 | CDK | CMGC | 3ns9 | A | | (2s,3s)-3-{[7-(benzylamino)-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-5-yl]amino}butane-1,2,4-triol | Human | 4575 | |
| CDK2 | CDK | CMGC | 3pj8 | A | A | (2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-ol | Human | 4375 | |
| CDK2 | CDK | CMGC | 3pj8 | A | B | (2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-ol | Human | 4454 | |
| CDK2 | CDK | CMGC | 3pxf | A | A | 8-anilino-1-naphthalene sulfonate | Human | 4047 | |
| CDK2 | CDK | CMGC | 3pxf | A | B | 8-anilino-1-naphthalene sulfonate | Human | 4301 | |
| CDK2 | CDK | CMGC | 3pxq | A | | 8-anilino-1-naphthalene sulfonate | Human | 3947 | |
| CDK2 | CDK | CMGC | 3pxr | A | A | - | Human | 3941 | |
| CDK2 | CDK | CMGC | 3pxr | A | B | - | Human | 4173 | |
| CDK2 | CDK | CMGC | 3pxy | A | A | 2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenol | Human | 4057 | |
| CDK2 | CDK | CMGC | 3pxy | A | B | 2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenol | Human | 3904 | |
| CDK2 | CDK | CMGC | 3pxz | A | | 8-anilino-1-naphthalene sulfonate | Human | 4251 | |
| CDK2 | CDK | CMGC | 3py0 | A | A | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 3995 | |
| CDK2 | CDK | CMGC | 3py0 | A | B | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 3869 | |
| CDK2 | CDK | CMGC | 3py1 | A | A | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 4361 | |
| CDK2 | CDK | CMGC | 3py1 | A | B | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 4444 | |
| CDK2 | CDK | CMGC | 3qhr | A | | adenosine-5'-diphosphate | Human | 4458 | |
| CDK2 | CDK | CMGC | 3qhr | C | | adenosine-5'-diphosphate | Human | 3879 | |
| CDK2 | CDK | CMGC | 3qhw | A | A | adenosine-5'-diphosphate | Human | 4346 | |
| CDK2 | CDK | CMGC | 3qhw | A | B | adenosine-5'-diphosphate | Human | 4156 | |
| CDK2 | CDK | CMGC | 3qhw | C | A | adenosine-5'-diphosphate | Human | 4129 | |
| CDK2 | CDK | CMGC | 3qhw | C | B | adenosine-5'-diphosphate | Human | 4143 | |
| CDK2 | CDK | CMGC | 3ql8 | A | A | 3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrile | Human | 3916 | |
| CDK2 | CDK | CMGC | 3ql8 | A | B | 3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrile | Human | 4306 | |
| CDK2 | CDK | CMGC | 3qqf | A | A | 5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4211 | |
| CDK2 | CDK | CMGC | 3qqf | A | B | 5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4287 | |
| CDK2 | CDK | CMGC | 3qqg | A | A | 4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 4130 | |
| CDK2 | CDK | CMGC | 3qqg | A | B | 4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 4310 | |
| CDK2 | CDK | CMGC | 3qqh | A | A | 2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenol | Human | 4393 | |
| CDK2 | CDK | CMGC | 3qqh | A | B | 2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenol | Human | 4533 | |
| CDK2 | CDK | CMGC | 3qqj | A | A | 2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 4113 | |
| CDK2 | CDK | CMGC | 3qqj | A | B | 2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 4204 | |
| CDK2 | CDK | CMGC | 3qqk | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 4568 | |
| CDK2 | CDK | CMGC | 3qqk | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 4514 | |
| CDK2 | CDK | CMGC | 3qql | A | A | (5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4341 | |
| CDK2 | CDK | CMGC | 3qql | A | B | (5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4378 | |
| CDK2 | CDK | CMGC | 3qrt | A | A | (5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 4586 | |
| CDK2 | CDK | CMGC | 3qrt | A | B | (5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 4536 | |
| CDK2 | CDK | CMGC | 3qru | A | A | (5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 4237 | |
| CDK2 | CDK | CMGC | 3qru | A | B | (5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 4516 | |
| CDK2 | CDK | CMGC | 3qtq | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4210 | |
| CDK2 | CDK | CMGC | 3qtq | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4103 | |
| CDK2 | CDK | CMGC | 3qtr | A | A | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 3874 | |
| CDK2 | CDK | CMGC | 3qtr | A | B | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 4243 | |
| CDK2 | CDK | CMGC | 3qts | A | A | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanone | Human | 4275 | |
| CDK2 | CDK | CMGC | 3qts | A | B | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanone | Human | 4564 | |
| CDK2 | CDK | CMGC | 3qtu | A | A | 4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4009 | |
| CDK2 | CDK | CMGC | 3qtu | A | B | 4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4323 | |
| CDK2 | CDK | CMGC | 3qtw | A | A | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4397 | |
| CDK2 | CDK | CMGC | 3qtw | A | B | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 3890 | |
| CDK2 | CDK | CMGC | 3qtx | A | A | 4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4339 | |
| CDK2 | CDK | CMGC | 3qtx | A | B | 4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4419 | |
| CDK2 | CDK | CMGC | 3qtz | A | A | 4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4109 | |
| CDK2 | CDK | CMGC | 3qtz | A | B | 4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4337 | |
| CDK2 | CDK | CMGC | 3qu0 | A | A | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4427 | |
| CDK2 | CDK | CMGC | 3qu0 | A | B | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4558 | |
| CDK2 | CDK | CMGC | 3qwj | A | A | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamide | Human | 4265 | |
| CDK2 | CDK | CMGC | 3qwj | A | B | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamide | Human | 4182 | |
| CDK2 | CDK | CMGC | 3qwk | A | A | 4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamide | Human | 4091 | |
| CDK2 | CDK | CMGC | 3qwk | A | B | 4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamide | Human | 4155 | |
| CDK2 | CDK | CMGC | 3qx2 | A | A | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamide | Human | 4031 | |
| CDK2 | CDK | CMGC | 3qx2 | A | B | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamide | Human | 4297 | |
| CDK2 | CDK | CMGC | 3qx4 | A | A | 4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4409 | |
| CDK2 | CDK | CMGC | 3qx4 | A | B | 4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 3990 | |
| CDK2 | CDK | CMGC | 3qxo | A | | 5-nitro-2-[(4-sulfamoylbenzyl)amino]benzamide | Human | 4282 | |
| CDK2 | CDK | CMGC | 3qxp | A | A | 4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4343 | |
| CDK2 | CDK | CMGC | 3qxp | A | B | 4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4482 | |
| CDK2 | CDK | CMGC | 3qzf | A | | 2-(4,6-diamino-1,3,5-triazin-2-yl)benzene-1,4-diol | Human | 4569 | |
| CDK2 | CDK | CMGC | 3qzg | A | A | 2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenol | Human | 4144 | |
| CDK2 | CDK | CMGC | 3qzg | A | B | 2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenol | Human | 4347 | |
| CDK2 | CDK | CMGC | 3qzh | A | | 4-methoxy-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 3954 | |
| CDK2 | CDK | CMGC | 3qzi | A | A | 4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamide | Human | 4094 | |
| CDK2 | CDK | CMGC | 3qzi | A | B | 4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamide | Human | 4500 | |
| CDK2 | CDK | CMGC | 3r1q | A | A | 4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamide | Human | 4224 | |
| CDK2 | CDK | CMGC | 3r1q | A | B | 4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamide | Human | 4507 | |
| CDK2 | CDK | CMGC | 3r1s | A | A | 2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamide | Human | 4263 | |
| CDK2 | CDK | CMGC | 3r1s | A | B | 2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamide | Human | 4358 | |
| CDK2 | CDK | CMGC | 3r1y | A | A | 2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4319 | |
| CDK2 | CDK | CMGC | 3r1y | A | B | 2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4405 | |
| CDK2 | CDK | CMGC | 3r28 | A | A | 4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamide | Human | 4052 | |
| CDK2 | CDK | CMGC | 3r28 | A | B | 4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamide | Human | 4293 | |
| CDK2 | CDK | CMGC | 3r6x | A | A | 4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4398 | |
| CDK2 | CDK | CMGC | 3r6x | A | B | 4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4107 | |
| CDK2 | CDK | CMGC | 3r71 | A | A | 4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 3962 | |
| CDK2 | CDK | CMGC | 3r71 | A | B | 4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4345 | |
| CDK2 | CDK | CMGC | 3r73 | A | A | 4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4187 | |
| CDK2 | CDK | CMGC | 3r73 | A | B | 4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 3899 | |
| CDK2 | CDK | CMGC | 3r7e | A | A | 5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamide | Human | 4159 | |
| CDK2 | CDK | CMGC | 3r7e | A | B | 5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamide | Human | 4447 | |
| CDK2 | CDK | CMGC | 3r7i | A | A | 4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acid | Human | 4450 | |
| CDK2 | CDK | CMGC | 3r7i | A | B | 4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acid | Human | 4070 | |
| CDK2 | CDK | CMGC | 3r7u | A | A | 2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamide | Human | 4510 | |
| CDK2 | CDK | CMGC | 3r7u | A | B | 2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamide | Human | 4023 | |
| CDK2 | CDK | CMGC | 3r7v | A | A | 5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamide | Human | 4380 | |
| CDK2 | CDK | CMGC | 3r7v | A | B | 5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamide | Human | 4183 | |
| CDK2 | CDK | CMGC | 3r7y | A | A | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamide | Human | 4476 | |
| CDK2 | CDK | CMGC | 3r7y | A | B | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamide | Human | 3975 | |
| CDK2 | CDK | CMGC | 3r83 | A | A | 4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamide | Human | 4234 | |
| CDK2 | CDK | CMGC | 3r83 | A | B | 4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamide | Human | 4543 | |
| CDK2 | CDK | CMGC | 3r8l | A | A | (5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4186 | |
| CDK2 | CDK | CMGC | 3r8l | A | B | (5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4523 | |
| CDK2 | CDK | CMGC | 3r8m | A | A | 1h-indazole-3-carbohydrazide | Human | 4111 | |
| CDK2 | CDK | CMGC | 3r8m | A | B | 1h-indazole-3-carbohydrazide | Human | 4451 | |
| CDK2 | CDK | CMGC | 3r8p | A | A | (5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4232 | |
| CDK2 | CDK | CMGC | 3r8p | A | B | (5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4538 | |
| CDK2 | CDK | CMGC | 3r8u | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | 3926 | |
| CDK2 | CDK | CMGC | 3r8u | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | 3864 | |
| CDK2 | CDK | CMGC | 3r8v | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | 3938 | |
| CDK2 | CDK | CMGC | 3r8v | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | 4191 | |
| CDK2 | CDK | CMGC | 3r8z | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanone | Human | 4137 | |
| CDK2 | CDK | CMGC | 3r8z | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanone | Human | 4140 | |
| CDK2 | CDK | CMGC | 3r9d | A | A | 4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4562 | |
| CDK2 | CDK | CMGC | 3r9d | A | B | 4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4565 | |
| CDK2 | CDK | CMGC | 3r9h | A | A | 4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 3958 | |
| CDK2 | CDK | CMGC | 3r9h | A | B | 4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4336 | |
| CDK2 | CDK | CMGC | 3r9n | A | A | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | 3885 | |
| CDK2 | CDK | CMGC | 3r9n | A | B | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | 3867 | |
| CDK2 | CDK | CMGC | 3r9o | A | | 4-amino-n-(3,5-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4279 | |
| CDK2 | CDK | CMGC | 3rah | A | A | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | 4438 | |
| CDK2 | CDK | CMGC | 3rah | A | B | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | 4206 | |
| CDK2 | CDK | CMGC | 3rai | A | A | 4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4441 | |
| CDK2 | CDK | CMGC | 3rai | A | B | 4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4002 | |
| CDK2 | CDK | CMGC | 3rak | A | A | 4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 4574 | |
| CDK2 | CDK | CMGC | 3rak | A | B | 4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 4331 | |
| CDK2 | CDK | CMGC | 3ral | A | A | 4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4017 | |
| CDK2 | CDK | CMGC | 3ral | A | B | 4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 3984 | |
| CDK2 | CDK | CMGC | 3rjc | A | A | {4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanone | Human | 4032 | |
| CDK2 | CDK | CMGC | 3rjc | A | B | {4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanone | Human | 4469 | |
| CDK2 | CDK | CMGC | 3rk5 | A | | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzoic acid | Human | 4160 | |
| CDK2 | CDK | CMGC | 3rk7 | A | | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzamide | Human | 4236 | |
| CDK2 | CDK | CMGC | 3rk9 | A | A | [4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4158 | |
| CDK2 | CDK | CMGC | 3rk9 | A | B | [4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4259 | |
| CDK2 | CDK | CMGC | 3rkb | A | A | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4460 | |
| CDK2 | CDK | CMGC | 3rkb | A | B | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4039 | |
| CDK2 | CDK | CMGC | 3rm6 | A | A | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamide | Human | 4262 | |
| CDK2 | CDK | CMGC | 3rm6 | A | B | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamide | Human | 4357 | |
| CDK2 | CDK | CMGC | 3rm7 | A | A | 2-[(4-hydroxybenzyl)amino]-5-nitrobenzamide | Human | 3893 | |
| CDK2 | CDK | CMGC | 3rm7 | A | B | 2-[(4-hydroxybenzyl)amino]-5-nitrobenzamide | Human | 4499 | |
| CDK2 | CDK | CMGC | 3rmf | A | A | 4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 3873 | |
| CDK2 | CDK | CMGC | 3rmf | A | B | 4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4014 | |
| CDK2 | CDK | CMGC | 3rni | A | A | 3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 3993 | |
| CDK2 | CDK | CMGC | 3rni | A | B | 3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 4420 | |
| CDK2 | CDK | CMGC | 3roy | A | A | 4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4131 | |
| CDK2 | CDK | CMGC | 3roy | A | B | 4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4239 | |
| CDK2 | CDK | CMGC | 3rpo | A | A | 4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acid | Human | 3966 | |
| CDK2 | CDK | CMGC | 3rpo | A | B | 4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acid | Human | 4098 | |
| CDK2 | CDK | CMGC | 3rpr | A | A | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanone | Human | 4452 | |
| CDK2 | CDK | CMGC | 3rpr | A | B | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanone | Human | 4241 | |
| CDK2 | CDK | CMGC | 3rpv | A | A | 4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4348 | |
| CDK2 | CDK | CMGC | 3rpv | A | B | 4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4372 | |
| CDK2 | CDK | CMGC | 3rpy | A | A | 4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4261 | |
| CDK2 | CDK | CMGC | 3rpy | A | B | 4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4519 | |
| CDK2 | CDK | CMGC | 3rzb | A | A | 4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamide | Human | 4264 | |
| CDK2 | CDK | CMGC | 3rzb | A | B | 4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamide | Human | 4395 | |
| CDK2 | CDK | CMGC | 3s00 | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanone | Human | 4208 | |
| CDK2 | CDK | CMGC | 3s00 | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanone | Human | 4248 | |
| CDK2 | CDK | CMGC | 3s0o | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanone | Human | 3898 | |
| CDK2 | CDK | CMGC | 3s0o | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanone | Human | 4123 | |
| CDK2 | CDK | CMGC | 3s1h | A | A | 4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4068 | |
| CDK2 | CDK | CMGC | 3s1h | A | B | 4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4226 | |
| CDK2 | CDK | CMGC | 3s2p | A | | (3s,4s)-1-{3-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-4-hydroxyphenyl}pyrrolidine-3,4-diol | Human | 4404 | |
| CDK2 | CDK | CMGC | 3sqq | A | A | 4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4231 | |
| CDK2 | CDK | CMGC | 3sqq | A | B | 4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 3925 | |
| CDK2 | CDK | CMGC | 3sw4 | A | A | n'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamine | Human | 4076 | |
| CDK2 | CDK | CMGC | 3sw4 | A | B | n'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamine | Human | 4439 | |
| CDK2 | CDK | CMGC | 3sw7 | A | A | n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamine | Human | 4198 | |
| CDK2 | CDK | CMGC | 3sw7 | A | B | n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamine | Human | 4584 | |
| CDK2 | CDK | CMGC | 3ti1 | A | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 4201 | |
| CDK2 | CDK | CMGC | 3ti1 | A | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 4213 | |
| CDK2 | CDK | CMGC | 3tiy | A | A | 2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-one | Human | 4413 | |
| CDK2 | CDK | CMGC | 3tiy | A | B | 2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-one | Human | 4488 | |
| CDK2 | CDK | CMGC | 3tiz | A | | 1-{(e)-[(4-hydroxyphenyl)imino]methyl}naphthalen-2-ol | Human | 4136 | |
| CDK2 | CDK | CMGC | 3tnw | A | A | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 4254 | |
| CDK2 | CDK | CMGC | 3tnw | A | B | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 3948 | |
| CDK2 | CDK | CMGC | 3tnw | C | A | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 3940 | |
| CDK2 | CDK | CMGC | 3tnw | C | B | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 4493 | |
| CDK2 | CDK | CMGC | 3uli | A | A | 1-(aminomethyl)-n-(3-{[6-bromo-2-(4-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-7-yl]amino}propyl)cyclopropanecarboxamide | Human | 4115 | |
| CDK2 | CDK | CMGC | 3unj | A | | 4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acid | Human | 4498 | |
| CDK2 | CDK | CMGC | 3unk | A | | 4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 4374 | |
| CDK2 | CDK | CMGC | 3wbl | A | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 3895 | |
| CDK2 | CDK | CMGC | 4acm | A | A | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 4247 | |
| CDK2 | CDK | CMGC | 4acm | A | B | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 3983 | |
| CDK2 | CDK | CMGC | 4bck | A | A | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4095 | |
| CDK2 | CDK | CMGC | 4bck | A | B | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 3960 | |
| CDK2 | CDK | CMGC | 4bck | A | C | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4433 | |
| CDK2 | CDK | CMGC | 4bck | A | D | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4563 | |
| CDK2 | CDK | CMGC | 4bck | C | A | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4268 | |
| CDK2 | CDK | CMGC | 4bck | C | B | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4506 | |
| CDK2 | CDK | CMGC | 4bck | C | C | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4029 | |
| CDK2 | CDK | CMGC | 4bck | C | D | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4080 | |
| CDK2 | CDK | CMGC | 4bcm | A | A | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 4290 | |
| CDK2 | CDK | CMGC | 4bcm | A | B | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 4203 | |
| CDK2 | CDK | CMGC | 4bcm | C | A | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 4227 | |
| CDK2 | CDK | CMGC | 4bcm | C | B | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 4124 | |
| CDK2 | CDK | CMGC | 4bcn | A | A | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4084 | |
| CDK2 | CDK | CMGC | 4bcn | A | B | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4298 | |
| CDK2 | CDK | CMGC | 4bcn | C | A | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4436 | |
| CDK2 | CDK | CMGC | 4bcn | C | B | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4150 | |
| CDK2 | CDK | CMGC | 4bco | A | A | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 3988 | |
| CDK2 | CDK | CMGC | 4bco | A | B | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4051 | |
| CDK2 | CDK | CMGC | 4bco | C | A | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4333 | |
| CDK2 | CDK | CMGC | 4bco | C | B | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4018 | |
| CDK2 | CDK | CMGC | 4bcp | A | A | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4552 | |
| CDK2 | CDK | CMGC | 4bcp | A | B | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4304 | |
| CDK2 | CDK | CMGC | 4bcp | C | A | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 3872 | |
| CDK2 | CDK | CMGC | 4bcp | C | B | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4501 | |
| CDK2 | CDK | CMGC | 4bcq | A | A | 4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrile | Human | 4396 | |
| CDK2 | CDK | CMGC | 4bcq | A | B | 4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrile | Human | 4415 | |
| CDK2 | CDK | CMGC | 4bcq | C | A | 4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrile | Human | 3996 | |
| CDK2 | CDK | CMGC | 4bcq | C | B | 4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrile | Human | 4120 | |
| CDK2 | CDK | CMGC | 4bgh | A | A | 4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamide | Human | 4073 | |
| CDK2 | CDK | CMGC | 4bgh | A | B | 4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamide | Human | 4509 | |
| CDK2 | CDK | CMGC | 4bzd | A | A | 6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amine | Human | 3865 | |
| CDK2 | CDK | CMGC | 4bzd | A | B | 6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amine | Human | 4490 | |
| CDK2 | CDK | CMGC | 4cfm | A | A | 6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amine | Human | 4207 | |
| CDK2 | CDK | CMGC | 4cfm | A | B | 6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amine | Human | 3986 | |
| CDK2 | CDK | CMGC | 4cfm | C | A | 6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amine | Human | 4260 | |
| CDK2 | CDK | CMGC | 4cfm | C | B | 6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amine | Human | 4005 | |
| CDK2 | CDK | CMGC | 4cfn | A | A | 6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amine | Human | 4285 | |
| CDK2 | CDK | CMGC | 4cfn | A | B | 6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amine | Human | 4437 | |
| CDK2 | CDK | CMGC | 4cfn | C | A | 6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amine | Human | 4355 | |
| CDK2 | CDK | CMGC | 4cfn | C | B | 6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amine | Human | 4567 | |
| CDK2 | CDK | CMGC | 4cfu | A | A | 3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acid | Human | 3905 | |
| CDK2 | CDK | CMGC | 4cfu | A | B | 3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acid | Human | 4308 | |
| CDK2 | CDK | CMGC | 4cfu | C | A | 3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acid | Human | 3967 | |
| CDK2 | CDK | CMGC | 4cfu | C | B | 3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acid | Human | 4539 | |
| CDK2 | CDK | CMGC | 4cfv | A | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenol | Human | 4180 | |
| CDK2 | CDK | CMGC | 4cfv | A | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenol | Human | 4328 | |
| CDK2 | CDK | CMGC | 4cfv | C | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenol | Human | 3999 | |
| CDK2 | CDK | CMGC | 4cfv | C | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenol | Human | 3979 | |
| CDK2 | CDK | CMGC | 4cfw | A | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4280 | |
| CDK2 | CDK | CMGC | 4cfw | A | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4557 | |
| CDK2 | CDK | CMGC | 4cfw | A | C | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4141 | |
| CDK2 | CDK | CMGC | 4cfw | C | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4549 | |
| CDK2 | CDK | CMGC | 4cfw | C | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4508 | |
| CDK2 | CDK | CMGC | 4cfw | C | C | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4102 | |
| CDK2 | CDK | CMGC | 4cfx | A | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4485 | |
| CDK2 | CDK | CMGC | 4cfx | A | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4086 | |
| CDK2 | CDK | CMGC | 4cfx | A | C | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 3963 | |
| CDK2 | CDK | CMGC | 4cfx | C | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4166 | |
| CDK2 | CDK | CMGC | 4cfx | C | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4257 | |
| CDK2 | CDK | CMGC | 4cfx | C | C | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4442 | |
| CDK2 | CDK | CMGC | 4d1x | A | | (4s)-2-(6-hydroxy-1,3-benzothiazol-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acid | Human | 4344 | |
| CDK2 | CDK | CMGC | 4d1z | A | | (4s)-2-(8-hydroxyquinolin-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acid | Human | 4486 | |
| CDK2 | CDK | CMGC | 4ek3 | A | A | - | Human | 3971 | |
| CDK2 | CDK | CMGC | 4ek3 | A | B | - | Human | 4202 | |
| CDK2 | CDK | CMGC | 4ek4 | A | A | 4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamide | Human | 4212 | |
| CDK2 | CDK | CMGC | 4ek4 | A | B | 4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamide | Human | 3957 | |
| CDK2 | CDK | CMGC | 4ek4 | A | C | 4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamide | Human | 4369 | |
| CDK2 | CDK | CMGC | 4ek5 | A | A | n-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamide | Human | 4037 | |
| CDK2 | CDK | CMGC | 4ek5 | A | B | n-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamide | Human | 4145 | |
| CDK2 | CDK | CMGC | 4ek6 | A | A | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamide | Human | 4359 | |
| CDK2 | CDK | CMGC | 4ek6 | A | B | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamide | Human | 4056 | |
| CDK2 | CDK | CMGC | 4ek8 | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amine | Human | 4079 | |
| CDK2 | CDK | CMGC | 4ek8 | A | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amine | Human | 3871 | |
| CDK2 | CDK | CMGC | 4eoi | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4307 | |
| CDK2 | CDK | CMGC | 4eoi | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4342 | |
| CDK2 | CDK | CMGC | 4eoi | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4522 | |
| CDK2 | CDK | CMGC | 4eoi | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4011 | |
| CDK2 | CDK | CMGC | 4eoj | A | A | adenosine-5'-triphosphate | Human | 4271 | |
| CDK2 | CDK | CMGC | 4eoj | A | B | adenosine-5'-triphosphate | Human | 4015 | |
| CDK2 | CDK | CMGC | 4eoj | C | A | adenosine-5'-triphosphate | Human | 4041 | |
| CDK2 | CDK | CMGC | 4eoj | C | B | adenosine-5'-triphosphate | Human | 4311 | |
| CDK2 | CDK | CMGC | 4eok | A | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 3913 | |
| CDK2 | CDK | CMGC | 4eok | C | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4385 | |
| CDK2 | CDK | CMGC | 4eol | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4089 | |
| CDK2 | CDK | CMGC | 4eol | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4270 | |
| CDK2 | CDK | CMGC | 4eol | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4235 | |
| CDK2 | CDK | CMGC | 4eol | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4521 | |
| CDK2 | CDK | CMGC | 4eom | A | A | adenosine-5'-triphosphate | Human | 4528 | |
| CDK2 | CDK | CMGC | 4eom | A | B | adenosine-5'-triphosphate | Human | 4472 | |
| CDK2 | CDK | CMGC | 4eom | C | A | adenosine-5'-triphosphate | Human | 4481 | |
| CDK2 | CDK | CMGC | 4eom | C | B | adenosine-5'-triphosphate | Human | 4423 | |
| CDK2 | CDK | CMGC | 4eon | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 3902 | |
| CDK2 | CDK | CMGC | 4eon | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4326 | |
| CDK2 | CDK | CMGC | 4eon | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4153 | |
| CDK2 | CDK | CMGC | 4eon | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4192 | |
| CDK2 | CDK | CMGC | 4eoo | A | A | adenosine-5'-triphosphate | Human | 4403 | |
| CDK2 | CDK | CMGC | 4eoo | A | B | adenosine-5'-triphosphate | Human | 4278 | |
| CDK2 | CDK | CMGC | 4eoo | C | A | adenosine-5'-triphosphate | Human | 4188 | |
| CDK2 | CDK | CMGC | 4eoo | C | B | adenosine-5'-triphosphate | Human | 4139 | |
| CDK2 | CDK | CMGC | 4eop | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4258 | |
| CDK2 | CDK | CMGC | 4eop | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4044 | |
| CDK2 | CDK | CMGC | 4eop | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4061 | |
| CDK2 | CDK | CMGC | 4eop | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4463 | |
| CDK2 | CDK | CMGC | 4eoq | A | A | adenosine-5'-triphosphate | Human | 4402 | |
| CDK2 | CDK | CMGC | 4eoq | A | B | adenosine-5'-triphosphate | Human | 4230 | |
| CDK2 | CDK | CMGC | 4eoq | C | A | adenosine-5'-triphosphate | Human | 4004 | |
| CDK2 | CDK | CMGC | 4eoq | C | B | adenosine-5'-triphosphate | Human | 3912 | |
| CDK2 | CDK | CMGC | 4eor | A | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4205 | |
| CDK2 | CDK | CMGC | 4eor | A | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 3934 | |
| CDK2 | CDK | CMGC | 4eor | C | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4221 | |
| CDK2 | CDK | CMGC | 4eor | C | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4487 | |
| CDK2 | CDK | CMGC | 4eos | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4340 | |
| CDK2 | CDK | CMGC | 4eos | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4028 | |
| CDK2 | CDK | CMGC | 4eos | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4008 | |
| CDK2 | CDK | CMGC | 4eos | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4181 | |
| CDK2 | CDK | CMGC | 4erw | A | | staurosporine | Human | 4370 | |
| CDK2 | CDK | CMGC | 4ez3 | A | | 4-[(e)-(6-hydroxy-2-oxo-1,2-dihydropyridin-3-yl)diazenyl]benzenesulfonamide | Human | 4551 | |
| CDK2 | CDK | CMGC | 4ez7 | A | | staurosporine | Human | 4240 | |
| CDK2 | CDK | CMGC | 4fkg | A | A | 4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acid | Human | 4020 | |
| CDK2 | CDK | CMGC | 4fkg | A | B | 4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acid | Human | 4559 | |
| CDK2 | CDK | CMGC | 4fki | A | A | n-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamide | Human | 4430 | |
| CDK2 | CDK | CMGC | 4fki | A | B | n-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamide | Human | 4272 | |
| CDK2 | CDK | CMGC | 4fkj | A | A | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamide | Human | 4387 | |
| CDK2 | CDK | CMGC | 4fkj | A | B | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamide | Human | 4164 | |
| CDK2 | CDK | CMGC | 4fkl | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4583 | |
| CDK2 | CDK | CMGC | 4fkl | A | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4134 | |
| CDK2 | CDK | CMGC | 4fko | A | A | 2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamine | Human | 4449 | |
| CDK2 | CDK | CMGC | 4fko | A | B | 2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamine | Human | 4534 | |
| CDK2 | CDK | CMGC | 4fkp | A | A | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4035 | |
| CDK2 | CDK | CMGC | 4fkp | A | B | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4313 | |
| CDK2 | CDK | CMGC | 4fkp | A | C | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4468 | |
| CDK2 | CDK | CMGC | 4fkq | A | A | 4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamide | Human | 3972 | |
| CDK2 | CDK | CMGC | 4fkq | A | B | 4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamide | Human | 4026 | |
| CDK2 | CDK | CMGC | 4fkr | A | A | (8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 4149 | |
| CDK2 | CDK | CMGC | 4fkr | A | B | (8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 4535 | |
| CDK2 | CDK | CMGC | 4fks | A | A | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4412 | |
| CDK2 | CDK | CMGC | 4fks | A | B | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4489 | |
| CDK2 | CDK | CMGC | 4fks | A | C | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4315 | |
| CDK2 | CDK | CMGC | 4fkt | A | A | n-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamide | Human | 4548 | |
| CDK2 | CDK | CMGC | 4fkt | A | B | n-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamide | Human | 4322 | |
| CDK2 | CDK | CMGC | 4fku | A | A | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 3863 | |
| CDK2 | CDK | CMGC | 4fku | A | B | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 4573 | |
| CDK2 | CDK | CMGC | 4fkv | A | A | (3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamide | Human | 4299 | |
| CDK2 | CDK | CMGC | 4fkv | A | B | (3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamide | Human | 3939 | |
| CDK2 | CDK | CMGC | 4fkw | A | A | 2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylate | Human | 4252 | |
| CDK2 | CDK | CMGC | 4fkw | A | B | 2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylate | Human | 4277 | |
| CDK2 | CDK | CMGC | 4fx3 | A | A | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 4518 | |
| CDK2 | CDK | CMGC | 4fx3 | A | B | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 3931 | |
| CDK2 | CDK | CMGC | 4fx3 | C | A | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 4349 | |
| CDK2 | CDK | CMGC | 4fx3 | C | B | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 4495 | |
| CDK2 | CDK | CMGC | 4gcj | A | A | 4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4138 | |
| CDK2 | CDK | CMGC | 4gcj | A | B | 4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4362 | |
| CDK2 | CDK | CMGC | 4i3z | A | | adenosine-5'-diphosphate | Human | 4148 | |
| CDK2 | CDK | CMGC | 4i3z | C | | adenosine-5'-diphosphate | Human | 3961 | |
| CDK2 | CDK | CMGC | 4ii5 | A | A | adenosine-5'-diphosphate | Human | 3930 | |
| CDK2 | CDK | CMGC | 4ii5 | A | B | adenosine-5'-diphosphate | Human | 4456 | |
| CDK2 | CDK | CMGC | 4ii5 | C | A | adenosine-5'-diphosphate | Human | 4530 | |
| CDK2 | CDK | CMGC | 4ii5 | C | B | adenosine-5'-diphosphate | Human | 4462 | |
| CDK2 | CDK | CMGC | 4kd1 | A | A | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 4585 | |
| CDK2 | CDK | CMGC | 4kd1 | A | B | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 4525 | |
| CDK2 | CDK | CMGC | 4lyn | A | | (2s)-n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)-2-phenylpropanamide | Human | 4550 | |
| CDK2 | CDK | CMGC | 4nj3 | A | A | 6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | 4075 | |
| CDK2 | CDK | CMGC | 4nj3 | A | B | 6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | 4366 | |
| CDK2 | CDK | CMGC | 4rj3 | A | A | 1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | 4244 | |
| CDK2 | CDK | CMGC | 4rj3 | A | B | 1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | 4127 | |
| CDK2 | CDK | CMGC | 5a14 | A | A | 1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea | Human | 3977 | |
| CDK2 | CDK | CMGC | 5a14 | A | B | 1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea | Human | 3901 | |
| CDK2 | CDK | CMGC | 5and | A | | 2-imidazol-1-yl-1h-benzimidazole | Human | 6543 | |
| CDK2 | CDK | CMGC | 5ane | A | | 6-methoxy-9h-purine | Human | 6542 | |
| CDK2 | CDK | CMGC | 5ang | A | | 7-hydroxy-4-(morpholinomethyl)chromen-2-one | Human | 6540 | |
| CDK2 | CDK | CMGC | 5ani | A | | 6-chloro-9h-purine | Human | 6539 | |
| CDK2 | CDK | CMGC | 5anj | A | | n-(9h-purin-6-yl)thiophene-2-carboxamide | Human | 6541 | |
| CDK2 | CDK | CMGC | 5ank | A | | 2,4,6-trioxo-1-phenyl-hexahydropyrimidine-5-carboxamide | Human | 6538 | |
| CDK2 | CDK | CMGC | 5ano | A | | - | Human | 6537 | |
| CDK2 | CDK | CMGC | 5cyi | A | A | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | 6052 | |
| CDK2 | CDK | CMGC | 5cyi | A | B | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | 6054 | |
| CDK2 | CDK | CMGC | 5cyi | C | A | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | 6055 | |
| CDK2 | CDK | CMGC | 5cyi | C | B | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | 6053 | |
| CDK2 | CDK | CMGC | 5d1j | A | | n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamide | Human | 4058 | |
| CDK2 | CDK | CMGC | 5fp5 | A | | 4-fluorobenzoic acid | Human | 6285 | |
| CDK2 | CDK | CMGC | 5fp6 | A | A | 3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-ol | Human | 6302 | |
| CDK2 | CDK | CMGC | 5fp6 | A | B | 3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-ol | Human | 6301 | |
| CDK2 | CDK | CMGC | 5iev | A | A | roniciclib | Human | 6567 | |
| CDK2 | CDK | CMGC | 5iev | A | B | roniciclib | Human | 6570 | |
| CDK2 | CDK | CMGC | 5iex | A | A | (2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-ol | Human | 6565 | |
| CDK2 | CDK | CMGC | 5iex | A | B | (2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-ol | Human | 6572 | |
| CDK2 | CDK | CMGC | 5iey | A | A | 4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamide | Human | 6566 | |
| CDK2 | CDK | CMGC | 5iey | A | B | 4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamide | Human | 6573 | |
| CDK2 | CDK | CMGC | 5if1 | A | A | - | Human | 6568 | |
| CDK2 | CDK | CMGC | 5if1 | A | B | - | Human | 6569 | |
| CDK2 | CDK | CMGC | 5if1 | C | A | - | Human | 6564 | |
| CDK2 | CDK | CMGC | 5if1 | C | B | - | Human | 6571 | |
| CDK2 | CDK | CMGC | 5jq5 | A | | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 7416 | |
| CDK2 | CDK | CMGC | 5jq8 | A | | (3s,4s)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 7417 | |
| CDK2 | CDK | CMGC | 5k4j | A | A | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 6751 | |
| CDK2 | CDK | CMGC | 5k4j | A | B | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 6750 | |
| CDK2 | CDK | CMGC | 5l2w | A | | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 6993 | |
| CDK2 | CDK | CMGC | 5lmk | A | A | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | 7399 | |
| CDK2 | CDK | CMGC | 5lmk | A | B | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | 7398 | |
| CDK2 | CDK | CMGC | 5lmk | C | A | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | 7396 | |
| CDK2 | CDK | CMGC | 5lmk | C | B | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | 7397 | |
| CDK2 | CDK | CMGC | 5mhq | A | A | (2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-ol | Human | 9409 | |
| CDK2 | CDK | CMGC | 5mhq | A | B | (2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-ol | Human | 9408 | |
| CDK2 | CDK | CMGC | 5nev | A | | 4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamide | Human | 8020 | |
| CDK2 | CDK | CMGC | 5nev | C | | 4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamide | Human | 8019 | |
| CDK2 | CDK | CMGC | 5oo0 | A | A | - | Human | 9744 | |
| CDK2 | CDK | CMGC | 5oo0 | A | C | - | Human | 9745 | |
| CDK2 | CDK | CMGC | 5oo1 | A | | ~{n}-(4-pyrimidin-2-ylphenyl)propanamide | Human | 10566 | |
| CDK2 | CDK | CMGC | 5oo3 | A | A | 1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-one | Human | 10569 | |
| CDK2 | CDK | CMGC | 5oo3 | A | B | 1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-one | Human | 10568 | |
| CDK2 | CDK | CMGC | 5osj | A | A | - | Human | 9743 | |
| CDK2 | CDK | CMGC | 5osj | A | B | - | Human | 9742 | |
| CDK2 | CDK | CMGC | 5osm | A | A | methyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylate | Human | 9741 | |
| CDK2 | CDK | CMGC | 5osm | A | B | methyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylate | Human | 9740 | |
| CDK2 | CDK | CMGC | 5uq1 | A | | - | Human | 8220 | |
| CDK2 | CDK | CMGC | 5uq1 | C | | - | Human | 8223 | |
| CDK2 | CDK | CMGC | 5uq2 | A | | - | Human | 8221 | |
| CDK2 | CDK | CMGC | 5uq3 | A | | - | Human | 8222 | |
| CDK2 | CDK | CMGC | 6ath | A | A | - | Human | 10567 | |
| CDK2 | CDK | CMGC | 6ath | A | B | - | Human | 10570 | |
| CDK2 | CDK | CMGC | 6gub | A | | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | 10764 | |
| CDK2 | CDK | CMGC | 6gub | C | | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | 10763 | |
| CDK2 | CDK | CMGC | 6guc | A | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 10767 | |
| CDK2 | CDK | CMGC | 6guc | C | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 10766 | |
| CDK2 | CDK | CMGC | 6gue | A | | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10771 | |
| CDK2 | CDK | CMGC | 6gue | C | | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10772 | |
| CDK2 | CDK | CMGC | 6guf | A | | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 10770 | |
| CDK2 | CDK | CMGC | 6guf | C | | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 10762 | |
| CDK2 | CDK | CMGC | 6guh | A | A | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10765 | |
| CDK2 | CDK | CMGC | 6guh | A | B | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10769 | |
| CDK2 | CDK | CMGC | 6guk | A | A | ~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamine | Human | 10773 | |
| CDK2 | CDK | CMGC | 6guk | A | B | ~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamine | Human | 10768 | |
| CDK2 | CDK | CMGC | 6gva | A | A | 5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | 11206 | |
| CDK2 | CDK | CMGC | 6gva | A | B | 5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | 11204 | |
| CDK2 | CDK | CMGC | 6inl | A | | 2,2'-{[6-{[(4-methoxyphenyl)methyl]amino}-9-(propan-2-yl)-9h-purin-2-yl]azanediyl}di(ethan-1-ol) | Human | 11794 | |
| CDK2 | CDK | CMGC | 6jgm | A | | 4-{[6-(cyclohexylmethoxy)-7h-purin-2-yl]amino}-n,n-diethylbenzamide | Human | 12008 | |
| CDK2 | CDK | CMGC | 6oqi | A | | 5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4s)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amine | Human | 12648 | |
| CDK2 | CDK | CMGC | 6p3w | A | A | - | Human | 11515 | |
| CDK2 | CDK | CMGC | 6p3w | A | B | - | Human | 11517 | |
| CDK2 | CDK | CMGC | 6p3w | C | A | - | Human | 11514 | |
| CDK2 | CDK | CMGC | 6p3w | C | B | - | Human | 11516 | |
| CDK2 | CDK | CMGC | 6q3b | A | A | 4-iodopyrazole | Human | 11177 | |
| CDK2 | CDK | CMGC | 6q3b | A | B | 4-iodopyrazole | Human | 11208 | |
| CDK2 | CDK | CMGC | 6q3c | A | A | 4-bromo-1h-pyrazole | Human | 11191 | |
| CDK2 | CDK | CMGC | 6q3c | A | B | 4-bromo-1h-pyrazole | Human | 11203 | |
| CDK2 | CDK | CMGC | 6q3c | A | C | - | Human | 11178 | |
| CDK2 | CDK | CMGC | 6q3f | A | A | - | Human | 11181 | |
| CDK2 | CDK | CMGC | 6q3f | A | B | - | Human | 11187 | |
| CDK2 | CDK | CMGC | 6q48 | A | A | 4-iodanyl-3~{h}-pyridin-2-one | Human | 11192 | |
| CDK2 | CDK | CMGC | 6q48 | A | B | 4-iodanyl-3~{h}-pyridin-2-one | Human | 11218 | |
| CDK2 | CDK | CMGC | 6q48 | A | C | 4-iodanyl-3~{h}-pyridin-2-one | Human | 11196 | |
| CDK2 | CDK | CMGC | 6q49 | A | A | - | Human | 11185 | |
| CDK2 | CDK | CMGC | 6q49 | A | B | - | Human | 11220 | |
| CDK2 | CDK | CMGC | 6q49 | A | C | - | Human | 11193 | |
| CDK2 | CDK | CMGC | 6q4a | A | A | 5-iodanylpyrimidine | Human | 11195 | |
| CDK2 | CDK | CMGC | 6q4a | A | B | 5-iodanylpyrimidine | Human | 11200 | |
| CDK2 | CDK | CMGC | 6q4a | A | C | 5-iodanylpyrimidine | Human | 11216 | |
| CDK2 | CDK | CMGC | 6q4b | A | A | 5-bromanylpyrimidine | Human | 11198 | |
| CDK2 | CDK | CMGC | 6q4b | A | B | 5-bromanylpyrimidine | Human | 11210 | |
| CDK2 | CDK | CMGC | 6q4b | A | C | 5-bromanylpyrimidine | Human | 11180 | |
| CDK2 | CDK | CMGC | 6q4c | A | A | 4-bromanyl-1,8-naphthyridine | Human | 11182 | |
| CDK2 | CDK | CMGC | 6q4c | A | B | 4-bromanyl-1,8-naphthyridine | Human | 11207 | |
| CDK2 | CDK | CMGC | 6q4c | A | C | 4-bromanyl-1,8-naphthyridine | Human | 11201 | |
| CDK2 | CDK | CMGC | 6q4d | A | A | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid | Human | 11184 | |
| CDK2 | CDK | CMGC | 6q4d | A | B | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid | Human | 11215 | |
| CDK2 | CDK | CMGC | 6q4d | A | C | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid | Human | 11188 | |
| CDK2 | CDK | CMGC | 6q4e | A | A | 6-iodanyl-7~{h}-purin-2-amine | Human | 11199 | |
| CDK2 | CDK | CMGC | 6q4e | A | B | 6-iodanyl-7~{h}-purin-2-amine | Human | 11205 | |
| CDK2 | CDK | CMGC | 6q4e | A | C | 6-iodanyl-7~{h}-purin-2-amine | Human | 11219 | |
| CDK2 | CDK | CMGC | 6q4f | A | A | pyridine-2,6-diamine | Human | 11202 | |
| CDK2 | CDK | CMGC | 6q4f | A | B | pyridine-2,6-diamine | Human | 11211 | |
| CDK2 | CDK | CMGC | 6q4f | A | C | pyridine-2,6-diamine | Human | 11212 | |
| CDK2 | CDK | CMGC | 6q4g | A | A | 2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acid | Human | 11214 | |
| CDK2 | CDK | CMGC | 6q4g | A | B | 2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acid | Human | 11217 | |
| CDK2 | CDK | CMGC | 6q4h | A | A | 2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acid | Human | 11194 | |
| CDK2 | CDK | CMGC | 6q4h | A | B | 2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acid | Human | 11190 | |
| CDK2 | CDK | CMGC | 6q4i | A | A | 2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acid | Human | 11183 | |
| CDK2 | CDK | CMGC | 6q4i | A | B | 2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acid | Human | 11197 | |
| CDK2 | CDK | CMGC | 6q4j | A | A | 2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acid | Human | 11209 | |
| CDK2 | CDK | CMGC | 6q4j | A | B | 2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acid | Human | 11213 | |
| CDK2 | CDK | CMGC | 6q4k | A | A | - | Human | 11179 | |
| CDK2 | CDK | CMGC | 6q4k | A | B | - | Human | 11186 | |
| CDK2 | CDK | CMGC | 6q4k | A | C | - | Human | 11189 | |
| CDK2 | CDK | CMGC | 6rij | A | A | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | 12623 | |
| CDK2 | CDK | CMGC | 6rij | A | B | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | 12624 | |
| CDK2 | CDK | CMGC | 6rij | C | A | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | 12625 | |
| CDK2 | CDK | CMGC | 6rij | C | B | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | 12622 | |
| CDK2 | CDK | CMGC | 6sg4 | A | A | - | Human | 13246 | |
| CDK2 | CDK | CMGC | 6sg4 | A | B | - | Human | 13247 | |
| CDK2 | CDK | CMGC | 6sg4 | C | A | - | Human | 13248 | |
| CDK2 | CDK | CMGC | 6sg4 | C | B | - | Human | 13245 | |
| CDK2 | CDK | CMGC | 6yl1 | A | A | methyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | 12497 | |
| CDK2 | CDK | CMGC | 6yl1 | A | B | methyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | 12496 | |
| CDK2 | CDK | CMGC | 6yl6 | A | A | - | Human | 12498 | |
| CDK2 | CDK | CMGC | 6yl6 | A | B | - | Human | 12495 | |
| CDK2 | CDK | CMGC | 6ylk | A | A | methyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | 12499 | |
| CDK2 | CDK | CMGC | 6ylk | A | B | methyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | 12494 | |
| CDK2 | CDK | CMGC | 7ack | A | A | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | 13451 | |
| CDK2 | CDK | CMGC | 7ack | A | B | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | 13453 | |
| CDK2 | CDK | CMGC | 7ack | C | A | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | 13450 | |
| CDK2 | CDK | CMGC | 7ack | C | B | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | 13452 | |
| CDK2 | CDK | CMGC | 7b5l | L | | - | Human | 13266 | |
| CDK2 | CDK | CMGC | 7b5r | L | | - | Human | 13265 | |
| CDK2 | CDK | CMGC | 7b7s | A | A | 7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxide | Human | 13833 | |
| CDK2 | CDK | CMGC | 7b7s | A | B | 7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxide | Human | 13834 | |
| CDK2 | CDK | CMGC | 7e34 | A | | - | Human | 13497 | |
| CDK2 | CDK | CMGC | 7kjs | A | | 6-(difluoromethyl)-8-[(1r,2r)-2-hydroxy-2-methylcyclopentyl]-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 13740 | |
| CDK2 | CDK | CMGC | 7m2f | A | A | [(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acid | Human | 13797 | |
| CDK2 | CDK | CMGC | 7m2f | A | B | [(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acid | Human | 13796 | |
| CDK2 | CDK | CMGC | 7mkx | A | | 2-[(5-bromo-2-{4-[(cyanomethyl)sulfamoyl]anilino}pyrimidin-4-yl)amino]-6-fluorobenzamide | Human | 14490 | |
| CDK2 | CDK | CMGC | 7nvq | A | | staurosporine | Human | 13627 | |
| CDK2 | CDK | CMGC | 7qhl | A | A | 5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidine | Human | 14275 | |
| CDK2 | CDK | CMGC | 7qhl | A | B | 5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidine | Human | 14276 | |
| CDK2 | CDK | CMGC | 7ra5 | A | A | 4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amine | Human | 13960 | |
| CDK2 | CDK | CMGC | 7ra5 | A | B | 4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amine | Human | 13959 | |
| CDK2 | CDK | CMGC | 7rwe | A | | 5-nitro-2-[(3-phenylpropyl)amino]benzoic acid | Human | 14345 | |
| CDK2 | CDK | CMGC | 7rwf | A | | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acid | Human | 14344 | |
| CDK2 | CDK | CMGC | 7rxo | A | A | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acid | Human | 14352 | |
| CDK2 | CDK | CMGC | 7rxo | A | B | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acid | Human | 14351 | |
| CDK2 | CDK | CMGC | 7s4t | A | A | 2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acid | Human | 14374 | |
| CDK2 | CDK | CMGC | 7s4t | A | B | 2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acid | Human | 14373 | |
| CDK2 | CDK | CMGC | 7s7a | A | A | 2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14427 | |
| CDK2 | CDK | CMGC | 7s7a | A | B | 2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14426 | |
| CDK2 | CDK | CMGC | 7s84 | A | A | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14424 | |
| CDK2 | CDK | CMGC | 7s84 | A | B | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14432 | |
| CDK2 | CDK | CMGC | 7s85 | A | | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethoxy)benzoic acid | Human | 14425 | |
| CDK2 | CDK | CMGC | 7s9x | A | A | 2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acid | Human | 14430 | |
| CDK2 | CDK | CMGC | 7s9x | A | B | 2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acid | Human | 14431 | |
| CDK2 | CDK | CMGC | 7sa0 | A | A | 2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14428 | |
| CDK2 | CDK | CMGC | 7sa0 | A | B | 2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14429 | |
| CDK2 | CDK | CMGC | 7ug1 | A | A | 8-(4-chloroanilino)naphthalene-1-sulfonic acid | Human | 14700 | |
| CDK2 | CDK | CMGC | 7ug1 | A | B | 8-(4-chloroanilino)naphthalene-1-sulfonic acid | Human | 14701 | |
| CDK2 | CDK | CMGC | 7uxi | A | A | - | Human | 14571 | |
| CDK2 | CDK | CMGC | 7uxi | A | B | - | Human | 14572 | |
| CDK2 | CDK | CMGC | 7uxk | A | | - | Human | 14570 | |
| CDK2 | CDK | CMGC | 7vdu | A | A | [1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanol | Human | 14136 | |
| CDK2 | CDK | CMGC | 7vdu | A | B | [1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanol | Human | 14137 | |
| CDK2 | CDK | CMGC | 7zpc | A | A | ~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamide | Human | 14606 | |
| CDK2 | CDK | CMGC | 7zpc | A | B | ~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamide | Human | 14607 | |
| CDK2 | CDK | CMGC | 8b54 | A | A | ~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | 14681 | |
| CDK2 | CDK | CMGC | 8b54 | A | B | ~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | 14680 | |
| CDK2 | CDK | CMGC | 8bya | A | | - | Human | 14814 | |
| CDK2 | CDK | CMGC | 8bzo | A | | - | Human | 14815 | |
| CDK2 | CDK | CMGC | 8cur | A | A | 6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | 14693 | |
| CDK2 | CDK | CMGC | 8cur | A | B | 6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | 14692 | |
| CDK2 | CDK | CMGC | 8erd | A | A | (2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanone | Human | 14949 | |
| CDK2 | CDK | CMGC | 8erd | A | B | (2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanone | Human | 14951 | |
| CDK2 | CDK | CMGC | 8ern | A | A | n,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamide | Human | 14948 | |
| CDK2 | CDK | CMGC | 8ern | A | B | n,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamide | Human | 14950 | |
| CDK2 | CDK | CMGC | 8fow | A | A | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 14759 | |
| CDK2 | CDK | CMGC | 8fow | A | B | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 14760 | |
| CDK2 | CDK | CMGC | 8fp0 | A | A | r-roscovitine | Human | 14758 | |
| CDK2 | CDK | CMGC | 8fp0 | A | B | r-roscovitine | Human | 14756 | |
| CDK2 | CDK | CMGC | 8fp5 | A | A | adenosine-5'-triphosphate | Human | 14761 | |
| CDK2 | CDK | CMGC | 8fp5 | A | B | adenosine-5'-triphosphate | Human | 14757 | |
| CDK2 | CDK | CMGC | 8h6p | A | | (7s,10r)-11-oxa-2,4,5,13,17,23-hexaazatetracyclo[17.3.1.1~3,6~.1~7,10~]pentacosa-1(23),3(25),5,19,21-pentaene-12,18-dione | Human | 14625 | |
| CDK2 | CDK | CMGC | 8h6t | A | | (1r,3s)-3-{3-[(pyridin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl propan-2-ylcarbamate | Human | 14626 | |
| CDK2 | CDK | CMGC | 8oy2 | A | | (1s,2s,11as)-1-methoxy-1,4,7,10-tetramethyl-2,9-bis(oxidanyl)-2,11a-dihydrobenzo[b][1,4]benzodioxepine-3,6-dione | Human | 15078 | |
| CDK2 | CDK | CMGC | 8ru8 | A | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 15329 | |
| CDK2 | CDK | CMGC | 8ru8 | A | B | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 15328 | |
| CDK2 | CDK | CMGC | 8uv0 | A | A | 1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-ol | Human | 15238 | |
| CDK2 | CDK | CMGC | 8uv0 | A | B | 1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-ol | Human | 15239 | |
| CDK4 | CDK | CMGC | 2w96 | B | A | - | Human | 3390 | |
| CDK4 | CDK | CMGC | 2w96 | B | B | - | Human | 3389 | |
| CDK4 | CDK | CMGC | 2w99 | B | | - | Human | 3385 | |
| CDK4 | CDK | CMGC | 2w9f | B | | - | Human | 3386 | |
| CDK4 | CDK | CMGC | 2w9z | B | A | - | Human | 3388 | |
| CDK4 | CDK | CMGC | 2w9z | B | B | - | Human | 3383 | |
| CDK4 | CDK | CMGC | 3g33 | A | | - | Human | 3387 | |
| CDK4 | CDK | CMGC | 3g33 | C | | - | Human | 3384 | |
| CDK4 | CDK | CMGC | 5fwk | K | | - | Human | 6747 | |
| CDK4 | CDK | CMGC | 5fwl | K | | - | Human | 6748 | |
| CDK4 | CDK | CMGC | 5fwm | K | | - | Human | 6749 | |
| CDK4 | CDK | CMGC | 5fwp | K | | - | Human | 7132 | |
| CDK4 | CDK | CMGC | 6p8e | B | | - | Human | 11891 | |
| CDK4 | CDK | CMGC | 6p8f | B | | - | Human | 11892 | |
| CDK4 | CDK | CMGC | 6p8g | B | | - | Human | 11893 | |
| CDK4 | CDK | CMGC | 6p8h | B | | - | Human | 11894 | |
| CDK4 | CDK | CMGC | 7sj3 | A | | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 14485 | |
| CDK5 | CDK | CMGC | 1h4l | A | | - | Human | 2788 | |
| CDK5 | CDK | CMGC | 1h4l | B | | - | Human | 2779 | |
| CDK5 | CDK | CMGC | 1ung | A | | 6-phenyl[5h]pyrrolo[2,3-b]pyrazine | Human | 2792 | |
| CDK5 | CDK | CMGC | 1ung | B | | 6-phenyl[5h]pyrrolo[2,3-b]pyrazine | Human | 2789 | |
| CDK5 | CDK | CMGC | 1unh | A | | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | 2780 | |
| CDK5 | CDK | CMGC | 1unh | B | | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | 2787 | |
| CDK5 | CDK | CMGC | 1unl | A | | r-roscovitine | Human | 2785 | |
| CDK5 | CDK | CMGC | 1unl | B | | - | Human | 2790 | |
| CDK5 | CDK | CMGC | 3o0g | A | | - | Human | 2782 | |
| CDK5 | CDK | CMGC | 3o0g | B | | {4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanone | Human | 2783 | |
| CDK5 | CDK | CMGC | 4au8 | A | A | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | 2784 | |
| CDK5 | CDK | CMGC | 4au8 | A | B | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | 2786 | |
| CDK5 | CDK | CMGC | 4au8 | B | A | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | 2791 | |
| CDK5 | CDK | CMGC | 4au8 | B | B | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | 2781 | |
| CDK5 | CDK | CMGC | 7vdp | A | | [1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanol | Human | 14145 | |
| CDK5 | CDK | CMGC | 7vdq | A | | 2-[[7-[[2-fluoranyl-4-[3-(hydroxymethyl)pyrazol-1-yl]phenyl]amino]-1,6-naphthyridin-2-yl]-(1-methylpiperidin-4-yl)amino]ethanoic acid | Human | 14144 | |
| CDK5 | CDK | CMGC | 7vdr | A | | (1r)-1-[7-[(2-fluoranyl-4-pyrazol-1-yl-phenyl)amino]-1,6-naphthyridin-2-yl]-1-(1-methylpiperidin-4-yl)ethanol | Human | 14146 | |
| CDK5 | CDK | CMGC | 7vds | A | A | 5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrile | Human | 14148 | |
| CDK5 | CDK | CMGC | 7vds | A | B | 5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrile | Human | 14147 | |
| CDK6 | CDK | CMGC | 1bi7 | A | | - | Human | 2798 | |
| CDK6 | CDK | CMGC | 1bi8 | A | | - | Human | 2796 | |
| CDK6 | CDK | CMGC | 1bi8 | C | | - | Human | 2799 | |
| CDK6 | CDK | CMGC | 1blx | A | | - | Human | 2802 | |
| CDK6 | CDK | CMGC | 1g3n | A | | - | Human | 2806 | |
| CDK6 | CDK | CMGC | 1g3n | E | | - | Human | 2805 | |
| CDK6 | CDK | CMGC | 1jow | B | | - | Human | 2793 | |
| CDK6 | CDK | CMGC | 1xo2 | B | | 3,7,3',4'-tetrahydroxyflavone | Human | 2794 | |
| CDK6 | CDK | CMGC | 2euf | B | | 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 2804 | |
| CDK6 | CDK | CMGC | 2f2c | B | | (2s)-2-({6-[(3-amino-5-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 2795 | |
| CDK6 | CDK | CMGC | 3nup | A | | 4-[3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(1-methylpiperidin-4-yl)pyrimidin-2-amine | Human | 2797 | |
| CDK6 | CDK | CMGC | 3nux | A | | 4-[5-chloro-3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amine | Human | 2807 | |
| CDK6 | CDK | CMGC | 4aua | A | | 1h-benzimidazol-2-yl(1h-pyrrol-2-yl)methanone | Human | 2801 | |
| CDK6 | CDK | CMGC | 4ez5 | A | | {5-[4-(dimethylamino)piperidin-1-yl]-1h-imidazo[4,5-b]pyridin-2-yl}[2-(isoquinolin-4-yl)pyridin-4-yl]methanone | Human | 2800 | |
| CDK6 | CDK | CMGC | 4tth | B | | 9-cyclopentyl-n-(5-piperazin-1-ylpyridin-2-yl)pyrido[4,5]pyrrolo[1,2-d]pyrimidin-2-amine | Human | 2803 | |
| CDK6 | CDK | CMGC | 5l2i | A | | 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6991 | |
| CDK6 | CDK | CMGC | 5l2s | A | | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 6990 | |
| CDK6 | CDK | CMGC | 5l2t | A | | 7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 6992 | |
| CDK6 | CDK | CMGC | 6oql | A | | 5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amine | Human | 12647 | |
| CDK6 | CDK | CMGC | 6oqo | A | | n-[5-(6-ethyl-2,6-diazaspiro[3.3]heptan-2-yl)pyridin-2-yl]-5-fluoro-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amine | Human | 12646 | |
| CDK6 | CDK | CMGC | 8i0m | A | | 2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 15164 | |
| CDK7 | CDK | CMGC | 1ua2 | A | | adenosine-5'-triphosphate | Human | 540 | |
| CDK7 | CDK | CMGC | 1ua2 | B | | adenosine-5'-triphosphate | Human | 541 | |
| CDK7 | CDK | CMGC | 1ua2 | C | | adenosine-5'-triphosphate | Human | 542 | |
| CDK7 | CDK | CMGC | 1ua2 | D | | adenosine-5'-triphosphate | Human | 543 | |
| CDK7 | CDK | CMGC | 6o9l | 8 | | - | Human | 11055 | |
| CDK7 | CDK | CMGC | 6xbz | J | | phosphothiophosphoric acid-adenylate ester | Human | 12773 | |
| CDK7 | CDK | CMGC | 6xd3 | J | | n-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamide | Human | 12772 | |
| CDK7 | CDK | CMGC | 7b5o | J | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13278 | |
| CDK7 | CDK | CMGC | 7b5o | J | B | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13279 | |
| CDK7 | CDK | CMGC | 7b5q | J | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13277 | |
| CDK7 | CDK | CMGC | 7b5q | J | B | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13280 | |
| CDK7 | CDK | CMGC | 7nvr | 8 | | - | Human | 13543 | |
| CDK7 | CDK | CMGC | 8bvw | I | | - | Human | 14733 | |
| CDK7 | CDK | CMGC | 8byq | I | | - | Human | 14732 | |
| CDK7 | CDK | CMGC | 8p4z | A | A | 2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine | Human | 14796 | |
| CDK7 | CDK | CMGC | 8p4z | A | B | 2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine | Human | 14797 | |
| CDK7 | CDK | CMGC | 8pyr | A | A | - | Human | 15254 | |
| CDK7 | CDK | CMGC | 8pyr | A | B | - | Human | 15253 | |
| CDK8 | CDK | CMGC | 3rgf | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 3841 | |
| CDK8 | CDK | CMGC | 3rgf | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 3846 | |
| CDK8 | CDK | CMGC | 4crl | A | | cortistatin a | Human | 6096 | |
| CDK8 | CDK | CMGC | 4f6s | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 3848 | |
| CDK8 | CDK | CMGC | 4f6u | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]urea | Human | 3849 | |
| CDK8 | CDK | CMGC | 4f6u | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]urea | Human | 3844 | |
| CDK8 | CDK | CMGC | 4f6w | A | | n-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-4-[2-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)ethyl]piperazine-1-carboxamide | Human | 3845 | |
| CDK8 | CDK | CMGC | 4f70 | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[2-(morpholin-4-yl)ethyl]urea | Human | 3852 | |
| CDK8 | CDK | CMGC | 4f7j | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)urea | Human | 3842 | |
| CDK8 | CDK | CMGC | 4f7j | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)urea | Human | 3843 | |
| CDK8 | CDK | CMGC | 4f7l | A | | tert-butyl [3-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)propyl]carbamate | Human | 3840 | |
| CDK8 | CDK | CMGC | 4f7n | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(5-hydroxypentyl)urea | Human | 3847 | |
| CDK8 | CDK | CMGC | 4f7s | A | A | n-(2-phenylethyl)quinazolin-4-amine | Human | 3850 | |
| CDK8 | CDK | CMGC | 4f7s | A | B | n-(2-phenylethyl)quinazolin-4-amine | Human | 3853 | |
| CDK8 | CDK | CMGC | 4g6l | A | | - | Human | 3851 | |
| CDK8 | CDK | CMGC | 5bnj | A | | 8-{3-chloro-5-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]pyridin-4-yl}-2,8-diazaspiro[4.5]decan-1-one | Human | 6152 | |
| CDK8 | CDK | CMGC | 5cei | A | A | 4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamide | Human | 6404 | |
| CDK8 | CDK | CMGC | 5cei | A | B | 4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamide | Human | 6403 | |
| CDK8 | CDK | CMGC | 5fgk | A | A | 8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-one | Human | 6391 | |
| CDK8 | CDK | CMGC | 5fgk | A | B | 8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-one | Human | 6388 | |
| CDK8 | CDK | CMGC | 5hbe | A | A | 8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one | Human | 6389 | |
| CDK8 | CDK | CMGC | 5hbe | A | B | 8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one | Human | 6386 | |
| CDK8 | CDK | CMGC | 5hbh | A | | 5-[5-chloranyl-4-[1-(2-methoxyethyl)-1,8-diazaspiro[4.5]decan-8-yl]pyridin-3-yl]-1-methyl-3~{h}-2,1-benzothiazole 2,2-dioxide | Human | 6387 | |
| CDK8 | CDK | CMGC | 5hbj | A | A | 8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-one | Human | 6390 | |
| CDK8 | CDK | CMGC | 5hbj | A | B | 8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-one | Human | 6385 | |
| CDK8 | CDK | CMGC | 5hnb | A | A | [6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanone | Human | 6562 | |
| CDK8 | CDK | CMGC | 5hnb | A | B | [6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanone | Human | 6563 | |
| CDK8 | CDK | CMGC | 5hvy | A | A | n-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}urea | Human | 6553 | |
| CDK8 | CDK | CMGC | 5hvy | A | B | n-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}urea | Human | 6552 | |
| CDK8 | CDK | CMGC | 5i5z | A | | n-methyl-8-(1-methyl-2,2-dioxo-2,3-dihydro-1h-2lambda~6~,1-benzothiazol-5-yl)-1,6-naphthyridine-2-carboxamide | Human | 6536 | |
| CDK8 | CDK | CMGC | 5icp | A | A | [(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanone | Human | 7318 | |
| CDK8 | CDK | CMGC | 5icp | A | B | [(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanone | Human | 7321 | |
| CDK8 | CDK | CMGC | 5idn | A | A | [(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanone | Human | 7322 | |
| CDK8 | CDK | CMGC | 5idn | A | B | [(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanone | Human | 7319 | |
| CDK8 | CDK | CMGC | 5idp | A | A | (3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanone | Human | 7317 | |
| CDK8 | CDK | CMGC | 5idp | A | B | (3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanone | Human | 7320 | |
| CDK8 | CDK | CMGC | 5xqx | A | | n-methyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamide | Human | 8313 | |
| CDK8 | CDK | CMGC | 5xs2 | A | A | 3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamide | Human | 8315 | |
| CDK8 | CDK | CMGC | 5xs2 | A | B | 3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamide | Human | 8314 | |
| CDK8 | CDK | CMGC | 6qtg | A | | 2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]-~{n},~{n}-dimethyl-ethanamide | Human | 12094 | |
| CDK8 | CDK | CMGC | 6qtj | A | | ~{n},~{n}-dimethyl-2-[4-[4-(2,6-naphthyridin-4-yl)phenyl]pyrazol-1-yl]ethanamide | Human | 12093 | |
| CDK8 | CDK | CMGC | 6r3s | A | A | 6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamide | Human | 12140 | |
| CDK8 | CDK | CMGC | 6r3s | A | B | 6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamide | Human | 12141 | |
| CDK8 | CDK | CMGC | 6t41 | A | | ~{n}-[(4-chlorophenyl)methyl]quinazolin-4-amine | Human | 11908 | |
| CDK8 | CDK | CMGC | 6tpa | A | | 1-[4-chloranyl-3-(trifluoromethyl)phenyl]-3-(5-oxidanylidene-6-pyridin-4-yl-pyrido[2,3-b][1,5]benzoxazepin-9-yl)urea | Human | 13160 | |
| CDK8 | CDK | CMGC | 6y0a | A | A | 6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamide | Human | 13306 | |
| CDK8 | CDK | CMGC | 6y0a | A | B | 6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamide | Human | 13305 | |
| CDK9 | CDK | CMGC | 3blh | A | | - | Human | 2251 | |
| CDK9 | CDK | CMGC | 3blq | A | | adenosine-5'-triphosphate | Human | 2248 | |
| CDK9 | CDK | CMGC | 3blr | A | | 2-(2-chloro-phenyl)-5,7-dihydroxy-8-(3-hydroxy-1-methyl-piperidin-4-yl)-4h-benzopyran-4-one | Human | 2236 | |
| CDK9 | CDK | CMGC | 3lq5 | A | | (2s)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 2253 | |
| CDK9 | CDK | CMGC | 3mi9 | A | | - | Human | 2239 | |
| CDK9 | CDK | CMGC | 3mia | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2242 | |
| CDK9 | CDK | CMGC | 3my1 | A | | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 2249 | |
| CDK9 | CDK | CMGC | 3tn8 | A | | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 2240 | |
| CDK9 | CDK | CMGC | 3tnh | A | | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 2232 | |
| CDK9 | CDK | CMGC | 3tni | A | | - | Human | 2250 | |
| CDK9 | CDK | CMGC | 4bcf | A | | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 2257 | |
| CDK9 | CDK | CMGC | 4bcg | A | | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 2255 | |
| CDK9 | CDK | CMGC | 4bch | A | | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 2246 | |
| CDK9 | CDK | CMGC | 4bci | A | | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 2243 | |
| CDK9 | CDK | CMGC | 4bcj | A | | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 2247 | |
| CDK9 | CDK | CMGC | 4ec8 | A | | - | Human | 2244 | |
| CDK9 | CDK | CMGC | 4ec9 | A | | - | Human | 2234 | |
| CDK9 | CDK | CMGC | 4imy | A | A | adenosine monophosphate | Human | 2238 | |
| CDK9 | CDK | CMGC | 4imy | A | B | adenosine monophosphate | Human | 2252 | |
| CDK9 | CDK | CMGC | 4imy | C | A | adenosine monophosphate | Human | 2237 | |
| CDK9 | CDK | CMGC | 4imy | C | B | adenosine monophosphate | Human | 2245 | |
| CDK9 | CDK | CMGC | 4imy | E | A | adenosine monophosphate | Human | 2258 | |
| CDK9 | CDK | CMGC | 4imy | E | B | adenosine monophosphate | Human | 2256 | |
| CDK9 | CDK | CMGC | 4ogr | A | | adenosine | Human | 2254 | |
| CDK9 | CDK | CMGC | 4ogr | E | | adenosine | Human | 2235 | |
| CDK9 | CDK | CMGC | 4ogr | I | | adenosine | Human | 2241 | |
| CDK9 | CDK | CMGC | 4or5 | A | | - | Human | 2233 | |
| CDK9 | CDK | CMGC | 4or5 | F | | - | Human | 2231 | |
| CDK9 | CDK | CMGC | 5l1z | A | | - | Human | 7121 | |
| CDK9 | CDK | CMGC | 6cyt | A | | - | Human | 10797 | |
| CDK9 | CDK | CMGC | 6gzh | A | | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10427 | |
| CDK9 | CDK | CMGC | 6w9e | A | A | (4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone | Human | 13859 | |
| CDK9 | CDK | CMGC | 6w9e | A | B | (4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone | Human | 13858 | |
| CDK9 | CDK | CMGC | 6w9e | A | C | (4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone | Human | 13861 | |
| CDK9 | CDK | CMGC | 6w9e | A | D | (4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone | Human | 13860 | |
| CDK9 | CDK | CMGC | 6z45 | A | | (1~{s},3~{r})-3-acetamido-~{n}-[5-chloranyl-4-(5,5-dimethyl-4,6-dihydropyrrolo[1,2-b]pyrazol-3-yl)pyridin-2-yl]cyclohexane-1-carboxamide | Human | 13115 | |
| CDK9 | CDK | CMGC | 7nwk | A | | n-((1r,3r)-3-(7-(4-fluoro-2-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-2-yl)cyclopentyl)acetamide | Human | 13951 | |
| CDK9 | CDK | CMGC | 8i0l | A | | 2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 15170 | |
| CDK9 | CDK | CMGC | 8k5r | A | | (1s,3s)-n3-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamine | Human | 15081 | |
| CDKL1 | CDKL | CMGC | 4agu | A | | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 761 | |
| CDKL1 | CDKL | CMGC | 4agu | B | | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 760 | |
| CDKL1 | CDKL | CMGC | 4agu | C | | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 762 | |
| CDKL2 | CDKL | CMGC | 4aaa | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 964 | |
| CDKL2 | CDKL | CMGC | 4aaa | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 962 | |
| CDKL2 | CDKL | CMGC | 4bbm | A | | 4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diol | Human | 963 | |
| CDKL2 | CDKL | CMGC | 4bbm | B | | 4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diol | Human | 965 | |
| CDKL3 | CDKL | CMGC | 3zdu | A | | [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4677 | |
| CDKL5 | CDKL | CMGC | 4bgq | A | A | [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 1425 | |
| CDKL5 | CDKL | CMGC | 4bgq | A | B | [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 1426 | |
| CDKL5 | CDKL | CMGC | 8cie | A | | 4-[[3,5-bis(fluoranyl)phenyl]carbonylamino]-~{n}-piperidin-4-yl-1~{h}-pyrazole-3-carboxamide | Human | 14778 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1ia8 | A | | - | Human | 1656 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvq | A | | 7-hydroxystaurosporine | Human | 1642 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvr | A | | staurosporine | Human | 1585 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvs | A | | rel-(9r,12s)-9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2h)-dione | Human | 1591 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1zlt | A | | (4z)-4-(2-amino-5-oxo-3,5-dihydro-4h-imidazol-4-ylidene)-2,3-dichloro-4,5,6,7-tetrahydropyrrolo[2,3-c]azepin-8(1h)-one | Human | 1596 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1zys | A | | n-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamide | Human | 1655 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ayp | A | | (3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-one | Human | 1682 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | A | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | 1677 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | B | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | 1571 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brb | A | | 2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanol | Human | 1582 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brg | A | | (5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-acetic | Human | 1589 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | A | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | 1694 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | B | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | 1654 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | A | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | 1621 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | B | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | 1643 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brn | A | | (2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-ol | Human | 1631 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2bro | A | | (2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diol | Human | 1686 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3j | A | | debromohymenialdisine | Human | 1551 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3k | A | | 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenol | Human | 1674 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3l | A | | 3-(1h-benzimidazol-2-yl)-1h-indazole | Human | 1612 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgu | A | | 2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acid | Human | 1697 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgv | A | | (2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-ol | Human | 1545 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgw | A | | 4,4'-(1-propyl-1h-1,2,4-triazole-3,5-diyl)bis(2,5-dihydro-1,2,5-oxadiazol-3-amine) | Human | 1683 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgx | A | | 2-[(6-amino-7h-purin-8-yl)thio]acetamide | Human | 1595 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9n | A | | 3-(4'-hydroxybiphenyl-4-yl)-n-(4-hydroxycyclohexyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamide | Human | 1690 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9o | A | | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | 1667 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9p | A | | 1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}urea | Human | 1618 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9u | A | | 18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-one | Human | 1584 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | A | | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | 1574 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | B | | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | 1638 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2gdo | A | | 4-[(3s)-1-azabicyclo[2.2.2]oct-3-ylamino]-3-(1h-benzimidazol-2-yl)-6-chloroquinolin-2(1h)-one | Human | 1606 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ghg | A | | 5-{5-[(s)-2-amino-3-(1h-indol-3-yl)-propoxyl]-pyridin-3-yl}-3-[1-(1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one | Human | 1581 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hog | A | | (5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanol | Human | 1653 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hxl | A | | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrile | Human | 1552 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hxq | A | | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-one | Human | 1587 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hy0 | A | | 3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-pyrazol-4-yl)quinolin-2(1h)-one | Human | 1555 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2qhm | A | | (3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylate | Human | 1669 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2qhn | A | | 5-ethyl-3-methyl-1,5-dihydro-4h-pyrazolo[4,3-c]quinolin-4-one | Human | 1675 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2r0u | A | | 6-(3-aminopropyl)-4-(3-hydroxyphenyl)-9-(1h-pyrazol-4-yl)benzo[h]isoquinolin-1(2h)-one | Human | 1632 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmq | A | | n-(4-oxo-5,6,7,8-tetrahydro-4h-[1,3]thiazolo[5,4-c]azepin-2-yl)acetamide | Human | 1647 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | A | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | 1609 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | B | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | 1604 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wms | A | | [4-amino-2-(tert-butylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 1657 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | A | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | 1576 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | B | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | 1685 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | A | 6-morpholin-4-yl-9h-purine | Human | 1662 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | B | 6-morpholin-4-yl-9h-purine | Human | 1578 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmv | A | | 1-[(2s)-4-(7h-purin-6-yl)morpholin-2-yl]methanamine | Human | 1562 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmw | A | | 1-[(2s)-4-(5-bromo-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | 1594 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmx | A | | 1-[(2s)-4-(5-phenyl-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | 1636 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | A | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1673 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | B | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1620 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8e | A | | 5-methyl-8-pyridin-4-yl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1548 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | A | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1699 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | B | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1558 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xey | A | | 3-(1h-indol-3-yl)-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | 1668 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xez | A | | 6-(1h-pyrazol-3-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | 1580 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xf0 | A | | 3-phenyl-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | 1534 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | A | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | 1684 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | B | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | 1579 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | A | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 1649 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | B | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 1687 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydk | A | | 2-(carbamoylamino)-5-phenyl-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | 1646 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | A | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | 1611 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | B | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | 1583 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | A | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1651 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | B | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1567 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | A | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1644 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | B | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1543 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | A | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1572 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | B | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1560 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym5 | A | | (3-{4-[(2s)-2-(aminomethyl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}phenyl)methanol | Human | 1627 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | A | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | 1563 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | B | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | 1559 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | A | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | 1650 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | B | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | 1645 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym8 | A | | (r)-5-(8-chloroisoquinolin-3-ylamino)-3-(1-(dimethylamino)propan-2-yloxy)pyrazine-2-carbonitrile | Human | 1588 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ywp | A | | 1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea | Human | 1658 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | A | - | Human | 1700 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | B | - | Human | 1666 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvr | A | | - | Human | 1625 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvs | A | | - | Human | 1630 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3nlb | A | | 3-methyl-5-[5-(1-methylethyl)-1h-benzimidazol-2-yl]-n-(1-methylpiperidin-4-yl)-1h-pyrazole-4-carboxamide | Human | 1641 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | A | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1696 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | B | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1602 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | A | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1569 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | B | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1590 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | 1691 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | 1635 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | 1592 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | 1566 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | A | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | 1676 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | B | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | 1544 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tkh | A | | 1-(morpholin-4-yl)-2-[4-(2-{[5-(pyridin-3-yl)-1,3-thiazol-2-yl]amino}pyridin-4-yl)piperazin-1-yl]ethanone | Human | 1665 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tki | A | | n-(2-aminoethyl)-5-(2-{[4-(morpholin-4-yl)pyridin-2-yl]amino}-1,3-thiazol-5-yl)pyridine-3-carboxamide | Human | 1599 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3u9n | A | | 2-(2,3-dihydro-1-benzofuran-5-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 1597 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | A | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | 1570 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | B | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | 1671 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | A | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | 1542 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | B | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | 1679 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | A | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | 1688 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | B | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | 1598 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | A | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | 1629 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | B | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | 1575 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | A | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | 1619 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | B | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | 1663 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | A | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | 1539 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | B | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | 1615 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | A | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1541 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | B | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1623 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | A | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | 1547 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | B | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | 1537 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | A | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | 1553 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | B | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | 1628 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | A | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | 1637 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | B | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | 1693 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | A | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | 1554 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | B | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | 1672 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | A | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1617 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | B | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1633 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | A | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1610 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | B | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1557 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | A | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | 1564 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | B | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | 1648 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | A | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | 1540 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | B | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | 1660 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | A | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | 1593 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | B | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | 1680 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | A | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | 1577 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | B | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | 1659 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | A | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | 1603 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | B | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | 1613 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | A | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | 1608 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | B | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | 1536 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | A | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | 1614 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | B | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | 1573 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | A | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | 1546 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | B | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | 1556 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | C | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | 1616 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | A | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | 1695 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | B | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | 1678 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | A | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | 1661 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | B | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | 1605 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | A | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | 1664 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | B | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | 1550 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | A | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | 1692 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | B | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | 1535 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | A | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1565 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | B | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1670 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | A | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1639 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | B | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1640 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | A | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1600 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | B | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1652 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | A | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | 1561 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | B | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | 1626 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | A | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 1538 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | B | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 1681 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4jik | A | | 2-(4-chlorophenyl)-8-[(3s)-piperidin-3-ylamino]imidazo[1,2-c]pyrimidine-5-carboxamide | Human | 1698 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qye | A | | 4-[6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | 1601 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyf | A | | 4-[3-amino-6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | 1622 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | A | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | 1568 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | B | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | 1607 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | A | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1689 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | B | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1586 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvk | A | | n-[3-(6-cyano-9h-pyrrolo[2,3-b:5,4-c']dipyridin-3-yl)phenyl]acetamide | Human | 1549 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvl | A | | 3-(2-hydroxyphenyl)-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1634 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvm | A | | 3-[4-(piperidin-1-ylmethyl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1624 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5dls | A | | 1-benzyl-n-(5-{5-[3-(dimethylamino)-2,2-dimethylpropoxy]-1h-indol-2-yl}-6-oxo-1,6-dihydropyridin-3-yl)-1h-pyrazole-4-carboxamide | Human | 6151 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | A | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | 6651 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | B | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | 6652 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 8612 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 8607 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oor | A | | staurosporine | Human | 8603 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oot | A | | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 8599 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8595 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8611 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op4 | A | | [4-[[4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-fluoranyl-5-methoxy-phenyl]-morpholin-4-yl-methanone | Human | 8613 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op5 | A | | 3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | 8600 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op7 | A | | [4-[[5-chloranyl-4-(methylamino)-7~{h}-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-phenyl]-morpholin-4-yl-methanone | Human | 8609 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | A | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | 8602 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | B | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | 8604 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opr | A | | 5-[4-(morpholin-4-ylmethyl)phenyl]-3-(1-propan-2-yl-1,2,3-triazol-4-yl)pyridin-2-amine | Human | 8614 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5ops | A | | 4-(3-hydroxyphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | 8598 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opu | A | | 6-azanyl-4-(3-methylphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | 8615 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opv | A | | 4-(3-methylphenyl)-6-[(1-methylpyrazol-3-yl)amino]-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | 8608 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq5 | A | | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 8597 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq6 | A | | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 8610 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8601 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8594 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8605 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8596 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq8 | A | | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8606 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | A | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | 9500 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | B | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | 9502 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | A | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | 9503 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | B | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | 9498 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | A | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | 9501 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | B | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | 9499 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | A | phosphothiophosphoric acid-adenylate ester | Human | 13489 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | B | phosphothiophosphoric acid-adenylate ester | Human | 13491 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | A | - | Human | 13494 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | B | - | Human | 13493 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | A | staurosporine | Human | 13490 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | B | staurosporine | Human | 13495 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | A | staurosporine | Human | 13492 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | B | staurosporine | Human | 13496 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | A | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | 13775 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | B | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | 13774 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | A | adenine | Human | 13767 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | B | adenine | Human | 13773 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | A | n,n-dimethyl-7h-purin-6-amine | Human | 13776 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | B | n,n-dimethyl-7h-purin-6-amine | Human | 13771 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | A | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 13777 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | B | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 13779 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjm | A | | 4-amino-6-{[(2-fluorophenyl)methyl]amino}-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13770 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjo | A | | 4-amino-6-(2,3-difluorophenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13780 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjr | A | | 4-amino-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13778 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | A | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13772 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | B | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13768 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk1 | A | | 4-amino-2-[(1,3-dimethyl-1h-pyrazol-4-yl)amino]-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13763 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk2 | A | | 4-amino-7-methyl-2-({5-methyl-1-[(3r)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13766 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk3 | A | | 4-amino-7-methyl-2-({5-methyl-1-[(3s)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13764 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bkn | A | | adenine | Human | 13769 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bko | A | | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 13765 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7mck | A | | n-{5-[(3s)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl}-6-(1-methyl-1h-pyrazol-4-yl)pyridine-2-carboxamide | Human | 13622 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | A | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | 14040 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | B | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | 14044 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | A | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | 14039 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | B | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | 14042 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suh | A | | 1-[5-chloro-4-({6-chloro-7-[1-(oxetan-3-yl)piperidin-4-yl]quinazolin-2-yl}amino)-1h-pyrazol-1-yl]-2-methylpropan-2-ol | Human | 14043 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sui | A | | (3r,4r)-4-{(3s,4s)-4-[6-chloro-2-({5-chloro-1-[(1r)-2,2-difluorocyclopropyl]-1h-pyrazol-4-yl}amino)quinazolin-7-yl]-3-fluoropiperidin-1-yl}oxolan-3-ol | Human | 14045 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suj | A | | (3r,4r)-4-{4-[6-chloro-2-({1-[(1r)-2,2-difluorocyclopropyl]-5-methyl-1h-pyrazol-4-yl}amino)quinazolin-7-yl]piperidin-1-yl}-4-methyloxolan-3-ol | Human | 14041 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e80 | A | | 2-[(1r,4r)-2-{(6p)-6-[(6m)-6-(1h-pyrazol-5-yl)-1h-indazol-1-yl]pyrimidin-4-yl}-2-azabicyclo[2.1.1]hexan-4-yl]propan-2-ol | Human | 14621 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e81 | A | | (1s)-1-[(1p)-1-{6-[(3r)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}-1h-indazol-6-yl]spiro[2.2]pentane-1-carbonitrile | Human | 14620 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siv | A | | n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)cyclopropanecarboxamide | Human | 14886 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siw | A | | (1s,2s)-n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)-2-(1-methyl-1h-pyrazol-4-yl)cyclopropane-1-carboxamide | Human | 14885 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8six | A | | (1s)-n-(7-chloro-6-{4-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperazin-1-yl}isoquinolin-3-yl)-6-oxaspiro[2.5]octane-1-carboxamide | Human | 14887 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2cn5 | A | | adenosine-5'-diphosphate | Human | 4789 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2cn8 | A | | debromohymenialdisine | Human | 4808 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2w0j | A | | 4,4'-diacetyldiphenylurea-bis(guanylhydrazone) | Human | 4811 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2w7x | A | A | n-[4-[(e)-n-carbamimidamido-c-methyl-carbonimidoyl]phenyl]-7-nitro-1h-indole-2-carboxamide | Human | 4784 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2w7x | A | B | n-[4-[(e)-n-carbamimidamido-c-methyl-carbonimidoyl]phenyl]-7-nitro-1h-indole-2-carboxamide | Human | 4780 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wtc | A | | 4-[2-amino-5-(4-hydroxy-3-methoxyphenyl)pyridin-3-yl]benzamide | Human | 4767 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wtd | A | | 4-[2-amino-5-(1,3-benzodioxol-4-yl)pyridin-3-yl]benzamide | Human | 4769 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wti | A | A | 4-[2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)pyridin-3-yl]benzamide | Human | 4812 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wti | A | B | 4-[2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)pyridin-3-yl]benzamide | Human | 4807 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wtj | A | A | 2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)-n-[2-(dimethylamino)ethyl]pyridine-3-carboxamide | Human | 4779 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wtj | A | B | 2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)-n-[2-(dimethylamino)ethyl]pyridine-3-carboxamide | Human | 4761 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xbj | A | | 4-fluoro-2-(4-{[(3s,4r)-4-(1-hydroxy-1-methylethyl)pyrrolidin-3-yl]amino}-6,7-dimethoxyquinazolin-2-yl)phenol | Human | 4783 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xk9 | A | | n-{4-[(1e)-n-(n-hydroxycarbamimidoyl)ethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamide | Human | 4771 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xm8 | A | | 2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenol | Human | 4773 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xm9 | A | A | 4-(1h-pyrazol-5-yl)-2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenol | Human | 4785 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xm9 | A | B | 4-(1h-pyrazol-5-yl)-2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenol | Human | 4803 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycf | A | A | (2e)-n-hydroxy-2-[1-(4-{[(4-{(1e)-1-[2-(n'-hydroxycarbamimidoyl)hydrazinylidene]ethyl}phenyl)carbamoyl]amino}phenyl)ethylidene]hydrazinecarboximidamide | Human | 4810 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycf | A | B | (2e)-n-hydroxy-2-[1-(4-{[(4-{(1e)-1-[2-(n'-hydroxycarbamimidoyl)hydrazinylidene]ethyl}phenyl)carbamoyl]amino}phenyl)ethylidene]hydrazinecarboximidamide | Human | 4774 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycq | A | A | n-{4-[(1e)-n-1h-imidazol-2-ylethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamide | Human | 4766 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycq | A | B | n-{4-[(1e)-n-1h-imidazol-2-ylethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamide | Human | 4790 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycr | A | A | 1,3-bis{4-[(1e)-n-(4,5-dihydro-1h-imidazol-2-yl)ethanehydrazonoyl]phenyl}urea | Human | 4760 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycr | A | B | 1,3-bis{4-[(1e)-n-(4,5-dihydro-1h-imidazol-2-yl)ethanehydrazonoyl]phenyl}urea | Human | 4775 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycs | A | A | n-{4-[(1e)-n-carbamimidoylethanehydrazonoyl]phenyl}-1h-indole-3-carboxamide | Human | 4804 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycs | A | B | n-{4-[(1e)-n-carbamimidoylethanehydrazonoyl]phenyl}-1h-indole-3-carboxamide | Human | 4764 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yiq | A | A | (e)-5-(1-(2-carbamimidoylhydrazono)ethyl)-n-(1h-indol-6-yl)-1h-indole-2-carboxamide | Human | 4791 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yiq | A | B | (e)-5-(1-(2-carbamimidoylhydrazono)ethyl)-n-(1h-indol-6-yl)-1h-indole-2-carboxamide | Human | 4800 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yir | A | | (e)-n-(5-(2-carbamimidoylhydrazono)-5,6,7,8-tetrahydronaphthalen-2-yl)-7-nitro-1h-indole-2-carboxamide | Human | 4768 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yit | A | A | n-{4-[(1e)-n-carbamimidoylbutanehydrazonoyl]phenyl}-5-methoxy-1h-indole-2-carboxamide | Human | 4777 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yit | A | B | n-{4-[(1e)-n-carbamimidoylbutanehydrazonoyl]phenyl}-5-methoxy-1h-indole-2-carboxamide | Human | 4770 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6u | A | | - | Human | 4798 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6u | B | | - | Human | 4787 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | A | | - | Human | 4813 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | B | | - | Human | 4792 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | C | | - | Human | 4802 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | D | | - | Human | 4805 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | E | | - | Human | 4806 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | F | | - | Human | 4776 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | G | | - | Human | 4793 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | H | | - | Human | 4799 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9r | A | | 2-[4-(4-chlorophenoxy)phenyl]-1h-benzimidazole-6-carboxamide | Human | 4763 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9s | A | A | 2-(4-(3-hydroxyphenoxy)phenyl)-1h-benzo[d]imidazole-5-carboxamide | Human | 4772 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9s | A | B | 2-(4-(3-hydroxyphenoxy)phenyl)-1h-benzo[d]imidazole-5-carboxamide | Human | 4801 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9t | A | | 2-(4-{[1-(4-chlorobenzyl)piperidin-4-yl]methoxy}phenyl)-1h-benzimidazole-5-carboxamide | Human | 4814 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9u | A | | 2-{4-[(1-benzylpiperidin-4-yl)methoxy]phenyl}-1h-benzimidazole-6-carboxamide | Human | 4778 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bda | A | | 3,4-dihydro[1,2,4]triazolo[1,5-a][3,1]benzimidazol-9-ium | Human | 4788 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdb | A | | 4-[(e)-c-methyl-n-oxidanyl-carbonimidoyl]benzene-1,3-diol | Human | 4797 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdc | A | | n-(furan-2-ylmethyl)quinoxaline-6-carboxamide | Human | 4794 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdd | A | | 1-(tert-butyl)-3-(quinoxalin-6-yl)urea | Human | 4786 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bde | A | | 6-methylquinazolin-4-amine | Human | 4781 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdf | A | | 5-methyl-3-phenyl-1h-pyrazole | Human | 4765 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdg | A | | 3-(pyridin-3-yl)-1h-pyrazol-5-amine | Human | 4796 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdh | A | | 3-methyl-4-(thiophen-2-yl)-1h-pyrazol-5-amine | Human | 4782 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdi | A | | 1-acetyl-n-(5-methylpyridin-2-yl)piperidine-4-carboxamide | Human | 4762 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdj | A | | 3-cyclopropyl-4-(furan-2-yl)-1h-pyrazolo[3,4-b]pyridine | Human | 4795 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdk | A | | n-[(4-methoxyphenyl)methyl]quinoxaline-6-carboxamide | Human | 4809 | |
| CHUK (IKKa) | IKK | Other | 5ebz | A | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7153 | |
| CHUK (IKKa) | IKK | Other | 5ebz | B | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7145 | |
| CHUK (IKKa) | IKK | Other | 5ebz | C | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7146 | |
| CHUK (IKKa) | IKK | Other | 5ebz | D | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7144 | |
| CHUK (IKKa) | IKK | Other | 5ebz | E | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7151 | |
| CHUK (IKKa) | IKK | Other | 5ebz | F | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7149 | |
| CHUK (IKKa) | IKK | Other | 5ebz | G | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7154 | |
| CHUK (IKKa) | IKK | Other | 5ebz | H | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7155 | |
| CHUK (IKKa) | IKK | Other | 5ebz | I | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7152 | |
| CHUK (IKKa) | IKK | Other | 5ebz | J | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7148 | |
| CHUK (IKKa) | IKK | Other | 5ebz | K | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7150 | |
| CHUK (IKKa) | IKK | Other | 5ebz | L | | 2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamide | Human | 7147 | |
| CHUK (IKKa) | IKK | Other | 5tqw | A | | - | Human | 7249 | |
| CHUK (IKKa) | IKK | Other | 5tqw | B | | - | Human | 7248 | |
| CHUK (IKKa) | IKK | Other | 5tqx | A | | - | Human | 7261 | |
| CHUK (IKKa) | IKK | Other | 5tqx | B | | - | Human | 7262 | |
| CHUK (IKKa) | IKK | Other | 5tqy | A | | - | Human | 7196 | |
| CHUK (IKKa) | IKK | Other | 5tqy | B | | - | Human | 7197 | |
| CLK1 | CLK | CMGC | 1z57 | A | A | debromohymenialdisine | Human | 106 | |
| CLK1 | CLK | CMGC | 1z57 | A | B | debromohymenialdisine | Human | 105 | |
| CLK1 | CLK | CMGC | 2vag | A | A | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 104 | |
| CLK1 | CLK | CMGC | 2vag | A | B | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 103 | |
| CLK1 | CLK | CMGC | 5j1v | A | | pyrido[3,4-g]quinazoline-2,10-diamine | Human | 6582 | |
| CLK1 | CLK | CMGC | 5j1v | B | | pyrido[3,4-g]quinazoline-2,10-diamine | Human | 6580 | |
| CLK1 | CLK | CMGC | 5j1v | C | | pyrido[3,4-g]quinazoline-2,10-diamine | Human | 6577 | |
| CLK1 | CLK | CMGC | 5j1w | A | A | pyrido[3,4-g]quinazolin-2-amine | Human | 6579 | |
| CLK1 | CLK | CMGC | 5j1w | A | B | pyrido[3,4-g]quinazolin-2-amine | Human | 6576 | |
| CLK1 | CLK | CMGC | 5j1w | B | A | pyrido[3,4-g]quinazolin-2-amine | Human | 6575 | |
| CLK1 | CLK | CMGC | 5j1w | B | B | pyrido[3,4-g]quinazolin-2-amine | Human | 6583 | |
| CLK1 | CLK | CMGC | 5j1w | C | A | pyrido[3,4-g]quinazolin-2-amine | Human | 6578 | |
| CLK1 | CLK | CMGC | 5j1w | C | B | pyrido[3,4-g]quinazolin-2-amine | Human | 6581 | |
| CLK1 | CLK | CMGC | 5x8i | A | | 5-[1-[(1s)-1-(4-fluorophenyl)ethyl]-[1,2,3]triazolo[4,5-c]quinolin-8-yl]-1,3-benzoxazole | Human | 8316 | |
| CLK1 | CLK | CMGC | 5x8i | B | | 5-[1-[(1s)-1-(4-fluorophenyl)ethyl]-[1,2,3]triazolo[4,5-c]quinolin-8-yl]-1,3-benzoxazole | Human | 8317 | |
| CLK1 | CLK | CMGC | 6ft8 | A | A | 3-(3-hydroxyphenyl)-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9895 | |
| CLK1 | CLK | CMGC | 6ft8 | A | B | 3-(3-hydroxyphenyl)-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9899 | |
| CLK1 | CLK | CMGC | 6ft9 | A | A | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9901 | |
| CLK1 | CLK | CMGC | 6ft9 | A | B | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9898 | |
| CLK1 | CLK | CMGC | 6ft9 | B | A | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9897 | |
| CLK1 | CLK | CMGC | 6ft9 | B | B | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9894 | |
| CLK1 | CLK | CMGC | 6ft9 | C | A | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9896 | |
| CLK1 | CLK | CMGC | 6ft9 | C | B | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9900 | |
| CLK1 | CLK | CMGC | 6fyo | A | A | 6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamide | Human | 10324 | |
| CLK1 | CLK | CMGC | 6fyo | A | B | 6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamide | Human | 10323 | |
| CLK1 | CLK | CMGC | 6g33 | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9819 | |
| CLK1 | CLK | CMGC | 6g33 | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9824 | |
| CLK1 | CLK | CMGC | 6g33 | A | C | - | Human | 9826 | |
| CLK1 | CLK | CMGC | 6g33 | B | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9821 | |
| CLK1 | CLK | CMGC | 6g33 | B | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9822 | |
| CLK1 | CLK | CMGC | 6g33 | B | C | - | Human | 9827 | |
| CLK1 | CLK | CMGC | 6g33 | C | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9825 | |
| CLK1 | CLK | CMGC | 6g33 | C | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9823 | |
| CLK1 | CLK | CMGC | 6g33 | C | C | - | Human | 9820 | |
| CLK1 | CLK | CMGC | 6i5h | A | A | 5-(1-methylpyrazol-4-yl)-3-(3-phenoxyphenyl)furo[3,2-b]pyridine | Human | 10848 | |
| CLK1 | CLK | CMGC | 6i5h | A | B | 5-(1-methylpyrazol-4-yl)-3-(3-phenoxyphenyl)furo[3,2-b]pyridine | Human | 10849 | |
| CLK1 | CLK | CMGC | 6i5i | A | A | 5-(1-methylpyrazol-4-yl)-3-[1-(phenylmethyl)pyrazol-4-yl]furo[3,2-b]pyridine | Human | 10845 | |
| CLK1 | CLK | CMGC | 6i5i | A | B | 5-(1-methylpyrazol-4-yl)-3-[1-(phenylmethyl)pyrazol-4-yl]furo[3,2-b]pyridine | Human | 10840 | |
| CLK1 | CLK | CMGC | 6i5k | A | A | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10844 | |
| CLK1 | CLK | CMGC | 6i5k | A | B | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10836 | |
| CLK1 | CLK | CMGC | 6i5k | B | A | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10842 | |
| CLK1 | CLK | CMGC | 6i5k | B | B | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10835 | |
| CLK1 | CLK | CMGC | 6i5k | C | A | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10834 | |
| CLK1 | CLK | CMGC | 6i5k | C | B | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10838 | |
| CLK1 | CLK | CMGC | 6i5l | A | A | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10837 | |
| CLK1 | CLK | CMGC | 6i5l | A | B | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10843 | |
| CLK1 | CLK | CMGC | 6i5l | B | A | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10846 | |
| CLK1 | CLK | CMGC | 6i5l | B | B | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10839 | |
| CLK1 | CLK | CMGC | 6i5l | C | A | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10833 | |
| CLK1 | CLK | CMGC | 6i5l | C | B | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10841 | |
| CLK1 | CLK | CMGC | 6khd | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11646 | |
| CLK1 | CLK | CMGC | 6khd | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11645 | |
| CLK1 | CLK | CMGC | 6khd | B | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11644 | |
| CLK1 | CLK | CMGC | 6khd | B | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11647 | |
| CLK1 | CLK | CMGC | 6khd | C | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11648 | |
| CLK1 | CLK | CMGC | 6khd | C | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11643 | |
| CLK1 | CLK | CMGC | 6q8k | A | A | ~{n}2-(3-morpholin-4-ylpropyl)pyrido[3,4-g]quinazoline-2,10-diamine | Human | 10902 | |
| CLK1 | CLK | CMGC | 6q8k | A | B | ~{n}2-(3-morpholin-4-ylpropyl)pyrido[3,4-g]quinazoline-2,10-diamine | Human | 10903 | |
| CLK1 | CLK | CMGC | 6q8p | A | | ~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amine | Human | 10899 | |
| CLK1 | CLK | CMGC | 6q8p | B | | ~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amine | Human | 10900 | |
| CLK1 | CLK | CMGC | 6q8p | C | | ~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amine | Human | 10901 | |
| CLK1 | CLK | CMGC | 6qty | A | A | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 12083 | |
| CLK1 | CLK | CMGC | 6qty | A | B | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 12084 | |
| CLK1 | CLK | CMGC | 6r3d | A | | 4-[6,7-bis(chloranyl)-1~{h}-indol-3-yl]pyrimidin-2-amine | Human | 12128 | |
| CLK1 | CLK | CMGC | 6r6e | A | | 5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amine | Human | 12232 | |
| CLK1 | CLK | CMGC | 6r6x | A | | 5-(1-methylindol-3-yl)pyrimidin-4-amine | Human | 12231 | |
| CLK1 | CLK | CMGC | 6r8j | A | A | 4-(1-methylindol-3-yl)pyrimidin-2-amine | Human | 12632 | |
| CLK1 | CLK | CMGC | 6r8j | A | B | 4-(1-methylindol-3-yl)pyrimidin-2-amine | Human | 12631 | |
| CLK1 | CLK | CMGC | 6raa | A | A | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11014 | |
| CLK1 | CLK | CMGC | 6raa | A | B | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11013 | |
| CLK1 | CLK | CMGC | 6tw2 | E | A | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 11962 | |
| CLK1 | CLK | CMGC | 6tw2 | E | B | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 11963 | |
| CLK1 | CLK | CMGC | 6yta | A | A | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 12423 | |
| CLK1 | CLK | CMGC | 6yta | A | B | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 12417 | |
| CLK1 | CLK | CMGC | 6ytd | A | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12418 | |
| CLK1 | CLK | CMGC | 6ytd | A | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12420 | |
| CLK1 | CLK | CMGC | 6yte | C | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12419 | |
| CLK1 | CLK | CMGC | 6yte | C | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12422 | |
| CLK1 | CLK | CMGC | 6ytg | A | A | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12416 | |
| CLK1 | CLK | CMGC | 6ytg | A | B | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12424 | |
| CLK1 | CLK | CMGC | 6yti | A | A | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 12413 | |
| CLK1 | CLK | CMGC | 6yti | A | B | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 12414 | |
| CLK1 | CLK | CMGC | 6z4z | A | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12315 | |
| CLK1 | CLK | CMGC | 6z4z | A | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12312 | |
| CLK1 | CLK | CMGC | 6z4z | B | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12310 | |
| CLK1 | CLK | CMGC | 6z4z | B | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12311 | |
| CLK1 | CLK | CMGC | 6z4z | C | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12309 | |
| CLK1 | CLK | CMGC | 6z4z | C | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12313 | |
| CLK1 | CLK | CMGC | 6z50 | A | A | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12314 | |
| CLK1 | CLK | CMGC | 6z50 | A | B | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12308 | |
| CLK1 | CLK | CMGC | 6zln | A | A | 4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 12711 | |
| CLK1 | CLK | CMGC | 6zln | A | B | 4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 12710 | |
| CLK1 | CLK | CMGC | 7ak3 | A | A | ~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 13142 | |
| CLK1 | CLK | CMGC | 7ak3 | A | B | ~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 13143 | |
| CLK1 | CLK | CMGC | 7o9y | A | | 4-(1~{h}-indol-3-yl)pyrimidin-2-amine | Human | 14208 | |
| CLK1 | CLK | CMGC | 7oa0 | A | | 5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amine | Human | 14207 | |
| CLK1 | CLK | CMGC | 7opg | A | A | 4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenol | Human | 13808 | |
| CLK1 | CLK | CMGC | 7opg | A | B | 4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenol | Human | 13809 | |
| CLK1 | CLK | CMGC | 8p04 | A | | (4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-one | Human | 14741 | |
| CLK1 | CLK | CMGC | 8p08 | A | | (4~{z})-4-(1,3-benzothiazol-6-ylmethylidene)-2-[[(2~{r})-1-methoxy-4-methyl-pentan-2-yl]amino]-1~{h}-imidazol-5-one | Human | 14742 | |
| CLK2 | CLK | CMGC | 3nr9 | A | | (5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 1927 | |
| CLK2 | CLK | CMGC | 3nr9 | B | | (5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 1928 | |
| CLK2 | CLK | CMGC | 3nr9 | C | | (5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 1929 | |
| CLK2 | CLK | CMGC | 5unp | A | | n~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamine | Human | 9887 | |
| CLK2 | CLK | CMGC | 5unp | B | | n~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamine | Human | 9888 | |
| CLK2 | CLK | CMGC | 6fyi | A | | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 10405 | |
| CLK2 | CLK | CMGC | 6fyk | A | A | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10406 | |
| CLK2 | CLK | CMGC | 6fyk | A | B | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10408 | |
| CLK2 | CLK | CMGC | 6fyk | B | A | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10407 | |
| CLK2 | CLK | CMGC | 6fyk | B | B | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10401 | |
| CLK2 | CLK | CMGC | 6fyk | C | A | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10402 | |
| CLK2 | CLK | CMGC | 6fyk | C | B | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10409 | |
| CLK2 | CLK | CMGC | 6fyl | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10403 | |
| CLK2 | CLK | CMGC | 6fyl | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10404 | |
| CLK2 | CLK | CMGC | 6khe | A | | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11651 | |
| CLK3 | CLK | CMGC | 2eu9 | A | A | - | Human | 1826 | |
| CLK3 | CLK | CMGC | 2eu9 | A | B | - | Human | 1830 | |
| CLK3 | CLK | CMGC | 2exe | A | A | - | Human | 1822 | |
| CLK3 | CLK | CMGC | 2exe | A | B | - | Human | 1819 | |
| CLK3 | CLK | CMGC | 2wu6 | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1823 | |
| CLK3 | CLK | CMGC | 2wu6 | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1821 | |
| CLK3 | CLK | CMGC | 2wu7 | A | A | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 1828 | |
| CLK3 | CLK | CMGC | 2wu7 | A | B | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 1827 | |
| CLK3 | CLK | CMGC | 3raw | A | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 1820 | |
| CLK3 | CLK | CMGC | 3raw | A | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 1829 | |
| CLK3 | CLK | CMGC | 3raw | B | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 1824 | |
| CLK3 | CLK | CMGC | 3raw | B | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 1825 | |
| CLK3 | CLK | CMGC | 6ft7 | A | A | 3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9905 | |
| CLK3 | CLK | CMGC | 6ft7 | A | B | 3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9903 | |
| CLK3 | CLK | CMGC | 6ft7 | B | A | 3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9904 | |
| CLK3 | CLK | CMGC | 6ft7 | B | B | 3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9902 | |
| CLK3 | CLK | CMGC | 6fyp | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10400 | |
| CLK3 | CLK | CMGC | 6fyp | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10397 | |
| CLK3 | CLK | CMGC | 6fyr | A | A | 6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamide | Human | 11407 | |
| CLK3 | CLK | CMGC | 6fyr | A | B | 6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamide | Human | 11406 | |
| CLK3 | CLK | CMGC | 6khf | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11650 | |
| CLK3 | CLK | CMGC | 6khf | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11649 | |
| CLK3 | CLK | CMGC | 6rct | A | A | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11127 | |
| CLK3 | CLK | CMGC | 6rct | A | B | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11126 | |
| CLK3 | CLK | CMGC | 6rct | B | A | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11128 | |
| CLK3 | CLK | CMGC | 6rct | B | B | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11129 | |
| CLK3 | CLK | CMGC | 6ytw | A | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12404 | |
| CLK3 | CLK | CMGC | 6ytw | A | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12407 | |
| CLK3 | CLK | CMGC | 6ytw | B | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12412 | |
| CLK3 | CLK | CMGC | 6ytw | B | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12410 | |
| CLK3 | CLK | CMGC | 6yty | A | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12409 | |
| CLK3 | CLK | CMGC | 6yty | A | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12406 | |
| CLK3 | CLK | CMGC | 6yu1 | a | A | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12403 | |
| CLK3 | CLK | CMGC | 6yu1 | a | B | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12408 | |
| CLK3 | CLK | CMGC | 6yu1 | c | A | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12405 | |
| CLK3 | CLK | CMGC | 6yu1 | c | B | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12411 | |
| CLK3 | CLK | CMGC | 6z2v | A | A | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12637 | |
| CLK3 | CLK | CMGC | 6z2v | A | B | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12636 | |
| CLK3 | CLK | CMGC | 6z51 | A | A | n-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide | Human | 12296 | |
| CLK3 | CLK | CMGC | 6z51 | A | B | n-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide | Human | 12304 | |
| CLK3 | CLK | CMGC | 6z52 | A | A | 11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12628 | |
| CLK3 | CLK | CMGC | 6z52 | A | B | 11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12627 | |
| CLK3 | CLK | CMGC | 6z52 | B | A | 11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12629 | |
| CLK3 | CLK | CMGC | 6z52 | B | B | 11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12626 | |
| CLK3 | CLK | CMGC | 6z53 | A | A | 6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12300 | |
| CLK3 | CLK | CMGC | 6z53 | A | B | 6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12305 | |
| CLK3 | CLK | CMGC | 6z54 | A | A | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12294 | |
| CLK3 | CLK | CMGC | 6z54 | A | B | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12295 | |
| CLK3 | CLK | CMGC | 6z55 | A | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12302 | |
| CLK3 | CLK | CMGC | 6z55 | A | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12298 | |
| CLK3 | CLK | CMGC | 6z55 | A | C | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12301 | |
| CLK3 | CLK | CMGC | 6z55 | B | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12303 | |
| CLK3 | CLK | CMGC | 6z55 | B | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12299 | |
| CLK3 | CLK | CMGC | 6z55 | B | C | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12297 | |
| CLK4 | CLK | CMGC | 6fyv | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10511 | |
| CLK4 | CLK | CMGC | 6fyv | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10510 | |
| COQ8A (ADCK3) | ABC1 | Atypical | 4ped | A | A | - | Human | 9121 | |
| COQ8A (ADCK3) | ABC1 | Atypical | 4ped | A | B | - | Human | 9120 | |
| COQ8A (ADCK3) | ABC1 | Atypical | 5i35 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 9122 | |
| COQ8A (ADCK3) | ABC1 | Atypical | 7udp | A | | 4-[(3,4,5-trimethoxyphenyl)amino]quinoline-7-carbonitrile | Human | 14589 | |
| COQ8A (ADCK3) | ABC1 | Atypical | 7udq | A | | 4-[(3,4,5-trimethoxyphenyl)amino]quinoline-7-carbonitrile | Human | 14588 | |
| CSF1R (FMS) | PDGFR | TK | 2i0v | A | | 6-chloro-3-(3-methylisoxazol-5-yl)-4-phenylquinolin-2(1h)-one | Human | 2303 | |
| CSF1R (FMS) | PDGFR | TK | 2i0y | A | | 5-cyano-furan-2-carboxylic acid [5-hydroxymethyl-2-(4-methyl-piperidin-1-yl)-phenyl]-amide | Human | 2315 | |
| CSF1R (FMS) | PDGFR | TK | 2i1m | A | | 5-cyano-furan-2-carboxylic acid [5-hydroxymethyl-2-(4-methyl-piperidin-1-yl)-phenyl]-amide | Human | 2306 | |
| CSF1R (FMS) | PDGFR | TK | 2ogv | A | | - | Human | 1243 | |
| CSF1R (FMS) | PDGFR | TK | 3bea | A | | 8-(2,3-dihydro-1h-inden-5-yl)-2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]phenyl}amino)-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 6761 | |
| CSF1R (FMS) | PDGFR | TK | 3dpk | A | A | 8-cyclohexyl-n-methoxy-5-oxo-2-{[4-(2-pyrrolidin-1-ylethyl)phenyl]amino}-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 2312 | |
| CSF1R (FMS) | PDGFR | TK | 3dpk | A | B | 8-cyclohexyl-n-methoxy-5-oxo-2-{[4-(2-pyrrolidin-1-ylethyl)phenyl]amino}-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 2305 | |
| CSF1R (FMS) | PDGFR | TK | 3krj | A | A | 4-cyano-n-(2-cyclohex-1-en-1-yl-4-piperidin-4-ylphenyl)-1h-imidazole-2-carboxamide | Human | 2302 | |
| CSF1R (FMS) | PDGFR | TK | 3krj | A | B | 4-cyano-n-(2-cyclohex-1-en-1-yl-4-piperidin-4-ylphenyl)-1h-imidazole-2-carboxamide | Human | 2310 | |
| CSF1R (FMS) | PDGFR | TK | 3krl | A | A | 5-cyano-n-[4-(4-methylpiperazin-1-yl)-2-piperidin-1-ylphenyl]furan-2-carboxamide | Human | 2309 | |
| CSF1R (FMS) | PDGFR | TK | 3krl | A | B | 5-cyano-n-[4-(4-methylpiperazin-1-yl)-2-piperidin-1-ylphenyl]furan-2-carboxamide | Human | 2311 | |
| CSF1R (FMS) | PDGFR | TK | 3lcd | A | A | n~3~-(2,6-dichlorobenzyl)-5-(4-{[(2r)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]carbonyl}phenyl)pyrazine-2,3-diamine | Human | 1241 | |
| CSF1R (FMS) | PDGFR | TK | 3lcd | A | B | n~3~-(2,6-dichlorobenzyl)-5-(4-{[(2r)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]carbonyl}phenyl)pyrazine-2,3-diamine | Human | 1242 | |
| CSF1R (FMS) | PDGFR | TK | 3lco | A | A | 3-({4-methoxy-5-[(4-methoxybenzyl)oxy]pyridin-2-yl}methoxy)-5-(1-methyl-1h-pyrazol-4-yl)pyrazin-2-amine | Human | 2314 | |
| CSF1R (FMS) | PDGFR | TK | 3lco | A | B | 3-({4-methoxy-5-[(4-methoxybenzyl)oxy]pyridin-2-yl}methoxy)-5-(1-methyl-1h-pyrazol-4-yl)pyrazin-2-amine | Human | 2313 | |
| CSF1R (FMS) | PDGFR | TK | 4hw7 | A | | 5-[(5-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-[4-(trifluoromethyl)benzyl]pyridin-2-amine | Human | 2304 | |
| CSF1R (FMS) | PDGFR | TK | 4r7h | A | | 5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amine | Human | 2308 | |
| CSF1R (FMS) | PDGFR | TK | 4r7i | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 2307 | |
| CSF1R (FMS) | PDGFR | TK | 6ig8 | A | A | (3-{4-[(4-cyclopropylphenyl)methoxy]-3-methoxyphenyl}azetidin-1-yl)(4-{[(2s)-2,3-dihydroxypropoxy]methyl}pyridin-2-yl)methanone | Human | 11519 | |
| CSF1R (FMS) | PDGFR | TK | 6ig8 | A | B | (3-{4-[(4-cyclopropylphenyl)methoxy]-3-methoxyphenyl}azetidin-1-yl)(4-{[(2s)-2,3-dihydroxypropoxy]methyl}pyridin-2-yl)methanone | Human | 11518 | |
| CSF1R (FMS) | PDGFR | TK | 6n33 | A | | 6-fluoro-n-[(5-fluoro-2-methoxypyridin-3-yl)methyl]-5-[(5-methyl-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]pyridin-2-amine | Human | 11634 | |
| CSF1R (FMS) | PDGFR | TK | 6t2w | A | | 2-[(4-methoxy-2-methyl-phenyl)amino]-7-methyl-9-(4-oxidanylcyclohexyl)purin-8-one | Human | 11905 | |
| CSF1R (FMS) | PDGFR | TK | 6wxj | A | | 4-(3-{[(2s)-2-(6-methoxypyridin-3-yl)-2,3-dihydro-1,4-benzodioxin-6-yl]methyl}-3h-imidazo[4,5-b]pyridin-6-yl)-2-methylbut-3-yn-2-amine | Human | 13337 | |
| CSF1R (FMS) | PDGFR | TK | 7mfc | A | A | vimseltinib | Human | 13990 | |
| CSF1R (FMS) | PDGFR | TK | 7mfc | A | B | vimseltinib | Human | 13989 | |
| CSF1R (FMS) | PDGFR | TK | 7tnh | A | | 2,2-dimethyl-n-[(6-methyl-5-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}pyridin-2-yl)carbamoyl]propanamide | Human | 14350 | |
| CSF1R (FMS) | PDGFR | TK | 8cgc | A | A | [4-[4-[methyl-[(3-methylphenyl)methyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]methanol | Human | 14766 | |
| CSF1R (FMS) | PDGFR | TK | 8cgc | A | B | [4-[4-[methyl-[(3-methylphenyl)methyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]methanol | Human | 14767 | |
| CSF1R (FMS) | PDGFR | TK | 8jot | A | | n-(2-(dimethylamino)ethyl)-1-(3-((4-((2-methyl-1h-indol-5-yl)oxy)pyrimidin-2-yl)amino)phenyl)methanesulfonamide | Human | 15255 | |
| CSK | Csk | TK | 1byg | A | | staurosporine | Human | 2943 | |
| CSK | Csk | TK | 3d7t | A | | staurosporine | Human | 2941 | |
| CSK | Csk | TK | 3d7u | A | | - | Human | 2942 | |
| CSK | Csk | TK | 3d7u | C | | - | Human | 2944 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 5fqd | C | | - | Human | 6415 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 5fqd | F | | - | Human | 6416 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 6gzd | A | A | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10560 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 6gzd | A | B | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10561 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 8g66 | C | | - | Human | 15006 | |
| Csnk1d (CK1d) | CK1 | CK1 | 4jjr | A | | - | Mouse | 5784 | |
| Csnk1d (CK1d) | CK1 | CK1 | 4jjr | B | | - | Mouse | 5785 | |
| Csnk1d (CK1d) | CK1 | CK1 | 5x17 | A | A | adenosine-5'-diphosphate | Mouse | 8546 | |
| Csnk1d (CK1d) | CK1 | CK1 | 5x17 | A | B | adenosine-5'-diphosphate | Mouse | 8544 | |
| Csnk1d (CK1d) | CK1 | CK1 | 5x17 | B | A | adenosine-5'-diphosphate | Mouse | 8545 | |
| Csnk1d (CK1d) | CK1 | CK1 | 5x17 | B | B | adenosine-5'-diphosphate | Mouse | 8547 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uys | A | | - | Human | 2183 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uys | B | | - | Human | 2159 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uys | C | | - | Human | 2149 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uys | D | | - | Human | 2180 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uyt | A | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2182 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uyt | B | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2166 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uyt | C | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2152 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uyt | D | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2163 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uzp | A | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2158 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uzp | B | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2177 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4hgt | A | | 2-{2-[(3,4-difluorophenoxy)methyl]-5-methoxypyridin-4-yl}-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 2181 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4hgt | B | | 2-{2-[(3,4-difluorophenoxy)methyl]-5-methoxypyridin-4-yl}-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 2179 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4hnf | A | | 3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 2194 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4hnf | B | | 3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 2193 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | A | A | 1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamine | Human | 2171 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | A | B | 1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamine | Human | 2161 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | B | A | n-benzyl-4-(pyridin-3-yl)pyrimidin-2-amine | Human | 2148 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | B | B | n-benzyl-4-(pyridin-3-yl)pyrimidin-2-amine | Human | 2147 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | C | A | 1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamine | Human | 2189 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | C | B | 1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamine | Human | 2164 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | D | A | n-benzyl-4-(pyridin-3-yl)pyrimidin-2-amine | Human | 2146 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | D | B | n-benzyl-4-(pyridin-3-yl)pyrimidin-2-amine | Human | 2188 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | A | A | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2151 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | A | B | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2141 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | B | A | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2191 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | B | B | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2175 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | C | A | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2172 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | C | B | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2184 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | D | A | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2160 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | D | B | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2142 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbc | A | A | {4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanol | Human | 2154 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbc | A | B | {4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanol | Human | 2156 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbc | B | A | {4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanol | Human | 2153 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbc | B | B | {4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanol | Human | 2150 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | A | A | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2192 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | A | B | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2176 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | B | A | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2174 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | B | B | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2187 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | C | A | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2169 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | C | B | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2165 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | D | A | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2190 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | D | B | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2145 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tn6 | A | A | 4-{4-(4-fluorophenyl)-1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1h-imidazol-5-yl}pyrimidin-2-amine | Human | 2168 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tn6 | A | B | 4-{4-(4-fluorophenyl)-1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1h-imidazol-5-yl}pyrimidin-2-amine | Human | 2186 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tn6 | B | A | - | Human | 2173 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tn6 | B | B | - | Human | 2162 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tw9 | A | A | octyl beta-l-talopyranoside | Human | 2143 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tw9 | A | B | octyl beta-l-talopyranoside | Human | 2155 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tw9 | B | A | n-(2,2-difluoro-5h-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-2-{[2-(trifluoromethoxy)benzoyl]amino}-1,3-thiazole-4-carboxamide | Human | 2178 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tw9 | B | B | n-(2,2-difluoro-5h-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-2-{[2-(trifluoromethoxy)benzoyl]amino}-1,3-thiazole-4-carboxamide | Human | 2167 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4twc | A | A | 2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamide | Human | 2185 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4twc | A | B | 2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamide | Human | 2157 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4twc | B | A | 2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamide | Human | 2170 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4twc | B | B | 2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamide | Human | 2144 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih4 | A | A | - | Human | 6530 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih4 | A | B | - | Human | 6534 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih4 | A | C | - | Human | 6529 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih4 | A | D | - | Human | 6531 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | A | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | 6527 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | B | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | 6533 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | C | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | 6526 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | D | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | 6528 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih6 | A | A | 6-(3-bromophenyl)pteridine-2,4,7-triamine | Human | 6535 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih6 | A | B | 6-(3-bromophenyl)pteridine-2,4,7-triamine | Human | 6532 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | A | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7532 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | A | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7534 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | B | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7542 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | B | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7540 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | C | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7541 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | C | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7535 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | D | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7537 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | D | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7539 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | E | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7543 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | E | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7538 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | F | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7536 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | F | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7533 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | A | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9862 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | A | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9861 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | B | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9860 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | B | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9857 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | C | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9858 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | C | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9859 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | D | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9855 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | D | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9856 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | A | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8174 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | A | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8177 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | B | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8173 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | B | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8179 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | C | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8175 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | C | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8178 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | D | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8176 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | D | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8180 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f1w | A | A | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10959 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f1w | A | B | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10957 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f1w | B | A | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10960 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f1w | B | B | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10961 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | A | A | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10955 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | A | B | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10953 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | A | C | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10954 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | B | A | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10958 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | B | B | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10956 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | B | C | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10952 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6gzm | A | A | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10426 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6gzm | A | B | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10425 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6gzm | B | A | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10423 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6gzm | B | B | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10424 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmp | A | A | - | Human | 11608 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmp | A | B | - | Human | 11609 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmp | B | A | - | Human | 11607 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmp | B | B | - | Human | 11610 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmr | A | A | - | Human | 11612 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmr | A | B | - | Human | 11606 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmr | B | A | - | Human | 11605 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmr | B | B | - | Human | 11611 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxn | A | A | - | Human | 11972 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxn | A | B | - | Human | 11977 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxn | B | A | - | Human | 11969 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxn | B | B | - | Human | 11978 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxo | A | A | - | Human | 11971 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxo | A | B | - | Human | 11976 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxo | B | A | - | Human | 11974 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxo | B | B | - | Human | 11975 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxp | A | | - | Human | 11970 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxp | B | | - | Human | 11973 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rcg | A | A | ~{n}-[[6,7-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(3-fluorophenyl)-2-morpholin-4-yl-purin-6-amine | Human | 12112 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rcg | A | B | ~{n}-[[6,7-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(3-fluorophenyl)-2-morpholin-4-yl-purin-6-amine | Human | 12109 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | A | A | ~{n}-[[4,5-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-naphthalen-2-yl-purin-6-amine | Human | 12108 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | A | B | ~{n}-[[4,5-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-naphthalen-2-yl-purin-6-amine | Human | 12107 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | A | C | ~{n}-[[4,5-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-naphthalen-2-yl-purin-6-amine | Human | 12111 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | B | A | - | Human | 12106 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | B | B | - | Human | 12110 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | B | C | - | Human | 12113 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru6 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 12260 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru6 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 12256 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru6 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 12259 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru6 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 12251 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru7 | A | A | adenosine-5'-diphosphate | Human | 12264 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru7 | A | B | adenosine-5'-diphosphate | Human | 12253 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru7 | B | A | adenosine-5'-diphosphate | Human | 12252 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru7 | B | B | adenosine-5'-diphosphate | Human | 12263 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | A | A | adenosine-5'-diphosphate | Human | 12258 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | A | B | adenosine-5'-diphosphate | Human | 12255 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | B | A | adenosine-5'-diphosphate | Human | 12265 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | B | B | adenosine-5'-diphosphate | Human | 12261 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | C | A | adenosine-5'-diphosphate | Human | 12266 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | C | B | adenosine-5'-diphosphate | Human | 12254 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | D | A | adenosine-5'-diphosphate | Human | 12262 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | D | B | adenosine-5'-diphosphate | Human | 12257 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7nzy | A | A | 9-chloranyl-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine | Human | 14381 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7nzy | A | B | 9-chloranyl-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine | Human | 14382 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7f | A | A | adenosine monophosphate | Human | 14188 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7f | A | B | adenosine monophosphate | Human | 14185 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7g | A | A | adenosine monophosphate | Human | 14187 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7g | A | B | adenosine monophosphate | Human | 14186 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7h | A | | adenosine monophosphate | Human | 14184 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qr9 | A | A | 4-[5-(4-fluorophenyl)-3-(pyridin-4-ylmethyl)imidazol-4-yl]-1~{h}-pyrrolo[2,3-b]pyridine | Human | 14579 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qr9 | A | B | 4-[5-(4-fluorophenyl)-3-(pyridin-4-ylmethyl)imidazol-4-yl]-1~{h}-pyrrolo[2,3-b]pyridine | Human | 14577 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qra | A | | 4-[3-cyclohexyl-5-(4-fluorophenyl)imidazol-4-yl]-1~{h}-pyrrolo[2,3-b]pyridine | Human | 14578 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qrb | A | A | 3-(dimethylamino)-~{n}-[4-[4-(4-fluorophenyl)-5-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)imidazol-1-yl]cyclohexyl]propane-1-sulfonamide | Human | 14580 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qrb | A | B | 3-(dimethylamino)-~{n}-[4-[4-(4-fluorophenyl)-5-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)imidazol-1-yl]cyclohexyl]propane-1-sulfonamide | Human | 14576 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8d7m | A | | - | Human | 14740 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8d7n | A | | - | Human | 14738 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8d7o | A | | - | Human | 14739 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8d7p | A | | - | Human | 14737 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8izc | A | A | ~{n}5-~{tert}-butyl-2-(3-chloranyl-4-fluoranyl-phenyl)-6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazine-3,5-dicarboxamide | Human | 15270 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8izc | A | B | ~{n}5-~{tert}-butyl-2-(3-chloranyl-4-fluoranyl-phenyl)-6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazine-3,5-dicarboxamide | Human | 15269 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hni | A | | 3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 1722 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hni | B | | 3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 1731 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | A | | - | Human | 1718 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | C | | - | Human | 1723 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | E | | - | Human | 1720 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | G | | - | Human | 1719 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | I | | - | Human | 1724 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | K | | - | Human | 1729 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | M | | - | Human | 1727 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | O | | - | Human | 1726 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | Q | | - | Human | 1730 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | S | | - | Human | 1721 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | U | | - | Human | 1725 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | W | | - | Human | 1728 | |
| CSNK1G1 (CK1g1) | CK1 | CK1 | 2cmw | A | A | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 5567 | |
| CSNK1G1 (CK1g1) | CK1 | CK1 | 2cmw | A | B | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 5566 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4618 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4621 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | B | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4622 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | B | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4620 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | C | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4619 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | C | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4624 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | D | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4623 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | D | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4617 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2chl | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 2220 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2chl | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 2217 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izr | A | A | {(2z)-4-amino-2-[(4-methoxyphenyl)imino]-2,3-dihydro-1,3-thiazol-5-yl}(4-methoxyphenyl)methanone | Human | 2222 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izr | A | B | {(2z)-4-amino-2-[(4-methoxyphenyl)imino]-2,3-dihydro-1,3-thiazol-5-yl}(4-methoxyphenyl)methanone | Human | 2221 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izs | A | A | {[4-amino-2-(3-chloroanilino)-1,3-thiazol-5-yl](4-fluorophenyl)methanone | Human | 2228 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izs | A | B | {[4-amino-2-(3-chloroanilino)-1,3-thiazol-5-yl](4-fluorophenyl)methanone | Human | 2223 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izt | A | A | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 2216 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izt | A | B | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 2215 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izu | A | A | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 2218 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izu | A | B | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 2225 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 4g16 | A | | 2-[(4-{[3-(trifluoromethyl)pyridin-2-yl]oxy}phenyl)amino]-1h-benzimidazole-6-carbonitrile | Human | 2219 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 4g17 | A | | 2-[(4-tert-butylphenyl)amino]-1h-benzimidazole-6-carbonitrile | Human | 2226 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 4hgl | A | | 2-[5-methoxy-2-(quinolin-3-yl)pyrimidin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 2227 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 4hgs | A | | 2-{2-[(3,4-difluorophenoxy)methyl]-5-methoxypyridin-4-yl}-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 2224 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 6gro | A | A | 4-[5-(2-azanylpyrimidin-4-yl)-4-(4-fluorophenyl)imidazol-1-yl]cyclohexan-1-ol | Human | 10002 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 6gro | A | B | 4-[5-(2-azanylpyrimidin-4-yl)-4-(4-fluorophenyl)imidazol-1-yl]cyclohexan-1-ol | Human | 10003 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1jwh | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5485 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1jwh | B | | - | Human | 5524 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1na7 | A | | - | Human | 5533 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1pjk | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5494 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1pjk | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5410 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 2pvr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5509 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 2pvr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5505 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 2zjw | A | | 2,3,7,8-tetrahydroxychromeno[5,4,3-cde]chromene-5,10-dione | Human | 5423 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3amy | A | | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 5506 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3at2 | A | A | - | Human | 5428 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3at2 | A | B | - | Human | 5492 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3at3 | A | | (1-{6-[6-(cyclopentylamino)-1h-indazol-1-yl]pyrazin-2-yl}-1h-pyrrol-3-yl)acetic acid | Human | 5504 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3at4 | A | | [1-(6-{6-[(1-methylethyl)amino]-1h-indazol-1-yl}pyrazin-2-yl)-1h-pyrrol-3-yl]acetic acid | Human | 5413 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3axw | A | | 4-(5-amino-1,3,4-thiadiazol-2-yl)benzoic acid | Human | 5440 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3bqc | A | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5486 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3bqc | A | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5490 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3c13 | A | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5530 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3c13 | A | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5472 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3fwq | A | | - | Human | 5507 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3fwq | B | | - | Human | 5479 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3h30 | A | A | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 5496 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3h30 | A | B | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 5460 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3h30 | B | A | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 5484 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3h30 | B | B | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 5480 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3juh | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5471 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3juh | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5456 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3juh | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 5431 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3juh | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 5421 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb6 | A | A | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 5424 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb6 | A | B | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 5499 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb6 | A | C | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 5529 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb7 | A | A | naphtho[2,1-b:7,8-b']difuran-2,9-dicarboxylic acid | Human | 5448 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb7 | A | B | naphtho[2,1-b:7,8-b']difuran-2,9-dicarboxylic acid | Human | 5455 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nga | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5422 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nga | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5515 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nga | B | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5441 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nga | B | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5511 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nsz | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5512 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nsz | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5503 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owj | A | A | 9-hydroxy-5,11-dimethyl-4,6-dihydro-1h-pyrido[4,3-b]carbazol-1-one | Human | 5452 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owj | A | B | 9-hydroxy-5,11-dimethyl-4,6-dihydro-1h-pyrido[4,3-b]carbazol-1-one | Human | 5470 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owk | A | A | 7-chloro-10-methyl-11h-benzo[g]pyrido[4,3-b]indol-3-ol | Human | 5467 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owk | A | B | 7-chloro-10-methyl-11h-benzo[g]pyrido[4,3-b]indol-3-ol | Human | 5433 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owl | A | A | 11-chloro-8-methyl-7h-benzo[e]pyrido[4,3-b]indol-3-ol | Human | 5502 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owl | A | B | 11-chloro-8-methyl-7h-benzo[e]pyrido[4,3-b]indol-3-ol | Human | 5416 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe1 | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5487 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe1 | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5500 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe2 | A | A | 5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5508 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe2 | A | B | 5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5519 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q04 | A | A | - | Human | 5514 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q04 | A | B | - | Human | 5419 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9w | A | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5436 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9w | A | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5420 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9x | A | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5446 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9x | A | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5488 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9x | B | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5516 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9x | B | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5417 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9y | A | A | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5493 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9y | A | B | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5526 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9z | A | A | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5510 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9z | A | B | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5437 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9z | B | A | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5426 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9z | B | B | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5430 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3qa0 | A | A | - | Human | 5425 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3qa0 | A | B | - | Human | 5451 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3qa0 | B | A | - | Human | 5495 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3qa0 | B | B | - | Human | 5528 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3r0t | A | A | 3-(cyclopropylamino)-5-{[3-(trifluoromethyl)phenyl]amino}pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5497 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3r0t | A | B | 3-(cyclopropylamino)-5-{[3-(trifluoromethyl)phenyl]amino}pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5517 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3rps | A | | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 5463 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3rps | B | | - | Human | 5450 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u4u | A | | 3-{5-(acetylamino)-3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1h-indol-1-yl}propanoic acid | Human | 5527 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u87 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5442 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u87 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 5513 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u9c | A | | 7-hydroxy-3h-phenoxazin-3-one | Human | 5461 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u9c | B | | 7-hydroxy-3h-phenoxazin-3-one | Human | 5523 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3w8l | A | | - | Human | 5427 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3w8l | B | | - | Human | 5469 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3war | A | A | nicotinic acid | Human | 5429 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3war | A | B | nicotinic acid | Human | 5464 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3wik | A | | n-[5-(4-nitrophenyl)-1,3,4-thiadiazol-2-yl]acetamide | Human | 5459 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3wil | A | | {[(2z)-2-(3,4-dimethoxybenzylidene)-3-oxo-2,3-dihydro-1-benzofuran-6-yl]oxy}acetic acid | Human | 5468 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3wow | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5445 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4dgl | C | | - | Human | 5474 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4dgl | D | | - | Human | 5521 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4fbx | A | | - | Human | 5415 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4grb | A | | 5-(2-{[4-(dimethylcarbamoyl)phenyl]amino}-4-methoxypyrimidin-5-yl)thiophene-3-carboxylic acid | Human | 5443 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4gub | A | | n-[5-({3-cyano-7-[(1-methyl-1h-imidazol-4-yl)amino]pyrazolo[1,5-a]pyrimidin-5-yl}amino)-2-methylphenyl]acetamide | Human | 5491 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | A | A | - | Human | 5501 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | A | B | - | Human | 5522 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | B | A | - | Human | 5532 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | B | B | - | Human | 5438 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | C | A | - | Human | 5498 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | C | B | - | Human | 5476 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4kwp | A | A | 4,5,6,7-tetrabromo-1-(2-deoxy-beta-d-erythro-pentofuranosyl)-1h-benzimidazole | Human | 5465 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4kwp | A | B | 4,5,6,7-tetrabromo-1-(2-deoxy-beta-d-erythro-pentofuranosyl)-1h-benzimidazole | Human | 5482 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md7 | E | | - | Human | 5435 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md7 | F | | - | Human | 5457 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md7 | G | | - | Human | 5409 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md7 | H | | - | Human | 5481 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md8 | E | | - | Human | 5439 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md8 | F | | - | Human | 5475 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md8 | G | | - | Human | 5478 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md8 | H | | - | Human | 5518 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | E | | - | Human | 5411 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | F | | - | Human | 5473 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | G | | - | Human | 5483 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | H | | - | Human | 5466 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | K | | - | Human | 5477 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | L | | - | Human | 5414 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | M | | - | Human | 5520 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | P | | - | Human | 5434 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4nh1 | A | | phosphomethylphosphonic acid adenylate ester | Human | 5412 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4nh1 | B | | phosphomethylphosphonic acid adenylate ester | Human | 5531 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4rll | A | A | 4-[(e)-(9h-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acid | Human | 5418 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4rll | A | B | 4-[(e)-(9h-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acid | Human | 5449 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ub7 | A | | 4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acid | Human | 5462 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4uba | A | | 4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acid | Human | 5432 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4uba | B | | 4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acid | Human | 5525 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5b0x | A | | 4-[2-[(4-methoxyphenyl)carbonylamino]-1,3-thiazol-5-yl]benzoic acid | Human | 6475 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5clp | A | A | 2-(3,4-dichlorophenyl)ethanamine | Human | 6922 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5clp | A | B | 2-(3,4-dichlorophenyl)ethanamine | Human | 6920 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5clp | B | A | 2-(3,4-dichlorophenyl)ethanamine | Human | 6909 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5clp | B | B | 2-(3,4-dichlorophenyl)ethanamine | Human | 6911 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqu | A | A | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6035 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqu | A | B | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6038 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqw | A | A | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6034 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqw | A | B | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6037 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqw | B | A | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6039 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqw | B | B | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6036 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cs6 | A | A | - | Human | 6915 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cs6 | A | B | - | Human | 6901 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cs6 | B | A | - | Human | 6919 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cs6 | B | B | - | Human | 6926 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csh | A | A | adenosine-5'-triphosphate | Human | 6918 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csh | A | B | adenosine-5'-triphosphate | Human | 6925 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csh | B | A | adenosine-5'-triphosphate | Human | 6923 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csh | B | B | adenosine-5'-triphosphate | Human | 6907 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csp | A | A | 2-hydroxy-5-methylbenzoic acid | Human | 6904 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csp | A | B | 2-hydroxy-5-methylbenzoic acid | Human | 6905 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csp | A | C | 2-hydroxy-5-methylbenzoic acid | Human | 6928 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csv | A | A | 3-aminobenzoic acid | Human | 6898 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csv | A | B | 3-aminobenzoic acid | Human | 6900 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ct0 | A | A | 3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-ol | Human | 7296 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ct0 | A | B | 3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-ol | Human | 7300 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ct0 | B | A | 3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-ol | Human | 7288 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ct0 | B | B | 3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-ol | Human | 7298 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ctp | A | A | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7304 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ctp | A | B | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7289 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ctp | B | A | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7297 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ctp | B | B | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7291 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu0 | A | A | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7299 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu0 | A | B | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7293 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu0 | B | A | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7295 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu0 | B | B | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7301 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu2 | A | A | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7303 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu2 | A | B | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7302 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu2 | B | A | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7292 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu2 | B | B | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7286 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu3 | A | A | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6902 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu3 | A | B | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6903 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu3 | B | A | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6921 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu3 | B | B | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6897 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu4 | A | A | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6924 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu4 | A | B | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6895 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu4 | A | C | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6916 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu6 | A | A | adenosine-5'-triphosphate | Human | 6899 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu6 | A | B | adenosine-5'-triphosphate | Human | 6906 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvf | A | A | adenosine-5'-triphosphate | Human | 6927 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvf | A | B | adenosine-5'-triphosphate | Human | 6910 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvg | A | A | - | Human | 6913 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvg | A | B | - | Human | 6908 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvh | A | A | adenosine-5'-diphosphate | Human | 6896 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvh | A | B | adenosine-5'-diphosphate | Human | 6912 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvh | B | A | adenosine-5'-diphosphate | Human | 6914 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvh | B | B | adenosine-5'-diphosphate | Human | 6917 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cx9 | A | A | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7287 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cx9 | A | B | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7290 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cx9 | B | A | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7285 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cx9 | B | B | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7294 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8b | A | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 6408 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8b | B | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 6406 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8e | A | | ~{n}-[2-[2-azanylethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 6409 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8e | B | | ~{n}-[2-[2-azanylethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 6407 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8g | A | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]ethanamide | Human | 6405 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ku8 | A | | ~{n}-[2-[(1~{s},2~{s})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 8664 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ku8 | B | | ~{n}-[2-[(1~{s},2~{s})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 8663 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5kwh | A | A | ~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 8617 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5kwh | A | B | ~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 8619 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5kwh | B | A | ~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 8618 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5kwh | B | B | ~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 8620 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m44 | A | | 3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acid | Human | 7404 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4c | A | A | 3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acid | Human | 7402 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4c | A | B | 3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acid | Human | 7403 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4f | A | A | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7405 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4f | A | B | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7401 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4i | A | | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7400 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmf | A | A | (3-chloranyl-4-phenyl-phenyl)methyl-propyl-azanium | Human | 7682 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmf | A | B | (3-chloranyl-4-phenyl-phenyl)methyl-propyl-azanium | Human | 7666 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmf | B | A | - | Human | 7696 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmf | B | B | - | Human | 7657 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmr | A | A | ~{n}'-[(3-chloranyl-4-phenyl-phenyl)methyl]butane-1,4-diamine | Human | 7668 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmr | A | B | ~{n}'-[(3-chloranyl-4-phenyl-phenyl)methyl]butane-1,4-diamine | Human | 7659 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmr | B | A | - | Human | 7651 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmr | B | B | - | Human | 7680 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo5 | A | A | ~{n}-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propyl]methanesulfonamide | Human | 7676 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo5 | A | B | ~{n}-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propyl]methanesulfonamide | Human | 7661 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo5 | B | A | - | Human | 7689 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo5 | B | B | - | Human | 7656 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo6 | A | A | 3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoic acid | Human | 7672 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo6 | A | B | 3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoic acid | Human | 7665 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo6 | B | A | - | Human | 7664 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo6 | B | B | - | Human | 7652 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo7 | A | A | 3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanamide | Human | 7669 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo7 | A | B | 3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanamide | Human | 7697 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo7 | B | A | - | Human | 7698 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo7 | B | B | - | Human | 7685 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo8 | A | A | 3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acid | Human | 7653 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo8 | A | B | 3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acid | Human | 7673 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo8 | B | A | 3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acid | Human | 7654 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo8 | B | B | 3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acid | Human | 7688 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mod | A | A | - | Human | 7678 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mod | A | B | - | Human | 7667 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mod | B | A | - | Human | 7679 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mod | B | B | - | Human | 7694 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moe | A | A | adenosine-5'-diphosphate | Human | 7650 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moe | A | B | adenosine-5'-diphosphate | Human | 7662 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moe | B | A | adenosine-5'-diphosphate | Human | 7693 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moe | B | B | adenosine-5'-diphosphate | Human | 7687 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moh | A | A | 2-(3-methoxy-4-oxidanyl-phenyl)ethanoic acid | Human | 7658 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moh | A | B | 2-(3-methoxy-4-oxidanyl-phenyl)ethanoic acid | Human | 7681 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mot | A | A | 4-hydroxybenzamide | Human | 7660 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mot | A | B | 4-hydroxybenzamide | Human | 7691 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mov | A | A | 4'-hydroxycinnamic acid | Human | 7655 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mov | A | B | 4'-hydroxycinnamic acid | Human | 7674 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mow | A | A | 5-bromopyridine-2,3-diamine | Human | 7670 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mow | A | B | 5-bromopyridine-2,3-diamine | Human | 7684 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mow | B | A | - | Human | 7671 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mow | B | B | - | Human | 7686 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mp8 | A | A | adenosine-5'-diphosphate | Human | 7690 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mp8 | A | B | adenosine-5'-diphosphate | Human | 7649 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mp8 | B | A | adenosine-5'-diphosphate | Human | 7695 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mp8 | B | B | adenosine-5'-diphosphate | Human | 7692 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mpj | A | A | adenosine-5'-diphosphate | Human | 7677 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mpj | A | B | adenosine-5'-diphosphate | Human | 7663 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mpj | B | A | - | Human | 7675 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mpj | B | B | - | Human | 7683 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n1v | A | A | pyrazolo-pyrimidine macrocycle | Human | 7588 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n1v | A | B | pyrazolo-pyrimidine macrocycle | Human | 7589 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n1v | B | A | pyrazolo-pyrimidine macrocycle | Human | 7587 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n1v | B | B | pyrazolo-pyrimidine macrocycle | Human | 7586 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9k | A | A | 1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diol | Human | 9682 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9k | A | B | 1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diol | Human | 9695 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9l | A | A | (4~{z})-6,7-bis(chloranyl)-4-[[(4-methylphenyl)amino]methylidene]-8-oxidanyl-1,2-dihydrodibenzofuran-3-one | Human | 9652 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9l | A | B | (4~{z})-6,7-bis(chloranyl)-4-[[(4-methylphenyl)amino]methylidene]-8-oxidanyl-1,2-dihydrodibenzofuran-3-one | Human | 9621 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9n | A | A | 1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diol | Human | 9661 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9n | A | B | 1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diol | Human | 9628 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5nqc | A | A | (3e)-6,7-dichloro-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-one | Human | 8112 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5nqc | A | B | (3e)-6,7-dichloro-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-one | Human | 8111 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5omy | A | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9457 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5omy | A | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9456 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oni | A | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9455 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oni | A | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9459 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oni | B | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9458 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oni | B | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9454 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oqu | A | A | adenosine-5'-diphosphate | Human | 9615 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oqu | A | B | adenosine-5'-diphosphate | Human | 9627 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oqu | B | A | adenosine-5'-diphosphate | Human | 9623 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oqu | B | B | adenosine-5'-diphosphate | Human | 9678 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orh | A | A | - | Human | 9620 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orh | A | B | - | Human | 9671 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orh | B | A | - | Human | 9694 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orh | B | B | - | Human | 9639 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orj | A | A | adenosine-5'-diphosphate | Human | 9653 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orj | A | B | adenosine-5'-diphosphate | Human | 9624 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orj | B | A | adenosine-5'-diphosphate | Human | 9607 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orj | B | B | adenosine-5'-diphosphate | Human | 9665 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ork | A | A | adenosine-5'-diphosphate | Human | 9693 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ork | A | B | adenosine-5'-diphosphate | Human | 9655 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ork | B | A | adenosine-5'-diphosphate | Human | 9674 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ork | B | B | adenosine-5'-diphosphate | Human | 9646 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os7 | A | A | adenosine-5'-triphosphate | Human | 9644 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os7 | A | B | adenosine-5'-triphosphate | Human | 9609 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os7 | B | A | adenosine-5'-triphosphate | Human | 9626 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os7 | B | B | adenosine-5'-triphosphate | Human | 9645 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os8 | A | A | adenosine-5'-triphosphate | Human | 9608 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os8 | A | B | adenosine-5'-triphosphate | Human | 9666 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osl | A | A | adenosine-5'-diphosphate | Human | 9673 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osl | A | B | adenosine-5'-diphosphate | Human | 9629 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osp | A | A | adenosine-5'-triphosphate | Human | 10587 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osp | A | B | adenosine-5'-triphosphate | Human | 10600 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osr | A | A | adenosine-5'-triphosphate | Human | 10601 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osr | A | B | adenosine-5'-triphosphate | Human | 10594 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osu | A | A | - | Human | 10595 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osu | A | B | - | Human | 10598 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osz | A | A | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azanium | Human | 9669 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osz | A | B | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azanium | Human | 9685 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osz | A | C | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azanium | Human | 9683 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot5 | A | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9656 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot5 | A | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9676 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot5 | B | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9689 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot5 | B | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9605 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot6 | A | A | (3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-pyrrol-2-yl)ethyl]azanium | Human | 9619 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot6 | A | B | (3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-pyrrol-2-yl)ethyl]azanium | Human | 9643 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot6 | B | A | - | Human | 9613 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot6 | B | B | - | Human | 9649 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otd | A | A | [2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azanium | Human | 9697 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otd | A | B | [2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azanium | Human | 9696 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otd | B | A | [2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azanium | Human | 9690 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otd | B | B | [2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azanium | Human | 9632 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oth | A | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9612 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oth | A | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9659 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oth | B | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9625 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oth | B | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9670 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oti | A | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9672 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oti | A | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9667 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otl | A | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9681 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otl | A | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9633 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otl | B | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9660 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otl | B | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9616 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oto | A | A | 2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9648 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oto | A | B | 2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9637 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oto | B | A | 2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9688 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oto | B | B | 2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9611 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otp | A | A | 2-[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 10588 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otp | A | B | 2-[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 10586 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otp | B | A | - | Human | 10602 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otp | B | B | - | Human | 10591 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otq | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methoxy-phenyl]methyl]ethanamine | Human | 9638 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otq | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methoxy-phenyl]methyl]ethanamine | Human | 9651 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otr | A | A | adenosine-5'-triphosphate | Human | 9640 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otr | A | B | adenosine-5'-triphosphate | Human | 9634 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ots | A | A | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3,5-bis(chloranyl)-4-phenyl-phenyl]methyl]azanium | Human | 10589 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ots | A | B | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3,5-bis(chloranyl)-4-phenyl-phenyl]methyl]azanium | Human | 10599 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oty | A | A | trifluoroacetic acid | Human | 9692 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oty | A | B | trifluoroacetic acid | Human | 9680 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otz | A | A | trifluoroacetic acid | Human | 9650 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otz | A | B | trifluoroacetic acid | Human | 9618 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oue | A | A | 3-methyl-5-oxidanyl-benzoic acid | Human | 9686 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oue | A | B | 3-methyl-5-oxidanyl-benzoic acid | Human | 9614 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oue | B | A | (3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-imidazol-4-yl)ethyl]azanium | Human | 9635 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oue | B | B | (3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-imidazol-4-yl)ethyl]azanium | Human | 9631 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oul | A | A | [3-chloranyl-4-(3-fluorophenyl)phenyl]methanamine | Human | 9622 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oul | A | B | [3-chloranyl-4-(3-fluorophenyl)phenyl]methanamine | Human | 9675 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oum | A | A | ~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]-2-(1~{h}-imidazol-2-yl)ethanamine | Human | 9668 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oum | A | B | ~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]-2-(1~{h}-imidazol-2-yl)ethanamine | Human | 9677 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oum | B | A | - | Human | 9679 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oum | B | B | - | Human | 9606 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ouu | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 9610 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ouu | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 9662 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ouu | B | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 9657 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ouu | B | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 9636 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owh | A | | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10597 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owl | A | A | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10593 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owl | A | B | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10596 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owl | B | A | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10590 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owl | B | B | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10592 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oyf | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methyl-phenyl]methyl]ethanamine | Human | 9617 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oyf | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methyl-phenyl]methyl]ethanamine | Human | 9658 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5t1h | A | A | 7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 8685 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5t1h | A | B | 7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 8682 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5t1h | B | A | 7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 8683 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5t1h | B | B | 7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 8684 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn0 | A | A | - | Human | 10697 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn0 | A | B | - | Human | 10699 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn0 | A | C | - | Human | 10704 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn0 | A | D | - | Human | 10709 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn1 | A | A | - | Human | 10696 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn1 | A | B | - | Human | 10707 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn2 | A | A | - | Human | 10698 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn2 | A | B | - | Human | 10702 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn3 | A | A | - | Human | 10703 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn3 | A | B | - | Human | 10706 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn4 | A | A | - | Human | 10700 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn4 | A | B | - | Human | 10708 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn5 | A | A | - | Human | 10705 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn5 | A | B | - | Human | 10701 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6a1c | A | A | 5-bromanyl-2-methoxy-4-[(e)-(3-methylsulfanyl-5-phenyl-1,2,4-triazol-4-yl)iminomethyl]phenol | Human | 11273 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6a1c | A | B | 5-bromanyl-2-methoxy-4-[(e)-(3-methylsulfanyl-5-phenyl-1,2,4-triazol-4-yl)iminomethyl]phenol | Human | 11286 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehk | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[3,5-bis(chloranyl)-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9641 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehk | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[3,5-bis(chloranyl)-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9663 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehu | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamine | Human | 9684 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehu | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamine | Human | 9691 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehu | B | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamine | Human | 9630 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehu | B | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamine | Human | 9664 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6eii | A | A | (3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azanium | Human | 9687 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6eii | A | B | (3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azanium | Human | 9647 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6eii | B | A | (3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azanium | Human | 9654 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6eii | B | B | (3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azanium | Human | 9642 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6fvf | A | A | - | Human | 11342 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6fvf | A | B | - | Human | 11341 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6fvg | A | A | adenosine-5'-triphosphate | Human | 11340 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6fvg | A | B | adenosine-5'-triphosphate | Human | 11339 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gih | A | A | - | Human | 9941 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gih | A | B | - | Human | 9942 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gmd | A | A | adenosine-5'-triphosphate | Human | 9993 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gmd | A | B | adenosine-5'-triphosphate | Human | 9990 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gmd | B | A | adenosine-5'-triphosphate | Human | 9991 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gmd | B | B | adenosine-5'-triphosphate | Human | 9992 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hbn | A | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11287 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hbn | A | B | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11284 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hbn | B | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11270 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hbn | B | B | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11272 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hme | A | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11275 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hme | A | B | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11283 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hme | B | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11279 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hme | B | B | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11282 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hnw | A | A | coumestrol | Human | 11523 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hnw | A | B | coumestrol | Human | 11521 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hny | A | A | boldine | Human | 11520 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hny | A | B | boldine | Human | 11522 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hop | A | A | 3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acid | Human | 11661 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hop | A | B | 4-hydroxy-3-methoxybenzaldehyde | Human | 11660 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hop | A | C | (~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-one | Human | 11662 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hop | A | D | (2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enal | Human | 11666 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hoq | A | A | 3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acid | Human | 11669 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hoq | A | B | 3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acid | Human | 11665 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hor | A | A | (~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-one | Human | 11668 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hor | A | B | (~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-one | Human | 11663 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hot | A | A | (2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enal | Human | 11667 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hot | A | B | (2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enal | Human | 11670 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hou | A | A | 4-hydroxy-3-methoxybenzaldehyde | Human | 11671 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hou | A | B | 4-hydroxy-3-methoxybenzaldehyde | Human | 11664 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6jwa | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 11467 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l1z | A | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12010 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l21 | A | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12011 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l22 | A | A | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12009 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l22 | A | B | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12014 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l23 | A | A | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 13455 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l23 | A | B | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 13454 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l24 | A | A | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12013 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l24 | A | B | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12012 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q38 | A | A | benzoic acid | Human | 11271 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q38 | A | B | benzoic acid | Human | 11285 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | A | A | benzoic acid | Human | 11281 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | A | B | benzoic acid | Human | 11276 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | A | C | benzoic acid | Human | 11277 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | B | A | benzoic acid | Human | 11274 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | B | B | benzoic acid | Human | 11278 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | B | C | benzoic acid | Human | 11280 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6qy7 | A | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12122 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6qy7 | A | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12123 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6qy7 | B | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12125 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6qy7 | B | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12124 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rb1 | A | A | (~{e})-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)-~{n}-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]prop-2-enamide | Human | 12145 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rb1 | A | B | (~{e})-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)-~{n}-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]prop-2-enamide | Human | 12142 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rcb | A | | (~{e})-2-cyano-~{n}-(2-hydroxyphenyl)-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12144 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rcm | A | A | (~{e})-~{n}-(5-~{tert}-butyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12150 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rcm | A | B | (~{e})-~{n}-(5-~{tert}-butyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12143 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rfe | A | A | (~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12148 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rfe | A | B | (~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12147 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rff | A | A | (~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-nitro-4-oxidanyl-phenyl)prop-2-enamide | Human | 12146 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rff | A | B | (~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-nitro-4-oxidanyl-phenyl)prop-2-enamide | Human | 12149 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6spw | A | A | - | Human | 11961 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6spw | A | B | - | Human | 11959 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6spx | A | | - | Human | 11960 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tei | A | A | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12461 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tei | A | B | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12459 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tei | B | A | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12460 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tei | B | B | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12457 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tll | A | A | 4,5,6,7-tetrabromobenzotriazole | Human | 13093 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tll | A | B | 4,5,6,7-tetrabromobenzotriazole | Human | 13081 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tll | A | C | 4,5,6,7-tetrabromobenzotriazole | Human | 13076 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tll | A | D | 4,5,6,7-tetrabromobenzotriazole | Human | 13087 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlo | A | A | 5,6,7-tris(bromanyl)-1~{h}-benzotriazole | Human | 13092 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlo | A | B | 5,6,7-tris(bromanyl)-1~{h}-benzotriazole | Human | 13074 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlo | A | C | - | Human | 13075 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlp | A | A | 5,6-dibromobenzotriazole | Human | 13080 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlp | A | B | 5,6-dibromobenzotriazole | Human | 13078 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlr | A | A | 4,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13089 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlr | A | B | 4,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13083 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tls | A | A | 5,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13077 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tls | A | B | 5,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13082 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlu | A | A | 6,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13091 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlu | A | B | 6,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13090 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlv | A | A | 6-bromanyl-1~{h}-benzotriazole | Human | 13079 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlv | A | B | 6-bromanyl-1~{h}-benzotriazole | Human | 13084 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlw | A | A | 7-bromanyl-1~{h}-benzotriazole | Human | 13088 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlw | A | B | 7-bromanyl-1~{h}-benzotriazole | Human | 13085 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlw | A | C | 7-bromanyl-1~{h}-benzotriazole | Human | 13086 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypg | A | A | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12425 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypg | A | B | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12432 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yph | A | A | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12433 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yph | A | B | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12431 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yph | B | A | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12428 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yph | B | B | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12429 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypj | A | A | 4-[(4-phenyl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12435 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypj | A | B | 4-[(4-phenyl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12434 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypk | A | A | - | Human | 12430 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypk | A | B | - | Human | 12426 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypn | B | A | adenosine-5'-diphosphate | Human | 12427 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypn | B | B | adenosine-5'-diphosphate | Human | 12436 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yul | A | | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12458 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yum | A | | 4-[5-[2-(2-hydroxyethyloxy)ethyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]pyrazolo[1,5-a]pyrimidin-3-yl]-2-oxidanyl-benzoic acid | Human | 12462 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yzh | A | A | adenosine-5'-diphosphate | Human | 13559 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yzh | A | B | adenosine-5'-diphosphate | Human | 13560 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6z83 | A | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamide | Human | 12652 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6z83 | B | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamide | Human | 12651 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6z84 | A | | ~{n}-[1-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]ethanamide | Human | 12650 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6z84 | B | | ~{n}-[1-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]ethanamide | Human | 12649 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a49 | A | | 6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13169 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a49 | B | | 6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13168 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4b | A | A | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13167 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4b | A | B | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13165 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4b | B | A | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13172 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4b | B | B | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13166 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4c | A | A | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13170 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4c | A | B | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13174 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4c | B | A | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13173 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4c | B | B | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13171 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4q | A | A | 2-methoxyimino-5-(quinolin-6-ylmethyl)-1,3-thiazol-4-one | Human | 14238 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4q | A | B | 2-methoxyimino-5-(quinolin-6-ylmethyl)-1,3-thiazol-4-one | Human | 14239 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7at5 | A | A | ~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamide | Human | 13840 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7at5 | A | B | ~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamide | Human | 13839 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7ay9 | A | | 7-(cyclopropylamino)-5-(5-(6-oxo-1,6-dihydropyridin-3-yl)-1-(2-(piperidin-1-yl)ethyl)-1h-1,2,3-triazol-4-yl)pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 13993 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7aya | A | A | ~{n}-[2-[(1~{r},2~{r})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 13991 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7aya | A | B | ~{n}-[2-[(1~{r},2~{r})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 13992 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8h | A | A | nicotinic acid | Human | 13260 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8h | A | B | nicotinic acid | Human | 13259 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8i | A | A | - | Human | 13263 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8i | A | B | - | Human | 13261 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8i | B | A | - | Human | 13264 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8i | B | B | - | Human | 13262 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7bu4 | A | A | 4-(6-aminocarbonyl-8-oxidanylidene-9-phenyl-7h-purin-2-yl)benzoic acid | Human | 13486 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7bu4 | A | B | 4-(6-aminocarbonyl-8-oxidanylidene-9-phenyl-7h-purin-2-yl)benzoic acid | Human | 13485 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7l1x | A | A | (2~{z})-6-[[2,6-bis(chloranyl)phenyl]methylsulfonyl]-2-[[4-oxidanyl-3-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methylidene]-4~{h}-1,4-benzothiazin-3-one | Human | 13847 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7l1x | A | B | (2~{z})-6-[[2,6-bis(chloranyl)phenyl]methylsulfonyl]-2-[[4-oxidanyl-3-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methylidene]-4~{h}-1,4-benzothiazin-3-one | Human | 13848 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7psu | A | A | - | Human | 14163 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7psu | A | B | - | Human | 14164 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgb | A | A | 5,6-dibromobenzotriazole | Human | 14468 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgb | A | B | 5,6-dibromobenzotriazole | Human | 14470 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgc | A | A | 5,6-dibromobenzotriazole | Human | 14433 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgc | A | B | 5,6-dibromobenzotriazole | Human | 14434 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgd | A | A | 5,6-dibromobenzotriazole | Human | 14472 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgd | A | B | 5,6-dibromobenzotriazole | Human | 14471 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qge | A | A | 4,5,6,7-tetrabromobenzotriazole | Human | 14469 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qge | A | B | 4,5,6,7-tetrabromobenzotriazole | Human | 14467 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qux | A | A | adenosine-5'-diphosphate | Human | 14574 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qux | A | B | adenosine-5'-diphosphate | Human | 14573 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7x4h | A | A | 5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrile | Human | 14595 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7x4h | A | B | 5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrile | Human | 14596 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7z39 | A | A | 2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamide | Human | 14449 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7z39 | A | B | 2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamide | Human | 14445 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwe | A | A | 7-(1~{h}-indol-2-yl)-5-methyl-~{n}-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine | Human | 14775 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwe | A | B | 7-(1~{h}-indol-2-yl)-5-methyl-~{n}-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine | Human | 14771 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwg | A | A | (5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dione | Human | 14772 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwg | A | B | (5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dione | Human | 14774 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwg | A | C | (5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dione | Human | 14773 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy0 | A | A | adenosine-5'-diphosphate | Human | 14452 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy0 | A | B | adenosine-5'-diphosphate | Human | 14439 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy2 | A | A | adenosine-5'-triphosphate | Human | 14443 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy2 | A | B | adenosine-5'-triphosphate | Human | 14458 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy5 | A | A | - | Human | 14457 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy5 | A | B | - | Human | 14453 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy8 | A | A | - | Human | 14441 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy8 | A | B | - | Human | 14454 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyd | A | A | adenosine-5'-triphosphate | Human | 14438 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyd | A | B | adenosine-5'-triphosphate | Human | 14450 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyk | A | A | adenosine-5'-diphosphate | Human | 14547 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyk | A | B | adenosine-5'-diphosphate | Human | 14546 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyo | A | A | adenosine-5'-triphosphate | Human | 14448 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyo | A | B | adenosine-5'-triphosphate | Human | 14440 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyr | A | A | adenosine-5'-triphosphate | Human | 14444 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyr | A | B | adenosine-5'-triphosphate | Human | 14456 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8ae7 | A | A | adenosine-5'-diphosphate | Human | 14682 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8ae7 | A | B | adenosine-5'-diphosphate | Human | 14684 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aec | A | A | adenosine-5'-triphosphate | Human | 14455 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aec | A | B | adenosine-5'-triphosphate | Human | 14451 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aec | A | C | adenosine-5'-triphosphate | Human | 14446 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aek | A | A | adenosine-5'-triphosphate | Human | 14442 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aek | A | B | adenosine-5'-triphosphate | Human | 14447 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aem | A | A | adenosine-5'-triphosphate | Human | 14685 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aem | A | B | adenosine-5'-triphosphate | Human | 14683 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8bgc | A | | 5-[(phenylmethyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 14545 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c5q | A | A | 2-methylpropyl 5-fluoranyl-3-[1-[[1-[2-[[4-(2-methylpropyl)phenyl]sulfonylamino]ethyl]piperidin-4-yl]methyl]-1,2,3-triazol-4-yl]-1~{h}-indole-2-carboxylate | Human | 15177 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c5q | A | B | 2-methylpropyl 5-fluoranyl-3-[1-[[1-[2-[[4-(2-methylpropyl)phenyl]sulfonylamino]ethyl]piperidin-4-yl]methyl]-1,2,3-triazol-4-yl]-1~{h}-indole-2-carboxylate | Human | 15175 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6l | A | A | 5-azanyl-3-[(~{z})-1-cyano-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]-3~{h}-pyrazole-4-carbonitrile | Human | 15275 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6l | A | B | 5-azanyl-3-[(~{z})-1-cyano-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]-3~{h}-pyrazole-4-carbonitrile | Human | 15280 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6m | A | A | (5~{z})-5-[(3-methoxy-4-oxidanyl-phenyl)methylidene]-1,3-thiazolidine-2,4-dione | Human | 15277 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6m | A | B | (5~{z})-5-[(3-methoxy-4-oxidanyl-phenyl)methylidene]-1,3-thiazolidine-2,4-dione | Human | 15278 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6n | A | A | (2~{z},5~{z})-5-[(4-methoxy-3-oxidanyl-phenyl)methylidene]-2-phenylimino-1,3-thiazolidin-4-one | Human | 15276 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6n | A | B | (2~{z},5~{z})-5-[(4-methoxy-3-oxidanyl-phenyl)methylidene]-2-phenylimino-1,3-thiazolidin-4-one | Human | 15279 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8p05 | A | | (4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-one | Human | 14744 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8p06 | A | | 7-(cyclopropylamino)-5-[[2-(1,2,4-triazol-4-yl)pyridin-4-yl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 14813 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8p07 | A | | 7-(cyclopropylamino)-5-[[3-(1,2,4-triazol-4-yl)phenyl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 14743 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8pvo | A | | 2-[1-(1,3-benzothiazol-6-ylsulfonyl)piperidin-4-yl]-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 14976 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8pvp | A | | ~{n}-[5-[(3-chloranyl-4-phenyl-phenyl)methylamino]pentyl]isoquinoline-5-sulfonamide | Human | 14977 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8qwy | A | | 4-[6-[(2-methoxy-5-propan-2-yloxy-phenyl)amino]pyrazin-2-yl]benzoic acid | Human | 15174 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8qwz | A | | 4-[6-(6-propan-2-yloxyindol-1-yl)pyrazin-2-yl]benzoic acid | Human | 15176 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 3e3b | X | | [1-(6-{6-[(1-methylethyl)amino]-1h-indazol-1-yl}pyrazin-2-yl)-1h-pyrrol-3-yl]acetic acid | Human | 2729 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 3ofm | A | A | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 2728 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 3ofm | A | B | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 2730 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5m4u | A | A | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7390 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5m4u | A | B | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7391 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5m56 | A | | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7388 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5m56 | B | | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7389 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ooi | A | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9447 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ooi | A | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9446 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ooi | B | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9445 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ooi | B | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9444 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5y9m | A | | nicotinic acid | Human | 9908 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5y9m | X | | nicotinic acid | Human | 9909 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5yf9 | B | A | nicotinic acid | Human | 11415 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5yf9 | B | B | nicotinic acid | Human | 11416 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5yf9 | X | A | nicotinic acid | Human | 11417 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5yf9 | X | B | nicotinic acid | Human | 11414 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ywm | X | | nicotinic acid | Human | 10759 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmb | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10994 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmb | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10995 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmc | A | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 10996 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmc | A | B | - | Human | 10993 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmd | A | A | 5-[2-(diethylamino)ethyl]-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 10997 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmd | A | B | - | Human | 10992 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmd | A | C | - | Human | 10990 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmq | A | A | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 10991 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmq | A | B | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 10998 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6l20 | A | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 11993 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6l20 | D | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 11996 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6l20 | G | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 11995 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6l20 | J | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 11994 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | A | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12117 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | A | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12120 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | B | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12114 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | B | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12121 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | C | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12115 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | C | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12119 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | D | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12116 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | D | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12118 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy9 | A | A | 3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrile | Human | 11012 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy9 | A | B | 3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrile | Human | 11011 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6te2 | A | A | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12444 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6te2 | A | B | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12446 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6tew | A | A | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12443 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6tew | A | B | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12447 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6tgu | A | A | 4-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxidanyl-benzoic acid | Human | 12448 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6tgu | A | B | 4-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxidanyl-benzoic acid | Human | 12445 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a1b | A | A | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13149 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a1b | A | B | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13144 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a1z | A | A | 6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13145 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a1z | A | B | 6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13147 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a22 | A | A | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13148 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a22 | A | B | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13151 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a2h | A | A | 5,6,7-tris(bromanyl)-1~{h}-imidazo[4,5-b]pyridine | Human | 13150 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a2h | A | B | 5,6,7-tris(bromanyl)-1~{h}-imidazo[4,5-b]pyridine | Human | 13146 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7at9 | A | A | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 13832 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7at9 | A | B | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 13829 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7at9 | A | C | 2-(3,4-dichlorophenyl)ethanamine | Human | 13830 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7atv | A | A | ~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamide | Human | 13831 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7atv | A | B | ~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamide | Human | 13828 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7xyh | A | | 5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrile | Human | 14587 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8q77 | A | A | (2~{s})-2-[[(2~{s})-2-[[(2~{s})-2-[12-[[4-[[5-(4-carboxyphenyl)-1,3-thiazol-2-yl]amino]-4-oxidanylidene-butanoyl]-(2-hydroxy-2-oxoethyl)amino]dodecanoylamino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]butanedioic acid | Human | 15024 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8q77 | A | B | (2~{s})-2-[[(2~{s})-2-[[(2~{s})-2-[12-[[4-[[5-(4-carboxyphenyl)-1,3-thiazol-2-yl]amino]-4-oxidanylidene-butanoyl]-(2-hydroxy-2-oxoethyl)amino]dodecanoylamino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]butanedioic acid | Human | 15022 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8q9s | A | A | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamide | Human | 15028 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8q9s | A | B | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamide | Human | 15031 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qbu | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 15029 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qbu | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 15025 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcd | A | A | 4,5,6,7-tetrabromobenzotriazole | Human | 15023 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcd | A | B | 4,5,6,7-tetrabromobenzotriazole | Human | 15019 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcg | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15026 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcg | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15030 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcg | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 15027 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qf1 | A | A | - | Human | 15020 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qf1 | A | B | - | Human | 15021 | |
| DAPK1 | DAPK | CAMK | 1ig1 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5615 | |
| DAPK1 | DAPK | CAMK | 1jkk | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5644 | |
| DAPK1 | DAPK | CAMK | 1jkl | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5685 | |
| DAPK1 | DAPK | CAMK | 1jkl | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5619 | |
| DAPK1 | DAPK | CAMK | 1jks | A | A | - | Human | 5657 | |
| DAPK1 | DAPK | CAMK | 1jks | A | B | - | Human | 5633 | |
| DAPK1 | DAPK | CAMK | 1jkt | A | | - | Human | 5650 | |
| DAPK1 | DAPK | CAMK | 1jkt | B | | - | Human | 5663 | |
| DAPK1 | DAPK | CAMK | 1p4f | A | A | 5,6-dihydro-benzo[h]cinnolin-3-ylamine | Human | 5625 | |
| DAPK1 | DAPK | CAMK | 1p4f | A | B | 5,6-dihydro-benzo[h]cinnolin-3-ylamine | Human | 5664 | |
| DAPK1 | DAPK | CAMK | 1wvw | A | | - | Human | 5652 | |
| DAPK1 | DAPK | CAMK | 1wvx | A | | 6-(3-aminopropyl)-4,9-dimethylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 5616 | |
| DAPK1 | DAPK | CAMK | 1wvy | A | | staurosporine | Human | 5661 | |
| DAPK1 | DAPK | CAMK | 2w4j | A | A | adenosine-5'-diphosphate | Human | 5678 | |
| DAPK1 | DAPK | CAMK | 2w4j | A | B | adenosine-5'-diphosphate | Human | 5682 | |
| DAPK1 | DAPK | CAMK | 2w4k | A | A | adenosine-5'-diphosphate | Human | 5653 | |
| DAPK1 | DAPK | CAMK | 2w4k | A | B | adenosine-5'-diphosphate | Human | 5660 | |
| DAPK1 | DAPK | CAMK | 2x0g | A | A | - | Human | 5672 | |
| DAPK1 | DAPK | CAMK | 2x0g | A | B | - | Human | 5676 | |
| DAPK1 | DAPK | CAMK | 2xuu | A | | adenosine-5'-diphosphate | Human | 5627 | |
| DAPK1 | DAPK | CAMK | 2xzs | A | A | - | Human | 5618 | |
| DAPK1 | DAPK | CAMK | 2xzs | A | B | - | Human | 5642 | |
| DAPK1 | DAPK | CAMK | 2xzs | B | A | - | Human | 5658 | |
| DAPK1 | DAPK | CAMK | 2xzs | B | B | - | Human | 5671 | |
| DAPK1 | DAPK | CAMK | 2y0a | A | | - | Human | 5651 | |
| DAPK1 | DAPK | CAMK | 2y4p | A | | - | Human | 5659 | |
| DAPK1 | DAPK | CAMK | 2y4p | B | | - | Human | 5626 | |
| DAPK1 | DAPK | CAMK | 2y4p | C | | - | Human | 5688 | |
| DAPK1 | DAPK | CAMK | 2y4p | D | | - | Human | 5640 | |
| DAPK1 | DAPK | CAMK | 2yak | A | A | ruthenium octasporine 4 | Human | 7259 | |
| DAPK1 | DAPK | CAMK | 2yak | A | B | ruthenium octasporine 4 | Human | 7260 | |
| DAPK1 | DAPK | CAMK | 3dfc | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 5645 | |
| DAPK1 | DAPK | CAMK | 3dfc | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 5620 | |
| DAPK1 | DAPK | CAMK | 3dgk | A | A | - | Human | 5656 | |
| DAPK1 | DAPK | CAMK | 3dgk | A | B | - | Human | 5629 | |
| DAPK1 | DAPK | CAMK | 3eh9 | A | A | adenosine-5'-diphosphate | Human | 5621 | |
| DAPK1 | DAPK | CAMK | 3eh9 | A | B | adenosine-5'-diphosphate | Human | 5622 | |
| DAPK1 | DAPK | CAMK | 3eh9 | A | C | adenosine-5'-diphosphate | Human | 5655 | |
| DAPK1 | DAPK | CAMK | 3eha | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5636 | |
| DAPK1 | DAPK | CAMK | 3eha | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5687 | |
| DAPK1 | DAPK | CAMK | 3eha | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 5647 | |
| DAPK1 | DAPK | CAMK | 3f5g | A | A | adenosine-5'-diphosphate | Human | 5635 | |
| DAPK1 | DAPK | CAMK | 3f5g | A | B | adenosine-5'-diphosphate | Human | 5675 | |
| DAPK1 | DAPK | CAMK | 3f5u | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5677 | |
| DAPK1 | DAPK | CAMK | 3f5u | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5632 | |
| DAPK1 | DAPK | CAMK | 3f5u | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 5630 | |
| DAPK1 | DAPK | CAMK | 3gu4 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5670 | |
| DAPK1 | DAPK | CAMK | 3gu4 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5681 | |
| DAPK1 | DAPK | CAMK | 3gu5 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5680 | |
| DAPK1 | DAPK | CAMK | 3gu5 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5669 | |
| DAPK1 | DAPK | CAMK | 3gu5 | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 5662 | |
| DAPK1 | DAPK | CAMK | 3gu6 | A | A | adenosine-5'-diphosphate | Human | 5631 | |
| DAPK1 | DAPK | CAMK | 3gu6 | A | B | adenosine-5'-diphosphate | Human | 5638 | |
| DAPK1 | DAPK | CAMK | 3gu7 | A | A | adenosine-5'-diphosphate | Human | 5624 | |
| DAPK1 | DAPK | CAMK | 3gu7 | A | B | adenosine-5'-diphosphate | Human | 5665 | |
| DAPK1 | DAPK | CAMK | 3gu8 | A | A | n6-cyclopentyladenosine | Human | 5679 | |
| DAPK1 | DAPK | CAMK | 3gu8 | A | B | n6-cyclopentyladenosine | Human | 5628 | |
| DAPK1 | DAPK | CAMK | 3gub | A | A | 9-alpha-l-lyxofuranosyl-n-(2-phenylethyl)-9h-purin-6-amine | Human | 5674 | |
| DAPK1 | DAPK | CAMK | 3gub | A | B | 9-alpha-l-lyxofuranosyl-n-(2-phenylethyl)-9h-purin-6-amine | Human | 5673 | |
| DAPK1 | DAPK | CAMK | 3zxt | A | | phosphomethylphosphonic acid adenylate ester | Human | 5634 | |
| DAPK1 | DAPK | CAMK | 3zxt | B | | phosphomethylphosphonic acid adenylate ester | Human | 5666 | |
| DAPK1 | DAPK | CAMK | 3zxt | C | | phosphomethylphosphonic acid adenylate ester | Human | 5646 | |
| DAPK1 | DAPK | CAMK | 3zxt | D | | phosphomethylphosphonic acid adenylate ester | Human | 5617 | |
| DAPK1 | DAPK | CAMK | 4b4l | A | A | - | Human | 5683 | |
| DAPK1 | DAPK | CAMK | 4b4l | A | B | - | Human | 5684 | |
| DAPK1 | DAPK | CAMK | 4pf4 | A | A | - | Human | 5643 | |
| DAPK1 | DAPK | CAMK | 4pf4 | A | B | - | Human | 5648 | |
| DAPK1 | DAPK | CAMK | 4tl0 | A | | - | Human | 5641 | |
| DAPK1 | DAPK | CAMK | 4txc | A | | 4-(3-{3-[(r)-{[2-(dimethylamino)ethyl]amino}(hydroxy)methyl]phenyl}imidazo[1,2-b]pyridazin-6-yl)-2-methoxyphenol | Human | 5668 | |
| DAPK1 | DAPK | CAMK | 4uv0 | A | | - | Human | 5639 | |
| DAPK1 | DAPK | CAMK | 4yo4 | A | A | phthalazine | Human | 5686 | |
| DAPK1 | DAPK | CAMK | 4yo4 | A | B | phthalazine | Human | 5649 | |
| DAPK1 | DAPK | CAMK | 4ypd | A | A | 4-methylpyridazine | Human | 5654 | |
| DAPK1 | DAPK | CAMK | 4ypd | A | B | 4-methylpyridazine | Human | 5623 | |
| DAPK1 | DAPK | CAMK | 5aut | A | | 8-anilino-1-naphthalene sulfonate | Human | 6137 | |
| DAPK1 | DAPK | CAMK | 5auu | A | | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4h-chromen-4-one | Human | 6145 | |
| DAPK1 | DAPK | CAMK | 5auv | A | | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 6139 | |
| DAPK1 | DAPK | CAMK | 5auw | A | | 3,5,7,3',4'-pentahydroxyflavone | Human | 6144 | |
| DAPK1 | DAPK | CAMK | 5aux | A | | 3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 6136 | |
| DAPK1 | DAPK | CAMK | 5auy | A | | 2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-one | Human | 6134 | |
| DAPK1 | DAPK | CAMK | 5auz | A | | genistein | Human | 6140 | |
| DAPK1 | DAPK | CAMK | 5av0 | A | | 3-(3,4-dihydroxyphenyl)-7-hydroxy-4h-chromen-4-one | Human | 6142 | |
| DAPK1 | DAPK | CAMK | 5av1 | A | | - | Human | 6138 | |
| DAPK1 | DAPK | CAMK | 5av2 | A | | 3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 6133 | |
| DAPK1 | DAPK | CAMK | 5av3 | A | | 3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 6143 | |
| DAPK1 | DAPK | CAMK | 5av4 | A | A | genistein | Human | 6135 | |
| DAPK1 | DAPK | CAMK | 5av4 | A | B | genistein | Human | 6141 | |
| DAPK1 | DAPK | CAMK | 6aar | A | | - | Human | 11468 | |
| DAPK1 | DAPK | CAMK | 6fha | A | A | - | Human | 11289 | |
| DAPK1 | DAPK | CAMK | 6fha | A | B | - | Human | 11288 | |
| DAPK1 | DAPK | CAMK | 6fhb | A | A | - | Human | 11290 | |
| DAPK1 | DAPK | CAMK | 6fhb | A | B | - | Human | 11291 | |
| DAPK1 | DAPK | CAMK | 6in4 | A | | - | Human | 11795 | |
| DAPK1 | DAPK | CAMK | 6qmo | A | A | - | Human | 11587 | |
| DAPK1 | DAPK | CAMK | 6qmo | A | B | - | Human | 11588 | |
| DAPK1 | DAPK | CAMK | 6qn4 | A | | - | Human | 11589 | |
| DAPK1 | DAPK | CAMK | 7ccu | A | A | resveratrol | Human | 13234 | |
| DAPK1 | DAPK | CAMK | 7ccu | A | B | resveratrol | Human | 13237 | |
| DAPK1 | DAPK | CAMK | 7ccv | A | A | piceatannol | Human | 13232 | |
| DAPK1 | DAPK | CAMK | 7ccv | A | B | piceatannol | Human | 13233 | |
| DAPK1 | DAPK | CAMK | 7ccw | A | A | resveratrol | Human | 13235 | |
| DAPK1 | DAPK | CAMK | 7ccw | A | B | resveratrol | Human | 13236 | |
| DAPK1 | DAPK | CAMK | 8ie5 | A | | trans-oxyresveratrol | Human | 14749 | |
| DAPK1 | DAPK | CAMK | 8ie6 | A | | 3-[(e)-2-(4-hydroxyphenyl)ethenyl]-5-methoxy-phenol | Human | 14751 | |
| DAPK1 | DAPK | CAMK | 8ie7 | A | | pterostilbene | Human | 14752 | |
| DAPK1 | DAPK | CAMK | 8ie8 | A | | 5-[(~{e})-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]benzene-1,3-diol | Human | 14750 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2ya9 | A | A | - | Mouse | 5749 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2ya9 | A | B | - | Mouse | 5752 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2ya9 | B | A | - | Mouse | 5743 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2ya9 | B | B | - | Mouse | 5744 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2yaa | A | A | adenosine-5'-triphosphate | Mouse | 5746 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2yaa | A | B | adenosine-5'-triphosphate | Mouse | 5747 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2yaa | B | A | adenosine-5'-triphosphate | Mouse | 5751 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2yaa | B | B | adenosine-5'-triphosphate | Mouse | 5754 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2yab | A | A | adenosine monophosphate | Mouse | 5750 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2yab | A | B | adenosine monophosphate | Mouse | 5753 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2yab | B | A | adenosine monophosphate | Mouse | 5748 | |
| Dapk2 (DAPK2) | DAPK | CAMK | 2yab | B | B | adenosine monophosphate | Mouse | 5745 | |
| DAPK2 | DAPK | CAMK | 1wmk | A | | - | Human | 1124 | |
| DAPK2 | DAPK | CAMK | 1wmk | B | | - | Human | 1140 | |
| DAPK2 | DAPK | CAMK | 1wmk | C | | - | Human | 1138 | |
| DAPK2 | DAPK | CAMK | 1wmk | D | | - | Human | 1139 | |
| DAPK2 | DAPK | CAMK | 1wmk | E | | - | Human | 1117 | |
| DAPK2 | DAPK | CAMK | 1wmk | F | | - | Human | 1126 | |
| DAPK2 | DAPK | CAMK | 1wmk | G | | - | Human | 1142 | |
| DAPK2 | DAPK | CAMK | 1wmk | H | | - | Human | 1151 | |
| DAPK2 | DAPK | CAMK | 1z9x | A | | - | Human | 1144 | |
| DAPK2 | DAPK | CAMK | 1z9x | B | | - | Human | 1136 | |
| DAPK2 | DAPK | CAMK | 1z9x | C | | - | Human | 1116 | |
| DAPK2 | DAPK | CAMK | 1zws | A | | - | Human | 1121 | |
| DAPK2 | DAPK | CAMK | 1zws | B | | - | Human | 1128 | |
| DAPK2 | DAPK | CAMK | 1zws | C | | - | Human | 1134 | |
| DAPK2 | DAPK | CAMK | 1zws | D | | - | Human | 1131 | |
| DAPK2 | DAPK | CAMK | 1zws | E | | - | Human | 1130 | |
| DAPK2 | DAPK | CAMK | 1zws | F | | - | Human | 1114 | |
| DAPK2 | DAPK | CAMK | 1zws | G | | - | Human | 1150 | |
| DAPK2 | DAPK | CAMK | 1zws | H | | - | Human | 1133 | |
| DAPK2 | DAPK | CAMK | 2a27 | A | | - | Human | 1113 | |
| DAPK2 | DAPK | CAMK | 2a27 | B | | - | Human | 1129 | |
| DAPK2 | DAPK | CAMK | 2a27 | C | | - | Human | 1125 | |
| DAPK2 | DAPK | CAMK | 2a27 | D | | - | Human | 1118 | |
| DAPK2 | DAPK | CAMK | 2a27 | E | | - | Human | 1147 | |
| DAPK2 | DAPK | CAMK | 2a27 | F | | - | Human | 1127 | |
| DAPK2 | DAPK | CAMK | 2a27 | G | | - | Human | 1146 | |
| DAPK2 | DAPK | CAMK | 2a27 | H | | - | Human | 1137 | |
| DAPK2 | DAPK | CAMK | 2a2a | A | A | - | Human | 1145 | |
| DAPK2 | DAPK | CAMK | 2a2a | A | B | - | Human | 1123 | |
| DAPK2 | DAPK | CAMK | 2a2a | B | A | - | Human | 1115 | |
| DAPK2 | DAPK | CAMK | 2a2a | B | B | - | Human | 1119 | |
| DAPK2 | DAPK | CAMK | 2a2a | C | A | - | Human | 1122 | |
| DAPK2 | DAPK | CAMK | 2a2a | C | B | - | Human | 1148 | |
| DAPK2 | DAPK | CAMK | 2a2a | D | A | - | Human | 1120 | |
| DAPK2 | DAPK | CAMK | 2a2a | D | B | - | Human | 1149 | |
| DAPK2 | DAPK | CAMK | 2cke | A | | n-(2-aminoethyl)isoquinoline-5-sulfonamide | Human | 1143 | |
| DAPK2 | DAPK | CAMK | 2cke | B | | n-(2-aminoethyl)isoquinoline-5-sulfonamide | Human | 1132 | |
| DAPK2 | DAPK | CAMK | 2cke | C | | n-(2-aminoethyl)isoquinoline-5-sulfonamide | Human | 1135 | |
| DAPK2 | DAPK | CAMK | 2cke | D | | n-(2-aminoethyl)isoquinoline-5-sulfonamide | Human | 1141 | |
| DAPK2 | DAPK | CAMK | 6paw | A | | - | Human | 12442 | |
| DAPK2 | DAPK | CAMK | 6paw | B | | - | Human | 12440 | |
| DAPK2 | DAPK | CAMK | 6paw | E | | - | Human | 12439 | |
| DAPK2 | DAPK | CAMK | 6paw | F | | - | Human | 12441 | |
| DAPK3 | DAPK | CAMK | 1yrp | A | | - | Human | 384 | |
| DAPK3 | DAPK | CAMK | 1yrp | B | | - | Human | 383 | |
| DAPK3 | DAPK | CAMK | 2j90 | A | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 387 | |
| DAPK3 | DAPK | CAMK | 2j90 | A | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 382 | |
| DAPK3 | DAPK | CAMK | 2j90 | B | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 378 | |
| DAPK3 | DAPK | CAMK | 2j90 | B | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 379 | |
| DAPK3 | DAPK | CAMK | 3bhy | A | A | (4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 385 | |
| DAPK3 | DAPK | CAMK | 3bhy | A | B | (4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 381 | |
| DAPK3 | DAPK | CAMK | 3bqr | A | A | 4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acid | Human | 380 | |
| DAPK3 | DAPK | CAMK | 3bqr | A | B | 4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acid | Human | 386 | |
| DAPK3 | DAPK | CAMK | 5a6n | A | A | 5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ide | Human | 6164 | |
| DAPK3 | DAPK | CAMK | 5a6n | A | B | 5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ide | Human | 6165 | |
| DAPK3 | DAPK | CAMK | 5a6n | B | A | - | Human | 6162 | |
| DAPK3 | DAPK | CAMK | 5a6n | B | B | - | Human | 6161 | |
| DAPK3 | DAPK | CAMK | 5a6o | A | A | - | Human | 6167 | |
| DAPK3 | DAPK | CAMK | 5a6o | A | B | - | Human | 6163 | |
| DAPK3 | DAPK | CAMK | 5a6o | B | A | - | Human | 6168 | |
| DAPK3 | DAPK | CAMK | 5a6o | B | B | - | Human | 6166 | |
| DAPK3 | DAPK | CAMK | 5vja | A | A | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10351 | |
| DAPK3 | DAPK | CAMK | 5vja | A | B | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10349 | |
| DAPK3 | DAPK | CAMK | 5vja | B | A | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10346 | |
| DAPK3 | DAPK | CAMK | 5vja | B | B | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10350 | |
| DAPK3 | DAPK | CAMK | 5vja | C | A | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10345 | |
| DAPK3 | DAPK | CAMK | 5vja | C | B | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10352 | |
| DAPK3 | DAPK | CAMK | 5vja | D | A | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10348 | |
| DAPK3 | DAPK | CAMK | 5vja | D | B | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10347 | |
| DCLK1 | DCAMKL | CAMK | 5jzj | A | A | amp phosphoramidate | Human | 6984 | |
| DCLK1 | DCAMKL | CAMK | 5jzj | A | B | amp phosphoramidate | Human | 6987 | |
| DCLK1 | DCAMKL | CAMK | 5jzj | B | A | amp phosphoramidate | Human | 6985 | |
| DCLK1 | DCAMKL | CAMK | 5jzj | B | B | amp phosphoramidate | Human | 6983 | |
| DCLK1 | DCAMKL | CAMK | 5jzn | A | | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 6986 | |
| DCLK1 | DCAMKL | CAMK | 5jzn | B | | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 6982 | |
| DCLK1 | DCAMKL | CAMK | 6kyq | A | A | - | Human | 12799 | |
| DCLK1 | DCAMKL | CAMK | 6kyq | A | B | - | Human | 12798 | |
| DCLK1 | DCAMKL | CAMK | 6kyq | B | A | - | Human | 12802 | |
| DCLK1 | DCAMKL | CAMK | 6kyq | B | B | - | Human | 12801 | |
| DCLK1 | DCAMKL | CAMK | 6kyr | A | A | - | Human | 12803 | |
| DCLK1 | DCAMKL | CAMK | 6kyr | A | B | - | Human | 12800 | |
| DCLK1 | DCAMKL | CAMK | 6kyr | B | A | - | Human | 12805 | |
| DCLK1 | DCAMKL | CAMK | 6kyr | B | B | - | Human | 12804 | |
| DCLK1 | DCAMKL | CAMK | 7f3g | A | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13853 | |
| DCLK1 | DCAMKL | CAMK | 7kx6 | A | | 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 13907 | |
| DCLK1 | DCAMKL | CAMK | 7kx8 | A | | 5-ethyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 13909 | |
| DCLK1 | DCAMKL | CAMK | 7kxw | A | | 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 13910 | |
| DCLK1 | DCAMKL | CAMK | 7kxw | B | | 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 13908 | |
| DDR1 | DDR | TK | 3zos | A | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3253 | |
| DDR1 | DDR | TK | 3zos | A | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3262 | |
| DDR1 | DDR | TK | 3zos | B | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3258 | |
| DDR1 | DDR | TK | 3zos | B | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3260 | |
| DDR1 | DDR | TK | 4bkj | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 3263 | |
| DDR1 | DDR | TK | 4bkj | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 3256 | |
| DDR1 | DDR | TK | 4bkj | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 3255 | |
| DDR1 | DDR | TK | 4bkj | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 3259 | |
| DDR1 | DDR | TK | 4ckr | A | A | 4-[(4-ethylpiperazin-1-yl)methyl]-n-{4-methyl-3-[(2-oxo-2,3-dihydro-1h-indol-5-yl)oxy]phenyl}-3-(trifluoromethyl)benzamide | Human | 3257 | |
| DDR1 | DDR | TK | 4ckr | A | B | 4-[(4-ethylpiperazin-1-yl)methyl]-n-{4-methyl-3-[(2-oxo-2,3-dihydro-1h-indol-5-yl)oxy]phenyl}-3-(trifluoromethyl)benzamide | Human | 3252 | |
| DDR1 | DDR | TK | 5bvk | A | | 1-(2-chlorophenyl)-3-(pyridin-3-ylmethyl)urea | Human | 3251 | |
| DDR1 | DDR | TK | 5bvn | A | | n-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 3261 | |
| DDR1 | DDR | TK | 5bvo | A | | n-(5-{(1s)-1-[(5-fluoro-1,3-benzoxazol-2-yl)amino]ethyl}-2-methylphenyl)imidazo[1,2-a]pyridine-3-carboxamide | Human | 3250 | |
| DDR1 | DDR | TK | 5bvw | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 3254 | |
| DDR1 | DDR | TK | 5fdp | A | | (4~{s})-4-methyl-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinoline-7-carboxamide | Human | 6676 | |
| DDR1 | DDR | TK | 5fdx | A | | 3-[(4-methylpiperazin-1-yl)methyl]-~{n}-[(4~{r})-4-methyl-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinolin-7-yl]-5-(trifluoromethyl)benzamide | Human | 7131 | |
| DDR1 | DDR | TK | 5fdx | B | | 3-[(4-methylpiperazin-1-yl)methyl]-~{n}-[(4~{r})-4-methyl-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinolin-7-yl]-5-(trifluoromethyl)benzamide | Human | 7130 | |
| DDR1 | DDR | TK | 5sau | A | A | 3-[(6-aminopyridin-3-yl)ethynyl]-n-[3-(trifluoromethyl)phenyl]benzamide | Human | 14253 | |
| DDR1 | DDR | TK | 5sau | A | B | 3-[(6-aminopyridin-3-yl)ethynyl]-n-[3-(trifluoromethyl)phenyl]benzamide | Human | 14258 | |
| DDR1 | DDR | TK | 5sav | A | A | n-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamide | Human | 14265 | |
| DDR1 | DDR | TK | 5sav | A | B | n-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamide | Human | 14261 | |
| DDR1 | DDR | TK | 5saw | A | A | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 14259 | |
| DDR1 | DDR | TK | 5saw | A | B | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 14251 | |
| DDR1 | DDR | TK | 5sax | A | A | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 14262 | |
| DDR1 | DDR | TK | 5sax | A | B | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 14263 | |
| DDR1 | DDR | TK | 5say | A | | n-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamide | Human | 14256 | |
| DDR1 | DDR | TK | 5saz | A | A | 2-chloro-5-{3-chloro-4-[(2-hydroxyethyl)amino]benzamido}-n-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamide | Human | 14255 | |
| DDR1 | DDR | TK | 5saz | A | B | 2-chloro-5-{3-chloro-4-[(2-hydroxyethyl)amino]benzamido}-n-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamide | Human | 14260 | |
| DDR1 | DDR | TK | 5sb0 | A | | n-{[(1r,2s)-2-{2-[(pyridin-3-yl)oxy]ethyl}cyclohexyl]methyl}-3-(trifluoromethoxy)benzamide | Human | 14264 | |
| DDR1 | DDR | TK | 5sb1 | A | A | 4-chloro-n-[(3s,4r)-4-phenylpyrrolidin-3-yl]-3-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | 14252 | |
| DDR1 | DDR | TK | 5sb1 | A | B | 4-chloro-n-[(3s,4r)-4-phenylpyrrolidin-3-yl]-3-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | 14257 | |
| DDR1 | DDR | TK | 5sb2 | A | A | 3-chloro-n-[(1r,2s)-2-phenylcyclopropyl]-5-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | 14250 | |
| DDR1 | DDR | TK | 5sb2 | A | B | 3-chloro-n-[(1r,2s)-2-phenylcyclopropyl]-5-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | 14254 | |
| DDR1 | DDR | TK | 6brj | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 10760 | |
| DDR1 | DDR | TK | 6bsd | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 10761 | |
| DDR1 | DDR | TK | 6few | A | A | 2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamide | Human | 10738 | |
| DDR1 | DDR | TK | 6few | A | B | 2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamide | Human | 10740 | |
| DDR1 | DDR | TK | 6fex | A | A | 2-[4-bromanyl-2-oxidanylidene-1'-(1~{h}-pyrazolo[4,3-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10741 | |
| DDR1 | DDR | TK | 6fex | A | B | 2-[4-bromanyl-2-oxidanylidene-1'-(1~{h}-pyrazolo[4,3-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10744 | |
| DDR1 | DDR | TK | 6fil | A | A | 2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamide | Human | 10746 | |
| DDR1 | DDR | TK | 6fil | A | B | 2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamide | Human | 10739 | |
| DDR1 | DDR | TK | 6fin | A | A | 3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-8-(1~{h}-indazol-5-ylcarbonyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one | Human | 10743 | |
| DDR1 | DDR | TK | 6fin | A | B | 3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-8-(1~{h}-indazol-5-ylcarbonyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one | Human | 10747 | |
| DDR1 | DDR | TK | 6fio | A | A | 2-[1'-(1~{h}-indazol-5-ylcarbonyl)-4-methyl-2-oxidanylidene-spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10748 | |
| DDR1 | DDR | TK | 6fio | A | B | 2-[1'-(1~{h}-indazol-5-ylcarbonyl)-4-methyl-2-oxidanylidene-spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10749 | |
| DDR1 | DDR | TK | 6fiq | A | | 1-(1~{h}-indazol-5-ylcarbonyl)-5'-methoxy-1'-[2-oxidanylidene-2-[(2~{s})-2-(trifluoromethyl)pyrrolidin-1-yl]ethyl]spiro[piperidine-4,3'-pyrrolo[3,2-b]pyridine]-2'-one | Human | 10742 | |
| DDR1 | DDR | TK | 6gwr | A | A | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamide | Human | 10485 | |
| DDR1 | DDR | TK | 6gwr | A | B | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamide | Human | 10484 | |
| DDR1 | DDR | TK | 6gwr | B | A | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamide | Human | 10486 | |
| DDR1 | DDR | TK | 6gwr | B | B | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamide | Human | 10487 | |
| DDR1 | DDR | TK | 6hp9 | A | | (2~{r})-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-2-(pyrimidin-5-ylamino)-2,3-dihydro-1~{h}-indene-5-carboxamide | Human | 10885 | |
| DDR1 | DDR | TK | 6hp9 | B | | (2~{r})-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-2-(pyrimidin-5-ylamino)-2,3-dihydro-1~{h}-indene-5-carboxamide | Human | 10884 | |
| DDR1 | DDR | TK | 6y23 | A | | - | Human | 12741 | |
| DDR1 | DDR | TK | 6y23 | B | | - | Human | 12742 | |
| DDR1 | DDR | TK | 6y23 | C | | - | Human | 12743 | |
| DDR1 | DDR | TK | 7bcm | A | | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 13379 | |
| DDR1 | DDR | TK | 7bcm | B | | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 13381 | |
| DDR1 | DDR | TK | 7be6 | A | A | 5-amino-n-(4-(((2s)-4-cyclohexyl-1-((1-(methylsulfonyl)piperidin-3-yl)amino)-1-oxobutan-2-yl)carbamoyl)benzyl)-1-phenyl-1h-pyrazole-4-carboxamide | Human | 13378 | |
| DDR1 | DDR | TK | 7be6 | A | B | 5-amino-n-(4-(((2s)-4-cyclohexyl-1-((1-(methylsulfonyl)piperidin-3-yl)amino)-1-oxobutan-2-yl)carbamoyl)benzyl)-1-phenyl-1h-pyrazole-4-carboxamide | Human | 13380 | |
| DDR1 | DDR | TK | 7feh | A | A | n-[(5-chloranyl-2-ethylsulfonyl-phenyl)methyl]-3-piperazin-1-yl-5-(trifluoromethyloxy)benzamide | Human | 14309 | |
| DDR1 | DDR | TK | 7feh | A | B | n-[(5-chloranyl-2-ethylsulfonyl-phenyl)methyl]-3-piperazin-1-yl-5-(trifluoromethyloxy)benzamide | Human | 14308 | |
| DDR2 | DDR | TK | 6fer | A | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10729 | |
| DDR2 | DDR | TK | 6fer | B | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10736 | |
| DDR2 | DDR | TK | 6fer | C | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10731 | |
| DDR2 | DDR | TK | 6fer | D | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10730 | |
| DDR2 | DDR | TK | 6fer | E | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10726 | |
| DDR2 | DDR | TK | 6fer | F | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10732 | |
| DDR2 | DDR | TK | 6fer | G | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10734 | |
| DDR2 | DDR | TK | 6fer | H | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10727 | |
| DDR2 | DDR | TK | 6fer | I | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10735 | |
| DDR2 | DDR | TK | 6fer | J | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10728 | |
| DDR2 | DDR | TK | 6fer | K | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10725 | |
| DDR2 | DDR | TK | 6fer | L | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10733 | |
| DDR2 | DDR | TK | 7aym | A | A | n-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 13071 | |
| DDR2 | DDR | TK | 7aym | A | B | n-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 13072 | |
| DMPK (DMPK1) | DMPK | AGC | 2vd5 | A | | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 1901 | |
| DMPK (DMPK1) | DMPK | AGC | 2vd5 | B | | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 1902 | |
| DYRK1A | DYRK | CMGC | 2vx3 | A | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3776 | |
| DYRK1A | DYRK | CMGC | 2vx3 | A | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3762 | |
| DYRK1A | DYRK | CMGC | 2vx3 | B | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3766 | |
| DYRK1A | DYRK | CMGC | 2vx3 | B | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3769 | |
| DYRK1A | DYRK | CMGC | 2vx3 | C | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3740 | |
| DYRK1A | DYRK | CMGC | 2vx3 | C | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3735 | |
| DYRK1A | DYRK | CMGC | 2vx3 | D | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3786 | |
| DYRK1A | DYRK | CMGC | 2vx3 | D | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3790 | |
| DYRK1A | DYRK | CMGC | 2wo6 | A | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3758 | |
| DYRK1A | DYRK | CMGC | 2wo6 | A | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3764 | |
| DYRK1A | DYRK | CMGC | 2wo6 | B | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3749 | |
| DYRK1A | DYRK | CMGC | 2wo6 | B | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3739 | |
| DYRK1A | DYRK | CMGC | 3anq | A | | (1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one | Human | 3767 | |
| DYRK1A | DYRK | CMGC | 3anq | B | | (1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one | Human | 3745 | |
| DYRK1A | DYRK | CMGC | 3anq | C | | (1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one | Human | 3791 | |
| DYRK1A | DYRK | CMGC | 3anq | D | | (1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one | Human | 3795 | |
| DYRK1A | DYRK | CMGC | 3anr | A | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 3778 | |
| DYRK1A | DYRK | CMGC | 3anr | B | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 3729 | |
| DYRK1A | DYRK | CMGC | 3anr | C | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 3783 | |
| DYRK1A | DYRK | CMGC | 3anr | D | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 3755 | |
| DYRK1A | DYRK | CMGC | 4aze | A | | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3761 | |
| DYRK1A | DYRK | CMGC | 4aze | B | | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3768 | |
| DYRK1A | DYRK | CMGC | 4aze | C | | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3788 | |
| DYRK1A | DYRK | CMGC | 4mq1 | A | A | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3796 | |
| DYRK1A | DYRK | CMGC | 4mq1 | A | B | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3736 | |
| DYRK1A | DYRK | CMGC | 4mq1 | B | A | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3773 | |
| DYRK1A | DYRK | CMGC | 4mq1 | B | B | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3770 | |
| DYRK1A | DYRK | CMGC | 4mq1 | C | A | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3781 | |
| DYRK1A | DYRK | CMGC | 4mq1 | C | B | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3750 | |
| DYRK1A | DYRK | CMGC | 4mq1 | D | A | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3744 | |
| DYRK1A | DYRK | CMGC | 4mq1 | D | B | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3763 | |
| DYRK1A | DYRK | CMGC | 4mq2 | A | A | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3752 | |
| DYRK1A | DYRK | CMGC | 4mq2 | A | B | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3771 | |
| DYRK1A | DYRK | CMGC | 4mq2 | B | A | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3792 | |
| DYRK1A | DYRK | CMGC | 4mq2 | B | B | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3787 | |
| DYRK1A | DYRK | CMGC | 4mq2 | C | A | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3730 | |
| DYRK1A | DYRK | CMGC | 4mq2 | C | B | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3780 | |
| DYRK1A | DYRK | CMGC | 4mq2 | D | A | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3757 | |
| DYRK1A | DYRK | CMGC | 4mq2 | D | B | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3734 | |
| DYRK1A | DYRK | CMGC | 4nct | A | | pkc412 | Human | 3794 | |
| DYRK1A | DYRK | CMGC | 4nct | B | | pkc412 | Human | 3743 | |
| DYRK1A | DYRK | CMGC | 4nct | C | | pkc412 | Human | 3779 | |
| DYRK1A | DYRK | CMGC | 4nct | D | | pkc412 | Human | 3751 | |
| DYRK1A | DYRK | CMGC | 4ylj | A | A | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3782 | |
| DYRK1A | DYRK | CMGC | 4ylj | A | B | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3746 | |
| DYRK1A | DYRK | CMGC | 4ylj | B | A | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3753 | |
| DYRK1A | DYRK | CMGC | 4ylj | B | B | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3785 | |
| DYRK1A | DYRK | CMGC | 4ylj | C | A | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3777 | |
| DYRK1A | DYRK | CMGC | 4ylj | C | B | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3748 | |
| DYRK1A | DYRK | CMGC | 4ylj | D | A | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3784 | |
| DYRK1A | DYRK | CMGC | 4ylj | D | B | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3793 | |
| DYRK1A | DYRK | CMGC | 4ylk | A | A | 10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3789 | |
| DYRK1A | DYRK | CMGC | 4ylk | A | B | 10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3756 | |
| DYRK1A | DYRK | CMGC | 4yll | A | A | 10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3747 | |
| DYRK1A | DYRK | CMGC | 4yll | A | B | 10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3772 | |
| DYRK1A | DYRK | CMGC | 4yll | A | C | 10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3731 | |
| DYRK1A | DYRK | CMGC | 4yu2 | A | A | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3774 | |
| DYRK1A | DYRK | CMGC | 4yu2 | A | B | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3765 | |
| DYRK1A | DYRK | CMGC | 4yu2 | B | A | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3737 | |
| DYRK1A | DYRK | CMGC | 4yu2 | B | B | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3738 | |
| DYRK1A | DYRK | CMGC | 4yu2 | C | A | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3741 | |
| DYRK1A | DYRK | CMGC | 4yu2 | C | B | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3775 | |
| DYRK1A | DYRK | CMGC | 4yu2 | D | A | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3760 | |
| DYRK1A | DYRK | CMGC | 4yu2 | D | B | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3733 | |
| DYRK1A | DYRK | CMGC | 5a3x | A | | n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6723 | |
| DYRK1A | DYRK | CMGC | 5a3x | B | | n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6724 | |
| DYRK1A | DYRK | CMGC | 5a3x | C | | n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6722 | |
| DYRK1A | DYRK | CMGC | 5a3x | D | | n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6718 | |
| DYRK1A | DYRK | CMGC | 5a4e | A | A | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6741 | |
| DYRK1A | DYRK | CMGC | 5a4e | A | B | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6740 | |
| DYRK1A | DYRK | CMGC | 5a4e | B | A | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6713 | |
| DYRK1A | DYRK | CMGC | 5a4e | B | B | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6726 | |
| DYRK1A | DYRK | CMGC | 5a4e | C | A | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6725 | |
| DYRK1A | DYRK | CMGC | 5a4e | C | B | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6727 | |
| DYRK1A | DYRK | CMGC | 5a4e | D | A | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6714 | |
| DYRK1A | DYRK | CMGC | 5a4e | D | B | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6733 | |
| DYRK1A | DYRK | CMGC | 5a4l | A | A | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6731 | |
| DYRK1A | DYRK | CMGC | 5a4l | A | B | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6728 | |
| DYRK1A | DYRK | CMGC | 5a4l | B | A | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6719 | |
| DYRK1A | DYRK | CMGC | 5a4l | B | B | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6735 | |
| DYRK1A | DYRK | CMGC | 5a4l | C | A | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6721 | |
| DYRK1A | DYRK | CMGC | 5a4l | C | B | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6711 | |
| DYRK1A | DYRK | CMGC | 5a4l | D | A | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6739 | |
| DYRK1A | DYRK | CMGC | 5a4l | D | B | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6730 | |
| DYRK1A | DYRK | CMGC | 5a4q | A | | n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6717 | |
| DYRK1A | DYRK | CMGC | 5a4q | B | | n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6729 | |
| DYRK1A | DYRK | CMGC | 5a4q | C | | n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6738 | |
| DYRK1A | DYRK | CMGC | 5a4q | D | | n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6737 | |
| DYRK1A | DYRK | CMGC | 5a4t | A | | n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide | Human | 6732 | |
| DYRK1A | DYRK | CMGC | 5a4t | B | | n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide | Human | 6715 | |
| DYRK1A | DYRK | CMGC | 5a4t | C | | n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide | Human | 6734 | |
| DYRK1A | DYRK | CMGC | 5a4t | D | | n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide | Human | 6712 | |
| DYRK1A | DYRK | CMGC | 5a54 | A | | n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide | Human | 6736 | |
| DYRK1A | DYRK | CMGC | 5a54 | B | | n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide | Human | 6716 | |
| DYRK1A | DYRK | CMGC | 5a54 | C | | n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide | Human | 6720 | |
| DYRK1A | DYRK | CMGC | 5a54 | D | | n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide | Human | 6710 | |
| DYRK1A | DYRK | CMGC | 5aik | A | | 4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine | Human | 3732 | |
| DYRK1A | DYRK | CMGC | 5aik | B | | 4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine | Human | 3759 | |
| DYRK1A | DYRK | CMGC | 5aik | C | | 4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine | Human | 3754 | |
| DYRK1A | DYRK | CMGC | 5aik | D | | 4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine | Human | 3742 | |
| DYRK1A | DYRK | CMGC | 6a1f | A | A | 8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amine | Human | 10522 | |
| DYRK1A | DYRK | CMGC | 6a1f | A | B | 8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amine | Human | 10521 | |
| DYRK1A | DYRK | CMGC | 6a1g | A | | 5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amine | Human | 10530 | |
| DYRK1A | DYRK | CMGC | 6a1g | B | | 5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amine | Human | 10539 | |
| DYRK1A | DYRK | CMGC | 6eif | A | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10534 | |
| DYRK1A | DYRK | CMGC | 6eif | B | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10544 | |
| DYRK1A | DYRK | CMGC | 6eif | C | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10525 | |
| DYRK1A | DYRK | CMGC | 6eif | D | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10532 | |
| DYRK1A | DYRK | CMGC | 6eij | A | | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | 10518 | |
| DYRK1A | DYRK | CMGC | 6eij | B | | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | 10516 | |
| DYRK1A | DYRK | CMGC | 6eij | C | | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | 10538 | |
| DYRK1A | DYRK | CMGC | 6eij | D | | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | 10559 | |
| DYRK1A | DYRK | CMGC | 6eil | A | | [3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone | Human | 10546 | |
| DYRK1A | DYRK | CMGC | 6eil | B | | [3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone | Human | 10557 | |
| DYRK1A | DYRK | CMGC | 6eil | C | | - | Human | 10552 | |
| DYRK1A | DYRK | CMGC | 6eil | D | | [3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone | Human | 10551 | |
| DYRK1A | DYRK | CMGC | 6eip | A | | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | 10555 | |
| DYRK1A | DYRK | CMGC | 6eip | B | | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | 10517 | |
| DYRK1A | DYRK | CMGC | 6eip | C | | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | 10533 | |
| DYRK1A | DYRK | CMGC | 6eip | D | | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | 10531 | |
| DYRK1A | DYRK | CMGC | 6eiq | A | | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | 10554 | |
| DYRK1A | DYRK | CMGC | 6eiq | B | | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | 10529 | |
| DYRK1A | DYRK | CMGC | 6eiq | C | | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | 10524 | |
| DYRK1A | DYRK | CMGC | 6eiq | D | | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | 10541 | |
| DYRK1A | DYRK | CMGC | 6eir | A | | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10550 | |
| DYRK1A | DYRK | CMGC | 6eir | B | | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10558 | |
| DYRK1A | DYRK | CMGC | 6eir | C | | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10528 | |
| DYRK1A | DYRK | CMGC | 6eir | D | | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10549 | |
| DYRK1A | DYRK | CMGC | 6eis | A | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10553 | |
| DYRK1A | DYRK | CMGC | 6eis | A | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10526 | |
| DYRK1A | DYRK | CMGC | 6eis | B | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10556 | |
| DYRK1A | DYRK | CMGC | 6eis | B | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10537 | |
| DYRK1A | DYRK | CMGC | 6eis | C | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10535 | |
| DYRK1A | DYRK | CMGC | 6eis | C | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10548 | |
| DYRK1A | DYRK | CMGC | 6eis | D | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10547 | |
| DYRK1A | DYRK | CMGC | 6eis | D | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10543 | |
| DYRK1A | DYRK | CMGC | 6eiv | A | | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10540 | |
| DYRK1A | DYRK | CMGC | 6eiv | B | | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10536 | |
| DYRK1A | DYRK | CMGC | 6eiv | C | | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10542 | |
| DYRK1A | DYRK | CMGC | 6eiv | D | | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10527 | |
| DYRK1A | DYRK | CMGC | 6ej4 | A | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10520 | |
| DYRK1A | DYRK | CMGC | 6ej4 | B | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10523 | |
| DYRK1A | DYRK | CMGC | 6ej4 | C | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10519 | |
| DYRK1A | DYRK | CMGC | 6ej4 | D | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10545 | |
| DYRK1A | DYRK | CMGC | 6ln1 | A | | 1,3,5,8-tetrakis(oxidanyl)xanthen-9-one | Human | 13935 | |
| DYRK1A | DYRK | CMGC | 6qu2 | A | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12085 | |
| DYRK1A | DYRK | CMGC | 6qu2 | A | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12092 | |
| DYRK1A | DYRK | CMGC | 6qu2 | B | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12086 | |
| DYRK1A | DYRK | CMGC | 6qu2 | B | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12088 | |
| DYRK1A | DYRK | CMGC | 6qu2 | C | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12090 | |
| DYRK1A | DYRK | CMGC | 6qu2 | C | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12087 | |
| DYRK1A | DYRK | CMGC | 6qu2 | D | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12091 | |
| DYRK1A | DYRK | CMGC | 6qu2 | D | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12089 | |
| DYRK1A | DYRK | CMGC | 6s11 | A | A | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11361 | |
| DYRK1A | DYRK | CMGC | 6s11 | A | B | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11364 | |
| DYRK1A | DYRK | CMGC | 6s11 | B | A | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11378 | |
| DYRK1A | DYRK | CMGC | 6s11 | B | B | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11372 | |
| DYRK1A | DYRK | CMGC | 6s14 | A | A | ~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11418 | |
| DYRK1A | DYRK | CMGC | 6s14 | A | B | ~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11421 | |
| DYRK1A | DYRK | CMGC | 6s17 | A | A | ~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11369 | |
| DYRK1A | DYRK | CMGC | 6s17 | A | B | ~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11375 | |
| DYRK1A | DYRK | CMGC | 6s1b | A | A | ~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11359 | |
| DYRK1A | DYRK | CMGC | 6s1b | A | B | ~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11377 | |
| DYRK1A | DYRK | CMGC | 6s1h | A | A | ~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 11419 | |
| DYRK1A | DYRK | CMGC | 6s1h | A | B | ~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 11420 | |
| DYRK1A | DYRK | CMGC | 6s1i | A | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11370 | |
| DYRK1A | DYRK | CMGC | 6s1i | A | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11376 | |
| DYRK1A | DYRK | CMGC | 6s1i | B | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11371 | |
| DYRK1A | DYRK | CMGC | 6s1i | B | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11367 | |
| DYRK1A | DYRK | CMGC | 6s1i | C | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11366 | |
| DYRK1A | DYRK | CMGC | 6s1i | C | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11373 | |
| DYRK1A | DYRK | CMGC | 6s1i | D | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11362 | |
| DYRK1A | DYRK | CMGC | 6s1i | D | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11379 | |
| DYRK1A | DYRK | CMGC | 6s1j | A | A | 3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazine | Human | 11365 | |
| DYRK1A | DYRK | CMGC | 6s1j | A | B | 3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazine | Human | 11360 | |
| DYRK1A | DYRK | CMGC | 6t6a | A | A | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11857 | |
| DYRK1A | DYRK | CMGC | 6t6a | A | B | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11858 | |
| DYRK1A | DYRK | CMGC | 6t6a | B | A | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11860 | |
| DYRK1A | DYRK | CMGC | 6t6a | B | B | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11861 | |
| DYRK1A | DYRK | CMGC | 6t6a | C | A | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11863 | |
| DYRK1A | DYRK | CMGC | 6t6a | C | B | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11859 | |
| DYRK1A | DYRK | CMGC | 6t6a | D | A | - | Human | 11862 | |
| DYRK1A | DYRK | CMGC | 6t6a | D | B | - | Human | 11856 | |
| DYRK1A | DYRK | CMGC | 6uip | A | | 4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide | Human | 12027 | |
| DYRK1A | DYRK | CMGC | 6uip | B | | 4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide | Human | 12025 | |
| DYRK1A | DYRK | CMGC | 6uip | C | | 4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide | Human | 12026 | |
| DYRK1A | DYRK | CMGC | 6uwy | A | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11989 | |
| DYRK1A | DYRK | CMGC | 6uwy | A | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11987 | |
| DYRK1A | DYRK | CMGC | 6uwy | B | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11983 | |
| DYRK1A | DYRK | CMGC | 6uwy | B | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11982 | |
| DYRK1A | DYRK | CMGC | 6uwy | C | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11984 | |
| DYRK1A | DYRK | CMGC | 6uwy | C | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11985 | |
| DYRK1A | DYRK | CMGC | 6uwy | D | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11988 | |
| DYRK1A | DYRK | CMGC | 6uwy | D | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11986 | |
| DYRK1A | DYRK | CMGC | 6yf8 | A | | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | 13462 | |
| DYRK1A | DYRK | CMGC | 6yf8 | B | | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | 13461 | |
| DYRK1A | DYRK | CMGC | 6yf8 | C | | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | 13463 | |
| DYRK1A | DYRK | CMGC | 6yf8 | D | | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | 13460 | |
| DYRK1A | DYRK | CMGC | 7a4o | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13744 | |
| DYRK1A | DYRK | CMGC | 7a4r | A | A | 2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-one | Human | 13751 | |
| DYRK1A | DYRK | CMGC | 7a4r | A | B | 2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-one | Human | 13743 | |
| DYRK1A | DYRK | CMGC | 7a4s | A | | 7-chlorothieno[3,2-c]pyridin-4-amine | Human | 13749 | |
| DYRK1A | DYRK | CMGC | 7a4w | A | | 6-(4-methoxyphenyl)pyrimidine-2,4-diamine | Human | 13754 | |
| DYRK1A | DYRK | CMGC | 7a4z | A | | 3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amine | Human | 13752 | |
| DYRK1A | DYRK | CMGC | 7a51 | A | | 4-azanyl-6-bromanyl-7-methyl-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13753 | |
| DYRK1A | DYRK | CMGC | 7a52 | A | A | 3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-one | Human | 13748 | |
| DYRK1A | DYRK | CMGC | 7a52 | A | B | 3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-one | Human | 13750 | |
| DYRK1A | DYRK | CMGC | 7a53 | A | A | (3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-one | Human | 13755 | |
| DYRK1A | DYRK | CMGC | 7a53 | A | B | (3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-one | Human | 13741 | |
| DYRK1A | DYRK | CMGC | 7a55 | A | | 3-(1-methylpyrazol-4-yl)-1~{h}-pyrazole-5-carboxylic acid | Human | 13746 | |
| DYRK1A | DYRK | CMGC | 7a5b | A | | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 13756 | |
| DYRK1A | DYRK | CMGC | 7a5d | A | A | 4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13742 | |
| DYRK1A | DYRK | CMGC | 7a5d | A | B | 4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13745 | |
| DYRK1A | DYRK | CMGC | 7a5l | A | A | 4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amine | Human | 13747 | |
| DYRK1A | DYRK | CMGC | 7a5l | A | B | 4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amine | Human | 13758 | |
| DYRK1A | DYRK | CMGC | 7a5n | A | | 5-(2-azanylpyridin-4-yl)-~{n}-[[2,6-bis(fluoranyl)phenyl]methyl]-2-methyl-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 13757 | |
| DYRK1A | DYRK | CMGC | 7aj2 | A | A | 4-(4-methoxyphenyl)pyridin-2-amine | Human | 13609 | |
| DYRK1A | DYRK | CMGC | 7aj2 | A | B | 4-(4-methoxyphenyl)pyridin-2-amine | Human | 13592 | |
| DYRK1A | DYRK | CMGC | 7aj4 | A | A | 4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amine | Human | 13605 | |
| DYRK1A | DYRK | CMGC | 7aj4 | A | B | 4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amine | Human | 13588 | |
| DYRK1A | DYRK | CMGC | 7aj5 | A | A | 4-(1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13602 | |
| DYRK1A | DYRK | CMGC | 7aj5 | A | B | 4-(1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13591 | |
| DYRK1A | DYRK | CMGC | 7aj7 | A | | 4-(3-methylbenzimidazol-5-yl)pyridine-2,6-diamine | Human | 13600 | |
| DYRK1A | DYRK | CMGC | 7aj8 | A | A | 4-(1-benzofuran-5-yl)pyridin-2-amine | Human | 13587 | |
| DYRK1A | DYRK | CMGC | 7aj8 | A | B | 4-(1-benzofuran-5-yl)pyridin-2-amine | Human | 13603 | |
| DYRK1A | DYRK | CMGC | 7aja | A | A | 1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazine | Human | 13610 | |
| DYRK1A | DYRK | CMGC | 7aja | A | B | 1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazine | Human | 13597 | |
| DYRK1A | DYRK | CMGC | 7ajm | A | A | ~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamide | Human | 13590 | |
| DYRK1A | DYRK | CMGC | 7ajm | A | B | ~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamide | Human | 13598 | |
| DYRK1A | DYRK | CMGC | 7ajs | A | A | 4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13599 | |
| DYRK1A | DYRK | CMGC | 7ajs | A | B | 4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13607 | |
| DYRK1A | DYRK | CMGC | 7ajv | A | | 4-(2,3-dibutylimidazo[4,5-b]pyridin-5-yl)pyridine-2,6-diamine | Human | 13594 | |
| DYRK1A | DYRK | CMGC | 7ajw | A | A | 4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13612 | |
| DYRK1A | DYRK | CMGC | 7ajw | A | B | 4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13611 | |
| DYRK1A | DYRK | CMGC | 7ajy | A | | 4-[2-methyl-3-[(2~{r})-2-phenoxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13606 | |
| DYRK1A | DYRK | CMGC | 7ak2 | A | | 4-[2-methyl-3-(2-pyridin-2-yloxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13593 | |
| DYRK1A | DYRK | CMGC | 7aka | A | A | 4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13596 | |
| DYRK1A | DYRK | CMGC | 7aka | A | B | 4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13595 | |
| DYRK1A | DYRK | CMGC | 7akb | A | A | 4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13608 | |
| DYRK1A | DYRK | CMGC | 7akb | A | B | 4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13604 | |
| DYRK1A | DYRK | CMGC | 7ake | A | | 4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13601 | |
| DYRK1A | DYRK | CMGC | 7akl | A | | 4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13589 | |
| DYRK1A | DYRK | CMGC | 7fhs | A | A | (5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | 14160 | |
| DYRK1A | DYRK | CMGC | 7fhs | A | B | (5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | 14159 | |
| DYRK1A | DYRK | CMGC | 7fht | A | A | (5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | 14161 | |
| DYRK1A | DYRK | CMGC | 7fht | A | B | (5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | 14162 | |
| DYRK1A | DYRK | CMGC | 7o7k | A | A | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 13988 | |
| DYRK1A | DYRK | CMGC | 7o7k | A | B | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 13987 | |
| DYRK1A | DYRK | CMGC | 7z5n | A | | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 14667 | |
| DYRK1A | DYRK | CMGC | 7zh8 | A | A | 6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridine | Human | 14489 | |
| DYRK1A | DYRK | CMGC | 7zh8 | A | B | 6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridine | Human | 14488 | |
| DYRK1A | DYRK | CMGC | 8c3g | A | A | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 15155 | |
| DYRK1A | DYRK | CMGC | 8c3g | A | B | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 15153 | |
| DYRK1A | DYRK | CMGC | 8c3q | A | A | rutin | Human | 15158 | |
| DYRK1A | DYRK | CMGC | 8c3q | A | B | rutin | Human | 15154 | |
| DYRK1A | DYRK | CMGC | 8c3r | A | A | gossypin | Human | 15156 | |
| DYRK1A | DYRK | CMGC | 8c3r | A | B | gossypin | Human | 15157 | |
| DYRK1B | DYRK | CMGC | 8c2z | A | A | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 15180 | |
| DYRK1B | DYRK | CMGC | 8c2z | A | B | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 15181 | |
| DYRK2 | DYRK | CMGC | 3k2l | A | A | - | Human | 3147 | |
| DYRK2 | DYRK | CMGC | 3k2l | A | B | - | Human | 3145 | |
| DYRK2 | DYRK | CMGC | 3kvw | A | A | (2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acid | Human | 3148 | |
| DYRK2 | DYRK | CMGC | 3kvw | A | B | (2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acid | Human | 3149 | |
| DYRK2 | DYRK | CMGC | 4azf | A | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3144 | |
| DYRK2 | DYRK | CMGC | 4azf | A | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3146 | |
| DYRK2 | DYRK | CMGC | 5lxc | A | A | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7122 | |
| DYRK2 | DYRK | CMGC | 5lxc | A | B | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7129 | |
| DYRK2 | DYRK | CMGC | 5lxc | B | A | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7125 | |
| DYRK2 | DYRK | CMGC | 5lxc | B | B | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7126 | |
| DYRK2 | DYRK | CMGC | 5lxd | A | A | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7124 | |
| DYRK2 | DYRK | CMGC | 5lxd | A | B | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7128 | |
| DYRK2 | DYRK | CMGC | 5lxd | B | A | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7123 | |
| DYRK2 | DYRK | CMGC | 5lxd | B | B | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7127 | |
| DYRK2 | DYRK | CMGC | 5ztn | A | | (1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | Human | 10482 | |
| DYRK2 | DYRK | CMGC | 5ztn | B | | (1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | Human | 10483 | |
| DYRK2 | DYRK | CMGC | 6hdp | A | A | scorzodihydrostilbene a | Human | 11572 | |
| DYRK2 | DYRK | CMGC | 6hdp | A | B | scorzodihydrostilbene a | Human | 11573 | |
| DYRK2 | DYRK | CMGC | 6hdr | A | A | curcumin | Human | 11570 | |
| DYRK2 | DYRK | CMGC | 6hdr | A | B | curcumin | Human | 11571 | |
| DYRK2 | DYRK | CMGC | 6k0j | A | | 3-(2,7-dimethoxyacridin-9-yl)sulfanylpropan-1-amine | Human | 11817 | |
| DYRK2 | DYRK | CMGC | 7akf | A | A | 4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13613 | |
| DYRK2 | DYRK | CMGC | 7akf | A | B | 4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13614 | |
| DYRK2 | DYRK | CMGC | 7akh | A | | 4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13615 | |
| DYRK2 | DYRK | CMGC | 7dg4 | A | | 2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine | Human | 13967 | |
| DYRK2 | DYRK | CMGC | 7dh3 | A | | 2,7-dimethoxy-9-piperidin-4-ylsulfanyl-acridine | Human | 13978 | |
| DYRK2 | DYRK | CMGC | 7dh9 | A | | [2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridin-4-yl]methanol | Human | 13976 | |
| DYRK2 | DYRK | CMGC | 7dhc | A | | 4-[bis(fluoranyl)methyl]-2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine | Human | 13973 | |
| DYRK2 | DYRK | CMGC | 7dhh | A | | [9-(azetidin-3-ylmethylsulfanyl)-2,7-dimethoxy-acridin-4-yl]methanol | Human | 13975 | |
| DYRK2 | DYRK | CMGC | 7dhk | A | | 2-methoxy-7-phenylmethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine | Human | 13977 | |
| DYRK2 | DYRK | CMGC | 7dhn | A | | 7-methoxy-2-methylsulfanyl-9-(piperidin-4-ylmethylsulfanyl)-[1,3]thiazolo[5,4-b]quinoline | Human | 13971 | |
| DYRK2 | DYRK | CMGC | 7dho | A | | 2-methoxy-9-(piperidin-4-ylmethylsulfanyl)-7-propan-2-yloxy-acridine | Human | 13972 | |
| DYRK2 | DYRK | CMGC | 7dhv | A | | 2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine-4-carboxylic acid | Human | 13974 | |
| DYRK2 | DYRK | CMGC | 7djo | A | | [2,7-dimethoxy-9-[[(3s)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanol | Human | 13994 | |
| DYRK2 | DYRK | CMGC | 7dl6 | A | | [2,7-dimethoxy-9-[[(3r)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanol | Human | 14013 | |
| DYRK2 | DYRK | CMGC | 7ejv | A | A | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | 14180 | |
| DYRK2 | DYRK | CMGC | 7ejv | A | B | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | 14181 | |
| DYRK2 | DYRK | CMGC | 7ejv | B | A | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | 14183 | |
| DYRK2 | DYRK | CMGC | 7ejv | B | B | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | 14182 | |
| DYRK2 | DYRK | CMGC | 8hlt | A | | (6-{[(4p)-4-(1,3-benzothiazol-5-yl)-5-fluoropyrimidin-2-yl]amino}pyridin-3-yl)(piperazin-1-yl)methanone | Human | 15091 | |
| DYRK3 | DYRK | CMGC | 5y86 | A | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 9876 | |
| EGFR | EGFR | TK | 1m14 | A | | - | Human | 826 | |
| EGFR | EGFR | TK | 1m17 | A | A | [6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amine | Human | 873 | |
| EGFR | EGFR | TK | 1m17 | A | B | [6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amine | Human | 905 | |
| EGFR | EGFR | TK | 1xkk | A | | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamine | Human | 844 | |
| EGFR | EGFR | TK | 2eb2 | A | | - | Human | 787 | |
| EGFR | EGFR | TK | 2eb3 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 816 | |
| EGFR | EGFR | TK | 2gs2 | A | | - | Human | 849 | |
| EGFR | EGFR | TK | 2gs6 | A | | - | Human | 815 | |
| EGFR | EGFR | TK | 2gs7 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 842 | |
| EGFR | EGFR | TK | 2gs7 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 795 | |
| EGFR | EGFR | TK | 2itn | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 879 | |
| EGFR | EGFR | TK | 2itn | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 833 | |
| EGFR | EGFR | TK | 2ito | A | | gefitinib | Human | 783 | |
| EGFR | EGFR | TK | 2itp | A | A | 6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 880 | |
| EGFR | EGFR | TK | 2itp | A | B | 6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 871 | |
| EGFR | EGFR | TK | 2itq | A | A | 1,2,3,4-tetrahydrogen staurosporine | Human | 813 | |
| EGFR | EGFR | TK | 2itq | A | B | 1,2,3,4-tetrahydrogen staurosporine | Human | 846 | |
| EGFR | EGFR | TK | 2itt | A | A | 6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 892 | |
| EGFR | EGFR | TK | 2itt | A | B | 6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 891 | |
| EGFR | EGFR | TK | 2itu | A | A | 1,2,3,4-tetrahydrogen staurosporine | Human | 779 | |
| EGFR | EGFR | TK | 2itu | A | B | 1,2,3,4-tetrahydrogen staurosporine | Human | 859 | |
| EGFR | EGFR | TK | 2itv | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 911 | |
| EGFR | EGFR | TK | 2itv | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 834 | |
| EGFR | EGFR | TK | 2itw | A | A | 1,2,3,4-tetrahydrogen staurosporine | Human | 817 | |
| EGFR | EGFR | TK | 2itw | A | B | 1,2,3,4-tetrahydrogen staurosporine | Human | 914 | |
| EGFR | EGFR | TK | 2itx | A | | phosphoaminophosphonic acid-adenylate ester | Human | 865 | |
| EGFR | EGFR | TK | 2ity | A | | gefitinib | Human | 790 | |
| EGFR | EGFR | TK | 2itz | A | | gefitinib | Human | 789 | |
| EGFR | EGFR | TK | 2j5e | A | | - | Human | 7215 | |
| EGFR | EGFR | TK | 2j5f | A | | n-[4-(3-bromo-phenylamino)-quinazolin-6-yl]-acrylamide | Human | 862 | |
| EGFR | EGFR | TK | 2j6m | A | | 6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 900 | |
| EGFR | EGFR | TK | 2jit | A | | - | Human | 888 | |
| EGFR | EGFR | TK | 2jit | B | | - | Human | 805 | |
| EGFR | EGFR | TK | 2jiu | A | | 6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 858 | |
| EGFR | EGFR | TK | 2jiu | B | | - | Human | 895 | |
| EGFR | EGFR | TK | 2jiv | A | A | n-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamide | Human | 893 | |
| EGFR | EGFR | TK | 2jiv | A | B | n-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamide | Human | 851 | |
| EGFR | EGFR | TK | 2jiv | B | A | n-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamide | Human | 830 | |
| EGFR | EGFR | TK | 2jiv | B | B | n-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamide | Human | 812 | |
| EGFR | EGFR | TK | 2rf9 | A | | - | Human | 876 | |
| EGFR | EGFR | TK | 2rf9 | B | | - | Human | 883 | |
| EGFR | EGFR | TK | 2rfd | A | | - | Human | 875 | |
| EGFR | EGFR | TK | 2rfd | B | | - | Human | 840 | |
| EGFR | EGFR | TK | 2rfe | A | | - | Human | 836 | |
| EGFR | EGFR | TK | 2rfe | B | | - | Human | 896 | |
| EGFR | EGFR | TK | 2rfe | C | | - | Human | 907 | |
| EGFR | EGFR | TK | 2rfe | D | | - | Human | 807 | |
| EGFR | EGFR | TK | 2rgp | A | | n-[1-(3-fluorobenzyl)-1h-indazol-5-yl]-5-[(piperidin-1-ylamino)methyl]pyrimidine-4,6-diamine | Human | 6757 | |
| EGFR | EGFR | TK | 3bel | A | | 4-amino-6-{[1-(3-fluorobenzyl)-1h-indazol-5-yl]amino}pyrimidine-5-carbaldehyde o-(2-methoxyethyl)oxime | Human | 6758 | |
| EGFR | EGFR | TK | 3gop | A | A | - | Human | 853 | |
| EGFR | EGFR | TK | 3gop | A | B | - | Human | 886 | |
| EGFR | EGFR | TK | 3gt8 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 908 | |
| EGFR | EGFR | TK | 3gt8 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 847 | |
| EGFR | EGFR | TK | 3gt8 | C | | phosphoaminophosphonic acid-adenylate ester | Human | 882 | |
| EGFR | EGFR | TK | 3gt8 | D | | phosphoaminophosphonic acid-adenylate ester | Human | 860 | |
| EGFR | EGFR | TK | 3ika | A | A | n-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | Human | 802 | |
| EGFR | EGFR | TK | 3ika | A | B | n-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | Human | 855 | |
| EGFR | EGFR | TK | 3ika | B | A | - | Human | 863 | |
| EGFR | EGFR | TK | 3ika | B | B | - | Human | 868 | |
| EGFR | EGFR | TK | 3lzb | A | | n-[3-(5-{2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}imidazo[2,1-b][1,3]thiazol-6-yl)phenyl]-2-phenylacetamide | Human | 800 | |
| EGFR | EGFR | TK | 3lzb | B | | n-[3-(5-{2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}imidazo[2,1-b][1,3]thiazol-6-yl)phenyl]-2-phenylacetamide | Human | 810 | |
| EGFR | EGFR | TK | 3lzb | C | | n-[3-(5-{2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}imidazo[2,1-b][1,3]thiazol-6-yl)phenyl]-2-phenylacetamide | Human | 808 | |
| EGFR | EGFR | TK | 3lzb | D | | n-[3-(5-{2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}imidazo[2,1-b][1,3]thiazol-6-yl)phenyl]-2-phenylacetamide | Human | 820 | |
| EGFR | EGFR | TK | 3poz | A | | n-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamide | Human | 7308 | |
| EGFR | EGFR | TK | 3ug1 | A | A | - | Human | 864 | |
| EGFR | EGFR | TK | 3ug1 | A | B | - | Human | 799 | |
| EGFR | EGFR | TK | 3ug2 | A | A | gefitinib | Human | 898 | |
| EGFR | EGFR | TK | 3ug2 | A | B | gefitinib | Human | 819 | |
| EGFR | EGFR | TK | 3vjn | A | | phosphoaminophosphonic acid-adenylate ester | Human | 872 | |
| EGFR | EGFR | TK | 3vjo | A | | phosphoaminophosphonic acid-adenylate ester | Human | 777 | |
| EGFR | EGFR | TK | 3w2o | A | A | n-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamide | Human | 9119 | |
| EGFR | EGFR | TK | 3w2o | A | B | n-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamide | Human | 9118 | |
| EGFR | EGFR | TK | 3w2p | A | A | n-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-4-(dimethylamino)butanamide | Human | 829 | |
| EGFR | EGFR | TK | 3w2p | A | B | n-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-4-(dimethylamino)butanamide | Human | 838 | |
| EGFR | EGFR | TK | 3w2q | A | A | n-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamide | Human | 845 | |
| EGFR | EGFR | TK | 3w2q | A | B | n-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamide | Human | 874 | |
| EGFR | EGFR | TK | 3w2r | A | A | 1-{3-[2-chloro-4-({5-[2-(2-hydroxyethoxy)ethyl]-5h-pyrrolo[3,2-d]pyrimidin-4-yl}amino)phenoxy]phenyl}-3-cyclohexylurea | Human | 822 | |
| EGFR | EGFR | TK | 3w2r | A | B | 1-{3-[2-chloro-4-({5-[2-(2-hydroxyethoxy)ethyl]-5h-pyrrolo[3,2-d]pyrimidin-4-yl}amino)phenoxy]phenyl}-3-cyclohexylurea | Human | 885 | |
| EGFR | EGFR | TK | 3w2s | A | A | 1-{3-[2-chloro-4-({5-[2-(2-hydroxyethoxy)ethyl]-5h-pyrrolo[3,2-d]pyrimidin-4-yl}amino)phenoxy]phenyl}-3-cyclohexylurea | Human | 778 | |
| EGFR | EGFR | TK | 3w2s | A | B | 1-{3-[2-chloro-4-({5-[2-(2-hydroxyethoxy)ethyl]-5h-pyrrolo[3,2-d]pyrimidin-4-yl}amino)phenoxy]phenyl}-3-cyclohexylurea | Human | 792 | |
| EGFR | EGFR | TK | 3w32 | A | | 4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-n-[2-(methylsulfonyl)ethyl]-8,9-dihydro-7h-pyrimido[4,5-b]azepine-6-carboxamide | Human | 784 | |
| EGFR | EGFR | TK | 3w33 | A | A | 4-{[4-(1-benzothiophen-4-yloxy)-3-chlorophenyl]amino}-n-(2-hydroxyethyl)-8,9-dihydro-7h-pyrimido[4,5-b]azepine-6-carboxamide | Human | 782 | |
| EGFR | EGFR | TK | 3w33 | A | B | 4-{[4-(1-benzothiophen-4-yloxy)-3-chlorophenyl]amino}-n-(2-hydroxyethyl)-8,9-dihydro-7h-pyrimido[4,5-b]azepine-6-carboxamide | Human | 869 | |
| EGFR | EGFR | TK | 4g5j | A | A | n-{4-[(3-chloro-4-fluorophenyl)amino]-7-[(3s)-tetrahydrofuran-3-yloxy]quinazolin-6-yl}-4-(dimethylamino)butanamide | Human | 794 | |
| EGFR | EGFR | TK | 4g5j | A | B | n-{4-[(3-chloro-4-fluorophenyl)amino]-7-[(3s)-tetrahydrofuran-3-yloxy]quinazolin-6-yl}-4-(dimethylamino)butanamide | Human | 852 | |
| EGFR | EGFR | TK | 4g5p | A | | n-{4-[(3-chloro-4-fluorophenyl)amino]-7-[(3s)-tetrahydrofuran-3-yloxy]quinazolin-6-yl}-4-(dimethylamino)butanamide | Human | 809 | |
| EGFR | EGFR | TK | 4g5p | B | | - | Human | 788 | |
| EGFR | EGFR | TK | 4hjo | A | | [6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amine | Human | 835 | |
| EGFR | EGFR | TK | 4i1z | A | A | - | Human | 903 | |
| EGFR | EGFR | TK | 4i1z | A | B | - | Human | 906 | |
| EGFR | EGFR | TK | 4i20 | A | | - | Human | 850 | |
| EGFR | EGFR | TK | 4i21 | A | | - | Human | 824 | |
| EGFR | EGFR | TK | 4i21 | B | | - | Human | 776 | |
| EGFR | EGFR | TK | 4i22 | A | | gefitinib | Human | 823 | |
| EGFR | EGFR | TK | 4i23 | A | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 870 | |
| EGFR | EGFR | TK | 4i24 | A | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 831 | |
| EGFR | EGFR | TK | 4i24 | B | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 910 | |
| EGFR | EGFR | TK | 4jq7 | A | | (2s)-2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]-2-phenylethanol | Human | 801 | |
| EGFR | EGFR | TK | 4jq8 | A | | n-[3-(4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-6-phenylfuro[2,3-d]pyrimidin-5-yl)phenyl]-n~3~,n~3~-dimethyl-beta-alaninamide | Human | 821 | |
| EGFR | EGFR | TK | 4jr3 | A | | n-[3-(4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-6-phenylfuro[2,3-d]pyrimidin-5-yl)phenyl]acetamide | Human | 915 | |
| EGFR | EGFR | TK | 4jrv | A | | 4-(dimethylamino)-n-[3-(4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-6-phenylfuro[2,3-d]pyrimidin-5-yl)phenyl]butanamide | Human | 857 | |
| EGFR | EGFR | TK | 4li5 | A | A | n-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-4-methoxyphenyl)propanamide | Human | 841 | |
| EGFR | EGFR | TK | 4li5 | A | B | n-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-4-methoxyphenyl)propanamide | Human | 797 | |
| EGFR | EGFR | TK | 4ll0 | A | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 804 | |
| EGFR | EGFR | TK | 4ll0 | B | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 796 | |
| EGFR | EGFR | TK | 4lqm | A | | n-[4-(3-bromo-phenylamino)-quinazolin-6-yl]-acrylamide | Human | 785 | |
| EGFR | EGFR | TK | 4lrm | A | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 901 | |
| EGFR | EGFR | TK | 4lrm | B | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 867 | |
| EGFR | EGFR | TK | 4lrm | C | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 781 | |
| EGFR | EGFR | TK | 4lrm | D | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 786 | |
| EGFR | EGFR | TK | 4lrm | E | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 825 | |
| EGFR | EGFR | TK | 4r3p | A | | - | Human | 827 | |
| EGFR | EGFR | TK | 4r3r | A | | - | Human | 887 | |
| EGFR | EGFR | TK | 4r5s | A | | n-[4-({[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino}methyl)phenyl]propanamide | Human | 775 | |
| EGFR | EGFR | TK | 4riw | B | | adenosine-5'-diphosphate | Human | 877 | |
| EGFR | EGFR | TK | 4riw | D | | adenosine-5'-diphosphate | Human | 848 | |
| EGFR | EGFR | TK | 4rix | B | | adenosine-5'-diphosphate | Human | 811 | |
| EGFR | EGFR | TK | 4rix | D | | adenosine-5'-diphosphate | Human | 909 | |
| EGFR | EGFR | TK | 4riy | B | | adenosine-5'-diphosphate | Human | 806 | |
| EGFR | EGFR | TK | 4riy | D | | adenosine-5'-diphosphate | Human | 856 | |
| EGFR | EGFR | TK | 4rj4 | A | | n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1-(propan-2-yl)-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | 866 | |
| EGFR | EGFR | TK | 4rj5 | A | | n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | 912 | |
| EGFR | EGFR | TK | 4rj6 | A | | n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-2-(1h-pyrazol-4-yl)-3h-imidazo[4,5-c]pyridin-6-amine | Human | 832 | |
| EGFR | EGFR | TK | 4rj7 | A | A | 2,6-dichloro-n-{2-[(2-{[(2s)-1-hydroxypropan-2-yl]amino}-6-methylpyrimidin-4-yl)amino]pyridin-4-yl}benzamide | Human | 793 | |
| EGFR | EGFR | TK | 4rj7 | A | B | 2,6-dichloro-n-{2-[(2-{[(2s)-1-hydroxypropan-2-yl]amino}-6-methylpyrimidin-4-yl)amino]pyridin-4-yl}benzamide | Human | 828 | |
| EGFR | EGFR | TK | 4rj8 | A | | 1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | 899 | |
| EGFR | EGFR | TK | 4tks | A | | - | Human | 897 | |
| EGFR | EGFR | TK | 4wd5 | A | | n-{2-methyl-5-[2-oxo-9-(1h-pyrazol-4-yl)benzo[h][1,6]naphthyridin-1(2h)-yl]phenyl}propanamide | Human | 6594 | |
| EGFR | EGFR | TK | 4wd5 | B | | - | Human | 6593 | |
| EGFR | EGFR | TK | 4wkq | A | A | gefitinib | Human | 889 | |
| EGFR | EGFR | TK | 4wkq | A | B | gefitinib | Human | 837 | |
| EGFR | EGFR | TK | 4wrg | A | A | - | Human | 854 | |
| EGFR | EGFR | TK | 4wrg | A | B | - | Human | 814 | |
| EGFR | EGFR | TK | 4zau | A | | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | 6221 | |
| EGFR | EGFR | TK | 4zjv | A | A | - | Human | 798 | |
| EGFR | EGFR | TK | 4zjv | A | B | - | Human | 843 | |
| EGFR | EGFR | TK | 4zjv | B | A | - | Human | 904 | |
| EGFR | EGFR | TK | 4zjv | B | B | - | Human | 780 | |
| EGFR | EGFR | TK | 4zse | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 6696 | |
| EGFR | EGFR | TK | 4zse | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 6697 | |
| EGFR | EGFR | TK | 4zse | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 6695 | |
| EGFR | EGFR | TK | 4zse | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 6699 | |
| EGFR | EGFR | TK | 4zse | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 6693 | |
| EGFR | EGFR | TK | 4zse | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 6698 | |
| EGFR | EGFR | TK | 4zse | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 6694 | |
| EGFR | EGFR | TK | 4zse | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 6700 | |
| EGFR | EGFR | TK | 5c8k | A | | 1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-imidazo[4,5-c]pyridin-6-amine | Human | 6201 | |
| EGFR | EGFR | TK | 5c8m | A | | 2-methyl-n-{2-[4-(methylsulfonyl)piperidin-1-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amine | Human | 6202 | |
| EGFR | EGFR | TK | 5c8n | A | | n-{2-[4-(2-aminoethyl)-4-methoxypiperidin-1-yl]pyrimidin-4-yl}-2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amine | Human | 6199 | |
| EGFR | EGFR | TK | 5cal | A | | 2,2-dimethyl-3-[(4-{[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]amino}pyrimidin-2-yl)amino]propanamide | Human | 6195 | |
| EGFR | EGFR | TK | 5can | A | | (3r)-3-methyl-1-(4-{[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]amino}pyrimidin-2-yl)pyrrolidine-3-carboxamide | Human | 6203 | |
| EGFR | EGFR | TK | 5cao | A | | n~2~-[2-methyl-2-(methylsulfonyl)propyl]-n~4~-[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]pyrimidine-2,4-diamine | Human | 6206 | |
| EGFR | EGFR | TK | 5cap | A | A | 2-methyl-n-[2-(2-methyl-2-methylsulfonyl-propoxy)pyrimidin-4-yl]-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amine | Human | 6200 | |
| EGFR | EGFR | TK | 5cap | A | B | 2-methyl-n-[2-(2-methyl-2-methylsulfonyl-propoxy)pyrimidin-4-yl]-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amine | Human | 6198 | |
| EGFR | EGFR | TK | 5caq | A | | n-[2-[(3r,4s)-3-fluoranyl-4-methoxy-piperidin-1-yl]pyrimidin-4-yl]-2-methyl-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amine | Human | 6204 | |
| EGFR | EGFR | TK | 5cas | A | | (1r)-1-{6-({2-[(3r,4s)-3-fluoro-4-methoxypiperidin-1-yl]pyrimidin-4-yl}amino)-1-[(2s)-1,1,1-trifluoropropan-2-yl]-1h-imidazo[4,5-c]pyridin-2-yl}ethanol | Human | 6205 | |
| EGFR | EGFR | TK | 5cau | A | | (1r)-1-{6-({2-[(3s,4r)-3-fluoro-4-methoxypiperidin-1-yl]pyrimidin-4-yl}amino)-1-[(2s)-1,1,1-trifluoropropan-2-yl]-1h-imidazo[4,5-c]pyridin-2-yl}ethanol | Human | 6196 | |
| EGFR | EGFR | TK | 5cav | A | | (1r)-1-{6-({2-[(3r,4s)-3-fluoro-4-methoxypiperidin-1-yl]pyrimidin-4-yl}amino)-1-[(2s)-1,1,1-trifluoropropan-2-yl]-1h-imidazo[4,5-c]pyridin-2-yl}ethanol | Human | 6197 | |
| EGFR | EGFR | TK | 5cnn | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 791 | |
| EGFR | EGFR | TK | 5cnn | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 902 | |
| EGFR | EGFR | TK | 5cnn | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 839 | |
| EGFR | EGFR | TK | 5cnn | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 803 | |
| EGFR | EGFR | TK | 5cno | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 884 | |
| EGFR | EGFR | TK | 5cno | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 894 | |
| EGFR | EGFR | TK | 5cno | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 878 | |
| EGFR | EGFR | TK | 5cno | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 861 | |
| EGFR | EGFR | TK | 5czh | A | | - | Human | 6111 | |
| EGFR | EGFR | TK | 5czi | A | | - | Human | 6110 | |
| EGFR | EGFR | TK | 5d41 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 6665 | |
| EGFR | EGFR | TK | 5d41 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 6667 | |
| EGFR | EGFR | TK | 5d41 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 6666 | |
| EGFR | EGFR | TK | 5d41 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 6664 | |
| EGFR | EGFR | TK | 5edp | A | | - | Human | 6252 | |
| EGFR | EGFR | TK | 5edq | A | | ~{n}-(7-chloranyl-1~{h}-indazol-3-yl)-7,7-dimethyl-2-(1~{h}-pyrazol-4-yl)-5~{h}-furo[3,4-d]pyrimidin-4-amine | Human | 6253 | |
| EGFR | EGFR | TK | 5edr | A | A | ~{n}-(1~{h}-indazol-3-yl)-7,7-dimethyl-2-(2-methylpyrazol-3-yl)-5~{h}-furo[3,4-d]pyrimidin-4-amine | Human | 6254 | |
| EGFR | EGFR | TK | 5edr | A | B | ~{n}-(1~{h}-indazol-3-yl)-7,7-dimethyl-2-(2-methylpyrazol-3-yl)-5~{h}-furo[3,4-d]pyrimidin-4-amine | Human | 6255 | |
| EGFR | EGFR | TK | 5em5 | A | | 4-[2-(4-chlorophenyl)ethylamino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamide | Human | 6307 | |
| EGFR | EGFR | TK | 5em6 | A | | 4-[(2-azanylpyrimidin-4-yl)amino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamide | Human | 6305 | |
| EGFR | EGFR | TK | 5em7 | A | A | 4-[(2-methoxyphenyl)amino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamide | Human | 6304 | |
| EGFR | EGFR | TK | 5em7 | A | B | 4-[(2-methoxyphenyl)amino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamide | Human | 6303 | |
| EGFR | EGFR | TK | 5em8 | A | | 4-[(2-methoxyphenyl)amino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamide | Human | 6306 | |
| EGFR | EGFR | TK | 5fed | A | | ~{n}-[7-methyl-1-[(3~{r})-1-propanoylazepan-3-yl]benzimidazol-2-yl]-3-(trifluoromethyl)benzamide | Human | 6882 | |
| EGFR | EGFR | TK | 5fee | A | | ~{n}-[7-methyl-1-[(3~{r})-1-propanoylazepan-3-yl]benzimidazol-2-yl]-3-(trifluoromethyl)benzamide | Human | 6881 | |
| EGFR | EGFR | TK | 5feq | A | | ~{n}-[1-[(3~{r})-1-[4-(dimethylamino)but-2-enoyl]azepan-3-yl]-7-methyl-benzimidazol-2-yl]-2-methyl-pyridine-4-carboxamide | Human | 6883 | |
| EGFR | EGFR | TK | 5gmp | A | A | n-[3-[2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-5-methyl-7-oxidanylidene-pyrido[2,3-d]pyrimidin-8-yl]phenyl]prop-2-enamide | Human | 8167 | |
| EGFR | EGFR | TK | 5gmp | A | B | n-[3-[2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-5-methyl-7-oxidanylidene-pyrido[2,3-d]pyrimidin-8-yl]phenyl]prop-2-enamide | Human | 8168 | |
| EGFR | EGFR | TK | 5gnk | A | A | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(1-methylimidazol-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 7525 | |
| EGFR | EGFR | TK | 5gnk | A | B | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(1-methylimidazol-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 7524 | |
| EGFR | EGFR | TK | 5gty | A | A | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8363 | |
| EGFR | EGFR | TK | 5gty | A | B | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8352 | |
| EGFR | EGFR | TK | 5gty | B | A | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8360 | |
| EGFR | EGFR | TK | 5gty | B | B | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8367 | |
| EGFR | EGFR | TK | 5gty | C | A | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8366 | |
| EGFR | EGFR | TK | 5gty | C | B | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8358 | |
| EGFR | EGFR | TK | 5gty | D | A | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8356 | |
| EGFR | EGFR | TK | 5gty | D | B | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8368 | |
| EGFR | EGFR | TK | 5gty | E | A | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8359 | |
| EGFR | EGFR | TK | 5gty | E | B | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8353 | |
| EGFR | EGFR | TK | 5gty | F | A | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8354 | |
| EGFR | EGFR | TK | 5gty | F | B | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8364 | |
| EGFR | EGFR | TK | 5gty | G | A | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8355 | |
| EGFR | EGFR | TK | 5gty | G | B | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8369 | |
| EGFR | EGFR | TK | 5gty | H | A | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8362 | |
| EGFR | EGFR | TK | 5gty | H | B | 1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-one | Human | 8357 | |
| EGFR | EGFR | TK | 5gtz | A | A | n-[5-[[5-chloranyl-4-[(2-propan-2-ylsulfonylphenyl)amino]pyrimidin-2-yl]amino]-2-(4-ethylpiperazin-1-yl)-4-methoxy-phenyl]prop-2-enamide | Human | 8365 | |
| EGFR | EGFR | TK | 5gtz | A | B | n-[5-[[5-chloranyl-4-[(2-propan-2-ylsulfonylphenyl)amino]pyrimidin-2-yl]amino]-2-(4-ethylpiperazin-1-yl)-4-methoxy-phenyl]prop-2-enamide | Human | 8361 | |
| EGFR | EGFR | TK | 5hcx | A | | ~{n}-[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]-2-methyl-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amine | Human | 7040 | |
| EGFR | EGFR | TK | 5hcy | A | | 6-[[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]amino]-~{n}-(oxan-4-yl)-1-propan-2-yl-pyrrolo[3,2-c]pyridine-3-carboxamide | Human | 7039 | |
| EGFR | EGFR | TK | 5hcz | A | | 2-[1-[1-[(2~{s})-butan-2-yl]-6-[[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]amino]pyrazolo[4,3-c]pyridin-3-yl]azetidin-3-yl]propan-2-ol | Human | 7041 | |
| EGFR | EGFR | TK | 5hg5 | A | A | n-{3-[(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy]phenyl}propanamide | Human | 6375 | |
| EGFR | EGFR | TK | 5hg5 | A | B | n-{3-[(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy]phenyl}propanamide | Human | 6376 | |
| EGFR | EGFR | TK | 5hg7 | A | | 1-{(3r,4r)-3-[({5-chloro-2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-methoxypyrrolidin-1-yl}propan-1-one | Human | 6367 | |
| EGFR | EGFR | TK | 5hg8 | A | A | n-[3-({2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)phenyl]propanamide | Human | 6380 | |
| EGFR | EGFR | TK | 5hg8 | A | B | n-[3-({2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)phenyl]propanamide | Human | 6378 | |
| EGFR | EGFR | TK | 5hg9 | A | A | 1-[(3r,4r)-3-[({2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-(trifluoromethyl)pyrrolidin-1-yl]propan-1-one | Human | 6379 | |
| EGFR | EGFR | TK | 5hg9 | A | B | 1-[(3r,4r)-3-[({2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-(trifluoromethyl)pyrrolidin-1-yl]propan-1-one | Human | 6377 | |
| EGFR | EGFR | TK | 5hib | A | | n-tert-butyl-5-{[(1-methyl-1h-pyrazol-5-yl)sulfonyl]amino}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 6490 | |
| EGFR | EGFR | TK | 5hic | A | | n-{2-[1-(cyclopropylsulfonyl)-1h-pyrazol-4-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amine | Human | 6491 | |
| EGFR | EGFR | TK | 5j9y | A | A | (r)-1-(3-(4-amino-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one | Human | 6946 | |
| EGFR | EGFR | TK | 5j9y | A | B | (r)-1-(3-(4-amino-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one | Human | 6945 | |
| EGFR | EGFR | TK | 5j9z | A | | (r)-1-(3-(4-amino-3-(1-methyl-1h-indol-3-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one | Human | 6947 | |
| EGFR | EGFR | TK | 5jeb | A | | 3-(furan-2-yl)-n-[5-(furan-2-yl)-2-methoxyphenyl]-1h-pyrazolo[3,4-d]pyrimidin-4-amine
| Human | 7038 | |
| EGFR | EGFR | TK | 5u8l | A | A | 4-[(4-{4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-6-[(prop-2-yn-1-yl)carbamoyl]pyrimidin-2-yl}piperazin-1-yl)methyl]benzene-1-sulfonyl fluoride | Human | 7387 | |
| EGFR | EGFR | TK | 5u8l | A | B | 4-[(4-{4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-6-[(prop-2-yn-1-yl)carbamoyl]pyrimidin-2-yl}piperazin-1-yl)methyl]benzene-1-sulfonyl fluoride | Human | 7386 | |
| EGFR | EGFR | TK | 5ug8 | A | A | n-[(3r,4r)-4-fluoro-1-{6-[(1-methyl-1h-pyrazol-4-yl)amino]-9-(propan-2-yl)-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 7519 | |
| EGFR | EGFR | TK | 5ug8 | A | B | n-[(3r,4r)-4-fluoro-1-{6-[(1-methyl-1h-pyrazol-4-yl)amino]-9-(propan-2-yl)-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 7514 | |
| EGFR | EGFR | TK | 5ug9 | A | A | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-(propan-2-yl)-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 7512 | |
| EGFR | EGFR | TK | 5ug9 | A | B | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-(propan-2-yl)-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 7513 | |
| EGFR | EGFR | TK | 5uga | A | A | 4-(4-{[2-{[(3s)-1-acetylpyrrolidin-3-yl]amino}-9-(propan-2-yl)-9h-purin-6-yl]amino}phenyl)-1-methylpiperazin-1-ium | Human | 7517 | |
| EGFR | EGFR | TK | 5uga | A | B | 4-(4-{[2-{[(3s)-1-acetylpyrrolidin-3-yl]amino}-9-(propan-2-yl)-9h-purin-6-yl]amino}phenyl)-1-methylpiperazin-1-ium | Human | 7511 | |
| EGFR | EGFR | TK | 5ugb | A | | 4-(4-{[2-{[(3s)-1-acetylpyrrolidin-3-yl]amino}-9-(propan-2-yl)-9h-purin-6-yl]amino}phenyl)-1-methylpiperazin-1-ium | Human | 7515 | |
| EGFR | EGFR | TK | 5ugc | A | A | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 7516 | |
| EGFR | EGFR | TK | 5ugc | A | B | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 7518 | |
| EGFR | EGFR | TK | 5uwd | A | | n-(3-{[2-{[4-(4-acetylpiperazin-1-yl)-2-methoxyphenyl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]amino}phenyl)propanamide | Human | 8568 | |
| EGFR | EGFR | TK | 5x26 | A | | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9536 | |
| EGFR | EGFR | TK | 5x27 | A | | 9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9534 | |
| EGFR | EGFR | TK | 5x28 | A | | 9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9538 | |
| EGFR | EGFR | TK | 5x2a | A | A | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9545 | |
| EGFR | EGFR | TK | 5x2a | A | B | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9530 | |
| EGFR | EGFR | TK | 5x2a | A | C | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9539 | |
| EGFR | EGFR | TK | 5x2a | B | A | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9526 | |
| EGFR | EGFR | TK | 5x2a | B | B | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9548 | |
| EGFR | EGFR | TK | 5x2a | B | C | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9543 | |
| EGFR | EGFR | TK | 5x2a | C | A | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9537 | |
| EGFR | EGFR | TK | 5x2a | C | B | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9531 | |
| EGFR | EGFR | TK | 5x2a | C | C | n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamine | Human | 9547 | |
| EGFR | EGFR | TK | 5x2a | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 9529 | |
| EGFR | EGFR | TK | 5x2a | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 9532 | |
| EGFR | EGFR | TK | 5x2a | D | C | phosphoaminophosphonic acid-adenylate ester | Human | 9533 | |
| EGFR | EGFR | TK | 5x2c | A | A | 9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9572 | |
| EGFR | EGFR | TK | 5x2c | A | B | 9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9567 | |
| EGFR | EGFR | TK | 5x2c | A | C | 9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9566 | |
| EGFR | EGFR | TK | 5x2c | B | A | 9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9569 | |
| EGFR | EGFR | TK | 5x2c | B | B | 9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9571 | |
| EGFR | EGFR | TK | 5x2c | B | C | 9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9570 | |
| EGFR | EGFR | TK | 5x2f | A | A | 9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9540 | |
| EGFR | EGFR | TK | 5x2f | A | B | 9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9535 | |
| EGFR | EGFR | TK | 5x2f | B | A | 9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9546 | |
| EGFR | EGFR | TK | 5x2f | B | B | 9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9541 | |
| EGFR | EGFR | TK | 5x2f | C | A | 9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9527 | |
| EGFR | EGFR | TK | 5x2f | C | B | 9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9542 | |
| EGFR | EGFR | TK | 5x2f | D | A | 9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9544 | |
| EGFR | EGFR | TK | 5x2f | D | B | 9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamine | Human | 9528 | |
| EGFR | EGFR | TK | 5x2k | A | | n-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | Human | 9568 | |
| EGFR | EGFR | TK | 5xdk | A | | n-[3-[[2-[[4-(4-ethanoylpiperazin-1-yl)-2-methoxy-phenyl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]prop-2-enamide | Human | 9065 | |
| EGFR | EGFR | TK | 5xdl | A | | n-[3-[[2-[[4-(4-ethanoylpiperazin-1-yl)-2-methoxy-phenyl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]prop-2-enamide | Human | 9066 | |
| EGFR | EGFR | TK | 5xgm | A | | 12-(2-cyanoethyl)-6,7,12,13-tetrahydro-13-methyl-5-oxo-5h-indolo[2,3-a]pyrrolo[3,4-c]carbazole | Human | 8552 | |
| EGFR | EGFR | TK | 5xgn | A | | 12-(2-cyanoethyl)-6,7,12,13-tetrahydro-13-methyl-5-oxo-5h-indolo[2,3-a]pyrrolo[3,4-c]carbazole | Human | 8553 | |
| EGFR | EGFR | TK | 5xgn | B | | - | Human | 8554 | |
| EGFR | EGFR | TK | 5y25 | A | | (2r)-n-[4-[(3-chloranyl-4-fluoranyl-phenyl)amino]-7-(3-morpholin-4-ylpropoxy)quinazolin-6-yl]-1-(2-fluoranylethanoyl)pyrrolidine-2-carboxamide | Human | 10373 | |
| EGFR | EGFR | TK | 5y9t | A | | 6-ethyl-3-[[4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-5-[(3r)-1-prop-2-enoylpyrrolidin-3-yl]oxy-pyrazine-2-carboxamide | Human | 10053 | |
| EGFR | EGFR | TK | 5yu9 | A | A | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 9430 | |
| EGFR | EGFR | TK | 5yu9 | A | B | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 9428 | |
| EGFR | EGFR | TK | 5yu9 | B | A | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 9433 | |
| EGFR | EGFR | TK | 5yu9 | B | B | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 9434 | |
| EGFR | EGFR | TK | 5yu9 | C | A | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 9432 | |
| EGFR | EGFR | TK | 5yu9 | C | B | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 9427 | |
| EGFR | EGFR | TK | 5yu9 | D | A | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 9431 | |
| EGFR | EGFR | TK | 5yu9 | D | B | 1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-one | Human | 9429 | |
| EGFR | EGFR | TK | 5zto | A | | n-{trans-4-[3-(2-chlorophenyl)-7-{[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]cyclohexyl}propanamide | Human | 11070 | |
| EGFR | EGFR | TK | 5zwj | A | | (2r)-2-(5-fluoro-2-hydroxyphenyl)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-(1,3-thiazol-2-yl)acetamide | Human | 10372 | |
| EGFR | EGFR | TK | 6d8e | A | | (4-fluorophenyl)methyl {2-[(1-methyl-1h-pyrazol-3-yl)amino]pyrimidin-4-yl}[3-(propanoylamino)phenyl]carbamate | Human | 10374 | |
| EGFR | EGFR | TK | 6duk | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 11067 | |
| EGFR | EGFR | TK | 6duk | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 11066 | |
| EGFR | EGFR | TK | 6duk | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 11060 | |
| EGFR | EGFR | TK | 6duk | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 11069 | |
| EGFR | EGFR | TK | 6duk | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 11061 | |
| EGFR | EGFR | TK | 6duk | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 11068 | |
| EGFR | EGFR | TK | 6duk | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 11064 | |
| EGFR | EGFR | TK | 6duk | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 11062 | |
| EGFR | EGFR | TK | 6duk | E | A | phosphoaminophosphonic acid-adenylate ester | Human | 11058 | |
| EGFR | EGFR | TK | 6duk | E | B | phosphoaminophosphonic acid-adenylate ester | Human | 11059 | |
| EGFR | EGFR | TK | 6duk | F | A | phosphoaminophosphonic acid-adenylate ester | Human | 11065 | |
| EGFR | EGFR | TK | 6duk | F | B | phosphoaminophosphonic acid-adenylate ester | Human | 11063 | |
| EGFR | EGFR | TK | 6jrj | A | | 6-(2-chloranyl-3-fluoranyl-phenyl)-5-methyl-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[(3s)-1-propanoylpiperidin-3-yl]pyrido[2,3-d]pyrimidin-7-one | Human | 12158 | |
| EGFR | EGFR | TK | 6jrk | A | | 6-(2-chloranyl-3-fluoranyl-phenyl)-5-methyl-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[(3s)-1-propanoylpiperidin-3-yl]pyrido[2,3-d]pyrimidin-7-one | Human | 12159 | |
| EGFR | EGFR | TK | 6jrx | A | | n-{trans-4-[3-(2-chlorophenyl)-7-{[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]cyclohexyl}propanamide | Human | 12157 | |
| EGFR | EGFR | TK | 6jwl | A | | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | 12173 | |
| EGFR | EGFR | TK | 6jx0 | A | | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | 12175 | |
| EGFR | EGFR | TK | 6jx4 | A | | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | 12176 | |
| EGFR | EGFR | TK | 6jxt | A | A | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | 12240 | |
| EGFR | EGFR | TK | 6jxt | A | B | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | 12239 | |
| EGFR | EGFR | TK | 6jz0 | A | | e-4-(dimethylamino)-n-[3-[4-[[(1s)-2-oxidanyl-1-phenyl-ethyl]amino]-6-phenyl-furo[2,3-d]pyrimidin-5-yl]phenyl]but-2-enamide | Human | 11845 | |
| EGFR | EGFR | TK | 6lub | A | A | n-[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]-7-(4-methylpiperazin-1-yl)-5-propan-2-yl-9-[2,2,2-tris(fluoranyl)ethoxy]pyrido[4,3-b]indol-3-amine | Human | 12918 | |
| EGFR | EGFR | TK | 6lub | A | B | n-[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]-7-(4-methylpiperazin-1-yl)-5-propan-2-yl-9-[2,2,2-tris(fluoranyl)ethoxy]pyrido[4,3-b]indol-3-amine | Human | 12917 | |
| EGFR | EGFR | TK | 6lud | A | | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | 12919 | |
| EGFR | EGFR | TK | 6p1d | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 11872 | |
| EGFR | EGFR | TK | 6p1d | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 11868 | |
| EGFR | EGFR | TK | 6p1d | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 11873 | |
| EGFR | EGFR | TK | 6p1d | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 11883 | |
| EGFR | EGFR | TK | 6p1d | C | A | 10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 11880 | |
| EGFR | EGFR | TK | 6p1d | C | B | 10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 11869 | |
| EGFR | EGFR | TK | 6p1d | D | A | 10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 11884 | |
| EGFR | EGFR | TK | 6p1d | D | B | 10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 11885 | |
| EGFR | EGFR | TK | 6p1l | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11878 | |
| EGFR | EGFR | TK | 6p1l | B | | phosphoaminophosphonic acid-adenylate ester | Human | 11886 | |
| EGFR | EGFR | TK | 6p1l | C | | phosphoaminophosphonic acid-adenylate ester | Human | 11876 | |
| EGFR | EGFR | TK | 6p1l | D | | phosphoaminophosphonic acid-adenylate ester | Human | 11870 | |
| EGFR | EGFR | TK | 6p8q | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 11875 | |
| EGFR | EGFR | TK | 6p8q | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 11882 | |
| EGFR | EGFR | TK | 6p8q | B | A | adenosine monophosphate | Human | 11867 | |
| EGFR | EGFR | TK | 6p8q | B | B | adenosine monophosphate | Human | 11874 | |
| EGFR | EGFR | TK | 6p8q | C | A | adenosine monophosphate | Human | 11881 | |
| EGFR | EGFR | TK | 6p8q | C | B | adenosine monophosphate | Human | 11879 | |
| EGFR | EGFR | TK | 6p8q | D | A | adenosine monophosphate | Human | 11871 | |
| EGFR | EGFR | TK | 6p8q | D | B | adenosine monophosphate | Human | 11877 | |
| EGFR | EGFR | TK | 6s89 | A | | ~{n}-[3-[6-[4-(4-methylpiperazin-1-yl)phenyl]-4-propan-2-yloxy-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | 11729 | |
| EGFR | EGFR | TK | 6s8a | A | | ~{n}-[3-[6-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-methylpropoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | 11728 | |
| EGFR | EGFR | TK | 6s9b | A | | 3-fluoranyl-~{n}-[1-(2-methyl-2-oxidanyl-propyl)benzimidazol-2-yl]-5-pyridin-3-yl-benzamide | Human | 11805 | |
| EGFR | EGFR | TK | 6s9c | A | A | ~{n}-[1-(2-methyl-2-oxidanyl-propyl)benzimidazol-2-yl]-2-phenyl-pyridine-4-carboxamide | Human | 11806 | |
| EGFR | EGFR | TK | 6s9c | A | B | ~{n}-[1-(2-methyl-2-oxidanyl-propyl)benzimidazol-2-yl]-2-phenyl-pyridine-4-carboxamide | Human | 11804 | |
| EGFR | EGFR | TK | 6s9d | A | | 8-oxa-14,21,23,28-tetraazapentacyclo[23.3.1.02,7.014,22.015,20]nonacosa-1(28),2(7),3,5,15,17,19,21,25(29),26-decaen-24-one | Human | 11803 | |
| EGFR | EGFR | TK | 6tfu | A | | ~{n}-[3-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | 12844 | |
| EGFR | EGFR | TK | 6tfu | B | | ~{n}-[3-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | 12842 | |
| EGFR | EGFR | TK | 6tfv | A | A | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | 12828 | |
| EGFR | EGFR | TK | 6tfv | A | B | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | 12832 | |
| EGFR | EGFR | TK | 6tfv | B | A | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | 12845 | |
| EGFR | EGFR | TK | 6tfv | B | B | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | 12827 | |
| EGFR | EGFR | TK | 6tfw | A | | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | 12838 | |
| EGFR | EGFR | TK | 6tfw | B | | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | 12837 | |
| EGFR | EGFR | TK | 6tfy | A | A | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamide | Human | 12825 | |
| EGFR | EGFR | TK | 6tfy | A | B | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamide | Human | 12841 | |
| EGFR | EGFR | TK | 6tfy | B | A | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamide | Human | 12847 | |
| EGFR | EGFR | TK | 6tfy | B | B | ~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamide | Human | 12831 | |
| EGFR | EGFR | TK | 6tfz | A | A | ~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | 12840 | |
| EGFR | EGFR | TK | 6tfz | A | B | ~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | 12846 | |
| EGFR | EGFR | TK | 6tfz | B | A | ~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | 12830 | |
| EGFR | EGFR | TK | 6tfz | B | B | ~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamide | Human | 12839 | |
| EGFR | EGFR | TK | 6tg0 | A | A | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | 12833 | |
| EGFR | EGFR | TK | 6tg0 | A | B | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | 12829 | |
| EGFR | EGFR | TK | 6tg0 | B | A | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | 12834 | |
| EGFR | EGFR | TK | 6tg0 | B | B | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamide | Human | 12835 | |
| EGFR | EGFR | TK | 6tg1 | A | A | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | 12826 | |
| EGFR | EGFR | TK | 6tg1 | A | B | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | 12843 | |
| EGFR | EGFR | TK | 6tg1 | B | A | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | 12836 | |
| EGFR | EGFR | TK | 6tg1 | B | B | ~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamide | Human | 12824 | |
| EGFR | EGFR | TK | 6v5n | A | A | 3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-ol | Human | 12170 | |
| EGFR | EGFR | TK | 6v5n | A | B | 3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-ol | Human | 12180 | |
| EGFR | EGFR | TK | 6v5n | B | A | 3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-ol | Human | 12227 | |
| EGFR | EGFR | TK | 6v5n | B | B | 3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-ol | Human | 12185 | |
| EGFR | EGFR | TK | 6v5n | C | A | 3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-ol | Human | 12197 | |
| EGFR | EGFR | TK | 6v5n | C | B | 3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-ol | Human | 12196 | |
| EGFR | EGFR | TK | 6v5n | D | A | 3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-ol | Human | 12199 | |
| EGFR | EGFR | TK | 6v5n | D | B | 3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-ol | Human | 12201 | |
| EGFR | EGFR | TK | 6v5p | A | A | 4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridine | Human | 12174 | |
| EGFR | EGFR | TK | 6v5p | A | B | 4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridine | Human | 12172 | |
| EGFR | EGFR | TK | 6v5p | B | A | 4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridine | Human | 12203 | |
| EGFR | EGFR | TK | 6v5p | B | B | 4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridine | Human | 12200 | |
| EGFR | EGFR | TK | 6v5p | C | A | 4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridine | Human | 12210 | |
| EGFR | EGFR | TK | 6v5p | C | B | 4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridine | Human | 12192 | |
| EGFR | EGFR | TK | 6v5p | D | A | 4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridine | Human | 12218 | |
| EGFR | EGFR | TK | 6v5p | D | B | 4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridine | Human | 12186 | |
| EGFR | EGFR | TK | 6v66 | A | A | n-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamide | Human | 12178 | |
| EGFR | EGFR | TK | 6v66 | A | B | n-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamide | Human | 12177 | |
| EGFR | EGFR | TK | 6v66 | B | A | n-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamide | Human | 12205 | |
| EGFR | EGFR | TK | 6v66 | B | B | n-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamide | Human | 12217 | |
| EGFR | EGFR | TK | 6v66 | C | A | n-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamide | Human | 12184 | |
| EGFR | EGFR | TK | 6v66 | C | B | n-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamide | Human | 12208 | |
| EGFR | EGFR | TK | 6v66 | D | A | n-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamide | Human | 12221 | |
| EGFR | EGFR | TK | 6v66 | D | B | n-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamide | Human | 12224 | |
| EGFR | EGFR | TK | 6v6k | A | A | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12179 | |
| EGFR | EGFR | TK | 6v6k | A | B | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12168 | |
| EGFR | EGFR | TK | 6v6k | B | A | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12202 | |
| EGFR | EGFR | TK | 6v6k | B | B | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12229 | |
| EGFR | EGFR | TK | 6v6k | C | A | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12207 | |
| EGFR | EGFR | TK | 6v6k | C | B | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12209 | |
| EGFR | EGFR | TK | 6v6k | D | A | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12223 | |
| EGFR | EGFR | TK | 6v6k | D | B | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12212 | |
| EGFR | EGFR | TK | 6v6k | E | A | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12187 | |
| EGFR | EGFR | TK | 6v6k | E | B | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12193 | |
| EGFR | EGFR | TK | 6v6k | F | A | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12204 | |
| EGFR | EGFR | TK | 6v6k | F | B | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12214 | |
| EGFR | EGFR | TK | 6v6k | G | A | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12195 | |
| EGFR | EGFR | TK | 6v6k | G | B | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12222 | |
| EGFR | EGFR | TK | 6v6k | H | A | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12216 | |
| EGFR | EGFR | TK | 6v6k | H | B | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12190 | |
| EGFR | EGFR | TK | 6v6o | A | A | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12169 | |
| EGFR | EGFR | TK | 6v6o | A | B | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12181 | |
| EGFR | EGFR | TK | 6v6o | B | A | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12198 | |
| EGFR | EGFR | TK | 6v6o | B | B | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12228 | |
| EGFR | EGFR | TK | 6v6o | C | A | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12188 | |
| EGFR | EGFR | TK | 6v6o | C | B | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12226 | |
| EGFR | EGFR | TK | 6v6o | D | A | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12213 | |
| EGFR | EGFR | TK | 6v6o | D | B | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12219 | |
| EGFR | EGFR | TK | 6v6o | E | A | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12225 | |
| EGFR | EGFR | TK | 6v6o | E | B | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12191 | |
| EGFR | EGFR | TK | 6v6o | F | A | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12206 | |
| EGFR | EGFR | TK | 6v6o | F | B | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12220 | |
| EGFR | EGFR | TK | 6v6o | G | A | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12215 | |
| EGFR | EGFR | TK | 6v6o | G | B | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12189 | |
| EGFR | EGFR | TK | 6v6o | H | A | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12194 | |
| EGFR | EGFR | TK | 6v6o | H | B | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12211 | |
| EGFR | EGFR | TK | 6vh4 | A | | n-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12183 | |
| EGFR | EGFR | TK | 6vhn | A | | n-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamide | Human | 12171 | |
| EGFR | EGFR | TK | 6vhp | A | | n-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamide | Human | 12182 | |
| EGFR | EGFR | TK | 6wa2 | A | A | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamide | Human | 13434 | |
| EGFR | EGFR | TK | 6wa2 | A | B | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamide | Human | 13442 | |
| EGFR | EGFR | TK | 6wa2 | B | A | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamide | Human | 13443 | |
| EGFR | EGFR | TK | 6wa2 | B | B | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamide | Human | 13444 | |
| EGFR | EGFR | TK | 6wa2 | C | A | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamide | Human | 13447 | |
| EGFR | EGFR | TK | 6wa2 | C | B | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamide | Human | 13436 | |
| EGFR | EGFR | TK | 6wa2 | D | A | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamide | Human | 13439 | |
| EGFR | EGFR | TK | 6wa2 | D | B | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamide | Human | 13437 | |
| EGFR | EGFR | TK | 6wak | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 13438 | |
| EGFR | EGFR | TK | 6wak | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 13440 | |
| EGFR | EGFR | TK | 6wak | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 13435 | |
| EGFR | EGFR | TK | 6wak | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 13448 | |
| EGFR | EGFR | TK | 6wak | C | A | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-[(1-oxo-1,3-dihydro-2h-isoindol-2-yl)methyl]benzamide | Human | 13449 | |
| EGFR | EGFR | TK | 6wak | C | B | n-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-[(1-oxo-1,3-dihydro-2h-isoindol-2-yl)methyl]benzamide | Human | 13441 | |
| EGFR | EGFR | TK | 6wak | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 13446 | |
| EGFR | EGFR | TK | 6wak | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 13445 | |
| EGFR | EGFR | TK | 6wxn | A | A | - | Human | 13558 | |
| EGFR | EGFR | TK | 6wxn | A | B | - | Human | 13557 | |
| EGFR | EGFR | TK | 6xl4 | A | | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 13759 | |
| EGFR | EGFR | TK | 6z4b | A | A | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 12975 | |
| EGFR | EGFR | TK | 6z4b | A | B | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 12974 | |
| EGFR | EGFR | TK | 6z4d | A | A | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 12971 | |
| EGFR | EGFR | TK | 6z4d | A | B | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 12972 | |
| EGFR | EGFR | TK | 6z4d | B | A | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 12979 | |
| EGFR | EGFR | TK | 6z4d | B | B | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 12978 | |
| EGFR | EGFR | TK | 7a2a | A | A | (2r)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-2-phenyl-n-(1,3-thiazol-2-yl)acetamide | Human | 12977 | |
| EGFR | EGFR | TK | 7a2a | A | B | (2r)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-2-phenyl-n-(1,3-thiazol-2-yl)acetamide | Human | 12976 | |
| EGFR | EGFR | TK | 7a2a | B | A | (2r)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-2-phenyl-n-(1,3-thiazol-2-yl)acetamide | Human | 12970 | |
| EGFR | EGFR | TK | 7a2a | B | B | (2r)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-2-phenyl-n-(1,3-thiazol-2-yl)acetamide | Human | 12973 | |
| EGFR | EGFR | TK | 7a6i | A | | ~{n}-[5-[4-chloranyl-2-[4-(4-methylpiperazin-1-yl)phenyl]-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]-2-methyl-phenyl]propanamide | Human | 14123 | |
| EGFR | EGFR | TK | 7a6j | A | A | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14125 | |
| EGFR | EGFR | TK | 7a6j | A | B | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14124 | |
| EGFR | EGFR | TK | 7a6k | A | A | propan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylate | Human | 14111 | |
| EGFR | EGFR | TK | 7a6k | A | B | propan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylate | Human | 14113 | |
| EGFR | EGFR | TK | 7a6k | A | C | propan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylate | Human | 14112 | |
| EGFR | EGFR | TK | 7aei | A | | 5-chloranyl-~{n}2-[4-[4-(dimethylamino)piperidin-1-yl]-2-methoxy-5-(1-methylpyrazol-4-yl)phenyl]-~{n}4-(2-dimethylphosphorylphenyl)pyrimidine-2,4-diamine | Human | 13619 | |
| EGFR | EGFR | TK | 7aem | A | | 5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamine | Human | 13482 | |
| EGFR | EGFR | TK | 7b85 | A | | propan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylate | Human | 14121 | |
| EGFR | EGFR | TK | 7er2 | A | | 5-chloranyl-n2-[3-chloranyl-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n4-(2-dimethylphosphorylphenyl)pyrimidine-2,4-diamine | Human | 14194 | |
| EGFR | EGFR | TK | 7jxi | A | A | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 13885 | |
| EGFR | EGFR | TK | 7jxi | A | B | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 13882 | |
| EGFR | EGFR | TK | 7jxk | A | A | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 13884 | |
| EGFR | EGFR | TK | 7jxk | A | B | n-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamide | Human | 13876 | |
| EGFR | EGFR | TK | 7jxl | A | A | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-5-{[4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-4-methoxyphenyl)propanamide | Human | 13878 | |
| EGFR | EGFR | TK | 7jxl | A | B | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-5-{[4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-4-methoxyphenyl)propanamide | Human | 13879 | |
| EGFR | EGFR | TK | 7jxm | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13883 | |
| EGFR | EGFR | TK | 7jxp | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 13881 | |
| EGFR | EGFR | TK | 7jxp | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 13874 | |
| EGFR | EGFR | TK | 7jxq | A | A | (2r)-2-(5-fluoro-2-hydroxyphenyl)-2-{6-[4-(1-methylpiperidin-4-yl)phenyl]-1-oxo-1,3-dihydro-2h-isoindol-2-yl}-n-(1,3-thiazol-2-yl)acetamide | Human | 13886 | |
| EGFR | EGFR | TK | 7jxq | A | B | (2r)-2-(5-fluoro-2-hydroxyphenyl)-2-{6-[4-(1-methylpiperidin-4-yl)phenyl]-1-oxo-1,3-dihydro-2h-isoindol-2-yl}-n-(1,3-thiazol-2-yl)acetamide | Human | 13880 | |
| EGFR | EGFR | TK | 7jxw | A | A | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | 13875 | |
| EGFR | EGFR | TK | 7jxw | A | B | n-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamide | Human | 13877 | |
| EGFR | EGFR | TK | 7k1h | A | | (2r)-2-(5-fluoro-2-hydroxyphenyl)-2-{6-[4-(1-methylpiperidin-4-yl)phenyl]-1-oxo-1,3-dihydro-2h-isoindol-2-yl}-n-(1,3-thiazol-2-yl)acetamide | Human | 13902 | |
| EGFR | EGFR | TK | 7k1i | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 13904 | |
| EGFR | EGFR | TK | 7k1i | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 13903 | |
| EGFR | EGFR | TK | 7kxz | A | | (20r)-10,15,20-trimethyl-2-[(4-methylpiperazin-1-yl)methyl]-18,19,20,21-tetrahydro-15h,17h-12,8-(metheno)pyrazolo[3',4':2,3][1,5,10,12]oxatriazacycloheptadecino[12,11-a]benzimidazol-7(6h)-one | Human | 14074 | |
| EGFR | EGFR | TK | 7ky0 | A | | (20r)-10,15,20-trimethyl-2-[(4-methylpiperazin-1-yl)methyl]-18,19,20,21-tetrahydro-15h,17h-12,8-(metheno)pyrazolo[3',4':2,3][1,5,10,12]oxatriazacycloheptadecino[12,11-a]benzimidazol-7(6h)-one | Human | 14073 | |
| EGFR | EGFR | TK | 7lg8 | A | | 6-ethyl-3-[[4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-5-[(3r)-1-prop-2-enoylpyrrolidin-3-yl]oxy-pyrazine-2-carboxamide | Human | 14120 | |
| EGFR | EGFR | TK | 7lgs | A | A | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 13906 | |
| EGFR | EGFR | TK | 7lgs | A | B | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 13905 | |
| EGFR | EGFR | TK | 7lgs | B | A | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 15372 | |
| EGFR | EGFR | TK | 7lgs | B | B | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 15373 | |
| EGFR | EGFR | TK | 7lgs | C | A | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 15371 | |
| EGFR | EGFR | TK | 7lgs | C | B | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 15376 | |
| EGFR | EGFR | TK | 7lgs | D | A | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 15370 | |
| EGFR | EGFR | TK | 7lgs | D | B | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 15374 | |
| EGFR | EGFR | TK | 7ltx | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14122 | |
| EGFR | EGFR | TK | 7oxb | A | | 2-[2-(3-methoxyphenyl)pyrimidin-4-yl]-1'-prop-2-enoyl-spiro[5,6-dihydro-1~{h}-pyrrolo[3,2-c]pyridine-7,4'-piperidine]-4-one | Human | 13948 | |
| EGFR | EGFR | TK | 7si1 | A | A | - | Human | 14478 | |
| EGFR | EGFR | TK | 7si1 | A | B | - | Human | 14480 | |
| EGFR | EGFR | TK | 7si1 | A | C | - | Human | 14479 | |
| EGFR | EGFR | TK | 7syd | A | B | - | Human | 14027 | |
| EGFR | EGFR | TK | 7sye | A | | - | Human | 14028 | |
| EGFR | EGFR | TK | 7sz0 | A | B | - | Human | 14031 | |
| EGFR | EGFR | TK | 7sz1 | A | | - | Human | 14029 | |
| EGFR | EGFR | TK | 7sz5 | A | | - | Human | 14030 | |
| EGFR | EGFR | TK | 7sz7 | A | | - | Human | 14016 | |
| EGFR | EGFR | TK | 7t4i | A | | propan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylate | Human | 14530 | |
| EGFR | EGFR | TK | 7t4j | A | | propan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylate | Human | 14529 | |
| EGFR | EGFR | TK | 7tvd | A | | - | Human | 14107 | |
| EGFR | EGFR | TK | 7u98 | A | | 19-chloro-18-fluoro-22-methoxy-8,9,11,12,14,15-hexahydro-21h-4,6-ethenopyrimido[5,4-m][1,4,7,10,15]benzotetraoxazacycloheptadecine | Human | 14526 | |
| EGFR | EGFR | TK | 7u99 | A | | 19-chloro-22-methoxy-8,9,11,12,14,15-hexahydro-21h-4,6-ethenopyrimido[5,4-m][1,4,7,10,15]benzotetraoxazacycloheptadecine | Human | 14533 | |
| EGFR | EGFR | TK | 7u9a | A | | 4-(5-chloro-4-fluoro-2-hydroxyanilino)-7-methoxyquinazolin-6-ol | Human | 14527 | |
| EGFR | EGFR | TK | 7ukv | A | | n-[5-{[(4p)-4-{4-[(dimethylamino)methyl]-3-phenyl-1h-pyrazol-1-yl}pyrimidin-2-yl]amino}-4-methoxy-2-(morpholin-4-yl)phenyl]propanamide | Human | 14528 | |
| EGFR | EGFR | TK | 7ukw | A | A | - | Human | 14531 | |
| EGFR | EGFR | TK | 7ukw | A | B | - | Human | 14532 | |
| EGFR | EGFR | TK | 7vra | A | A | 25-chloro-11-(ethylsulfonyl)-44-morpholino-11h-5,12-dioxa-3-aza-1(3,6)-indola-2(4,2)-pyrimidina-4(1,3)-benzenacyclododecaphane | Human | 14235 | |
| EGFR | EGFR | TK | 7vra | A | B | 25-chloro-11-(ethylsulfonyl)-44-morpholino-11h-5,12-dioxa-3-aza-1(3,6)-indola-2(4,2)-pyrimidina-4(1,3)-benzenacyclododecaphane | Human | 14237 | |
| EGFR | EGFR | TK | 7vre | A | | 5-chloranyl-n-[5-chloranyl-2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-4-(1-ethylsulfonylindol-3-yl)pyrimidin-2-amine | Human | 14236 | |
| EGFR | EGFR | TK | 7zym | A | | 5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamine | Human | 14726 | |
| EGFR | EGFR | TK | 7zyn | A | A | n-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | Human | 14727 | |
| EGFR | EGFR | TK | 7zyn | A | B | n-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | Human | 14728 | |
| EGFR | EGFR | TK | 7zyp | A | | propan-2-yl 2-[[4-(4-azanylpiperidin-1-yl)-2-methoxy-phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylate | Human | 14731 | |
| EGFR | EGFR | TK | 7zyq | A | A | phenyl 2-[[4-[4-(dimethylamino)piperidin-1-yl]-2-methoxy-phenyl]amino]-4-(1h-indol-3-yl)pyrimidine-5-carboxylate | Human | 14730 | |
| EGFR | EGFR | TK | 7zyq | A | B | phenyl 2-[[4-[4-(dimethylamino)piperidin-1-yl]-2-methoxy-phenyl]amino]-4-(1h-indol-3-yl)pyrimidine-5-carboxylate | Human | 14729 | |
| EGFR | EGFR | TK | 8a27 | A | A | (2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamide | Human | 14462 | |
| EGFR | EGFR | TK | 8a27 | A | B | (2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamide | Human | 14465 | |
| EGFR | EGFR | TK | 8a2a | A | A | (2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamide | Human | 14466 | |
| EGFR | EGFR | TK | 8a2a | A | B | (2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamide | Human | 14460 | |
| EGFR | EGFR | TK | 8a2b | A | A | (2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamide | Human | 14464 | |
| EGFR | EGFR | TK | 8a2b | A | B | (2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamide | Human | 14459 | |
| EGFR | EGFR | TK | 8a2d | A | A | (2r)-2-[4-[bis(fluoranyl)methyl]-6-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-7-methyl-indazol-2-yl]-2-spiro[6,7-dihydropyrrolo[1,2-c]imidazole-5,1'-cyclopropane]-1-yl-n-(1,3-thiazol-2-yl)ethanamide | Human | 14463 | |
| EGFR | EGFR | TK | 8a2d | A | B | (2r)-2-[4-[bis(fluoranyl)methyl]-6-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-7-methyl-indazol-2-yl]-2-spiro[6,7-dihydropyrrolo[1,2-c]imidazole-5,1'-cyclopropane]-1-yl-n-(1,3-thiazol-2-yl)ethanamide | Human | 14461 | |
| EGFR | EGFR | TK | 8d73 | A | A | (3s,4r)-3-fluoro-1-(4-{[4-(methylamino)-1-(propan-2-yl)pyrido[3,4-d]pyridazin-7-yl]amino}pyrimidin-2-yl)piperidin-4-ol | Human | 14312 | |
| EGFR | EGFR | TK | 8d73 | A | B | (3s,4r)-3-fluoro-1-(4-{[4-(methylamino)-1-(propan-2-yl)pyrido[3,4-d]pyridazin-7-yl]amino}pyrimidin-2-yl)piperidin-4-ol | Human | 14310 | |
| EGFR | EGFR | TK | 8d76 | A | A | (3s,4r)-3-fluoro-1-(4-{[8-{3-[(methanesulfonyl)methyl]azetidin-1-yl}-5-(propan-2-yl)-2,7-naphthyridin-3-yl]amino}pyrimidin-2-yl)-3-methylpiperidin-4-ol | Human | 14311 | |
| EGFR | EGFR | TK | 8d76 | A | B | (3s,4r)-3-fluoro-1-(4-{[8-{3-[(methanesulfonyl)methyl]azetidin-1-yl}-5-(propan-2-yl)-2,7-naphthyridin-3-yl]amino}pyrimidin-2-yl)-3-methylpiperidin-4-ol | Human | 14313 | |
| EGFR | EGFR | TK | 8dsw | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14946 | |
| EGFR | EGFR | TK | 8eme | A | | - | Human | 14938 | |
| EGFR | EGFR | TK | 8eme | B | | n-{7-methyl-1-[(3s)-1-(prop-2-enoyl)azepan-3-yl]-1h-benzimidazol-2-yl}-5-(prop-2-enamido)thiophene-3-carboxamide | Human | 15375 | |
| EGFR | EGFR | TK | 8f1h | A | | n-[(5p,8s,10r)-4-amino-6-methyl-5-(quinolin-3-yl)-8,9-dihydropyrimido[5,4-b]indolizin-8-yl]prop-2-enamide | Human | 14947 | |
| EGFR | EGFR | TK | 8f1w | A | | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14944 | |
| EGFR | EGFR | TK | 8f1x | A | A | propan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylate | Human | 14942 | |
| EGFR | EGFR | TK | 8f1x | A | B | propan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylate | Human | 14943 | |
| EGFR | EGFR | TK | 8f1y | A | | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14940 | |
| EGFR | EGFR | TK | 8f1z | A | | (2p)-3-(3-chloro-2-methoxyanilino)-2-[3-(2-methoxy-2-methylpropoxy)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 14939 | |
| EGFR | EGFR | TK | 8fv3 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15168 | |
| EGFR | EGFR | TK | 8fv3 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15167 | |
| EGFR | EGFR | TK | 8fv4 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15166 | |
| EGFR | EGFR | TK | 8fv4 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15165 | |
| EGFR | EGFR | TK | 8g63 | A | | ralimetinib | Human | 14937 | |
| EGFR | EGFR | TK | 8gb4 | A | A | 2-[(r)-(1h-benzimidazol-2-yl)(3-fluorophenyl)methyl]-6-[4-(1-methylpiperidin-4-yl)phenyl]-2,3-dihydro-1h-isoindol-1-one | Human | 15236 | |
| EGFR | EGFR | TK | 8gb4 | A | B | 2-[(r)-(1h-benzimidazol-2-yl)(3-fluorophenyl)methyl]-6-[4-(1-methylpiperidin-4-yl)phenyl]-2,3-dihydro-1h-isoindol-1-one | Human | 15235 | |
| EGFR | EGFR | TK | 8gk5 | A | | ~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamide | Human | 15327 | |
| EGFR | EGFR | TK | 8h7x | A | | 5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamine | Human | 14945 | |
| EGFR | EGFR | TK | 8hv1 | A | | 3-(3-bromophenyl)-1,4-dihydro-1,2,4-triazole-5-thione | Human | 15072 | |
| EGFR | EGFR | TK | 8hv2 | A | A | ~{n}-pyridin-2-ylprop-2-enamide | Human | 15077 | |
| EGFR | EGFR | TK | 8hv2 | A | B | ~{n}-pyridin-2-ylprop-2-enamide | Human | 15068 | |
| EGFR | EGFR | TK | 8hv3 | A | | ~{n}-pyridin-2-ylprop-2-enamide | Human | 15067 | |
| EGFR | EGFR | TK | 8hv4 | A | | ~{n}-pyridin-2-ylprop-2-enamide | Human | 15075 | |
| EGFR | EGFR | TK | 8hv5 | A | A | ~{n}-(1-methylbenzimidazol-4-yl)prop-2-enamide | Human | 15069 | |
| EGFR | EGFR | TK | 8hv5 | A | B | ~{n}-(1-methylbenzimidazol-4-yl)prop-2-enamide | Human | 15065 | |
| EGFR | EGFR | TK | 8hv6 | A | A | ~{n}-quinolin-7-ylprop-2-enamide | Human | 15071 | |
| EGFR | EGFR | TK | 8hv6 | A | B | ~{n}-quinolin-7-ylprop-2-enamide | Human | 15064 | |
| EGFR | EGFR | TK | 8hv7 | A | | ~{n}-[7-(dimethylamino)-2-methyl-pyrazolo[1,5-a]pyrimidin-5-yl]prop-2-enamide | Human | 15066 | |
| EGFR | EGFR | TK | 8hv8 | A | | ~{n}-pyrazolo[1,5-a]pyridin-2-ylprop-2-enamide | Human | 15073 | |
| EGFR | EGFR | TK | 8hv9 | A | A | ~{n}-(4-phenylpyridin-2-yl)prop-2-enamide | Human | 15063 | |
| EGFR | EGFR | TK | 8hv9 | A | B | ~{n}-(4-phenylpyridin-2-yl)prop-2-enamide | Human | 15070 | |
| EGFR | EGFR | TK | 8hva | A | | ~{n}-[6-(1-methylindol-3-yl)pyrimidin-4-yl]prop-2-enamide | Human | 15076 | |
| EGFR | EGFR | TK | 8hy7 | A | | ~{n}-[3-[[6-fluoranyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]quinazolin-4-yl]amino]phenyl]prop-2-enamide | Human | 14941 | |
| EGFR | EGFR | TK | 8kfq | A | | ~{n}-[3-[[6-chloranyl-2-[(1-ethylpyrazol-4-yl)amino]quinazolin-4-yl]amino]phenyl]prop-2-enamide | Human | 15367 | |
| EGFR | EGFR | TK | 8sc7 | A | A | n-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide | Human | 15325 | |
| EGFR | EGFR | TK | 8sc7 | A | B | n-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide | Human | 15324 | |
| EGFR | EGFR | TK | 8sc7 | A | C | n-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide | Human | 15326 | |
| EGFR | EGFR | TK | 8tjl | A | | 1-{3-[(4-amino-1-tert-butyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)oxy]azetidin-1-yl}propan-1-one | Human | 15237 | |
| EGFR | EGFR | TK | 8to3 | A | A | 3-hydroxy-n-{(3p)-3-[(4p)-2-(methylsulfanyl)-5-{2-[4-(piperazin-1-yl)anilino]pyridin-4-yl}-1h-imidazol-4-yl]phenyl}-2-[(1-oxo-1,3-dihydro-2h-isoindol-2-yl)methyl]benzamide | Human | 15388 | |
| EGFR | EGFR | TK | 8to3 | A | B | 3-hydroxy-n-{(3p)-3-[(4p)-2-(methylsulfanyl)-5-{2-[4-(piperazin-1-yl)anilino]pyridin-4-yl}-1h-imidazol-4-yl]phenyl}-2-[(1-oxo-1,3-dihydro-2h-isoindol-2-yl)methyl]benzamide | Human | 15389 | |
| EGFR | EGFR | TK | 8to4 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15391 | |
| EGFR | EGFR | TK | 8to4 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15390 | |
| EGFR | EGFR | TK | 8wd4 | A | | ~{n}-[3,3-bis(fluoranyl)propyl]-4-[[(2~{s})-butan-2-yl]amino]-6-[[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]amino]pyridine-3-carboxamide | Human | 15074 | |
| EIF2AK2 (PKR) | PEK | Other | 2a19 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 920 | |
| EIF2AK2 (PKR) | PEK | Other | 2a19 | C | | phosphoaminophosphonic acid-adenylate ester | Human | 918 | |
| EIF2AK2 (PKR) | PEK | Other | 2a1a | B | | - | Human | 919 | |
| EIF2AK2 (PKR) | PEK | Other | 3uiu | A | | - | Human | 917 | |
| EIF2AK2 (PKR) | PEK | Other | 3uiu | B | | - | Human | 916 | |
| EIF2AK2 (PKR) | PEK | Other | 6d3k | A | | adenosine-5'-diphosphate | Human | 11386 | |
| EIF2AK2 (PKR) | PEK | Other | 6d3k | B | | adenosine-5'-diphosphate | Human | 11385 | |
| EIF2AK2 (PKR) | PEK | Other | 6d3k | C | | adenosine-5'-diphosphate | Human | 11387 | |
| EIF2AK2 (PKR) | PEK | Other | 6d3l | A | | - | Human | 11384 | |
| EIF2AK2 (PKR) | PEK | Other | 8qel | B | | (3~{z})-3-[(4-methyl-1~{h}-imidazol-5-yl)methylidene]-2-oxidanylidene-1~{h}-indole-5-carboxamide | Human | 14954 | |
| Eif2ak3 (PEK) | PEK | Other | 3qd2 | B | | - | Mouse | 5802 | |
| EIF2AK3 (PEK) | PEK | Other | 4g31 | A | A | 1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanone | Human | 2672 | |
| EIF2AK3 (PEK) | PEK | Other | 4g31 | A | B | 1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanone | Human | 2671 | |
| EIF2AK3 (PEK) | PEK | Other | 4g34 | A | A | 1-[5-(4-aminothieno[3,2-c]pyridin-3-yl)-2,3-dihydro-1h-indol-1-yl]-2-phenylethanone | Human | 2674 | |
| EIF2AK3 (PEK) | PEK | Other | 4g34 | A | B | 1-[5-(4-aminothieno[3,2-c]pyridin-3-yl)-2,3-dihydro-1h-indol-1-yl]-2-phenylethanone | Human | 2670 | |
| EIF2AK3 (PEK) | PEK | Other | 4m7i | A | | 1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-1h-indol-1-yl]-2-(6-methylpyridin-2-yl)ethanone | Human | 2673 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7h | A | A | n-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1h-pyrazole-4-carboxamide | Human | 7247 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7h | A | B | n-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1h-pyrazole-4-carboxamide | Human | 7240 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7j | A | A | 2-amino-n-[4-methoxy-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamide | Human | 6848 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7j | A | B | 2-amino-n-[4-methoxy-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamide | Human | 6841 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7k | A | A | 4-{2-amino-3-[5-fluoro-2-(methylamino)quinazolin-6-yl]-4-methylbenzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | 7246 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7k | A | B | 4-{2-amino-3-[5-fluoro-2-(methylamino)quinazolin-6-yl]-4-methylbenzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | 7242 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7l | A | A | 4-{2-amino-4-methyl-3-[2-(methylamino)-1,3-benzothiazol-6-yl]benzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | 6844 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7l | A | B | 4-{2-amino-4-methyl-3-[2-(methylamino)-1,3-benzothiazol-6-yl]benzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | 6843 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7n | A | A | 4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | 7245 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7n | A | B | 4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-one | Human | 7241 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7o | A | A | 1-[5-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanone | Human | 7243 | |
| EIF2AK3 (PEK) | PEK | Other | 4x7o | A | B | 1-[5-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanone | Human | 7244 | |
| EIF2AK3 (PEK) | PEK | Other | 7mf0 | A | | 2-amino-n-cyclopropyl-5-(4-{[(2r)-2-(3,5-difluorophenyl)-2-hydroxyacetyl]amino}-2-methylphenyl)pyridine-3-carboxamide | Human | 13577 | |
| EIF2AK3 (PEK) | PEK | Other | 8eq9 | A | A | (2r)-n-[(4m)-4-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamide | Human | 14524 | |
| EIF2AK3 (PEK) | PEK | Other | 8eq9 | A | B | (2r)-n-[(4m)-4-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamide | Human | 14521 | |
| EIF2AK3 (PEK) | PEK | Other | 8eqd | A | | (2r)-n-[(4m)-4-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamide | Human | 14523 | |
| EIF2AK3 (PEK) | PEK | Other | 8eqe | A | | (2r)-n-[(4m)-4-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-hydroxy-2-[3-(trifluoromethyl)phenyl]acetamide | Human | 14522 | |
| EIF2AK4 (GCN2) | PEK | Other | 6n3l | A | A | n-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamide | Human | 11691 | |
| EIF2AK4 (GCN2) | PEK | Other | 6n3l | A | B | n-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamide | Human | 11694 | |
| EIF2AK4 (GCN2) | PEK | Other | 6n3l | B | A | n-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamide | Human | 11693 | |
| EIF2AK4 (GCN2) | PEK | Other | 6n3l | B | B | n-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamide | Human | 11692 | |
| EIF2AK4 (GCN2) | PEK | Other | 6n3n | A | | n-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-2,5-dichloro-3-(hydroxymethyl)benzene-1-sulfonamide | Human | 11690 | |
| EIF2AK4 (GCN2) | PEK | Other | 6n3o | A | | n-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-5-chloro-2-methoxypyridine-3-sulfonamide | Human | 11695 | |
| EIF2AK4 (GCN2) | PEK | Other | 7qq6 | A | | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 14116 | |
| EIF2AK4 (GCN2) | PEK | Other | 7qwk | A | | (2~{s})-~{n}-[(1~{s})-1-[4-[(6-pyridin-4-ylquinazolin-2-yl)amino]phenyl]ethyl]piperidine-2-carboxamide | Human | 14209 | |
| EIF2AK4 (GCN2) | PEK | Other | 8t7t | A | A | - | Human | 15229 | |
| EIF2AK4 (GCN2) | PEK | Other | 8t7t | A | B | - | Human | 15230 | |
| EPHA2 (EphA2) | Eph | TK | 1mqb | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2088 | |
| EPHA2 (EphA2) | Eph | TK | 1mqb | B | | phosphoaminophosphonic acid-adenylate ester | Human | 2089 | |
| EPHA2 (EphA2) | Eph | TK | 4p2k | A | | - | Human | 2091 | |
| EPHA2 (EphA2) | Eph | TK | 4pdo | A | | - | Human | 2086 | |
| EPHA2 (EphA2) | Eph | TK | 4pdo | B | | - | Human | 2087 | |
| EPHA2 (EphA2) | Eph | TK | 4trl | A | | - | Human | 2090 | |
| EPHA2 (EphA2) | Eph | TK | 5ek7 | A | | - | Human | 6322 | |
| EPHA2 (EphA2) | Eph | TK | 5ek7 | B | | - | Human | 6321 | |
| EPHA2 (EphA2) | Eph | TK | 5i9u | A | A | - | Human | 7190 | |
| EPHA2 (EphA2) | Eph | TK | 5i9u | A | B | - | Human | 7185 | |
| EPHA2 (EphA2) | Eph | TK | 5i9v | A | A | phosphothiophosphoric acid-adenylate ester | Human | 7188 | |
| EPHA2 (EphA2) | Eph | TK | 5i9v | A | B | phosphothiophosphoric acid-adenylate ester | Human | 7173 | |
| EPHA2 (EphA2) | Eph | TK | 5i9w | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 7187 | |
| EPHA2 (EphA2) | Eph | TK | 5i9w | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 7178 | |
| EPHA2 (EphA2) | Eph | TK | 5i9x | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 7182 | |
| EPHA2 (EphA2) | Eph | TK | 5i9x | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 7177 | |
| EPHA2 (EphA2) | Eph | TK | 5i9y | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7194 | |
| EPHA2 (EphA2) | Eph | TK | 5i9y | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7176 | |
| EPHA2 (EphA2) | Eph | TK | 5i9z | A | A | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 7180 | |
| EPHA2 (EphA2) | Eph | TK | 5i9z | A | B | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 7181 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | A | A | alisertib | Human | 7169 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | A | B | alisertib | Human | 7171 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | B | A | alisertib | Human | 7174 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | B | B | alisertib | Human | 7179 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | C | A | alisertib | Human | 7186 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | C | B | alisertib | Human | 7175 | |
| EPHA2 (EphA2) | Eph | TK | 5ia1 | A | | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 7191 | |
| EPHA2 (EphA2) | Eph | TK | 5ia2 | A | A | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 7170 | |
| EPHA2 (EphA2) | Eph | TK | 5ia2 | A | B | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 7172 | |
| EPHA2 (EphA2) | Eph | TK | 5ia3 | A | A | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Human | 7193 | |
| EPHA2 (EphA2) | Eph | TK | 5ia3 | A | B | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Human | 7184 | |
| EPHA2 (EphA2) | Eph | TK | 5ia4 | A | A | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 7189 | |
| EPHA2 (EphA2) | Eph | TK | 5ia4 | A | B | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 7168 | |
| EPHA2 (EphA2) | Eph | TK | 5ia5 | A | A | golvatinib | Human | 7192 | |
| EPHA2 (EphA2) | Eph | TK | 5ia5 | A | B | golvatinib | Human | 7183 | |
| EPHA2 (EphA2) | Eph | TK | 5njz | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8093 | |
| EPHA2 (EphA2) | Eph | TK | 5njz | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8085 | |
| EPHA2 (EphA2) | Eph | TK | 5nk0 | A | A | 2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8095 | |
| EPHA2 (EphA2) | Eph | TK | 5nk0 | A | B | 2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8096 | |
| EPHA2 (EphA2) | Eph | TK | 5nk1 | A | A | 2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8064 | |
| EPHA2 (EphA2) | Eph | TK | 5nk1 | A | B | 2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8059 | |
| EPHA2 (EphA2) | Eph | TK | 5nk2 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8100 | |
| EPHA2 (EphA2) | Eph | TK | 5nk2 | A | B | - | Human | 8060 | |
| EPHA2 (EphA2) | Eph | TK | 5nk2 | A | C | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8065 | |
| EPHA2 (EphA2) | Eph | TK | 5nk3 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8092 | |
| EPHA2 (EphA2) | Eph | TK | 5nk3 | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8080 | |
| EPHA2 (EphA2) | Eph | TK | 5nk4 | A | A | 2-[[3-[[(4~{r})-3,3-bis(fluoranyl)piperidin-4-yl]carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8070 | |
| EPHA2 (EphA2) | Eph | TK | 5nk4 | A | B | 2-[[3-[[(4~{r})-3,3-bis(fluoranyl)piperidin-4-yl]carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8076 | |
| EPHA2 (EphA2) | Eph | TK | 5nk5 | A | A | 2-[[3-[(3-aminophenyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8068 | |
| EPHA2 (EphA2) | Eph | TK | 5nk5 | A | B | 2-[[3-[(3-aminophenyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8066 | |
| EPHA2 (EphA2) | Eph | TK | 5nk5 | A | C | - | Human | 8091 | |
| EPHA2 (EphA2) | Eph | TK | 5nk6 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(4-oxidanylcyclohexyl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8094 | |
| EPHA2 (EphA2) | Eph | TK | 5nk6 | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(4-oxidanylcyclohexyl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8061 | |
| EPHA2 (EphA2) | Eph | TK | 5nk7 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8089 | |
| EPHA2 (EphA2) | Eph | TK | 5nk7 | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8081 | |
| EPHA2 (EphA2) | Eph | TK | 5nk8 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(2,2,6,6-tetramethyl-1-oxidanyl-piperidin-4-yl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8062 | |
| EPHA2 (EphA2) | Eph | TK | 5nk8 | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(2,2,6,6-tetramethyl-1-oxidanyl-piperidin-4-yl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8088 | |
| EPHA2 (EphA2) | Eph | TK | 5nk9 | A | A | (2~{z})-~{n}-(2-chloranyl-6-methyl-phenyl)-2-[3-[(4-methyl-4-oxidanyl-cyclohexyl)carbamoyl]phenyl]imino-1,3-thiazolidine-5-carboxamide | Human | 8073 | |
| EPHA2 (EphA2) | Eph | TK | 5nk9 | A | B | (2~{z})-~{n}-(2-chloranyl-6-methyl-phenyl)-2-[3-[(4-methyl-4-oxidanyl-cyclohexyl)carbamoyl]phenyl]imino-1,3-thiazolidine-5-carboxamide | Human | 8067 | |
| EPHA2 (EphA2) | Eph | TK | 5nka | A | A | 4-[[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylamino]cyclohexane-1-carboxylic acid | Human | 8075 | |
| EPHA2 (EphA2) | Eph | TK | 5nka | A | B | 4-[[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylamino]cyclohexane-1-carboxylic acid | Human | 8086 | |
| EPHA2 (EphA2) | Eph | TK | 5nka | A | C | - | Human | 8083 | |
| EPHA2 (EphA2) | Eph | TK | 5nkb | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3,5-dimorpholin-4-ylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 8098 | |
| EPHA2 (EphA2) | Eph | TK | 5nkb | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3,5-dimorpholin-4-ylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 8097 | |
| EPHA2 (EphA2) | Eph | TK | 5nkc | A | A | (3~{s})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidine-3-carboxylic acid | Human | 8099 | |
| EPHA2 (EphA2) | Eph | TK | 5nkc | A | B | (3~{s})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidine-3-carboxylic acid | Human | 8072 | |
| EPHA2 (EphA2) | Eph | TK | 5nkd | A | A | 2-[(3~{r})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidin-3-yl]ethanoic acid | Human | 8058 | |
| EPHA2 (EphA2) | Eph | TK | 5nkd | A | B | 2-[(3~{r})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidin-3-yl]ethanoic acid | Human | 8082 | |
| EPHA2 (EphA2) | Eph | TK | 5nke | A | A | 2-[[3-bromanyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8078 | |
| EPHA2 (EphA2) | Eph | TK | 5nke | A | B | 2-[[3-bromanyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8063 | |
| EPHA2 (EphA2) | Eph | TK | 5nkf | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)-5-(trifluoromethyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8087 | |
| EPHA2 (EphA2) | Eph | TK | 5nkf | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)-5-(trifluoromethyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8071 | |
| EPHA2 (EphA2) | Eph | TK | 5nkg | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-ethyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8079 | |
| EPHA2 (EphA2) | Eph | TK | 5nkg | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-ethyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8090 | |
| EPHA2 (EphA2) | Eph | TK | 5nkh | A | A | 2-[[3-(2-aminophenyl)-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8074 | |
| EPHA2 (EphA2) | Eph | TK | 5nkh | A | B | 2-[[3-(2-aminophenyl)-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8077 | |
| EPHA2 (EphA2) | Eph | TK | 5nki | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]-1,3-thiazole-5-carboxamide | Human | 8084 | |
| EPHA2 (EphA2) | Eph | TK | 5nki | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]-1,3-thiazole-5-carboxamide | Human | 8069 | |
| EPHA2 (EphA2) | Eph | TK | 6fnf | A | A | 4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10417 | |
| EPHA2 (EphA2) | Eph | TK | 6fnf | A | B | 4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10420 | |
| EPHA2 (EphA2) | Eph | TK | 6fng | A | A | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10414 | |
| EPHA2 (EphA2) | Eph | TK | 6fng | A | B | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10416 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | A | A | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10422 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | A | B | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10418 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | B | A | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10421 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | B | B | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10413 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | C | A | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10415 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | C | B | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10419 | |
| EPHA2 (EphA2) | Eph | TK | 6hes | A | A | 4-methyl-3-[(2-pyridin-3-ylquinazolin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11550 | |
| EPHA2 (EphA2) | Eph | TK | 6hes | A | B | 4-methyl-3-[(2-pyridin-3-ylquinazolin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11566 | |
| EPHA2 (EphA2) | Eph | TK | 6hes | A | C | - | Human | 11554 | |
| EPHA2 (EphA2) | Eph | TK | 6het | A | A | ~{n}-(3-chlorophenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 11564 | |
| EPHA2 (EphA2) | Eph | TK | 6het | A | B | ~{n}-(3-chlorophenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 11560 | |
| EPHA2 (EphA2) | Eph | TK | 6het | A | C | - | Human | 11562 | |
| EPHA2 (EphA2) | Eph | TK | 6heu | A | A | 3-[(4,6-dipyridin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11563 | |
| EPHA2 (EphA2) | Eph | TK | 6heu | A | B | 3-[(4,6-dipyridin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11552 | |
| EPHA2 (EphA2) | Eph | TK | 6hev | A | A | 4-methyl-3-[(2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11561 | |
| EPHA2 (EphA2) | Eph | TK | 6hev | A | B | 4-methyl-3-[(2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11565 | |
| EPHA2 (EphA2) | Eph | TK | 6hew | A | A | 4-methyl-3-[(1-methyl-6-pyrimidin-5-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11549 | |
| EPHA2 (EphA2) | Eph | TK | 6hew | A | B | 4-methyl-3-[(1-methyl-6-pyrimidin-5-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11556 | |
| EPHA2 (EphA2) | Eph | TK | 6hew | A | C | - | Human | 11553 | |
| EPHA2 (EphA2) | Eph | TK | 6hex | A | A | 4-methyl-3-[(1-methyl-6-pyrazin-2-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11559 | |
| EPHA2 (EphA2) | Eph | TK | 6hex | A | B | 4-methyl-3-[(1-methyl-6-pyrazin-2-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11555 | |
| EPHA2 (EphA2) | Eph | TK | 6hex | A | C | - | Human | 11551 | |
| EPHA2 (EphA2) | Eph | TK | 6hey | A | A | 3-[(4,6-dipyridin-3-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11557 | |
| EPHA2 (EphA2) | Eph | TK | 6hey | A | B | 3-[(4,6-dipyridin-3-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11558 | |
| EPHA2 (EphA2) | Eph | TK | 6q7b | A | A | 3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11927 | |
| EPHA2 (EphA2) | Eph | TK | 6q7b | A | B | 3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11935 | |
| EPHA2 (EphA2) | Eph | TK | 6q7c | A | A | 3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpiperidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11931 | |
| EPHA2 (EphA2) | Eph | TK | 6q7c | A | B | 3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpiperidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11930 | |
| EPHA2 (EphA2) | Eph | TK | 6q7d | A | A | 3-[[4-imidazol-1-yl-6-(4-oxidanylpiperidin-1-yl)-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11937 | |
| EPHA2 (EphA2) | Eph | TK | 6q7d | A | B | 3-[[4-imidazol-1-yl-6-(4-oxidanylpiperidin-1-yl)-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11928 | |
| EPHA2 (EphA2) | Eph | TK | 6q7e | A | A | 3-[[4-imidazol-1-yl-6-[(3~{r})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11926 | |
| EPHA2 (EphA2) | Eph | TK | 6q7e | A | B | 3-[[4-imidazol-1-yl-6-[(3~{r})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11932 | |
| EPHA2 (EphA2) | Eph | TK | 6q7f | A | A | 3-[(4-imidazol-1-yl-6-piperazin-1-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11929 | |
| EPHA2 (EphA2) | Eph | TK | 6q7f | A | B | 3-[(4-imidazol-1-yl-6-piperazin-1-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11936 | |
| EPHA2 (EphA2) | Eph | TK | 6q7g | A | A | 3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11933 | |
| EPHA2 (EphA2) | Eph | TK | 6q7g | A | B | 3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11938 | |
| EPHA2 (EphA2) | Eph | TK | 6q7g | A | C | 3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11934 | |
| EPHA2 (EphA2) | Eph | TK | 7kja | A | A | phosphomethylphosphonic acid adenylate ester | Human | 13250 | |
| EPHA2 (EphA2) | Eph | TK | 7kja | A | B | phosphomethylphosphonic acid adenylate ester | Human | 13255 | |
| EPHA2 (EphA2) | Eph | TK | 7kja | B | A | phosphomethylphosphonic acid adenylate ester | Human | 13249 | |
| EPHA2 (EphA2) | Eph | TK | 7kja | B | B | phosphomethylphosphonic acid adenylate ester | Human | 13251 | |
| EPHA2 (EphA2) | Eph | TK | 7kjb | A | | - | Human | 13253 | |
| EPHA2 (EphA2) | Eph | TK | 7kjc | A | A | phosphomethylphosphonic acid adenylate ester | Human | 13257 | |
| EPHA2 (EphA2) | Eph | TK | 7kjc | A | B | phosphomethylphosphonic acid adenylate ester | Human | 13256 | |
| EPHA2 (EphA2) | Eph | TK | 7kjc | B | A | phosphomethylphosphonic acid adenylate ester | Human | 13252 | |
| EPHA2 (EphA2) | Eph | TK | 7kjc | B | B | phosphomethylphosphonic acid adenylate ester | Human | 13254 | |
| EPHA2 (EphA2) | Eph | TK | 8bin | A | A | 8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14514 | |
| EPHA2 (EphA2) | Eph | TK | 8bin | A | B | 8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14515 | |
| EPHA2 (EphA2) | Eph | TK | 8bin | A | C | 8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14512 | |
| EPHA2 (EphA2) | Eph | TK | 8bio | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-5-(trifluoromethyl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14513 | |
| EPHA2 (EphA2) | Eph | TK | 8bk0 | A | A | ~{n}-(2-chlorophenyl)-6-piperidin-4-yl-imidazo[1,2-a]pyridine-3-carboxamide | Human | 14504 | |
| EPHA2 (EphA2) | Eph | TK | 8bk0 | A | B | ~{n}-(2-chlorophenyl)-6-piperidin-4-yl-imidazo[1,2-a]pyridine-3-carboxamide | Human | 14503 | |
| EPHA2 (EphA2) | Eph | TK | 8boc | A | A | ~{n}-[3,5-bis(trifluoromethyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 15003 | |
| EPHA2 (EphA2) | Eph | TK | 8boc | A | B | ~{n}-[3,5-bis(trifluoromethyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 15002 | |
| EPHA2 (EphA2) | Eph | TK | 8bod | A | A | ~{n}-[3,5-bis(chloranyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14657 | |
| EPHA2 (EphA2) | Eph | TK | 8bod | A | B | ~{n}-[3,5-bis(chloranyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14646 | |
| EPHA2 (EphA2) | Eph | TK | 8bof | A | A | 4-methyl-~{n}-(3-methylphenyl)-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14656 | |
| EPHA2 (EphA2) | Eph | TK | 8bof | A | B | 4-methyl-~{n}-(3-methylphenyl)-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14652 | |
| EPHA2 (EphA2) | Eph | TK | 8bog | A | A | ~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamide | Human | 14650 | |
| EPHA2 (EphA2) | Eph | TK | 8bog | A | B | ~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamide | Human | 14649 | |
| EPHA2 (EphA2) | Eph | TK | 8bog | A | C | ~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamide | Human | 14654 | |
| EPHA2 (EphA2) | Eph | TK | 8boh | A | A | 4-methyl-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14647 | |
| EPHA2 (EphA2) | Eph | TK | 8boh | A | B | 4-methyl-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14651 | |
| EPHA2 (EphA2) | Eph | TK | 8boi | A | A | 4-methyl-~{n}-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14645 | |
| EPHA2 (EphA2) | Eph | TK | 8boi | A | B | 4-methyl-~{n}-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14655 | |
| EPHA2 (EphA2) | Eph | TK | 8bok | A | A | ~{n}-(3,5-dimethoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14648 | |
| EPHA2 (EphA2) | Eph | TK | 8bok | A | B | ~{n}-(3,5-dimethoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14659 | |
| EPHA2 (EphA2) | Eph | TK | 8bom | A | A | ~{n}-(3-methoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14658 | |
| EPHA2 (EphA2) | Eph | TK | 8bom | A | B | ~{n}-(3-methoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14653 | |
| EPHA2 (EphA2) | Eph | TK | 8qqy | A | A | 6-(4-fluoranyl-3-methoxy-phenyl)-13$l^{6}-thia-2,4,8,12,19-pentazatricyclo[12.3.1.1^{3,7}]nonadeca-1(18),3,5,7(19),14,16-hexaene 13,13-dioxide | Human | 15001 | |
| EPHA2 (EphA2) | Eph | TK | 8qqy | A | B | 6-(4-fluoranyl-3-methoxy-phenyl)-13$l^{6}-thia-2,4,8,12,19-pentazatricyclo[12.3.1.1^{3,7}]nonadeca-1(18),3,5,7(19),14,16-hexaene 13,13-dioxide | Human | 15000 | |
| EPHA2 (EphA2) | Eph | TK | 8xpv | A | A | 1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}urea | Human | 15134 | |
| EPHA2 (EphA2) | Eph | TK | 8xpv | A | B | 1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}urea | Human | 15135 | |
| EPHA3 (EphA3) | Eph | TK | 2gsf | A | | - | Human | 2861 | |
| EPHA3 (EphA3) | Eph | TK | 2qo2 | A | A | - | Human | 2880 | |
| EPHA3 (EphA3) | Eph | TK | 2qo2 | A | B | - | Human | 2886 | |
| EPHA3 (EphA3) | Eph | TK | 2qo7 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2874 | |
| EPHA3 (EphA3) | Eph | TK | 2qo7 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2857 | |
| EPHA3 (EphA3) | Eph | TK | 2qo7 | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 2839 | |
| EPHA3 (EphA3) | Eph | TK | 2qo9 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2862 | |
| EPHA3 (EphA3) | Eph | TK | 2qo9 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2864 | |
| EPHA3 (EphA3) | Eph | TK | 2qob | A | A | - | Human | 2889 | |
| EPHA3 (EphA3) | Eph | TK | 2qob | A | B | - | Human | 2872 | |
| EPHA3 (EphA3) | Eph | TK | 2qob | A | C | - | Human | 2850 | |
| EPHA3 (EphA3) | Eph | TK | 2qoc | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2882 | |
| EPHA3 (EphA3) | Eph | TK | 2qoc | A | B | - | Human | 2856 | |
| EPHA3 (EphA3) | Eph | TK | 2qoc | A | C | - | Human | 2871 | |
| EPHA3 (EphA3) | Eph | TK | 2qod | A | A | - | Human | 2869 | |
| EPHA3 (EphA3) | Eph | TK | 2qod | A | B | - | Human | 2842 | |
| EPHA3 (EphA3) | Eph | TK | 2qod | A | C | - | Human | 2866 | |
| EPHA3 (EphA3) | Eph | TK | 2qof | A | A | - | Human | 2888 | |
| EPHA3 (EphA3) | Eph | TK | 2qof | A | B | - | Human | 2859 | |
| EPHA3 (EphA3) | Eph | TK | 2qof | A | C | - | Human | 2870 | |
| EPHA3 (EphA3) | Eph | TK | 2qoi | A | A | - | Human | 2855 | |
| EPHA3 (EphA3) | Eph | TK | 2qoi | A | B | - | Human | 2891 | |
| EPHA3 (EphA3) | Eph | TK | 2qok | A | A | - | Human | 2873 | |
| EPHA3 (EphA3) | Eph | TK | 2qok | A | B | - | Human | 2876 | |
| EPHA3 (EphA3) | Eph | TK | 2qok | A | C | - | Human | 2884 | |
| EPHA3 (EphA3) | Eph | TK | 2qol | A | A | - | Human | 2863 | |
| EPHA3 (EphA3) | Eph | TK | 2qol | A | B | - | Human | 2836 | |
| EPHA3 (EphA3) | Eph | TK | 2qol | A | C | - | Human | 2845 | |
| EPHA3 (EphA3) | Eph | TK | 2qol | A | D | - | Human | 2877 | |
| EPHA3 (EphA3) | Eph | TK | 2qon | A | A | - | Human | 2867 | |
| EPHA3 (EphA3) | Eph | TK | 2qon | A | B | - | Human | 2853 | |
| EPHA3 (EphA3) | Eph | TK | 2qoo | A | A | - | Human | 2847 | |
| EPHA3 (EphA3) | Eph | TK | 2qoo | A | B | - | Human | 2881 | |
| EPHA3 (EphA3) | Eph | TK | 2qoq | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2890 | |
| EPHA3 (EphA3) | Eph | TK | 2qoq | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2849 | |
| EPHA3 (EphA3) | Eph | TK | 2qoq | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 2879 | |
| EPHA3 (EphA3) | Eph | TK | 3dzq | A | A | n-[2-methyl-5-({[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamide | Human | 2852 | |
| EPHA3 (EphA3) | Eph | TK | 3dzq | A | B | n-[2-methyl-5-({[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamide | Human | 2868 | |
| EPHA3 (EphA3) | Eph | TK | 3fxx | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2883 | |
| EPHA3 (EphA3) | Eph | TK | 3fxx | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2860 | |
| EPHA3 (EphA3) | Eph | TK | 3fy2 | A | A | - | Human | 2851 | |
| EPHA3 (EphA3) | Eph | TK | 3fy2 | A | B | - | Human | 2837 | |
| EPHA3 (EphA3) | Eph | TK | 4g2f | A | A | 1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-one | Human | 2843 | |
| EPHA3 (EphA3) | Eph | TK | 4g2f | A | B | 1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-one | Human | 2838 | |
| EPHA3 (EphA3) | Eph | TK | 4gk2 | A | A | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2841 | |
| EPHA3 (EphA3) | Eph | TK | 4gk2 | A | B | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2858 | |
| EPHA3 (EphA3) | Eph | TK | 4gk3 | A | A | 8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2844 | |
| EPHA3 (EphA3) | Eph | TK | 4gk3 | A | B | 8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2885 | |
| EPHA3 (EphA3) | Eph | TK | 4gk4 | A | A | 8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2854 | |
| EPHA3 (EphA3) | Eph | TK | 4gk4 | A | B | 8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2840 | |
| EPHA3 (EphA3) | Eph | TK | 4p4c | A | | 2-amino-1-(3-methoxyphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 2875 | |
| EPHA3 (EphA3) | Eph | TK | 4p5q | A | A | 2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 2892 | |
| EPHA3 (EphA3) | Eph | TK | 4p5q | A | B | 2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 2878 | |
| EPHA3 (EphA3) | Eph | TK | 4p5z | A | | 2-amino-1-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenyl]-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 2887 | |
| EPHA3 (EphA3) | Eph | TK | 4twn | A | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 2846 | |
| EPHA3 (EphA3) | Eph | TK | 4twn | A | B | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 2865 | |
| EPHA3 (EphA3) | Eph | TK | 4two | A | A | 5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acid | Human | 2893 | |
| EPHA3 (EphA3) | Eph | TK | 4two | A | B | 5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acid | Human | 2848 | |
| EPHA3 (EphA3) | Eph | TK | 6in0 | A | A | 1,4,7,10,13,16-hexaoxacyclooctadecane | Human | 11792 | |
| EPHA3 (EphA3) | Eph | TK | 6in0 | A | B | 1,4,7,10,13,16-hexaoxacyclooctadecane | Human | 11793 | |
| Epha4 (EphA4) | Eph | TK | 2hel | A | | - | Mouse | 5812 | |
| Epha4 (EphA4) | Eph | TK | 2xyu | A | | 5-(5-fluoro-2-methylphenyl)-6,7,8,9-tetrahydro-3h-pyrazolo[3,4-c]isoquinolin-1-amine | Mouse | 5810 | |
| Epha4 (EphA4) | Eph | TK | 2y6m | A | A | - | Mouse | 5809 | |
| Epha4 (EphA4) | Eph | TK | 2y6m | A | B | - | Mouse | 5813 | |
| Epha4 (EphA4) | Eph | TK | 2y6o | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5814 | |
| Epha4 (EphA4) | Eph | TK | 2y6o | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5811 | |
| EPHA5 (EphA5) | Eph | TK | 2r2p | A | A | - | Human | 3412 | |
| EPHA5 (EphA5) | Eph | TK | 2r2p | A | B | - | Human | 3413 | |
| EPHA7 (EphA7) | Eph | TK | 2rei | A | A | - | Human | 4 | |
| EPHA7 (EphA7) | Eph | TK | 2rei | A | B | - | Human | 2 | |
| EPHA7 (EphA7) | Eph | TK | 3dko | A | A | 5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamide | Human | 1 | |
| EPHA7 (EphA7) | Eph | TK | 3dko | A | B | 5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamide | Human | 3 | |
| EPHA7 (EphA7) | Eph | TK | 7eec | A | A | - | Human | 13792 | |
| EPHA7 (EphA7) | Eph | TK | 7eec | A | B | - | Human | 13790 | |
| EPHA7 (EphA7) | Eph | TK | 7eed | A | | - | Human | 13791 | |
| EPHA7 (EphA7) | Eph | TK | 7eef | A | | - | Human | 13793 | |
| EPHA8 (EphA8) | Eph | TK | 3kul | A | A | - | Human | 1251 | |
| EPHA8 (EphA8) | Eph | TK | 3kul | A | B | - | Human | 1252 | |
| EPHA8 (EphA8) | Eph | TK | 3kul | B | A | - | Human | 1249 | |
| EPHA8 (EphA8) | Eph | TK | 3kul | B | B | - | Human | 1250 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | A | | - | Human | 560 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | B | | - | Human | 558 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | C | | - | Human | 557 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | D | | - | Human | 552 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | E | | - | Human | 555 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | F | | - | Human | 553 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | G | | - | Human | 554 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | H | | - | Human | 556 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | I | | - | Human | 559 | |
| EPHB1 (EphB1) | Eph | TK | 5mja | A | | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | 7582 | |
| EPHB1 (EphB1) | Eph | TK | 5mja | B | | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | 7583 | |
| EPHB1 (EphB1) | Eph | TK | 5mjb | A | | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | 7584 | |
| EPHB1 (EphB1) | Eph | TK | 5mjb | B | | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | 7585 | |
| EPHB1 (EphB1) | Eph | TK | 6umw | A | A | - | Human | 12924 | |
| EPHB1 (EphB1) | Eph | TK | 6umw | A | B | - | Human | 12923 | |
| EPHB1 (EphB1) | Eph | TK | 7kpl | A | A | - | Human | 13384 | |
| EPHB1 (EphB1) | Eph | TK | 7kpl | A | B | - | Human | 13383 | |
| EPHB1 (EphB1) | Eph | TK | 7kpm | A | A | adenosine-5'-diphosphate | Human | 13385 | |
| EPHB1 (EphB1) | Eph | TK | 7kpm | A | B | adenosine-5'-diphosphate | Human | 13382 | |
| Ephb2 (EphB2) | Eph | TK | 1jpa | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5806 | |
| Ephb2 (EphB2) | Eph | TK | 1jpa | B | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5805 | |
| Ephb2 (EphB2) | Eph | TK | 2hen | A | | adenosine-5'-diphosphate | Mouse | 5807 | |
| Ephb2 (EphB2) | Eph | TK | 2hen | B | | adenosine-5'-diphosphate | Mouse | 5804 | |
| Ephb2 (EphB2) | Eph | TK | 2hen | C | | adenosine-5'-diphosphate | Mouse | 5808 | |
| Ephb2 (EphB2) | Eph | TK | 2hen | D | | adenosine-5'-diphosphate | Mouse | 5803 | |
| EPHB2 (EphB2) | Eph | TK | 3zfm | A | | - | Human | 2731 | |
| EPHB3 (EphB3) | Eph | TK | 3zfy | A | A | - | Human | 537 | |
| EPHB3 (EphB3) | Eph | TK | 3zfy | A | B | - | Human | 538 | |
| EPHB3 (EphB3) | Eph | TK | 3zfy | B | A | - | Human | 539 | |
| EPHB3 (EphB3) | Eph | TK | 3zfy | B | B | - | Human | 536 | |
| EPHB3 (EphB3) | Eph | TK | 5l6o | A | | 1-(4-phenylazanylquinazolin-7-yl)ethanone | Human | 6938 | |
| EPHB3 (EphB3) | Eph | TK | 5l6p | A | | ~{n}-(4-phenylazanylquinazolin-7-yl)ethanamide | Human | 6937 | |
| EPHB4 (EphB4) | Eph | TK | 2vwu | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin-4-amine | Human | 370 | |
| EPHB4 (EphB4) | Eph | TK | 2vwv | A | A | n'-(3-chloro-4-methoxy-phenyl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazine-2,4-diamine | Human | 365 | |
| EPHB4 (EphB4) | Eph | TK | 2vwv | A | B | n'-(3-chloro-4-methoxy-phenyl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazine-2,4-diamine | Human | 369 | |
| EPHB4 (EphB4) | Eph | TK | 2vww | A | A | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3,4,5- trimethoxyphenyl)pyrimidine-2,4-diamine | Human | 356 | |
| EPHB4 (EphB4) | Eph | TK | 2vww | A | B | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3,4,5- trimethoxyphenyl)pyrimidine-2,4-diamine | Human | 358 | |
| EPHB4 (EphB4) | Eph | TK | 2vwx | A | A | 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 361 | |
| EPHB4 (EphB4) | Eph | TK | 2vwx | A | B | 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 350 | |
| EPHB4 (EphB4) | Eph | TK | 2vwy | A | A | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-methylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 353 | |
| EPHB4 (EphB4) | Eph | TK | 2vwy | A | B | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-methylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 355 | |
| EPHB4 (EphB4) | Eph | TK | 2vwz | A | A | n-[3-[[4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl]amino]phenyl]methanesulfonamide | Human | 360 | |
| EPHB4 (EphB4) | Eph | TK | 2vwz | A | B | n-[3-[[4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl]amino]phenyl]methanesulfonamide | Human | 362 | |
| EPHB4 (EphB4) | Eph | TK | 2vx0 | A | A | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-morpholin-4-ylphenyl)pyrimidine-2,4-diamine | Human | 375 | |
| EPHB4 (EphB4) | Eph | TK | 2vx0 | A | B | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-morpholin-4-ylphenyl)pyrimidine-2,4-diamine | Human | 368 | |
| EPHB4 (EphB4) | Eph | TK | 2vx1 | A | A | 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzamide | Human | 371 | |
| EPHB4 (EphB4) | Eph | TK | 2vx1 | A | B | 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzamide | Human | 374 | |
| EPHB4 (EphB4) | Eph | TK | 2x9f | A | A | n^4^-1h-indazol-4-yl-n^2^-[3-(methylsulfonyl)phenyl]pyrimidine-2,4-diamine | Human | 354 | |
| EPHB4 (EphB4) | Eph | TK | 2x9f | A | B | n^4^-1h-indazol-4-yl-n^2^-[3-(methylsulfonyl)phenyl]pyrimidine-2,4-diamine | Human | 359 | |
| EPHB4 (EphB4) | Eph | TK | 2xvd | A | A | {4-methyl-3-[(1-methylethyl)(2-{[3-(methylsulfonyl)-5-morpholin-4-ylphenyl]amino}pyrimidin-4-yl)amino]phenyl}methanol | Human | 363 | |
| EPHB4 (EphB4) | Eph | TK | 2xvd | A | B | {4-methyl-3-[(1-methylethyl)(2-{[3-(methylsulfonyl)-5-morpholin-4-ylphenyl]amino}pyrimidin-4-yl)amino]phenyl}methanol | Human | 372 | |
| EPHB4 (EphB4) | Eph | TK | 2yn8 | A | | staurosporine | Human | 352 | |
| EPHB4 (EphB4) | Eph | TK | 2yn8 | B | | staurosporine | Human | 349 | |
| EPHB4 (EphB4) | Eph | TK | 3zew | A | A | staurosporine | Human | 373 | |
| EPHB4 (EphB4) | Eph | TK | 3zew | A | B | staurosporine | Human | 377 | |
| EPHB4 (EphB4) | Eph | TK | 3zew | B | A | staurosporine | Human | 351 | |
| EPHB4 (EphB4) | Eph | TK | 3zew | B | B | staurosporine | Human | 357 | |
| EPHB4 (EphB4) | Eph | TK | 4aw5 | A | A | (3z)-5-[(1-ethylpiperidin-4-yl)amino]-3-[(5-methoxy-1h-benzimidazol-2-yl)(phenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 367 | |
| EPHB4 (EphB4) | Eph | TK | 4aw5 | A | B | (3z)-5-[(1-ethylpiperidin-4-yl)amino]-3-[(5-methoxy-1h-benzimidazol-2-yl)(phenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 376 | |
| EPHB4 (EphB4) | Eph | TK | 4bb4 | A | A | n-(2-methoxyethyl)-4-[(6-pyridin-4-ylquinazolin-2-yl)amino]benzamide | Human | 364 | |
| EPHB4 (EphB4) | Eph | TK | 4bb4 | A | B | n-(2-methoxyethyl)-4-[(6-pyridin-4-ylquinazolin-2-yl)amino]benzamide | Human | 366 | |
| EPHB4 (EphB4) | Eph | TK | 6fni | A | A | 4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10338 | |
| EPHB4 (EphB4) | Eph | TK | 6fni | A | B | 4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10333 | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | A | A | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10336 | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | A | B | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10334 | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | B | A | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10340 | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | B | B | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10341 | |
| EPHB4 (EphB4) | Eph | TK | 6fnk | A | A | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10344 | |
| EPHB4 (EphB4) | Eph | TK | 6fnk | A | B | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10337 | |
| EPHB4 (EphB4) | Eph | TK | 6fnl | A | A | - | Human | 10343 | |
| EPHB4 (EphB4) | Eph | TK | 6fnl | A | B | - | Human | 10335 | |
| EPHB4 (EphB4) | Eph | TK | 6fnm | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 10342 | |
| EPHB4 (EphB4) | Eph | TK | 6fnm | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 10339 | |
| ERBB2 (ErbB2) | EGFR | TK | 3pp0 | A | A | 2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanol | Human | 4815 | |
| ERBB2 (ErbB2) | EGFR | TK | 3pp0 | A | B | 2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanol | Human | 4820 | |
| ERBB2 (ErbB2) | EGFR | TK | 3pp0 | B | A | 2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanol | Human | 4816 | |
| ERBB2 (ErbB2) | EGFR | TK | 3pp0 | B | B | 2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanol | Human | 4819 | |
| ERBB2 (ErbB2) | EGFR | TK | 3rcd | A | | n-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamide | Human | 9325 | |
| ERBB2 (ErbB2) | EGFR | TK | 3rcd | B | | - | Human | 9322 | |
| ERBB2 (ErbB2) | EGFR | TK | 3rcd | C | | n-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamide | Human | 9323 | |
| ERBB2 (ErbB2) | EGFR | TK | 3rcd | D | | - | Human | 9324 | |
| ERBB2 (ErbB2) | EGFR | TK | 7jxh | A | A | (2e)-n-[3-cyano-7-ethoxy-4-({3-methyl-4-[([1,2,4]triazolo[1,5-a]pyridin-7-yl)oxy]phenyl}amino)quinolin-6-yl]-4-(dimethylamino)but-2-enamide | Human | 13888 | |
| ERBB2 (ErbB2) | EGFR | TK | 7jxh | A | B | (2e)-n-[3-cyano-7-ethoxy-4-({3-methyl-4-[([1,2,4]triazolo[1,5-a]pyridin-7-yl)oxy]phenyl}amino)quinolin-6-yl]-4-(dimethylamino)but-2-enamide | Human | 13887 | |
| ERBB2 (ErbB2) | EGFR | TK | 7pcd | A | A | 1-[4-[4-[[3,5-bis(chloranyl)-4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)phenyl]amino]pyrimido[5,4-d]pyrimidin-6-yl]piperazin-1-yl]-4-(3-fluoranylazetidin-1-yl)butan-1-one | Human | 14320 | |
| ERBB2 (ErbB2) | EGFR | TK | 7pcd | A | B | 1-[4-[4-[[3,5-bis(chloranyl)-4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)phenyl]amino]pyrimido[5,4-d]pyrimidin-6-yl]piperazin-1-yl]-4-(3-fluoranylazetidin-1-yl)butan-1-one | Human | 14319 | |
| ERBB2 (ErbB2) | EGFR | TK | 8u8x | A | A | 1-{(1r,3r,5s)-3-[(3m)-4-methyl-3-{3-methyl-4-[(1-methyl-1h-benzimidazol-5-yl)oxy]phenyl}-1h-pyrazolo[3,4-d]pyrimidin-1-yl]-8-azabicyclo[3.2.1]octan-8-yl}propan-1-one | Human | 15345 | |
| ERBB2 (ErbB2) | EGFR | TK | 8u8x | A | B | 1-{(1r,3r,5s)-3-[(3m)-4-methyl-3-{3-methyl-4-[(1-methyl-1h-benzimidazol-5-yl)oxy]phenyl}-1h-pyrazolo[3,4-d]pyrimidin-1-yl]-8-azabicyclo[3.2.1]octan-8-yl}propan-1-one | Human | 15344 | |
| ERBB3 (ErbB3) | EGFR | TK | 3kex | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1939 | |
| ERBB3 (ErbB3) | EGFR | TK | 3kex | B | | phosphoaminophosphonic acid-adenylate ester | Human | 1933 | |
| ERBB3 (ErbB3) | EGFR | TK | 3lmg | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1935 | |
| ERBB3 (ErbB3) | EGFR | TK | 3lmg | B | | phosphoaminophosphonic acid-adenylate ester | Human | 1936 | |
| ERBB3 (ErbB3) | EGFR | TK | 4riw | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1930 | |
| ERBB3 (ErbB3) | EGFR | TK | 4riw | C | | phosphoaminophosphonic acid-adenylate ester | Human | 1932 | |
| ERBB3 (ErbB3) | EGFR | TK | 4rix | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1931 | |
| ERBB3 (ErbB3) | EGFR | TK | 4rix | C | | phosphoaminophosphonic acid-adenylate ester | Human | 1934 | |
| ERBB3 (ErbB3) | EGFR | TK | 4riy | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1937 | |
| ERBB3 (ErbB3) | EGFR | TK | 4riy | C | | phosphoaminophosphonic acid-adenylate ester | Human | 1938 | |
| ERBB3 (ErbB3) | EGFR | TK | 6op9 | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 11545 | |
| ERBB3 (ErbB3) | EGFR | TK | 6op9 | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 11544 | |
| ERBB3 (ErbB3) | EGFR | TK | 7mn5 | A | | - | Human | 13953 | |
| ERBB3 (ErbB3) | EGFR | TK | 7mn6 | A | | - | Human | 13952 | |
| ERBB3 (ErbB3) | EGFR | TK | 7mn8 | A | | - | Human | 13966 | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | A | A | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | 2822 | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | A | B | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | 2827 | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | B | A | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | 2818 | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | B | B | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | 2823 | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbt | B | | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamine | Human | 2825 | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbt | D | | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamine | Human | 2819 | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbw | A | | - | Human | 2820 | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbw | B | | - | Human | 2817 | |
| ERBB4 (ErbB4) | EGFR | TK | 3bce | A | | - | Human | 2821 | |
| ERBB4 (ErbB4) | EGFR | TK | 3bce | B | | - | Human | 2826 | |
| ERBB4 (ErbB4) | EGFR | TK | 3bce | C | | - | Human | 2824 | |
| Ern1 (IRE1) | IRE | Other | 4pl3 | A | | adenosine-5'-diphosphate | Mouse | 5769 | |
| Ern1 (IRE1) | IRE | Other | 4pl3 | B | | adenosine-5'-diphosphate | Mouse | 5768 | |
| Ern1 (IRE1) | IRE | Other | 4pl4 | A | | adenosine-5'-diphosphate | Mouse | 5770 | |
| Ern1 (IRE1) | IRE | Other | 4pl4 | B | | adenosine-5'-diphosphate | Mouse | 5767 | |
| Ern1 (IRE1) | IRE | Other | 4pl4 | C | | adenosine-5'-diphosphate | Mouse | 5761 | |
| Ern1 (IRE1) | IRE | Other | 4pl4 | D | | adenosine-5'-diphosphate | Mouse | 5765 | |
| Ern1 (IRE1) | IRE | Other | 4pl5 | A | | adenosine-5'-diphosphate | Mouse | 5762 | |
| Ern1 (IRE1) | IRE | Other | 4pl5 | B | | adenosine-5'-diphosphate | Mouse | 5764 | |
| Ern1 (IRE1) | IRE | Other | 4pl5 | C | | adenosine-5'-diphosphate | Mouse | 5766 | |
| Ern1 (IRE1) | IRE | Other | 4pl5 | D | | adenosine-5'-diphosphate | Mouse | 5763 | |
| ERN1 (IRE1) | IRE | Other | 3p23 | A | | adenosine-5'-diphosphate | Human | 1795 | |
| ERN1 (IRE1) | IRE | Other | 3p23 | B | | adenosine-5'-diphosphate | Human | 1797 | |
| ERN1 (IRE1) | IRE | Other | 3p23 | C | | adenosine-5'-diphosphate | Human | 1798 | |
| ERN1 (IRE1) | IRE | Other | 3p23 | D | | adenosine-5'-diphosphate | Human | 1800 | |
| ERN1 (IRE1) | IRE | Other | 4u6r | A | | n-{4-[(3-{2-[(trans-4-aminocyclohexyl)amino]pyrimidin-4-yl}pyridin-2-yl)oxy]-3-methylnaphthalen-1-yl}-2-chlorobenzenesulfonamide | Human | 1802 | |
| ERN1 (IRE1) | IRE | Other | 4yz9 | A | A | (5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamide | Human | 6233 | |
| ERN1 (IRE1) | IRE | Other | 4yz9 | A | B | (5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamide | Human | 6224 | |
| ERN1 (IRE1) | IRE | Other | 4yz9 | B | A | (5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamide | Human | 6225 | |
| ERN1 (IRE1) | IRE | Other | 4yz9 | B | B | (5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamide | Human | 6229 | |
| ERN1 (IRE1) | IRE | Other | 4yz9 | C | A | (5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamide | Human | 6223 | |
| ERN1 (IRE1) | IRE | Other | 4yz9 | C | B | (5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamide | Human | 6222 | |
| ERN1 (IRE1) | IRE | Other | 4yzc | A | A | staurosporine | Human | 6235 | |
| ERN1 (IRE1) | IRE | Other | 4yzc | A | B | staurosporine | Human | 6232 | |
| ERN1 (IRE1) | IRE | Other | 4yzc | B | A | staurosporine | Human | 6227 | |
| ERN1 (IRE1) | IRE | Other | 4yzc | B | B | staurosporine | Human | 6231 | |
| ERN1 (IRE1) | IRE | Other | 4yzd | A | A | adenosine-5'-diphosphate | Human | 6234 | |
| ERN1 (IRE1) | IRE | Other | 4yzd | A | B | adenosine-5'-diphosphate | Human | 6228 | |
| ERN1 (IRE1) | IRE | Other | 4yzd | B | A | adenosine-5'-diphosphate | Human | 6236 | |
| ERN1 (IRE1) | IRE | Other | 4yzd | B | B | adenosine-5'-diphosphate | Human | 6230 | |
| ERN1 (IRE1) | IRE | Other | 4yzd | C | A | adenosine-5'-diphosphate | Human | 6237 | |
| ERN1 (IRE1) | IRE | Other | 4yzd | C | B | adenosine-5'-diphosphate | Human | 6226 | |
| ERN1 (IRE1) | IRE | Other | 4z7g | A | | - | Human | 1799 | |
| ERN1 (IRE1) | IRE | Other | 4z7g | B | | - | Human | 1796 | |
| ERN1 (IRE1) | IRE | Other | 4z7h | A | | 2-methoxy-4-[6-(propan-2-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 1794 | |
| ERN1 (IRE1) | IRE | Other | 4z7h | B | | 2-methoxy-4-[6-(propan-2-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 1801 | |
| ERN1 (IRE1) | IRE | Other | 5hgi | A | | - | Human | 6669 | |
| ERN1 (IRE1) | IRE | Other | 6hv0 | A | | 6-chloranyl-3-(2~{h}-indazol-5-yl)-~{n}-propan-2-yl-imidazo[1,2-b]pyridazin-8-amine | Human | 10928 | |
| ERN1 (IRE1) | IRE | Other | 6hx1 | A | A | 6-chloranyl-~{n}-(cyclopropylmethyl)-3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-8-amine | Human | 10927 | |
| ERN1 (IRE1) | IRE | Other | 6hx1 | A | B | 6-chloranyl-~{n}-(cyclopropylmethyl)-3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-8-amine | Human | 10929 | |
| ERN1 (IRE1) | IRE | Other | 6urc | A | | 2-chloro-n-(6-methyl-5-{[3-(2-{[(3s)-piperidin-3-yl]amino}pyrimidin-4-yl)pyridin-2-yl]oxy}naphthalen-1-yl)benzene-1-sulfonamide | Human | 11799 | |
| ERN1 (IRE1) | IRE | Other | 6urc | B | | 2-chloro-n-(6-methyl-5-{[3-(2-{[(3s)-piperidin-3-yl]amino}pyrimidin-4-yl)pyridin-2-yl]oxy}naphthalen-1-yl)benzene-1-sulfonamide | Human | 11798 | |
| ERN1 (IRE1) | IRE | Other | 6w39 | A | A | ethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamate | Human | 13120 | |
| ERN1 (IRE1) | IRE | Other | 6w39 | A | B | ethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamate | Human | 13122 | |
| ERN1 (IRE1) | IRE | Other | 6w39 | B | A | ethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamate | Human | 13117 | |
| ERN1 (IRE1) | IRE | Other | 6w39 | B | B | ethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamate | Human | 13124 | |
| ERN1 (IRE1) | IRE | Other | 6w3a | A | A | ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]but-2-ynamide | Human | 13125 | |
| ERN1 (IRE1) | IRE | Other | 6w3a | A | B | ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]but-2-ynamide | Human | 13116 | |
| ERN1 (IRE1) | IRE | Other | 6w3a | B | A | ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]but-2-ynamide | Human | 13118 | |
| ERN1 (IRE1) | IRE | Other | 6w3a | B | B | ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]but-2-ynamide | Human | 13119 | |
| ERN1 (IRE1) | IRE | Other | 6w3b | A | | - | Human | 13039 | |
| ERN1 (IRE1) | IRE | Other | 6w3c | A | | - | Human | 13040 | |
| ERN1 (IRE1) | IRE | Other | 6w3c | B | | - | Human | 13038 | |
| ERN1 (IRE1) | IRE | Other | 6w3c | C | | - | Human | 13036 | |
| ERN1 (IRE1) | IRE | Other | 6w3c | D | | - | Human | 13037 | |
| ERN1 (IRE1) | IRE | Other | 6w3e | A | | methyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamate | Human | 13121 | |
| ERN1 (IRE1) | IRE | Other | 6w3e | B | | methyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamate | Human | 13126 | |
| ERN1 (IRE1) | IRE | Other | 6w3k | A | | 4-[5-[2,6-bis(fluoranyl)phenyl]-2~{h}-pyrazolo[3,4-b]pyridin-3-yl]-2-(4-oxidanylpiperidin-1-yl)-1~{h}-pyrimidin-6-one | Human | 13123 | |
| ERN1 (IRE1) | IRE | Other | 6xdb | A | | 4-amino-n-(6-chloro-2-fluoro-3-{[(2-fluorophenyl)sulfonyl]amino}phenyl)-6-(1,3-dimethyl-1h-pyrazol-4-yl)quinazoline-8-carboxamide | Human | 13531 | |
| ERN1 (IRE1) | IRE | Other | 6xdd | A | | 4-[(trans-4-aminocyclohexyl)amino]-n-(6-chloro-3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)thieno[3,2-d]pyrimidine-7-carboxamide | Human | 13529 | |
| ERN1 (IRE1) | IRE | Other | 6xdd | B | | 4-[(trans-4-aminocyclohexyl)amino]-n-(6-chloro-3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)thieno[3,2-d]pyrimidine-7-carboxamide | Human | 13530 | |
| ERN1 (IRE1) | IRE | Other | 6xdf | B | A | - | Human | 13508 | |
| ERN1 (IRE1) | IRE | Other | 6xdf | B | B | - | Human | 13507 | |
| ERN1 (IRE1) | IRE | Other | 7bmk | A | A | 2,2,2-tris(fluoranyl)-~{n}-[4-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxynaphthalen-1-yl]ethanesulfonamide | Human | 13911 | |
| ERN1 (IRE1) | IRE | Other | 7bmk | A | B | 2,2,2-tris(fluoranyl)-~{n}-[4-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxynaphthalen-1-yl]ethanesulfonamide | Human | 13912 | |
| FES | Fer | TK | 3bkb | A | A | staurosporine | Human | 2810 | |
| FES | Fer | TK | 3bkb | A | B | staurosporine | Human | 2813 | |
| FES | Fer | TK | 3bkb | A | C | staurosporine | Human | 2812 | |
| FES | Fer | TK | 3cbl | A | A | staurosporine | Human | 2808 | |
| FES | Fer | TK | 3cbl | A | B | staurosporine | Human | 2811 | |
| FES | Fer | TK | 3cd3 | A | A | staurosporine | Human | 2814 | |
| FES | Fer | TK | 3cd3 | A | B | staurosporine | Human | 2815 | |
| FES | Fer | TK | 4e93 | A | A | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 2816 | |
| FES | Fer | TK | 4e93 | A | B | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 2809 | |
| FES | Fer | TK | 6jmf | A | | 6-{[(1r,2s)-2-aminocyclohexyl]amino}-5-cyano-2-[(3-methylphenyl)amino]pyridine-3-carboxamide | Human | 11140 | |
| FGFR1 | FGFR | TK | 1agw | A | A | 3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone | Human | 3520 | |
| FGFR1 | FGFR | TK | 1agw | A | B | 3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone | Human | 3528 | |
| FGFR1 | FGFR | TK | 1agw | B | A | 3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone | Human | 3568 | |
| FGFR1 | FGFR | TK | 1agw | B | B | 3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinone | Human | 3510 | |
| FGFR1 | FGFR | TK | 1fgi | A | A | 3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinone | Human | 3555 | |
| FGFR1 | FGFR | TK | 1fgi | A | B | 3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinone | Human | 3552 | |
| FGFR1 | FGFR | TK | 1fgi | B | A | 3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinone | Human | 3586 | |
| FGFR1 | FGFR | TK | 1fgi | B | B | 3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinone | Human | 3580 | |
| FGFR1 | FGFR | TK | 1fgk | A | A | - | Human | 3592 | |
| FGFR1 | FGFR | TK | 1fgk | A | B | - | Human | 3546 | |
| FGFR1 | FGFR | TK | 1fgk | B | A | - | Human | 3513 | |
| FGFR1 | FGFR | TK | 1fgk | B | B | - | Human | 3557 | |
| FGFR1 | FGFR | TK | 2fgi | A | | 1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-urea | Human | 3490 | |
| FGFR1 | FGFR | TK | 2fgi | B | | 1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-urea | Human | 3541 | |
| FGFR1 | FGFR | TK | 3c4f | A | A | 3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridine | Human | 3515 | |
| FGFR1 | FGFR | TK | 3c4f | A | B | 3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridine | Human | 3564 | |
| FGFR1 | FGFR | TK | 3c4f | B | A | 3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridine | Human | 3573 | |
| FGFR1 | FGFR | TK | 3c4f | B | B | 3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridine | Human | 3562 | |
| FGFR1 | FGFR | TK | 3gqi | A | | phosphomethylphosphonic acid adenylate ester | Human | 3566 | |
| FGFR1 | FGFR | TK | 3gql | A | | (e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanol | Human | 3509 | |
| FGFR1 | FGFR | TK | 3gql | B | | (e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanol | Human | 3506 | |
| FGFR1 | FGFR | TK | 3gql | C | | (e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanol | Human | 3536 | |
| FGFR1 | FGFR | TK | 3js2 | A | | 5-(2-thienyl)nicotinic acid | Human | 3523 | |
| FGFR1 | FGFR | TK | 3js2 | B | | 5-(2-thienyl)nicotinic acid | Human | 3504 | |
| FGFR1 | FGFR | TK | 3kxx | A | | - | Human | 3495 | |
| FGFR1 | FGFR | TK | 3kxx | B | | - | Human | 3575 | |
| FGFR1 | FGFR | TK | 3kxx | C | | - | Human | 3549 | |
| FGFR1 | FGFR | TK | 3kxx | D | | - | Human | 3503 | |
| FGFR1 | FGFR | TK | 3ky2 | A | | - | Human | 3534 | |
| FGFR1 | FGFR | TK | 3ky2 | B | | - | Human | 3525 | |
| FGFR1 | FGFR | TK | 3rhx | A | | (6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amine | Human | 3554 | |
| FGFR1 | FGFR | TK | 3rhx | B | | (6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amine | Human | 3522 | |
| FGFR1 | FGFR | TK | 3tt0 | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylurea | Human | 3567 | |
| FGFR1 | FGFR | TK | 3tt0 | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylurea | Human | 3538 | |
| FGFR1 | FGFR | TK | 3tt0 | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylurea | Human | 3547 | |
| FGFR1 | FGFR | TK | 3tt0 | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylurea | Human | 3581 | |
| FGFR1 | FGFR | TK | 4f63 | A | | 5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamine | Human | 3563 | |
| FGFR1 | FGFR | TK | 4f63 | B | | 5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamine | Human | 3574 | |
| FGFR1 | FGFR | TK | 4f64 | A | A | 5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | 3548 | |
| FGFR1 | FGFR | TK | 4f64 | A | B | 5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | 3589 | |
| FGFR1 | FGFR | TK | 4f64 | B | A | 5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | 3576 | |
| FGFR1 | FGFR | TK | 4f64 | B | B | 5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | 3553 | |
| FGFR1 | FGFR | TK | 4f65 | A | A | 5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamine | Human | 3558 | |
| FGFR1 | FGFR | TK | 4f65 | A | B | 5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamine | Human | 3508 | |
| FGFR1 | FGFR | TK | 4f65 | B | A | 5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamine | Human | 3545 | |
| FGFR1 | FGFR | TK | 4f65 | B | B | 5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamine | Human | 3502 | |
| FGFR1 | FGFR | TK | 4nk9 | A | | n~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | 3550 | |
| FGFR1 | FGFR | TK | 4nk9 | B | | n~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | 3535 | |
| FGFR1 | FGFR | TK | 4nka | A | | n~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | 3501 | |
| FGFR1 | FGFR | TK | 4nka | B | | n~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine | Human | 3539 | |
| FGFR1 | FGFR | TK | 4nks | A | A | n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamine | Human | 3570 | |
| FGFR1 | FGFR | TK | 4nks | A | B | n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamine | Human | 3561 | |
| FGFR1 | FGFR | TK | 4nks | B | A | n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamine | Human | 3492 | |
| FGFR1 | FGFR | TK | 4nks | B | B | n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamine | Human | 3577 | |
| FGFR1 | FGFR | TK | 4rwi | A | A | - | Human | 3499 | |
| FGFR1 | FGFR | TK | 4rwi | A | B | - | Human | 3551 | |
| FGFR1 | FGFR | TK | 4rwi | B | A | - | Human | 3569 | |
| FGFR1 | FGFR | TK | 4rwi | B | B | - | Human | 3527 | |
| FGFR1 | FGFR | TK | 4rwj | A | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3584 | |
| FGFR1 | FGFR | TK | 4rwj | A | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3519 | |
| FGFR1 | FGFR | TK | 4rwj | B | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3579 | |
| FGFR1 | FGFR | TK | 4rwj | B | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3559 | |
| FGFR1 | FGFR | TK | 4rwk | A | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3500 | |
| FGFR1 | FGFR | TK | 4rwk | A | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3517 | |
| FGFR1 | FGFR | TK | 4rwk | B | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3591 | |
| FGFR1 | FGFR | TK | 4rwk | B | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3530 | |
| FGFR1 | FGFR | TK | 4rwl | A | | - | Human | 3516 | |
| FGFR1 | FGFR | TK | 4rwl | B | | 6-({7-[(1-aminocyclopropyl)methoxy]-6-methoxyquinolin-4-yl}oxy)-n-methylnaphthalene-1-carboxamide | Human | 3596 | |
| FGFR1 | FGFR | TK | 4uwb | A | A | n-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamide | Human | 6020 | |
| FGFR1 | FGFR | TK | 4uwb | A | B | n-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamide | Human | 6023 | |
| FGFR1 | FGFR | TK | 4uwb | B | A | n-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamide | Human | 6018 | |
| FGFR1 | FGFR | TK | 4uwb | B | B | n-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamide | Human | 6022 | |
| FGFR1 | FGFR | TK | 4uwc | A | A | 3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamide | Human | 6019 | |
| FGFR1 | FGFR | TK | 4uwc | A | B | 3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamide | Human | 6017 | |
| FGFR1 | FGFR | TK | 4uwc | B | A | 3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamide | Human | 6021 | |
| FGFR1 | FGFR | TK | 4uwc | B | B | 3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamide | Human | 6016 | |
| FGFR1 | FGFR | TK | 4uwy | A | A | - | Human | 3489 | |
| FGFR1 | FGFR | TK | 4uwy | A | B | - | Human | 3582 | |
| FGFR1 | FGFR | TK | 4uwy | B | A | - | Human | 3537 | |
| FGFR1 | FGFR | TK | 4uwy | B | B | - | Human | 3583 | |
| FGFR1 | FGFR | TK | 4v01 | A | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3556 | |
| FGFR1 | FGFR | TK | 4v01 | A | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3590 | |
| FGFR1 | FGFR | TK | 4v01 | B | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3497 | |
| FGFR1 | FGFR | TK | 4v01 | B | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3594 | |
| FGFR1 | FGFR | TK | 4v04 | A | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3542 | |
| FGFR1 | FGFR | TK | 4v04 | A | B | - | Human | 3571 | |
| FGFR1 | FGFR | TK | 4v04 | B | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3524 | |
| FGFR1 | FGFR | TK | 4v04 | B | B | - | Human | 3496 | |
| FGFR1 | FGFR | TK | 4v05 | A | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3560 | |
| FGFR1 | FGFR | TK | 4v05 | A | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3593 | |
| FGFR1 | FGFR | TK | 4v05 | B | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3518 | |
| FGFR1 | FGFR | TK | 4v05 | B | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3493 | |
| FGFR1 | FGFR | TK | 4wun | A | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3511 | |
| FGFR1 | FGFR | TK | 4wun | A | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3595 | |
| FGFR1 | FGFR | TK | 4wun | B | A | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3529 | |
| FGFR1 | FGFR | TK | 4wun | B | B | n-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamide | Human | 3565 | |
| FGFR1 | FGFR | TK | 4zsa | A | A | 4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamide | Human | 3491 | |
| FGFR1 | FGFR | TK | 4zsa | A | B | 4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamide | Human | 3487 | |
| FGFR1 | FGFR | TK | 4zsa | B | A | 4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamide | Human | 3572 | |
| FGFR1 | FGFR | TK | 4zsa | B | B | 4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamide | Human | 3512 | |
| FGFR1 | FGFR | TK | 5a46 | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3532 | |
| FGFR1 | FGFR | TK | 5a46 | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3505 | |
| FGFR1 | FGFR | TK | 5a46 | B | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3526 | |
| FGFR1 | FGFR | TK | 5a46 | B | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3578 | |
| FGFR1 | FGFR | TK | 5a4c | A | A | 1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea | Human | 3543 | |
| FGFR1 | FGFR | TK | 5a4c | A | B | 1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea | Human | 3498 | |
| FGFR1 | FGFR | TK | 5a4c | B | A | 1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea | Human | 3585 | |
| FGFR1 | FGFR | TK | 5a4c | B | B | 1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea | Human | 3540 | |
| FGFR1 | FGFR | TK | 5am6 | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3494 | |
| FGFR1 | FGFR | TK | 5am6 | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3514 | |
| FGFR1 | FGFR | TK | 5am6 | B | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3587 | |
| FGFR1 | FGFR | TK | 5am6 | B | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3521 | |
| FGFR1 | FGFR | TK | 5am7 | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3533 | |
| FGFR1 | FGFR | TK | 5am7 | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3488 | |
| FGFR1 | FGFR | TK | 5am7 | B | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3588 | |
| FGFR1 | FGFR | TK | 5am7 | B | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 3531 | |
| FGFR1 | FGFR | TK | 5b7v | A | | [5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanone | Human | 6705 | |
| FGFR1 | FGFR | TK | 5b7v | B | | [5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanone | Human | 6704 | |
| FGFR1 | FGFR | TK | 5ew8 | A | A | ~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamine | Human | 6470 | |
| FGFR1 | FGFR | TK | 5ew8 | A | B | ~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamine | Human | 6461 | |
| FGFR1 | FGFR | TK | 5ew8 | B | A | ~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamine | Human | 6474 | |
| FGFR1 | FGFR | TK | 5ew8 | B | B | ~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamine | Human | 6471 | |
| FGFR1 | FGFR | TK | 5flf | A | A | - | Human | 6462 | |
| FGFR1 | FGFR | TK | 5flf | A | B | - | Human | 6464 | |
| FGFR1 | FGFR | TK | 5flf | B | A | - | Human | 6465 | |
| FGFR1 | FGFR | TK | 5flf | B | B | - | Human | 6467 | |
| FGFR1 | FGFR | TK | 5flf | C | A | - | Human | 6469 | |
| FGFR1 | FGFR | TK | 5flf | C | B | - | Human | 6466 | |
| FGFR1 | FGFR | TK | 5flf | D | A | - | Human | 6468 | |
| FGFR1 | FGFR | TK | 5flf | D | B | - | Human | 6463 | |
| FGFR1 | FGFR | TK | 5flf | E | A | - | Human | 6473 | |
| FGFR1 | FGFR | TK | 5flf | E | B | - | Human | 6472 | |
| FGFR1 | FGFR | TK | 5o49 | A | A | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoate | Human | 9560 | |
| FGFR1 | FGFR | TK | 5o49 | A | B | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoate | Human | 9556 | |
| FGFR1 | FGFR | TK | 5o49 | B | A | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoate | Human | 9561 | |
| FGFR1 | FGFR | TK | 5o49 | B | B | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoate | Human | 9557 | |
| FGFR1 | FGFR | TK | 5o4a | A | A | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoate | Human | 9554 | |
| FGFR1 | FGFR | TK | 5o4a | A | B | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoate | Human | 9558 | |
| FGFR1 | FGFR | TK | 5o4a | B | A | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoate | Human | 9559 | |
| FGFR1 | FGFR | TK | 5o4a | B | B | [(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoate | Human | 9555 | |
| FGFR1 | FGFR | TK | 5uq0 | A | A | 2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamide | Human | 7456 | |
| FGFR1 | FGFR | TK | 5uq0 | A | B | 2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamide | Human | 7458 | |
| FGFR1 | FGFR | TK | 5uq0 | B | A | 2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamide | Human | 7459 | |
| FGFR1 | FGFR | TK | 5uq0 | B | B | 2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamide | Human | 7457 | |
| FGFR1 | FGFR | TK | 5ur1 | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 7970 | |
| FGFR1 | FGFR | TK | 5ur1 | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 7972 | |
| FGFR1 | FGFR | TK | 5ur1 | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 7969 | |
| FGFR1 | FGFR | TK | 5ur1 | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 7971 | |
| FGFR1 | FGFR | TK | 5vnd | A | A | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamide | Human | 7646 | |
| FGFR1 | FGFR | TK | 5vnd | A | B | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamide | Human | 7648 | |
| FGFR1 | FGFR | TK | 5vnd | B | A | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamide | Human | 7647 | |
| FGFR1 | FGFR | TK | 5vnd | B | B | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamide | Human | 7645 | |
| FGFR1 | FGFR | TK | 5z0s | A | A | 1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridine | Human | 10813 | |
| FGFR1 | FGFR | TK | 5z0s | A | B | 1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridine | Human | 10815 | |
| FGFR1 | FGFR | TK | 5z0s | B | A | 1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridine | Human | 10812 | |
| FGFR1 | FGFR | TK | 5z0s | B | B | 1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridine | Human | 10814 | |
| FGFR1 | FGFR | TK | 5zv2 | A | | 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide | Human | 10055 | |
| FGFR1 | FGFR | TK | 5zv2 | B | | 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide | Human | 10054 | |
| FGFR1 | FGFR | TK | 6c18 | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 11155 | |
| FGFR1 | FGFR | TK | 6c18 | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 11168 | |
| FGFR1 | FGFR | TK | 6c18 | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 10854 | |
| FGFR1 | FGFR | TK | 6c18 | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 11170 | |
| FGFR1 | FGFR | TK | 6c19 | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 11163 | |
| FGFR1 | FGFR | TK | 6c19 | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 10859 | |
| FGFR1 | FGFR | TK | 6c19 | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 10855 | |
| FGFR1 | FGFR | TK | 6c19 | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 10862 | |
| FGFR1 | FGFR | TK | 6c1b | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 11169 | |
| FGFR1 | FGFR | TK | 6c1b | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 10861 | |
| FGFR1 | FGFR | TK | 6c1b | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 10856 | |
| FGFR1 | FGFR | TK | 6c1b | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 11167 | |
| FGFR1 | FGFR | TK | 6c1c | A | A | 7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 11164 | |
| FGFR1 | FGFR | TK | 6c1c | A | B | 7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 10853 | |
| FGFR1 | FGFR | TK | 6c1c | B | A | 7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 10858 | |
| FGFR1 | FGFR | TK | 6c1c | B | B | 7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 11158 | |
| FGFR1 | FGFR | TK | 6c1o | A | A | n-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamide | Human | 11159 | |
| FGFR1 | FGFR | TK | 6c1o | A | B | n-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamide | Human | 11166 | |
| FGFR1 | FGFR | TK | 6c1o | B | A | n-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamide | Human | 11160 | |
| FGFR1 | FGFR | TK | 6c1o | B | B | n-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamide | Human | 11154 | |
| FGFR1 | FGFR | TK | 6itj | A | A | 4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-one | Human | 11773 | |
| FGFR1 | FGFR | TK | 6itj | A | B | 4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-one | Human | 11774 | |
| FGFR1 | FGFR | TK | 6itj | B | A | 4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-one | Human | 11775 | |
| FGFR1 | FGFR | TK | 6itj | B | B | 4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-one | Human | 11772 | |
| FGFR1 | FGFR | TK | 6mzq | A | A | 1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one | Human | 10860 | |
| FGFR1 | FGFR | TK | 6mzq | A | B | 1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one | Human | 11156 | |
| FGFR1 | FGFR | TK | 6mzq | B | A | 1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one | Human | 11161 | |
| FGFR1 | FGFR | TK | 6mzq | B | B | 1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one | Human | 11171 | |
| FGFR1 | FGFR | TK | 6mzw | A | A | 1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one | Human | 11162 | |
| FGFR1 | FGFR | TK | 6mzw | A | B | 1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one | Human | 11157 | |
| FGFR1 | FGFR | TK | 6mzw | B | A | 1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one | Human | 11165 | |
| FGFR1 | FGFR | TK | 6mzw | B | B | 1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-one | Human | 10857 | |
| FGFR1 | FGFR | TK | 6nvl | A | A | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11400 | |
| FGFR1 | FGFR | TK | 6nvl | A | B | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11401 | |
| FGFR1 | FGFR | TK | 6nvl | B | A | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11403 | |
| FGFR1 | FGFR | TK | 6nvl | B | B | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11399 | |
| FGFR1 | FGFR | TK | 6nvl | C | A | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11404 | |
| FGFR1 | FGFR | TK | 6nvl | C | B | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11405 | |
| FGFR1 | FGFR | TK | 6nvl | D | A | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11402 | |
| FGFR1 | FGFR | TK | 6nvl | D | B | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11398 | |
| FGFR1 | FGFR | TK | 6p68 | A | | n-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamide | Human | 11336 | |
| FGFR1 | FGFR | TK | 6p68 | B | | n-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamide | Human | 11334 | |
| FGFR1 | FGFR | TK | 6p68 | C | | n-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamide | Human | 11332 | |
| FGFR1 | FGFR | TK | 6p69 | A | A | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamide | Human | 11333 | |
| FGFR1 | FGFR | TK | 6p69 | A | B | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamide | Human | 11330 | |
| FGFR1 | FGFR | TK | 6p69 | B | A | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamide | Human | 11331 | |
| FGFR1 | FGFR | TK | 6p69 | B | B | n-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamide | Human | 11335 | |
| FGFR1 | FGFR | TK | 7ozb | A | A | 4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenol | Human | 14010 | |
| FGFR1 | FGFR | TK | 7ozb | A | B | 4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenol | Human | 14008 | |
| FGFR1 | FGFR | TK | 7ozd | A | A | n-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamide | Human | 14007 | |
| FGFR1 | FGFR | TK | 7ozd | A | B | n-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamide | Human | 14009 | |
| FGFR1 | FGFR | TK | 7ozf | A | A | n-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamide | Human | 14011 | |
| FGFR1 | FGFR | TK | 7ozf | A | B | n-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamide | Human | 14006 | |
| FGFR1 | FGFR | TK | 7wcl | A | A | 11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-one | Human | 14364 | |
| FGFR1 | FGFR | TK | 7wcl | A | B | 11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-one | Human | 14363 | |
| FGFR1 | FGFR | TK | 8jmz | A | A | n-(2-(dimethylamino)ethyl)-1-(3-((4-((2-methyl-1h-indol-5-yl)oxy)pyrimidin-2-yl)amino)phenyl)methanesulfonamide | Human | 15228 | |
| FGFR1 | FGFR | TK | 8jmz | A | B | n-(2-(dimethylamino)ethyl)-1-(3-((4-((2-methyl-1h-indol-5-yl)oxy)pyrimidin-2-yl)amino)phenyl)methanesulfonamide | Human | 15227 | |
| FGFR2 | FGFR | TK | 1gjo | A | | - | Human | 478 | |
| FGFR2 | FGFR | TK | 1oec | A | | 4-aryl-2-phenylamino pyrimidine | Human | 479 | |
| FGFR2 | FGFR | TK | 2psq | A | | - | Human | 515 | |
| FGFR2 | FGFR | TK | 2psq | B | | - | Human | 530 | |
| FGFR2 | FGFR | TK | 2pvf | A | | phosphomethylphosphonic acid adenylate ester | Human | 525 | |
| FGFR2 | FGFR | TK | 2pvy | A | | phosphomethylphosphonic acid adenylate ester | Human | 489 | |
| FGFR2 | FGFR | TK | 2pvy | B | | phosphomethylphosphonic acid adenylate ester | Human | 504 | |
| FGFR2 | FGFR | TK | 2pvy | C | | phosphomethylphosphonic acid adenylate ester | Human | 501 | |
| FGFR2 | FGFR | TK | 2pvy | D | | phosphomethylphosphonic acid adenylate ester | Human | 482 | |
| FGFR2 | FGFR | TK | 2pwl | A | | phosphomethylphosphonic acid adenylate ester | Human | 523 | |
| FGFR2 | FGFR | TK | 2pwl | B | | phosphomethylphosphonic acid adenylate ester | Human | 534 | |
| FGFR2 | FGFR | TK | 2py3 | A | | phosphomethylphosphonic acid adenylate ester | Human | 509 | |
| FGFR2 | FGFR | TK | 2py3 | B | | phosphomethylphosphonic acid adenylate ester | Human | 484 | |
| FGFR2 | FGFR | TK | 2pz5 | A | | phosphomethylphosphonic acid adenylate ester | Human | 511 | |
| FGFR2 | FGFR | TK | 2pz5 | B | | phosphomethylphosphonic acid adenylate ester | Human | 513 | |
| FGFR2 | FGFR | TK | 2pzp | A | | phosphomethylphosphonic acid adenylate ester | Human | 497 | |
| FGFR2 | FGFR | TK | 2pzp | B | | phosphomethylphosphonic acid adenylate ester | Human | 524 | |
| FGFR2 | FGFR | TK | 2pzr | A | | phosphomethylphosphonic acid adenylate ester | Human | 526 | |
| FGFR2 | FGFR | TK | 2pzr | B | | phosphomethylphosphonic acid adenylate ester | Human | 508 | |
| FGFR2 | FGFR | TK | 2q0b | A | | phosphomethylphosphonic acid adenylate ester | Human | 512 | |
| FGFR2 | FGFR | TK | 2q0b | B | | phosphomethylphosphonic acid adenylate ester | Human | 499 | |
| FGFR2 | FGFR | TK | 3b2t | A | | 5'-o-[(s)-hydroxy{[(s)-hydroxy(methyl)phosphoryl]oxy}phosphoryl]adenosine | Human | 520 | |
| FGFR2 | FGFR | TK | 3b2t | B | | 5'-o-[(s)-hydroxy{[(s)-hydroxy(methyl)phosphoryl]oxy}phosphoryl]adenosine | Human | 517 | |
| FGFR2 | FGFR | TK | 3cly | A | | phosphomethylphosphonic acid adenylate ester | Human | 522 | |
| FGFR2 | FGFR | TK | 3ri1 | A | | (6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amine | Human | 503 | |
| FGFR2 | FGFR | TK | 3ri1 | B | | (6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amine | Human | 528 | |
| FGFR2 | FGFR | TK | 4j95 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 529 | |
| FGFR2 | FGFR | TK | 4j95 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 477 | |
| FGFR2 | FGFR | TK | 4j95 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 498 | |
| FGFR2 | FGFR | TK | 4j95 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 519 | |
| FGFR2 | FGFR | TK | 4j95 | C | A | phosphomethylphosphonic acid adenylate ester | Human | 531 | |
| FGFR2 | FGFR | TK | 4j95 | C | B | phosphomethylphosphonic acid adenylate ester | Human | 502 | |
| FGFR2 | FGFR | TK | 4j95 | D | A | phosphomethylphosphonic acid adenylate ester | Human | 490 | |
| FGFR2 | FGFR | TK | 4j95 | D | B | phosphomethylphosphonic acid adenylate ester | Human | 492 | |
| FGFR2 | FGFR | TK | 4j96 | A | A | - | Human | 473 | |
| FGFR2 | FGFR | TK | 4j96 | A | B | - | Human | 470 | |
| FGFR2 | FGFR | TK | 4j96 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 485 | |
| FGFR2 | FGFR | TK | 4j96 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 486 | |
| FGFR2 | FGFR | TK | 4j97 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 496 | |
| FGFR2 | FGFR | TK | 4j97 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 527 | |
| FGFR2 | FGFR | TK | 4j97 | A | C | phosphomethylphosphonic acid adenylate ester | Human | 521 | |
| FGFR2 | FGFR | TK | 4j97 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 476 | |
| FGFR2 | FGFR | TK | 4j97 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 493 | |
| FGFR2 | FGFR | TK | 4j97 | B | C | phosphomethylphosphonic acid adenylate ester | Human | 510 | |
| FGFR2 | FGFR | TK | 4j97 | C | A | phosphomethylphosphonic acid adenylate ester | Human | 488 | |
| FGFR2 | FGFR | TK | 4j97 | C | B | phosphomethylphosphonic acid adenylate ester | Human | 487 | |
| FGFR2 | FGFR | TK | 4j97 | C | C | phosphomethylphosphonic acid adenylate ester | Human | 483 | |
| FGFR2 | FGFR | TK | 4j97 | D | A | phosphomethylphosphonic acid adenylate ester | Human | 507 | |
| FGFR2 | FGFR | TK | 4j97 | D | B | phosphomethylphosphonic acid adenylate ester | Human | 532 | |
| FGFR2 | FGFR | TK | 4j97 | D | C | phosphomethylphosphonic acid adenylate ester | Human | 514 | |
| FGFR2 | FGFR | TK | 4j98 | A | A | - | Human | 500 | |
| FGFR2 | FGFR | TK | 4j98 | A | B | - | Human | 475 | |
| FGFR2 | FGFR | TK | 4j98 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 516 | |
| FGFR2 | FGFR | TK | 4j98 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 472 | |
| FGFR2 | FGFR | TK | 4j99 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 474 | |
| FGFR2 | FGFR | TK | 4j99 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 494 | |
| FGFR2 | FGFR | TK | 4j99 | A | C | phosphomethylphosphonic acid adenylate ester | Human | 469 | |
| FGFR2 | FGFR | TK | 4j99 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 518 | |
| FGFR2 | FGFR | TK | 4j99 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 495 | |
| FGFR2 | FGFR | TK | 4j99 | B | C | phosphomethylphosphonic acid adenylate ester | Human | 491 | |
| FGFR2 | FGFR | TK | 4j99 | C | A | phosphomethylphosphonic acid adenylate ester | Human | 505 | |
| FGFR2 | FGFR | TK | 4j99 | C | B | phosphomethylphosphonic acid adenylate ester | Human | 506 | |
| FGFR2 | FGFR | TK | 4j99 | C | C | phosphomethylphosphonic acid adenylate ester | Human | 471 | |
| FGFR2 | FGFR | TK | 4j99 | D | A | phosphomethylphosphonic acid adenylate ester | Human | 533 | |
| FGFR2 | FGFR | TK | 4j99 | D | B | phosphomethylphosphonic acid adenylate ester | Human | 481 | |
| FGFR2 | FGFR | TK | 4j99 | D | C | phosphomethylphosphonic acid adenylate ester | Human | 480 | |
| FGFR2 | FGFR | TK | 5eg3 | A | | phosphomethylphosphonic acid adenylate ester | Human | 6368 | |
| FGFR2 | FGFR | TK | 5ugl | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 7442 | |
| FGFR2 | FGFR | TK | 5ugl | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 7452 | |
| FGFR2 | FGFR | TK | 5ugl | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 7450 | |
| FGFR2 | FGFR | TK | 5ugl | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 7449 | |
| FGFR2 | FGFR | TK | 5ugx | A | A | phosphomethylphosphonic acid adenylate ester | Human | 7443 | |
| FGFR2 | FGFR | TK | 5ugx | A | B | phosphomethylphosphonic acid adenylate ester | Human | 7448 | |
| FGFR2 | FGFR | TK | 5ugx | B | A | phosphomethylphosphonic acid adenylate ester | Human | 7454 | |
| FGFR2 | FGFR | TK | 5ugx | B | B | phosphomethylphosphonic acid adenylate ester | Human | 7445 | |
| FGFR2 | FGFR | TK | 5uhn | A | A | phosphomethylphosphonic acid adenylate ester | Human | 7455 | |
| FGFR2 | FGFR | TK | 5uhn | A | B | phosphomethylphosphonic acid adenylate ester | Human | 7441 | |
| FGFR2 | FGFR | TK | 5uhn | B | A | phosphomethylphosphonic acid adenylate ester | Human | 7451 | |
| FGFR2 | FGFR | TK | 5uhn | B | B | phosphomethylphosphonic acid adenylate ester | Human | 7444 | |
| FGFR2 | FGFR | TK | 5ui0 | A | A | - | Human | 7446 | |
| FGFR2 | FGFR | TK | 5ui0 | A | B | - | Human | 7447 | |
| FGFR2 | FGFR | TK | 5ui0 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 7453 | |
| FGFR2 | FGFR | TK | 5ui0 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 7440 | |
| FGFR2 | FGFR | TK | 6agx | A | A | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | 11541 | |
| FGFR2 | FGFR | TK | 6agx | A | B | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | 11542 | |
| FGFR2 | FGFR | TK | 6agx | B | A | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | 11540 | |
| FGFR2 | FGFR | TK | 6agx | B | B | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | 11536 | |
| FGFR2 | FGFR | TK | 6agx | C | A | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | 11538 | |
| FGFR2 | FGFR | TK | 6agx | C | B | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | 11537 | |
| FGFR2 | FGFR | TK | 6agx | D | A | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | 11543 | |
| FGFR2 | FGFR | TK | 6agx | D | B | ethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetate | Human | 11539 | |
| FGFR2 | FGFR | TK | 6lvk | A | | n-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamide | Human | 12131 | |
| FGFR2 | FGFR | TK | 6lvk | B | | n-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamide | Human | 12129 | |
| FGFR2 | FGFR | TK | 6lvl | A | | n-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamide | Human | 12132 | |
| FGFR2 | FGFR | TK | 6lvl | B | | n-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamide | Human | 12130 | |
| FGFR2 | FGFR | TK | 6v6q | A | | phosphomethylphosphonic acid adenylate ester | Human | 12968 | |
| FGFR2 | FGFR | TK | 6v6q | B | | phosphomethylphosphonic acid adenylate ester | Human | 12966 | |
| FGFR2 | FGFR | TK | 6v6q | C | | phosphomethylphosphonic acid adenylate ester | Human | 12969 | |
| FGFR2 | FGFR | TK | 6v6q | D | | phosphomethylphosphonic acid adenylate ester | Human | 12967 | |
| FGFR2 | FGFR | TK | 7kia | A | A | 1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-one | Human | 13283 | |
| FGFR2 | FGFR | TK | 7kia | A | B | 1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-one | Human | 13285 | |
| FGFR2 | FGFR | TK | 7kia | B | A | 1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-one | Human | 13281 | |
| FGFR2 | FGFR | TK | 7kia | B | B | 1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-one | Human | 13288 | |
| FGFR2 | FGFR | TK | 7kie | A | A | n-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamide | Human | 13287 | |
| FGFR2 | FGFR | TK | 7kie | A | B | n-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamide | Human | 13286 | |
| FGFR2 | FGFR | TK | 7kie | B | A | n-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamide | Human | 13282 | |
| FGFR2 | FGFR | TK | 7kie | B | B | n-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamide | Human | 13284 | |
| FGFR2 | FGFR | TK | 7ozy | A | A | 4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenol | Human | 13999 | |
| FGFR2 | FGFR | TK | 7ozy | A | B | 4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenol | Human | 13998 | |
| FGFR2 | FGFR | TK | 8e1x | A | | (5m)-n-methyl-5-{(6m,8s)-5-{[(3s)-oxolan-3-yl]amino}-6-[1-(propan-2-yl)-1h-pyrazol-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl}pyridine-3-carboxamide | Human | 14511 | |
| FGFR2 | FGFR | TK | 8h75 | A | | 4-[9-(2-chlorophenyl)-6-methyl-2,4,5,8,12-pentazatricyclo[8.4.0.0^{3,7}]tetradeca-1(10),3,6,8,11,13-hexaen-13-yl]morpholine | Human | 14860 | |
| FGFR2 | FGFR | TK | 8stg | A | | n-{4-[(5p)-4-amino-5-{3-fluoro-4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}-2-methylprop-2-enamide | Human | 14762 | |
| FGFR2 | FGFR | TK | 8swe | A | A | n-{4-[4-amino-5-(4-methoxyphenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}prop-2-enamide | Human | 15200 | |
| FGFR2 | FGFR | TK | 8swe | A | B | n-{4-[4-amino-5-(4-methoxyphenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}prop-2-enamide | Human | 15201 | |
| FGFR2 | FGFR | TK | 8u1f | A | | n-[4-(4-amino-7-methyl-5-{4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7h-pyrrolo[2,3-d]pyrimidin-6-yl)phenyl]-2-methylpropanamide | Human | 15202 | |
| FGFR3 | FGFR | TK | 4k33 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 1871 | |
| FGFR3 | FGFR | TK | 4k33 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 1870 | |
| FGFR3 | FGFR | TK | 6lvm | A | | 2-[[5-[2-(3,5-dimethoxyphenyl)ethyl]-2-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]pyrimidin-4-yl]amino]-n-ethyl-benzenesulfonamide | Human | 12134 | |
| FGFR3 | FGFR | TK | 6pnx | A | A | phosphomethylphosphonic acid adenylate ester | Human | 11948 | |
| FGFR3 | FGFR | TK | 6pnx | A | B | phosphomethylphosphonic acid adenylate ester | Human | 11946 | |
| FGFR3 | FGFR | TK | 6pnx | B | A | phosphomethylphosphonic acid adenylate ester | Human | 11947 | |
| FGFR3 | FGFR | TK | 6pnx | B | B | phosphomethylphosphonic acid adenylate ester | Human | 11949 | |
| FGFR3 | FGFR | TK | 7dhl | A | | 5-[2-(3,5-dimethoxyphenyl)ethyl]-n-[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]pyrimidin-2-amine | Human | 13258 | |
| FGFR3 | FGFR | TK | 8udt | A | | 3-[(1-cyclopropyl-4,6-difluoro-1h-benzimidazol-5-yl)ethynyl]-1-[(3r,5r)-5-(methoxymethyl)-1-propanoylpyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamide | Human | 15206 | |
| FGFR3 | FGFR | TK | 8udu | A | A | 3-[(6-chloro-1-cyclopropyl-1h-benzimidazol-5-yl)ethynyl]-1-[(3s,5s)-5-(methoxymethyl)-1-(prop-2-enoyl)pyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamide | Human | 15205 | |
| FGFR3 | FGFR | TK | 8udu | A | B | 3-[(6-chloro-1-cyclopropyl-1h-benzimidazol-5-yl)ethynyl]-1-[(3s,5s)-5-(methoxymethyl)-1-(prop-2-enoyl)pyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamide | Human | 15204 | |
| FGFR3 | FGFR | TK | 8udv | A | | 3-[(6-chloro-1-cyclopropyl-1h-benzimidazol-5-yl)ethynyl]-1-[(3s,5s)-5-(methoxymethyl)-1-(prop-2-enoyl)pyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamide | Human | 15203 | |
| FGFR4 | FGFR | TK | 4qq5 | A | | n-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamide | Human | 921 | |
| FGFR4 | FGFR | TK | 4qqc | A | A | n-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamide | Human | 934 | |
| FGFR4 | FGFR | TK | 4qqc | A | B | n-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamide | Human | 932 | |
| FGFR4 | FGFR | TK | 4qqj | A | | - | Human | 935 | |
| FGFR4 | FGFR | TK | 4qqt | A | | - | Human | 922 | |
| FGFR4 | FGFR | TK | 4qrc | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 923 | |
| FGFR4 | FGFR | TK | 4r6v | A | | n-[4-({[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino}methyl)phenyl]propanamide | Human | 931 | |
| FGFR4 | FGFR | TK | 4tye | A | | - | Human | 927 | |
| FGFR4 | FGFR | TK | 4tyg | A | A | - | Human | 929 | |
| FGFR4 | FGFR | TK | 4tyg | A | B | - | Human | 933 | |
| FGFR4 | FGFR | TK | 4tyi | A | | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 926 | |
| FGFR4 | FGFR | TK | 4tyj | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 925 | |
| FGFR4 | FGFR | TK | 4uxq | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 930 | |
| FGFR4 | FGFR | TK | 4xcu | A | A | n-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamide | Human | 928 | |
| FGFR4 | FGFR | TK | 4xcu | A | B | n-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamide | Human | 924 | |
| FGFR4 | FGFR | TK | 5jkg | A | | 2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanol | Human | 7089 | |
| FGFR4 | FGFR | TK | 5nud | A | | 3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amine | Human | 9787 | |
| FGFR4 | FGFR | TK | 5nud | B | | 3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amine | Human | 9790 | |
| FGFR4 | FGFR | TK | 5nwz | A | | ~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamide | Human | 9789 | |
| FGFR4 | FGFR | TK | 5nwz | B | | ~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamide | Human | 9788 | |
| FGFR4 | FGFR | TK | 5xff | A | | 2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanol | Human | 10375 | |
| FGFR4 | FGFR | TK | 5xfj | A | | 2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanol | Human | 10376 | |
| FGFR4 | FGFR | TK | 6iuo | A | | n-({4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}methyl)prop-2-enamide | Human | 11757 | |
| FGFR4 | FGFR | TK | 6iup | A | A | n-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamide | Human | 11797 | |
| FGFR4 | FGFR | TK | 6iup | A | B | n-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamide | Human | 11796 | |
| FGFR4 | FGFR | TK | 6jpe | A | | n-[2-[[6-[2-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]amino]pyridin-3-yl]pyrimidin-4-yl]amino]-3-methyl-phenyl]prop-2-enamide | Human | 12230 | |
| FGFR4 | FGFR | TK | 6jpj | A | | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 11051 | |
| FGFR4 | FGFR | TK | 6nvg | A | | n-[3,5-dichloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)phenyl]propanamide | Human | 11394 | |
| FGFR4 | FGFR | TK | 6nvh | A | A | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11388 | |
| FGFR4 | FGFR | TK | 6nvh | A | B | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamide | Human | 11393 | |
| FGFR4 | FGFR | TK | 6nvi | A | A | n-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamide | Human | 11392 | |
| FGFR4 | FGFR | TK | 6nvi | A | B | n-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamide | Human | 11389 | |
| FGFR4 | FGFR | TK | 6nvj | A | | n-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-fluorophenyl]propanamide | Human | 11391 | |
| FGFR4 | FGFR | TK | 6nvk | A | A | n-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamide | Human | 11395 | |
| FGFR4 | FGFR | TK | 6nvk | A | B | n-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamide | Human | 11390 | |
| FGFR4 | FGFR | TK | 6v9c | A | A | n-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamide | Human | 12096 | |
| FGFR4 | FGFR | TK | 6v9c | A | B | n-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamide | Human | 12095 | |
| FGFR4 | FGFR | TK | 6yi8 | A | A | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 12812 | |
| FGFR4 | FGFR | TK | 6yi8 | A | B | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 12811 | |
| FGFR4 | FGFR | TK | 6yi8 | B | A | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 12813 | |
| FGFR4 | FGFR | TK | 6yi8 | B | B | n-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 12814 | |
| FGFR4 | FGFR | TK | 7dtz | A | | n-[2-[[5-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]methoxy]pyrimidin-2-yl]amino]-3-methyl-phenyl]-2-fluoranyl-prop-2-enamide | Human | 13506 | |
| FGFR4 | FGFR | TK | 7f3m | A | | 6-[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]-2-(methylamino)-8-[3-(4-prop-2-enoylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidin-7-one | Human | 14034 | |
| FGFR4 | FGFR | TK | 7v29 | A | | n-[2-[[3-(3,5-dimethoxyphenyl)-2-oxidanylidene-1-[3-(4-propanoylpiperazin-1-yl)propyl]-4h-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]propanamide | Human | 14165 | |
| FGFR4 | FGFR | TK | 7vjl | A | | n-[5-(aminomethyl)-4-(2-methoxyethylamino)pyridin-2-yl]-7-[2,2,2-tris(fluoranyl)ethanoyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamide | Human | 14109 | |
| FGFR4 | FGFR | TK | 7wct | A | | ~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamide | Human | 14167 | |
| FGFR4 | FGFR | TK | 7wcw | A | | ~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamide | Human | 14168 | |
| FGFR4 | FGFR | TK | 7wcx | A | | ~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamide | Human | 14166 | |
| FGFR4 | FGFR | TK | 7ybo | A | | ~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14499 | |
| FGFR4 | FGFR | TK | 7ybp | A | | ~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14500 | |
| FGFR4 | FGFR | TK | 7ybx | A | | ~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14502 | |
| FGFR4 | FGFR | TK | 7yc1 | A | | ~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-propyl-pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14498 | |
| FGFR4 | FGFR | TK | 7yc3 | A | | 6-bromanyl-~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamide | Human | 14501 | |
| FGFR4 | FGFR | TK | 8kh6 | A | | - | Human | 15287 | |
| FGFR4 | FGFR | TK | 8kh7 | A | | - | Human | 15286 | |
| FGFR4 | FGFR | TK | 8kh8 | A | | - | Human | 15285 | |
| FGFR4 | FGFR | TK | 8kh9 | A | | - | Human | 15284 | |
| FGFR4 | FGFR | TK | 8w5c | A | | - | Human | 15288 | |
| FGR | Src | TK | 7uy0 | A | A | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14568 | |
| FGR | Src | TK | 7uy0 | A | B | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14563 | |
| FGR | Src | TK | 7uy0 | A | C | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14564 | |
| FGR | Src | TK | 7uy0 | B | A | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14566 | |
| FGR | Src | TK | 7uy0 | B | B | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14565 | |
| FGR | Src | TK | 7uy0 | B | C | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14562 | |
| FGR | Src | TK | 7uy3 | A | | 3-[(6,7-dimethoxyquinazolin-4-yl)oxy]-n-{4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-4-methylbenzamide | Human | 14567 | |
| FLT1 | VEGFR | TK | 3hng | A | A | n-(4-chlorophenyl)-2-[(pyridin-4-ylmethyl)amino]benzamide | Human | 3837 | |
| FLT1 | VEGFR | TK | 3hng | A | B | n-(4-chlorophenyl)-2-[(pyridin-4-ylmethyl)amino]benzamide | Human | 3838 | |
| FLT3 | PDGFR | TK | 1rjb | A | | - | Human | 625 | |
| FLT3 | PDGFR | TK | 4rt7 | A | A | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)urea | Human | 626 | |
| FLT3 | PDGFR | TK | 4rt7 | A | B | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)urea | Human | 627 | |
| FLT3 | PDGFR | TK | 4xuf | A | | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)urea | Human | 624 | |
| FLT3 | PDGFR | TK | 4xuf | B | | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)urea | Human | 623 | |
| FLT3 | PDGFR | TK | 5x02 | A | | n-[(2s)-1-[5-[2-[(4-cyanophenyl)amino]-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxidanylidene-propan-2-yl]-4-(dimethylamino)-n-methyl-but-2-enamide | Human | 9522 | |
| FLT3 | PDGFR | TK | 6il3 | A | A | 7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)-3-(pyridin-2-yl)imidazo[1,2-a]pyridine | Human | 10785 | |
| FLT3 | PDGFR | TK | 6il3 | A | B | 7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)-3-(pyridin-2-yl)imidazo[1,2-a]pyridine | Human | 10786 | |
| FLT3 | PDGFR | TK | 6jqr | A | | 6-ethyl-3-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-5-(oxan-4-ylamino)pyrazine-2-carboxamide | Human | 11802 | |
| FYN | Src | TK | 2dq7 | X | | staurosporine | Human | 1941 | |
| GAK | NAK | Other | 4c57 | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 341 | |
| GAK | NAK | Other | 4c57 | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 340 | |
| GAK | NAK | Other | 4c57 | B | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 334 | |
| GAK | NAK | Other | 4c57 | B | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 348 | |
| GAK | NAK | Other | 4c58 | A | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 336 | |
| GAK | NAK | Other | 4c58 | A | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 333 | |
| GAK | NAK | Other | 4c59 | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 337 | |
| GAK | NAK | Other | 4c59 | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 346 | |
| GAK | NAK | Other | 4o38 | A | A | - | Human | 345 | |
| GAK | NAK | Other | 4o38 | A | B | - | Human | 335 | |
| GAK | NAK | Other | 4o38 | B | A | - | Human | 338 | |
| GAK | NAK | Other | 4o38 | B | B | - | Human | 343 | |
| GAK | NAK | Other | 4y8d | A | A | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | 344 | |
| GAK | NAK | Other | 4y8d | A | B | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | 339 | |
| GAK | NAK | Other | 4y8d | B | A | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | 347 | |
| GAK | NAK | Other | 4y8d | B | B | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | 342 | |
| GAK | NAK | Other | 5y7z | A | | gefitinib | Human | 10332 | |
| GAK | NAK | Other | 5y7z | B | | gefitinib | Human | 10331 | |
| GAK | NAK | Other | 5y80 | A | A | gefitinib | Human | 10329 | |
| GAK | NAK | Other | 5y80 | A | B | gefitinib | Human | 10330 | |
| GRK2 (BARK1) | GRK | AGC | 3cik | A | | - | Human | 1706 | |
| GRK2 (BARK1) | GRK | AGC | 3krw | A | | balanol | Human | 1707 | |
| GRK2 (BARK1) | GRK | AGC | 3krx | A | | balanol | Human | 1709 | |
| GRK2 (BARK1) | GRK | AGC | 3v5w | A | A | paroxetine | Human | 1705 | |
| GRK2 (BARK1) | GRK | AGC | 3v5w | A | B | paroxetine | Human | 1711 | |
| GRK2 (BARK1) | GRK | AGC | 4mk0 | A | A | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-one | Human | 1710 | |
| GRK2 (BARK1) | GRK | AGC | 4mk0 | A | B | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-one | Human | 1704 | |
| GRK2 (BARK1) | GRK | AGC | 4pnk | A | A | (4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide | Human | 1703 | |
| GRK2 (BARK1) | GRK | AGC | 4pnk | A | B | (4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide | Human | 1708 | |
| GRK2 (BARK1) | GRK | AGC | 5he1 | A | A | (4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamide | Human | 6605 | |
| GRK2 (BARK1) | GRK | AGC | 5he1 | A | B | (4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamide | Human | 6606 | |
| GRK2 (BARK1) | GRK | AGC | 5ukk | A | A | 5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamide | Human | 7529 | |
| GRK2 (BARK1) | GRK | AGC | 5ukk | A | B | 5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamide | Human | 7530 | |
| GRK2 (BARK1) | GRK | AGC | 5ukl | A | A | 2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamide | Human | 7528 | |
| GRK2 (BARK1) | GRK | AGC | 5ukl | A | B | 2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamide | Human | 7531 | |
| GRK2 (BARK1) | GRK | AGC | 5uuu | A | A | 3-({[4-methyl-5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)-n-[2-(trifluoromethyl)benzyl]benzamide | Human | 8255 | |
| GRK2 (BARK1) | GRK | AGC | 5uuu | A | B | 3-({[4-methyl-5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)-n-[2-(trifluoromethyl)benzyl]benzamide | Human | 8254 | |
| GRK2 (BARK1) | GRK | AGC | 5uvc | A | | n-benzyl-3-({[5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)benzamide | Human | 8256 | |
| GRK2 (BARK1) | GRK | AGC | 5wg3 | A | | 2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(1h-pyrazol-3-yl)methyl]benzamide | Human | 9439 | |
| GRK2 (BARK1) | GRK | AGC | 5wg4 | A | A | 2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamide | Human | 9441 | |
| GRK2 (BARK1) | GRK | AGC | 5wg4 | A | B | 2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamide | Human | 9438 | |
| GRK2 (BARK1) | GRK | AGC | 5wg5 | A | A | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazole | Human | 9437 | |
| GRK2 (BARK1) | GRK | AGC | 5wg5 | A | B | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazole | Human | 9440 | |
| GRK2 (BARK1) | GRK | AGC | 6c2y | A | | (4r,5r,6s)-4-[4-fluoro-3-({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}carbamoyl)phenyl]-n-(2h-indazol-5-yl)-6-methyl-2-oxohexahydropyrimidine-5-carboxamide | Human | 9854 | |
| GRK2 (BARK1) | GRK | AGC | 6u7c | A | | 5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(2h-indazol-3-yl)methyl]benzamide | Human | 12162 | |
| GRK2 (BARK1) | GRK | AGC | 7k7l | A | A | 3-benzyl-6-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | 12960 | |
| GRK2 (BARK1) | GRK | AGC | 7k7l | A | B | 3-benzyl-6-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | 12958 | |
| GRK2 (BARK1) | GRK | AGC | 7k7z | A | A | 3-benzyl-7-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | 12959 | |
| GRK2 (BARK1) | GRK | AGC | 7k7z | A | B | 3-benzyl-7-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | 12961 | |
| GRK2 (BARK1) | GRK | AGC | 7pwd | A | A | 4-chloranyl-n-[2-(4-chlorophenyl)ethyl]thieno[2,3-c]pyridine-2-carboxamide | Human | 13949 | |
| GRK2 (BARK1) | GRK | AGC | 7pwd | A | B | 4-chloranyl-n-[2-(4-chlorophenyl)ethyl]thieno[2,3-c]pyridine-2-carboxamide | Human | 13950 | |
| GRK4 (GPRK4) | GRK | AGC | 4yhj | A | | amp phosphoramidate | Human | 422 | |
| GRK4 (GPRK4) | GRK | AGC | 4yhj | B | | amp phosphoramidate | Human | 423 | |
| GRK5 (GPRK5) | GRK | AGC | 4tnb | A | | sangivamycin | Human | 3276 | |
| GRK5 (GPRK5) | GRK | AGC | 4tnd | A | | phosphoaminophosphonic acid-adenylate ester | Human | 3275 | |
| GRK5 (GPRK5) | GRK | AGC | 6pjx | A | A | sangivamycin | Human | 13042 | |
| GRK5 (GPRK5) | GRK | AGC | 6pjx | A | B | sangivamycin | Human | 13041 | |
| GRK5 (GPRK5) | GRK | AGC | 8uap | A | | (3z)-3-{[4-(2-chloroacetamido)-3,5-dimethyl-1h-pyrrol-2-yl]methylidene}-n-[(1r)-1-(4-fluorophenyl)ethyl]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 15093 | |
| GRK5 (GPRK5) | GRK | AGC | 8uaq | A | | (3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-[(4-{[(2s)-2-(furan-2-yl)-2-hydroxyacetyl]amino}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 15092 | |
| GRK6 (GPRK6) | GRK | AGC | 2acx | A | | phosphoaminophosphonic acid-adenylate ester | Human | 420 | |
| GRK6 (GPRK6) | GRK | AGC | 2acx | B | | phosphoaminophosphonic acid-adenylate ester | Human | 417 | |
| GRK6 (GPRK6) | GRK | AGC | 3nyn | A | | sangivamycin | Human | 419 | |
| GRK6 (GPRK6) | GRK | AGC | 3nyn | B | | sangivamycin | Human | 416 | |
| GRK6 (GPRK6) | GRK | AGC | 3nyo | A | | adenosine monophosphate | Human | 418 | |
| GRK6 (GPRK6) | GRK | AGC | 3nyo | B | | adenosine monophosphate | Human | 421 | |
| GSK3A | GSK | CMGC | 7sxf | A | A | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 14781 | |
| GSK3A | GSK | CMGC | 7sxf | A | B | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 14780 | |
| GSK3A | GSK | CMGC | 7sxg | A | A | (4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-ol | Human | 14783 | |
| GSK3A | GSK | CMGC | 7sxg | A | B | (4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-ol | Human | 14782 | |
| Gsk3b (GSK3B) | GSK | CMGC | 4nu1 | A | A | adenosine-5'-diphosphate | Mouse | 5699 | |
| Gsk3b (GSK3B) | GSK | CMGC | 4nu1 | A | B | adenosine-5'-diphosphate | Mouse | 5700 | |
| Gsk3b (GSK3B) | GSK | CMGC | 5air | A | | - | Mouse | 6863 | |
| Gsk3b (GSK3B) | GSK | CMGC | 5air | B | | - | Mouse | 6864 | |
| Gsk3b (GSK3B) | GSK | CMGC | 6ae3 | A | | 2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-one | Mouse | 10607 | |
| Gsk3b (GSK3B) | GSK | CMGC | 6ae3 | B | | 2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-one | Mouse | 10606 | |
| Gsk3b (GSK3B) | GSK | CMGC | 6ae3 | C | | - | Mouse | 10605 | |
| Gsk3b (GSK3B) | GSK | CMGC | 6ae3 | D | | - | Mouse | 10604 | |
| Gsk3b (GSK3B) | GSK | CMGC | 8vme | A | A | adenosine-5'-diphosphate | Mouse | 15398 | |
| Gsk3b (GSK3B) | GSK | CMGC | 8vme | A | B | adenosine-5'-diphosphate | Mouse | 15399 | |
| Gsk3b (GSK3B) | GSK | CMGC | 8vmf | A | A | adenosine-5'-diphosphate | Mouse | 15400 | |
| Gsk3b (GSK3B) | GSK | CMGC | 8vmf | A | B | adenosine-5'-diphosphate | Mouse | 15401 | |
| Gsk3b (GSK3B) | GSK | CMGC | 8vmg | A | A | adenosine-5'-diphosphate | Mouse | 15397 | |
| Gsk3b (GSK3B) | GSK | CMGC | 8vmg | A | B | adenosine-5'-diphosphate | Mouse | 15396 | |
| GSK3B | GSK | CMGC | 1gng | A | | - | Human | 665 | |
| GSK3B | GSK | CMGC | 1gng | B | | - | Human | 700 | |
| GSK3B | GSK | CMGC | 1h8f | A | | - | Human | 745 | |
| GSK3B | GSK | CMGC | 1h8f | B | | - | Human | 666 | |
| GSK3B | GSK | CMGC | 1i09 | A | | - | Human | 630 | |
| GSK3B | GSK | CMGC | 1i09 | B | | - | Human | 638 | |
| GSK3B | GSK | CMGC | 1j1b | A | | phosphoaminophosphonic acid-adenylate ester | Human | 707 | |
| GSK3B | GSK | CMGC | 1j1b | B | | phosphoaminophosphonic acid-adenylate ester | Human | 657 | |
| GSK3B | GSK | CMGC | 1j1c | A | | adenosine-5'-diphosphate | Human | 696 | |
| GSK3B | GSK | CMGC | 1j1c | B | | adenosine-5'-diphosphate | Human | 677 | |
| GSK3B | GSK | CMGC | 1o9u | A | | 9-methyl-9h-purin-6-amine | Human | 708 | |
| GSK3B | GSK | CMGC | 1pyx | A | | phosphoaminophosphonic acid-adenylate ester | Human | 645 | |
| GSK3B | GSK | CMGC | 1pyx | B | | phosphoaminophosphonic acid-adenylate ester | Human | 663 | |
| GSK3B | GSK | CMGC | 1q3d | A | | staurosporine | Human | 705 | |
| GSK3B | GSK | CMGC | 1q3d | B | | staurosporine | Human | 752 | |
| GSK3B | GSK | CMGC | 1q3w | A | | 9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-one | Human | 635 | |
| GSK3B | GSK | CMGC | 1q3w | B | | 9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-one | Human | 693 | |
| GSK3B | GSK | CMGC | 1q41 | A | | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | 628 | |
| GSK3B | GSK | CMGC | 1q41 | B | | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | 658 | |
| GSK3B | GSK | CMGC | 1q4l | A | | 2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acid | Human | 714 | |
| GSK3B | GSK | CMGC | 1q4l | B | | 2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acid | Human | 655 | |
| GSK3B | GSK | CMGC | 1q5k | A | | n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea | Human | 680 | |
| GSK3B | GSK | CMGC | 1q5k | B | | n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea | Human | 651 | |
| GSK3B | GSK | CMGC | 1r0e | A | A | 3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 733 | |
| GSK3B | GSK | CMGC | 1r0e | A | B | 3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 672 | |
| GSK3B | GSK | CMGC | 1r0e | B | A | 3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 687 | |
| GSK3B | GSK | CMGC | 1r0e | B | B | 3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 639 | |
| GSK3B | GSK | CMGC | 1uv5 | A | | 6-bromoindirubin-3'-oxime | Human | 759 | |
| GSK3B | GSK | CMGC | 2jld | A | A | ruthenium pyridocarbazole | Human | 7213 | |
| GSK3B | GSK | CMGC | 2jld | A | B | ruthenium pyridocarbazole | Human | 7214 | |
| GSK3B | GSK | CMGC | 2jld | B | A | ruthenium pyridocarbazole | Human | 7205 | |
| GSK3B | GSK | CMGC | 2jld | B | B | ruthenium pyridocarbazole | Human | 7209 | |
| GSK3B | GSK | CMGC | 2o5k | A | | 2-(2,4-dichloro-phenyl)-7-hydroxy-1h-benzoimidazole-4-carboxylic acid [2-(4-methanesulfonylamino-phenyl)-ethyl]-amide | Human | 633 | |
| GSK3B | GSK | CMGC | 2ow3 | A | | bis-(indole)maleimide pyridinophane | Human | 698 | |
| GSK3B | GSK | CMGC | 2ow3 | B | | bis-(indole)maleimide pyridinophane | Human | 649 | |
| GSK3B | GSK | CMGC | 3du8 | A | | (7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 701 | |
| GSK3B | GSK | CMGC | 3du8 | B | | (7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 737 | |
| GSK3B | GSK | CMGC | 3f7z | A | A | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 743 | |
| GSK3B | GSK | CMGC | 3f7z | A | B | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 647 | |
| GSK3B | GSK | CMGC | 3f7z | A | C | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 685 | |
| GSK3B | GSK | CMGC | 3f7z | B | A | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 749 | |
| GSK3B | GSK | CMGC | 3f7z | B | B | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 670 | |
| GSK3B | GSK | CMGC | 3f7z | B | C | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 686 | |
| GSK3B | GSK | CMGC | 3f88 | A | A | 5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 741 | |
| GSK3B | GSK | CMGC | 3f88 | A | B | 5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 679 | |
| GSK3B | GSK | CMGC | 3f88 | B | A | 5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 744 | |
| GSK3B | GSK | CMGC | 3f88 | B | B | 5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 756 | |
| GSK3B | GSK | CMGC | 3gb2 | A | A | 2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazole | Human | 727 | |
| GSK3B | GSK | CMGC | 3gb2 | A | B | 2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazole | Human | 734 | |
| GSK3B | GSK | CMGC | 3i4b | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamide | Human | 646 | |
| GSK3B | GSK | CMGC | 3i4b | B | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamide | Human | 629 | |
| GSK3B | GSK | CMGC | 3l1s | A | | (4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-one | Human | 757 | |
| GSK3B | GSK | CMGC | 3l1s | B | | (4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-one | Human | 713 | |
| GSK3B | GSK | CMGC | 3m1s | A | A | ruthenium pyridocarbazole | Human | 7212 | |
| GSK3B | GSK | CMGC | 3m1s | A | B | ruthenium pyridocarbazole | Human | 7206 | |
| GSK3B | GSK | CMGC | 3m1s | B | A | ruthenium pyridocarbazole | Human | 7210 | |
| GSK3B | GSK | CMGC | 3m1s | B | B | ruthenium pyridocarbazole | Human | 7208 | |
| GSK3B | GSK | CMGC | 3pup | A | | ruthenium octasporine | Human | 7207 | |
| GSK3B | GSK | CMGC | 3pup | B | | ruthenium octasporine | Human | 7211 | |
| GSK3B | GSK | CMGC | 3q3b | A | | 4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-one | Human | 660 | |
| GSK3B | GSK | CMGC | 3q3b | B | | 4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-one | Human | 674 | |
| GSK3B | GSK | CMGC | 3say | A | A | (3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamide | Human | 738 | |
| GSK3B | GSK | CMGC | 3say | A | B | (3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamide | Human | 661 | |
| GSK3B | GSK | CMGC | 3say | B | A | (3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamide | Human | 682 | |
| GSK3B | GSK | CMGC | 3say | B | B | (3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamide | Human | 710 | |
| GSK3B | GSK | CMGC | 3sd0 | A | | 3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dione | Human | 720 | |
| GSK3B | GSK | CMGC | 3sd0 | B | | 3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dione | Human | 673 | |
| GSK3B | GSK | CMGC | 3zdi | A | | 3,6-diamino-4-(2-chlorophenyl)thieno[2,3-b]pyridine-2,5-dicarbonitrile | Human | 748 | |
| GSK3B | GSK | CMGC | 3zrk | A | A | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 675 | |
| GSK3B | GSK | CMGC | 3zrk | A | B | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 644 | |
| GSK3B | GSK | CMGC | 3zrk | A | C | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 697 | |
| GSK3B | GSK | CMGC | 3zrk | B | A | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 637 | |
| GSK3B | GSK | CMGC | 3zrk | B | B | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 662 | |
| GSK3B | GSK | CMGC | 3zrk | B | C | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 731 | |
| GSK3B | GSK | CMGC | 3zrl | A | A | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 712 | |
| GSK3B | GSK | CMGC | 3zrl | A | B | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 725 | |
| GSK3B | GSK | CMGC | 3zrl | A | C | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 654 | |
| GSK3B | GSK | CMGC | 3zrl | B | A | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 718 | |
| GSK3B | GSK | CMGC | 3zrl | B | B | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 691 | |
| GSK3B | GSK | CMGC | 3zrl | B | C | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 676 | |
| GSK3B | GSK | CMGC | 3zrm | A | A | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 751 | |
| GSK3B | GSK | CMGC | 3zrm | A | B | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 648 | |
| GSK3B | GSK | CMGC | 3zrm | A | C | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 724 | |
| GSK3B | GSK | CMGC | 3zrm | B | A | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 753 | |
| GSK3B | GSK | CMGC | 3zrm | B | B | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 652 | |
| GSK3B | GSK | CMGC | 3zrm | B | C | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 706 | |
| GSK3B | GSK | CMGC | 4acc | A | | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 704 | |
| GSK3B | GSK | CMGC | 4acc | B | | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 669 | |
| GSK3B | GSK | CMGC | 4acd | A | | 3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 723 | |
| GSK3B | GSK | CMGC | 4acd | B | | 3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 692 | |
| GSK3B | GSK | CMGC | 4acg | A | | 2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamide | Human | 681 | |
| GSK3B | GSK | CMGC | 4acg | B | | 2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamide | Human | 721 | |
| GSK3B | GSK | CMGC | 4ach | A | | 3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamide | Human | 653 | |
| GSK3B | GSK | CMGC | 4ach | B | | 3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamide | Human | 702 | |
| GSK3B | GSK | CMGC | 4afj | A | A | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 632 | |
| GSK3B | GSK | CMGC | 4afj | A | B | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 683 | |
| GSK3B | GSK | CMGC | 4afj | A | C | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 742 | |
| GSK3B | GSK | CMGC | 4afj | B | A | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 678 | |
| GSK3B | GSK | CMGC | 4afj | B | B | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 726 | |
| GSK3B | GSK | CMGC | 4afj | B | C | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 711 | |
| GSK3B | GSK | CMGC | 4b7t | A | | (5z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-methyl-2-(propan-2-ylamino)imidazol-4-one | Human | 732 | |
| GSK3B | GSK | CMGC | 4dit | A | | n-(pyridin-3-yl)-2-(thiophen-3-yl)-3h-imidazo[4,5-b]pyridine-7-carboxamide | Human | 689 | |
| GSK3B | GSK | CMGC | 4iq6 | A | | 6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amine | Human | 728 | |
| GSK3B | GSK | CMGC | 4iq6 | B | | 6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amine | Human | 750 | |
| GSK3B | GSK | CMGC | 4j1r | A | | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 709 | |
| GSK3B | GSK | CMGC | 4j1r | B | | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 656 | |
| GSK3B | GSK | CMGC | 4j1r | C | | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 688 | |
| GSK3B | GSK | CMGC | 4j1r | D | | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 736 | |
| GSK3B | GSK | CMGC | 4j71 | A | A | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 642 | |
| GSK3B | GSK | CMGC | 4j71 | A | B | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 690 | |
| GSK3B | GSK | CMGC | 4j71 | B | A | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 641 | |
| GSK3B | GSK | CMGC | 4j71 | B | B | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 739 | |
| GSK3B | GSK | CMGC | 4nm0 | A | A | adenosine-5'-diphosphate | Human | 715 | |
| GSK3B | GSK | CMGC | 4nm0 | A | B | adenosine-5'-diphosphate | Human | 671 | |
| GSK3B | GSK | CMGC | 4nm3 | A | A | adenosine-5'-diphosphate | Human | 730 | |
| GSK3B | GSK | CMGC | 4nm3 | A | B | adenosine-5'-diphosphate | Human | 640 | |
| GSK3B | GSK | CMGC | 4nm5 | A | A | adenosine-5'-diphosphate | Human | 755 | |
| GSK3B | GSK | CMGC | 4nm5 | A | B | adenosine-5'-diphosphate | Human | 694 | |
| GSK3B | GSK | CMGC | 4nm7 | A | A | adenosine-5'-diphosphate | Human | 695 | |
| GSK3B | GSK | CMGC | 4nm7 | A | B | adenosine-5'-diphosphate | Human | 684 | |
| GSK3B | GSK | CMGC | 4ptc | A | A | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | 664 | |
| GSK3B | GSK | CMGC | 4ptc | A | B | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | 659 | |
| GSK3B | GSK | CMGC | 4ptc | B | A | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | 747 | |
| GSK3B | GSK | CMGC | 4ptc | B | B | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | 758 | |
| GSK3B | GSK | CMGC | 4pte | A | A | n-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamide | Human | 716 | |
| GSK3B | GSK | CMGC | 4pte | A | B | n-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamide | Human | 717 | |
| GSK3B | GSK | CMGC | 4pte | B | A | n-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamide | Human | 722 | |
| GSK3B | GSK | CMGC | 4pte | B | B | n-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamide | Human | 667 | |
| GSK3B | GSK | CMGC | 4ptg | A | A | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamide | Human | 735 | |
| GSK3B | GSK | CMGC | 4ptg | A | B | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamide | Human | 634 | |
| GSK3B | GSK | CMGC | 4ptg | B | A | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamide | Human | 740 | |
| GSK3B | GSK | CMGC | 4ptg | B | B | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamide | Human | 754 | |
| GSK3B | GSK | CMGC | 5f94 | A | A | 2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamide | Human | 6374 | |
| GSK3B | GSK | CMGC | 5f94 | A | B | 2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamide | Human | 6369 | |
| GSK3B | GSK | CMGC | 5f94 | B | A | 2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamide | Human | 6372 | |
| GSK3B | GSK | CMGC | 5f94 | B | B | 2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamide | Human | 6371 | |
| GSK3B | GSK | CMGC | 5f95 | A | | 2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamide | Human | 6373 | |
| GSK3B | GSK | CMGC | 5f95 | B | | 2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamide | Human | 6370 | |
| GSK3B | GSK | CMGC | 5hln | A | | chir99021 | Human | 6649 | |
| GSK3B | GSK | CMGC | 5hln | B | | chir99021 | Human | 6650 | |
| GSK3B | GSK | CMGC | 5hlp | A | A | 4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-one | Human | 6647 | |
| GSK3B | GSK | CMGC | 5hlp | A | B | 4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-one | Human | 6648 | |
| GSK3B | GSK | CMGC | 5hlp | B | A | 4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-one | Human | 6646 | |
| GSK3B | GSK | CMGC | 5hlp | B | B | 4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-one | Human | 6645 | |
| GSK3B | GSK | CMGC | 5k5n | A | | 5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamide | Human | 7411 | |
| GSK3B | GSK | CMGC | 5k5n | B | | 5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamide | Human | 7410 | |
| GSK3B | GSK | CMGC | 5kpk | A | | (4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9735 | |
| GSK3B | GSK | CMGC | 5kpk | B | | (4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9731 | |
| GSK3B | GSK | CMGC | 5kpl | A | A | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9729 | |
| GSK3B | GSK | CMGC | 5kpl | A | B | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9730 | |
| GSK3B | GSK | CMGC | 5kpl | B | A | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9728 | |
| GSK3B | GSK | CMGC | 5kpl | B | B | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9733 | |
| GSK3B | GSK | CMGC | 5kpm | A | | (4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9732 | |
| GSK3B | GSK | CMGC | 5kpm | B | | (4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9734 | |
| GSK3B | GSK | CMGC | 5oy4 | A | | ~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamide | Human | 8621 | |
| GSK3B | GSK | CMGC | 5oy4 | B | | ~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamide | Human | 8622 | |
| GSK3B | GSK | CMGC | 5t31 | A | | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9565 | |
| GSK3B | GSK | CMGC | 5t31 | B | | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9564 | |
| GSK3B | GSK | CMGC | 6b8j | A | A | chir99021 | Human | 8658 | |
| GSK3B | GSK | CMGC | 6b8j | A | B | chir99021 | Human | 8659 | |
| GSK3B | GSK | CMGC | 6gjo | A | | (3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-one | Human | 10974 | |
| GSK3B | GSK | CMGC | 6gjo | B | | (3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-one | Human | 10973 | |
| GSK3B | GSK | CMGC | 6gn1 | A | | ~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamide | Human | 9997 | |
| GSK3B | GSK | CMGC | 6gn1 | B | | ~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamide | Human | 9996 | |
| GSK3B | GSK | CMGC | 6h0u | A | | (2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamide | Human | 11049 | |
| GSK3B | GSK | CMGC | 6h0u | B | | (2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamide | Human | 11050 | |
| GSK3B | GSK | CMGC | 6hk3 | A | A | 3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11425 | |
| GSK3B | GSK | CMGC | 6hk3 | A | B | 3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11426 | |
| GSK3B | GSK | CMGC | 6hk3 | B | A | 3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11422 | |
| GSK3B | GSK | CMGC | 6hk3 | B | B | 3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11424 | |
| GSK3B | GSK | CMGC | 6hk4 | A | A | 3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamide | Human | 11429 | |
| GSK3B | GSK | CMGC | 6hk4 | A | B | 3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamide | Human | 11423 | |
| GSK3B | GSK | CMGC | 6hk4 | B | A | 3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamide | Human | 11430 | |
| GSK3B | GSK | CMGC | 6hk4 | B | B | 3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamide | Human | 11427 | |
| GSK3B | GSK | CMGC | 6hk7 | A | | 3-azanyl-~{n}-(2-methoxyethyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11428 | |
| GSK3B | GSK | CMGC | 6tcu | A | A | 5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamide | Human | 12780 | |
| GSK3B | GSK | CMGC | 6tcu | A | B | 5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamide | Human | 12781 | |
| GSK3B | GSK | CMGC | 6v6l | A | A | - | Human | 11913 | |
| GSK3B | GSK | CMGC | 6v6l | A | B | - | Human | 11912 | |
| GSK3B | GSK | CMGC | 6y9r | A | A | ~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamide | Human | 12287 | |
| GSK3B | GSK | CMGC | 6y9r | A | B | ~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamide | Human | 12289 | |
| GSK3B | GSK | CMGC | 6y9s | A | A | ~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamide | Human | 12286 | |
| GSK3B | GSK | CMGC | 6y9s | A | B | ~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamide | Human | 12290 | |
| GSK3B | GSK | CMGC | 6y9s | B | A | ~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamide | Human | 12285 | |
| GSK3B | GSK | CMGC | 6y9s | B | B | ~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamide | Human | 12288 | |
| GSK3B | GSK | CMGC | 7b6f | A | A | 3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrile | Human | 13069 | |
| GSK3B | GSK | CMGC | 7b6f | A | B | 3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrile | Human | 13070 | |
| GSK3B | GSK | CMGC | 7oy5 | A | A | ~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamine | Human | 14118 | |
| GSK3B | GSK | CMGC | 7oy5 | A | B | ~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamine | Human | 14119 | |
| GSK3B | GSK | CMGC | 7sxh | A | A | (4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-ol | Human | 14787 | |
| GSK3B | GSK | CMGC | 7sxh | A | B | (4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-ol | Human | 14784 | |
| GSK3B | GSK | CMGC | 7sxj | A | A | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 14785 | |
| GSK3B | GSK | CMGC | 7sxj | A | B | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 14786 | |
| GSK3B | GSK | CMGC | 7u2z | A | A | (3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamide | Human | 14203 | |
| GSK3B | GSK | CMGC | 7u2z | A | B | (3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamide | Human | 14202 | |
| GSK3B | GSK | CMGC | 7u31 | A | A | 5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amine | Human | 14199 | |
| GSK3B | GSK | CMGC | 7u31 | A | B | 5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amine | Human | 14201 | |
| GSK3B | GSK | CMGC | 7u33 | A | A | 3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamide | Human | 14198 | |
| GSK3B | GSK | CMGC | 7u33 | A | B | 3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamide | Human | 14200 | |
| GSK3B | GSK | CMGC | 7u36 | A | | (3s)-1-[(2-fluorophenoxy)acetyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamide | Human | 14204 | |
| GSK3B | GSK | CMGC | 7z1f | A | | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 14663 | |
| GSK3B | GSK | CMGC | 7z1g | A | | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 14662 | |
| GSK3B | GSK | CMGC | 8auz | A | A | 8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxaline | Human | 14707 | |
| GSK3B | GSK | CMGC | 8auz | A | B | 8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxaline | Human | 14708 | |
| GSK3B | GSK | CMGC | 8av1 | A | A | 2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxaline | Human | 14706 | |
| GSK3B | GSK | CMGC | 8av1 | A | B | 2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxaline | Human | 14709 | |
| GSK3B | GSK | CMGC | 8djc | A | A | (4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamide | Human | 14672 | |
| GSK3B | GSK | CMGC | 8djc | A | B | (4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamide | Human | 14669 | |
| GSK3B | GSK | CMGC | 8djd | A | A | 2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamide | Human | 14673 | |
| GSK3B | GSK | CMGC | 8djd | A | B | 2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamide | Human | 14668 | |
| GSK3B | GSK | CMGC | 8dje | A | A | (4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamide | Human | 14670 | |
| GSK3B | GSK | CMGC | 8dje | A | B | (4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamide | Human | 14671 | |
| GSK3B | GSK | CMGC | 8ff8 | A | | 2-(4-cyanoanilino)-n-(4-phenylpyridin-3-yl)pyrimidine-4-carboxamide | Human | 14763 | |
| GSK3B | GSK | CMGC | 8qji | A | | n-[4-[5-(1,2,4-oxadiazol-3-yl)thiophen-2-yl]pyridin-2-yl]cyclopropanecarboxamide | Human | 15386 | |
| GUCY2C (HSER) | RGC | RGC | 8fx4 | D | | - | Human | 14837 | |
| HASPIN (Haspin) | Haspin | Other | 2vuw | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 3809 | |
| HASPIN (Haspin) | Haspin | Other | 2vuw | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 3801 | |
| HASPIN (Haspin) | Haspin | Other | 2wb8 | A | A | - | Human | 3802 | |
| HASPIN (Haspin) | Haspin | Other | 2wb8 | A | B | - | Human | 3815 | |
| HASPIN (Haspin) | Haspin | Other | 3dlz | A | A | adenosine monophosphate | Human | 3804 | |
| HASPIN (Haspin) | Haspin | Other | 3dlz | A | B | adenosine monophosphate | Human | 3808 | |
| HASPIN (Haspin) | Haspin | Other | 3e7v | A | A | 3-(3-aminophenyl)-n-(3-chlorophenyl)pyrazolo[1,5-a]pyrimidin-5-amine | Human | 3814 | |
| HASPIN (Haspin) | Haspin | Other | 3e7v | A | B | 3-(3-aminophenyl)-n-(3-chlorophenyl)pyrazolo[1,5-a]pyrimidin-5-amine | Human | 3799 | |
| HASPIN (Haspin) | Haspin | Other | 3f2n | A | A | (2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-ol | Human | 3803 | |
| HASPIN (Haspin) | Haspin | Other | 3f2n | A | B | (2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-ol | Human | 3813 | |
| HASPIN (Haspin) | Haspin | Other | 3fmd | A | A | n-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamide | Human | 3798 | |
| HASPIN (Haspin) | Haspin | Other | 3fmd | A | B | n-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamide | Human | 3810 | |
| HASPIN (Haspin) | Haspin | Other | 3iq7 | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 3807 | |
| HASPIN (Haspin) | Haspin | Other | 3iq7 | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 3811 | |
| HASPIN (Haspin) | Haspin | Other | 4ouc | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 3806 | |
| HASPIN (Haspin) | Haspin | Other | 4ouc | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 3812 | |
| HASPIN (Haspin) | Haspin | Other | 4qtc | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 3805 | |
| HASPIN (Haspin) | Haspin | Other | 4qtc | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 3800 | |
| HASPIN (Haspin) | Haspin | Other | 5htb | A | A | - | Human | 6620 | |
| HASPIN (Haspin) | Haspin | Other | 5htb | A | B | - | Human | 6621 | |
| HASPIN (Haspin) | Haspin | Other | 5htc | A | A | - | Human | 6445 | |
| HASPIN (Haspin) | Haspin | Other | 5htc | A | B | - | Human | 6446 | |
| HASPIN (Haspin) | Haspin | Other | 5htc | A | C | - | Human | 6444 | |
| HASPIN (Haspin) | Haspin | Other | 6g34 | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9832 | |
| HASPIN (Haspin) | Haspin | Other | 6g34 | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9846 | |
| HASPIN (Haspin) | Haspin | Other | 6g35 | A | A | 5-bromotubercidin | Human | 9843 | |
| HASPIN (Haspin) | Haspin | Other | 6g35 | A | B | 5-bromotubercidin | Human | 9841 | |
| HASPIN (Haspin) | Haspin | Other | 6g35 | A | C | - | Human | 9837 | |
| HASPIN (Haspin) | Haspin | Other | 6g35 | A | D | - | Human | 9829 | |
| HASPIN (Haspin) | Haspin | Other | 6g36 | A | A | 5-chlorotubercidin | Human | 9834 | |
| HASPIN (Haspin) | Haspin | Other | 6g36 | A | B | 5-chlorotubercidin | Human | 9844 | |
| HASPIN (Haspin) | Haspin | Other | 6g37 | A | A | 5-fluorotubercidin | Human | 9840 | |
| HASPIN (Haspin) | Haspin | Other | 6g37 | A | B | 5-fluorotubercidin | Human | 9845 | |
| HASPIN (Haspin) | Haspin | Other | 6g38 | A | A | '2-(4-amino-pyrrolo[2,3-d]pyrimidin-7-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol | Human | 9830 | |
| HASPIN (Haspin) | Haspin | Other | 6g38 | A | B | '2-(4-amino-pyrrolo[2,3-d]pyrimidin-7-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diol | Human | 9842 | |
| HASPIN (Haspin) | Haspin | Other | 6g39 | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9839 | |
| HASPIN (Haspin) | Haspin | Other | 6g39 | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9831 | |
| HASPIN (Haspin) | Haspin | Other | 6g39 | A | C | - | Human | 9838 | |
| HASPIN (Haspin) | Haspin | Other | 6g39 | A | D | - | Human | 9833 | |
| HASPIN (Haspin) | Haspin | Other | 6g3a | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9836 | |
| HASPIN (Haspin) | Haspin | Other | 6g3a | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9835 | |
| HASPIN (Haspin) | Haspin | Other | 6z56 | A | A | 6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12322 | |
| HASPIN (Haspin) | Haspin | Other | 6z56 | A | B | 6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12333 | |
| HASPIN (Haspin) | Haspin | Other | 6z56 | A | C | 6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12320 | |
| HASPIN (Haspin) | Haspin | Other | 6z57 | A | A | 10-(2-morpholin-4-ylethyl)-7-oxa-10,13,17,18,21-pentazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene | Human | 12321 | |
| HASPIN (Haspin) | Haspin | Other | 6z57 | A | B | 10-(2-morpholin-4-ylethyl)-7-oxa-10,13,17,18,21-pentazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene | Human | 12323 | |
| HASPIN (Haspin) | Haspin | Other | 6z58 | A | A | 8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-one | Human | 12327 | |
| HASPIN (Haspin) | Haspin | Other | 6z58 | A | B | 8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-one | Human | 12332 | |
| HASPIN (Haspin) | Haspin | Other | 6z59 | A | A | 11-oxa-8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-one | Human | 12326 | |
| HASPIN (Haspin) | Haspin | Other | 6z59 | A | B | 11-oxa-8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-one | Human | 12316 | |
| HASPIN (Haspin) | Haspin | Other | 6z5a | A | A | n-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide | Human | 12328 | |
| HASPIN (Haspin) | Haspin | Other | 6z5a | A | B | n-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide | Human | 12324 | |
| HASPIN (Haspin) | Haspin | Other | 6z5b | A | A | 6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12331 | |
| HASPIN (Haspin) | Haspin | Other | 6z5b | A | B | 6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12334 | |
| HASPIN (Haspin) | Haspin | Other | 6z5c | A | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12319 | |
| HASPIN (Haspin) | Haspin | Other | 6z5c | A | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12318 | |
| HASPIN (Haspin) | Haspin | Other | 6z5d | A | A | 11-methyl-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one | Human | 12325 | |
| HASPIN (Haspin) | Haspin | Other | 6z5d | A | B | 11-methyl-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one | Human | 12330 | |
| HASPIN (Haspin) | Haspin | Other | 6z5e | A | A | 11-cyclopropyl-14-(2-hydroxyethyl)-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one | Human | 12317 | |
| HASPIN (Haspin) | Haspin | Other | 6z5e | A | B | 11-cyclopropyl-14-(2-hydroxyethyl)-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one | Human | 12329 | |
| HASPIN (Haspin) | Haspin | Other | 7avq | A | A | (2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-ol | Human | 13176 | |
| HASPIN (Haspin) | Haspin | Other | 7avq | A | B | (2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-ol | Human | 13175 | |
| HASPIN (Haspin) | Haspin | Other | 7ops | A | | 2-methylsulfanyl-10-nitro-pyrido[3,4-g]quinazoline | Human | 13815 | |
| HASPIN (Haspin) | Haspin | Other | 7sqm | A | A | 1-[(4s)-5-(2,4-difluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-4-methylpiperidin-4-amine | Human | 14033 | |
| HASPIN (Haspin) | Haspin | Other | 7sqm | A | B | 1-[(4s)-5-(2,4-difluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-4-methylpiperidin-4-amine | Human | 14032 | |
| HASPIN (Haspin) | Haspin | Other | 8rdk | A | | 3-pyridin-4-yl-1~{h}-pyrrolo[3,2-g]isoquinoline | Human | 15259 | |
| HCK | Src | TK | 1ad5 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 9480 | |
| HCK | Src | TK | 1ad5 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 9483 | |
| HCK | Src | TK | 1qcf | A | | 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 2641 | |
| HCK | Src | TK | 2c0i | A | A | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2662 | |
| HCK | Src | TK | 2c0i | A | B | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2649 | |
| HCK | Src | TK | 2c0i | B | A | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2650 | |
| HCK | Src | TK | 2c0i | B | B | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2640 | |
| HCK | Src | TK | 2c0o | A | A | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2666 | |
| HCK | Src | TK | 2c0o | A | B | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2652 | |
| HCK | Src | TK | 2c0o | B | A | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2663 | |
| HCK | Src | TK | 2c0o | B | B | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2657 | |
| HCK | Src | TK | 2c0t | A | A | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2653 | |
| HCK | Src | TK | 2c0t | A | B | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2667 | |
| HCK | Src | TK | 2c0t | B | A | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2642 | |
| HCK | Src | TK | 2c0t | B | B | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2634 | |
| HCK | Src | TK | 2hck | A | | 3,5,7,3',4'-pentahydroxyflavone | Human | 9481 | |
| HCK | Src | TK | 2hck | B | | 3,5,7,3',4'-pentahydroxyflavone | Human | 9482 | |
| HCK | Src | TK | 2hk5 | A | | 3-{[2-(1h-benzimidazol-1-yl)-6-{[2-(diethylamino)ethyl]amino}pyrimidin-4-yl]amino}-4-methylphenol | Human | 2639 | |
| HCK | Src | TK | 3vry | A | | 4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentane | Human | 2647 | |
| HCK | Src | TK | 3vry | B | | 4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentane | Human | 2646 | |
| HCK | Src | TK | 3vrz | A | | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-benzylurea | Human | 2658 | |
| HCK | Src | TK | 3vrz | B | | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-benzylurea | Human | 2661 | |
| HCK | Src | TK | 3vs0 | A | | n-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]benzamide | Human | 2633 | |
| HCK | Src | TK | 3vs0 | B | | n-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]benzamide | Human | 2644 | |
| HCK | Src | TK | 3vs1 | A | | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-phenylurea | Human | 2635 | |
| HCK | Src | TK | 3vs1 | B | | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-phenylurea | Human | 2636 | |
| HCK | Src | TK | 3vs2 | A | | 7-[cis-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2651 | |
| HCK | Src | TK | 3vs2 | B | | 7-[cis-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2632 | |
| HCK | Src | TK | 3vs3 | A | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2643 | |
| HCK | Src | TK | 3vs3 | B | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2665 | |
| HCK | Src | TK | 3vs4 | A | | 5-(4-phenoxyphenyl)-7-(tetrahydro-2h-pyran-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2654 | |
| HCK | Src | TK | 3vs4 | B | | 5-(4-phenoxyphenyl)-7-(tetrahydro-2h-pyran-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2638 | |
| HCK | Src | TK | 3vs5 | A | | 7-(1-methylpiperidin-4-yl)-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2645 | |
| HCK | Src | TK | 3vs5 | B | | 7-(1-methylpiperidin-4-yl)-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2669 | |
| HCK | Src | TK | 3vs6 | A | | tert-butyl {4-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl}carbamate | Human | 2664 | |
| HCK | Src | TK | 3vs6 | B | | tert-butyl {4-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl}carbamate | Human | 2656 | |
| HCK | Src | TK | 3vs7 | A | | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 2659 | |
| HCK | Src | TK | 3vs7 | B | | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 2648 | |
| HCK | Src | TK | 4lud | A | | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | 2660 | |
| HCK | Src | TK | 4lud | B | | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | 2637 | |
| HCK | Src | TK | 4lue | A | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2655 | |
| HCK | Src | TK | 4lue | B | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2668 | |
| HCK | Src | TK | 5h09 | A | | ethyl (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-4-methyl-pentanoate | Human | 8537 | |
| HCK | Src | TK | 5h0b | A | | (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]azaniumyl]-4-methyl-pentanoate | Human | 8567 | |
| HCK | Src | TK | 5h0e | A | | (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-4-methyl-pentanamide | Human | 8538 | |
| HCK | Src | TK | 5h0g | A | | (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-~{n},4-dimethyl-pentanamide | Human | 8536 | |
| HCK | Src | TK | 5h0h | A | | (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-~{n},~{n},4-trimethyl-pentanamide | Human | 8539 | |
| HCK | Src | TK | 5zj6 | A | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9987 | |
| HCK | Src | TK | 5zj6 | B | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9988 | |
| HIPK2 | DYRK | CMGC | 6p5s | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11512 | |
| HIPK2 | DYRK | CMGC | 6p5s | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11513 | |
| HIPK2 | DYRK | CMGC | 7ncf | A | | 3-(4-tert-butylphenyl)-5-(1h-pyrazol-4-yl)furo[3,2-b]pyridine | Human | 13393 | |
| HIPK3 | DYRK | CMGC | 7o7i | A | | - | Human | 13996 | |
| HIPK3 | DYRK | CMGC | 7o7j | A | | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 13997 | |
| Igf1r (IGF1R) | InsR | TK | 6pyh | A | | - | Mouse | 11777 | |
| Igf1r (IGF1R) | InsR | TK | 6pyh | D | | - | Mouse | 11776 | |
| IGF1R | InsR | TK | 1jqh | A | | phosphoaminophosphonic acid-adenylate ester | Human | 999 | |
| IGF1R | InsR | TK | 1jqh | B | | phosphoaminophosphonic acid-adenylate ester | Human | 994 | |
| IGF1R | InsR | TK | 1jqh | C | | phosphoaminophosphonic acid-adenylate ester | Human | 1038 | |
| IGF1R | InsR | TK | 1k3a | A | | phosphomethylphosphonic acid adenylate ester | Human | 1028 | |
| IGF1R | InsR | TK | 1m7n | A | | - | Human | 1007 | |
| IGF1R | InsR | TK | 1m7n | B | | - | Human | 1012 | |
| IGF1R | InsR | TK | 1p4o | A | | - | Human | 1002 | |
| IGF1R | InsR | TK | 1p4o | B | | - | Human | 1026 | |
| IGF1R | InsR | TK | 2oj9 | A | | 3-[5-(1h-imidazol-1-yl)-7-methyl-1h-benzimidazol-2-yl]-4-[(pyridin-2-ylmethyl)amino]pyridin-2(1h)-one | Human | 1017 | |
| IGF1R | InsR | TK | 2zm3 | A | | (4z)-6-bromo-4-({[4-(pyrrolidin-1-ylmethyl)phenyl]amino}methylidene)isoquinoline-1,3(2h,4h)-dione | Human | 1004 | |
| IGF1R | InsR | TK | 2zm3 | B | | (4z)-6-bromo-4-({[4-(pyrrolidin-1-ylmethyl)phenyl]amino}methylidene)isoquinoline-1,3(2h,4h)-dione | Human | 1000 | |
| IGF1R | InsR | TK | 2zm3 | C | | (4z)-6-bromo-4-({[4-(pyrrolidin-1-ylmethyl)phenyl]amino}methylidene)isoquinoline-1,3(2h,4h)-dione | Human | 1010 | |
| IGF1R | InsR | TK | 2zm3 | D | | (4z)-6-bromo-4-({[4-(pyrrolidin-1-ylmethyl)phenyl]amino}methylidene)isoquinoline-1,3(2h,4h)-dione | Human | 1023 | |
| IGF1R | InsR | TK | 3d94 | A | A | 3-[cis-3-(4-methylpiperazin-1-yl)cyclobutyl]-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-8-amine | Human | 6759 | |
| IGF1R | InsR | TK | 3d94 | A | B | 3-[cis-3-(4-methylpiperazin-1-yl)cyclobutyl]-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-8-amine | Human | 6760 | |
| IGF1R | InsR | TK | 3f5p | A | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 995 | |
| IGF1R | InsR | TK | 3f5p | B | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1044 | |
| IGF1R | InsR | TK | 3f5p | C | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1022 | |
| IGF1R | InsR | TK | 3f5p | D | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1015 | |
| IGF1R | InsR | TK | 3f5p | E | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1042 | |
| IGF1R | InsR | TK | 3f5p | F | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1029 | |
| IGF1R | InsR | TK | 3f5p | G | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1005 | |
| IGF1R | InsR | TK | 3f5p | H | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1006 | |
| IGF1R | InsR | TK | 3f5p | I | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1016 | |
| IGF1R | InsR | TK | 3f5p | J | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1040 | |
| IGF1R | InsR | TK | 3f5p | K | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1013 | |
| IGF1R | InsR | TK | 3f5p | L | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1039 | |
| IGF1R | InsR | TK | 3f5p | M | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1001 | |
| IGF1R | InsR | TK | 3f5p | R | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1019 | |
| IGF1R | InsR | TK | 3f5p | S | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 996 | |
| IGF1R | InsR | TK | 3f5p | T | | 4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrile | Human | 1037 | |
| IGF1R | InsR | TK | 3i81 | A | | 1-{4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}-n-(6-fluoropyridin-3-yl)-2-methyl-l-prolinamide | Human | 1041 | |
| IGF1R | InsR | TK | 3lvp | A | | 3-(4-chloro-1h-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dimethoxy-1-methyl-1h-pyrrolo[3,2-b]pyridine | Human | 1032 | |
| IGF1R | InsR | TK | 3lvp | B | | 3-(4-chloro-1h-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dimethoxy-1-methyl-1h-pyrrolo[3,2-b]pyridine | Human | 1035 | |
| IGF1R | InsR | TK | 3lvp | C | | 3-(4-chloro-1h-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dimethoxy-1-methyl-1h-pyrrolo[3,2-b]pyridine | Human | 1003 | |
| IGF1R | InsR | TK | 3lvp | D | | 3-(4-chloro-1h-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dimethoxy-1-methyl-1h-pyrrolo[3,2-b]pyridine | Human | 1009 | |
| IGF1R | InsR | TK | 3lw0 | A | A | - | Human | 1021 | |
| IGF1R | InsR | TK | 3lw0 | A | B | - | Human | 1031 | |
| IGF1R | InsR | TK | 3lw0 | B | A | - | Human | 993 | |
| IGF1R | InsR | TK | 3lw0 | B | B | - | Human | 1008 | |
| IGF1R | InsR | TK | 3lw0 | C | A | - | Human | 1011 | |
| IGF1R | InsR | TK | 3lw0 | C | B | - | Human | 1025 | |
| IGF1R | InsR | TK | 3lw0 | D | A | - | Human | 1033 | |
| IGF1R | InsR | TK | 3lw0 | D | B | - | Human | 1027 | |
| IGF1R | InsR | TK | 3nw5 | A | | n-(5-cyclopropyl-1h-pyrazol-3-yl)-2-{(2r)-1-[(6-fluoropyridin-3-yl)carbonyl]pyrrolidin-2-yl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 998 | |
| IGF1R | InsR | TK | 3nw6 | A | | n-(5-cyclopropyl-1h-pyrazol-3-yl)-2-{(2s)-1-[(6-fluoropyridin-3-yl)carbonyl]pyrrolidin-2-yl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 1043 | |
| IGF1R | InsR | TK | 3nw7 | A | | n-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}methyl)-6-fluoropyridine-3-carboxamide | Human | 1030 | |
| IGF1R | InsR | TK | 3o23 | A | | (5s)-5-methyl-1-(quinolin-4-ylmethyl)-3-{4-[(trifluoromethyl)sulfonyl]phenyl}imidazolidine-2,4-dione | Human | 1036 | |
| IGF1R | InsR | TK | 3qqu | A | | n~2~-[3-methoxy-4-(morpholin-4-yl)phenyl]-n~4~-(quinolin-3-yl)pyrimidine-2,4-diamine | Human | 1024 | |
| IGF1R | InsR | TK | 3qqu | B | | n~2~-[3-methoxy-4-(morpholin-4-yl)phenyl]-n~4~-(quinolin-3-yl)pyrimidine-2,4-diamine | Human | 1020 | |
| IGF1R | InsR | TK | 3qqu | C | | n~2~-[3-methoxy-4-(morpholin-4-yl)phenyl]-n~4~-(quinolin-3-yl)pyrimidine-2,4-diamine | Human | 1014 | |
| IGF1R | InsR | TK | 3qqu | D | | n~2~-[3-methoxy-4-(morpholin-4-yl)phenyl]-n~4~-(quinolin-3-yl)pyrimidine-2,4-diamine | Human | 997 | |
| IGF1R | InsR | TK | 4d2r | A | A | n-{2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]phenyl}-4-(1h-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 1018 | |
| IGF1R | InsR | TK | 4d2r | A | B | n-{2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]phenyl}-4-(1h-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 1034 | |
| IGF1R | InsR | TK | 5fxq | A | | 5-chloranyl-4-imidazo[1,2-a]pyridin-3-yl-n-(5-methyl-1-piperidin-4-yl-pyrazol-4-yl)pyrimidin-2-amine | Human | 7093 | |
| IGF1R | InsR | TK | 5fxr | A | A | 5-chloranyl-4-imidazo[1,2-a]pyridin-3-yl-n-(3-methyl-1-piperidin-4-yl-pyrazol-4-yl)pyrimidin-2-amine | Human | 7095 | |
| IGF1R | InsR | TK | 5fxr | A | B | 5-chloranyl-4-imidazo[1,2-a]pyridin-3-yl-n-(3-methyl-1-piperidin-4-yl-pyrazol-4-yl)pyrimidin-2-amine | Human | 7094 | |
| IGF1R | InsR | TK | 5fxs | A | A | 2-[4-[4-[[(6z)-5-chloranyl-6-pyrazolo[1,5-a]pyridin-3-ylidene-1h-pyrimidin-2-yl]amino]-3,5-dimethyl-pyrazol-1-yl]piperidin-1-yl]-n,n-dimethyl-ethanamide | Human | 7096 | |
| IGF1R | InsR | TK | 5fxs | A | B | 2-[4-[4-[[(6z)-5-chloranyl-6-pyrazolo[1,5-a]pyridin-3-ylidene-1h-pyrimidin-2-yl]amino]-3,5-dimethyl-pyrazol-1-yl]piperidin-1-yl]-n,n-dimethyl-ethanamide | Human | 7097 | |
| IGF1R | InsR | TK | 5hzn | A | | 7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6493 | |
| IGF1R | InsR | TK | 5hzn | B | | 7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6495 | |
| IGF1R | InsR | TK | 5hzn | C | | 7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6498 | |
| IGF1R | InsR | TK | 5hzn | D | | 7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6496 | |
| IGF1R | InsR | TK | 5hzn | E | | 7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6494 | |
| IGF1R | InsR | TK | 5hzn | F | | 7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6497 | |
| IGF1R | InsR | TK | 5hzn | G | | 7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6499 | |
| IGF1R | InsR | TK | 5hzn | H | | 7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6492 | |
| IGF1R | InsR | TK | 6jk8 | A | A | - | Human | 12015 | |
| IGF1R | InsR | TK | 6jk8 | A | B | - | Human | 12016 | |
| IGF1R | InsR | TK | 6jk8 | B | A | - | Human | 12018 | |
| IGF1R | InsR | TK | 6jk8 | B | B | - | Human | 12017 | |
| IGF1R | InsR | TK | 8pyi | A | | 3-[8-azanyl-1-(4-ethoxy-8-fluoranyl-2-phenyl-quinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl]-1-methyl-cyclobutan-1-ol | Human | 14903 | |
| IGF1R | InsR | TK | 8pyj | A | | 5,5-dimethyl-1-(quinolin-4-ylmethyl)-3-[4-(trifluoromethylsulfonyl)phenyl]imidazolidine-2,4-dione | Human | 14905 | |
| IGF1R | InsR | TK | 8pyk | A | A | 5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-3-[4-(trifluoromethylsulfanyl)phenyl]imidazolidine-2,4-dione | Human | 14900 | |
| IGF1R | InsR | TK | 8pyk | A | B | 5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-3-[4-(trifluoromethylsulfanyl)phenyl]imidazolidine-2,4-dione | Human | 14904 | |
| IGF1R | InsR | TK | 8pyl | A | | (5s)-5-methyl-1-(1h-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfanyl)phenyl]imidazolidine-2,4-dione | Human | 14906 | |
| IGF1R | InsR | TK | 8pym | A | | 5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfanyl)phenyl]imidazolidine-2,4-dione | Human | 14901 | |
| IGF1R | InsR | TK | 8pyn | A | A | 5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfonyl)phenyl]imidazolidine-2,4-dione | Human | 14902 | |
| IGF1R | InsR | TK | 8pyn | A | B | 5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfonyl)phenyl]imidazolidine-2,4-dione | Human | 14907 | |
| IKBKB (IKKb) | IKK | Other | 4e3c | A | | - | Human | 297 | |
| IKBKB (IKKb) | IKK | Other | 4e3c | B | | - | Human | 294 | |
| IKBKB (IKKb) | IKK | Other | 4e3c | C | | - | Human | 296 | |
| IKBKB (IKKb) | IKK | Other | 4e3c | D | | - | Human | 291 | |
| IKBKB (IKKb) | IKK | Other | 4e3c | E | | - | Human | 289 | |
| IKBKB (IKKb) | IKK | Other | 4e3c | F | | - | Human | 292 | |
| IKBKB (IKKb) | IKK | Other | 4kik | A | A | k-252a | Human | 290 | |
| IKBKB (IKKb) | IKK | Other | 4kik | A | B | k-252a | Human | 288 | |
| IKBKB (IKKb) | IKK | Other | 4kik | B | A | k-252a | Human | 295 | |
| IKBKB (IKKb) | IKK | Other | 4kik | B | B | k-252a | Human | 293 | |
| IKBKB (IKKb) | IKK | Other | 8omv | A | | - | Human | 15271 | |
| ILK | MLK | TKL | 3kmu | A | | - | Human | 4606 | |
| ILK | MLK | TKL | 3kmw | A | | adenosine-5'-triphosphate | Human | 4605 | |
| ILK | MLK | TKL | 3rep | A | | adenosine-5'-triphosphate | Human | 4604 | |
| ILK | MLK | TKL | 6mib | A | | - | Human | 10687 | |
| Insr (INSR) | InsR | TK | 7sl4 | A | | - | Mouse | 14172 | |
| Insr (INSR) | InsR | TK | 7sl6 | A | | - | Mouse | 14171 | |
| Insr (INSR) | InsR | TK | 7sl7 | A | | - | Mouse | 14169 | |
| Insr (INSR) | InsR | TK | 7stj | A | | - | Mouse | 14170 | |
| Insr (INSR) | InsR | TK | 8dtl | B | | - | Mouse | 14362 | |
| Insr (INSR) | InsR | TK | 8eyx | A | | - | Mouse | 14496 | |
| Insr (INSR) | InsR | TK | 8eyy | A | | - | Mouse | 14497 | |
| INSR | InsR | TK | 1gag | A | | - | Human | 586 | |
| INSR | InsR | TK | 1i44 | A | | phosphomethylphosphonic acid adenylate ester | Human | 582 | |
| INSR | InsR | TK | 1ir3 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 602 | |
| INSR | InsR | TK | 1irk | A | A | - | Human | 596 | |
| INSR | InsR | TK | 1irk | A | B | - | Human | 603 | |
| INSR | InsR | TK | 1p14 | A | | - | Human | 593 | |
| INSR | InsR | TK | 1rqq | A | | thiophosphoric acid o-((adenosyl-phospho)phospho)-s-acetamidyl-diester | Human | 7407 | |
| INSR | InsR | TK | 1rqq | B | | thiophosphoric acid o-((adenosyl-phospho)phospho)-s-acetamidyl-diester | Human | 7406 | |
| INSR | InsR | TK | 2auh | A | | - | Human | 584 | |
| INSR | InsR | TK | 2b4s | B | | - | Human | 585 | |
| INSR | InsR | TK | 2b4s | D | | - | Human | 583 | |
| INSR | InsR | TK | 2z8c | A | | [4-({5-(aminocarbonyl)-4-[(3-methylphenyl)amino]pyrimidin-2-yl}amino)phenyl]acetic acid | Human | 587 | |
| INSR | InsR | TK | 3bu3 | A | | - | Human | 591 | |
| INSR | InsR | TK | 3bu5 | A | | adenosine-5'-triphosphate | Human | 595 | |
| INSR | InsR | TK | 3bu6 | A | | - | Human | 601 | |
| INSR | InsR | TK | 3ekk | A | A | 2-[(2-{[1-(n,n-dimethylglycyl)-5-methoxy-1h-indol-6-yl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-6-fluoro-n-methylbenzamide | Human | 578 | |
| INSR | InsR | TK | 3ekk | A | B | 2-[(2-{[1-(n,n-dimethylglycyl)-5-methoxy-1h-indol-6-yl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-6-fluoro-n-methylbenzamide | Human | 581 | |
| INSR | InsR | TK | 3ekn | A | A | 2-fluoro-6-{[2-({2-methoxy-4-[4-(1-methylethyl)piperazin-1-yl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide | Human | 597 | |
| INSR | InsR | TK | 3ekn | A | B | 2-fluoro-6-{[2-({2-methoxy-4-[4-(1-methylethyl)piperazin-1-yl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide | Human | 594 | |
| INSR | InsR | TK | 3eta | A | A | 1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea | Human | 590 | |
| INSR | InsR | TK | 3eta | A | B | 1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea | Human | 579 | |
| INSR | InsR | TK | 3eta | B | A | 1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea | Human | 588 | |
| INSR | InsR | TK | 3eta | B | B | 1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)urea | Human | 600 | |
| INSR | InsR | TK | 4ibm | A | A | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-one | Human | 589 | |
| INSR | InsR | TK | 4ibm | A | B | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-one | Human | 598 | |
| INSR | InsR | TK | 4ibm | B | A | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-one | Human | 604 | |
| INSR | InsR | TK | 4ibm | B | B | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-one | Human | 599 | |
| INSR | InsR | TK | 4xlv | A | | phosphomethylphosphonic acid adenylate ester | Human | 577 | |
| INSR | InsR | TK | 5e1s | A | A | (5r)-n-(1-{2-[4-(2-methoxyethyl)piperazin-1-yl]ethyl}-1h-pyrazol-3-yl)-5,8-dimethyl-9-phenyl-6,8-dihydro-5h-pyrazolo[3,4-h]quinazolin-2-amine | Human | 6146 | |
| INSR | InsR | TK | 5e1s | A | B | (5r)-n-(1-{2-[4-(2-methoxyethyl)piperazin-1-yl]ethyl}-1h-pyrazol-3-yl)-5,8-dimethyl-9-phenyl-6,8-dihydro-5h-pyrazolo[3,4-h]quinazolin-2-amine | Human | 6147 | |
| INSR | InsR | TK | 5hhw | A | A | 7-[3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-[[(2~{r})-oxan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6523 | |
| INSR | InsR | TK | 5hhw | A | B | 7-[3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-[[(2~{r})-oxan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6522 | |
| INSR | InsR | TK | 6pxv | A | | - | Human | 11592 | |
| INSR | InsR | TK | 6pxv | C | | - | Human | 11590 | |
| INSR | InsR | TK | 6pxw | A | | - | Human | 11593 | |
| INSR | InsR | TK | 6pxw | B | | - | Human | 11591 | |
| INSR | InsR | TK | 7bw7 | A | | - | Human | 13504 | |
| INSR | InsR | TK | 7bw7 | C | | - | Human | 13505 | |
| INSR | InsR | TK | 7bw8 | A | | - | Human | 13502 | |
| INSR | InsR | TK | 7bw8 | C | | - | Human | 13503 | |
| INSR | InsR | TK | 7pg0 | A | | - | Human | 14097 | |
| INSR | InsR | TK | 7pg2 | A | | - | Human | 14098 | |
| INSR | InsR | TK | 7pg3 | A | | - | Human | 14099 | |
| INSR | InsR | TK | 7pg4 | A | | - | Human | 14100 | |
| INSR | InsR | TK | 8dwn | A | | - | Human | 14975 | |
| INSR | InsR | TK | 8u4b | A | | - | Human | 15258 | |
| INSRR (IRR) | InsR | TK | 7tyk | A | | - | Human | 14612 | |
| INSRR (IRR) | InsR | TK | 7tym | A | | - | Human | 14611 | |
| IRAK1 | IRAK | TKL | 6bfn | A | A | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamide | Human | 8698 | |
| IRAK1 | IRAK | TKL | 6bfn | A | B | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamide | Human | 8700 | |
| IRAK1 | IRAK | TKL | 6bfn | B | A | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamide | Human | 8701 | |
| IRAK1 | IRAK | TKL | 6bfn | B | B | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamide | Human | 8699 | |
| IRAK3 | IRAK | TKL | 6ruu | A | | - | Human | 12770 | |
| IRAK3 | IRAK | TKL | 6ruu | B | | - | Human | 12769 | |
| IRAK3 | IRAK | TKL | 6ruu | C | | - | Human | 12771 | |
| IRAK3 | IRAK | TKL | 6ziw | I | | phosphothiophosphoric acid-adenylate ester | Human | 12483 | |
| IRAK4 | IRAK | TKL | 2nru | A | A | 1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalate | Human | 1748 | |
| IRAK4 | IRAK | TKL | 2nru | A | B | 1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalate | Human | 1760 | |
| IRAK4 | IRAK | TKL | 2nru | B | A | 1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalate | Human | 1773 | |
| IRAK4 | IRAK | TKL | 2nru | B | B | 1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalate | Human | 1749 | |
| IRAK4 | IRAK | TKL | 2nru | C | A | 1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalate | Human | 1776 | |
| IRAK4 | IRAK | TKL | 2nru | C | B | 1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalate | Human | 1771 | |
| IRAK4 | IRAK | TKL | 2nru | D | A | 1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalate | Human | 1762 | |
| IRAK4 | IRAK | TKL | 2nru | D | B | 1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalate | Human | 1787 | |
| IRAK4 | IRAK | TKL | 2nry | A | A | staurosporine | Human | 1753 | |
| IRAK4 | IRAK | TKL | 2nry | A | B | staurosporine | Human | 1777 | |
| IRAK4 | IRAK | TKL | 2nry | B | A | staurosporine | Human | 1758 | |
| IRAK4 | IRAK | TKL | 2nry | B | B | staurosporine | Human | 1772 | |
| IRAK4 | IRAK | TKL | 2nry | C | A | staurosporine | Human | 1779 | |
| IRAK4 | IRAK | TKL | 2nry | C | B | staurosporine | Human | 1750 | |
| IRAK4 | IRAK | TKL | 2nry | D | A | staurosporine | Human | 1789 | |
| IRAK4 | IRAK | TKL | 2nry | D | B | staurosporine | Human | 1746 | |
| IRAK4 | IRAK | TKL | 2o8y | A | | - | Human | 1744 | |
| IRAK4 | IRAK | TKL | 2o8y | B | | - | Human | 1732 | |
| IRAK4 | IRAK | TKL | 2oib | A | A | - | Human | 1756 | |
| IRAK4 | IRAK | TKL | 2oib | A | B | - | Human | 1766 | |
| IRAK4 | IRAK | TKL | 2oib | B | A | - | Human | 1785 | |
| IRAK4 | IRAK | TKL | 2oib | B | B | - | Human | 1743 | |
| IRAK4 | IRAK | TKL | 2oib | C | A | - | Human | 1781 | |
| IRAK4 | IRAK | TKL | 2oib | C | B | - | Human | 1741 | |
| IRAK4 | IRAK | TKL | 2oib | D | A | - | Human | 1736 | |
| IRAK4 | IRAK | TKL | 2oib | D | B | - | Human | 1783 | |
| IRAK4 | IRAK | TKL | 2oic | A | | staurosporine | Human | 1739 | |
| IRAK4 | IRAK | TKL | 2oic | B | | staurosporine | Human | 1752 | |
| IRAK4 | IRAK | TKL | 2oic | C | | staurosporine | Human | 1734 | |
| IRAK4 | IRAK | TKL | 2oic | D | | staurosporine | Human | 1755 | |
| IRAK4 | IRAK | TKL | 2oid | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1764 | |
| IRAK4 | IRAK | TKL | 2oid | B | | phosphoaminophosphonic acid-adenylate ester | Human | 1759 | |
| IRAK4 | IRAK | TKL | 2oid | C | | phosphoaminophosphonic acid-adenylate ester | Human | 1775 | |
| IRAK4 | IRAK | TKL | 2oid | D | | phosphoaminophosphonic acid-adenylate ester | Human | 1733 | |
| IRAK4 | IRAK | TKL | 4rmz | A | A | 3-nitro-n-[1-phenyl-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl]benzamide | Human | 6349 | |
| IRAK4 | IRAK | TKL | 4rmz | A | B | 3-nitro-n-[1-phenyl-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl]benzamide | Human | 6352 | |
| IRAK4 | IRAK | TKL | 4rmz | B | A | 3-nitro-n-[1-phenyl-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl]benzamide | Human | 6351 | |
| IRAK4 | IRAK | TKL | 4rmz | B | B | 3-nitro-n-[1-phenyl-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl]benzamide | Human | 6350 | |
| IRAK4 | IRAK | TKL | 4u97 | A | | staurosporine | Human | 1754 | |
| IRAK4 | IRAK | TKL | 4u97 | B | | staurosporine | Human | 1742 | |
| IRAK4 | IRAK | TKL | 4u9a | A | | staurosporine | Human | 1751 | |
| IRAK4 | IRAK | TKL | 4u9a | B | | staurosporine | Human | 1792 | |
| IRAK4 | IRAK | TKL | 4xs2 | A | | (1r,2s,3r,5r)-3-({5-(1,3-benzothiazol-2-yl)-6-chloro-2-[(3-methoxypropyl)amino]pyrimidin-4-yl}amino)-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 1765 | |
| IRAK4 | IRAK | TKL | 4xs2 | B | | (1r,2s,3r,5r)-3-({5-(1,3-benzothiazol-2-yl)-6-chloro-2-[(3-methoxypropyl)amino]pyrimidin-4-yl}amino)-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 1778 | |
| IRAK4 | IRAK | TKL | 4xs2 | C | | (1r,2s,3r,5r)-3-({5-(1,3-benzothiazol-2-yl)-6-chloro-2-[(3-methoxypropyl)amino]pyrimidin-4-yl}amino)-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 1791 | |
| IRAK4 | IRAK | TKL | 4xs2 | D | | (1r,2s,3r,5r)-3-({5-(1,3-benzothiazol-2-yl)-6-chloro-2-[(3-methoxypropyl)amino]pyrimidin-4-yl}amino)-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 1738 | |
| IRAK4 | IRAK | TKL | 4y73 | A | A | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 9123 | |
| IRAK4 | IRAK | TKL | 4y73 | A | B | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 9129 | |
| IRAK4 | IRAK | TKL | 4y73 | B | A | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 9128 | |
| IRAK4 | IRAK | TKL | 4y73 | B | B | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 9125 | |
| IRAK4 | IRAK | TKL | 4y73 | C | A | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 9130 | |
| IRAK4 | IRAK | TKL | 4y73 | C | B | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 9124 | |
| IRAK4 | IRAK | TKL | 4y73 | D | A | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 9127 | |
| IRAK4 | IRAK | TKL | 4y73 | D | B | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 9126 | |
| IRAK4 | IRAK | TKL | 4yo6 | A | A | n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1793 | |
| IRAK4 | IRAK | TKL | 4yo6 | A | B | n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1763 | |
| IRAK4 | IRAK | TKL | 4yo6 | B | A | n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1747 | |
| IRAK4 | IRAK | TKL | 4yo6 | B | B | n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1769 | |
| IRAK4 | IRAK | TKL | 4yo6 | C | A | n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1780 | |
| IRAK4 | IRAK | TKL | 4yo6 | C | B | n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1737 | |
| IRAK4 | IRAK | TKL | 4yo6 | D | A | n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1768 | |
| IRAK4 | IRAK | TKL | 4yo6 | D | B | n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1788 | |
| IRAK4 | IRAK | TKL | 4yp8 | A | | n-{1-(4-cyclopropyl-2-fluorophenyl)-3-[1-(propan-2-yl)piperidin-4-yl]-1h-pyrazol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1740 | |
| IRAK4 | IRAK | TKL | 4yp8 | B | | n-{1-(4-cyclopropyl-2-fluorophenyl)-3-[1-(propan-2-yl)piperidin-4-yl]-1h-pyrazol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1786 | |
| IRAK4 | IRAK | TKL | 4yp8 | C | | n-{1-(4-cyclopropyl-2-fluorophenyl)-3-[1-(propan-2-yl)piperidin-4-yl]-1h-pyrazol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1735 | |
| IRAK4 | IRAK | TKL | 4yp8 | D | | n-{1-(4-cyclopropyl-2-fluorophenyl)-3-[1-(propan-2-yl)piperidin-4-yl]-1h-pyrazol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 1745 | |
| IRAK4 | IRAK | TKL | 4ztl | A | A | (1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 6003 | |
| IRAK4 | IRAK | TKL | 4ztl | A | B | (1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 5994 | |
| IRAK4 | IRAK | TKL | 4ztl | B | A | (1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 6009 | |
| IRAK4 | IRAK | TKL | 4ztl | B | B | (1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 6004 | |
| IRAK4 | IRAK | TKL | 4ztl | C | A | (1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 5998 | |
| IRAK4 | IRAK | TKL | 4ztl | C | B | (1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 5990 | |
| IRAK4 | IRAK | TKL | 4ztl | D | A | (1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 5996 | |
| IRAK4 | IRAK | TKL | 4ztl | D | B | (1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diol | Human | 6000 | |
| IRAK4 | IRAK | TKL | 4ztm | A | | 5-(1,3-benzothiazol-2-yl)-2-(cyclopropylamino)-6-{[(1r,2s,3r,4r)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino}pyrimidin-4(3h)-one | Human | 5997 | |
| IRAK4 | IRAK | TKL | 4ztm | B | | 5-(1,3-benzothiazol-2-yl)-2-(cyclopropylamino)-6-{[(1r,2s,3r,4r)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino}pyrimidin-4(3h)-one | Human | 5992 | |
| IRAK4 | IRAK | TKL | 4ztm | C | | 5-(1,3-benzothiazol-2-yl)-2-(cyclopropylamino)-6-{[(1r,2s,3r,4r)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino}pyrimidin-4(3h)-one | Human | 6006 | |
| IRAK4 | IRAK | TKL | 4ztm | D | | 5-(1,3-benzothiazol-2-yl)-2-(cyclopropylamino)-6-{[(1r,2s,3r,4r)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino}pyrimidin-4(3h)-one | Human | 5999 | |
| IRAK4 | IRAK | TKL | 4ztn | A | A | 5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-one | Human | 5993 | |
| IRAK4 | IRAK | TKL | 4ztn | A | B | 5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-one | Human | 6007 | |
| IRAK4 | IRAK | TKL | 4ztn | B | A | 5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-one | Human | 6005 | |
| IRAK4 | IRAK | TKL | 4ztn | B | B | 5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-one | Human | 6001 | |
| IRAK4 | IRAK | TKL | 4ztn | C | A | 5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-one | Human | 6008 | |
| IRAK4 | IRAK | TKL | 4ztn | C | B | 5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-one | Human | 5991 | |
| IRAK4 | IRAK | TKL | 4ztn | D | A | 5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-one | Human | 5995 | |
| IRAK4 | IRAK | TKL | 4ztn | D | B | 5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-one | Human | 6002 | |
| IRAK4 | IRAK | TKL | 5k72 | A | | ~{n}4,~{n}4-dimethyl-~{n}1-[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]cyclohexane-1,4-diamine | Human | 8720 | |
| IRAK4 | IRAK | TKL | 5k72 | B | | ~{n}4,~{n}4-dimethyl-~{n}1-[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]cyclohexane-1,4-diamine | Human | 8711 | |
| IRAK4 | IRAK | TKL | 5k72 | C | | ~{n}4,~{n}4-dimethyl-~{n}1-[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]cyclohexane-1,4-diamine | Human | 8723 | |
| IRAK4 | IRAK | TKL | 5k72 | D | | ~{n}4,~{n}4-dimethyl-~{n}1-[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]cyclohexane-1,4-diamine | Human | 8721 | |
| IRAK4 | IRAK | TKL | 5k75 | A | A | ~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamine | Human | 8725 | |
| IRAK4 | IRAK | TKL | 5k75 | A | B | ~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamine | Human | 8727 | |
| IRAK4 | IRAK | TKL | 5k75 | B | A | ~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamine | Human | 8713 | |
| IRAK4 | IRAK | TKL | 5k75 | B | B | ~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamine | Human | 8717 | |
| IRAK4 | IRAK | TKL | 5k75 | C | A | ~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamine | Human | 8724 | |
| IRAK4 | IRAK | TKL | 5k75 | C | B | ~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamine | Human | 8710 | |
| IRAK4 | IRAK | TKL | 5k75 | D | A | ~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamine | Human | 8718 | |
| IRAK4 | IRAK | TKL | 5k75 | D | B | ~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamine | Human | 8714 | |
| IRAK4 | IRAK | TKL | 5k76 | A | A | ~{n}-(4-morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 8712 | |
| IRAK4 | IRAK | TKL | 5k76 | A | B | ~{n}-(4-morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 8715 | |
| IRAK4 | IRAK | TKL | 5k76 | B | A | ~{n}-(4-morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 8709 | |
| IRAK4 | IRAK | TKL | 5k76 | B | B | ~{n}-(4-morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 8708 | |
| IRAK4 | IRAK | TKL | 5k7g | A | | (3~{a}~{s},7~{a}~{r})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-one | Human | 8722 | |
| IRAK4 | IRAK | TKL | 5k7g | B | | (3~{a}~{s},7~{a}~{r})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-one | Human | 8706 | |
| IRAK4 | IRAK | TKL | 5k7g | C | | (3~{a}~{s},7~{a}~{r})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-one | Human | 8707 | |
| IRAK4 | IRAK | TKL | 5k7g | D | | (3~{a}~{s},7~{a}~{r})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-one | Human | 8716 | |
| IRAK4 | IRAK | TKL | 5k7i | A | | (3~{a}~{r},7~{a}~{s})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-one | Human | 9521 | |
| IRAK4 | IRAK | TKL | 5k7i | B | | (3~{a}~{r},7~{a}~{s})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-one | Human | 9520 | |
| IRAK4 | IRAK | TKL | 5kx7 | A | | - | Human | 6956 | |
| IRAK4 | IRAK | TKL | 5kx7 | B | | ~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-6-(1-methylpyrazol-4-yl)pyridine-2-carboxamide | Human | 6957 | |
| IRAK4 | IRAK | TKL | 5kx8 | A | | ~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-5-piperazin-1-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 6958 | |
| IRAK4 | IRAK | TKL | 5kx8 | B | | ~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-5-piperazin-1-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 6959 | |
| IRAK4 | IRAK | TKL | 5kx8 | C | | ~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-5-piperazin-1-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 6960 | |
| IRAK4 | IRAK | TKL | 5kx8 | D | | ~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-5-piperazin-1-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 6961 | |
| IRAK4 | IRAK | TKL | 5t1s | A | | 5-[3-(3,5-dimethylphenyl)-4-[4-(methylamino)butyl]quinolin-6-yl]pyridin-3-ol | Human | 7568 | |
| IRAK4 | IRAK | TKL | 5t1s | B | | 5-[3-(3,5-dimethylphenyl)-4-[4-(methylamino)butyl]quinolin-6-yl]pyridin-3-ol | Human | 7566 | |
| IRAK4 | IRAK | TKL | 5t1s | C | | 5-[3-(3,5-dimethylphenyl)-4-[4-(methylamino)butyl]quinolin-6-yl]pyridin-3-ol | Human | 7561 | |
| IRAK4 | IRAK | TKL | 5t1s | D | | 5-[3-(3,5-dimethylphenyl)-4-[4-(methylamino)butyl]quinolin-6-yl]pyridin-3-ol | Human | 7563 | |
| IRAK4 | IRAK | TKL | 5t1t | A | | ~{n},~{n}-dimethyl-4-(6-nitroquinazolin-4-yl)oxy-cyclohexan-1-amine | Human | 7567 | |
| IRAK4 | IRAK | TKL | 5t1t | B | | ~{n},~{n}-dimethyl-4-(6-nitroquinazolin-4-yl)oxy-cyclohexan-1-amine | Human | 7562 | |
| IRAK4 | IRAK | TKL | 5t1t | C | | ~{n},~{n}-dimethyl-4-(6-nitroquinazolin-4-yl)oxy-cyclohexan-1-amine | Human | 7564 | |
| IRAK4 | IRAK | TKL | 5t1t | D | | ~{n},~{n}-dimethyl-4-(6-nitroquinazolin-4-yl)oxy-cyclohexan-1-amine | Human | 7565 | |
| IRAK4 | IRAK | TKL | 5uiq | A | A | 2-[(propan-2-yl)oxy]benzamide | Human | 7596 | |
| IRAK4 | IRAK | TKL | 5uiq | A | B | 2-[(propan-2-yl)oxy]benzamide | Human | 7612 | |
| IRAK4 | IRAK | TKL | 5uiq | B | A | 2-[(propan-2-yl)oxy]benzamide | Human | 7617 | |
| IRAK4 | IRAK | TKL | 5uiq | B | B | 2-[(propan-2-yl)oxy]benzamide | Human | 7619 | |
| IRAK4 | IRAK | TKL | 5uiq | C | A | 2-[(propan-2-yl)oxy]benzamide | Human | 7616 | |
| IRAK4 | IRAK | TKL | 5uiq | C | B | 2-[(propan-2-yl)oxy]benzamide | Human | 7608 | |
| IRAK4 | IRAK | TKL | 5uiq | D | A | 2-[(propan-2-yl)oxy]benzamide | Human | 7620 | |
| IRAK4 | IRAK | TKL | 5uiq | D | B | 2-[(propan-2-yl)oxy]benzamide | Human | 7610 | |
| IRAK4 | IRAK | TKL | 5uir | A | A | 5-(4-cyanophenyl)-3-[(propan-2-yl)oxy]naphthalene-2-carboxamide | Human | 7599 | |
| IRAK4 | IRAK | TKL | 5uir | A | B | 5-(4-cyanophenyl)-3-[(propan-2-yl)oxy]naphthalene-2-carboxamide | Human | 7600 | |
| IRAK4 | IRAK | TKL | 5uir | B | A | 5-(4-cyanophenyl)-3-[(propan-2-yl)oxy]naphthalene-2-carboxamide | Human | 7595 | |
| IRAK4 | IRAK | TKL | 5uir | B | B | 5-(4-cyanophenyl)-3-[(propan-2-yl)oxy]naphthalene-2-carboxamide | Human | 7605 | |
| IRAK4 | IRAK | TKL | 5uis | A | A | 4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamide | Human | 7604 | |
| IRAK4 | IRAK | TKL | 5uis | A | B | 4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamide | Human | 7598 | |
| IRAK4 | IRAK | TKL | 5uis | B | A | 4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamide | Human | 7601 | |
| IRAK4 | IRAK | TKL | 5uis | B | B | 4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamide | Human | 7618 | |
| IRAK4 | IRAK | TKL | 5uis | C | A | 4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamide | Human | 7611 | |
| IRAK4 | IRAK | TKL | 5uis | C | B | 4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamide | Human | 7613 | |
| IRAK4 | IRAK | TKL | 5uis | D | A | 4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamide | Human | 7602 | |
| IRAK4 | IRAK | TKL | 5uis | D | B | 4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamide | Human | 7614 | |
| IRAK4 | IRAK | TKL | 5uit | A | | 1-{[(2s)-5-oxopyrrolidin-2-yl]methoxy}-7-[(propan-2-yl)oxy]isoquinoline-6-carboxamide | Human | 7606 | |
| IRAK4 | IRAK | TKL | 5uit | B | | 1-{[(2s)-5-oxopyrrolidin-2-yl]methoxy}-7-[(propan-2-yl)oxy]isoquinoline-6-carboxamide | Human | 7597 | |
| IRAK4 | IRAK | TKL | 5uiu | A | A | 1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide | Human | 7603 | |
| IRAK4 | IRAK | TKL | 5uiu | A | B | 1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide | Human | 7615 | |
| IRAK4 | IRAK | TKL | 5uiu | B | A | 1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide | Human | 7607 | |
| IRAK4 | IRAK | TKL | 5uiu | B | B | 1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide | Human | 7609 | |
| IRAK4 | IRAK | TKL | 5w84 | A | | 4-(benzylamino)-6-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]pyridine-3-carboxamide | Human | 8559 | |
| IRAK4 | IRAK | TKL | 5w84 | B | | 4-(benzylamino)-6-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]pyridine-3-carboxamide | Human | 8561 | |
| IRAK4 | IRAK | TKL | 5w85 | A | | 6-[(1,3-benzothiazol-6-yl)amino]-4-{[(2s)-1-hydroxy-3-phenylpropan-2-yl]amino}-n-methylpyridine-3-carboxamide | Human | 8560 | |
| IRAK4 | IRAK | TKL | 5w85 | B | | 6-[(1,3-benzothiazol-6-yl)amino]-4-{[(2s)-1-hydroxy-3-phenylpropan-2-yl]amino}-n-methylpyridine-3-carboxamide | Human | 8558 | |
| IRAK4 | IRAK | TKL | 6eg9 | A | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 10906 | |
| IRAK4 | IRAK | TKL | 6eg9 | A | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 10905 | |
| IRAK4 | IRAK | TKL | 6eg9 | B | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 10909 | |
| IRAK4 | IRAK | TKL | 6eg9 | B | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 10911 | |
| IRAK4 | IRAK | TKL | 6ega | A | A | 3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}-n-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 10908 | |
| IRAK4 | IRAK | TKL | 6ega | A | B | 3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}-n-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 10907 | |
| IRAK4 | IRAK | TKL | 6ega | B | A | 3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}-n-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 10912 | |
| IRAK4 | IRAK | TKL | 6ega | B | B | 3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}-n-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 10910 | |
| IRAK4 | IRAK | TKL | 6egd | A | A | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-2-(pyridin-3-yl)-1,3-thiazole-5-carboxamide | Human | 10895 | |
| IRAK4 | IRAK | TKL | 6egd | A | B | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-2-(pyridin-3-yl)-1,3-thiazole-5-carboxamide | Human | 10892 | |
| IRAK4 | IRAK | TKL | 6egd | D | A | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-2-(pyridin-3-yl)-1,3-thiazole-5-carboxamide | Human | 10894 | |
| IRAK4 | IRAK | TKL | 6egd | D | B | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-2-(pyridin-3-yl)-1,3-thiazole-5-carboxamide | Human | 10890 | |
| IRAK4 | IRAK | TKL | 6ege | A | A | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamide | Human | 10897 | |
| IRAK4 | IRAK | TKL | 6ege | A | B | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamide | Human | 10891 | |
| IRAK4 | IRAK | TKL | 6ege | D | A | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamide | Human | 10896 | |
| IRAK4 | IRAK | TKL | 6ege | D | B | n-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamide | Human | 10889 | |
| IRAK4 | IRAK | TKL | 6egf | B | | phosphoaminophosphonic acid-adenylate ester | Human | 10893 | |
| IRAK4 | IRAK | TKL | 6f3d | A | | 4-[4-[[4-(dimethylamino)cyclohexyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]cyclohexane-1-carboxamide | Human | 9925 | |
| IRAK4 | IRAK | TKL | 6f3d | B | | 4-[4-[[4-(dimethylamino)cyclohexyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]cyclohexane-1-carboxamide | Human | 9924 | |
| IRAK4 | IRAK | TKL | 6f3e | A | | 2-[(3~{r})-12-(4-morpholin-4-ylcyclohexyl)oxy-7-thia-9,11-diazatricyclo[6.4.0.0^{2,6}]dodeca-1(8),2(6),9,11-tetraen-3-yl]ethanamide | Human | 9923 | |
| IRAK4 | IRAK | TKL | 6f3e | B | | 2-[(3~{r})-12-(4-morpholin-4-ylcyclohexyl)oxy-7-thia-9,11-diazatricyclo[6.4.0.0^{2,6}]dodeca-1(8),2(6),9,11-tetraen-3-yl]ethanamide | Human | 9926 | |
| IRAK4 | IRAK | TKL | 6f3g | A | | ~{n}4,~{n}4-dimethyl-~{n}1-(5-propan-2-ylpyrrolo[3,2-d]pyrimidin-4-yl)cyclohexane-1,4-diamine | Human | 9921 | |
| IRAK4 | IRAK | TKL | 6f3g | B | | ~{n}4,~{n}4-dimethyl-~{n}1-(5-propan-2-ylpyrrolo[3,2-d]pyrimidin-4-yl)cyclohexane-1,4-diamine | Human | 9927 | |
| IRAK4 | IRAK | TKL | 6f3i | A | | (3~{r})-3-[4-[[4-(4-ethanoylpiperazin-1-yl)cyclohexyl]amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]butanamide | Human | 9928 | |
| IRAK4 | IRAK | TKL | 6f3i | B | | (3~{r})-3-[4-[[4-(4-ethanoylpiperazin-1-yl)cyclohexyl]amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]butanamide | Human | 9922 | |
| IRAK4 | IRAK | TKL | 6lxy | B | | n-[(2r)-2-fluoranyl-3-methyl-3-oxidanyl-butyl]-6-[(6-fluoranylpyrazolo[1,5-a]pyrimidin-5-yl)amino]-4-(propan-2-ylamino)pyridine-3-carboxamide | Human | 13163 | |
| IRAK4 | IRAK | TKL | 6lxy | D | | n-[(2r)-2-fluoranyl-3-methyl-3-oxidanyl-butyl]-6-[(6-fluoranylpyrazolo[1,5-a]pyrimidin-5-yl)amino]-4-(propan-2-ylamino)pyridine-3-carboxamide | Human | 13161 | |
| IRAK4 | IRAK | TKL | 6lxy | E | | n-[(2r)-2-fluoranyl-3-methyl-3-oxidanyl-butyl]-6-[(6-fluoranylpyrazolo[1,5-a]pyrimidin-5-yl)amino]-4-(propan-2-ylamino)pyridine-3-carboxamide | Human | 13162 | |
| IRAK4 | IRAK | TKL | 6mom | A | A | 6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amine | Human | 11742 | |
| IRAK4 | IRAK | TKL | 6mom | A | B | 6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amine | Human | 11740 | |
| IRAK4 | IRAK | TKL | 6mom | B | A | 6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amine | Human | 11743 | |
| IRAK4 | IRAK | TKL | 6mom | B | B | 6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amine | Human | 11745 | |
| IRAK4 | IRAK | TKL | 6mom | C | A | 6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amine | Human | 11738 | |
| IRAK4 | IRAK | TKL | 6mom | C | B | 6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amine | Human | 11739 | |
| IRAK4 | IRAK | TKL | 6mom | D | A | 6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amine | Human | 11744 | |
| IRAK4 | IRAK | TKL | 6mom | D | B | 6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amine | Human | 11741 | |
| IRAK4 | IRAK | TKL | 6n8g | A | A | n-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide | Human | 10796 | |
| IRAK4 | IRAK | TKL | 6n8g | A | B | n-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide | Human | 10795 | |
| IRAK4 | IRAK | TKL | 6n8g | B | A | n-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide | Human | 10791 | |
| IRAK4 | IRAK | TKL | 6n8g | B | B | n-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide | Human | 10790 | |
| IRAK4 | IRAK | TKL | 6n8g | C | A | n-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide | Human | 10794 | |
| IRAK4 | IRAK | TKL | 6n8g | C | B | n-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide | Human | 10793 | |
| IRAK4 | IRAK | TKL | 6n8g | D | A | n-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide | Human | 10792 | |
| IRAK4 | IRAK | TKL | 6n8g | D | B | n-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamide | Human | 10789 | |
| IRAK4 | IRAK | TKL | 6o8u | A | A | n-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11113 | |
| IRAK4 | IRAK | TKL | 6o8u | A | B | n-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11121 | |
| IRAK4 | IRAK | TKL | 6o8u | B | A | n-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11120 | |
| IRAK4 | IRAK | TKL | 6o8u | B | B | n-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11096 | |
| IRAK4 | IRAK | TKL | 6o8u | C | A | n-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11116 | |
| IRAK4 | IRAK | TKL | 6o8u | C | B | n-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11093 | |
| IRAK4 | IRAK | TKL | 6o8u | D | A | n-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11119 | |
| IRAK4 | IRAK | TKL | 6o8u | D | B | n-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11103 | |
| IRAK4 | IRAK | TKL | 6o94 | A | A | n-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11092 | |
| IRAK4 | IRAK | TKL | 6o94 | A | B | n-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11091 | |
| IRAK4 | IRAK | TKL | 6o94 | B | A | n-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11098 | |
| IRAK4 | IRAK | TKL | 6o94 | B | B | n-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11117 | |
| IRAK4 | IRAK | TKL | 6o94 | C | A | n-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11118 | |
| IRAK4 | IRAK | TKL | 6o94 | C | B | n-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11095 | |
| IRAK4 | IRAK | TKL | 6o94 | D | A | n-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11111 | |
| IRAK4 | IRAK | TKL | 6o94 | D | B | n-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11108 | |
| IRAK4 | IRAK | TKL | 6o95 | A | A | n-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11104 | |
| IRAK4 | IRAK | TKL | 6o95 | A | B | n-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11102 | |
| IRAK4 | IRAK | TKL | 6o95 | B | A | n-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11090 | |
| IRAK4 | IRAK | TKL | 6o95 | B | B | n-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11106 | |
| IRAK4 | IRAK | TKL | 6o95 | C | A | n-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11110 | |
| IRAK4 | IRAK | TKL | 6o95 | C | B | n-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11097 | |
| IRAK4 | IRAK | TKL | 6o95 | D | A | n-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11105 | |
| IRAK4 | IRAK | TKL | 6o95 | D | B | n-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11101 | |
| IRAK4 | IRAK | TKL | 6o9d | A | A | n-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11099 | |
| IRAK4 | IRAK | TKL | 6o9d | A | B | n-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11109 | |
| IRAK4 | IRAK | TKL | 6o9d | B | A | n-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11107 | |
| IRAK4 | IRAK | TKL | 6o9d | B | B | n-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11094 | |
| IRAK4 | IRAK | TKL | 6o9d | C | A | n-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11115 | |
| IRAK4 | IRAK | TKL | 6o9d | C | B | n-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11112 | |
| IRAK4 | IRAK | TKL | 6o9d | D | A | n-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11100 | |
| IRAK4 | IRAK | TKL | 6o9d | D | B | n-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11114 | |
| IRAK4 | IRAK | TKL | 6rfi | A | A | methyl 4-[4-[(6-cyanoquinazolin-4-yl)amino]cyclohexyl]piperazine-1-carboxylate | Human | 11788 | |
| IRAK4 | IRAK | TKL | 6rfi | A | B | methyl 4-[4-[(6-cyanoquinazolin-4-yl)amino]cyclohexyl]piperazine-1-carboxylate | Human | 11787 | |
| IRAK4 | IRAK | TKL | 6rfi | B | A | methyl 4-[4-[(6-cyanoquinazolin-4-yl)amino]cyclohexyl]piperazine-1-carboxylate | Human | 11790 | |
| IRAK4 | IRAK | TKL | 6rfi | B | B | methyl 4-[4-[(6-cyanoquinazolin-4-yl)amino]cyclohexyl]piperazine-1-carboxylate | Human | 11791 | |
| IRAK4 | IRAK | TKL | 6rfj | A | | methyl 4-[4-[[6-(cyanomethyl)-2-[(1-methylpyrazol-4-yl)amino]pyrido[3,2-d]pyrimidin-4-yl]amino]cyclohexyl]piperazine-1-carboxylate | Human | 11786 | |
| IRAK4 | IRAK | TKL | 6rfj | B | | methyl 4-[4-[[6-(cyanomethyl)-2-[(1-methylpyrazol-4-yl)amino]pyrido[3,2-d]pyrimidin-4-yl]amino]cyclohexyl]piperazine-1-carboxylate | Human | 11789 | |
| IRAK4 | IRAK | TKL | 6thw | A | | 7-fluoranyl-4-(1-methylcyclopropyl)oxy-~{n}-[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]-6-(2-methylpyrimidin-5-yl)pyrido[3,2-d]pyrimidin-2-amine | Human | 12950 | |
| IRAK4 | IRAK | TKL | 6thw | B | | 7-fluoranyl-4-(1-methylcyclopropyl)oxy-~{n}-[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]-6-(2-methylpyrimidin-5-yl)pyrido[3,2-d]pyrimidin-2-amine | Human | 12956 | |
| IRAK4 | IRAK | TKL | 6thx | A | | 2-[4-[(1-methylcyclopropyl)amino]-2-[(1-methylpyrazol-4-yl)amino]pyrido[3,2-d]pyrimidin-6-yl]ethanenitrile | Human | 12944 | |
| IRAK4 | IRAK | TKL | 6thx | B | | 2-[4-[(1-methylcyclopropyl)amino]-2-[(1-methylpyrazol-4-yl)amino]pyrido[3,2-d]pyrimidin-6-yl]ethanenitrile | Human | 12953 | |
| IRAK4 | IRAK | TKL | 6thz | A | | 7-fluoranyl-~{n}-[1-(2-methyl-2-azaspiro[3.3]heptan-6-yl)pyrazol-4-yl]-4-(1-methylcyclopropyl)oxy-6-(2-methylpyrimidin-5-yl)pyrido[3,2-d]pyrimidin-2-amine | Human | 12948 | |
| IRAK4 | IRAK | TKL | 6thz | B | | 7-fluoranyl-~{n}-[1-(2-methyl-2-azaspiro[3.3]heptan-6-yl)pyrazol-4-yl]-4-(1-methylcyclopropyl)oxy-6-(2-methylpyrimidin-5-yl)pyrido[3,2-d]pyrimidin-2-amine | Human | 12951 | |
| IRAK4 | IRAK | TKL | 6ti8 | A | A | ~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamide | Human | 12947 | |
| IRAK4 | IRAK | TKL | 6ti8 | A | B | ~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamide | Human | 12954 | |
| IRAK4 | IRAK | TKL | 6ti8 | B | A | ~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamide | Human | 12949 | |
| IRAK4 | IRAK | TKL | 6ti8 | B | B | ~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamide | Human | 12952 | |
| IRAK4 | IRAK | TKL | 6ti8 | C | A | ~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamide | Human | 12945 | |
| IRAK4 | IRAK | TKL | 6ti8 | C | B | ~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamide | Human | 12946 | |
| IRAK4 | IRAK | TKL | 6ti8 | D | A | ~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamide | Human | 12957 | |
| IRAK4 | IRAK | TKL | 6ti8 | D | B | ~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamide | Human | 12942 | |
| IRAK4 | IRAK | TKL | 6tia | A | | 4-(1-methylcyclopropyl)oxy-~{n}-[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]-6-(1-methylpyrazol-4-yl)pyrido[3,2-d]pyrimidin-2-amine | Human | 12955 | |
| IRAK4 | IRAK | TKL | 6tia | B | | 4-(1-methylcyclopropyl)oxy-~{n}-[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]-6-(1-methylpyrazol-4-yl)pyrido[3,2-d]pyrimidin-2-amine | Human | 12943 | |
| IRAK4 | IRAK | TKL | 6uya | A | A | n-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11810 | |
| IRAK4 | IRAK | TKL | 6uya | A | B | n-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11811 | |
| IRAK4 | IRAK | TKL | 6uya | B | A | n-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11807 | |
| IRAK4 | IRAK | TKL | 6uya | B | B | n-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11812 | |
| IRAK4 | IRAK | TKL | 6uya | C | A | n-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11814 | |
| IRAK4 | IRAK | TKL | 6uya | C | B | n-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11808 | |
| IRAK4 | IRAK | TKL | 6uya | D | A | n-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11813 | |
| IRAK4 | IRAK | TKL | 6uya | D | B | n-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11809 | |
| IRAK4 | IRAK | TKL | 6vql | A | | 6-[(1,3-benzothiazol-6-yl)amino]-4-(cyclopropylamino)-n-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide | Human | 12395 | |
| IRAK4 | IRAK | TKL | 6vql | B | | 6-[(1,3-benzothiazol-6-yl)amino]-4-(cyclopropylamino)-n-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide | Human | 12394 | |
| IRAK4 | IRAK | TKL | 6vql | C | | 6-[(1,3-benzothiazol-6-yl)amino]-4-(cyclopropylamino)-n-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide | Human | 12393 | |
| IRAK4 | IRAK | TKL | 6vql | D | | 6-[(1,3-benzothiazol-6-yl)amino]-4-(cyclopropylamino)-n-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamide | Human | 12392 | |
| IRAK4 | IRAK | TKL | 7c2v | A | A | 2-(2-methylpyridin-4-yl)-n-[2-morpholin-4-yl-5-[(3r)-3-oxidanylpyrrolidin-1-yl]-[1,3]oxazolo[4,5-b]pyridin-6-yl]-1,3-oxazole-4-carboxamide | Human | 12997 | |
| IRAK4 | IRAK | TKL | 7c2v | A | B | 2-(2-methylpyridin-4-yl)-n-[2-morpholin-4-yl-5-[(3r)-3-oxidanylpyrrolidin-1-yl]-[1,3]oxazolo[4,5-b]pyridin-6-yl]-1,3-oxazole-4-carboxamide | Human | 13001 | |
| IRAK4 | IRAK | TKL | 7c2v | C | A | 2-(2-methylpyridin-4-yl)-n-[2-morpholin-4-yl-5-[(3r)-3-oxidanylpyrrolidin-1-yl]-[1,3]oxazolo[4,5-b]pyridin-6-yl]-1,3-oxazole-4-carboxamide | Human | 12999 | |
| IRAK4 | IRAK | TKL | 7c2v | C | B | 2-(2-methylpyridin-4-yl)-n-[2-morpholin-4-yl-5-[(3r)-3-oxidanylpyrrolidin-1-yl]-[1,3]oxazolo[4,5-b]pyridin-6-yl]-1,3-oxazole-4-carboxamide | Human | 13003 | |
| IRAK4 | IRAK | TKL | 7c2w | A | A | - | Human | 12996 | |
| IRAK4 | IRAK | TKL | 7c2w | B | A | - | Human | 12998 | |
| IRAK4 | IRAK | TKL | 7c2w | C | A | - | Human | 13002 | |
| IRAK4 | IRAK | TKL | 7c2w | D | A | - | Human | 13000 | |
| IRAK4 | IRAK | TKL | 7qg1 | A | | methyl 4-[4-[[6-(cyanomethyl)-2-[(1-methylpyrazol-4-yl)amino]-5-oxidanylidene-pyrido[4,3-d]pyrimidin-4-yl]amino]cyclohexyl]piperazine-1-carboxylate | Human | 14212 | |
| IRAK4 | IRAK | TKL | 7qg2 | A | A | 6-methyl-4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[4,3-d]pyrimidin-5-one | Human | 14210 | |
| IRAK4 | IRAK | TKL | 7qg2 | A | B | 6-methyl-4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[4,3-d]pyrimidin-5-one | Human | 14215 | |
| IRAK4 | IRAK | TKL | 7qg3 | A | | 6-[(2~{s})-2-fluoranylpropyl]-4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[4,3-d]pyrimidin-5-one | Human | 14213 | |
| IRAK4 | IRAK | TKL | 7qg5 | A | A | 4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-6-pyrimidin-5-yl-pyrido[4,3-d]pyrimidin-5-one | Human | 14211 | |
| IRAK4 | IRAK | TKL | 7qg5 | A | B | 4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-6-pyrimidin-5-yl-pyrido[4,3-d]pyrimidin-5-one | Human | 14214 | |
| IRAK4 | IRAK | TKL | 8atb | A | A | ~{n}-[6-ethoxy-2-[2-(4-methylpiperazin-1-yl)-2-oxidanylidene-ethyl]indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 15080 | |
| IRAK4 | IRAK | TKL | 8atb | A | B | ~{n}-[6-ethoxy-2-[2-(4-methylpiperazin-1-yl)-2-oxidanylidene-ethyl]indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 15079 | |
| IRAK4 | IRAK | TKL | 8atl | A | A | ~{n}-[6-methoxy-2-(2-morpholin-4-yl-2-oxidanylidene-ethyl)indazol-5-yl]-6-[(1~{r})-2,2,2-tris(fluoranyl)-1-oxidanyl-ethyl]pyridine-2-carboxamide | Human | 14964 | |
| IRAK4 | IRAK | TKL | 8atl | A | B | ~{n}-[6-methoxy-2-(2-morpholin-4-yl-2-oxidanylidene-ethyl)indazol-5-yl]-6-[(1~{r})-2,2,2-tris(fluoranyl)-1-oxidanyl-ethyl]pyridine-2-carboxamide | Human | 14959 | |
| IRAK4 | IRAK | TKL | 8atl | B | A | ~{n}-[6-methoxy-2-(2-morpholin-4-yl-2-oxidanylidene-ethyl)indazol-5-yl]-6-[(1~{r})-2,2,2-tris(fluoranyl)-1-oxidanyl-ethyl]pyridine-2-carboxamide | Human | 14961 | |
| IRAK4 | IRAK | TKL | 8atl | B | B | ~{n}-[6-methoxy-2-(2-morpholin-4-yl-2-oxidanylidene-ethyl)indazol-5-yl]-6-[(1~{r})-2,2,2-tris(fluoranyl)-1-oxidanyl-ethyl]pyridine-2-carboxamide | Human | 14966 | |
| IRAK4 | IRAK | TKL | 8atn | A | A | ~{n}-[3-methyl-2-(3-methyl-3-oxidanyl-butyl)-6-(2-oxidanylpropan-2-yl)benzimidazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 14965 | |
| IRAK4 | IRAK | TKL | 8atn | A | B | ~{n}-[3-methyl-2-(3-methyl-3-oxidanyl-butyl)-6-(2-oxidanylpropan-2-yl)benzimidazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 14962 | |
| IRAK4 | IRAK | TKL | 8br5 | A | A | ~{n}-[2,3-dimethyl-6-(1~{h}-pyrazol-5-yl)benzimidazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 15187 | |
| IRAK4 | IRAK | TKL | 8br5 | A | B | ~{n}-[2,3-dimethyl-6-(1~{h}-pyrazol-5-yl)benzimidazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 15189 | |
| IRAK4 | IRAK | TKL | 8br6 | A | A | ~{n}-[6-methoxy-2-(2-methylsulfonylethyl)-1,3-dihydroindazol-5-yl]-6-(2-oxidanylpropan-2-yl)pyridine-2-carboxamide | Human | 15191 | |
| IRAK4 | IRAK | TKL | 8br6 | A | B | ~{n}-[6-methoxy-2-(2-methylsulfonylethyl)-1,3-dihydroindazol-5-yl]-6-(2-oxidanylpropan-2-yl)pyridine-2-carboxamide | Human | 15190 | |
| IRAK4 | IRAK | TKL | 8br7 | A | | 3-nitro-~{n}-[2-[2-oxidanylidene-2-[4-(phenylcarbonyl)piperazin-1-yl]ethyl]indazol-5-yl]benzamide | Human | 15188 | |
| IRAK4 | IRAK | TKL | 8dks | A | A | (1s,2s,3r,4r)-3-({2-[3-(pyrrolidine-1-carbonyl)anilino]thieno[3,2-d]pyrimidin-4-yl}amino)bicyclo[2.2.1]hept-5-ene-2-carboxamide | Human | 14316 | |
| IRAK4 | IRAK | TKL | 8dks | A | B | (1s,2s,3r,4r)-3-({2-[3-(pyrrolidine-1-carbonyl)anilino]thieno[3,2-d]pyrimidin-4-yl}amino)bicyclo[2.2.1]hept-5-ene-2-carboxamide | Human | 14315 | |
| IRAK4 | IRAK | TKL | 8tvm | A | A | n-{1-[(1r,2r)-2-fluorocyclopropyl]-2-oxo-1,2-dihydropyridin-3-yl}-2-[(1r,4r)-1-methyl-2-oxabicyclo[2.1.1]hexan-4-yl]-6-[(propan-2-yl)oxy]-2h-pyrazolo[3,4-b]pyridine-5-carboxamide | Human | 15337 | |
| IRAK4 | IRAK | TKL | 8tvm | A | B | n-{1-[(1r,2r)-2-fluorocyclopropyl]-2-oxo-1,2-dihydropyridin-3-yl}-2-[(1r,4r)-1-methyl-2-oxabicyclo[2.1.1]hexan-4-yl]-6-[(propan-2-yl)oxy]-2h-pyrazolo[3,4-b]pyridine-5-carboxamide | Human | 15336 | |
| IRAK4 | IRAK | TKL | 8tvn | A | A | n-{1-[(1r,2s)-2-fluorocyclopropyl]-2-oxo-1,2-dihydropyridin-3-yl}-2-[(1r,4r)-1-methyl-2-oxabicyclo[2.1.1]hexan-4-yl]-6-[(propan-2-yl)oxy]-2h-pyrazolo[3,4-b]pyridine-5-carboxamide | Human | 15339 | |
| IRAK4 | IRAK | TKL | 8tvn | A | B | n-{1-[(1r,2s)-2-fluorocyclopropyl]-2-oxo-1,2-dihydropyridin-3-yl}-2-[(1r,4r)-1-methyl-2-oxabicyclo[2.1.1]hexan-4-yl]-6-[(propan-2-yl)oxy]-2h-pyrazolo[3,4-b]pyridine-5-carboxamide | Human | 15341 | |
| IRAK4 | IRAK | TKL | 8tx0 | A | | ~{n}-(1-cyclopropyl-2-oxidanylidene-pyridin-3-yl)-2-(1-methyl-2-oxabicyclo[2.1.1]hexan-4-yl)-7-propan-2-yloxy-imidazo[1,2-a]pyrimidine-6-carboxamide | Human | 15340 | |
| IRAK4 | IRAK | TKL | 8ucb | A | | 6-(difluoromethyl)-n-[(4r)-7-ethoxy-2-{[(3r)-oxolan-3-yl]methyl}imidazo[1,2-a]pyridin-6-yl]pyridine-2-carboxamide | Human | 15338 | |
| IRAK4 | IRAK | TKL | 8ucc | A | | (4s)-2-[(1r,4s)-1-methyl-2-oxabicyclo[2.1.1]hexan-4-yl]-n-[(8s)-6-methylpyrazolo[1,5-a]pyrimidin-3-yl]-7-[(propan-2-yl)oxy]imidazo[1,2-a]pyrimidine-6-carboxamide | Human | 15332 | |
| IRAK4 | IRAK | TKL | 8ucc | B | | (4s)-2-[(1r,4s)-1-methyl-2-oxabicyclo[2.1.1]hexan-4-yl]-n-[(8s)-6-methylpyrazolo[1,5-a]pyrimidin-3-yl]-7-[(propan-2-yl)oxy]imidazo[1,2-a]pyrimidine-6-carboxamide | Human | 15342 | |
| IRAK4 | IRAK | TKL | 8v1o | A | | n-[2-(3-hydroxy-3-methylbutyl)-6-(2-hydroxypropan-2-yl)-2h-indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 15334 | |
| IRAK4 | IRAK | TKL | 8v2f | A | A | n-{2-[(1r,4r)-4-(hydroxymethyl)cyclohexyl]-6-(2-hydroxypropan-2-yl)-2h-indazol-5-yl}-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 15333 | |
| IRAK4 | IRAK | TKL | 8v2f | A | B | n-{2-[(1r,4r)-4-(hydroxymethyl)cyclohexyl]-6-(2-hydroxypropan-2-yl)-2h-indazol-5-yl}-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 15330 | |
| IRAK4 | IRAK | TKL | 8v2l | A | A | n-{2-[4-(hydroxymethyl)phenyl]-6-(2-hydroxypropan-2-yl)-2h-indazol-5-yl}-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 15331 | |
| IRAK4 | IRAK | TKL | 8v2l | A | B | n-{2-[4-(hydroxymethyl)phenyl]-6-(2-hydroxypropan-2-yl)-2h-indazol-5-yl}-6-(trifluoromethyl)pyridine-2-carboxamide | Human | 15335 | |
| IRAK4 | IRAK | TKL | 8wtf | A | A | 1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide | Human | 14960 | |
| IRAK4 | IRAK | TKL | 8wtf | A | B | 1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide | Human | 14963 | |
| ITK | Tec | TK | 1sm2 | A | | staurosporine | Human | 74 | |
| ITK | Tec | TK | 1sm2 | B | | staurosporine | Human | 73 | |
| ITK | Tec | TK | 1snu | A | | staurosporine | Human | 82 | |
| ITK | Tec | TK | 1snu | B | | staurosporine | Human | 33 | |
| ITK | Tec | TK | 1snx | A | | - | Human | 61 | |
| ITK | Tec | TK | 1snx | B | | - | Human | 62 | |
| ITK | Tec | TK | 3miy | A | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 46 | |
| ITK | Tec | TK | 3miy | B | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 8 | |
| ITK | Tec | TK | 3mj1 | A | | 7-[(4-methylpiperazin-1-yl)methyl]-4-[(3-methyl-1h-pyrazol-5-yl)amino]-2-(tetrahydro-2h-pyran-4-yl)phthalazin-1(2h)-one | Human | 27 | |
| ITK | Tec | TK | 3mj2 | A | | n-[5-({5-[(4-acetylpiperazin-1-yl)carbonyl]-4-methoxy-2-methylphenyl}sulfanyl)-1,3-thiazol-2-yl]-4-({[(1s)-1,2,2-trimethylpropyl]amino}methyl)benzamide | Human | 67 | |
| ITK | Tec | TK | 3qgw | A | A | 3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamide | Human | 11 | |
| ITK | Tec | TK | 3qgw | A | B | 3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamide | Human | 57 | |
| ITK | Tec | TK | 3qgw | B | A | n-(6-oxo-1,6-dihydro-3,4'-bipyridin-5-yl)benzamide | Human | 65 | |
| ITK | Tec | TK | 3qgw | B | B | n-(6-oxo-1,6-dihydro-3,4'-bipyridin-5-yl)benzamide | Human | 14 | |
| ITK | Tec | TK | 3qgy | A | A | 3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamide | Human | 35 | |
| ITK | Tec | TK | 3qgy | A | B | 3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamide | Human | 72 | |
| ITK | Tec | TK | 3qgy | B | A | n-{5-[2-(methylamino)pyrimidin-4-yl]-2-oxo-1,2-dihydropyridin-3-yl}-4-(piperidin-1-yl)benzamide | Human | 52 | |
| ITK | Tec | TK | 3qgy | B | B | n-{5-[2-(methylamino)pyrimidin-4-yl]-2-oxo-1,2-dihydropyridin-3-yl}-4-(piperidin-1-yl)benzamide | Human | 66 | |
| ITK | Tec | TK | 3t9t | A | A | (2z)-4-(dimethylamino)-n-{7-fluoro-4-[(2-methylphenyl)amino]imidazo[1,5-a]quinoxalin-8-yl}-n-methylbut-2-enamide | Human | 16 | |
| ITK | Tec | TK | 3t9t | A | B | (2z)-4-(dimethylamino)-n-{7-fluoro-4-[(2-methylphenyl)amino]imidazo[1,5-a]quinoxalin-8-yl}-n-methylbut-2-enamide | Human | 83 | |
| ITK | Tec | TK | 3v5j | A | | 3-{4-[2-(morpholin-4-yl)ethoxy]-2-(4lambda~4~-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl}pentan-3-ol | Human | 80 | |
| ITK | Tec | TK | 3v5j | B | | 3-{4-[2-(morpholin-4-yl)ethoxy]-2-(4lambda~4~-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl}pentan-3-ol | Human | 60 | |
| ITK | Tec | TK | 3v5l | A | | 3-[3-(4-methoxyphenyl)-2-(1h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-ol | Human | 30 | |
| ITK | Tec | TK | 3v5l | B | | 3-[3-(4-methoxyphenyl)-2-(1h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-ol | Human | 54 | |
| ITK | Tec | TK | 3v5l | C | | 3-[3-(4-methoxyphenyl)-2-(1h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-ol | Human | 26 | |
| ITK | Tec | TK | 3v5l | D | | 3-[3-(4-methoxyphenyl)-2-(1h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-ol | Human | 56 | |
| ITK | Tec | TK | 3v8t | A | A | 3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-ol | Human | 55 | |
| ITK | Tec | TK | 3v8t | A | B | 3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-ol | Human | 5 | |
| ITK | Tec | TK | 3v8t | B | A | 3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-ol | Human | 39 | |
| ITK | Tec | TK | 3v8t | B | B | 3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-ol | Human | 49 | |
| ITK | Tec | TK | 3v8w | A | | 3-[2-(5-phenyl-2h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-ol | Human | 43 | |
| ITK | Tec | TK | 3v8w | B | | 3-[2-(5-phenyl-2h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-ol | Human | 10 | |
| ITK | Tec | TK | 4hct | A | | 3-{1-[(3r)-1-acryloylpiperidin-3-yl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-n-(3-tert-butylphenyl)benzamide | Human | 44 | |
| ITK | Tec | TK | 4hcu | A | | 3-{4-amino-1-[(3r)-1-propanoylpiperidin-3-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-n-[4-(propan-2-yl)phenyl]benzamide | Human | 81 | |
| ITK | Tec | TK | 4hcv | A | | 3-{4-amino-1-[(3s)-1-propanoylpiperidin-3-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-n-[4-(propan-2-yl)phenyl]benzamide | Human | 32 | |
| ITK | Tec | TK | 4kio | A | A | 1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-one | Human | 76 | |
| ITK | Tec | TK | 4kio | A | B | 1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-one | Human | 79 | |
| ITK | Tec | TK | 4kio | B | A | 1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-one | Human | 36 | |
| ITK | Tec | TK | 4kio | B | B | 1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-one | Human | 48 | |
| ITK | Tec | TK | 4kio | C | A | 1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]propan-1-one | Human | 75 | |
| ITK | Tec | TK | 4kio | C | B | 1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-one | Human | 7 | |
| ITK | Tec | TK | 4kio | D | A | 1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]propan-1-one | Human | 6 | |
| ITK | Tec | TK | 4kio | D | B | 1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]propan-1-one | Human | 85 | |
| ITK | Tec | TK | 4l7s | A | A | trans-4-({4-[difluoro(4-fluorophenyl)methyl]-6-[(5-methoxy[1,3]thiazolo[5,4-b]pyridin-2-yl)amino]pyrimidin-2-yl}amino)cyclohexanol | Human | 50 | |
| ITK | Tec | TK | 4l7s | A | B | trans-4-({4-[difluoro(4-fluorophenyl)methyl]-6-[(5-methoxy[1,3]thiazolo[5,4-b]pyridin-2-yl)amino]pyrimidin-2-yl}amino)cyclohexanol | Human | 64 | |
| ITK | Tec | TK | 4l7s | B | A | trans-4-({4-[difluoro(4-fluorophenyl)methyl]-6-[(5-methoxy[1,3]thiazolo[5,4-b]pyridin-2-yl)amino]pyrimidin-2-yl}amino)cyclohexanol | Human | 37 | |
| ITK | Tec | TK | 4l7s | B | B | trans-4-({4-[difluoro(4-fluorophenyl)methyl]-6-[(5-methoxy[1,3]thiazolo[5,4-b]pyridin-2-yl)amino]pyrimidin-2-yl}amino)cyclohexanol | Human | 25 | |
| ITK | Tec | TK | 4m0y | A | A | 4-(carbamoylamino)-1-(naphthalen-1-yl)-1h-pyrazole-3-carboxamide | Human | 9 | |
| ITK | Tec | TK | 4m0y | A | B | 4-(carbamoylamino)-1-(naphthalen-1-yl)-1h-pyrazole-3-carboxamide | Human | 70 | |
| ITK | Tec | TK | 4m0z | A | A | 4-(carbamoylamino)-1-(7-methoxynaphthalen-1-yl)-1h-pyrazole-3-carboxamide | Human | 45 | |
| ITK | Tec | TK | 4m0z | A | B | 4-(carbamoylamino)-1-(7-methoxynaphthalen-1-yl)-1h-pyrazole-3-carboxamide | Human | 47 | |
| ITK | Tec | TK | 4m12 | A | A | - | Human | 22 | |
| ITK | Tec | TK | 4m12 | A | B | - | Human | 51 | |
| ITK | Tec | TK | 4m13 | A | A | - | Human | 17 | |
| ITK | Tec | TK | 4m13 | A | B | - | Human | 15 | |
| ITK | Tec | TK | 4m14 | A | | 4-(carbamoylamino)-1-[7-(propan-2-yloxy)naphthalen-1-yl]-1h-pyrazole-3-carboxamide | Human | 58 | |
| ITK | Tec | TK | 4m15 | A | | adenosine-5'-diphosphate | Human | 31 | |
| ITK | Tec | TK | 4mf0 | A | | (1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(pyridin-3-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamide | Human | 77 | |
| ITK | Tec | TK | 4mf0 | B | | (1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(pyridin-3-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamide | Human | 28 | |
| ITK | Tec | TK | 4mf1 | A | A | (1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(1h-pyrazol-4-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamide | Human | 41 | |
| ITK | Tec | TK | 4mf1 | A | B | (1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(1h-pyrazol-4-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamide | Human | 34 | |
| ITK | Tec | TK | 4mf1 | B | A | (1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(1h-pyrazol-4-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamide | Human | 12 | |
| ITK | Tec | TK | 4mf1 | B | B | (1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(1h-pyrazol-4-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamide | Human | 18 | |
| ITK | Tec | TK | 4pp9 | A | | n-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-2h-indazole-3-carboxamide | Human | 20 | |
| ITK | Tec | TK | 4pp9 | B | | n-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-2h-indazole-3-carboxamide | Human | 40 | |
| ITK | Tec | TK | 4ppa | A | | n-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamide | Human | 38 | |
| ITK | Tec | TK | 4ppa | B | | n-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamide | Human | 21 | |
| ITK | Tec | TK | 4ppb | A | | n-{1-[(1s)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamide | Human | 29 | |
| ITK | Tec | TK | 4ppb | B | | n-{1-[(1s)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamide | Human | 84 | |
| ITK | Tec | TK | 4ppc | A | A | n-{1-[(1r)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamide | Human | 53 | |
| ITK | Tec | TK | 4ppc | A | B | n-{1-[(1r)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamide | Human | 13 | |
| ITK | Tec | TK | 4ppc | B | A | n-{1-[(1r)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamide | Human | 78 | |
| ITK | Tec | TK | 4ppc | B | B | n-{1-[(1r)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamide | Human | 63 | |
| ITK | Tec | TK | 4pqn | A | A | n-{1-[(1s)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6,6-dimethyl-4,5,6,7-tetrahydro-1h-indazole-3-carboxamide | Human | 42 | |
| ITK | Tec | TK | 4pqn | A | B | n-{1-[(1s)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6,6-dimethyl-4,5,6,7-tetrahydro-1h-indazole-3-carboxamide | Human | 19 | |
| ITK | Tec | TK | 4qd6 | A | A | trans-4-({6-[(5-phenyl-1h-pyrazol-3-yl)amino]-4-(phenylsulfonyl)pyridin-2-yl}amino)cyclohexanol | Human | 23 | |
| ITK | Tec | TK | 4qd6 | A | B | trans-4-({6-[(5-phenyl-1h-pyrazol-3-yl)amino]-4-(phenylsulfonyl)pyridin-2-yl}amino)cyclohexanol | Human | 59 | |
| ITK | Tec | TK | 4qd6 | B | A | trans-4-({6-[(5-phenyl-1h-pyrazol-3-yl)amino]-4-(phenylsulfonyl)pyridin-2-yl}amino)cyclohexanol | Human | 24 | |
| ITK | Tec | TK | 4qd6 | B | B | trans-4-({6-[(5-phenyl-1h-pyrazol-3-yl)amino]-4-(phenylsulfonyl)pyridin-2-yl}amino)cyclohexanol | Human | 71 | |
| ITK | Tec | TK | 4rfm | A | A | (4as,5ar)-n-{1-[(r)-[(2r)-1,1-dioxidotetrahydro-2h-thiopyran-2-yl](phenyl)methyl]-1h-pyrazol-4-yl}-5,5-difluoro-5a-methyl-1,4,4a,5,5a,6-hexahydrocyclopropa[f]indazole-3-carboxamide | Human | 68 | |
| ITK | Tec | TK | 4rfm | A | B | (4as,5ar)-n-{1-[(r)-[(2r)-1,1-dioxidotetrahydro-2h-thiopyran-2-yl](phenyl)methyl]-1h-pyrazol-4-yl}-5,5-difluoro-5a-methyl-1,4,4a,5,5a,6-hexahydrocyclopropa[f]indazole-3-carboxamide | Human | 69 | |
| Jak1 (JAK1) | JakA | TK | 8ewy | A | | - | Mouse | 14664 | |
| JAK1 | JakA | TK | 3eyg | A | A | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 1445 | |
| JAK1 | JakA | TK | 3eyg | A | B | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 1453 | |
| JAK1 | JakA | TK | 3eyh | A | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 1462 | |
| JAK1 | JakA | TK | 4e4l | A | A | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1450 | |
| JAK1 | JakA | TK | 4e4l | A | B | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1488 | |
| JAK1 | JakA | TK | 4e4l | B | A | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1464 | |
| JAK1 | JakA | TK | 4e4l | B | B | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1466 | |
| JAK1 | JakA | TK | 4e4l | D | A | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1455 | |
| JAK1 | JakA | TK | 4e4l | D | B | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1468 | |
| JAK1 | JakA | TK | 4e4l | E | A | - | Human | 1469 | |
| JAK1 | JakA | TK | 4e4l | E | B | - | Human | 1484 | |
| JAK1 | JakA | TK | 4e4n | A | | tert-butyl [(1r,3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)cyclopentyl]carbamate | Human | 1443 | |
| JAK1 | JakA | TK | 4e4n | B | | tert-butyl [(1r,3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)cyclopentyl]carbamate | Human | 1454 | |
| JAK1 | JakA | TK | 4e5w | A | A | [4-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl][(2s)-1-(propan-2-yl)pyrrolidin-2-yl]methanone | Human | 1452 | |
| JAK1 | JakA | TK | 4e5w | A | B | [4-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl][(2s)-1-(propan-2-yl)pyrrolidin-2-yl]methanone | Human | 1473 | |
| JAK1 | JakA | TK | 4e5w | B | A | [4-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl][(2s)-1-(propan-2-yl)pyrrolidin-2-yl]methanone | Human | 1447 | |
| JAK1 | JakA | TK | 4e5w | B | B | [4-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl][(2s)-1-(propan-2-yl)pyrrolidin-2-yl]methanone | Human | 1477 | |
| JAK1 | JakA | TK | 4ehz | A | A | 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1482 | |
| JAK1 | JakA | TK | 4ehz | A | B | 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1463 | |
| JAK1 | JakA | TK | 4ehz | B | A | 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1448 | |
| JAK1 | JakA | TK | 4ehz | B | B | 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1481 | |
| JAK1 | JakA | TK | 4ehz | C | A | 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1470 | |
| JAK1 | JakA | TK | 4ehz | C | B | 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1476 | |
| JAK1 | JakA | TK | 4ehz | D | A | 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1485 | |
| JAK1 | JakA | TK | 4ehz | D | B | 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 1451 | |
| JAK1 | JakA | TK | 4ei4 | A | | (1r,3r)-3-(2-methylimidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(8h)-yl)cyclohexanol | Human | 1480 | |
| JAK1 | JakA | TK | 4ei4 | B | | (1r,3r)-3-(2-methylimidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(8h)-yl)cyclohexanol | Human | 1483 | |
| JAK1 | JakA | TK | 4fk6 | A | A | n-({1-[(1r,2r,4s)-bicyclo[2.2.1]hept-2-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2-yl}methyl)methanesulfonamide | Human | 1465 | |
| JAK1 | JakA | TK | 4fk6 | A | B | n-({1-[(1r,2r,4s)-bicyclo[2.2.1]hept-2-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2-yl}methyl)methanesulfonamide | Human | 1460 | |
| JAK1 | JakA | TK | 4fk6 | B | A | n-({1-[(1r,2r,4s)-bicyclo[2.2.1]hept-2-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2-yl}methyl)methanesulfonamide | Human | 1487 | |
| JAK1 | JakA | TK | 4fk6 | B | B | n-({1-[(1r,2r,4s)-bicyclo[2.2.1]hept-2-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2-yl}methyl)methanesulfonamide | Human | 1459 | |
| JAK1 | JakA | TK | 4i5c | A | A | 3-oxo-3-[(3r)-3-(pyrrolo[2,3-b][1,2,3]triazolo[4,5-d]pyridin-1(6h)-yl)piperidin-1-yl]propanenitrile | Human | 1446 | |
| JAK1 | JakA | TK | 4i5c | A | B | 3-oxo-3-[(3r)-3-(pyrrolo[2,3-b][1,2,3]triazolo[4,5-d]pyridin-1(6h)-yl)piperidin-1-yl]propanenitrile | Human | 1471 | |
| JAK1 | JakA | TK | 4i5c | B | A | 3-oxo-3-[(3r)-3-(pyrrolo[2,3-b][1,2,3]triazolo[4,5-d]pyridin-1(6h)-yl)piperidin-1-yl]propanenitrile | Human | 1467 | |
| JAK1 | JakA | TK | 4i5c | B | B | 3-oxo-3-[(3r)-3-(pyrrolo[2,3-b][1,2,3]triazolo[4,5-d]pyridin-1(6h)-yl)piperidin-1-yl]propanenitrile | Human | 1458 | |
| JAK1 | JakA | TK | 4ivb | A | A | trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrile | Human | 1486 | |
| JAK1 | JakA | TK | 4ivb | A | B | trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrile | Human | 1479 | |
| JAK1 | JakA | TK | 4ivb | B | A | trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrile | Human | 1472 | |
| JAK1 | JakA | TK | 4ivb | B | B | trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrile | Human | 1444 | |
| JAK1 | JakA | TK | 4ivc | A | | (trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)acetonitrile | Human | 1461 | |
| JAK1 | JakA | TK | 4ivc | B | | (trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)acetonitrile | Human | 1456 | |
| JAK1 | JakA | TK | 4ivd | A | A | 3-(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)propanenitrile | Human | 1489 | |
| JAK1 | JakA | TK | 4ivd | A | B | 3-(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)propanenitrile | Human | 1474 | |
| JAK1 | JakA | TK | 4ivd | B | A | 3-(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)propanenitrile | Human | 1490 | |
| JAK1 | JakA | TK | 4ivd | B | B | 3-(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)propanenitrile | Human | 1457 | |
| JAK1 | JakA | TK | 4k6z | A | | (1r,2s)-2-{[8-oxo-2-(1h-pyrazol-4-yl)-5,8-dihydropyrido[3,4-d]pyrimidin-4-yl]amino}cyclopentanecarbonitrile | Human | 1478 | |
| JAK1 | JakA | TK | 4k77 | A | | 4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-8(7h)-one | Human | 1449 | |
| JAK1 | JakA | TK | 4k77 | B | | 4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-8(7h)-one | Human | 1475 | |
| JAK1 | JakA | TK | 5e1e | A | A | 6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amine | Human | 6250 | |
| JAK1 | JakA | TK | 5e1e | A | B | 6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amine | Human | 6248 | |
| JAK1 | JakA | TK | 5e1e | B | A | 6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amine | Human | 6249 | |
| JAK1 | JakA | TK | 5e1e | B | B | 6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amine | Human | 6251 | |
| JAK1 | JakA | TK | 5hx8 | A | A | 4-[(4-aminocyclohexyl)amino]-3-(1h-benzimidazol-2-yl)-1h-pyridin-2-one | Human | 6441 | |
| JAK1 | JakA | TK | 5hx8 | A | B | 4-[(4-aminocyclohexyl)amino]-3-(1h-benzimidazol-2-yl)-1h-pyridin-2-one | Human | 6438 | |
| JAK1 | JakA | TK | 5hx8 | B | A | 4-[(4-aminocyclohexyl)amino]-3-(1h-benzimidazol-2-yl)-1h-pyridin-2-one | Human | 6440 | |
| JAK1 | JakA | TK | 5hx8 | B | B | 4-[(4-aminocyclohexyl)amino]-3-(1h-benzimidazol-2-yl)-1h-pyridin-2-one | Human | 6439 | |
| JAK1 | JakA | TK | 5khw | A | | adenosine-5'-diphosphate | Human | 7164 | |
| JAK1 | JakA | TK | 5khw | B | | adenosine-5'-diphosphate | Human | 7165 | |
| JAK1 | JakA | TK | 5khx | A | A | ~{n}-[3-[methyl(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl]methanesulfonamide | Human | 7167 | |
| JAK1 | JakA | TK | 5khx | A | B | ~{n}-[3-[methyl(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl]methanesulfonamide | Human | 7166 | |
| JAK1 | JakA | TK | 5wo4 | A | A | 3-[(4-chloro-3-methoxyphenyl)amino]-1-[(3r,4s)-4-cyanooxan-3-yl]-1h-pyrazole-4-carboxamide | Human | 8702 | |
| JAK1 | JakA | TK | 5wo4 | A | B | 3-[(4-chloro-3-methoxyphenyl)amino]-1-[(3r,4s)-4-cyanooxan-3-yl]-1h-pyrazole-4-carboxamide | Human | 8705 | |
| JAK1 | JakA | TK | 5wo4 | B | A | 3-[(4-chloro-3-methoxyphenyl)amino]-1-[(3r,4s)-4-cyanooxan-3-yl]-1h-pyrazole-4-carboxamide | Human | 8704 | |
| JAK1 | JakA | TK | 5wo4 | B | B | 3-[(4-chloro-3-methoxyphenyl)amino]-1-[(3r,4s)-4-cyanooxan-3-yl]-1h-pyrazole-4-carboxamide | Human | 8703 | |
| JAK1 | JakA | TK | 6aah | A | A | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10392 | |
| JAK1 | JakA | TK | 6aah | A | B | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10396 | |
| JAK1 | JakA | TK | 6aah | B | A | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10394 | |
| JAK1 | JakA | TK | 6aah | B | B | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10395 | |
| JAK1 | JakA | TK | 6bbu | A | A | n-{cis-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide | Human | 9497 | |
| JAK1 | JakA | TK | 6bbu | A | B | n-{cis-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide | Human | 9496 | |
| JAK1 | JakA | TK | 6c7y | A | A | adenosine-5'-diphosphate | Human | 9866 | |
| JAK1 | JakA | TK | 6c7y | A | B | adenosine-5'-diphosphate | Human | 9867 | |
| JAK1 | JakA | TK | 6dbn | A | A | [(1s)-2,2-difluorocyclopropyl][(1r,5s)-3-{2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octan-8-yl]methanone | Human | 10393 | |
| JAK1 | JakA | TK | 6dbn | A | B | [(1s)-2,2-difluorocyclopropyl][(1r,5s)-3-{2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octan-8-yl]methanone | Human | 10391 | |
| JAK1 | JakA | TK | 6elr | A | A | [3-[[5-methyl-2-[[3-(4-methylpiperazin-1-yl)-5-methylsulfonyl-phenyl]amino]pyrimidin-4-yl]amino]phenyl]methanol | Human | 10618 | |
| JAK1 | JakA | TK | 6elr | A | B | [3-[[5-methyl-2-[[3-(4-methylpiperazin-1-yl)-5-methylsulfonyl-phenyl]amino]pyrimidin-4-yl]amino]phenyl]methanol | Human | 10616 | |
| JAK1 | JakA | TK | 6elr | B | A | [3-[[5-methyl-2-[[3-(4-methylpiperazin-1-yl)-5-methylsulfonyl-phenyl]amino]pyrimidin-4-yl]amino]phenyl]methanol | Human | 10619 | |
| JAK1 | JakA | TK | 6elr | B | B | [3-[[5-methyl-2-[[3-(4-methylpiperazin-1-yl)-5-methylsulfonyl-phenyl]amino]pyrimidin-4-yl]amino]phenyl]methanol | Human | 10617 | |
| JAK1 | JakA | TK | 6ggh | A | A | ~{n}-[5-methyl-4-[7-[[(2~{r})-2-(4-methylpiperazin-1-yl)propanoyl]amino]-1~{h}-indol-3-yl]pyrimidin-2-yl]cyclopropanecarboxamide | Human | 11087 | |
| JAK1 | JakA | TK | 6ggh | A | B | ~{n}-[5-methyl-4-[7-[[(2~{r})-2-(4-methylpiperazin-1-yl)propanoyl]amino]-1~{h}-indol-3-yl]pyrimidin-2-yl]cyclopropanecarboxamide | Human | 11088 | |
| JAK1 | JakA | TK | 6ggh | B | A | ~{n}-[5-methyl-4-[7-[[(2~{r})-2-(4-methylpiperazin-1-yl)propanoyl]amino]-1~{h}-indol-3-yl]pyrimidin-2-yl]cyclopropanecarboxamide | Human | 11089 | |
| JAK1 | JakA | TK | 6ggh | B | B | ~{n}-[5-methyl-4-[7-[[(2~{r})-2-(4-methylpiperazin-1-yl)propanoyl]amino]-1~{h}-indol-3-yl]pyrimidin-2-yl]cyclopropanecarboxamide | Human | 11086 | |
| JAK1 | JakA | TK | 6hzu | A | A | 2-[4-[8-oxidanylidene-2-[(~{e})-(2-oxidanylidenepyridin-3-ylidene)amino]-7~{h}-purin-9-yl]cyclohexyl]ethanenitrile | Human | 11764 | |
| JAK1 | JakA | TK | 6hzu | A | B | 2-[4-[8-oxidanylidene-2-[(~{e})-(2-oxidanylidenepyridin-3-ylidene)amino]-7~{h}-purin-9-yl]cyclohexyl]ethanenitrile | Human | 11762 | |
| JAK1 | JakA | TK | 6hzu | B | A | 2-[4-[8-oxidanylidene-2-[(~{e})-(2-oxidanylidenepyridin-3-ylidene)amino]-7~{h}-purin-9-yl]cyclohexyl]ethanenitrile | Human | 11765 | |
| JAK1 | JakA | TK | 6hzu | B | B | 2-[4-[8-oxidanylidene-2-[(~{e})-(2-oxidanylidenepyridin-3-ylidene)amino]-7~{h}-purin-9-yl]cyclohexyl]ethanenitrile | Human | 11763 | |
| JAK1 | JakA | TK | 6n77 | A | A | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11024 | |
| JAK1 | JakA | TK | 6n77 | A | B | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11021 | |
| JAK1 | JakA | TK | 6n77 | A | C | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11029 | |
| JAK1 | JakA | TK | 6n77 | B | A | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11030 | |
| JAK1 | JakA | TK | 6n77 | B | B | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11018 | |
| JAK1 | JakA | TK | 6n77 | B | C | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11034 | |
| JAK1 | JakA | TK | 6n78 | A | A | n-{3-[5-chloro-2-(difluoromethoxy)phenyl]-1-methyl-1h-pyrazol-4-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11019 | |
| JAK1 | JakA | TK | 6n78 | A | B | n-{3-[5-chloro-2-(difluoromethoxy)phenyl]-1-methyl-1h-pyrazol-4-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11022 | |
| JAK1 | JakA | TK | 6n79 | A | | n-{5-[5-chloro-2-(difluoromethoxy)phenyl]-1h-pyrazol-4-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11031 | |
| JAK1 | JakA | TK | 6n7a | A | A | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-2-methyl-2h-pyrazolo[4,3-c]pyridine-7-carboxamide | Human | 11017 | |
| JAK1 | JakA | TK | 6n7a | A | B | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-2-methyl-2h-pyrazolo[4,3-c]pyridine-7-carboxamide | Human | 11028 | |
| JAK1 | JakA | TK | 6n7a | B | A | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-2-methyl-2h-pyrazolo[4,3-c]pyridine-7-carboxamide | Human | 11015 | |
| JAK1 | JakA | TK | 6n7a | B | B | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-2-methyl-2h-pyrazolo[4,3-c]pyridine-7-carboxamide | Human | 11026 | |
| JAK1 | JakA | TK | 6n7b | A | | n-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-1h-pyrazolo[4,3-c]pyridine-7-carboxamide | Human | 11020 | |
| JAK1 | JakA | TK | 6n7c | A | A | n-[5-(3-methoxynaphthalen-2-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11016 | |
| JAK1 | JakA | TK | 6n7c | A | B | n-[5-(3-methoxynaphthalen-2-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11027 | |
| JAK1 | JakA | TK | 6n7c | B | A | n-[5-(3-methoxynaphthalen-2-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11033 | |
| JAK1 | JakA | TK | 6n7c | B | B | n-[5-(3-methoxynaphthalen-2-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11023 | |
| JAK1 | JakA | TK | 6n7d | A | A | n-[5-(6-methoxy-1h-indazol-5-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11032 | |
| JAK1 | JakA | TK | 6n7d | A | B | n-[5-(6-methoxy-1h-indazol-5-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 11025 | |
| JAK1 | JakA | TK | 6rsb | A | | 1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[[4-(cyclohexen-1-yl)phenyl]methyl]-3-fluoranyl-piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12482 | |
| JAK1 | JakA | TK | 6rsb | B | | 1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[[4-(cyclohexen-1-yl)phenyl]methyl]-3-fluoranyl-piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12479 | |
| JAK1 | JakA | TK | 6rsc | A | A | 1-[4-(cyanomethyl)-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12477 | |
| JAK1 | JakA | TK | 6rsc | A | B | 1-[4-(cyanomethyl)-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12468 | |
| JAK1 | JakA | TK | 6rsc | B | A | 1-[4-(cyanomethyl)-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12474 | |
| JAK1 | JakA | TK | 6rsc | B | B | 1-[4-(cyanomethyl)-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12469 | |
| JAK1 | JakA | TK | 6rsd | A | A | 1-[4-(cyanomethyl)-1-[(3-oxidanyl-4-phenyl-phenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12472 | |
| JAK1 | JakA | TK | 6rsd | A | B | 1-[4-(cyanomethyl)-1-[(3-oxidanyl-4-phenyl-phenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12478 | |
| JAK1 | JakA | TK | 6rsd | B | A | 1-[4-(cyanomethyl)-1-[(3-oxidanyl-4-phenyl-phenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12466 | |
| JAK1 | JakA | TK | 6rsd | B | B | 1-[4-(cyanomethyl)-1-[(3-oxidanyl-4-phenyl-phenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12475 | |
| JAK1 | JakA | TK | 6rse | A | A | methyl ~{n}-[4-aminocarbonyl-1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[(4-ethenyl-2-fluoranyl-5-oxidanyl-phenyl)methyl]-3-fluoranyl-piperidin-4-yl]pyrazol-3-yl]carbamate | Human | 12481 | |
| JAK1 | JakA | TK | 6rse | A | B | methyl ~{n}-[4-aminocarbonyl-1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[(4-ethenyl-2-fluoranyl-5-oxidanyl-phenyl)methyl]-3-fluoranyl-piperidin-4-yl]pyrazol-3-yl]carbamate | Human | 12476 | |
| JAK1 | JakA | TK | 6rse | B | A | methyl ~{n}-[4-aminocarbonyl-1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[(4-ethenyl-2-fluoranyl-5-oxidanyl-phenyl)methyl]-3-fluoranyl-piperidin-4-yl]pyrazol-3-yl]carbamate | Human | 12465 | |
| JAK1 | JakA | TK | 6rse | B | B | methyl ~{n}-[4-aminocarbonyl-1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[(4-ethenyl-2-fluoranyl-5-oxidanyl-phenyl)methyl]-3-fluoranyl-piperidin-4-yl]pyrazol-3-yl]carbamate | Human | 12471 | |
| JAK1 | JakA | TK | 6rsh | A | A | 1-[(3~{r},4~{r})-4-(cyanomethyl)-3-fluoranyl-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12470 | |
| JAK1 | JakA | TK | 6rsh | A | B | 1-[(3~{r},4~{r})-4-(cyanomethyl)-3-fluoranyl-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12473 | |
| JAK1 | JakA | TK | 6rsh | B | A | 1-[(3~{r},4~{r})-4-(cyanomethyl)-3-fluoranyl-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12467 | |
| JAK1 | JakA | TK | 6rsh | B | B | 1-[(3~{r},4~{r})-4-(cyanomethyl)-3-fluoranyl-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamide | Human | 12480 | |
| JAK1 | JakA | TK | 6sm8 | A | A | 2-chloranyl-6-[(3~{s})-3-[(1~{s})-2-cyano-1-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethyl]pyrrolidin-1-yl]benzenecarbonitrile | Human | 12248 | |
| JAK1 | JakA | TK | 6sm8 | A | B | 2-chloranyl-6-[(3~{s})-3-[(1~{s})-2-cyano-1-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethyl]pyrrolidin-1-yl]benzenecarbonitrile | Human | 12250 | |
| JAK1 | JakA | TK | 6sm8 | B | A | 2-chloranyl-6-[(3~{s})-3-[(1~{s})-2-cyano-1-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethyl]pyrrolidin-1-yl]benzenecarbonitrile | Human | 12245 | |
| JAK1 | JakA | TK | 6sm8 | B | B | 2-chloranyl-6-[(3~{s})-3-[(1~{s})-2-cyano-1-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethyl]pyrrolidin-1-yl]benzenecarbonitrile | Human | 12249 | |
| JAK1 | JakA | TK | 6smb | A | A | ~{n}-[3-[2-[(3-methoxy-1-methyl-pyrazol-4-yl)amino]-5-methyl-pyrimidin-4-yl]-1~{h}-indol-7-yl]-2-methyl-pyridine-3-carboxamide | Human | 12246 | |
| JAK1 | JakA | TK | 6smb | A | B | ~{n}-[3-[2-[(3-methoxy-1-methyl-pyrazol-4-yl)amino]-5-methyl-pyrimidin-4-yl]-1~{h}-indol-7-yl]-2-methyl-pyridine-3-carboxamide | Human | 12247 | |
| JAK1 | JakA | TK | 6smb | B | A | ~{n}-[3-[2-[(3-methoxy-1-methyl-pyrazol-4-yl)amino]-5-methyl-pyrimidin-4-yl]-1~{h}-indol-7-yl]-2-methyl-pyridine-3-carboxamide | Human | 12244 | |
| JAK1 | JakA | TK | 6smb | B | B | ~{n}-[3-[2-[(3-methoxy-1-methyl-pyrazol-4-yl)amino]-5-methyl-pyrimidin-4-yl]-1~{h}-indol-7-yl]-2-methyl-pyridine-3-carboxamide | Human | 12243 | |
| JAK1 | JakA | TK | 6tpe | A | | 2-[4-(3-methyl-6-oxidanylidene-1,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]ethanenitrile | Human | 12364 | |
| JAK1 | JakA | TK | 6tpe | B | | 2-[4-(3-methyl-6-oxidanylidene-1,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]ethanenitrile | Human | 12368 | |
| JAK1 | JakA | TK | 6tpf | A | A | (1~{s})-2,2-bis(fluoranyl)-~{n}-[4-(3-methyl-6-oxidanylidene-2,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]cyclopropane-1-carboxamide | Human | 12366 | |
| JAK1 | JakA | TK | 6tpf | A | B | (1~{s})-2,2-bis(fluoranyl)-~{n}-[4-(3-methyl-6-oxidanylidene-2,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]cyclopropane-1-carboxamide | Human | 12365 | |
| JAK1 | JakA | TK | 6tpf | B | A | (1~{s})-2,2-bis(fluoranyl)-~{n}-[4-(3-methyl-6-oxidanylidene-2,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]cyclopropane-1-carboxamide | Human | 12363 | |
| JAK1 | JakA | TK | 6tpf | B | B | (1~{s})-2,2-bis(fluoranyl)-~{n}-[4-(3-methyl-6-oxidanylidene-2,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]cyclopropane-1-carboxamide | Human | 12367 | |
| JAK1 | JakA | TK | 6w8l | A | | n-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropanecarboxamide | Human | 12133 | |
| JAK1-b | JakB | TK | 4l00 | A | A | - | Human | 1421 | |
| JAK1-b | JakB | TK | 4l00 | A | B | - | Human | 1420 | |
| JAK1-b | JakB | TK | 4l00 | B | A | - | Human | 1422 | |
| JAK1-b | JakB | TK | 4l00 | B | B | - | Human | 1423 | |
| JAK1-b | JakB | TK | 4l01 | A | A | - | Human | 1424 | |
| JAK1-b | JakB | TK | 4l01 | A | B | - | Human | 1418 | |
| JAK1-b | JakB | TK | 4l01 | B | A | - | Human | 1417 | |
| JAK1-b | JakB | TK | 4l01 | B | B | - | Human | 1419 | |
| Jak2 (JAK2) | JakA | TK | 4gl9 | A | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6933 | |
| Jak2 (JAK2) | JakA | TK | 4gl9 | B | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6936 | |
| Jak2 (JAK2) | JakA | TK | 4gl9 | C | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6934 | |
| Jak2 (JAK2) | JakA | TK | 4gl9 | D | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6935 | |
| JAK2 | JakA | TK | 2b7a | A | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 3708 | |
| JAK2 | JakA | TK | 2b7a | B | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 3728 | |
| JAK2 | JakA | TK | 2w1i | A | | 4-[(2-{4-[(cyclopropylcarbamoyl)amino]-1h-pyrazol-3-yl}-1h-benzimidazol-6-yl)methyl]morpholin-4-ium | Human | 3652 | |
| JAK2 | JakA | TK | 2w1i | B | | - | Human | 3648 | |
| JAK2 | JakA | TK | 2xa4 | A | A | 5-chloro-n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(5-methyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine | Human | 3664 | |
| JAK2 | JakA | TK | 2xa4 | A | B | 5-chloro-n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(5-methyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine | Human | 3623 | |
| JAK2 | JakA | TK | 2xa4 | B | A | 5-chloro-n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(5-methyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine | Human | 3628 | |
| JAK2 | JakA | TK | 2xa4 | B | B | 5-chloro-n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(5-methyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine | Human | 3707 | |
| JAK2 | JakA | TK | 3e62 | A | A | 5-bromo-1h-indazol-3-amine | Human | 3665 | |
| JAK2 | JakA | TK | 3e62 | A | B | 5-bromo-1h-indazol-3-amine | Human | 3630 | |
| JAK2 | JakA | TK | 3e63 | A | A | 5-phenyl-1h-indazol-3-amine | Human | 3675 | |
| JAK2 | JakA | TK | 3e63 | A | B | 5-phenyl-1h-indazol-3-amine | Human | 3711 | |
| JAK2 | JakA | TK | 3e64 | A | A | 4-(3-amino-1h-indazol-5-yl)-n-tert-butylbenzenesulfonamide | Human | 3646 | |
| JAK2 | JakA | TK | 3e64 | A | B | 4-(3-amino-1h-indazol-5-yl)-n-tert-butylbenzenesulfonamide | Human | 3653 | |
| JAK2 | JakA | TK | 3fup | A | | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 3721 | |
| JAK2 | JakA | TK | 3fup | B | | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 3654 | |
| JAK2 | JakA | TK | 3io7 | A | | (3s)-1-[6-(2-aminopyrazolo[1,5-a]pyrimidin-3-yl)pyrimidin-4-yl]-n,n-diethylpiperidine-3-carboxamide | Human | 3636 | |
| JAK2 | JakA | TK | 3iok | A | A | 3-(6-{[(1s)-1-(4-fluorophenyl)ethyl]amino}pyrimidin-4-yl)pyrazolo[1,5-a]pyrimidin-2-amine | Human | 3694 | |
| JAK2 | JakA | TK | 3iok | A | B | 3-(6-{[(1s)-1-(4-fluorophenyl)ethyl]amino}pyrimidin-4-yl)pyrazolo[1,5-a]pyrimidin-2-amine | Human | 3718 | |
| JAK2 | JakA | TK | 3jy9 | A | A | (3s)-3-(4-hydroxyphenyl)-1,5-dihydro-1,5,12-triazabenzo[4,5]cycloocta[1,2,3-cd]inden-4(3h)-one | Human | 3668 | |
| JAK2 | JakA | TK | 3jy9 | A | B | (3s)-3-(4-hydroxyphenyl)-1,5-dihydro-1,5,12-triazabenzo[4,5]cycloocta[1,2,3-cd]inden-4(3h)-one | Human | 3716 | |
| JAK2 | JakA | TK | 3kck | A | A | 3-chloro-4-(4h-3,4,7-triazadibenzo[cd,f]azulen-6-yl)phenol | Human | 3683 | |
| JAK2 | JakA | TK | 3kck | A | B | 3-chloro-4-(4h-3,4,7-triazadibenzo[cd,f]azulen-6-yl)phenol | Human | 3722 | |
| JAK2 | JakA | TK | 3krr | A | A | 8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-(1-piperidin-4-yl-1h-pyrazol-4-yl)quinoxaline | Human | 3643 | |
| JAK2 | JakA | TK | 3krr | A | B | 8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-(1-piperidin-4-yl-1h-pyrazol-4-yl)quinoxaline | Human | 3695 | |
| JAK2 | JakA | TK | 3lpb | A | A | n-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]benzenesulfonamide | Human | 3672 | |
| JAK2 | JakA | TK | 3lpb | A | B | n-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]benzenesulfonamide | Human | 3698 | |
| JAK2 | JakA | TK | 3lpb | B | A | n-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]benzenesulfonamide | Human | 3635 | |
| JAK2 | JakA | TK | 3lpb | B | B | n-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]benzenesulfonamide | Human | 3681 | |
| JAK2 | JakA | TK | 3q32 | A | | 2-(2,6-difluoro-4-methoxyphenyl)-1-(4-{4-[(3-methyl-1h-pyrazol-5-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}piperazin-1-yl)ethanone | Human | 3700 | |
| JAK2 | JakA | TK | 3q32 | B | | 2-(2,6-difluoro-4-methoxyphenyl)-1-(4-{4-[(3-methyl-1h-pyrazol-5-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}piperazin-1-yl)ethanone | Human | 3639 | |
| JAK2 | JakA | TK | 3rvg | A | | 1-(cyclohexylamino)-7-(1-methyl-1h-pyrazol-4-yl)-5h-pyrido[4,3-b]indole-4-carboxamide | Human | 3638 | |
| JAK2 | JakA | TK | 3tjc | A | | 4-amino-n-methyl-2-[4-(morpholin-4-yl)phenyl]thieno[3,2-c]pyridine-7-carboxamide | Human | 3685 | |
| JAK2 | JakA | TK | 3tjc | B | | 4-amino-n-methyl-2-[4-(morpholin-4-yl)phenyl]thieno[3,2-c]pyridine-7-carboxamide | Human | 3688 | |
| JAK2 | JakA | TK | 3tjd | A | | 4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-n-methylthieno[3,2-c]pyridine-7-carboxamide | Human | 3677 | |
| JAK2 | JakA | TK | 3tjd | B | | 4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-n-methylthieno[3,2-c]pyridine-7-carboxamide | Human | 3626 | |
| JAK2 | JakA | TK | 3ugc | A | A | 5-{[6-(acetylamino)pyrimidin-4-yl]oxy}-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-2,3-dihydro-1h-indole-1-carboxamide | Human | 3632 | |
| JAK2 | JakA | TK | 3ugc | A | B | 5-{[6-(acetylamino)pyrimidin-4-yl]oxy}-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-2,3-dihydro-1h-indole-1-carboxamide | Human | 3651 | |
| JAK2 | JakA | TK | 3zmm | A | A | 5-fluoro-4-[(1s)-1-(5-fluoropyrimidin-2-yl)ethoxy]-n-(5-methyl-1h-pyrazol-3-yl)-6-morpholino-pyrimidin-2-amine | Human | 3674 | |
| JAK2 | JakA | TK | 3zmm | A | B | 5-fluoro-4-[(1s)-1-(5-fluoropyrimidin-2-yl)ethoxy]-n-(5-methyl-1h-pyrazol-3-yl)-6-morpholino-pyrimidin-2-amine | Human | 3667 | |
| JAK2 | JakA | TK | 3zmm | B | A | 5-fluoro-4-[(1s)-1-(5-fluoropyrimidin-2-yl)ethoxy]-n-(5-methyl-1h-pyrazol-3-yl)-6-morpholino-pyrimidin-2-amine | Human | 3709 | |
| JAK2 | JakA | TK | 3zmm | B | B | 5-fluoro-4-[(1s)-1-(5-fluoropyrimidin-2-yl)ethoxy]-n-(5-methyl-1h-pyrazol-3-yl)-6-morpholino-pyrimidin-2-amine | Human | 3678 | |
| JAK2 | JakA | TK | 4aqc | A | A | 8-(4-methylsulfonylphenyl)-n-(4-morpholin-4-ylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine | Human | 3720 | |
| JAK2 | JakA | TK | 4aqc | A | B | 8-(4-methylsulfonylphenyl)-n-(4-morpholin-4-ylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine | Human | 3696 | |
| JAK2 | JakA | TK | 4aqc | B | A | 8-(4-methylsulfonylphenyl)-n-(4-morpholin-4-ylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine | Human | 3679 | |
| JAK2 | JakA | TK | 4aqc | B | B | 8-(4-methylsulfonylphenyl)-n-(4-morpholin-4-ylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amine | Human | 3676 | |
| JAK2 | JakA | TK | 4bbe | A | | n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]ethanamide | Human | 3670 | |
| JAK2 | JakA | TK | 4bbe | B | | n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]ethanamide | Human | 3727 | |
| JAK2 | JakA | TK | 4bbe | C | | n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]ethanamide | Human | 3649 | |
| JAK2 | JakA | TK | 4bbe | D | | n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]ethanamide | Human | 3726 | |
| JAK2 | JakA | TK | 4bbf | A | | (2r)-n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]pyrrolidine-2-carboxamide | Human | 3723 | |
| JAK2 | JakA | TK | 4bbf | B | | (2r)-n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]pyrrolidine-2-carboxamide | Human | 3717 | |
| JAK2 | JakA | TK | 4bbf | C | | (2r)-n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]pyrrolidine-2-carboxamide | Human | 3644 | |
| JAK2 | JakA | TK | 4bbf | D | | (2r)-n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]pyrrolidine-2-carboxamide | Human | 3663 | |
| JAK2 | JakA | TK | 4c61 | A | | n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-7-methyl-n4-(1-methylimidazol-4-yl)thieno[3,2-d]pyrimidine-2,4-diamine | Human | 3661 | |
| JAK2 | JakA | TK | 4c61 | B | | n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-7-methyl-n4-(1-methylimidazol-4-yl)thieno[3,2-d]pyrimidine-2,4-diamine | Human | 3645 | |
| JAK2 | JakA | TK | 4c62 | A | | n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(1-methylimidazol-4-yl)-6-morpholino-1,3,5-triazine-2,4-diamine | Human | 3655 | |
| JAK2 | JakA | TK | 4c62 | B | | n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(1-methylimidazol-4-yl)-6-morpholino-1,3,5-triazine-2,4-diamine | Human | 3625 | |
| JAK2 | JakA | TK | 4d0w | A | A | 5-(2-aminopyrimidin-4-yl)-2-(5-chloro-2-methylphenyl)-1h-pyrrole-3-carboxamide | Human | 3666 | |
| JAK2 | JakA | TK | 4d0w | A | B | 5-(2-aminopyrimidin-4-yl)-2-(5-chloro-2-methylphenyl)-1h-pyrrole-3-carboxamide | Human | 3650 | |
| JAK2 | JakA | TK | 4d0x | A | A | 5-(2-aminopyrimidin-4-yl)-2-[2-chloro-5-(trifluoromethyl)phenyl]-1h-pyrrole-3-carboxamide | Human | 3699 | |
| JAK2 | JakA | TK | 4d0x | A | B | 5-(2-aminopyrimidin-4-yl)-2-[2-chloro-5-(trifluoromethyl)phenyl]-1h-pyrrole-3-carboxamide | Human | 3642 | |
| JAK2 | JakA | TK | 4d1s | A | A | 2-(5-chloro-2-methylphenyl)-1-methyl-5-(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1h-pyrrole-3-carboxamide | Human | 3634 | |
| JAK2 | JakA | TK | 4d1s | A | B | 2-(5-chloro-2-methylphenyl)-1-methyl-5-(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1h-pyrrole-3-carboxamide | Human | 3627 | |
| JAK2 | JakA | TK | 4e4m | A | | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 3713 | |
| JAK2 | JakA | TK | 4e4m | B | | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 3712 | |
| JAK2 | JakA | TK | 4e4m | D | | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 3669 | |
| JAK2 | JakA | TK | 4e4m | E | | 1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 3637 | |
| JAK2 | JakA | TK | 4e6d | A | A | 3-[(3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl]-3-oxopropanenitrile | Human | 3689 | |
| JAK2 | JakA | TK | 4e6d | A | B | 3-[(3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl]-3-oxopropanenitrile | Human | 3656 | |
| JAK2 | JakA | TK | 4e6d | B | A | 3-[(3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl]-3-oxopropanenitrile | Human | 3631 | |
| JAK2 | JakA | TK | 4e6d | B | B | 3-[(3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl]-3-oxopropanenitrile | Human | 3647 | |
| JAK2 | JakA | TK | 4e6q | A | | 1-(1-benzylpiperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 3624 | |
| JAK2 | JakA | TK | 4e6q | B | | 1-(1-benzylpiperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 3671 | |
| JAK2 | JakA | TK | 4f08 | A | | 1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 3662 | |
| JAK2 | JakA | TK | 4f08 | B | | 1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 3719 | |
| JAK2 | JakA | TK | 4f09 | A | | 2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine | Human | 3622 | |
| JAK2 | JakA | TK | 4gfm | A | A | 2,6-dichloro-n-(2-oxo-2,5-dihydropyridin-4-yl)benzamide | Human | 3680 | |
| JAK2 | JakA | TK | 4gfm | A | B | 2,6-dichloro-n-(2-oxo-2,5-dihydropyridin-4-yl)benzamide | Human | 3705 | |
| JAK2 | JakA | TK | 4gmy | A | | 2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamide | Human | 3684 | |
| JAK2 | JakA | TK | 4hge | A | A | n-[1-(3-chlorophenyl)-3-methyl-1h-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 3703 | |
| JAK2 | JakA | TK | 4hge | A | B | n-[1-(3-chlorophenyl)-3-methyl-1h-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 3658 | |
| JAK2 | JakA | TK | 4hge | B | A | n-[1-(3-chlorophenyl)-3-methyl-1h-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 3706 | |
| JAK2 | JakA | TK | 4hge | B | B | n-[1-(3-chlorophenyl)-3-methyl-1h-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 3715 | |
| JAK2 | JakA | TK | 4iva | A | A | trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrile | Human | 3673 | |
| JAK2 | JakA | TK | 4iva | A | B | trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrile | Human | 3725 | |
| JAK2 | JakA | TK | 4iva | A | C | trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrile | Human | 3714 | |
| JAK2 | JakA | TK | 4ji9 | A | | n-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamide | Human | 3692 | |
| JAK2 | JakA | TK | 4ji9 | B | | n-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamide | Human | 3724 | |
| JAK2 | JakA | TK | 4jia | A | A | 5-(4-methoxyphenyl)-n-[4-(4-methylpiperazin-1-yl)phenyl][1,2,4]triazolo[1,5-a]pyridin-2-amine | Human | 3691 | |
| JAK2 | JakA | TK | 4jia | A | B | 5-(4-methoxyphenyl)-n-[4-(4-methylpiperazin-1-yl)phenyl][1,2,4]triazolo[1,5-a]pyridin-2-amine | Human | 3640 | |
| JAK2 | JakA | TK | 4p7e | A | | n-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide | Human | 3682 | |
| JAK2 | JakA | TK | 4p7e | B | | n-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide | Human | 3701 | |
| JAK2 | JakA | TK | 4ytc | A | A | n~3~-phenyl-1-[6-(phenylamino)pyrimidin-4-yl]-1h-1,2,4-triazole-3,5-diamine | Human | 3633 | |
| JAK2 | JakA | TK | 4ytc | A | B | n~3~-phenyl-1-[6-(phenylamino)pyrimidin-4-yl]-1h-1,2,4-triazole-3,5-diamine | Human | 3687 | |
| JAK2 | JakA | TK | 4ytf | A | A | n~2~-[2-(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl]-n-(2,2,2-trifluoroethyl)-l-alaninamide | Human | 3690 | |
| JAK2 | JakA | TK | 4ytf | A | B | n~2~-[2-(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl]-n-(2,2,2-trifluoroethyl)-l-alaninamide | Human | 3693 | |
| JAK2 | JakA | TK | 4yth | A | A | n~2~-[2-(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl]-2-methyl-n-(2,2,2-trifluoroethyl)-d-alaninamide | Human | 3710 | |
| JAK2 | JakA | TK | 4yth | A | B | n~2~-[2-(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl]-2-methyl-n-(2,2,2-trifluoroethyl)-d-alaninamide | Human | 3702 | |
| JAK2 | JakA | TK | 4yti | A | A | (2r)-2-methyl-2-[[2-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl]amino]-n-[2,2,2-tris(fluoranyl)ethyl]butanamide | Human | 3641 | |
| JAK2 | JakA | TK | 4yti | A | B | (2r)-2-methyl-2-[[2-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl]amino]-n-[2,2,2-tris(fluoranyl)ethyl]butanamide | Human | 3657 | |
| JAK2 | JakA | TK | 4zim | A | A | 3-(3,4-dichlorophenyl)-6-(morpholin-4-ylcarbonyl)-9h-carbazole-1-carboxamide | Human | 3704 | |
| JAK2 | JakA | TK | 4zim | A | B | 3-(3,4-dichlorophenyl)-6-(morpholin-4-ylcarbonyl)-9h-carbazole-1-carboxamide | Human | 3659 | |
| JAK2 | JakA | TK | 4zim | B | A | 3-(3,4-dichlorophenyl)-6-(morpholin-4-ylcarbonyl)-9h-carbazole-1-carboxamide | Human | 3660 | |
| JAK2 | JakA | TK | 4zim | B | B | 3-(3,4-dichlorophenyl)-6-(morpholin-4-ylcarbonyl)-9h-carbazole-1-carboxamide | Human | 3697 | |
| JAK2 | JakA | TK | 5aep | A | A | 1-(5-chloro-2-methylphenyl)-4-(pyrrolo[2,1-f][1,2,4]triazin-4-yl)-1h-pyrrole-2-carboxamide | Human | 3629 | |
| JAK2 | JakA | TK | 5aep | A | B | 1-(5-chloro-2-methylphenyl)-4-(pyrrolo[2,1-f][1,2,4]triazin-4-yl)-1h-pyrrole-2-carboxamide | Human | 3686 | |
| JAK2 | JakA | TK | 5cf4 | A | | n,n-dicyclopropyl-6-ethyl-4-[(3-methoxypropyl)amino]-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5980 | |
| JAK2 | JakA | TK | 5cf4 | B | | n,n-dicyclopropyl-6-ethyl-4-[(3-methoxypropyl)amino]-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5982 | |
| JAK2 | JakA | TK | 5cf5 | A | | n,n-dicyclopropyl-4-[(4,5-dimethyl-1,3-thiazol-2-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5984 | |
| JAK2 | JakA | TK | 5cf5 | B | | n,n-dicyclopropyl-4-[(4,5-dimethyl-1,3-thiazol-2-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5976 | |
| JAK2 | JakA | TK | 5cf6 | A | | n,n-dicyclopropyl-6-[(2s)-2,3-dihydroxypropyl]-1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5979 | |
| JAK2 | JakA | TK | 5cf6 | B | | n,n-dicyclopropyl-6-[(2s)-2,3-dihydroxypropyl]-1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5977 | |
| JAK2 | JakA | TK | 5cf8 | A | A | n,n-dicyclopropyl-4-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5978 | |
| JAK2 | JakA | TK | 5cf8 | A | B | n,n-dicyclopropyl-4-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5981 | |
| JAK2 | JakA | TK | 5cf8 | B | A | n,n-dicyclopropyl-4-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5985 | |
| JAK2 | JakA | TK | 5cf8 | B | B | n,n-dicyclopropyl-4-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamide | Human | 5983 | |
| JAK2 | JakA | TK | 5hez | A | | n-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamide | Human | 7254 | |
| JAK2 | JakA | TK | 5hez | B | | n-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamide | Human | 7255 | |
| JAK2 | JakA | TK | 5hez | C | | n-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamide | Human | 7253 | |
| JAK2 | JakA | TK | 5hez | D | | n-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamide | Human | 7252 | |
| JAK2 | JakA | TK | 5l3a | A | A | ~{n}-(1~{h}-indazol-4-yl)methanesulfonamide | Human | 6561 | |
| JAK2 | JakA | TK | 5l3a | A | B | ~{n}-(1~{h}-indazol-4-yl)methanesulfonamide | Human | 6560 | |
| JAK2 | JakA | TK | 5tq3 | A | A | 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-3-ethylphenol | Human | 7359 | |
| JAK2 | JakA | TK | 5tq3 | A | B | 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-3-ethylphenol | Human | 7356 | |
| JAK2 | JakA | TK | 5tq3 | B | A | 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-3-ethylphenol | Human | 7360 | |
| JAK2 | JakA | TK | 5tq3 | B | B | 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-3-ethylphenol | Human | 7352 | |
| JAK2 | JakA | TK | 5tq4 | A | | 6-(2-ethyl-4-hydroxyphenyl)-1h-indazole-3-carboxamide | Human | 7351 | |
| JAK2 | JakA | TK | 5tq5 | A | | 6-(2-ethyl-4-hydroxyphenyl)-n-(6-methylpyridin-3-yl)-1h-indazole-3-carboxamide | Human | 7358 | |
| JAK2 | JakA | TK | 5tq6 | A | | {(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}(pyrrolidin-1-yl)methanone | Human | 7354 | |
| JAK2 | JakA | TK | 5tq6 | B | | {(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}(pyrrolidin-1-yl)methanone | Human | 7361 | |
| JAK2 | JakA | TK | 5tq7 | A | | {(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}[(3r)-3-(phenylsulfonyl)pyrrolidin-1-yl]methanone | Human | 7355 | |
| JAK2 | JakA | TK | 5tq7 | B | | {(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}[(3r)-3-(phenylsulfonyl)pyrrolidin-1-yl]methanone | Human | 7353 | |
| JAK2 | JakA | TK | 5tq8 | A | | {2-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-2h-indazol-3-yl]-3,4,6,7-tetrahydro-5h-imidazo[4,5-c]pyridin-5-yl}[5-(piperidin-1-yl)pyrazin-2-yl]methanone | Human | 7357 | |
| JAK2 | JakA | TK | 5usy | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8101 | |
| JAK2 | JakA | TK | 5usy | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8102 | |
| JAK2 | JakA | TK | 5usy | B | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8103 | |
| JAK2 | JakA | TK | 5usy | B | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8104 | |
| JAK2 | JakA | TK | 5wev | A | A | n-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamide | Human | 8377 | |
| JAK2 | JakA | TK | 5wev | A | B | n-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamide | Human | 8376 | |
| JAK2 | JakA | TK | 6aaj | A | | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10515 | |
| JAK2 | JakA | TK | 6aaj | B | | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10514 | |
| JAK2 | JakA | TK | 6bbv | A | | n-{cis-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamide | Human | 9504 | |
| JAK2 | JakA | TK | 6drw | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 10512 | |
| JAK2 | JakA | TK | 6drw | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 10513 | |
| JAK2 | JakA | TK | 6tpd | A | | 3-methyl-4-phenyl-2,7-dihydropyrazolo[3,4-b]pyridin-6-one | Human | 12350 | |
| JAK2 | JakA | TK | 6vgl | A | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13223 | |
| JAK2 | JakA | TK | 6vgl | B | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13222 | |
| JAK2 | JakA | TK | 6vgl | C | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13221 | |
| JAK2 | JakA | TK | 6vgl | D | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13220 | |
| JAK2 | JakA | TK | 6vn8 | A | | baricitinib | Human | 13291 | |
| JAK2 | JakA | TK | 6vn8 | B | | baricitinib | Human | 13301 | |
| JAK2 | JakA | TK | 6vnb | A | | (3s)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13298 | |
| JAK2 | JakA | TK | 6vnc | A | | (3r)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13359 | |
| JAK2 | JakA | TK | 6vnc | B | | (3r)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13348 | |
| JAK2 | JakA | TK | 6vne | A | | n-tert-butyl-3-{[5-methyl-2-({4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}amino)pyrimidin-4-yl]amino}benzenesulfonamide | Human | 13296 | |
| JAK2 | JakA | TK | 6vne | B | | n-tert-butyl-3-{[5-methyl-2-({4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}amino)pyrimidin-4-yl]amino}benzenesulfonamide | Human | 13302 | |
| JAK2 | JakA | TK | 6vnf | A | A | n~4~-[1-(tert-butylsulfonyl)-2,3-dihydro-1h-indol-6-yl]-n~2~-[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]-5-methylpyrimidine-2,4-diamine | Human | 13347 | |
| JAK2 | JakA | TK | 6vnf | A | B | n~4~-[1-(tert-butylsulfonyl)-2,3-dihydro-1h-indol-6-yl]-n~2~-[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]-5-methylpyrimidine-2,4-diamine | Human | 13357 | |
| JAK2 | JakA | TK | 6vnf | B | A | n~4~-[1-(tert-butylsulfonyl)-2,3-dihydro-1h-indol-6-yl]-n~2~-[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]-5-methylpyrimidine-2,4-diamine | Human | 13346 | |
| JAK2 | JakA | TK | 6vnf | B | B | n~4~-[1-(tert-butylsulfonyl)-2,3-dihydro-1h-indol-6-yl]-n~2~-[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]-5-methylpyrimidine-2,4-diamine | Human | 13352 | |
| JAK2 | JakA | TK | 6vng | A | | n-{2-fluoro-5-[(2-{[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]phenyl}-2-methylpropane-2-sulfonamide | Human | 13358 | |
| JAK2 | JakA | TK | 6vng | B | | n-{2-fluoro-5-[(2-{[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]phenyl}-2-methylpropane-2-sulfonamide | Human | 13341 | |
| JAK2 | JakA | TK | 6vnh | A | | n-{5-[(2-{[3,5-difluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]-2-fluorophenyl}-2-methylpropane-2-sulfonamide | Human | 13344 | |
| JAK2 | JakA | TK | 6vnh | B | | n-{5-[(2-{[3,5-difluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]-2-fluorophenyl}-2-methylpropane-2-sulfonamide | Human | 13342 | |
| JAK2 | JakA | TK | 6vni | A | | 2-{5-[(2-{[3,5-difluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]-2-fluorophenyl}-1lambda~6~,2-thiazolidine-1,1-dione | Human | 13294 | |
| JAK2 | JakA | TK | 6vnj | A | A | 3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13340 | |
| JAK2 | JakA | TK | 6vnj | B | A | 3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13355 | |
| JAK2 | JakA | TK | 6vnk | A | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13293 | |
| JAK2 | JakA | TK | 6vnk | B | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13295 | |
| JAK2 | JakA | TK | 6vnk | C | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13304 | |
| JAK2 | JakA | TK | 6vnk | D | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13292 | |
| JAK2 | JakA | TK | 6vnl | A | | 4-[[4-[[3-(~{tert}-butylsulfonylamino)-4-chloranyl-phenyl]amino]-5-methyl-pyrimidin-2-yl]amino]-2-fluoranyl-~{n}-(1-methylpiperidin-4-yl)benzamide | Human | 13303 | |
| JAK2 | JakA | TK | 6vnl | B | | 4-[[4-[[3-(~{tert}-butylsulfonylamino)-4-chloranyl-phenyl]amino]-5-methyl-pyrimidin-2-yl]amino]-2-fluoranyl-~{n}-(1-methylpiperidin-4-yl)benzamide | Human | 13299 | |
| JAK2 | JakA | TK | 6vnl | C | | 4-[[4-[[3-(~{tert}-butylsulfonylamino)-4-chloranyl-phenyl]amino]-5-methyl-pyrimidin-2-yl]amino]-2-fluoranyl-~{n}-(1-methylpiperidin-4-yl)benzamide | Human | 13300 | |
| JAK2 | JakA | TK | 6vnl | D | | 4-[[4-[[3-(~{tert}-butylsulfonylamino)-4-chloranyl-phenyl]amino]-5-methyl-pyrimidin-2-yl]amino]-2-fluoranyl-~{n}-(1-methylpiperidin-4-yl)benzamide | Human | 13297 | |
| JAK2 | JakA | TK | 6vnm | A | | 4-[1-(but-3-en-1-yl)-1h-pyrazol-4-yl]-n-[4-(piperidin-4-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-2-amine | Human | 13354 | |
| JAK2 | JakA | TK | 6vnm | B | | 4-[1-(but-3-en-1-yl)-1h-pyrazol-4-yl]-n-[4-(piperidin-4-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-2-amine | Human | 13351 | |
| JAK2 | JakA | TK | 6vs3 | A | | (3r)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13349 | |
| JAK2 | JakA | TK | 6vs3 | B | | (3r)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13345 | |
| JAK2 | JakA | TK | 6vsn | A | | (3s)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13353 | |
| JAK2 | JakA | TK | 6vsn | B | | (3s)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13356 | |
| JAK2 | JakA | TK | 6vsn | C | | (3s)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13350 | |
| JAK2 | JakA | TK | 6vsn | D | | (3s)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13343 | |
| JAK2 | JakA | TK | 6wtn | A | A | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13538 | |
| JAK2 | JakA | TK | 6wtn | A | B | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13540 | |
| JAK2 | JakA | TK | 6wto | A | A | baricitinib | Human | 13536 | |
| JAK2 | JakA | TK | 6wto | A | B | baricitinib | Human | 13539 | |
| JAK2 | JakA | TK | 6wtp | A | A | tert-butyl 4-[(4-{1-[3-(cyanomethyl)-1-(ethylsulfonyl)azetidin-3-yl]-1h-pyrazol-4-yl}-7h-pyrrolo[2,3-d]pyrimidin-2-yl)amino]benzoate | Human | 13541 | |
| JAK2 | JakA | TK | 6wtp | A | B | tert-butyl 4-[(4-{1-[3-(cyanomethyl)-1-(ethylsulfonyl)azetidin-3-yl]-1h-pyrazol-4-yl}-7h-pyrrolo[2,3-d]pyrimidin-2-yl)amino]benzoate | Human | 13542 | |
| JAK2 | JakA | TK | 6wtq | A | A | n-methyl-4-{[4-(1-propyl-1h-pyrazol-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-2-yl]amino}benzamide | Human | 13535 | |
| JAK2 | JakA | TK | 6wtq | A | B | n-methyl-4-{[4-(1-propyl-1h-pyrazol-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-2-yl]amino}benzamide | Human | 13537 | |
| JAK2 | JakA | TK | 6x8e | A | A | [3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrile | Human | 13154 | |
| JAK2 | JakA | TK | 6x8e | A | B | [3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrile | Human | 13152 | |
| JAK2 | JakA | TK | 6x8e | B | A | [3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrile | Human | 13155 | |
| JAK2 | JakA | TK | 6x8e | B | B | [3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrile | Human | 13153 | |
| JAK2 | JakA | TK | 7ll4 | A | A | {1-(ethylsulfonyl)-3-[4-(2-{[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]azetidin-3-yl}acetonitrile | Human | 14035 | |
| JAK2 | JakA | TK | 7ll4 | A | B | {1-(ethylsulfonyl)-3-[4-(2-{[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]azetidin-3-yl}acetonitrile | Human | 14037 | |
| JAK2 | JakA | TK | 7ll5 | A | A | {1-(ethylsulfonyl)-3-[4-(2-{[4-(1-methylpiperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]azetidin-3-yl}acetonitrile | Human | 14036 | |
| JAK2 | JakA | TK | 7ll5 | A | B | {1-(ethylsulfonyl)-3-[4-(2-{[4-(1-methylpiperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]azetidin-3-yl}acetonitrile | Human | 14038 | |
| JAK2 | JakA | TK | 7q7i | A | A | 4-[8-methoxy-2-[(1-methylpyrazol-4-yl)amino]quinazolin-6-yl]phenol | Human | 14085 | |
| JAK2 | JakA | TK | 7q7i | A | B | 4-[8-methoxy-2-[(1-methylpyrazol-4-yl)amino]quinazolin-6-yl]phenol | Human | 14088 | |
| JAK2 | JakA | TK | 7q7k | A | A | 4-(2-azanyl-8-methoxy-quinazolin-6-yl)phenol | Human | 14091 | |
| JAK2 | JakA | TK | 7q7k | A | B | 4-(2-azanyl-8-methoxy-quinazolin-6-yl)phenol | Human | 14086 | |
| JAK2 | JakA | TK | 7q7l | A | A | 4-[2-azanyl-8-[[(2~{s})-1-oxidanylpropan-2-yl]amino]quinazolin-6-yl]-5-ethyl-2-fluoranyl-phenol | Human | 14092 | |
| JAK2 | JakA | TK | 7q7l | A | B | 4-[2-azanyl-8-[[(2~{s})-1-oxidanylpropan-2-yl]amino]quinazolin-6-yl]-5-ethyl-2-fluoranyl-phenol | Human | 14090 | |
| JAK2 | JakA | TK | 7q7w | A | A | 4-[2-[5-(dimethylamino)pentylamino]-8-[[(2~{s})-1-oxidanylpropan-2-yl]amino]quinazolin-6-yl]-5-ethyl-2-fluoranyl-phenol | Human | 14087 | |
| JAK2 | JakA | TK | 7q7w | A | B | 4-[2-[5-(dimethylamino)pentylamino]-8-[[(2~{s})-1-oxidanylpropan-2-yl]amino]quinazolin-6-yl]-5-ethyl-2-fluoranyl-phenol | Human | 14089 | |
| JAK2 | JakA | TK | 7ree | A | A | [3-(4-{2-[3,5-difluoro-4-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)anilino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}-1h-pyrazol-1-yl)-1-(ethanesulfonyl)azetidin-3-yl]acetonitrile | Human | 13855 | |
| JAK2 | JakA | TK | 7ree | A | B | [3-(4-{2-[3,5-difluoro-4-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)anilino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}-1h-pyrazol-1-yl)-1-(ethanesulfonyl)azetidin-3-yl]acetonitrile | Human | 13856 | |
| JAK2 | JakA | TK | 7rn6 | A | A | 5-{[6-(acetylamino)pyrimidin-4-yl]oxy}-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-2,3-dihydro-1h-indole-1-carboxamide | Human | 13956 | |
| JAK2 | JakA | TK | 7rn6 | A | B | 5-{[6-(acetylamino)pyrimidin-4-yl]oxy}-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-2,3-dihydro-1h-indole-1-carboxamide | Human | 13955 | |
| JAK2 | JakA | TK | 7teu | A | A | 3-{(4s)-2-[(cyclopropanecarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}-4-methylbenzamide | Human | 14806 | |
| JAK2 | JakA | TK | 7teu | A | B | 3-{(4s)-2-[(cyclopropanecarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}-4-methylbenzamide | Human | 14811 | |
| JAK2 | JakA | TK | 7uyw | A | A | 2-(2,6-difluorophenyl)-4-[4-(pyrrolidine-1-carbonyl)anilino]-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 14333 | |
| JAK2 | JakA | TK | 7uyw | A | B | 2-(2,6-difluorophenyl)-4-[4-(pyrrolidine-1-carbonyl)anilino]-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 14334 | |
| JAK2 | JakA | TK | 8bm2 | A | A | 3-[(4-chloranyl-2-fluoranyl-phenyl)methyl]-2-methyl-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)-8-(morpholin-4-ylmethyl)imidazo[1,2-b]pyridazin-6-amine | Human | 15043 | |
| JAK2 | JakA | TK | 8bm2 | A | B | 3-[(4-chloranyl-2-fluoranyl-phenyl)methyl]-2-methyl-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)-8-(morpholin-4-ylmethyl)imidazo[1,2-b]pyridazin-6-amine | Human | 15035 | |
| JAK2 | JakA | TK | 8bpv | A | A | 11-(2-pyrrolidin-1-yl-ethoxy)-14,19-dioxa-5,7,26-triaza-tetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaene | Human | 15040 | |
| JAK2 | JakA | TK | 8bpv | A | B | 11-(2-pyrrolidin-1-yl-ethoxy)-14,19-dioxa-5,7,26-triaza-tetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaene | Human | 15036 | |
| JAK2 | JakA | TK | 8bpw | A | A | lestaurtinib | Human | 15044 | |
| JAK2 | JakA | TK | 8bpw | A | B | lestaurtinib | Human | 15039 | |
| JAK2 | JakA | TK | 8bx6 | A | A | cerdulatinib | Human | 15033 | |
| JAK2 | JakA | TK | 8bx6 | A | B | cerdulatinib | Human | 15042 | |
| JAK2 | JakA | TK | 8bx9 | A | A | ilginatinib | Human | 15038 | |
| JAK2 | JakA | TK | 8bx9 | A | B | ilginatinib | Human | 15034 | |
| JAK2 | JakA | TK | 8bxc | A | A | itacitinib | Human | 15037 | |
| JAK2 | JakA | TK | 8bxc | A | B | itacitinib | Human | 15041 | |
| JAK2 | JakA | TK | 8bxh | A | A | momelotinib | Human | 15032 | |
| JAK2 | JakA | TK | 8bxh | A | B | momelotinib | Human | 15045 | |
| JAK2 | JakA | TK | 8g6z | A | A | (3r)-3-cyclopentyl-3-[(4m)-4-{5-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-1h-pyrazol-1-yl]propanenitrile | Human | 14808 | |
| JAK2 | JakA | TK | 8g6z | A | B | (3r)-3-cyclopentyl-3-[(4m)-4-{5-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-1h-pyrazol-1-yl]propanenitrile | Human | 14810 | |
| JAK2 | JakA | TK | 8g8o | A | A | [1-{5-methyl-2-[(3-methyl-1,2-thiazol-5-yl)amino]pyrimidin-4-yl}-3-(4-methylpiperazin-1-yl)azetidin-3-yl]acetonitrile | Human | 14807 | |
| JAK2 | JakA | TK | 8g8o | A | B | [1-{5-methyl-2-[(3-methyl-1,2-thiazol-5-yl)amino]pyrimidin-4-yl}-3-(4-methylpiperazin-1-yl)azetidin-3-yl]acetonitrile | Human | 14809 | |
| JAK2 | JakA | TK | 8g8x | A | A | 3-cyclopropyl-1-{5-methyl-2-[(3-methyl-1,2-thiazol-5-yl)amino]pyrimidin-4-yl}azetidin-3-ol | Human | 14804 | |
| JAK2 | JakA | TK | 8g8x | A | B | 3-cyclopropyl-1-{5-methyl-2-[(3-methyl-1,2-thiazol-5-yl)amino]pyrimidin-4-yl}azetidin-3-ol | Human | 14805 | |
| JAK2-b | JakB | TK | 4fvp | A | | - | Human | 1222 | |
| JAK2-b | JakB | TK | 4fvq | A | | adenosine-5'-triphosphate | Human | 1224 | |
| JAK2-b | JakB | TK | 4fvr | A | | adenosine-5'-triphosphate | Human | 1223 | |
| JAK2-b | JakB | TK | 5i4n | A | A | adenosine-5'-triphosphate | Human | 6525 | |
| JAK2-b | JakB | TK | 5i4n | A | B | adenosine-5'-triphosphate | Human | 6524 | |
| JAK2-b | JakB | TK | 5usz | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8048 | |
| JAK2-b | JakB | TK | 5usz | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 8043 | |
| JAK2-b | JakB | TK | 5ut0 | A | A | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 8041 | |
| JAK2-b | JakB | TK | 5ut0 | A | B | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 8047 | |
| JAK2-b | JakB | TK | 5ut1 | A | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 8046 | |
| JAK2-b | JakB | TK | 5ut1 | A | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 8049 | |
| JAK2-b | JakB | TK | 5ut2 | A | A | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamide | Human | 8040 | |
| JAK2-b | JakB | TK | 5ut2 | A | B | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamide | Human | 8039 | |
| JAK2-b | JakB | TK | 5ut3 | A | | 5-phenyl-2-ureidothiophene-3-carboxamide | Human | 8044 | |
| JAK2-b | JakB | TK | 5ut4 | A | | 8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-(1-piperidin-4-yl-1h-pyrazol-4-yl)quinoxaline | Human | 8038 | |
| JAK2-b | JakB | TK | 5ut5 | A | A | n-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide | Human | 8042 | |
| JAK2-b | JakB | TK | 5ut5 | A | B | n-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamide | Human | 8037 | |
| JAK2-b | JakB | TK | 5ut6 | A | A | 4-({4-amino-6-[3-(hydroxymethyl)-1h-pyrazol-1-yl]pyrimidin-2-yl}amino)benzonitrile | Human | 8036 | |
| JAK2-b | JakB | TK | 5ut6 | A | B | 4-({4-amino-6-[3-(hydroxymethyl)-1h-pyrazol-1-yl]pyrimidin-2-yl}amino)benzonitrile | Human | 8045 | |
| JAK2-b | JakB | TK | 5wij | A | | 4-{[6-(cyclohexylmethoxy)-7h-purin-2-yl]amino}-n,n-diethylbenzamide | Human | 10388 | |
| JAK2-b | JakB | TK | 5wik | B | | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 10387 | |
| JAK2-b | JakB | TK | 5wil | A | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 10379 | |
| JAK2-b | JakB | TK | 5wim | A | | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 10385 | |
| JAK2-b | JakB | TK | 5win | A | | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 10378 | |
| JAK2-b | JakB | TK | 6brw | A | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 10382 | |
| JAK2-b | JakB | TK | 6brw | A | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 10377 | |
| JAK2-b | JakB | TK | 6bs0 | A | A | 4-(5-aminopyrazin-2-yl)-1h-pyrrolo[2,3-b]pyridin-6-amine | Human | 10380 | |
| JAK2-b | JakB | TK | 6bs0 | A | B | 4-(5-aminopyrazin-2-yl)-1h-pyrrolo[2,3-b]pyridin-6-amine | Human | 10381 | |
| JAK2-b | JakB | TK | 6bss | A | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 10386 | |
| JAK2-b | JakB | TK | 6d2i | A | | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 10967 | |
| JAK2-b | JakB | TK | 6d2i | B | | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 10966 | |
| JAK2-b | JakB | TK | 6g3c | A | A | 2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-one | Human | 10978 | |
| JAK2-b | JakB | TK | 6g3c | A | B | 2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-one | Human | 10976 | |
| JAK2-b | JakB | TK | 6g3c | B | A | 2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-one | Human | 10977 | |
| JAK2-b | JakB | TK | 6g3c | B | B | 2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-one | Human | 10975 | |
| JAK2-b | JakB | TK | 6m9h | A | A | 4-({4-amino-6-[4-(2-hydroxyethyl)-1h-imidazol-1-yl]pyrimidin-2-yl}amino)benzonitrile | Human | 10384 | |
| JAK2-b | JakB | TK | 6m9h | A | B | 4-({4-amino-6-[4-(2-hydroxyethyl)-1h-imidazol-1-yl]pyrimidin-2-yl}amino)benzonitrile | Human | 10383 | |
| JAK2-b | JakB | TK | 6oav | A | | 5-amino-3-[(4-cyanophenyl)amino]-n-phenyl-1h-1,2,4-triazole-1-carboxamide | Human | 12099 | |
| JAK2-b | JakB | TK | 6obb | A | | 5-amino-n-phenyl-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carboxamide | Human | 12097 | |
| JAK2-b | JakB | TK | 6obf | A | | [4-({5-amino-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenoxy]acetic acid | Human | 12098 | |
| JAK2-b | JakB | TK | 6obl | A | | [4-({5-amino-3-[(4-cyanophenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenoxy]acetic acid | Human | 12101 | |
| JAK2-b | JakB | TK | 6occ | A | | 2-[4-({5-amino-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenyl]-1,3-oxazole-4-carboxylic acid | Human | 12100 | |
| JAK3 | JakA | TK | 1yvj | A | A | 1,2,3,4-tetrahydrogen-staurosporine | Human | 460 | |
| JAK3 | JakA | TK | 1yvj | A | B | 1,2,3,4-tetrahydrogen-staurosporine | Human | 451 | |
| JAK3 | JakA | TK | 3lxk | A | | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 436 | |
| JAK3 | JakA | TK | 3lxl | A | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 434 | |
| JAK3 | JakA | TK | 3lxl | A | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 443 | |
| JAK3 | JakA | TK | 3pjc | A | | 3-(1h-indol-3-yl)-4-[2-(4-oxopiperidin-1-yl)-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrrole-2,5-dione | Human | 444 | |
| JAK3 | JakA | TK | 3zc6 | A | A | n-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 442 | |
| JAK3 | JakA | TK | 3zc6 | A | B | n-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 461 | |
| JAK3 | JakA | TK | 3zc6 | B | A | n-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 449 | |
| JAK3 | JakA | TK | 3zc6 | B | B | n-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 447 | |
| JAK3 | JakA | TK | 3zc6 | C | A | n-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 433 | |
| JAK3 | JakA | TK | 3zc6 | C | B | n-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 445 | |
| JAK3 | JakA | TK | 3zc6 | D | A | n-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 446 | |
| JAK3 | JakA | TK | 3zc6 | D | B | n-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 459 | |
| JAK3 | JakA | TK | 3zep | A | A | 2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 448 | |
| JAK3 | JakA | TK | 3zep | A | B | 2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 456 | |
| JAK3 | JakA | TK | 3zep | B | A | 2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 430 | |
| JAK3 | JakA | TK | 3zep | B | B | 2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 437 | |
| JAK3 | JakA | TK | 3zep | C | A | 2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 439 | |
| JAK3 | JakA | TK | 3zep | C | B | 2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 462 | |
| JAK3 | JakA | TK | 3zep | D | A | 2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 454 | |
| JAK3 | JakA | TK | 3zep | D | B | 2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 457 | |
| JAK3 | JakA | TK | 4hvd | A | | 2-cyclopropyl-n-[(2s)-3,3-dimethylbutan-2-yl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 431 | |
| JAK3 | JakA | TK | 4hvg | A | | 2-cyclopropyl-n-[(2s)-3-hydroxy-3-methylbutan-2-yl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 450 | |
| JAK3 | JakA | TK | 4hvh | A | | 2-cyclopropyl-n-[(2r)-3-hydroxy-3-methylbutan-2-yl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 441 | |
| JAK3 | JakA | TK | 4hvi | A | | 2-cyclopropyl-n-[(2r)-1-oxo-1-(piperidin-1-yl)propan-2-yl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 438 | |
| JAK3 | JakA | TK | 4i6q | A | | n-[(1s)-1-cyclopropylethyl]-2-phenoxy-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 432 | |
| JAK3 | JakA | TK | 4qps | A | A | n-{1-[6-(phenylamino)pyrazin-2-yl]-1h-benzimidazol-6-yl}prop-2-enamide | Human | 453 | |
| JAK3 | JakA | TK | 4qps | A | B | n-{1-[6-(phenylamino)pyrazin-2-yl]-1h-benzimidazol-6-yl}prop-2-enamide | Human | 458 | |
| JAK3 | JakA | TK | 4qps | C | A | n-{1-[6-(phenylamino)pyrazin-2-yl]-1h-benzimidazol-6-yl}prop-2-enamide | Human | 435 | |
| JAK3 | JakA | TK | 4qps | C | B | n-{1-[6-(phenylamino)pyrazin-2-yl]-1h-benzimidazol-6-yl}prop-2-enamide | Human | 455 | |
| JAK3 | JakA | TK | 4qt1 | A | | 1-{(3s)-1-[(2-methylpropyl)sulfonyl]piperidin-3-yl}-3-(5h-pyrrolo[2,3-b]pyrazin-2-yl)urea | Human | 452 | |
| JAK3 | JakA | TK | 4rio | A | | 4-{[(1r,2s)-2-fluoro-2-methylcyclopentyl]amino}pyrrolo[1,2-b]pyridazine-3-carboxamide | Human | 440 | |
| JAK3 | JakA | TK | 4v0g | A | A | n-[3-(2-{3-amino-6-[1-(1-methylpiperidin-4-yl)-1h-pyrazol-4-yl]pyrazin-2-yl}-1h-benzimidazol-1-yl)phenyl]propanamide | Human | 6347 | |
| JAK3 | JakA | TK | 4v0g | A | B | n-[3-(2-{3-amino-6-[1-(1-methylpiperidin-4-yl)-1h-pyrazol-4-yl]pyrazin-2-yl}-1h-benzimidazol-1-yl)phenyl]propanamide | Human | 6346 | |
| JAK3 | JakA | TK | 4v0g | B | A | n-[3-(2-{3-amino-6-[1-(1-methylpiperidin-4-yl)-1h-pyrazol-4-yl]pyrazin-2-yl}-1h-benzimidazol-1-yl)phenyl]propanamide | Human | 6348 | |
| JAK3 | JakA | TK | 4v0g | B | B | n-[3-(2-{3-amino-6-[1-(1-methylpiperidin-4-yl)-1h-pyrazol-4-yl]pyrazin-2-yl}-1h-benzimidazol-1-yl)phenyl]propanamide | Human | 6345 | |
| JAK3 | JakA | TK | 4z16 | A | | n-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamide | Human | 6395 | |
| JAK3 | JakA | TK | 4z16 | B | | n-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamide | Human | 6396 | |
| JAK3 | JakA | TK | 4z16 | C | | n-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamide | Human | 6397 | |
| JAK3 | JakA | TK | 4z16 | D | | n-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamide | Human | 6394 | |
| JAK3 | JakA | TK | 5lwm | A | A | 2-cyano-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1,4,6,8,11-pentaen-4-yl)furan-2-yl]-~{n},~{n}-dimethyl-prop-2-enamide | Human | 7115 | |
| JAK3 | JakA | TK | 5lwm | A | B | 2-cyano-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1,4,6,8,11-pentaen-4-yl)furan-2-yl]-~{n},~{n}-dimethyl-prop-2-enamide | Human | 7118 | |
| JAK3 | JakA | TK | 5lwn | A | A | (~{z})-2-cyano-~{n},~{n}-dimethyl-3-[5-[3-[(1~{s},2~{r})-2-methylcyclohexyl]-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1,4,6,8,11-pentaen-4-yl]furan-2-yl]prop-2-enamide | Human | 7117 | |
| JAK3 | JakA | TK | 5lwn | A | B | (2~{s})-2-cyano-~{n},~{n}-dimethyl-3-[5-[3-[(1~{s},2~{r})-2-methylcyclohexyl]-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1,4,6,8,11-pentaen-4-yl]furan-2-yl]propanamide | Human | 7116 | |
| JAK3 | JakA | TK | 5toz | A | | 1-{(2s,5r)-2-methyl-5-[(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}propan-1-one | Human | 7163 | |
| JAK3 | JakA | TK | 5tts | A | | 1-{(3r)-3-[(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}propan-1-one | Human | 7439 | |
| JAK3 | JakA | TK | 5ttu | A | A | 1-[(3ar,7ar)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)octahydro-6h-pyrrolo[2,3-c]pyridin-6-yl]propan-1-one | Human | 7435 | |
| JAK3 | JakA | TK | 5ttu | A | B | 1-[(3ar,7ar)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)octahydro-6h-pyrrolo[2,3-c]pyridin-6-yl]propan-1-one | Human | 7438 | |
| JAK3 | JakA | TK | 5ttv | A | A | n-[3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]propanamide | Human | 7437 | |
| JAK3 | JakA | TK | 5ttv | A | B | n-[3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]propanamide | Human | 7436 | |
| JAK3 | JakA | TK | 5vo6 | A | | 4-{[(1r,3s)-3-amino-2,2,3-trimethylcyclopentyl]amino}-6-phenylpyrrolo[1,2-b]pyridazine-3-carboxamide | Human | 7960 | |
| JAK3 | JakA | TK | 5w86 | A | A | 4-(benzylamino)-6-({4-[(1-methylpiperidin-4-yl)carbamoyl]phenyl}amino)pyridine-3-carboxamide | Human | 8549 | |
| JAK3 | JakA | TK | 5w86 | B | A | 4-(benzylamino)-6-({4-[(1-methylpiperidin-4-yl)carbamoyl]phenyl}amino)pyridine-3-carboxamide | Human | 8551 | |
| JAK3 | JakA | TK | 5w86 | C | A | 4-(benzylamino)-6-({4-[(1-methylpiperidin-4-yl)carbamoyl]phenyl}amino)pyridine-3-carboxamide | Human | 8550 | |
| JAK3 | JakA | TK | 5w86 | D | A | 4-(benzylamino)-6-({4-[(1-methylpiperidin-4-yl)carbamoyl]phenyl}amino)pyridine-3-carboxamide | Human | 8548 | |
| JAK3 | JakA | TK | 5wfj | A | | 4-({[3-(propanoylamino)phenyl]methyl}amino)pyrrolo[1,2-b]pyridazine-3-carboxamide | Human | 8535 | |
| JAK3 | JakA | TK | 6aak | A | | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10366 | |
| JAK3 | JakA | TK | 6aak | B | | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10367 | |
| JAK3 | JakA | TK | 6aak | C | | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10368 | |
| JAK3 | JakA | TK | 6aak | D | | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10365 | |
| JAK3 | JakA | TK | 6da4 | A | | (z)-1-{2,2-difluoro-6-[5-(2-methoxyethyl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]-2,3-dihydro-4h-1,4-benzoxazin-4-yl}methanimine | Human | 10723 | |
| JAK3 | JakA | TK | 6db3 | A | A | [(1s)-1-methyl-6-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]cyanamide | Human | 10718 | |
| JAK3 | JakA | TK | 6db3 | A | B | [(1s)-1-methyl-6-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]cyanamide | Human | 10719 | |
| JAK3 | JakA | TK | 6db4 | A | A | n-[(1s)-6-(5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]imidoformamide | Human | 10724 | |
| JAK3 | JakA | TK | 6db4 | A | B | n-[(1s)-6-(5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]imidoformamide | Human | 10721 | |
| JAK3 | JakA | TK | 6dud | A | A | n-[(1s)-6-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]imidoformamide | Human | 10722 | |
| JAK3 | JakA | TK | 6dud | A | B | n-[(1s)-6-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]imidoformamide | Human | 10720 | |
| JAK3 | JakA | TK | 6gl9 | A | A | (~{e})-3-[3-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)phenyl]prop-2-enenitrile | Human | 10014 | |
| JAK3 | JakA | TK | 6gl9 | A | B | (~{e})-3-[3-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)phenyl]prop-2-enenitrile | Human | 10016 | |
| JAK3 | JakA | TK | 6gl9 | B | A | (~{e})-3-[3-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)phenyl]prop-2-enenitrile | Human | 10019 | |
| JAK3 | JakA | TK | 6gl9 | B | B | (~{e})-3-[3-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)phenyl]prop-2-enenitrile | Human | 10013 | |
| JAK3 | JakA | TK | 6gla | A | A | (~{e})-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]prop-2-enenitrile | Human | 10018 | |
| JAK3 | JakA | TK | 6gla | A | B | (~{e})-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]prop-2-enenitrile | Human | 10012 | |
| JAK3 | JakA | TK | 6gla | B | A | (~{e})-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]prop-2-enenitrile | Human | 10017 | |
| JAK3 | JakA | TK | 6gla | B | B | (~{e})-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]prop-2-enenitrile | Human | 10022 | |
| JAK3 | JakA | TK | 6glb | A | A | 3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]propanenitrile | Human | 10020 | |
| JAK3 | JakA | TK | 6glb | A | B | 3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]propanenitrile | Human | 10023 | |
| JAK3 | JakA | TK | 6glb | B | A | 3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]propanenitrile | Human | 10021 | |
| JAK3 | JakA | TK | 6glb | B | B | 3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]propanenitrile | Human | 10015 | |
| JAK3 | JakA | TK | 6hzv | A | A | 3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile | Human | 11756 | |
| JAK3 | JakA | TK | 6hzv | A | B | 3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile | Human | 11751 | |
| JAK3 | JakA | TK | 6hzv | B | A | 3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile | Human | 11753 | |
| JAK3 | JakA | TK | 6hzv | B | B | 3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile | Human | 11754 | |
| JAK3 | JakA | TK | 6hzv | C | A | 3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile | Human | 11752 | |
| JAK3 | JakA | TK | 6hzv | C | B | 3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile | Human | 11755 | |
| JAK3 | JakA | TK | 6hzv | D | A | 3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile | Human | 11749 | |
| JAK3 | JakA | TK | 6hzv | D | B | 3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrile | Human | 11750 | |
| JAK3 | JakA | TK | 6ny4 | A | | 4-{[(2r,3r)-1,3-dihydroxybutan-2-yl]amino}-6-phenylpyrrolo[1,2-b]pyridazine-3-carboxamide | Human | 11052 | |
| JAK3 | JakA | TK | 7apf | A | A | 3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 13141 | |
| JAK3 | JakA | TK | 7apf | A | B | 3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 13130 | |
| JAK3 | JakA | TK | 7apf | B | A | 3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 13137 | |
| JAK3 | JakA | TK | 7apf | B | B | 3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 13132 | |
| JAK3 | JakA | TK | 7apg | A | A | ~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamide | Human | 13134 | |
| JAK3 | JakA | TK | 7apg | A | B | ~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamide | Human | 13135 | |
| JAK3 | JakA | TK | 7apg | B | A | ~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamide | Human | 13131 | |
| JAK3 | JakA | TK | 7apg | B | B | ~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamide | Human | 13136 | |
| JAK3 | JakA | TK | 7apg | C | A | ~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamide | Human | 13140 | |
| JAK3 | JakA | TK | 7apg | C | B | ~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamide | Human | 13139 | |
| JAK3 | JakA | TK | 7apg | D | A | ~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamide | Human | 13138 | |
| JAK3 | JakA | TK | 7apg | D | B | ~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamide | Human | 13133 | |
| JAK3 | JakA | TK | 7c3n | A | A | 3-[(3s,4r)-3-methyl-7-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1,7-diazaspiro[3.4]octan-1-yl]-3-oxidanylidene-propanenitrile | Human | 12389 | |
| JAK3 | JakA | TK | 7c3n | A | B | 3-[(3s,4r)-3-methyl-7-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1,7-diazaspiro[3.4]octan-1-yl]-3-oxidanylidene-propanenitrile | Human | 12391 | |
| JAK3 | JakA | TK | 7c3n | A | C | 3-[(3s,4r)-3-methyl-7-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1,7-diazaspiro[3.4]octan-1-yl]-3-oxidanylidene-propanenitrile | Human | 12390 | |
| JAK3 | JakA | TK | 7q6h | A | A | 1-[4-[[2-[(1-methylpyrazol-4-yl)amino]quinazolin-8-yl]amino]piperidin-1-yl]ethanone | Human | 14080 | |
| JAK3 | JakA | TK | 7q6h | A | B | 1-[4-[[2-[(1-methylpyrazol-4-yl)amino]quinazolin-8-yl]amino]piperidin-1-yl]ethanone | Human | 14082 | |
| JAK3 | JakA | TK | 7q6h | A | C | 1-[4-[[2-[(1-methylpyrazol-4-yl)amino]quinazolin-8-yl]amino]piperidin-1-yl]ethanone | Human | 14081 | |
| JAK3 | JakA | TK | 7uyv | A | A | 6-{[(2m)-2-(2-chloro-6-fluorophenyl)-5-oxo-5h-pyrrolo[3,4-b]pyridin-4-yl]amino}-n-ethylpyridine-3-carboxamide | Human | 14331 | |
| JAK3 | JakA | TK | 7uyv | A | B | 6-{[(2m)-2-(2-chloro-6-fluorophenyl)-5-oxo-5h-pyrrolo[3,4-b]pyridin-4-yl]amino}-n-ethylpyridine-3-carboxamide | Human | 14332 | |
| KDR | VEGFR | TK | 1vr2 | A | | - | Human | 5338 | |
| KDR | VEGFR | TK | 1y6a | A | A | n-[5-(ethylsulfonyl)-2-methoxyphenyl]-5-[3-(2-pyridinyl)phenyl]-1,3-oxazol-2-amine | Human | 5339 | |
| KDR | VEGFR | TK | 1y6a | A | B | n-[5-(ethylsulfonyl)-2-methoxyphenyl]-5-[3-(2-pyridinyl)phenyl]-1,3-oxazol-2-amine | Human | 5323 | |
| KDR | VEGFR | TK | 1y6b | A | | n-(cyclopropylmethyl)-4-(methyloxy)-3-({5-[3-(3-pyridinyl)phenyl]-1,3-oxazol-2-yl}amino)benzenesulfonamide | Human | 5345 | |
| KDR | VEGFR | TK | 1ywn | A | | n-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl]phenyl}-n'-[2-fluoro-5-(trifluoromethyl)phenyl]urea | Human | 5314 | |
| KDR | VEGFR | TK | 2oh4 | A | A | methyl (5-{4-[({[2-fluoro-5-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-1h-benzimidazol-2-yl)carbamate | Human | 5347 | |
| KDR | VEGFR | TK | 2oh4 | A | B | methyl (5-{4-[({[2-fluoro-5-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-1h-benzimidazol-2-yl)carbamate | Human | 5324 | |
| KDR | VEGFR | TK | 2p2h | A | | 4-(2-anilinopyridin-3-yl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazin-2-amine | Human | 5310 | |
| KDR | VEGFR | TK | 2p2i | A | | n-(4-phenoxyphenyl)-2-[(pyridin-4-ylmethyl)amino]nicotinamide | Human | 5326 | |
| KDR | VEGFR | TK | 2p2i | B | | n-(4-phenoxyphenyl)-2-[(pyridin-4-ylmethyl)amino]nicotinamide | Human | 5315 | |
| KDR | VEGFR | TK | 2qu5 | A | | 4-[[2-[[4-chloro-3-(trifluoromethyl)phenyl]amino]-3h-benzimidazol-5-yl]oxy]-n-methyl-pyridine-2-carboxamide | Human | 5317 | |
| KDR | VEGFR | TK | 2qu6 | A | | 4-({2-[(4-chloro-3-{[(2s)-1-methylpyrrolidin-2-yl]methoxy}phenyl)amino]-1,3-benzoxazol-5-yl}oxy)-n-methylpyridine-2-carboxamide | Human | 5316 | |
| KDR | VEGFR | TK | 2qu6 | B | | 4-({2-[(4-chloro-3-{[(2s)-1-methylpyrrolidin-2-yl]methoxy}phenyl)amino]-1,3-benzoxazol-5-yl}oxy)-n-methylpyridine-2-carboxamide | Human | 5340 | |
| KDR | VEGFR | TK | 2rl5 | A | | n-(4-chlorophenyl)-7-[(6,7-dimethoxyquinolin-4-yl)oxy]-2,3-dihydro-1,4-benzoxazine-4-carboxamide | Human | 5348 | |
| KDR | VEGFR | TK | 2xir | A | | n,2-dimethyl-6-{[7-(2-morpholin-4-ylethoxy)quinolin-4-yl]oxy}-1-benzofuran-3-carboxamide | Human | 6789 | |
| KDR | VEGFR | TK | 3b8q | A | | n-(4-chlorophenyl)-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamide | Human | 5332 | |
| KDR | VEGFR | TK | 3b8q | B | | n-(4-chlorophenyl)-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamide | Human | 5319 | |
| KDR | VEGFR | TK | 3b8r | A | | n-cyclopropyl-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamide | Human | 5327 | |
| KDR | VEGFR | TK | 3b8r | B | | n-cyclopropyl-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamide | Human | 5341 | |
| KDR | VEGFR | TK | 3be2 | A | | n-{3-[3-(dimethylamino)propyl]-5-(trifluoromethyl)phenyl}-4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]benzamide | Human | 5337 | |
| KDR | VEGFR | TK | 3c7q | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 5334 | |
| KDR | VEGFR | TK | 3cjf | A | A | n~4~-(3-methyl-1h-indazol-6-yl)-n~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamine | Human | 6792 | |
| KDR | VEGFR | TK | 3cjf | A | B | n~4~-(3-methyl-1h-indazol-6-yl)-n~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamine | Human | 6794 | |
| KDR | VEGFR | TK | 3cjg | A | A | n~4~-methyl-n~4~-(3-methyl-1h-indazol-6-yl)-n~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamine | Human | 6791 | |
| KDR | VEGFR | TK | 3cjg | A | B | n~4~-methyl-n~4~-(3-methyl-1h-indazol-6-yl)-n~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamine | Human | 6788 | |
| KDR | VEGFR | TK | 3cp9 | A | | 3-(2-aminoquinazolin-6-yl)-1-(3,3-dimethylindolin-6-yl)-4-methylpyridin-2(1h)-one | Human | 6786 | |
| KDR | VEGFR | TK | 3cp9 | B | | 3-(2-aminoquinazolin-6-yl)-1-(3,3-dimethylindolin-6-yl)-4-methylpyridin-2(1h)-one | Human | 6790 | |
| KDR | VEGFR | TK | 3cpb | A | | n'-(6-aminopyridin-3-yl)-n-(2-cyclopentylethyl)-4-methyl-benzene-1,3-dicarboxamide | Human | 6787 | |
| KDR | VEGFR | TK | 3cpb | B | | n'-(6-aminopyridin-3-yl)-n-(2-cyclopentylethyl)-4-methyl-benzene-1,3-dicarboxamide | Human | 6793 | |
| KDR | VEGFR | TK | 3cpc | A | | 3-(2-aminoquinazolin-6-yl)-4-methyl-1-[3-(trifluoromethyl)phenyl]pyridin-2(1h)-one | Human | 5346 | |
| KDR | VEGFR | TK | 3cpc | B | | 3-(2-aminoquinazolin-6-yl)-4-methyl-1-[3-(trifluoromethyl)phenyl]pyridin-2(1h)-one | Human | 5309 | |
| KDR | VEGFR | TK | 3dtw | A | | 6-chloro-n-pyrimidin-5-yl-3-{[3-(trifluoromethyl)phenyl]amino}-1,2-benzisoxazole-7-carboxamide | Human | 5313 | |
| KDR | VEGFR | TK | 3dtw | B | | 6-chloro-n-pyrimidin-5-yl-3-{[3-(trifluoromethyl)phenyl]amino}-1,2-benzisoxazole-7-carboxamide | Human | 5308 | |
| KDR | VEGFR | TK | 3efl | A | | n-(3,3-dimethyl-2,3-dihydro-1h-indol-6-yl)-2-[(pyridin-4-ylmethyl)amino]pyridine-3-carboxamide | Human | 5344 | |
| KDR | VEGFR | TK | 3efl | B | | n-(3,3-dimethyl-2,3-dihydro-1h-indol-6-yl)-2-[(pyridin-4-ylmethyl)amino]pyridine-3-carboxamide | Human | 5330 | |
| KDR | VEGFR | TK | 3ewh | A | | n-[4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)naphthalen-1-yl]-6-(trifluoromethyl)-1h-benzimidazol-2-amine | Human | 5351 | |
| KDR | VEGFR | TK | 3u6j | A | | n-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamide | Human | 5318 | |
| KDR | VEGFR | TK | 3vhe | A | | 1-{2-fluoro-4-[(5-methyl-5h-pyrrolo[3,2-d]pyrimidin-4-yl)oxy]phenyl}-3-[3-(trifluoromethyl)phenyl]urea | Human | 5331 | |
| KDR | VEGFR | TK | 3vhk | A | | {3-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methoxy]phenyl}methanol | Human | 5342 | |
| KDR | VEGFR | TK | 3vid | A | | 4,5,6,11-tetrahydro-1h-pyrazolo[4',3':6,7]cyclohepta[1,2-b]indole | Human | 5335 | |
| KDR | VEGFR | TK | 3vnt | A | A | 2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamide | Human | 5312 | |
| KDR | VEGFR | TK | 3vnt | A | B | 2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamide | Human | 5328 | |
| KDR | VEGFR | TK | 3vo3 | A | A | n-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}oxy)phenyl]-1,3-dimethyl-1h-pyrazole-5-carboxamide | Human | 5329 | |
| KDR | VEGFR | TK | 3vo3 | A | B | n-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}oxy)phenyl]-1,3-dimethyl-1h-pyrazole-5-carboxamide | Human | 5321 | |
| KDR | VEGFR | TK | 3wzd | A | A | 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide | Human | 5325 | |
| KDR | VEGFR | TK | 3wzd | A | B | 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide | Human | 5350 | |
| KDR | VEGFR | TK | 3wze | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5336 | |
| KDR | VEGFR | TK | 3wze | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5320 | |
| KDR | VEGFR | TK | 4ag8 | A | | axitinib | Human | 5311 | |
| KDR | VEGFR | TK | 4agc | A | | axitinib | Human | 5343 | |
| KDR | VEGFR | TK | 4agd | A | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 5322 | |
| KDR | VEGFR | TK | 4asd | A | | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5333 | |
| KDR | VEGFR | TK | 4ase | A | | tivozanib | Human | 5349 | |
| KDR | VEGFR | TK | 5ew3 | A | | 2-(pyridin-4-ylmethylamino)-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 6289 | |
| KDR | VEGFR | TK | 5ew3 | B | | 2-(pyridin-4-ylmethylamino)-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 6290 | |
| KDR | VEGFR | TK | 6gqo | A | A | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10580 | |
| KDR | VEGFR | TK | 6gqo | A | B | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10583 | |
| KDR | VEGFR | TK | 6gqp | A | A | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10582 | |
| KDR | VEGFR | TK | 6gqp | A | B | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10584 | |
| KDR | VEGFR | TK | 6gqq | A | A | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10581 | |
| KDR | VEGFR | TK | 6gqq | A | B | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10585 | |
| KDR | VEGFR | TK | 6xvj | A | | ~{n}-[3-[(dimethylamino)methyl]-5-methyl-phenyl]-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12274 | |
| KDR | VEGFR | TK | 6xvk | A | | ~{n}-(4,4-dimethyl-2-prop-1-ynyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12273 | |
| KIT | PDGFR | TK | 1pkg | A | | adenosine-5'-diphosphate | Human | 397 | |
| KIT | PDGFR | TK | 1pkg | B | | adenosine-5'-diphosphate | Human | 402 | |
| KIT | PDGFR | TK | 1t45 | A | A | - | Human | 399 | |
| KIT | PDGFR | TK | 1t45 | A | B | - | Human | 394 | |
| KIT | PDGFR | TK | 1t46 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 393 | |
| KIT | PDGFR | TK | 1t46 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 404 | |
| KIT | PDGFR | TK | 3g0e | A | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 401 | |
| KIT | PDGFR | TK | 3g0e | A | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 398 | |
| KIT | PDGFR | TK | 3g0f | A | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 395 | |
| KIT | PDGFR | TK | 3g0f | B | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 400 | |
| KIT | PDGFR | TK | 4hvs | A | | 5-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-n-[4-(trifluoromethyl)benzyl]pyridin-2-amine | Human | 403 | |
| KIT | PDGFR | TK | 4u0i | A | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 405 | |
| KIT | PDGFR | TK | 4u0i | A | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 396 | |
| KIT | PDGFR | TK | 6gqj | A | A | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10364 | |
| KIT | PDGFR | TK | 6gqj | A | B | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10354 | |
| KIT | PDGFR | TK | 6gqj | B | A | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10358 | |
| KIT | PDGFR | TK | 6gqj | B | B | 2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamide | Human | 10356 | |
| KIT | PDGFR | TK | 6gqk | A | A | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10355 | |
| KIT | PDGFR | TK | 6gqk | A | B | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10353 | |
| KIT | PDGFR | TK | 6gqk | B | A | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10363 | |
| KIT | PDGFR | TK | 6gqk | B | B | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamide | Human | 10360 | |
| KIT | PDGFR | TK | 6gql | A | | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10362 | |
| KIT | PDGFR | TK | 6gql | B | | ~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10357 | |
| KIT | PDGFR | TK | 6gqm | A | | ~{n}-[4-[[5-fluoranyl-7-(2-methoxyethoxy)quinazolin-4-yl]amino]phenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10359 | |
| KIT | PDGFR | TK | 6gqm | B | | ~{n}-[4-[[5-fluoranyl-7-(2-methoxyethoxy)quinazolin-4-yl]amino]phenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamide | Human | 10361 | |
| KIT | PDGFR | TK | 6hh1 | A | A | ~{n}-(2,3-dimethylphenyl)-5-(4-pyridin-4-yloxyphenyl)-4~{h}-1,2,4-triazol-3-amine | Human | 11629 | |
| KIT | PDGFR | TK | 6hh1 | A | B | ~{n}-(2,3-dimethylphenyl)-5-(4-pyridin-4-yloxyphenyl)-4~{h}-1,2,4-triazol-3-amine | Human | 11628 | |
| KIT | PDGFR | TK | 6itt | A | A | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11826 | |
| KIT | PDGFR | TK | 6itt | A | B | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11824 | |
| KIT | PDGFR | TK | 6itt | B | A | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11821 | |
| KIT | PDGFR | TK | 6itt | B | B | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11820 | |
| KIT | PDGFR | TK | 6itv | A | A | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11822 | |
| KIT | PDGFR | TK | 6itv | A | B | n-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]urea | Human | 11827 | |
| KIT | PDGFR | TK | 6kla | A | A | n-[6-(4-ethylpiperazin-1-yl)-2-methyl-pyrimidin-4-yl]-5-pyridin-4-yl-1,3-thiazol-2-amine | Human | 11825 | |
| KIT | PDGFR | TK | 6kla | A | B | n-[6-(4-ethylpiperazin-1-yl)-2-methyl-pyrimidin-4-yl]-5-pyridin-4-yl-1,3-thiazol-2-amine | Human | 11823 | |
| KIT | PDGFR | TK | 6mob | A | A | n-{4-chloro-5-[1-ethyl-7-(methylamino)-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl]-2-fluorophenyl}-n'-phenylurea | Human | 11469 | |
| KIT | PDGFR | TK | 6mob | A | B | n-{4-chloro-5-[1-ethyl-7-(methylamino)-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl]-2-fluorophenyl}-n'-phenylurea | Human | 11470 | |
| KIT | PDGFR | TK | 6xv9 | A | | ~{n}-[3-[(dimethylamino)methyl]-5-methyl-phenyl]-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12282 | |
| KIT | PDGFR | TK | 6xv9 | B | | ~{n}-[3-[(dimethylamino)methyl]-5-methyl-phenyl]-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12283 | |
| KIT | PDGFR | TK | 6xva | A | | ~{n}-[[3-[2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanoylamino]-5-methyl-phenyl]methyl]propanamide | Human | 12284 | |
| KIT | PDGFR | TK | 6xva | B | | ~{n}-[[3-[2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanoylamino]-5-methyl-phenyl]methyl]propanamide | Human | 12281 | |
| KIT | PDGFR | TK | 6xvb | A | | ~{n}-(4,4-dimethyl-2-propyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12279 | |
| KIT | PDGFR | TK | 6xvb | B | | ~{n}-(4,4-dimethyl-2-propyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamide | Human | 12280 | |
| KIT | PDGFR | TK | 7khg | A | A | 5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amine | Human | 13786 | |
| KIT | PDGFR | TK | 7khg | A | B | 5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amine | Human | 13788 | |
| KIT | PDGFR | TK | 7khj | A | | 2-phenyl-5-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 13789 | |
| KIT | PDGFR | TK | 7khk | A | | 4,5-dimethyl-n-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazole-3-carboxamide | Human | 13787 | |
| KIT | PDGFR | TK | 7zw8 | A | A | ~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amine | Human | 14622 | |
| KIT | PDGFR | TK | 7zw8 | A | B | ~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amine | Human | 14624 | |
| KIT | PDGFR | TK | 7zy6 | A | | 5-imidazo[1,2-a]pyridin-3-yl-~{n}-[(1~{r})-1-(6-pyrrolidin-1-ylpyridin-3-yl)ethyl]pyridin-3-amine | Human | 14623 | |
| KIT | PDGFR | TK | 8dfm | A | | - | Human | 14677 | |
| KIT | PDGFR | TK | 8dfp | A | | - | Human | 14678 | |
| KIT | PDGFR | TK | 8dfq | A | | - | Human | 14679 | |
| KIT | PDGFR | TK | 8pq9 | A | A | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15118 | |
| KIT | PDGFR | TK | 8pq9 | A | B | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15125 | |
| KIT | PDGFR | TK | 8pqa | A | A | 6-(1-methylpyrazol-4-yl)-4-(4-pyrimidin-2-ylpiperazin-1-yl)pyrrolo[2,1-f][1,2,4]triazine | Human | 15124 | |
| KIT | PDGFR | TK | 8pqa | A | B | 6-(1-methylpyrazol-4-yl)-4-(4-pyrimidin-2-ylpiperazin-1-yl)pyrrolo[2,1-f][1,2,4]triazine | Human | 15115 | |
| KIT | PDGFR | TK | 8pqb | A | A | (1~{s})-1-(4-fluorophenyl)-~{n},~{n}-dimethyl-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15121 | |
| KIT | PDGFR | TK | 8pqb | A | B | (1~{s})-1-(4-fluorophenyl)-~{n},~{n}-dimethyl-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15120 | |
| KIT | PDGFR | TK | 8pqc | A | A | (1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15122 | |
| KIT | PDGFR | TK | 8pqc | A | B | (1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15123 | |
| KIT | PDGFR | TK | 8pqd | A | A | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]ethanamide | Human | 15113 | |
| KIT | PDGFR | TK | 8pqd | A | B | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]ethanamide | Human | 15126 | |
| KIT | PDGFR | TK | 8pqe | A | A | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]prop-2-enamide | Human | 15119 | |
| KIT | PDGFR | TK | 8pqe | A | B | ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]prop-2-enamide | Human | 15117 | |
| KIT | PDGFR | TK | 8pqf | A | A | methyl ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]carbamate | Human | 15116 | |
| KIT | PDGFR | TK | 8pqf | A | B | methyl ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]carbamate | Human | 15127 | |
| KIT | PDGFR | TK | 8pqg | A | A | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15114 | |
| KIT | PDGFR | TK | 8pqg | A | B | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15112 | |
| KSR1 | RAF | TKL | 7juw | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12855 | |
| KSR1 | RAF | TKL | 7jux | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14018 | |
| KSR1 | RAF | TKL | 7juy | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12920 | |
| KSR1 | RAF | TKL | 7juz | A | | - | Human | 12856 | |
| KSR1 | RAF | TKL | 7juz | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12851 | |
| KSR1 | RAF | TKL | 7jv0 | A | | - | Human | 12848 | |
| KSR1 | RAF | TKL | 7jv0 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12853 | |
| KSR1 | RAF | TKL | 7jv1 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12854 | |
| KSR1 | RAF | TKL | 7jv1 | D | | - | Human | 12849 | |
| KSR2 | RAF | TKL | 2y4i | B | | adenosine-5'-triphosphate | Human | 1244 | |
| KSR2 | RAF | TKL | 5kkr | B | | 6,7-dimethoxy-~{n}-(2-methyl-4-phenoxy-phenyl)quinazolin-4-amine | Human | 7027 | |
| KSR2 | RAF | TKL | 7juq | B | | adenosine-5'-diphosphate | Human | 12821 | |
| KSR2 | RAF | TKL | 7jur | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12822 | |
| KSR2 | RAF | TKL | 7jus | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12823 | |
| KSR2 | RAF | TKL | 7jut | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12818 | |
| KSR2 | RAF | TKL | 7juu | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12820 | |
| KSR2 | RAF | TKL | 7juv | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12819 | |
| LCK | Src | TK | 1qpc | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2291 | |
| LCK | Src | TK | 1qpd | A | | staurosporine | Human | 2267 | |
| LCK | Src | TK | 1qpe | A | | 1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 2271 | |
| LCK | Src | TK | 1qpj | A | | staurosporine | Human | 2283 | |
| LCK | Src | TK | 2of2 | A | | 2,3-diphenyl-n-(2-piperazin-1-ylethyl)furo[2,3-b]pyridin-4-amine | Human | 2261 | |
| LCK | Src | TK | 2of4 | A | | 5,6-diphenyl-n-(2-piperazin-1-ylethyl)furo[2,3-d]pyrimidin-4-amine | Human | 2296 | |
| LCK | Src | TK | 2ofu | A | | 2,6-dimethylphenyl 2-(3,5-dimethoxy-4-(3-(4-methylpiperazin-1-yl)propoxy)phenylamino)pyrimidin- 4-yl(2,4-dimethoxyphenyl)carbamate | Human | 2259 | |
| LCK | Src | TK | 2ofv | A | | 3-(2-aminoquinazolin-6-yl)-4-methyl-n-[3-(trifluoromethyl)phenyl]benzamide | Human | 2280 | |
| LCK | Src | TK | 2ofv | B | | 3-(2-aminoquinazolin-6-yl)-4-methyl-n-[3-(trifluoromethyl)phenyl]benzamide | Human | 2294 | |
| LCK | Src | TK | 2og8 | A | | n-{2-[(n,n-diethylglycyl)amino]-5-(trifluoromethyl)phenyl}-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamide | Human | 2286 | |
| LCK | Src | TK | 2og8 | B | | n-{2-[(n,n-diethylglycyl)amino]-5-(trifluoromethyl)phenyl}-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamide | Human | 2282 | |
| LCK | Src | TK | 2pl0 | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 2290 | |
| LCK | Src | TK | 2zm1 | A | | n-(2-chlorophenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine | Human | 2273 | |
| LCK | Src | TK | 2zm4 | A | | n-(2-chloro-6-methylphenyl)-8-[(3s)-3-methylpiperazin-1-yl]imidazo[1,5-a]quinoxalin-4-amine | Human | 2262 | |
| LCK | Src | TK | 2zyb | A | | n-(2,6-dimethylphenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine | Human | 2275 | |
| LCK | Src | TK | 3ac1 | A | | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-3-[(3,5-dimethoxyphenyl)amino]pyrazine-2-carboxamide | Human | 2287 | |
| LCK | Src | TK | 3ac2 | A | | 7-[(2-amino-2-methylpropyl)amino]-2-[(3,5-dimethoxyphenyl)amino]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2266 | |
| LCK | Src | TK | 3ac3 | A | | 2-[(3,5-dimethoxyphenyl)amino]-5-ethyl-7-[(2r)-2-(hydroxymethyl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2292 | |
| LCK | Src | TK | 3ac4 | A | | 5-[(2-amino-1,1-dimethylethyl)amino]-7-[(3,5-dimethoxyphenyl)amino][1,2,4]triazolo[4,3-c]pyrimidine-8-carboxamide | Human | 2278 | |
| LCK | Src | TK | 3ac5 | A | | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-7-[(3,5-dimethoxyphenyl)amino]-2-(3-hydroxyphenyl)[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxamide | Human | 2277 | |
| LCK | Src | TK | 3ac8 | A | | 7-[(2-amino-2-methylpropyl)amino]-5-cyclopropyl-2-[(3,5-dimethoxyphenyl)amino]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2300 | |
| LCK | Src | TK | 3acj | A | | 7-(3,4-dimethoxyphenyl)-5-(ethylsulfanyl)imidazo[1,2-c]pyrimidine | Human | 2260 | |
| LCK | Src | TK | 3ack | A | | 6-(5-methoxy-1-methyl-1h-indol-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 2284 | |
| LCK | Src | TK | 3ad4 | A | | (4-chlorophenyl)(5-methoxy-1-benzofuran-2-yl)methanone | Human | 2268 | |
| LCK | Src | TK | 3ad5 | A | | 4-[4-(benzyloxy)phenyl]-5-{[2-(4-chlorophenyl)-2-oxoethyl]sulfanyl}-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 2270 | |
| LCK | Src | TK | 3ad6 | A | | 7-[(cyclopropylmethyl)amino]-2-[(4-methoxyphenyl)amino]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2274 | |
| LCK | Src | TK | 3b2w | A | | n-[5-({[2-fluoro-3-(trifluoromethyl)phenyl]amino}carbonyl)-2-methylphenyl]-4-methoxy-2-[(4-piperazin-1-ylphenyl)amino]pyrimidine-5-carboxamide | Human | 2299 | |
| LCK | Src | TK | 3bym | A | | n-phenyl-1-{4-[(3,4,5-trimethoxyphenyl)amino]-1,3,5-triazin-2-yl}-1h-benzimidazol-2-amine | Human | 2264 | |
| LCK | Src | TK | 3byo | A | | 6-(2,6-dimethylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimido[5',4':5,6]pyrimido[1,2-a]benzimidazol-5(6h)-one | Human | 2272 | |
| LCK | Src | TK | 3bys | A | | 4-methyl-n~3~-(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-5-yl)-n~1~-[3-(trifluoromethyl)phenyl]benzene-1,3-dicarboxamide | Human | 2293 | |
| LCK | Src | TK | 3byu | A | | 2-methyl-n-{4-methyl-3-[(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-5-yl)carbamoyl]phenyl}-3-(trifluoromethyl)benzamide | Human | 2288 | |
| LCK | Src | TK | 3kmm | A | | 3-(2,6-dichlorophenyl)-7-({4-[2-(diethylamino)ethoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 2265 | |
| LCK | Src | TK | 3kxz | A | | 3-[7-[(3-hydroxyphenyl)amino]pyrazolo[1,5-a]pyrimidin-2-yl]-n-(1-hydroxy-2,2,6,6-tetramethyl-piperidin-4-yl)benzamide | Human | 2281 | |
| LCK | Src | TK | 3lck | A | A | - | Human | 2263 | |
| LCK | Src | TK | 3lck | A | B | - | Human | 2301 | |
| LCK | Src | TK | 3mpm | A | A | 4-{(6r,7r)-7-amino-3-[3-(4-methylpiperazin-1-yl)phenyl]-6,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl}phenol | Human | 2279 | |
| LCK | Src | TK | 3mpm | A | B | 4-{(6r,7r)-7-amino-3-[3-(4-methylpiperazin-1-yl)phenyl]-6,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl}phenol | Human | 2295 | |
| LCK | Src | TK | 4c3f | A | A | n-phenyl-4-(5-phenyl-1h-pyrazol-4-yl)pyrimidin-2-amine | Human | 2276 | |
| LCK | Src | TK | 4c3f | A | B | n-phenyl-4-(5-phenyl-1h-pyrazol-4-yl)pyrimidin-2-amine | Human | 2297 | |
| LCK | Src | TK | 6pdj | A | A | n-{4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]-3-methylphenyl}-1-methyl-1h-indazole-3-carboxamide | Human | 11698 | |
| LCK | Src | TK | 6pdj | A | B | n-{4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]-3-methylphenyl}-1-methyl-1h-indazole-3-carboxamide | Human | 11699 | |
| LIMK1 | LISK | TKL | 3s95 | A | A | staurosporine | Human | 1246 | |
| LIMK1 | LISK | TKL | 3s95 | A | B | staurosporine | Human | 1248 | |
| LIMK1 | LISK | TKL | 3s95 | B | A | staurosporine | Human | 1245 | |
| LIMK1 | LISK | TKL | 3s95 | B | B | staurosporine | Human | 1247 | |
| LIMK1 | LISK | TKL | 5hvj | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 6599 | |
| LIMK1 | LISK | TKL | 5hvj | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 6598 | |
| LIMK1 | LISK | TKL | 5hvj | B | A | - | Human | 6597 | |
| LIMK1 | LISK | TKL | 5hvj | B | B | - | Human | 6595 | |
| LIMK1 | LISK | TKL | 5hvk | A | | phosphoaminophosphonic acid-adenylate ester | Human | 6600 | |
| LIMK1 | LISK | TKL | 5hvk | C | | phosphoaminophosphonic acid-adenylate ester | Human | 6596 | |
| LIMK1 | LISK | TKL | 5l6w | L | | phosphothiophosphoric acid-adenylate ester | Human | 6668 | |
| LIMK1 | LISK | TKL | 5nxc | L | | (2~{r})-2-azanyl-2-cyclohexyl-~{n}-[2-(1-methylpyrazol-4-yl)-9-oxidanylidene-3,10,11-triazatricyclo[6.4.1.0^{4,13}]trideca-1,4,6,8(13),11-pentaen-6-yl]ethanamide | Human | 7592 | |
| LIMK1 | LISK | TKL | 7ats | A | | n-[3-[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]benzenesulfonamide | Human | 13164 | |
| LIMK1 | LISK | TKL | 7atu | A | | (s)-2-benzyl-6-(8-chloro-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-7-oxo-4,5,6,7-tetrahydro-2h-pyrazolo[3,4-c]pyridine-3-carboxamide | Human | 14019 | |
| LIMK1 | LISK | TKL | 7b8w | A | | 2-(2-methylpropanoylamino)-~{n}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamide | Human | 14126 | |
| LIMK1 | LISK | TKL | 8aau | L | A | ~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamide | Human | 14555 | |
| LIMK1 | LISK | TKL | 8aau | L | B | ~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamide | Human | 14554 | |
| LIMK2 | LISK | TKL | 4tpt | A | | n-{4-[(1s)-1,2-dihydroxyethyl]benzyl}-n-methyl-4-(phenylsulfamoyl)benzamide | Human | 2476 | |
| LIMK2 | LISK | TKL | 4tpt | B | | n-{4-[(1s)-1,2-dihydroxyethyl]benzyl}-n-methyl-4-(phenylsulfamoyl)benzamide | Human | 2475 | |
| LIMK2 | LISK | TKL | 5nxd | A | A | 4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamide | Human | 7623 | |
| LIMK2 | LISK | TKL | 5nxd | A | B | 4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamide | Human | 7621 | |
| LIMK2 | LISK | TKL | 5nxd | B | A | 4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamide | Human | 7624 | |
| LIMK2 | LISK | TKL | 5nxd | B | B | 4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamide | Human | 7622 | |
| LIMK2 | LISK | TKL | 7qhg | A | A | 2-(2-methylpropanoylamino)-~{n}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamide | Human | 14021 | |
| LIMK2 | LISK | TKL | 7qhg | A | B | 2-(2-methylpropanoylamino)-~{n}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamide | Human | 14020 | |
| LIMK2 | LISK | TKL | 8wsw | A | A | ~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamide | Human | 14862 | |
| LIMK2 | LISK | TKL | 8wsw | A | B | ~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamide | Human | 14861 | |
| LMTK3 (LMR3) | Lmr | TK | 6seq | A | A | - | Human | 12994 | |
| LMTK3 (LMR3) | Lmr | TK | 6seq | A | B | - | Human | 12995 | |
| LRRK1 | LRRK | TKL | 8e04 | A | | - | Human | 14879 | |
| LRRK1 | LRRK | TKL | 8e05 | A | | - | Human | 14882 | |
| LRRK1 | LRRK | TKL | 8e06 | A | | - | Human | 14881 | |
| LRRK1 | LRRK | TKL | 8fac | A | | - | Human | 14880 | |
| LRRK2 | LRRK | TKL | 6vno | A | 1 | - | Human | 12735 | |
| LRRK2 | LRRK | TKL | 6vno | A | 10 | - | Human | 12717 | |
| LRRK2 | LRRK | TKL | 6vno | A | 2 | - | Human | 12725 | |
| LRRK2 | LRRK | TKL | 6vno | A | 3 | - | Human | 12731 | |
| LRRK2 | LRRK | TKL | 6vno | A | 4 | - | Human | 12719 | |
| LRRK2 | LRRK | TKL | 6vno | A | 5 | - | Human | 12715 | |
| LRRK2 | LRRK | TKL | 6vno | A | 6 | - | Human | 12732 | |
| LRRK2 | LRRK | TKL | 6vno | A | 7 | - | Human | 12712 | |
| LRRK2 | LRRK | TKL | 6vno | A | 8 | - | Human | 12718 | |
| LRRK2 | LRRK | TKL | 6vno | A | 9 | - | Human | 12728 | |
| LRRK2 | LRRK | TKL | 6vp6 | A | | - | Human | 12714 | |
| LRRK2 | LRRK | TKL | 6vp6 | B | | - | Human | 12726 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 1 | - | Human | 12713 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 10 | - | Human | 12730 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 2 | - | Human | 12724 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 3 | - | Human | 12733 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 4 | - | Human | 12720 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 5 | - | Human | 12716 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 6 | - | Human | 12721 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 7 | - | Human | 12727 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 8 | - | Human | 12722 | |
| LRRK2 | LRRK | TKL | 6vp7 | A | 9 | - | Human | 12729 | |
| LRRK2 | LRRK | TKL | 6vp8 | A | | - | Human | 12723 | |
| LRRK2 | LRRK | TKL | 6vp8 | B | | - | Human | 12734 | |
| LRRK2 | LRRK | TKL | 7lht | A | | - | Human | 13623 | |
| LRRK2 | LRRK | TKL | 7lhw | A | | - | Human | 13625 | |
| LRRK2 | LRRK | TKL | 7li3 | A | | - | Human | 13626 | |
| LRRK2 | LRRK | TKL | 7li4 | A | | - | Human | 13624 | |
| LRRK2 | LRRK | TKL | 8fo8 | C | | - | Human | 15133 | |
| LRRK2 | LRRK | TKL | 8fo9 | A | | - | Human | 15132 | |
| LRRK2 | LRRK | TKL | 8txz | A | A | - | Human | 15056 | |
| LRRK2 | LRRK | TKL | 8txz | A | B | - | Human | 15057 | |
| LRRK2 | LRRK | TKL | 8tyq | A | A | 4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-3-[(1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]benzamide | Human | 15058 | |
| LRRK2 | LRRK | TKL | 8tyq | A | B | 4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-3-[(1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]benzamide | Human | 15055 | |
| LRRK2 | LRRK | TKL | 8tzb | A | | - | Human | 15052 | |
| LRRK2 | LRRK | TKL | 8tzc | A | | - | Human | 15050 | |
| LRRK2 | LRRK | TKL | 8tze | A | | 4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-3-[(1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]benzamide | Human | 15054 | |
| LRRK2 | LRRK | TKL | 8tzf | A | | - | Human | 15059 | |
| LRRK2 | LRRK | TKL | 8tzg | A | A | - | Human | 15051 | |
| LRRK2 | LRRK | TKL | 8tzg | A | B | - | Human | 15053 | |
| LRRK2 | LRRK | TKL | 8u1b | A | | - | Human | 15387 | |
| LRRK2 | LRRK | TKL | 8u7l | A | | - | Human | 15184 | |
| LRRK2 | LRRK | TKL | 8u8b | A | | - | Human | 15185 | |
| Lyn (LYN) | Src | TK | 2zv7 | A | | - | Mouse | 5771 | |
| Lyn (LYN) | Src | TK | 2zv8 | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5772 | |
| Lyn (LYN) | Src | TK | 2zv9 | A | | 1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Mouse | 5773 | |
| Lyn (LYN) | Src | TK | 2zva | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5774 | |
| LYN | Src | TK | 3a4o | X | | staurosporine | Human | 1812 | |
| LYN | Src | TK | 5xy1 | A | | n-(1h-indazol-6-yl)-8-piperidin-4-yloxy-6-propyl-quinazolin-2-amine | Human | 8271 | |
| MAP2K1 | STE7 | STE | 1s9j | A | | adenosine-5'-triphosphate | Human | 3316 | |
| MAP2K1 | STE7 | STE | 2p55 | A | | 2-[(4-ethynyl-2-fluorophenyl)amino]-3,4-difluoro-n-(2-hydroxyethoxy)benzamide | Human | 3327 | |
| MAP2K1 | STE7 | STE | 3dv3 | A | A | adenosine-5'-triphosphate | Human | 3322 | |
| MAP2K1 | STE7 | STE | 3dv3 | A | B | adenosine-5'-triphosphate | Human | 3311 | |
| MAP2K1 | STE7 | STE | 3dy7 | A | | adenosine-5'-triphosphate | Human | 3282 | |
| MAP2K1 | STE7 | STE | 3e8n | A | | adenosine-5'-triphosphate | Human | 3323 | |
| MAP2K1 | STE7 | STE | 3eqb | A | A | adenosine-5'-triphosphate | Human | 3324 | |
| MAP2K1 | STE7 | STE | 3eqb | A | B | adenosine-5'-triphosphate | Human | 3310 | |
| MAP2K1 | STE7 | STE | 3eqc | A | A | 2-[(2-chloro-4-iodophenyl)amino]-n-{[(2r)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamide | Human | 3280 | |
| MAP2K1 | STE7 | STE | 3eqc | A | B | 2-[(2-chloro-4-iodophenyl)amino]-n-{[(2r)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamide | Human | 3300 | |
| MAP2K1 | STE7 | STE | 3eqd | A | | phosphothiophosphoric acid-adenylate ester | Human | 3284 | |
| MAP2K1 | STE7 | STE | 3eqf | A | | k-252a | Human | 3317 | |
| MAP2K1 | STE7 | STE | 3eqg | A | | adenosine-5'-diphosphate | Human | 3304 | |
| MAP2K1 | STE7 | STE | 3eqh | A | | (2z)-bis{amino[(2-aminophenyl)sulfanyl]methylidene}butanedinitrile | Human | 3290 | |
| MAP2K1 | STE7 | STE | 3eqi | A | | adenosine-5'-diphosphate | Human | 3308 | |
| MAP2K1 | STE7 | STE | 3mbl | A | A | adenosine-5'-diphosphate | Human | 3292 | |
| MAP2K1 | STE7 | STE | 3mbl | A | B | adenosine-5'-diphosphate | Human | 3318 | |
| MAP2K1 | STE7 | STE | 3orn | A | | phosphoaminophosphonic acid-adenylate ester | Human | 3277 | |
| MAP2K1 | STE7 | STE | 3os3 | A | | adenosine-5'-triphosphate | Human | 3281 | |
| MAP2K1 | STE7 | STE | 3pp1 | A | A | adenosine-5'-triphosphate | Human | 3294 | |
| MAP2K1 | STE7 | STE | 3pp1 | A | B | adenosine-5'-triphosphate | Human | 3285 | |
| MAP2K1 | STE7 | STE | 3sls | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 9486 | |
| MAP2K1 | STE7 | STE | 3sls | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 9485 | |
| MAP2K1 | STE7 | STE | 3sls | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 9487 | |
| MAP2K1 | STE7 | STE | 3sls | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 9484 | |
| MAP2K1 | STE7 | STE | 3v01 | A | | n-{[(2r)-2,3-dihydroxypropyl]oxy}-3-[(2-fluoro-4-iodophenyl)amino]furo[3,2-c]pyridine-2-carboxamide | Human | 3291 | |
| MAP2K1 | STE7 | STE | 3v04 | A | | 4-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)-1h-indazole-5-carboxamide | Human | 3325 | |
| MAP2K1 | STE7 | STE | 3vvh | A | A | adenosine-5'-triphosphate | Human | 3288 | |
| MAP2K1 | STE7 | STE | 3vvh | A | B | adenosine-5'-triphosphate | Human | 3296 | |
| MAP2K1 | STE7 | STE | 3vvh | B | A | adenosine-5'-triphosphate | Human | 3321 | |
| MAP2K1 | STE7 | STE | 3vvh | B | B | adenosine-5'-triphosphate | Human | 3289 | |
| MAP2K1 | STE7 | STE | 3vvh | C | A | adenosine-5'-triphosphate | Human | 3306 | |
| MAP2K1 | STE7 | STE | 3vvh | C | B | adenosine-5'-triphosphate | Human | 3287 | |
| MAP2K1 | STE7 | STE | 3w8q | A | | phosphothiophosphoric acid-adenylate ester | Human | 3298 | |
| MAP2K1 | STE7 | STE | 3wig | A | | phosphoaminophosphonic acid-adenylate ester | Human | 3329 | |
| MAP2K1 | STE7 | STE | 3zls | A | | 1h-pyrrolo[2,3-b]pyridine-3-carboxylic acid | Human | 3279 | |
| MAP2K1 | STE7 | STE | 3zlw | A | | (1r)-1-hydroxy-1-methyl-2,3,6,7-tetrahydro-1h,5h-pyrido[3,2,1-ij]quinolin-5-one | Human | 3278 | |
| MAP2K1 | STE7 | STE | 3zlx | A | | 7-choro-6-[(3r)-pyrrolidin-3-ylmethoxy]isoquinolin-1(2h)-one | Human | 3312 | |
| MAP2K1 | STE7 | STE | 3zly | A | | 3-amino-1h-indazole-4-carbonitrile | Human | 3320 | |
| MAP2K1 | STE7 | STE | 3zm4 | A | | 7-chloranyl-6-[(3s)-pyrrolidin-3-yl]oxy-2h-isoquinolin-1-one | Human | 3303 | |
| MAP2K1 | STE7 | STE | 4an2 | A | A | [3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]-[3-oxidanyl-3-[(2s)-piperidin-2-yl]azetidin-1-yl]methanone | Human | 3309 | |
| MAP2K1 | STE7 | STE | 4an2 | A | B | [3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]-[3-oxidanyl-3-[(2s)-piperidin-2-yl]azetidin-1-yl]methanone | Human | 3326 | |
| MAP2K1 | STE7 | STE | 4an3 | A | | adenosine-5'-triphosphate | Human | 3295 | |
| MAP2K1 | STE7 | STE | 4an9 | A | | phosphomethylphosphonic acid adenylate ester | Human | 3330 | |
| MAP2K1 | STE7 | STE | 4anb | A | | [3-(aminomethyl)-3-oxidanyl-azetidin-1-yl]-[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]methanone | Human | 3302 | |
| MAP2K1 | STE7 | STE | 4ark | A | | adenosine-5'-diphosphate | Human | 3299 | |
| MAP2K1 | STE7 | STE | 4lmn | A | | phosphoaminophosphonic acid-adenylate ester | Human | 3283 | |
| MAP2K1 | STE7 | STE | 4mne | A | A | phosphomethylphosphonic acid adenylate ester | Human | 3293 | |
| MAP2K1 | STE7 | STE | 4mne | A | B | phosphomethylphosphonic acid adenylate ester | Human | 3307 | |
| MAP2K1 | STE7 | STE | 4mne | D | A | phosphomethylphosphonic acid adenylate ester | Human | 3313 | |
| MAP2K1 | STE7 | STE | 4mne | D | B | phosphomethylphosphonic acid adenylate ester | Human | 3315 | |
| MAP2K1 | STE7 | STE | 4mne | E | A | phosphomethylphosphonic acid adenylate ester | Human | 3314 | |
| MAP2K1 | STE7 | STE | 4mne | E | B | phosphomethylphosphonic acid adenylate ester | Human | 3286 | |
| MAP2K1 | STE7 | STE | 4mne | H | A | phosphomethylphosphonic acid adenylate ester | Human | 3319 | |
| MAP2K1 | STE7 | STE | 4mne | H | B | phosphomethylphosphonic acid adenylate ester | Human | 3328 | |
| MAP2K1 | STE7 | STE | 4u7z | A | | 5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamide | Human | 3297 | |
| MAP2K1 | STE7 | STE | 4u80 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 3305 | |
| MAP2K1 | STE7 | STE | 4u81 | A | | 8-[(4-cyclopropyl-2-fluorophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-7-carboxamide | Human | 3301 | |
| MAP2K1 | STE7 | STE | 5bx0 | A | | ethyl 2h-indazole-5-carboxylate | Human | 6300 | |
| MAP2K1 | STE7 | STE | 5eym | A | A | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 6966 | |
| MAP2K1 | STE7 | STE | 5eym | A | B | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 6969 | |
| MAP2K1 | STE7 | STE | 5eym | B | A | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 6968 | |
| MAP2K1 | STE7 | STE | 5eym | B | B | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 6967 | |
| MAP2K1 | STE7 | STE | 5hze | A | A | (3s,4r,8s,9s,11e)-8,9,16-trihydroxy-3,4-dimethyl-14-(methylamino)-3,4,5,6,9,10-hexahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 7569 | |
| MAP2K1 | STE7 | STE | 5hze | A | B | (3s,4r,8s,9s,11e)-8,9,16-trihydroxy-3,4-dimethyl-14-(methylamino)-3,4,5,6,9,10-hexahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 7570 | |
| MAP2K1 | STE7 | STE | 5yt3 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 10692 | |
| MAP2K1 | STE7 | STE | 5yt3 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 10694 | |
| MAP2K1 | STE7 | STE | 5yt3 | C | | phosphoaminophosphonic acid-adenylate ester | Human | 10693 | |
| MAP2K1 | STE7 | STE | 5yt3 | D | | phosphoaminophosphonic acid-adenylate ester | Human | 10695 | |
| MAP2K1 | STE7 | STE | 6nyb | B | | adenosine-5'-diphosphate | Human | 11719 | |
| MAP2K1 | STE7 | STE | 6pp9 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 11716 | |
| MAP2K1 | STE7 | STE | 6pp9 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 11720 | |
| MAP2K1 | STE7 | STE | 6q0j | C | A | 5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamide | Human | 11721 | |
| MAP2K1 | STE7 | STE | 6q0j | C | B | 5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamide | Human | 11713 | |
| MAP2K1 | STE7 | STE | 6q0j | D | A | 5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamide | Human | 11714 | |
| MAP2K1 | STE7 | STE | 6q0j | D | B | 5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamide | Human | 11718 | |
| MAP2K1 | STE7 | STE | 6q0t | C | A | 5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamide | Human | 11715 | |
| MAP2K1 | STE7 | STE | 6q0t | C | B | 5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamide | Human | 11717 | |
| MAP2K1 | STE7 | STE | 6u2g | A | | phosphomethylphosphonic acid adenylate ester | Human | 11574 | |
| MAP2K1 | STE7 | STE | 6v2w | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 13015 | |
| MAP2K1 | STE7 | STE | 6v2w | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 13017 | |
| MAP2K1 | STE7 | STE | 7b3m | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13365 | |
| MAP2K1 | STE7 | STE | 7b3m | B | | phosphoaminophosphonic acid-adenylate ester | Human | 13363 | |
| MAP2K1 | STE7 | STE | 7b7r | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13397 | |
| MAP2K1 | STE7 | STE | 7b7r | B | | phosphoaminophosphonic acid-adenylate ester | Human | 13400 | |
| MAP2K1 | STE7 | STE | 7b94 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 13364 | |
| MAP2K1 | STE7 | STE | 7b9l | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 13402 | |
| MAP2K1 | STE7 | STE | 7b9l | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 13401 | |
| MAP2K1 | STE7 | STE | 7b9l | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 13398 | |
| MAP2K1 | STE7 | STE | 7b9l | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 13399 | |
| MAP2K1 | STE7 | STE | 7f2x | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14243 | |
| MAP2K1 | STE7 | STE | 7m0t | B | | 5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamide | Human | 13512 | |
| MAP2K1 | STE7 | STE | 7m0u | B | | 5-[(4-bromo-2-fluorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamide | Human | 13517 | |
| MAP2K1 | STE7 | STE | 7m0v | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 13518 | |
| MAP2K1 | STE7 | STE | 7m0v | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 13511 | |
| MAP2K1 | STE7 | STE | 7m0w | B | | phosphoaminophosphonic acid-adenylate ester | Human | 13515 | |
| MAP2K1 | STE7 | STE | 7m0x | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 13514 | |
| MAP2K1 | STE7 | STE | 7m0x | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 13519 | |
| MAP2K1 | STE7 | STE | 7m0y | B | | phosphoaminophosphonic acid-adenylate ester | Human | 13513 | |
| MAP2K1 | STE7 | STE | 7m0z | B | | phosphoaminophosphonic acid-adenylate ester | Human | 13516 | |
| MAP2K1 | STE7 | STE | 7mfd | B | | n-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-n'-methylsulfuric diamide | Human | 14076 | |
| MAP2K1 | STE7 | STE | 7pqv | A | A | 8-(2-chloranyl-4-methoxy-phenyl)-7-fluoranyl-1-piperidin-4-yl-imidazo[4,5-c]quinoline | Human | 14157 | |
| MAP2K1 | STE7 | STE | 7pqv | A | B | 8-(2-chloranyl-4-methoxy-phenyl)-7-fluoranyl-1-piperidin-4-yl-imidazo[4,5-c]quinoline | Human | 14158 | |
| MAP2K1 | STE7 | STE | 7umb | B | | phosphoaminophosphonic acid-adenylate ester | Human | 14989 | |
| MAP2K1 | STE7 | STE | 7xlp | A | | (1~{r},3~{s})-3-[[6-[2-chloranyl-4-(4-methylpyrimidin-2-yl)oxy-phenyl]-3-methyl-1~{h}-indazol-4-yl]oxy]cyclohexan-1-amine | Human | 14644 | |
| MAP2K1 | STE7 | STE | 7xnc | A | | ~{n}-[4-[[6-(3-chloranylpyridin-4-yl)-3-methyl-1~{h}-indazol-4-yl]oxy]cyclohexyl]ethanamide | Human | 14643 | |
| MAP2K1 | STE7 | STE | 8chf | E | | - | Human | 15261 | |
| MAP2K1 | STE7 | STE | 8dgs | B | A | phosphothiophosphoric acid-adenylate ester | Human | 14825 | |
| MAP2K1 | STE7 | STE | 8dgs | B | B | phosphothiophosphoric acid-adenylate ester | Human | 14826 | |
| MAP2K1 | STE7 | STE | 8dgt | B | A | phosphothiophosphoric acid-adenylate ester | Human | 14828 | |
| MAP2K1 | STE7 | STE | 8dgt | B | B | phosphothiophosphoric acid-adenylate ester | Human | 14827 | |
| MAP2K2 | STE7 | STE | 1s9i | A | | adenosine-5'-triphosphate | Human | 2772 | |
| MAP2K2 | STE7 | STE | 1s9i | B | | adenosine-5'-triphosphate | Human | 2770 | |
| MAP2K4 | STE7 | STE | 3aln | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2832 | |
| MAP2K4 | STE7 | STE | 3aln | B | | phosphoaminophosphonic acid-adenylate ester | Human | 2830 | |
| MAP2K4 | STE7 | STE | 3aln | C | | phosphoaminophosphonic acid-adenylate ester | Human | 2831 | |
| MAP2K4 | STE7 | STE | 3alo | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2835 | |
| MAP2K4 | STE7 | STE | 3vut | A | | - | Human | 2834 | |
| MAP2K4 | STE7 | STE | 3vut | B | | - | Human | 2833 | |
| MAP2K6 | STE7 | STE | 3enm | A | A | - | Human | 1225 | |
| MAP2K6 | STE7 | STE | 3enm | A | B | - | Human | 1229 | |
| MAP2K6 | STE7 | STE | 3enm | B | A | - | Human | 1227 | |
| MAP2K6 | STE7 | STE | 3enm | B | B | - | Human | 1232 | |
| MAP2K6 | STE7 | STE | 3enm | C | A | - | Human | 1234 | |
| MAP2K6 | STE7 | STE | 3enm | C | B | - | Human | 1226 | |
| MAP2K6 | STE7 | STE | 3enm | D | A | - | Human | 1230 | |
| MAP2K6 | STE7 | STE | 3enm | D | B | - | Human | 1233 | |
| MAP2K6 | STE7 | STE | 3fme | A | | staurosporine | Human | 1231 | |
| MAP2K6 | STE7 | STE | 3vn9 | A | | 9-{5-o-[(r)-hydroxy{[(s)-hydroxy(phosphonoamino)phosphoryl]oxy}phosphoryl]-beta-l-ribofuranosyl}-9h-purin-6-amine | Human | 1228 | |
| MAP2K6 | STE7 | STE | 8a8m | B | | phosphomethylphosphonic acid adenosyl ester | Human | 14292 | |
| MAP2K6 | STE7 | STE | 8p7j | A | | n-[3-(1h-pyrrolo[2,3-b]pyridin-4-yl)phenyl]prop-2-enamide | Human | 14833 | |
| MAP2K6 | STE7 | STE | 8pm3 | A | | ~{n}-[3-(2-azanylpyridin-4-yl)phenyl]propanamide | Human | 14994 | |
| MAP2K7 | STE7 | STE | 2dyl | A | | - | Human | 1240 | |
| MAP2K7 | STE7 | STE | 3wzu | A | | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 1239 | |
| MAP2K7 | STE7 | STE | 5b2k | A | | - | Human | 6503 | |
| MAP2K7 | STE7 | STE | 5b2l | A | A | - | Human | 6501 | |
| MAP2K7 | STE7 | STE | 5b2l | A | B | - | Human | 6502 | |
| MAP2K7 | STE7 | STE | 5b2m | A | | - | Human | 6500 | |
| MAP2K7 | STE7 | STE | 5y8u | A | | - | Human | 8556 | |
| MAP2K7 | STE7 | STE | 5y90 | A | A | - | Human | 8555 | |
| MAP2K7 | STE7 | STE | 5y90 | A | B | - | Human | 8557 | |
| MAP2K7 | STE7 | STE | 5z1d | A | | n-[3-(6-methyl-1h-indazol-3-yl)phenyl]prop-2-enamide | Human | 10827 | |
| MAP2K7 | STE7 | STE | 5z1e | A | | n-[3-(6-methyl-1h-indazol-3-yl)phenyl]prop-2-enamide | Human | 10828 | |
| MAP2K7 | STE7 | STE | 6ib0 | A | | 1-[(3~{r})-3-(4-azanyl-3-ethynyl-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]prop-2-en-1-one | Human | 10922 | |
| MAP2K7 | STE7 | STE | 6ib2 | A | | 1-[(3~{r})-3-[4-azanyl-3-[1-(4-ethanoylphenyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 10921 | |
| MAP2K7 | STE7 | STE | 6qfl | A | | - | Human | 11080 | |
| MAP2K7 | STE7 | STE | 6qfr | A | | - | Human | 11081 | |
| MAP2K7 | STE7 | STE | 6qft | A | | 1-[(3~{r})-3-(4-azanyl-3-iodanyl-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]propan-1-one | Human | 11085 | |
| MAP2K7 | STE7 | STE | 6qg4 | A | | 1-[(3~{r})-3-[4-azanyl-3-(4-hydroxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 11084 | |
| MAP2K7 | STE7 | STE | 6qg7 | A | | (r)-1-(3-(4-amino-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one | Human | 11083 | |
| MAP2K7 | STE7 | STE | 6qho | A | | 1-[(3~{r})-3-(4-azanylpyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]propan-1-one | Human | 11079 | |
| MAP2K7 | STE7 | STE | 6qhr | A | | 1-[(3~{r})-3-[4-azanyl-3-(1~{h}-pyrrolo[2,3-b]pyridin-5-yl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 11082 | |
| MAP2K7 | STE7 | STE | 6yfz | A | A | - | Human | 12679 | |
| MAP2K7 | STE7 | STE | 6yfz | A | B | - | Human | 12682 | |
| MAP2K7 | STE7 | STE | 6yg0 | A | | - | Human | 12695 | |
| MAP2K7 | STE7 | STE | 6yg1 | A | A | - | Human | 12690 | |
| MAP2K7 | STE7 | STE | 6yg1 | A | B | - | Human | 12684 | |
| MAP2K7 | STE7 | STE | 6yg1 | B | A | - | Human | 12691 | |
| MAP2K7 | STE7 | STE | 6yg1 | B | B | - | Human | 12680 | |
| MAP2K7 | STE7 | STE | 6yg1 | C | A | - | Human | 12692 | |
| MAP2K7 | STE7 | STE | 6yg1 | C | B | - | Human | 12688 | |
| MAP2K7 | STE7 | STE | 6yg2 | A | A | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 12678 | |
| MAP2K7 | STE7 | STE | 6yg2 | A | B | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 12686 | |
| MAP2K7 | STE7 | STE | 6yg3 | A | A | n-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamide | Human | 12689 | |
| MAP2K7 | STE7 | STE | 6yg3 | A | B | n-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamide | Human | 12681 | |
| MAP2K7 | STE7 | STE | 6yg4 | A | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 12693 | |
| MAP2K7 | STE7 | STE | 6yg5 | A | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}amino)phenyl]acetonitrile | Human | 12677 | |
| MAP2K7 | STE7 | STE | 6yg6 | A | A | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | 12676 | |
| MAP2K7 | STE7 | STE | 6yg6 | A | B | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | 12687 | |
| MAP2K7 | STE7 | STE | 6yg6 | B | A | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | 12673 | |
| MAP2K7 | STE7 | STE | 6yg6 | B | B | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | 12694 | |
| MAP2K7 | STE7 | STE | 6yg7 | A | A | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | 12683 | |
| MAP2K7 | STE7 | STE | 6yg7 | A | B | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | 12674 | |
| MAP2K7 | STE7 | STE | 6yg7 | B | A | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | 12696 | |
| MAP2K7 | STE7 | STE | 6yg7 | B | B | ~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamide | Human | 12685 | |
| MAP2K7 | STE7 | STE | 6yz4 | A | A | - | Human | 12697 | |
| MAP2K7 | STE7 | STE | 6yz4 | A | B | - | Human | 12675 | |
| MAP2K7 | STE7 | STE | 7cbx | A | A | 3-(1h-indazol-3-yl)-5-(prop-2-enoylamino)-n-prop-2-ynyl-benzamide | Human | 12815 | |
| MAP2K7 | STE7 | STE | 7cbx | A | B | 3-(1h-indazol-3-yl)-5-(prop-2-enoylamino)-n-prop-2-ynyl-benzamide | Human | 12816 | |
| MAP2K7 | STE7 | STE | 7ovi | A | | 1-[(3~{r})-3-[4-azanyl-3-[1-(2-phenylethyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 14301 | |
| MAP2K7 | STE7 | STE | 7ovj | A | A | 1-[(3~{r})-3-[4-azanyl-3-[1-[2,2-bis(fluoranyl)-2-phenyl-ethyl]-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 14306 | |
| MAP2K7 | STE7 | STE | 7ovj | A | B | 1-[(3~{r})-3-[4-azanyl-3-[1-[2,2-bis(fluoranyl)-2-phenyl-ethyl]-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 14299 | |
| MAP2K7 | STE7 | STE | 7ovk | A | | 1-[(3~{r})-3-[4-azanyl-3-[1-(5-bromanyl-2-oxidanyl-phenyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Human | 14298 | |
| MAP2K7 | STE7 | STE | 7ovl | A | A | 3-(2~{h}-indazol-3-yl)-~{n}-[[1-[(1~{r},2~{r})-2-methoxycyclohexyl]-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamide | Human | 14307 | |
| MAP2K7 | STE7 | STE | 7ovl | A | B | 3-(2~{h}-indazol-3-yl)-~{n}-[[1-[(1~{r},2~{r})-2-methoxycyclohexyl]-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamide | Human | 14304 | |
| MAP2K7 | STE7 | STE | 7ovm | A | A | ~{n}-[(1-cyclobutyl-1,2,3-triazol-4-yl)methyl]-3-(1~{h}-indazol-3-yl)-5-(propanoylamino)benzamide | Human | 14305 | |
| MAP2K7 | STE7 | STE | 7ovm | A | B | ~{n}-[(1-cyclobutyl-1,2,3-triazol-4-yl)methyl]-3-(1~{h}-indazol-3-yl)-5-(propanoylamino)benzamide | Human | 14302 | |
| MAP2K7 | STE7 | STE | 7ovn | A | A | 3-(1~{h}-indazol-3-yl)-~{n}-[[1-(2-methylphenyl)-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamide | Human | 14303 | |
| MAP2K7 | STE7 | STE | 7ovn | A | B | 3-(1~{h}-indazol-3-yl)-~{n}-[[1-(2-methylphenyl)-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamide | Human | 14300 | |
| MAP3K12 (DLK) | MLK | TKL | 5cen | A | A | - | Human | 6157 | |
| MAP3K12 (DLK) | MLK | TKL | 5cen | A | B | - | Human | 6160 | |
| MAP3K12 (DLK) | MLK | TKL | 5ceo | A | A | 2-[[6-[3,3-bis(fluoranyl)pyrrolidin-1-yl]-4-[1-(oxetan-3-yl)piperidin-4-yl]pyridin-2-yl]amino]pyridine-4-carbonitrile | Human | 6156 | |
| MAP3K12 (DLK) | MLK | TKL | 5ceo | A | B | 2-[[6-[3,3-bis(fluoranyl)pyrrolidin-1-yl]-4-[1-(oxetan-3-yl)piperidin-4-yl]pyridin-2-yl]amino]pyridine-4-carbonitrile | Human | 6155 | |
| MAP3K12 (DLK) | MLK | TKL | 5cep | A | A | n-(5-piperidin-4-yl-1-propan-2-yl-pyrazol-3-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | 6158 | |
| MAP3K12 (DLK) | MLK | TKL | 5cep | A | B | n-(5-piperidin-4-yl-1-propan-2-yl-pyrazol-3-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | 6154 | |
| MAP3K12 (DLK) | MLK | TKL | 5ceq | A | A | 2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrile | Human | 6159 | |
| MAP3K12 (DLK) | MLK | TKL | 5ceq | A | B | 2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrile | Human | 6153 | |
| MAP3K12 (DLK) | MLK | TKL | 5vo1 | A | A | 5-{5-[(1r,5s,6r)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | 8540 | |
| MAP3K12 (DLK) | MLK | TKL | 5vo1 | A | B | 5-{5-[(1r,5s,6r)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | 8541 | |
| MAP3K12 (DLK) | MLK | TKL | 5vo2 | A | A | 5-{5-[1-(oxetan-3-yl)piperidin-4-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | 8543 | |
| MAP3K12 (DLK) | MLK | TKL | 5vo2 | A | B | 5-{5-[1-(oxetan-3-yl)piperidin-4-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | 8542 | |
| MAP3K12 (DLK) | MLK | TKL | 8deg | A | | methyl (1s,4s)-5-{(4p)-4-[5-amino-6-(difluoromethoxy)pyrazin-2-yl]-6-[(1r,4r)-2-azabicyclo[2.1.1]hexan-2-yl]pyridin-2-yl}-2,5-diazabicyclo[2.2.1]heptane-2-carboxylate | Human | 14557 | |
| MAP3K12 (DLK) | MLK | TKL | 8our | A | A | 5-[1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)-2-propan-2-yl-imidazol-4-yl]-3-(trifluoromethyloxy)pyridin-2-amine | Human | 14856 | |
| MAP3K12 (DLK) | MLK | TKL | 8our | A | B | 5-[1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)-2-propan-2-yl-imidazol-4-yl]-3-(trifluoromethyloxy)pyridin-2-amine | Human | 14852 | |
| MAP3K12 (DLK) | MLK | TKL | 8ous | A | A | (1s)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2-methyl-propan-1-ol | Human | 14857 | |
| MAP3K12 (DLK) | MLK | TKL | 8ous | A | B | (1s)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2-methyl-propan-1-ol | Human | 14854 | |
| MAP3K12 (DLK) | MLK | TKL | 8out | A | A | (1r)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-fluoranyl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2,2,2-tris(fluoranyl)ethanol | Human | 14853 | |
| MAP3K12 (DLK) | MLK | TKL | 8out | A | B | (1r)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-fluoranyl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2,2,2-tris(fluoranyl)ethanol | Human | 14855 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3c | A | A | - | Mouse | 5797 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3c | A | B | - | Mouse | 5786 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3c | B | A | - | Mouse | 5792 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3c | B | B | - | Mouse | 5787 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3e | A | A | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | 5790 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3e | A | B | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | 5795 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3e | B | A | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | 5796 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3e | B | B | (2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-ol | Mouse | 5794 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3f | A | A | 3-{2-[(5-fluoro-2-hydroxyphenyl)amino]-1,3-thiazol-4-yl}benzonitrile | Mouse | 5789 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3f | A | B | 3-{2-[(5-fluoro-2-hydroxyphenyl)amino]-1,3-thiazol-4-yl}benzonitrile | Mouse | 5788 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3g | A | A | 4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenol | Mouse | 5793 | |
| Map3k14 (NIK) | STE-Unique | STE | 4g3g | A | B | 4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenol | Mouse | 5791 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8o | A | A | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | 7373 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8o | A | B | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | 7371 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8o | B | A | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | 7372 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8o | B | B | 10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamide | Mouse | 7378 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8p | A | A | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | 7368 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8p | A | B | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | 7377 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8p | B | A | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | 7376 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8p | B | B | 6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamide | Mouse | 7379 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8q | A | A | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | 7370 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8q | A | B | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | 7369 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8q | B | A | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | 7374 | |
| Map3k14 (NIK) | STE-Unique | STE | 5t8q | B | B | 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide | Mouse | 7375 | |
| Map3k14 (NIK) | STE-Unique | STE | 6g4y | A | A | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | 10041 | |
| Map3k14 (NIK) | STE-Unique | STE | 6g4y | A | B | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | 10043 | |
| Map3k14 (NIK) | STE-Unique | STE | 6g4y | B | A | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | 10047 | |
| Map3k14 (NIK) | STE-Unique | STE | 6g4y | B | B | 10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamide | Mouse | 10045 | |
| Map3k14 (NIK) | STE-Unique | STE | 6g4z | A | A | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | 10044 | |
| Map3k14 (NIK) | STE-Unique | STE | 6g4z | A | B | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | 10046 | |
| Map3k14 (NIK) | STE-Unique | STE | 6g4z | B | A | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | 10048 | |
| Map3k14 (NIK) | STE-Unique | STE | 6g4z | B | B | 5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamide | Mouse | 10042 | |
| Map3k14 (NIK) | STE-Unique | STE | 6myn | A | A | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | 11525 | |
| Map3k14 (NIK) | STE-Unique | STE | 6myn | A | B | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | 11526 | |
| Map3k14 (NIK) | STE-Unique | STE | 6myn | B | A | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | 11524 | |
| Map3k14 (NIK) | STE-Unique | STE | 6myn | B | B | (5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Mouse | 11527 | |
| Map3k14 (NIK) | STE-Unique | STE | 7szr | A | A | 1-(3-{[(1r,4r,5s)-4-hydroxy-2-methyl-3-oxo-2-azabicyclo[3.1.0]hexan-4-yl]ethynyl}phenyl)-1h-pyrazolo[3,4-b]pyridine-3-carboxamide | Mouse | 14777 | |
| Map3k14 (NIK) | STE-Unique | STE | 7szr | A | B | 1-(3-{[(1r,4r,5s)-4-hydroxy-2-methyl-3-oxo-2-azabicyclo[3.1.0]hexan-4-yl]ethynyl}phenyl)-1h-pyrazolo[3,4-b]pyridine-3-carboxamide | Mouse | 14776 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4dn5 | A | | phosphothiophosphoric acid-adenylate ester | Human | 2205 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4dn5 | B | | phosphothiophosphoric acid-adenylate ester | Human | 2202 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4g3d | A | | - | Human | 2208 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4g3d | B | | - | Human | 2209 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4g3d | D | | - | Human | 2212 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4g3d | E | | - | Human | 2214 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4idt | A | A | 11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amine | Human | 2203 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4idt | A | B | 11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amine | Human | 2204 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4idt | B | A | 11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amine | Human | 2210 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4idt | B | B | 11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amine | Human | 2207 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4idv | A | A | 4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-ol | Human | 2211 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4idv | B | A | 4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-ol | Human | 2206 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4idv | C | A | 4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-ol | Human | 2201 | |
| MAP3K14 (NIK) | STE-Unique | STE | 4idv | D | A | 4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-ol | Human | 2213 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6wpp | A | A | 5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amine | Human | 12737 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6wpp | A | B | 5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amine | Human | 12736 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6wpp | B | A | 5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amine | Human | 12738 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6wpp | B | B | 5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amine | Human | 12739 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6z1q | A | A | desf-3r/4076 | Human | 12451 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6z1q | A | B | desf-3r/4076 | Human | 12454 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6z1q | B | A | desf-3r/4076 | Human | 12455 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6z1q | B | B | desf-3r/4076 | Human | 12449 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6z1t | A | A | 4s/3694 | Human | 12450 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6z1t | A | B | 4s/3694 | Human | 12456 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6z1t | B | A | 4s/3694 | Human | 12453 | |
| MAP3K14 (NIK) | STE-Unique | STE | 6z1t | B | B | 4s/3694 | Human | 12452 | |
| MAP3K14 (NIK) | STE-Unique | STE | 8yhw | A | | phosphothiophosphoric acid-adenylate ester | Human | 15233 | |
| MAP3K20 (ZAK) | MLK | TKL | 5hes | A | A | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6460 | |
| MAP3K20 (ZAK) | MLK | TKL | 5hes | A | B | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6458 | |
| MAP3K20 (ZAK) | MLK | TKL | 5hes | B | A | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6459 | |
| MAP3K20 (ZAK) | MLK | TKL | 5hes | B | B | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6457 | |
| MAP3K20 (ZAK) | MLK | TKL | 5x5o | A | A | n-[2,4-bis(fluoranyl)-3-[2-(3-methoxy-1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-bromanyl-benzenesulfonamide | Human | 9449 | |
| MAP3K20 (ZAK) | MLK | TKL | 5x5o | A | B | n-[2,4-bis(fluoranyl)-3-[2-(3-methoxy-1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-bromanyl-benzenesulfonamide | Human | 9448 | |
| MAP3K20 (ZAK) | MLK | TKL | 6jut | A | | ~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]-3-bromanyl-benzenesulfonamide | Human | 11462 | |
| MAP3K20 (ZAK) | MLK | TKL | 6juu | A | A | ~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamide | Human | 12167 | |
| MAP3K20 (ZAK) | MLK | TKL | 6juu | A | B | ~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamide | Human | 12166 | |
| MAP3K20 (ZAK) | MLK | TKL | 7yaw | A | A | ~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamide | Human | 14891 | |
| MAP3K20 (ZAK) | MLK | TKL | 7yaw | A | B | ~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamide | Human | 14893 | |
| MAP3K20 (ZAK) | MLK | TKL | 7yaz | A | A | ~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamide | Human | 14894 | |
| MAP3K20 (ZAK) | MLK | TKL | 7yaz | A | B | ~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamide | Human | 14892 | |
| MAP3K21 (MLK4) | MLK | TKL | 4uya | A | | phosphothiophosphoric acid-adenylate ester | Human | 6126 | |
| MAP3K5 | STE11 | STE | 2clq | A | A | staurosporine | Human | 4740 | |
| MAP3K5 | STE11 | STE | 2clq | A | B | staurosporine | Human | 4736 | |
| MAP3K5 | STE11 | STE | 2clq | B | A | staurosporine | Human | 4755 | |
| MAP3K5 | STE11 | STE | 2clq | B | B | staurosporine | Human | 4732 | |
| MAP3K5 | STE11 | STE | 3vw6 | A | A | 4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | 4747 | |
| MAP3K5 | STE11 | STE | 3vw6 | A | B | 4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | 4752 | |
| MAP3K5 | STE11 | STE | 3vw6 | B | A | 4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | 4738 | |
| MAP3K5 | STE11 | STE | 3vw6 | B | B | 4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | 4737 | |
| MAP3K5 | STE11 | STE | 4bf2 | A | | staurosporine | Human | 4743 | |
| MAP3K5 | STE11 | STE | 4bf2 | B | | staurosporine | Human | 4745 | |
| MAP3K5 | STE11 | STE | 4bhn | A | A | 4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | 4754 | |
| MAP3K5 | STE11 | STE | 4bhn | A | B | 4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | 4758 | |
| MAP3K5 | STE11 | STE | 4bhn | B | A | 4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | 4734 | |
| MAP3K5 | STE11 | STE | 4bhn | B | B | 4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamide | Human | 4748 | |
| MAP3K5 | STE11 | STE | 4bib | A | A | 3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamide | Human | 4750 | |
| MAP3K5 | STE11 | STE | 4bib | A | B | 3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamide | Human | 4759 | |
| MAP3K5 | STE11 | STE | 4bib | B | A | 3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamide | Human | 4733 | |
| MAP3K5 | STE11 | STE | 4bib | B | B | 3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamide | Human | 4749 | |
| MAP3K5 | STE11 | STE | 4bic | A | | n-(2-aminoethyl)-5-{1h-pyrrolo[2,3-b]pyridin-3-yl}thiophene-2-sulfonamide | Human | 4739 | |
| MAP3K5 | STE11 | STE | 4bic | B | | - | Human | 4741 | |
| MAP3K5 | STE11 | STE | 4bid | A | A | 5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridine | Human | 4756 | |
| MAP3K5 | STE11 | STE | 4bid | A | B | 5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridine | Human | 4753 | |
| MAP3K5 | STE11 | STE | 4bid | B | A | 5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridine | Human | 4742 | |
| MAP3K5 | STE11 | STE | 4bid | B | B | 5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridine | Human | 4744 | |
| MAP3K5 | STE11 | STE | 4bie | A | A | n-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide | Human | 4746 | |
| MAP3K5 | STE11 | STE | 4bie | A | B | n-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide | Human | 4757 | |
| MAP3K5 | STE11 | STE | 4bie | B | A | n-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide | Human | 4735 | |
| MAP3K5 | STE11 | STE | 4bie | B | B | n-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamide | Human | 4751 | |
| MAP3K5 | STE11 | STE | 5uor | A | | 6-{[(2s)-4-methylmorpholin-2-yl]methoxy}-2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-one | Human | 8107 | |
| MAP3K5 | STE11 | STE | 5uor | B | | 6-{[(2s)-4-methylmorpholin-2-yl]methoxy}-2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-one | Human | 8108 | |
| MAP3K5 | STE11 | STE | 5uox | A | | 2-(6-{4-[(2r)-1-hydroxypropan-2-yl]-4h-1,2,4-triazol-3-yl}pyridin-2-yl)-6-[(propan-2-yl)oxy]-2,3-dihydro-1h-isoindol-1-one | Human | 8109 | |
| MAP3K5 | STE11 | STE | 5uox | B | | 2-(6-{4-[(2r)-1-hydroxypropan-2-yl]-4h-1,2,4-triazol-3-yl}pyridin-2-yl)-6-[(propan-2-yl)oxy]-2,3-dihydro-1h-isoindol-1-one | Human | 8106 | |
| MAP3K5 | STE11 | STE | 5up3 | A | | 2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-one | Human | 8105 | |
| MAP3K5 | STE11 | STE | 5up3 | B | | 2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-one | Human | 8110 | |
| MAP3K5 | STE11 | STE | 5v19 | A | | n-(1-ethyl-1h-pyrazol-4-yl)furan-3-carboxamide | Human | 8025 | |
| MAP3K5 | STE11 | STE | 5v19 | B | | n-(1-ethyl-1h-pyrazol-4-yl)furan-3-carboxamide | Human | 8024 | |
| MAP3K5 | STE11 | STE | 5v24 | A | A | 2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamide | Human | 8022 | |
| MAP3K5 | STE11 | STE | 5v24 | A | B | 2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamide | Human | 8021 | |
| MAP3K5 | STE11 | STE | 5v24 | B | A | 2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamide | Human | 8026 | |
| MAP3K5 | STE11 | STE | 5v24 | B | B | 2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamide | Human | 8023 | |
| MAP3K5 | STE11 | STE | 5vil | A | | 2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamide | Human | 9512 | |
| MAP3K5 | STE11 | STE | 5vil | B | | 2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamide | Human | 9509 | |
| MAP3K5 | STE11 | STE | 5vil | C | | 2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamide | Human | 9506 | |
| MAP3K5 | STE11 | STE | 5vil | D | | 2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamide | Human | 9508 | |
| MAP3K5 | STE11 | STE | 5vio | A | | 4-methoxy-n~1~-methyl-n~3~-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzene-1,3-dicarboxamide | Human | 9510 | |
| MAP3K5 | STE11 | STE | 5vio | B | | 4-methoxy-n~1~-methyl-n~3~-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzene-1,3-dicarboxamide | Human | 9507 | |
| MAP3K5 | STE11 | STE | 5vio | C | | - | Human | 9511 | |
| MAP3K5 | STE11 | STE | 5vio | D | | 4-methoxy-n~1~-methyl-n~3~-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzene-1,3-dicarboxamide | Human | 9505 | |
| MAP3K5 | STE11 | STE | 6e2m | A | | n-[3-(4-methyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide | Human | 10575 | |
| MAP3K5 | STE11 | STE | 6e2m | B | | n-[3-(4-methyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide | Human | 10576 | |
| MAP3K5 | STE11 | STE | 6e2n | A | | n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl][3,4'-bipyridine]-2'-carboxamide | Human | 10577 | |
| MAP3K5 | STE11 | STE | 6e2n | B | | n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl][3,4'-bipyridine]-2'-carboxamide | Human | 10572 | |
| MAP3K5 | STE11 | STE | 6e2o | A | | 4-(4-cyclopropyl-1h-imidazol-1-yl)-n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide | Human | 10574 | |
| MAP3K5 | STE11 | STE | 6e2o | B | | 4-(4-cyclopropyl-1h-imidazol-1-yl)-n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamide | Human | 10573 | |
| MAP3K5 | STE11 | STE | 6oyt | A | | 5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamide | Human | 11837 | |
| MAP3K5 | STE11 | STE | 6oyt | B | | 5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamide | Human | 11835 | |
| MAP3K5 | STE11 | STE | 6oyt | C | | 5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamide | Human | 11840 | |
| MAP3K5 | STE11 | STE | 6oyt | D | | 5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamide | Human | 11844 | |
| MAP3K5 | STE11 | STE | 6oyw | A | A | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | 11836 | |
| MAP3K5 | STE11 | STE | 6oyw | A | B | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | 11842 | |
| MAP3K5 | STE11 | STE | 6oyw | B | A | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | 11839 | |
| MAP3K5 | STE11 | STE | 6oyw | B | B | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | 11841 | |
| MAP3K5 | STE11 | STE | 6oyw | C | A | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | 11838 | |
| MAP3K5 | STE11 | STE | 6oyw | C | B | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | 11843 | |
| MAP3K5 | STE11 | STE | 6oyw | D | A | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | 11834 | |
| MAP3K5 | STE11 | STE | 6oyw | D | B | (19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-one | Human | 11833 | |
| MAP3K5 | STE11 | STE | 6vre | A | A | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | 12236 | |
| MAP3K5 | STE11 | STE | 6vre | A | B | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | 12233 | |
| MAP3K5 | STE11 | STE | 6vre | B | A | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | 12235 | |
| MAP3K5 | STE11 | STE | 6vre | B | B | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | 12234 | |
| MAP3K5 | STE11 | STE | 6xih | A | A | (2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamide | Human | 12703 | |
| MAP3K5 | STE11 | STE | 6xih | A | B | (2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamide | Human | 12700 | |
| MAP3K5 | STE11 | STE | 6xih | B | A | (2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamide | Human | 12702 | |
| MAP3K5 | STE11 | STE | 6xih | B | B | (2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamide | Human | 12701 | |
| MAP3K5 | STE11 | STE | 7mu7 | A | A | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | 14221 | |
| MAP3K5 | STE11 | STE | 7mu7 | A | B | 3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamide | Human | 14220 | |
| MAP3K5 | STE11 | STE | 8qgy | A | | - | Human | 15268 | |
| MAP3K7 (TAK1) | MLK | TKL | 2eva | A | A | adenosine | Human | 1884 | |
| MAP3K7 (TAK1) | MLK | TKL | 2eva | A | B | adenosine | Human | 1882 | |
| MAP3K7 (TAK1) | MLK | TKL | 2yiy | A | | (1e)-1-[5-tert-butyl-2-(3-fluorophenyl)-1h-pyrazol-3-ylidene]-3-(4-pyridin-3-yloxyphenyl)urea | Human | 1890 | |
| MAP3K7 (TAK1) | MLK | TKL | 4gs6 | A | A | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 1885 | |
| MAP3K7 (TAK1) | MLK | TKL | 4gs6 | A | B | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 1886 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l3p | A | | 2-(1-benzothiophen-7-yl)-4-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[2,3-c]pyridin-7-amine | Human | 1891 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l52 | A | A | 1-(4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}piperidin-1-yl)ethanone | Human | 1883 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l52 | A | B | 1-(4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}piperidin-1-yl)ethanone | Human | 1889 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l53 | A | A | trans-4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}cyclohexanol | Human | 1887 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l53 | A | B | trans-4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}cyclohexanol | Human | 1892 | |
| MAP3K7 (TAK1) | MLK | TKL | 4o91 | A | | n-{4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-4-methyl-3-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)benzamide | Human | 1888 | |
| MAP3K7 (TAK1) | MLK | TKL | 5e7r | A | | 2-chloro-n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}acetamide | Human | 7412 | |
| MAP3K7 (TAK1) | MLK | TKL | 5gjd | A | | 1-(4-((1h-pyrrolo[2,3-b]pyridin-4-yl)oxy)phenyl)-3-(5-(4-methylpiperazin-1-yl)naphthalen-2-yl)urea | Human | 7263 | |
| MAP3K7 (TAK1) | MLK | TKL | 5gjf | A | | n-(2-isopropoxy-4-(4-methylpiperazine-1-carbonyl)phenyl)-2-(3-(3-phenylureido)phenyl)thiazole-4-carboxamide | Human | 7264 | |
| MAP3K7 (TAK1) | MLK | TKL | 5gjg | A | | n-(2-isopropoxy-4-(4-methylpiperazine-1-carbonyl)phenyl)-2-(3-(phenylcarbamoyl)phenyl)thiazole-4-carboxamide | Human | 7265 | |
| MAP3K7 (TAK1) | MLK | TKL | 5j7s | A | | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 7429 | |
| MAP3K7 (TAK1) | MLK | TKL | 5j8i | A | | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | Human | 7428 | |
| MAP3K7 (TAK1) | MLK | TKL | 5j9l | A | | n-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamide | Human | 7426 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jga | A | | n-[5-(4-methylpiperazine-1-carbonyl)[1,1'-biphenyl]-2-yl]-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamide | Human | 6886 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jgb | A | | n-(2-methoxy-4-{[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamide | Human | 6885 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jgd | A | | n-(2-isopropoxy-3-(4-methylpiperazine-1-carbonyl)phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamide | Human | 6884 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jh6 | A | | 2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl prop-2-enoate | Human | 7427 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jk3 | A | | ~{n}-[2-[5-chloranyl-2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]oxyphenyl]prop-2-enamide | Human | 7430 | |
| MAP3K7 (TAK1) | MLK | TKL | 5v5n | A | A | n~1~-(1-propyl-1,3-dihydro-2h-benzimidazol-2-ylidene)benzene-1,3-dicarboxamide | Human | 8350 | |
| MAP3K7 (TAK1) | MLK | TKL | 5v5n | A | B | n~1~-(1-propyl-1,3-dihydro-2h-benzimidazol-2-ylidene)benzene-1,3-dicarboxamide | Human | 8351 | |
| MAP3K7 (TAK1) | MLK | TKL | 7nth | A | A | 2-[[5-[[2-[bis(fluoranyl)methoxy]phenyl]methyl-[(2~{r})-1-(methylamino)-1-oxidanylidene-propan-2-yl]carbamoyl]-1~{h}-imidazol-2-yl]carbonyl]isoindole-5-carboxamide | Human | 13456 | |
| MAP3K7 (TAK1) | MLK | TKL | 7nth | A | B | 2-[[5-[[2-[bis(fluoranyl)methoxy]phenyl]methyl-[(2~{r})-1-(methylamino)-1-oxidanylidene-propan-2-yl]carbamoyl]-1~{h}-imidazol-2-yl]carbonyl]isoindole-5-carboxamide | Human | 13458 | |
| MAP3K7 (TAK1) | MLK | TKL | 7nti | A | A | ~{n}-[[2-[bis(fluoranyl)methoxy]phenyl]methyl]-~{n}-[2-(methylamino)-2-oxidanylidene-ethyl]-2-pyrrolidin-1-ylcarbonyl-1~{h}-imidazole-4-carboxamide | Human | 13459 | |
| MAP3K7 (TAK1) | MLK | TKL | 7nti | A | B | ~{n}-[[2-[bis(fluoranyl)methoxy]phenyl]methyl]-~{n}-[2-(methylamino)-2-oxidanylidene-ethyl]-2-pyrrolidin-1-ylcarbonyl-1~{h}-imidazole-4-carboxamide | Human | 13457 | |
| MAP3K7 (TAK1) | MLK | TKL | 8gw3 | A | | - | Human | 14877 | |
| MAP3K8 (COT) | STE-Unique | STE | 4y83 | A | | 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 428 | |
| MAP3K8 (COT) | STE-Unique | STE | 4y83 | B | | 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 426 | |
| MAP3K8 (COT) | STE-Unique | STE | 4y83 | C | | 5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 425 | |
| MAP3K8 (COT) | STE-Unique | STE | 4y85 | A | | 5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine | Human | 427 | |
| MAP3K8 (COT) | STE-Unique | STE | 4y85 | B | | 5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine | Human | 429 | |
| MAP3K8 (COT) | STE-Unique | STE | 4y85 | C | | 5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amine | Human | 424 | |
| MAP3K8 (COT) | STE-Unique | STE | 5iu2 | A | A | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | 6980 | |
| MAP3K8 (COT) | STE-Unique | STE | 5iu2 | A | B | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | 6981 | |
| MAP3K8 (COT) | STE-Unique | STE | 5iu2 | B | A | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | 6979 | |
| MAP3K8 (COT) | STE-Unique | STE | 5iu2 | B | B | n-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amine | Human | 6978 | |
| MAP3K9 (MLK1) | MLK | TKL | 3dtc | A | | 12-(2-hydroxyethyl)-2-(1-methylethoxy)-13,14-dihydronaphtho[2,1-a]pyrrolo[3,4-c]carbazol-5(12h)-one | Human | 3839 | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | A | A | - | Human | 6127 | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | A | B | - | Human | 6128 | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | B | A | - | Human | 6129 | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | B | B | - | Human | 6130 | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqd | A | | phosphoaminophosphonic acid-adenylate ester | Human | 10803 | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqd | B | | phosphoaminophosphonic acid-adenylate ester | Human | 10801 | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqe | A | A | - | Human | 10802 | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqe | A | B | - | Human | 10804 | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqe | B | A | - | Human | 10805 | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqe | B | B | - | Human | 10800 | |
| MAP4K1 (HPK1) | STE20 | STE | 6cqf | A | | n-{2-(3,3-difluoropyrrolidin-1-yl)-6-[(3r)-pyrrolidin-3-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-pyrazolo[4,3-c]pyridin-6-amine | Human | 10806 | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfy | A | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 11075 | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfy | A | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 11072 | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfy | B | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 11076 | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfy | B | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 11077 | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfz | A | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 11078 | |
| MAP4K1 (HPK1) | STE20 | STE | 6nfz | B | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 11074 | |
| MAP4K1 (HPK1) | STE20 | STE | 6ng0 | A | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 11071 | |
| MAP4K1 (HPK1) | STE20 | STE | 6ng0 | B | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 11073 | |
| MAP4K1 (HPK1) | STE20 | STE | 7kac | A | | 5-{[4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-5-(1,3,4-oxadiazol-2-yl)pyrimidin-2-yl]amino}-3,3-dimethyl-2-benzofuran-1(3h)-one | Human | 13231 | |
| MAP4K1 (HPK1) | STE20 | STE | 7kac | B | | 5-{[4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-5-(1,3,4-oxadiazol-2-yl)pyrimidin-2-yl]amino}-3,3-dimethyl-2-benzofuran-1(3h)-one | Human | 13230 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | A | A | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | 13416 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | A | B | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | 13418 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | B | A | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | 13422 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | B | B | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | 13426 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | C | A | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | 13423 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | C | B | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | 13417 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | D | A | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | 13415 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l24 | D | B | 6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridine | Human | 13421 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l25 | A | A | 6-(2-fluoro-6-methoxyphenyl)-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[4,3-c]pyridine | Human | 13428 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l25 | A | B | 6-(2-fluoro-6-methoxyphenyl)-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[4,3-c]pyridine | Human | 13424 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l25 | B | A | 6-(2-fluoro-6-methoxyphenyl)-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[4,3-c]pyridine | Human | 13413 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l25 | B | B | 6-(2-fluoro-6-methoxyphenyl)-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[4,3-c]pyridine | Human | 13425 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l26 | A | A | 6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrile | Human | 13427 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l26 | A | B | 6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrile | Human | 13429 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l26 | B | A | 6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrile | Human | 13430 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l26 | B | B | 6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrile | Human | 13414 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l26 | C | A | 6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrile | Human | 13419 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l26 | C | B | 6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrile | Human | 13420 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l26 | D | A | 6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrile | Human | 13431 | |
| MAP4K1 (HPK1) | STE20 | STE | 7l26 | D | B | 6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrile | Human | 13432 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0k | A | A | 4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13480 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0k | A | B | 4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13481 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0k | B | A | 4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13476 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0k | B | B | 4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13470 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0k | C | A | 4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13473 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0k | C | B | 4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13474 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0k | D | A | 4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13479 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0k | D | B | 4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13471 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0l | A | | 4-(2-bromoanilino)-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13475 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0l | B | | 4-(2-bromoanilino)-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13466 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0l | C | | 4-(2-bromoanilino)-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13478 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0l | D | | 4-(2-bromoanilino)-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13468 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0m | A | A | 4-[2-fluoro-6-(trifluoromethyl)anilino]-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13469 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0m | A | B | 4-[2-fluoro-6-(trifluoromethyl)anilino]-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13477 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0m | B | A | 4-[2-fluoro-6-(trifluoromethyl)anilino]-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13467 | |
| MAP4K1 (HPK1) | STE20 | STE | 7m0m | B | B | 4-[2-fluoro-6-(trifluoromethyl)anilino]-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamide | Human | 13472 | |
| MAP4K1 (HPK1) | STE20 | STE | 7r9l | A | | 2-amino-n,n-dimethyl-5-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamide | Human | 14026 | |
| MAP4K1 (HPK1) | STE20 | STE | 7r9n | A | A | n-{2-(3,3-difluoropyrrolidin-1-yl)-6-[(3r)-pyrrolidin-3-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-pyrazolo[4,3-c]pyridin-6-amine | Human | 14025 | |
| MAP4K1 (HPK1) | STE20 | STE | 7r9n | A | B | n-{2-(3,3-difluoropyrrolidin-1-yl)-6-[(3r)-pyrrolidin-3-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-pyrazolo[4,3-c]pyridin-6-amine | Human | 14023 | |
| MAP4K1 (HPK1) | STE20 | STE | 7r9p | A | | 6-amino-2-fluoro-n,n-dimethyl-3-(4'-methylspiro[cyclopropane-1,3'-pyrrolo[2,3-b]pyridin]-5'-yl)benzamide | Human | 14022 | |
| MAP4K1 (HPK1) | STE20 | STE | 7r9t | A | | 6-amino-3-[(1s,3r)-4'-chloro-3-hydroxy-1',2'-dihydrospiro[cyclopentane-1,3'-pyrrolo[2,3-b]pyridin]-5'-yl]-2-fluoro-n,n-dimethylbenzamide | Human | 14024 | |
| MAP4K1 (HPK1) | STE20 | STE | 7siu | A | | 6-[(5r)-5-benzamidocyclohex-1-en-1-yl]-3-[(1-methyl-1h-pyrazol-4-yl)amino]pyrazine-2-carboxamide | Human | 14117 | |
| MAP4K1 (HPK1) | STE20 | STE | 8cdw | A | A | ~{n}-[4-(1-methylpiperidin-4-yl)phenyl]-7-(1-methylpyrazol-4-yl)quinazolin-2-amine | Human | 14896 | |
| MAP4K1 (HPK1) | STE20 | STE | 8cdw | A | B | ~{n}-[4-(1-methylpiperidin-4-yl)phenyl]-7-(1-methylpyrazol-4-yl)quinazolin-2-amine | Human | 14895 | |
| MAP4K1 (HPK1) | STE20 | STE | 8cij | A | | 2-[[8-azanyl-7-fluoranyl-6-(8-methyl-2,3-dihydro-1~{h}-pyrido[2,3-b][1,4]oxazin-7-yl)isoquinolin-3-yl]amino]-6-propan-2-yl-5,8-dihydro-4~{h}-pyrazolo[1,5-d][1,4]diazepin-7-one | Human | 14897 | |
| MAP4K1 (HPK1) | STE20 | STE | 8fh4 | A | A | (3p)-3-[6-chloro-4-(9-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | 14688 | |
| MAP4K1 (HPK1) | STE20 | STE | 8fh4 | A | B | (3p)-3-[6-chloro-4-(9-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | 14690 | |
| MAP4K1 (HPK1) | STE20 | STE | 8fjz | A | | (3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | Human | 14691 | |
| MAP4K1 (HPK1) | STE20 | STE | 8fko | A | | (3p)-3-{4-[(2s,5r)-5-amino-2-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | Human | 14689 | |
| MAP4K1 (HPK1) | STE20 | STE | 8par | A | | ~{n}-[3,5-bis(fluoranyl)-4-[[3-[1-(trifluoromethyl)cyclopropyl]-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-2,9-dioxa-4-azaspiro[5.5]undec-3-en-3-amine | Human | 15319 | |
| MAP4K1 (HPK1) | STE20 | STE | 8pas | A | | 4-[2,6-bis(fluoranyl)-4-(3-morpholin-4-ylpropylcarbamoylamino)phenoxy]-~{n}-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1~{h}-pyrrolo[2,3-b]pyridine-3-carboxamide | Human | 15318 | |
| MAP4K1 (HPK1) | STE20 | STE | 8pau | A | | [(5~{r})-2-[[3,5-bis(fluoranyl)-4-[[3-(trifluoromethyl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]amino]-5-fluoranyl-4,6-dihydro-1,3-oxazin-5-yl]methanol | Human | 15317 | |
| MAP4K3 (KHS2) | STE20 | STE | 5j5t | A | | 5-[2-(piperidin-4-yl)-1,3-thiazol-5-yl]-3-[(pyridin-4-yl)methoxy]pyridin-2-amine | Human | 7133 | |
| MAP4K4 (HGK) | STE20 | STE | 4obo | A | A | 6-(3-chlorophenyl)quinazolin-4-amine | Human | 2746 | |
| MAP4K4 (HGK) | STE20 | STE | 4obo | A | B | 6-(3-chlorophenyl)quinazolin-4-amine | Human | 2744 | |
| MAP4K4 (HGK) | STE20 | STE | 4obo | B | A | - | Human | 2762 | |
| MAP4K4 (HGK) | STE20 | STE | 4obo | B | B | - | Human | 2748 | |
| MAP4K4 (HGK) | STE20 | STE | 4obp | A | A | 6-(2-fluoropyridin-4-yl)pyrido[3,2-d]pyrimidin-4-amine | Human | 2750 | |
| MAP4K4 (HGK) | STE20 | STE | 4obp | A | B | 6-(2-fluoropyridin-4-yl)pyrido[3,2-d]pyrimidin-4-amine | Human | 2761 | |
| MAP4K4 (HGK) | STE20 | STE | 4obp | B | A | - | Human | 2754 | |
| MAP4K4 (HGK) | STE20 | STE | 4obp | B | B | - | Human | 2757 | |
| MAP4K4 (HGK) | STE20 | STE | 4obq | A | A | n-[3-(4-aminoquinazolin-6-yl)-5-fluorophenyl]-2-(pyrrolidin-1-yl)acetamide | Human | 2758 | |
| MAP4K4 (HGK) | STE20 | STE | 4obq | A | B | n-[3-(4-aminoquinazolin-6-yl)-5-fluorophenyl]-2-(pyrrolidin-1-yl)acetamide | Human | 2755 | |
| MAP4K4 (HGK) | STE20 | STE | 4obq | B | A | - | Human | 2736 | |
| MAP4K4 (HGK) | STE20 | STE | 4obq | B | B | - | Human | 2742 | |
| MAP4K4 (HGK) | STE20 | STE | 4rvt | A | A | 3-hexanoyl-4-hydroxy-5-(4-hydroxyphenyl)pyridin-2(1h)-one | Human | 2751 | |
| MAP4K4 (HGK) | STE20 | STE | 4rvt | A | B | 3-hexanoyl-4-hydroxy-5-(4-hydroxyphenyl)pyridin-2(1h)-one | Human | 2760 | |
| MAP4K4 (HGK) | STE20 | STE | 4rvt | B | A | - | Human | 2749 | |
| MAP4K4 (HGK) | STE20 | STE | 4rvt | B | B | - | Human | 2739 | |
| MAP4K4 (HGK) | STE20 | STE | 4u3y | A | A | - | Human | 6339 | |
| MAP4K4 (HGK) | STE20 | STE | 4u3y | A | B | - | Human | 6340 | |
| MAP4K4 (HGK) | STE20 | STE | 4u3y | B | A | - | Human | 6344 | |
| MAP4K4 (HGK) | STE20 | STE | 4u3y | B | B | - | Human | 6343 | |
| MAP4K4 (HGK) | STE20 | STE | 4u3z | A | A | - | Human | 6333 | |
| MAP4K4 (HGK) | STE20 | STE | 4u3z | A | B | - | Human | 6326 | |
| MAP4K4 (HGK) | STE20 | STE | 4u3z | B | A | - | Human | 6336 | |
| MAP4K4 (HGK) | STE20 | STE | 4u3z | B | B | - | Human | 6327 | |
| MAP4K4 (HGK) | STE20 | STE | 4u40 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 6332 | |
| MAP4K4 (HGK) | STE20 | STE | 4u40 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 6329 | |
| MAP4K4 (HGK) | STE20 | STE | 4u40 | B | A | - | Human | 6342 | |
| MAP4K4 (HGK) | STE20 | STE | 4u40 | B | B | - | Human | 6331 | |
| MAP4K4 (HGK) | STE20 | STE | 4u41 | A | A | 6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amine | Human | 6338 | |
| MAP4K4 (HGK) | STE20 | STE | 4u41 | A | B | 6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amine | Human | 6334 | |
| MAP4K4 (HGK) | STE20 | STE | 4u41 | B | A | - | Human | 6341 | |
| MAP4K4 (HGK) | STE20 | STE | 4u41 | B | B | - | Human | 6328 | |
| MAP4K4 (HGK) | STE20 | STE | 4u42 | A | A | 6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amine | Human | 6335 | |
| MAP4K4 (HGK) | STE20 | STE | 4u42 | A | B | 6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amine | Human | 6337 | |
| MAP4K4 (HGK) | STE20 | STE | 4u42 | B | A | 6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amine | Human | 6330 | |
| MAP4K4 (HGK) | STE20 | STE | 4u42 | B | B | 6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amine | Human | 6325 | |
| MAP4K4 (HGK) | STE20 | STE | 4u43 | A | A | n-(pyridin-3-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 2763 | |
| MAP4K4 (HGK) | STE20 | STE | 4u43 | A | B | n-(pyridin-3-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 2738 | |
| MAP4K4 (HGK) | STE20 | STE | 4u43 | B | A | - | Human | 2753 | |
| MAP4K4 (HGK) | STE20 | STE | 4u43 | B | B | - | Human | 2743 | |
| MAP4K4 (HGK) | STE20 | STE | 4u44 | A | A | 6-phenyl-n-(pyridin-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 2752 | |
| MAP4K4 (HGK) | STE20 | STE | 4u44 | A | B | 6-phenyl-n-(pyridin-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 2745 | |
| MAP4K4 (HGK) | STE20 | STE | 4u44 | B | A | - | Human | 2737 | |
| MAP4K4 (HGK) | STE20 | STE | 4u44 | B | B | - | Human | 2740 | |
| MAP4K4 (HGK) | STE20 | STE | 4u45 | A | A | 6-(1h-pyrazol-4-yl)-n-(pyridin-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 2747 | |
| MAP4K4 (HGK) | STE20 | STE | 4u45 | A | B | 6-(1h-pyrazol-4-yl)-n-(pyridin-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 2759 | |
| MAP4K4 (HGK) | STE20 | STE | 4u45 | B | A | - | Human | 2741 | |
| MAP4K4 (HGK) | STE20 | STE | 4u45 | B | B | - | Human | 2756 | |
| MAP4K4 (HGK) | STE20 | STE | 4zk5 | A | | 8-amino-n-[1-(cyclopropylcarbonyl)azetidin-3-yl]-2-(3-fluorophenyl)-1,7-naphthyridine-5-carboxamide | Human | 6015 | |
| MAP4K4 (HGK) | STE20 | STE | 4zk5 | B | | - | Human | 6014 | |
| MAP4K4 (HGK) | STE20 | STE | 4zp5 | A | | 4-[5-(4-chlorophenyl)-1,3-oxazol-2-yl]benzamide | Human | 7091 | |
| MAP4K4 (HGK) | STE20 | STE | 4zp5 | B | | - | Human | 7090 | |
| MAP4K4 (HGK) | STE20 | STE | 5di1 | A | | 4-{6-amino-5-[4-(methylsulfonyl)phenyl]pyridin-3-yl}phenol | Human | 6354 | |
| MAP4K4 (HGK) | STE20 | STE | 5di1 | B | | - | Human | 6353 | |
| MAP4K4 (HGK) | STE20 | STE | 5j95 | A | | 1-{4-[6-amino-5-(4-chlorophenyl)pyridin-3-yl]phenyl}cyclopentane-1-carboxylic acid | Human | 7999 | |
| MAP4K4 (HGK) | STE20 | STE | 5j95 | B | | - | Human | 8000 | |
| MAP4K4 (HGK) | STE20 | STE | 5w5q | A | A | (5s,7s)-n~3~-methyl-10-[3-methyl-3-(5-methyl-1,3-oxazol-2-yl)but-1-yn-1-yl]-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Human | 10008 | |
| MAP4K4 (HGK) | STE20 | STE | 5w5q | A | B | (5s,7s)-n~3~-methyl-10-[3-methyl-3-(5-methyl-1,3-oxazol-2-yl)but-1-yn-1-yl]-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamide | Human | 10005 | |
| MAP4K4 (HGK) | STE20 | STE | 5w5q | B | A | - | Human | 10007 | |
| MAP4K4 (HGK) | STE20 | STE | 5w5q | B | B | - | Human | 10006 | |
| MAPK1 (Erk2) | MAPK | CMGC | 1pme | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 2583 | |
| MAPK1 (Erk2) | MAPK | CMGC | 1tvo | A | | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 2581 | |
| MAPK1 (Erk2) | MAPK | CMGC | 1wzy | A | | 1-allyl-5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 2618 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2ojg | A | | n,n-dimethyl-4-(4-phenyl-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamide | Human | 2603 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2oji | A | | n-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamide | Human | 2570 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2ojj | A | | (s)-n-(1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamide | Human | 2612 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2y9q | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2626 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2y9q | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2556 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2y9q | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 2567 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3i5z | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamide | Human | 2579 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3i60 | A | | 4-{2-[(2-chlorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-phenylethyl]-1h-pyrrole-2-carboxamide | Human | 2584 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3sa0 | A | A | norathyriol | Human | 2596 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3sa0 | A | B | norathyriol | Human | 2557 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3tei | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2608 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3w55 | A | | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 2573 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fmq | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2604 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fmq | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2619 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fux | A | | trans-4-{[4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)pyrimidin-2-yl]amino}cyclohexanol | Human | 2568 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fuy | A | A | {4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanone | Human | 2622 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fuy | A | B | {4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanone | Human | 2587 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv0 | A | A | n-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amine | Human | 2562 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv0 | A | B | n-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amine | Human | 2599 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv1 | A | A | n-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamide | Human | 2594 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv1 | A | B | n-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamide | Human | 2613 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv2 | A | A | 4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamide | Human | 2592 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv2 | A | B | 4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamide | Human | 2571 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv3 | A | A | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 2617 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv3 | A | B | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 2580 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv4 | A | A | 9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrile | Human | 2623 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv4 | A | B | 9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrile | Human | 2558 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv5 | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-(5-methyl-2-phenylpyrimidin-4-yl)-1h-pyrrole-2-carboxamide | Human | 2598 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv6 | A | | n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-4-(2-{[(2s)-1-hydroxybutan-2-yl]amino}-5-methylpyrimidin-4-yl)-1h-pyrrole-2-carboxamide | Human | 2551 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv7 | A | A | 4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrile | Human | 2572 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv7 | A | B | 4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrile | Human | 2614 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv8 | A | A | 6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-one | Human | 2625 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv8 | A | B | 6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-one | Human | 2601 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv9 | A | A | 3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 2582 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv9 | A | B | 3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 2552 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4g6n | A | A | 3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazole | Human | 2609 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4g6n | A | B | 3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazole | Human | 2593 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4g6o | A | | 4-{4-[4-(aminomethyl)-3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamide | Human | 2565 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4h3p | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2624 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4h3p | D | | phosphoaminophosphonic acid-adenylate ester | Human | 2575 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4h3q | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2611 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | A | | adenosine-5'-diphosphate | Human | 2554 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | B | | adenosine-5'-diphosphate | Human | 2600 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | C | | adenosine-5'-diphosphate | Human | 2595 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | D | | adenosine-5'-diphosphate | Human | 2578 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | A | A | - | Human | 2615 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | A | B | - | Human | 2577 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | C | A | - | Human | 2569 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | C | B | - | Human | 2597 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | A | A | - | Human | 2586 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | A | B | - | Human | 2607 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | C | A | - | Human | 2588 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | C | B | - | Human | 2627 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4n0s | A | A | caffeic acid | Human | 2589 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4n0s | A | B | caffeic acid | Human | 2555 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 2585 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 2566 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | E | A | phosphoaminophosphonic acid-adenylate ester | Human | 2621 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | E | B | phosphoaminophosphonic acid-adenylate ester | Human | 2591 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4o6e | A | A | n-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamide | Human | 2559 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4o6e | A | B | n-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamide | Human | 2553 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp1 | A | | n-benzyl-9h-purin-6-amine | Human | 6092 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp1 | B | | n-benzyl-9h-purin-6-amine | Human | 6080 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp2 | A | | 5-chloro-1,3-benzoxazol-2-amine | Human | 6078 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp2 | B | | - | Human | 6081 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp3 | A | | (2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-ol | Human | 6084 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp3 | B | | (2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-ol | Human | 6079 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | A | A | n-cyclohexyl-9h-purin-6-amine | Human | 6088 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | A | B | n-cyclohexyl-9h-purin-6-amine | Human | 6075 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | B | A | n-cyclohexyl-9h-purin-6-amine | Human | 6086 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | B | B | n-cyclohexyl-9h-purin-6-amine | Human | 6083 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp6 | A | | 5h-pyrrolo[2,3-b]pyrazine | Human | 6089 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp6 | B | | 5h-pyrrolo[2,3-b]pyrazine | Human | 6091 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp7 | A | | 2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6082 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp7 | B | | 2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6093 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp8 | A | | 2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6087 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp8 | B | | 2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6076 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp9 | A | | 7-(1-propyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6085 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qpa | A | | 7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6077 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qpa | B | | 7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6090 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 2602 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 2576 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qte | A | A | 4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamide | Human | 2590 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qte | A | B | 4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamide | Human | 2564 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4xj0 | A | | 1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-one | Human | 6048 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4xj0 | B | | 1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-one | Human | 6049 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zxt | A | A | catechol | Human | 6654 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zxt | A | B | catechol | Human | 6653 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzm | A | | 7-ethylsulfonyl-n-(oxan-4-yl)-6,8-dihydro-5h-pyrido[3,4-d]pyrimidin-2-amine | Human | 2616 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzn | A | A | 2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamide | Human | 2605 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzn | A | B | 2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamide | Human | 2610 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzo | A | A | n-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 2620 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzo | A | B | n-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 2606 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5ax3 | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 6398 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bue | A | | 1-benzyl-4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-one | Human | 2574 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bui | A | | 3-(4-fluorophenyl)-5-(pyridin-2-yl)-4,5,6,7-tetrahydro-2h-pyrazolo[4,3-c]pyridine | Human | 2563 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5buj | A | A | 4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-one | Human | 2560 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5buj | A | B | 4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-one | Human | 2561 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvd | A | A | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-one | Human | 6030 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvd | A | B | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-one | Human | 6028 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bve | A | A | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6029 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bve | A | B | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6026 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvf | A | A | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6031 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvf | A | B | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6027 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5k4i | A | | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 6744 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lcj | A | A | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 6833 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lcj | A | B | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 6834 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lck | A | A | ~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 6835 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lck | A | B | ~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 6836 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5ngu | A | | 2-[2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-one | Human | 7991 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhf | A | | 2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-5-(phenylmethyl)-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7997 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhh | A | | 5-(2-methoxyethyl)-2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7996 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhj | A | | 5-(2-methoxyethyl)-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7994 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhl | A | | (6~{r})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7992 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nho | A | | (6~{s})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7993 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhp | A | | 5-(2-methoxyethyl)-1-methyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydropyrrolo[3,2-c]pyridin-4-one | Human | 7998 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhv | A | | 7-[2-(oxan-4-ylamino)pyrimidin-4-yl]-3,4-dihydro-2~{h}-pyrrolo[1,2-a]pyrazin-1-one | Human | 7995 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v60 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 8261 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v60 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 8263 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v61 | A | A | - | Human | 8265 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v61 | A | B | - | Human | 8266 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v62 | A | A | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 8264 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v62 | A | B | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 8262 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5wp1 | A | A | 5,7-dihydroxy-4h-1-benzopyran-4-one | Human | 10441 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5wp1 | A | B | 5,7-dihydroxy-4h-1-benzopyran-4-one | Human | 10440 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6d5y | A | | - | Human | 10939 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6dmg | A | A | - | Human | 10811 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6dmg | A | B | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 10810 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6dmg | A | C | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 10809 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g54 | A | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10938 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g54 | A | B | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10937 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g8x | A | A | 4-chloranyl-1~{h}-indazol-3-amine | Human | 9957 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g8x | A | B | 4-chloranyl-1~{h}-indazol-3-amine | Human | 9954 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g91 | A | A | 5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amine | Human | 9965 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g91 | A | B | 5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amine | Human | 9956 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g92 | A | A | ~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amine | Human | 11409 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g92 | A | B | ~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amine | Human | 11411 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g93 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-one | Human | 9955 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g93 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-one | Human | 9959 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g97 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-one | Human | 9960 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g97 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-one | Human | 9970 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9a | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-one | Human | 11408 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9a | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-one | Human | 11412 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9d | A | A | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamide | Human | 9972 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9d | A | B | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamide | Human | 9953 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9h | A | A | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamide | Human | 9971 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9h | A | B | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamide | Human | 9958 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9j | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamide | Human | 9952 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9j | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamide | Human | 9949 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9k | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamide | Human | 9966 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9k | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamide | Human | 9947 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9m | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamide | Human | 9964 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9m | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamide | Human | 9944 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9n | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamide | Human | 11410 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9n | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamide | Human | 11413 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdm | A | A | (3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamide | Human | 9968 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdm | A | B | (3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamide | Human | 9946 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdq | A | A | 4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamide | Human | 9948 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdq | A | B | 4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamide | Human | 9973 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6ge0 | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamide | Human | 9950 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6ge0 | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamide | Human | 9961 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjb | A | A | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 10832 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjb | A | B | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 10831 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjd | A | A | cyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamate | Human | 10829 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjd | A | B | cyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamate | Human | 10830 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6nbs | A | A | - | Human | 11510 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6nbs | A | B | - | Human | 11508 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6opg | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11507 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6oph | A | | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 11509 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6opi | A | | (3r)-n-[3-(2-cyclopropylpyridin-4-yl)-1h-indazol-5-yl]-3-(methoxymethyl)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]-3,6-dihydropyridin-1(2h)-yl}ethyl)pyrrolidine-3-carboxamide | Human | 11511 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7k | A | | 1h-imidazol-2-amine | Human | 10985 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7s | A | A | - | Human | 11349 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7s | A | B | - | Human | 11343 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7t | A | A | 1,2-oxazol-3-amine | Human | 11350 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7t | A | B | 1,2-oxazol-3-amine | Human | 11347 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa1 | A | A | pyridin-2-amine | Human | 11352 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa1 | A | B | pyridin-2-amine | Human | 11346 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa3 | A | A | pyrazole | Human | 11353 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa3 | A | B | pyrazole | Human | 11345 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa4 | A | A | 1~{h}-pyridin-2-one | Human | 11344 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa4 | A | B | 1~{h}-pyridin-2-one | Human | 11351 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qag | A | A | 1~{h}-1,2,3-triazole | Human | 10988 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qag | A | B | 1~{h}-1,2,3-triazole | Human | 10982 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qah | A | A | 1-azanylpropylideneazanium | Human | 11354 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qah | A | B | 1-azanylpropylideneazanium | Human | 11348 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qal | A | A | 1,1-bis(oxidanylidene)thietan-3-ol | Human | 10987 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qal | A | B | 1,1-bis(oxidanylidene)thietan-3-ol | Human | 10981 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaq | A | A | thiophen-3-ylmethylazanium | Human | 10983 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaq | A | B | thiophen-3-ylmethylazanium | Human | 10989 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaw | A | A | [1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazanium | Human | 10984 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaw | A | B | [1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazanium | Human | 10986 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rfo | A | | - | Human | 12341 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rq4 | A | A | 6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-one | Human | 11854 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rq4 | A | B | 6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-one | Human | 11855 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6slg | A | A | (6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-one | Human | 11815 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6slg | A | B | (6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-one | Human | 11816 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7auv | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13925 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7auv | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13930 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7e73 | A | | - | Human | 14114 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7e75 | A | | - | Human | 14115 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqq | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamide | Human | 13926 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqq | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamide | Human | 13928 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqw | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13927 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqw | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13924 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr3 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13923 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr3 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13922 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr5 | A | A | (2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13921 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr5 | A | B | (2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13934 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr8 | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamide | Human | 13933 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr8 | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamide | Human | 13929 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr9 | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamide | Human | 13932 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr9 | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamide | Human | 13931 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7opm | A | A | 1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]urea | Human | 14084 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7opm | A | B | 1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]urea | Human | 14083 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7w5o | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14110 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7x4u | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14660 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7x4u | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14661 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7xc1 | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14665 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao2 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)propanamide | Human | 14415 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao2 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)propanamide | Human | 14394 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao3 | A | A | 2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14386 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao3 | A | B | 2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14414 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao4 | A | A | ~{n}-(1~{h}-indazol-5-yl)ethanesulfonamide | Human | 14416 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao4 | A | B | ~{n}-(1~{h}-indazol-5-yl)ethanesulfonamide | Human | 14399 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao5 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamide | Human | 14392 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao5 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamide | Human | 14400 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao6 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14397 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao6 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14396 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao7 | A | A | ~{n}-[(1-methylindazol-6-yl)methyl]propanamide | Human | 14389 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao7 | A | B | ~{n}-[(1-methylindazol-6-yl)methyl]propanamide | Human | 14398 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao8 | A | A | 1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-one | Human | 14410 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao8 | A | B | 1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-one | Human | 14405 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | A | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | 14420 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | B | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | 14390 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | C | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | 14401 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoa | A | A | ~{n}-pyridin-3-ylprop-2-enamide | Human | 14391 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoa | A | B | ~{n}-pyridin-3-ylpropanamide | Human | 14407 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aob | A | A | ~{n}-[(1-methylindazol-3-yl)methyl]propanamide | Human | 14402 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aob | A | B | ~{n}-[(1-methylindazol-3-yl)methyl]propanamide | Human | 14413 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoc | A | A | ~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamide | Human | 14409 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoc | A | B | ~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamide | Human | 14406 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aod | A | A | 1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-one | Human | 14417 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aod | A | B | 1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-one | Human | 14388 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoe | A | A | ~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamide | Human | 14395 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoe | A | B | ~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamide | Human | 14411 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aof | A | A | ~{n}-(2-methylpyrimidin-5-yl)propanamide | Human | 14419 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aof | A | B | ~{n}-(2-methylpyrimidin-5-yl)propanamide | Human | 14408 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aog | A | A | ~{n}-(5-methyl-1,2-oxazol-3-yl)propanamide | Human | 14403 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aog | A | B | ~{n}-(5-methyl-1,2-oxazol-3-yl)propanamide | Human | 14421 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoh | A | A | ~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamide | Human | 14385 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoh | A | B | ~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamide | Human | 14404 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoi | A | A | 1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-one | Human | 14387 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoi | A | B | 1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-one | Human | 14393 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoj | A | A | 1-[(2~{s})-2-(5-methyl-3-pyridin-4-yl-1~{h}-pyrazol-4-yl)pyrrolidin-1-yl]propan-1-one | Human | 14412 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoj | A | B | - | Human | 14418 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15300 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15298 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pst | A | A | - | Human | 15311 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pst | A | B | - | Human | 15299 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psw | A | A | - | Human | 15310 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psw | A | B | - | Human | 15303 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psy | A | | - | Human | 15308 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt0 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15297 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt0 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15307 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15302 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15309 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt3 | A | A | - | Human | 15304 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt3 | A | B | - | Human | 15305 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt5 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15306 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt5 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15301 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8u8j | A | | (4m)-4-{(4r)-3-[(2s)-2-methylbutyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(1-methyl-1h-pyrazol-5-yl)pyrimidin-2-amine | Human | 15224 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8u8k | A | | (4m)-4-{(4s)-3-[(2-chloropyridin-3-yl)methyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(oxan-4-yl)pyrimidin-2-amine | Human | 15225 | |
| MAPK10 (JNK3) | MAPK | CMGC | 1jnk | A | | phosphoaminophosphonic acid-adenylate ester | Human | 3451 | |
| MAPK10 (JNK3) | MAPK | CMGC | 1pmn | A | | cyclopropyl-{4-[5-(3,4-dichlorophenyl)-2-[(1-methyl)-piperidin]-4-yl-3-propyl-3h-imidazol-4-yl]-pyrimidin-2-yl}amine | Human | 3439 | |
| MAPK10 (JNK3) | MAPK | CMGC | 1pmu | A | | 9-(4-hydroxyphenyl)-2,7-phenanthroline | Human | 3474 | |
| MAPK10 (JNK3) | MAPK | CMGC | 1pmv | A | | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | 3434 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2b1p | A | | 3-{6-[(2-chlorophenyl)amino]-1h-indazol-3-yl}-5-{[4-(dimethylamino)butanoyl]amino}benzoic acid | Human | 3464 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2exc | X | | n-{2'-[(4-fluorophenyl)amino]-4,4'-bipyridin-2-yl}-4-methoxycyclohexanecarboxamide | Human | 3478 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2o0u | A | | n-{3-cyano-6-[3-(1-piperidinyl)propanoyl]-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-yl}1-naphthalenecarboxamide | Human | 3415 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2o2u | A | | n-(3-cyano-4,5,6,7-tetrahydro-1-benzothien-2-yl)-2-fluorobenzamide | Human | 3457 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2ok1 | A | A | n-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamide | Human | 3444 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2ok1 | A | B | n-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamide | Human | 3473 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2p33 | A | | 4-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-n-ethylpiperidine-1-carboxamide | Human | 3455 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2r9s | A | | n-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamide | Human | 3450 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2r9s | B | | n-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamide | Human | 3420 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2waj | A | A | 1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinoline | Human | 3472 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2waj | A | B | 1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinoline | Human | 3471 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2zdt | A | A | 4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acid | Human | 3421 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2zdt | A | B | 4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acid | Human | 3424 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2zdu | A | | 4-[(4-{[6-bromo-3-(methoxycarbonyl)-1-oxo-4-phenylisoquinolin-2(1h)-yl]methyl}phenyl)amino]-4-oxobutanoic acid | Human | 3479 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3cgf | A | | n-cyclohexyl-4-imidazo[1,2-a]pyridin-3-yl-n-methylpyrimidin-2-amine | Human | 6770 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3cgo | A | | 2-{4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidin-1-yl}-n-methylacetamide | Human | 6771 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3da6 | A | | n-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)naphthalen-1-yl]-1h-benzimidazol-2-amine | Human | 3476 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fi2 | A | A | 3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | 3463 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fi2 | A | B | 3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | 3452 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fi3 | A | A | 3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | 3442 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fi3 | A | B | 3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | 3445 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fv8 | A | A | 5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamide | Human | 3468 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fv8 | A | B | 5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamide | Human | 3426 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3g90 | X | | (3e)-5-fluoro-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-1h-indole-2,3-dione 3-oxime | Human | 3477 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3g9l | X | | (3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-[(e)-2-phenylethenyl]-1h-indole-2,3-dione 3-oxime | Human | 3435 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3g9n | A | | (3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-phenyl-1h-indole-2,3-dione 3-oxime | Human | 3416 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3kvx | A | A | n-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)aniline | Human | 3433 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3kvx | A | B | n-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)aniline | Human | 3430 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3oxi | A | | methyl 3-[(thiophen-2-ylacetyl)amino]thiophene-2-carboxylate | Human | 3423 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3oy1 | A | | 5-[2-(cyclohexylamino)pyridin-4-yl]-4-naphthalen-2-yl-2-(tetrahydro-2h-pyran-4-yl)-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 3469 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3ptg | A | | n-[4-methyl-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamide | Human | 3470 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3rtp | A | | n-[4-cyano-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamide | Human | 3467 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3tti | A | | trans-4-({9-[(3s)-tetrahydrofuran-3-yl]-8-[(2,4,6-trifluorophenyl)amino]-9h-purin-2-yl}amino)cyclohexanol | Human | 3456 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3ttj | A | A | 9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamine | Human | 3458 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3ttj | A | B | 9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamine | Human | 3428 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6r | A | A | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3441 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6r | A | B | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3436 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6r | B | A | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3427 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6r | B | B | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3417 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6s | A | B | 3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3449 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6s | B | B | 3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3425 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h36 | A | A | - | Human | 3459 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h36 | A | B | - | Human | 3461 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h39 | A | A | - | Human | 3460 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h39 | A | B | - | Human | 3462 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | A | A | - | Human | 3480 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | A | B | - | Human | 3454 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | A | C | - | Human | 3453 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | C | A | - | Human | 3475 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | C | B | - | Human | 3465 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | C | C | - | Human | 3446 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4kke | A | | adenosine monophosphate | Human | 3448 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4kkg | A | | - | Human | 3443 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4kkh | A | | cyclopropyl[(3r)-3-({4-[6-hydroxy-2-(naphthalen-2-yl)-1h-benzimidazol-1-yl]pyrimidin-2-yl}amino)piperidin-1-yl]methanone | Human | 3419 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4u79 | A | | n-{4-[(3-{2-[(trans-4-aminocyclohexyl)amino]pyrimidin-4-yl}pyridin-2-yl)oxy]naphthalen-1-yl}benzenesulfonamide | Human | 3466 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4w4v | A | | 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamide | Human | 3437 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4w4w | A | | n-(2-methylpyridin-4-yl)-3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}benzamide | Human | 3418 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4w4x | A | | 3-(4-{[(4-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamide | Human | 3440 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4w4y | A | | 3-(4-{[(4-methylphenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamide | Human | 3447 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4whz | A | A | 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamide | Human | 3429 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4whz | A | B | 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamide | Human | 3422 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4x21 | A | | n-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamide | Human | 6240 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4x21 | B | | n-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamide | Human | 6239 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4y46 | A | | 1-{trans-4-[(8-cyclopentyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]cyclohexyl}-3-propan-2-ylurea | Human | 3414 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4y5h | A | | 1-(trans-4-{[7-oxo-8-(propan-2-yl)-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}cyclohexyl)-3-propan-2-ylurea | Human | 3431 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4z9l | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 3432 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4z9l | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 3438 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6ekd | A | A | 4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10498 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6ekd | A | B | 4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10502 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | A | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10508 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | A | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10503 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | B | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10506 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | B | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10501 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | C | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10507 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | C | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10505 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | D | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10497 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | D | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10496 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 10500 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 10509 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 10504 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 10499 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ksi | A | | 4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13387 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ksj | A | | 4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13388 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ksk | A | | 4-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13386 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ore | A | A | 4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamide | Human | 13811 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ore | A | B | 4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamide | Human | 13810 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ore | A | C | 4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamide | Human | 13813 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7orf | A | A | n-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamide | Human | 13812 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7orf | A | B | n-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamide | Human | 13814 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7s1n | A | A | 4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13958 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7s1n | A | B | 4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13957 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7yl1 | A | | 7-hexyl-3-methyl-8-sulfanylidene-9h-purine-2,6-dione | Human | 14845 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8bzp | A | A | 2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamide | Human | 14859 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8bzp | A | B | 2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamide | Human | 14858 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8enj | A | | n-[3-({(4p)-4-[(3m)-1-tert-butyl-3-(3-hydroxyphenyl)-1h-pyrazol-4-yl]pyridin-2-yl}amino)propyl]-4-hydroxybenzene-1-sulfonamide | Human | 14884 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8wgf | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15046 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8wgf | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15047 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gc8 | A | | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 2766 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gc8 | B | | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 2769 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gc9 | A | | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 2765 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gc9 | B | | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 2767 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gp0 | A | A | nilotinib | Human | 2768 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gp0 | A | B | nilotinib | Human | 2764 | |
| MAPK11 (p38b) | MAPK | CMGC | 8ygw | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 15234 | |
| MAPK12 (p38g) | MAPK | CMGC | 1cm8 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 4625 | |
| MAPK12 (p38g) | MAPK | CMGC | 1cm8 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 4626 | |
| MAPK12 (p38g) | MAPK | CMGC | 6una | A | A | - | Human | 11898 | |
| MAPK12 (p38g) | MAPK | CMGC | 6una | A | B | - | Human | 11900 | |
| MAPK12 (p38g) | MAPK | CMGC | 6una | B | A | - | Human | 11901 | |
| MAPK12 (p38g) | MAPK | CMGC | 6una | B | B | - | Human | 11899 | |
| MAPK12 (p38g) | MAPK | CMGC | 7cga | A | | - | Human | 13762 | |
| MAPK13 (p38d) | MAPK | CMGC | 3coi | A | A | - | Human | 2948 | |
| MAPK13 (p38d) | MAPK | CMGC | 3coi | A | B | - | Human | 2946 | |
| MAPK13 (p38d) | MAPK | CMGC | 4eyj | A | | 1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-yloxy)phenyl]urea | Human | 2949 | |
| MAPK13 (p38d) | MAPK | CMGC | 4eym | A | | 2-(morpholin-4-yl)-n-[4-(pyridin-4-yloxy)phenyl]pyridine-4-carboxamide | Human | 2945 | |
| MAPK13 (p38d) | MAPK | CMGC | 4myg | A | | - | Human | 2951 | |
| MAPK13 (p38d) | MAPK | CMGC | 4myg | B | | - | Human | 2950 | |
| MAPK13 (p38d) | MAPK | CMGC | 4yno | A | | - | Human | 2947 | |
| MAPK13 (p38d) | MAPK | CMGC | 5ekn | A | | 1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-ylsulfanyl)phenyl]urea | Human | 6745 | |
| MAPK13 (p38d) | MAPK | CMGC | 5eko | A | | 3-(4-methyl-1h-imidazol-1-yl)-n-[4-(pyridin-4-yloxy)phenyl]benzamide | Human | 6746 | |
| MAPK13 (p38d) | MAPK | CMGC | 8x23 | A | A | - | Human | 15129 | |
| MAPK13 (p38d) | MAPK | CMGC | 8x23 | A | B | - | Human | 15128 | |
| Mapk14 (p38a) | MAPK | CMGC | 1lew | A | | - | Mouse | 5864 | |
| Mapk14 (p38a) | MAPK | CMGC | 1lez | A | | - | Mouse | 5863 | |
| Mapk14 (p38a) | MAPK | CMGC | 1yw2 | A | | 2-(ethoxymethyl)-4-(4-fluorophenyl)-3-[2-(2-hydroxyphenoxy)pyrimidin-4-yl]isoxazol-5(2h)-one | Mouse | 5869 | |
| Mapk14 (p38a) | MAPK | CMGC | 1ywr | A | | 4-(4-fluorophenyl)-1-methyl-5-(2-{[(1s)-1-phenylethyl]amino}pyrimidin-4-yl)-2-piperidin-4-yl-1,2-dihydro-3h-pyrazol-3-one | Mouse | 5840 | |
| Mapk14 (p38a) | MAPK | CMGC | 2ewa | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 5859 | |
| Mapk14 (p38a) | MAPK | CMGC | 2ewa | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 5870 | |
| Mapk14 (p38a) | MAPK | CMGC | 2ghl | A | | 3-(2-chlorophenyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)urea | Mouse | 5871 | |
| Mapk14 (p38a) | MAPK | CMGC | 2ghm | A | | 3-(2-chlorobenzyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)urea | Mouse | 5845 | |
| Mapk14 (p38a) | MAPK | CMGC | 2gtm | A | | 8-(2-chlorophenylamino)-2-(2,6-difluorophenylamino)-9-ethyl-9h-purine-1,7-diium | Mouse | 5867 | |
| Mapk14 (p38a) | MAPK | CMGC | 2gtn | A | | 2-(2,6-difluorophenoxy)-n-(2-fluorophenyl)-9-isopropyl-9h-purin-8-amine | Mouse | 5860 | |
| Mapk14 (p38a) | MAPK | CMGC | 2oza | B | | - | Mouse | 5862 | |
| Mapk14 (p38a) | MAPK | CMGC | 2puu | A | | 5-tert-butyl-2-(4-methylphenyl)-3-{[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]-1-naphthyl}amino)carbonyl]amino}-1h-pyrazol-2-ium | Mouse | 6866 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p4k | A | | - | Mouse | 5842 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p5k | A | | 1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylurea | Mouse | 5854 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p78 | A | | 1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-2-ylurea | Mouse | 5866 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p79 | A | | 1-{3-tert-butyl-1-[2-(1,1-dioxidothiomorpholin-4-yl)-2-oxoethyl]-1h-pyrazol-5-yl}-3-naphthalen-2-ylurea | Mouse | 5849 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p7a | A | | 1-[5-tert-butyl-2-(1,1-dioxidothiomorpholin-4-yl)thiophen-3-yl]-3-naphthalen-1-ylurea | Mouse | 5853 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p7b | A | | 1-{5-tert-butyl-3-[(5-oxo-1,4-diazepan-1-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylurea | Mouse | 5856 | |
| Mapk14 (p38a) | MAPK | CMGC | 3p7c | A | | 1-[5-tert-butyl-3-({4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepan-1-yl}carbonyl)thiophen-2-yl]-3-(2,3-dichlorophenyl)urea | Mouse | 5838 | |
| Mapk14 (p38a) | MAPK | CMGC | 3py3 | A | | - | Mouse | 5857 | |
| Mapk14 (p38a) | MAPK | CMGC | 3tg1 | A | | - | Mouse | 5850 | |
| Mapk14 (p38a) | MAPK | CMGC | 4ka3 | A | | - | Mouse | 5852 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loo | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5851 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loo | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5832 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5848 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5861 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | B | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5839 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | B | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5831 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | C | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5847 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | C | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5855 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | D | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5865 | |
| Mapk14 (p38a) | MAPK | CMGC | 4lop | D | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5837 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5872 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5836 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | B | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5834 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | B | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5833 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | C | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5858 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | C | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5846 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | D | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5835 | |
| Mapk14 (p38a) | MAPK | CMGC | 4loq | D | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 5843 | |
| Mapk14 (p38a) | MAPK | CMGC | 4tyh | B | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Mouse | 5841 | |
| Mapk14 (p38a) | MAPK | CMGC | 4tyh | B | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Mouse | 5844 | |
| Mapk14 (p38a) | MAPK | CMGC | 5lar | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 6753 | |
| Mapk14 (p38a) | MAPK | CMGC | 5lar | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 6752 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | E | A | phosphothiophosphoric acid-adenylate ester | Mouse | 9981 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | E | B | phosphothiophosphoric acid-adenylate ester | Mouse | 9980 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | F | A | phosphothiophosphoric acid-adenylate ester | Mouse | 9983 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | F | B | phosphothiophosphoric acid-adenylate ester | Mouse | 9979 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | G | A | phosphothiophosphoric acid-adenylate ester | Mouse | 9977 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | G | B | phosphothiophosphoric acid-adenylate ester | Mouse | 9982 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | H | A | phosphothiophosphoric acid-adenylate ester | Mouse | 9978 | |
| Mapk14 (p38a) | MAPK | CMGC | 5nzz | H | B | phosphothiophosphoric acid-adenylate ester | Mouse | 9984 | |
| Mapk14 (p38a) | MAPK | CMGC | 5o90 | A | | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 9525 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8u | A | A | 3,4-dihydro-2~{h}-chromene-6-carboxamide | Mouse | 12555 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8u | A | B | 3,4-dihydro-2~{h}-chromene-6-carboxamide | Mouse | 12583 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8v | A | A | - | Mouse | 12553 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8v | A | B | - | Mouse | 12556 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8w | A | A | - | Mouse | 12535 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8w | A | B | - | Mouse | 12534 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8x | A | A | - | Mouse | 12573 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8x | A | B | - | Mouse | 12521 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8y | A | A | thiophene-2-carbothioamide | Mouse | 12584 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8y | A | B | thiophene-2-carbothioamide | Mouse | 12524 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8z | A | A | 6-methoxypyridine-3-carbothioamide | Mouse | 12575 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r8z | A | B | 6-methoxypyridine-3-carbothioamide | Mouse | 12544 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r90 | A | A | 2,5-diphenyl-4~{h}-pyrazol-3-one | Mouse | 12603 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r90 | A | B | 2,5-diphenyl-4~{h}-pyrazol-3-one | Mouse | 12582 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r91 | A | A | - | Mouse | 12560 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r91 | A | B | - | Mouse | 12539 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r92 | A | A | (3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamide | Mouse | 12590 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r92 | A | B | (3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamide | Mouse | 12620 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r93 | A | A | - | Mouse | 12571 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r93 | A | B | - | Mouse | 12545 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r94 | A | A | - | Mouse | 12532 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r94 | A | B | - | Mouse | 12589 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r95 | A | A | - | Mouse | 12586 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r95 | A | B | - | Mouse | 12597 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r96 | A | A | - | Mouse | 12610 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r96 | A | B | - | Mouse | 12559 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r97 | A | A | 4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amine | Mouse | 12529 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r97 | A | B | 4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amine | Mouse | 12525 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r98 | A | A | - | Mouse | 12563 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r98 | A | B | - | Mouse | 12606 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r99 | A | A | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | 12572 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r99 | A | B | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | 12533 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9a | A | A | - | Mouse | 12565 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9a | A | B | - | Mouse | 12604 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9b | A | A | - | Mouse | 12577 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9b | A | B | - | Mouse | 12540 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9c | A | A | - | Mouse | 12591 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9c | A | B | - | Mouse | 12522 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9d | A | A | benzyl hydroxycarbamate | Mouse | 12550 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9d | A | B | benzyl hydroxycarbamate | Mouse | 12554 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9e | A | A | - | Mouse | 12602 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9e | A | B | - | Mouse | 12564 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9f | A | A | - | Mouse | 12526 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9f | A | B | - | Mouse | 12569 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9g | A | A | - | Mouse | 12547 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9g | A | B | - | Mouse | 12595 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9h | A | A | - | Mouse | 12615 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9h | A | B | - | Mouse | 12587 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9i | A | A | methyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoate | Mouse | 12548 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9i | A | B | methyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoate | Mouse | 12551 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9j | A | A | 3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dione | Mouse | 12609 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9j | A | B | 3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dione | Mouse | 12527 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9k | A | A | 2,3-dihydro-1-benzoxepine-5-carboxylic acid | Mouse | 12611 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9k | A | B | 2,3-dihydro-1-benzoxepine-5-carboxylic acid | Mouse | 12549 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9l | A | A | (3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-ol | Mouse | 12562 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9l | A | B | (3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-ol | Mouse | 12523 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9m | A | A | - | Mouse | 12574 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9m | A | B | - | Mouse | 12570 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9n | A | A | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | 12593 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9n | A | B | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | 12596 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9o | A | A | - | Mouse | 12588 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9o | A | B | - | Mouse | 12616 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9p | A | A | 4-amino-n-(pyridin-2-yl)benzenesulfonamide | Mouse | 12518 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9p | A | B | 4-amino-n-(pyridin-2-yl)benzenesulfonamide | Mouse | 12576 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9q | A | A | 1-phenylmethoxyurea | Mouse | 12557 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9q | A | B | 1-phenylmethoxyurea | Mouse | 12612 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9r | A | A | 4-acetyl-n-ethylpiperazine-1-carboxamide | Mouse | 12519 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9r | A | B | 4-acetyl-n-ethylpiperazine-1-carboxamide | Mouse | 12536 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9s | A | A | - | Mouse | 12531 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9s | A | B | - | Mouse | 12561 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9t | A | A | - | Mouse | 12618 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9t | A | B | - | Mouse | 12538 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9u | A | A | [4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanone | Mouse | 12541 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9u | A | B | [4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanone | Mouse | 12546 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9v | A | A | - | Mouse | 12530 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9v | A | B | - | Mouse | 12528 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9w | A | A | ~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamide | Mouse | 12605 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9w | A | B | ~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamide | Mouse | 12542 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9x | A | A | - | Mouse | 12566 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9x | A | B | - | Mouse | 12543 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9y | A | A | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | 12537 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9y | A | B | 3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrile | Mouse | 12621 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9z | A | A | - | Mouse | 12580 | |
| Mapk14 (p38a) | MAPK | CMGC | 5r9z | A | B | - | Mouse | 12613 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra0 | A | A | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | 12592 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra0 | A | B | [4-(1h-benzimidazol-1-yl)phenyl]methanol | Mouse | 12617 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra1 | A | A | 2-phenoxyacetamide | Mouse | 12600 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra1 | A | B | 2-phenoxyacetamide | Mouse | 12579 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra2 | A | A | 1-(3-methylpyridin-2-yl)-1,4-diazepane | Mouse | 12568 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra2 | A | B | 1-(3-methylpyridin-2-yl)-1,4-diazepane | Mouse | 12520 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra3 | A | A | - | Mouse | 12599 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra3 | A | B | - | Mouse | 12581 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra4 | A | A | - | Mouse | 12552 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra4 | A | B | - | Mouse | 12594 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra5 | A | A | - | Mouse | 12558 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra5 | A | B | - | Mouse | 12619 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra6 | A | A | 1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thiourea | Mouse | 12614 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra6 | A | B | 1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thiourea | Mouse | 12598 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra7 | A | A | 4-methylbenzamide | Mouse | 12567 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra7 | A | B | 4-methylbenzamide | Mouse | 12578 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra8 | A | A | 5-(trifluoromethyl)-1,2-benzoxazol-3-amine | Mouse | 12585 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra8 | A | B | 5-(trifluoromethyl)-1,2-benzoxazol-3-amine | Mouse | 12608 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra9 | A | A | 4-chloranylthieno[3,2-d]pyrimidine | Mouse | 12601 | |
| Mapk14 (p38a) | MAPK | CMGC | 5ra9 | A | B | 4-chloranylthieno[3,2-d]pyrimidine | Mouse | 12607 | |
| Mapk14 (p38a) | MAPK | CMGC | 5uoj | A | | - | Mouse | 7466 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so1 | A | A | - | Mouse | 11681 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so1 | A | B | - | Mouse | 11675 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so2 | A | A | - | Mouse | 11678 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so2 | A | B | - | Mouse | 11679 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so4 | A | A | - | Mouse | 11627 | |
| Mapk14 (p38a) | MAPK | CMGC | 6so4 | A | B | - | Mouse | 11626 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sod | A | A | - | Mouse | 11673 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sod | A | B | - | Mouse | 11674 | |
| Mapk14 (p38a) | MAPK | CMGC | 6soi | A | A | - | Mouse | 11676 | |
| Mapk14 (p38a) | MAPK | CMGC | 6soi | A | B | - | Mouse | 11682 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sot | A | A | - | Mouse | 11689 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sot | A | B | - | Mouse | 11688 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sou | A | A | 2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanone | Mouse | 11680 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sou | A | B | 2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanone | Mouse | 11672 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sov | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11685 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sov | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11677 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sp9 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11684 | |
| Mapk14 (p38a) | MAPK | CMGC | 6sp9 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11686 | |
| Mapk14 (p38a) | MAPK | CMGC | 6spl | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11687 | |
| Mapk14 (p38a) | MAPK | CMGC | 6spl | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 11683 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4t | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12030 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4t | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12036 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4u | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12035 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4u | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12038 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4v | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12037 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4v | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12031 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4w | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12034 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4w | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12033 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4x | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12039 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y4x | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12032 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y6v | A | A | 5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12066 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y6v | A | B | 5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12067 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7w | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12065 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7w | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12071 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7x | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12072 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7x | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12060 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7y | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12063 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7y | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12076 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7z | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12070 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y7z | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12082 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y80 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12081 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y80 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12080 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y81 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12079 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y81 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12073 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y82 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12077 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y82 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12061 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y85 | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12069 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y85 | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12068 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y8h | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12075 | |
| Mapk14 (p38a) | MAPK | CMGC | 6y8h | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12078 | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycu | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12152 | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycu | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12154 | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycw | A | A | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12153 | |
| Mapk14 (p38a) | MAPK | CMGC | 6ycw | A | B | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Mouse | 12151 | |
| Mapk14 (p38a) | MAPK | CMGC | 6yjc | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12437 | |
| Mapk14 (p38a) | MAPK | CMGC | 6yjc | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12438 | |
| Mapk14 (p38a) | MAPK | CMGC | 6yk7 | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12163 | |
| Mapk14 (p38a) | MAPK | CMGC | 6yk7 | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12164 | |
| Mapk14 (p38a) | MAPK | CMGC | 6zwr | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12708 | |
| Mapk14 (p38a) | MAPK | CMGC | 6zwr | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 12709 | |
| Mapk14 (p38a) | MAPK | CMGC | 7bdo | A | A | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Mouse | 13409 | |
| Mapk14 (p38a) | MAPK | CMGC | 7bdo | A | B | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Mouse | 13405 | |
| Mapk14 (p38a) | MAPK | CMGC | 7bdq | A | | ~{n}-[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]-4-[[(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]benzamide | Mouse | 13408 | |
| Mapk14 (p38a) | MAPK | CMGC | 7be4 | A | | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Mouse | 13406 | |
| Mapk14 (p38a) | MAPK | CMGC | 7be5 | A | | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-methyl-pyrazole-4-carboxamide | Mouse | 13407 | |
| Mapk14 (p38a) | MAPK | CMGC | 7pvu | A | A | - | Mouse | 14747 | |
| Mapk14 (p38a) | MAPK | CMGC | 7pvu | A | B | - | Mouse | 14748 | |
| Mapk14 (p38a) | MAPK | CMGC | 7z6i | A | A | 4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridine | Mouse | 14801 | |
| Mapk14 (p38a) | MAPK | CMGC | 7z6i | A | B | 4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridine | Mouse | 14800 | |
| Mapk14 (p38a) | MAPK | CMGC | 7z9t | A | | n-(2-cyclobutyl-1h-1,3-benzodiazol-5-yl)benzenesulfonamide | Mouse | 14799 | |
| Mapk14 (p38a) | MAPK | CMGC | 8acm | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 15096 | |
| Mapk14 (p38a) | MAPK | CMGC | 8aco | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 15095 | |
| Mapk14 (p38a) | MAPK | CMGC | 8aco | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Mouse | 15094 | |
| Mapk14 (p38a) | MAPK | CMGC | 8efj | A | | (4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamide | Mouse | 14995 | |
| MAPK14 (p38a) | MAPK | CMGC | 1a9u | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5229 | |
| MAPK14 (p38a) | MAPK | CMGC | 1bl6 | A | | 4-(4-fluorophenyl)-1-cycloropropylmethyl-5-(4-pyridyl)-imidazole | Human | 5243 | |
| MAPK14 (p38a) | MAPK | CMGC | 1bl7 | A | | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Human | 5193 | |
| MAPK14 (p38a) | MAPK | CMGC | 1bmk | A | | 4-(fluorophenyl)-1-cyclopropylmethyl-5-(2-amino-4-pyrimidinyl)imidazole | Human | 5235 | |
| MAPK14 (p38a) | MAPK | CMGC | 1di9 | A | | 4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazoline | Human | 5251 | |
| MAPK14 (p38a) | MAPK | CMGC | 1kv1 | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5252 | |
| MAPK14 (p38a) | MAPK | CMGC | 1kv2 | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 5255 | |
| MAPK14 (p38a) | MAPK | CMGC | 1m7q | A | | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2(1h)-one | Human | 5128 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ouk | A | | 4-[5-[2-(1-phenyl-ethylamino)-pyrimidin-4-yl]-1-methyl-4-(3-trifluoromethylphenyl)-1h-imidazol-2-yl]-piperidine | Human | 5146 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ouy | A | | 1-(2,6-dichlorophenyl)-6-[(2,4-difluorophenyl)sulfanyl]-7-(1,2,3,6-tetrahydro-4-pyridinyl)-3,4-dihydropyrido[3,2-d]pyrimidin-2(1h)-one | Human | 7258 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | A | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | 5178 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | B | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | 5087 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | C | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | 5199 | |
| MAPK14 (p38a) | MAPK | CMGC | 1oz1 | A | A | 3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-ol | Human | 5230 | |
| MAPK14 (p38a) | MAPK | CMGC | 1oz1 | A | B | 3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-ol | Human | 5261 | |
| MAPK14 (p38a) | MAPK | CMGC | 1r39 | A | | - | Human | 5116 | |
| MAPK14 (p38a) | MAPK | CMGC | 1r3c | A | A | - | Human | 5170 | |
| MAPK14 (p38a) | MAPK | CMGC | 1r3c | A | B | - | Human | 4996 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w7h | A | | 3-(benzyloxy)pyridin-2-amine | Human | 5023 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w82 | A | | n-[(3z)-5-tert-butyl-2-phenyl-1,2-dihydro-3h-pyrazol-3-ylidene]-n'-(4-chlorophenyl)urea | Human | 5165 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w83 | A | | n-[4-chloro-3-(pyridin-3-yloxymethyl)-phenyl]-3-fluoro- | Human | 4986 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w84 | A | | 3-(2-pyridin-4-ylethyl)-1h-indole | Human | 5065 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbn | A | | n-(3-tert-butyl-1h-pyrazol-5-yl)-n'-{4-chloro-3-[(pyridin-3-yloxy)methyl]phenyl}urea | Human | 5257 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbo | A | | 2-chlorophenol | Human | 5039 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbs | A | | 3-fluoro-5-morpholin-4-yl-n-[3-(2-pyridin-4-ylethyl)-1h-indol-5-yl]benzamide | Human | 5258 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbt | A | | 3-fluoro-5-morpholin-4-yl-n-[1-(2-pyridin-4-ylethyl)-1h-indol-6-yl]benzamide | Human | 5082 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbv | A | | 3-fluoro-n-1h-indol-5-yl-5-morpholin-4-ylbenzamide | Human | 5148 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbw | A | | 3-(1-naphthylmethoxy)pyridin-2-amine | Human | 5179 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wfc | A | | - | Human | 4989 | |
| MAPK14 (p38a) | MAPK | CMGC | 1yqj | A | | 6((s)-3-benzylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyrazine | Human | 5152 | |
| MAPK14 (p38a) | MAPK | CMGC | 1zyj | A | | 4-phenoxy-n-(pyridin-2-ylmethyl)benzamide | Human | 5058 | |
| MAPK14 (p38a) | MAPK | CMGC | 1zz2 | A | | n-[3-(4-fluorophenoxy)phenyl]-4-[(2-hydroxybenzyl)amino]piperidine-1-sulfonamide | Human | 5164 | |
| MAPK14 (p38a) | MAPK | CMGC | 1zzl | A | | 6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-3-isopropyl[1,2,4]triazolo[4,3-a]pyridine | Human | 5249 | |
| MAPK14 (p38a) | MAPK | CMGC | 2baj | A | | 1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2,3-dichlorophenyl)urea | Human | 5176 | |
| MAPK14 (p38a) | MAPK | CMGC | 2bak | A | | n-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamide | Human | 5114 | |
| MAPK14 (p38a) | MAPK | CMGC | 2bal | A | | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl][3-(piperidin-4-yloxy)phenyl]methanone | Human | 5260 | |
| MAPK14 (p38a) | MAPK | CMGC | 2baq | A | | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | 5184 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fsl | X | | - | Human | 5264 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fsm | X | | - | Human | 5044 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fso | X | | - | Human | 5117 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fst | X | A | - | Human | 5080 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fst | X | B | - | Human | 5195 | |
| MAPK14 (p38a) | MAPK | CMGC | 2gfs | A | A | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | 5227 | |
| MAPK14 (p38a) | MAPK | CMGC | 2gfs | A | B | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | 5050 | |
| MAPK14 (p38a) | MAPK | CMGC | 2i0h | A | A | 2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dione | Human | 5062 | |
| MAPK14 (p38a) | MAPK | CMGC | 2i0h | A | B | 2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dione | Human | 5009 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 1 | - | Human | 5021 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 10 | - | Human | 5063 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 2 | - | Human | 5093 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 3 | - | Human | 5040 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 4 | - | Human | 5067 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 5 | - | Human | 5107 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 6 | - | Human | 5219 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 7 | - | Human | 5161 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 8 | - | Human | 5078 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 9 | - | Human | 5127 | |
| MAPK14 (p38a) | MAPK | CMGC | 2npq | A | | - | Human | 5205 | |
| MAPK14 (p38a) | MAPK | CMGC | 2okr | A | | - | Human | 5136 | |
| MAPK14 (p38a) | MAPK | CMGC | 2okr | D | | - | Human | 5100 | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | A | | - | Human | 5177 | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | B | | - | Human | 5007 | |
| MAPK14 (p38a) | MAPK | CMGC | 2qd9 | A | | 1-[(3ar)-5-{[3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8h)-yl]carbonyl}-6-methoxy-3ah-pyrrolo[2,3-b]pyridin-3-yl]-2-[(3r)-3-hydroxypyrrolidin-1-yl]-2-oxoethanone | Human | 5197 | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg5 | A | | n-ethyl-4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5254 | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg6 | A | | 4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methyl-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5228 | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | A | - | Human | 5079 | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | B | - | Human | 5030 | |
| MAPK14 (p38a) | MAPK | CMGC | 2yis | A | | 1-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1h-pyrazol-5-yl]-3-{2-[(3-{2-[(2-hydroxyethyl)sulfanyl]phenyl}[1,2,4]triazolo[4,3-a]pyridin-6-yl)sulfanyl]benzyl}urea | Human | 5240 | |
| MAPK14 (p38a) | MAPK | CMGC | 2yiw | A | | 1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | 4988 | |
| MAPK14 (p38a) | MAPK | CMGC | 2yix | A | | 1-ethyl-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | 5143 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | A | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | 4980 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | B | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | 5034 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | A | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | 5099 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | B | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | 5147 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | A | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | 5038 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | B | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | 5103 | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv2 | A | | 5-methyl-4-[(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)amino]-n-(1-phenylethenyl)pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5191 | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv3 | A | | 5-methyl-4-[(2-methyl-5-{[(3-morpholin-4-ylphenyl)carbonyl]amino}phenyl)amino]-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5207 | |
| MAPK14 (p38a) | MAPK | CMGC | 3bx5 | A | | n-[2-methyl-5-(methylcarbamoyl)phenyl]-2-{[(1r)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamide | Human | 5000 | |
| MAPK14 (p38a) | MAPK | CMGC | 3c5u | A | | 6-[4-(2-fluorophenyl)-1,3-oxazol-5-yl]-n-(1-methylethyl)-1,3-benzothiazol-2-amine | Human | 5125 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ctq | A | | n-benzyl-1-[5-({5-tert-butyl-2-methoxy-3-[(methylsulfonyl)amino]phenyl}carbamoyl)-2-methylphenyl]-1h-1,2,3-triazole-4-carboxamide | Human | 5220 | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | A | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | 5247 | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | B | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | 5108 | |
| MAPK14 (p38a) | MAPK | CMGC | 3d83 | A | | n-{4'-[(cyclopropylmethyl)carbamoyl]-6-methylbiphenyl-3-yl}-2-morpholin-4-ylpyridine-4-carboxamide | Human | 5028 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | A | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5074 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | B | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5188 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | C | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5182 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | D | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5123 | |
| MAPK14 (p38a) | MAPK | CMGC | 3dt1 | A | | n-cyclopropyl-4-methyl-3-{2-[(2-morpholin-4-ylethyl)amino]quinazolin-6-yl}benzamide | Human | 5086 | |
| MAPK14 (p38a) | MAPK | CMGC | 3e92 | A | | n-cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamide | Human | 5149 | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | A | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | 5241 | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | B | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | 5004 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fc1 | X | | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 5110 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fi4 | A | | (2s)-1-{[3-(2-chlorophenyl)-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-ol | Human | 5051 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkl | A | | n-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-2h-pyran-4-ylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]benzamide | Human | 5172 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkn | A | | 3-[2-chloro-5-(methylsulfonyl)phenyl]-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidine | Human | 5049 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fko | A | | 3-(2-chlorophenyl)-6-(2-fluorophenoxy)-2h-indazole | Human | 5075 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fl4 | A | | 6-(2,4-difluorophenoxy)-3-(2-methylphenyl)-1h-pyrazolo[3,4-d]pyrimidine | Human | 5151 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fln | C | | 6-(2,4-difluorophenoxy)-8-methyl-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5090 | |
| MAPK14 (p38a) | MAPK | CMGC | 3flq | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5168 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fls | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5119 | |
| MAPK14 (p38a) | MAPK | CMGC | 3flw | A | | 6-(2,4-difluorophenoxy)-2-{[3-hydroxy-1-(2-hydroxyethyl)propyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5153 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fly | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-[(1-methylethyl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5113 | |
| MAPK14 (p38a) | MAPK | CMGC | 3flz | A | | 8-methyl-6-phenoxy-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5204 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmh | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5024 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmj | A | | 4-(5-methyl-3-phenylisoxazol-4-yl)pyrimidin-2-amine | Human | 5129 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmk | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5209 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fml | A | | 6-(2,4-difluorophenoxy)-n-[(1s)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 5010 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmm | A | | 6-(2,4-difluorophenoxy)-n-[(1r)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 5186 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmn | A | A | 6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 5196 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmn | A | B | 6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 4995 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fsf | A | | 3-(2,6-dichlorophenyl)-7-({4-[(diethylamino)methoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 5097 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fsk | A | | 3-(2-chlorophenyl)-7-[(trans-4-hydroxycyclohexyl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 5008 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gc7 | A | A | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 5061 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gc7 | A | B | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 5256 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcp | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5194 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcp | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5157 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcq | A | A | 1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5066 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcq | A | B | 1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5053 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcs | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5077 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcs | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5052 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | A | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5032 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | A | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5162 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | B | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5175 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | B | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5126 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcv | A | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5088 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcv | A | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5174 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gfe | A | | n-cyclopropyl-3-{[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-4-yl]amino}-4-methylbenzamide | Human | 4991 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gi3 | A | | n-{5-tert-butyl-2-methoxy-3-[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]naphthalen-1-yl}carbamoyl)amino]phenyl}methanesulfonamide | Human | 5226 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ha8 | A | A | n~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamide | Human | 5253 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ha8 | A | B | n~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamide | Human | 5187 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hec | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 5166 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hec | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 5035 | |
| MAPK14 (p38a) | MAPK | CMGC | 3heg | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5112 | |
| MAPK14 (p38a) | MAPK | CMGC | 3heg | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5218 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hl7 | A | | 2-{4-[5-(4-chlorophenyl)-4-pyrimidin-4-yl-1h-pyrazol-3-yl]piperidin-1-yl}-2-oxoethanol | Human | 5236 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hll | A | A | 3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamide | Human | 5115 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hll | A | B | 3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamide | Human | 5104 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp2 | A | A | 1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-one | Human | 5217 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp2 | A | B | 1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-one | Human | 5031 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp5 | A | | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 5158 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hrb | A | | [3-amino-2-(2-methylphenyl)-1-oxidopyridin-4-yl](2,4-difluorophenyl)methanone | Human | 5202 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hub | A | | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | 5029 | |
| MAPK14 (p38a) | MAPK | CMGC | 3huc | A | A | n-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamide | Human | 5027 | |
| MAPK14 (p38a) | MAPK | CMGC | 3huc | A | B | n-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamide | Human | 5111 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv3 | A | A | 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5012 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv3 | A | B | 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5232 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv4 | A | | 1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5121 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv4 | B | | 1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5064 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5203 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5263 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | B | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5085 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | B | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5137 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv6 | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(2-morpholin-4-ylethoxy)phenyl]urea | Human | 5101 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv7 | A | | 1-[1-(3-aminophenyl)-3-tert-butyl-1h-pyrazol-5-yl]-3-naphthalen-1-ylurea | Human | 5223 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hvc | A | | 4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridine | Human | 5054 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iph | A | A | 6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamide | Human | 4999 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iph | A | B | 6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamide | Human | 5156 | |
| MAPK14 (p38a) | MAPK | CMGC | 3itz | A | | 4-chloro-n-cyclopropyl-3-{[1-(2,6-difluorophenyl)-1h-pyrazolo[3,4-d]pyridazin-4-yl]amino}benzamide | Human | 5135 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw5 | A | | n-[2-(3-{[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl}-1h-indol-1-yl)ethyl]-3-(trifluoromethyl)benzamide | Human | 5076 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | A | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | 4990 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | B | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | 5154 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw7 | A | | 2-({4-[(4-benzylpiperidin-1-yl)carbonyl]benzyl}sulfanyl)-3h-imidazo[4,5-c]pyridine | Human | 5084 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw8 | A | | 1-{4-[(1s)-1-amino-2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-(3-chloro-4-fluorophenyl)urea | Human | 5181 | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | A | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | 5212 | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | B | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | 5022 | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3j | A | | 2-(4-fluorophenyl)-3-oxo-6-pyridin-4-yl-n-[2-(trifluoromethyl)benzyl]-2,3-dihydropyridazine-4-carboxamide | Human | 5047 | |
| MAPK14 (p38a) | MAPK | CMGC | 3kf7 | A | | 3-{6-[2-(2,4-difluorophenyl)ethyl][1,2,4]triazolo[4,3-a]pyridin-3-yl}-4-methylbenzamide | Human | 5201 | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | A | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | 5081 | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | B | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | 5057 | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8s | A | | 3-[(4-bromo-2,6-difluorobenzyl)oxy]-5-{[(4-pyrrolidin-1-ylbutyl)carbamoyl]amino}isothiazole-4-carboxamide | Human | 5055 | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8x | A | | n,4-dimethyl-3-[(1-phenyl-1h-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 5041 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfa | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 5018 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | 4998 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | 5001 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfc | A | | (4-{5-[({4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}carbamoyl)amino]-3-tert-butyl-1h-pyrazol-1-yl}phenyl)acetic acid | Human | 5160 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfd | A | | 1-{4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5102 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfe | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-4-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | 5173 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | A | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | 5140 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | B | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | 5120 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lhj | A | | n-cyclopropyl-3-[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamide | Human | 5234 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mgy | A | | - | Human | 5171 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh0 | A | | - | Human | 5124 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh1 | A | | - | Human | 5003 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh2 | A | | - | Human | 4985 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh3 | A | | - | Human | 5109 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpa | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5026 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | A | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | 5224 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | B | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | 5246 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | A | | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5060 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | B | | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5091 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | A | | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 4993 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | B | | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5210 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mw1 | A | | 8-(2,6-dichlorophenyl)-4-(2,4-difluorophenyl)-2-piperidin-4-yl-1,7-naphthyridine 7-oxide | Human | 5072 | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | A | - | Human | 5025 | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | B | - | Human | 5248 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | A | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | 5094 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | B | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | 5059 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | A | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | 5037 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | B | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | 5046 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | A | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | 5139 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | B | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | 5138 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnx | A | | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | 5002 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nww | A | | 1-[2-(2-{[2-(dimethylamino)ethyl]amino}-6-{2-[(1-methylethyl)amino]-1,3-thiazol-5-yl}pyrimidin-4-yl)benzyl]-3-ethylurea | Human | 5068 | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8p | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5071 | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8t | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5167 | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8u | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5250 | |
| MAPK14 (p38a) | MAPK | CMGC | 3obg | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5211 | |
| MAPK14 (p38a) | MAPK | CMGC | 3obj | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 4994 | |
| MAPK14 (p38a) | MAPK | CMGC | 3oc1 | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5019 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ocg | A | | 5-amino-n-[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]-1-phenyl-1h-pyrazole-4-carboxamide | Human | 4984 | |
| MAPK14 (p38a) | MAPK | CMGC | 3od6 | X | | - | Human | 5134 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ody | X | | - | Human | 5233 | |
| MAPK14 (p38a) | MAPK | CMGC | 3odz | X | | - | Human | 5069 | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | A | - | Human | 5163 | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | B | - | Human | 5231 | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | 5122 | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | 5096 | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | A | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | 5006 | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | B | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | 5262 | |
| MAPK14 (p38a) | MAPK | CMGC | 3que | A | | 2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-one | Human | 5095 | |
| MAPK14 (p38a) | MAPK | CMGC | 3rin | A | | n-cyclopropyl-4-methyl-3-(2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indol]-6'-yl)benzamide | Human | 5239 | |
| MAPK14 (p38a) | MAPK | CMGC | 3roc | A | | 3-{5-chloro-4-[(2,4-difluorobenzyl)oxy]-6-oxopyrimidin-1(6h)-yl}-n-(2-hydroxyethyl)-4-methylbenzamide | Human | 5011 | |
| MAPK14 (p38a) | MAPK | CMGC | 3s3i | A | | 3-(3-tert-butyl[1,2,4]triazolo[4,3-a]pyridin-7-yl)-n-cyclopropyl-4-methylbenzamide | Human | 5169 | |
| MAPK14 (p38a) | MAPK | CMGC | 3s4q | A | | 3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-n-cyclopropyl-4-methylbenzamide | Human | 5133 | |
| MAPK14 (p38a) | MAPK | CMGC | 3u8w | A | | 3-[3-(2-chloro-6-fluorophenyl)-5-ethyl-6-oxo-5,6-dihydro[1,2,4]triazolo[4,3-b]pyridazin-7-yl]-n-cyclopropyl-4-methylbenzamide | Human | 5192 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | A | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | 5070 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | B | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | 5155 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | A | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | 5183 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | B | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | 5214 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | 6880 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | 6879 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 4987 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 4977 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | A | tak-715 | Human | 5033 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | B | tak-715 | Human | 5098 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | A | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | 5216 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | B | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | 5118 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | A | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 5056 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | B | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 4983 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | A | 2-amino-phenylamino-dibenzosuberone | Human | 5105 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | B | 2-amino-phenylamino-dibenzosuberone | Human | 5089 | |
| MAPK14 (p38a) | MAPK | CMGC | 4a9y | A | | n-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamide | Human | 5073 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | A | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | 5213 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | B | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | 5132 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa4 | A | | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]furan-3-carboxamide | Human | 5045 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa5 | A | | n-cyclopropyl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]benzamide | Human | 5206 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aac | A | | n-isoxazol-3-yl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxo-quinazolin-3-yl]benzamide | Human | 5048 | |
| MAPK14 (p38a) | MAPK | CMGC | 4dli | A | | - | Human | 5092 | |
| MAPK14 (p38a) | MAPK | CMGC | 4dlj | A | | 2-phenyl-n~4~-(2-phenylethyl)quinazoline-4,7-diamine | Human | 5242 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | A | - | Human | 5189 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | B | - | Human | 5222 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5b | A | | - | Human | 5221 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6a | A | | - | Human | 5238 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6c | A | | - | Human | 5015 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e8a | A | | - | Human | 4979 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh2 | A | | 3-phenylquinazolin-4(3h)-one | Human | 5244 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh3 | A | | naringenin | Human | 5042 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh4 | A | | phenyl(piperidin-1-yl)methanone | Human | 5043 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh5 | A | | benzyl pyridine-3-carboxylate | Human | 5185 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh6 | A | | n-phenylpyridine-3-carboxamide | Human | 5083 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh7 | A | A | (3-phenoxyphenyl)methanol | Human | 5208 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh7 | A | B | (3-phenoxyphenyl)methanol | Human | 5020 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh8 | A | A | [3-(benzyloxy)phenyl]methanol | Human | 4978 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh8 | A | B | [3-(benzyloxy)phenyl]methanol | Human | 5014 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh9 | A | | - | Human | 4982 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ehv | A | A | - | Human | 4997 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ehv | A | B | - | Human | 4981 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ewq | A | A | 3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazine | Human | 5200 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ewq | A | B | 3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazine | Human | 5245 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9w | A | A | n,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5130 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9w | A | B | n,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5106 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9y | A | A | n,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5225 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9y | A | B | n,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5017 | |
| MAPK14 (p38a) | MAPK | CMGC | 4fa2 | A | A | trans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanol | Human | 5150 | |
| MAPK14 (p38a) | MAPK | CMGC | 4fa2 | A | B | trans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanol | Human | 5145 | |
| MAPK14 (p38a) | MAPK | CMGC | 4geo | A | | - | Human | 5190 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | A | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5237 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | B | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5131 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | C | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5142 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | D | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5144 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kip | A | | 2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamide | Human | 5159 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kip | B | | 2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamide | Human | 5180 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | A | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5141 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | B | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5013 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | C | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5215 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | D | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5016 | |
| MAPK14 (p38a) | MAPK | CMGC | 4l8m | A | A | n-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamide | Human | 5005 | |
| MAPK14 (p38a) | MAPK | CMGC | 4l8m | A | B | n-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamide | Human | 4992 | |
| MAPK14 (p38a) | MAPK | CMGC | 4r3c | A | A | 6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine | Human | 5198 | |
| MAPK14 (p38a) | MAPK | CMGC | 4r3c | A | B | 6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine | Human | 5036 | |
| MAPK14 (p38a) | MAPK | CMGC | 4zth | A | A | 6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazine | Human | 6706 | |
| MAPK14 (p38a) | MAPK | CMGC | 4zth | A | B | 6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazine | Human | 6707 | |
| MAPK14 (p38a) | MAPK | CMGC | 5eta | A | | - | Human | 7136 | |
| MAPK14 (p38a) | MAPK | CMGC | 5eta | B | | - | Human | 7137 | |
| MAPK14 (p38a) | MAPK | CMGC | 5etc | A | | - | Human | 6361 | |
| MAPK14 (p38a) | MAPK | CMGC | 5etf | A | A | - | Human | 7134 | |
| MAPK14 (p38a) | MAPK | CMGC | 5etf | A | B | - | Human | 7135 | |
| MAPK14 (p38a) | MAPK | CMGC | 5eti | A | | - | Human | 6362 | |
| MAPK14 (p38a) | MAPK | CMGC | 5ml5 | A | | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-methylsulfanyl-1~{h}-imidazol-5-yl]pyridin-2-yl]propanamide | Human | 7544 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mtx | A | A | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamide | Human | 8382 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mtx | A | B | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamide | Human | 8379 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mty | A | | ~{n}-[2,4-bis(fluoranyl)-5-[[14-(2-hydroxyethylcarbamoyl)-2-oxidanylidene-6-tricyclo[9.4.0.0^{3,8}]pentadeca-1(15),3(8),4,6,11,13-hexaenyl]amino]phenyl]thiophene-2-carboxamide | Human | 8383 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mz3 | A | A | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | 8680 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mz3 | A | B | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | 8681 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n63 | A | | - | Human | 8526 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n64 | A | | - | Human | 8527 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n65 | A | | 2-phenyl-~{n}4-(2-thiophen-2-ylethyl)quinazoline-4,7-diamine | Human | 8525 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n66 | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 8524 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n67 | A | A | - | Human | 8523 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n67 | A | B | - | Human | 8521 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n68 | A | | - | Human | 8522 | |
| MAPK14 (p38a) | MAPK | CMGC | 5o8u | A | | - | Human | 8381 | |
| MAPK14 (p38a) | MAPK | CMGC | 5o8v | A | | - | Human | 8380 | |
| MAPK14 (p38a) | MAPK | CMGC | 5omg | A | A | 3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | 11246 | |
| MAPK14 (p38a) | MAPK | CMGC | 5omg | A | B | 3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | 11245 | |
| MAPK14 (p38a) | MAPK | CMGC | 5omh | A | | 1-(3-chlorophenyl)-3-methyl-4~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | 11251 | |
| MAPK14 (p38a) | MAPK | CMGC | 5tbe | A | | ~{n}-[2,4-bis(fluoranyl)-5-[[9-(2-morpholin-4-ylethylcarbamoyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulen-3-yl]amino]phenyl]thiophene-2-carboxamide | Human | 8032 | |
| MAPK14 (p38a) | MAPK | CMGC | 5tco | A | | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulene-9-carboxamide | Human | 8031 | |
| MAPK14 (p38a) | MAPK | CMGC | 5wjj | A | A | n-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamide | Human | 9514 | |
| MAPK14 (p38a) | MAPK | CMGC | 5wjj | A | B | n-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamide | Human | 9516 | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyx | A | A | n-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amine | Human | 9519 | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyx | A | B | n-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amine | Human | 9517 | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyy | A | | 3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-4h-1,2,4-triazol-3-yl)phenol | Human | 9513 | |
| MAPK14 (p38a) | MAPK | CMGC | 6anl | A | A | tak-715 | Human | 9515 | |
| MAPK14 (p38a) | MAPK | CMGC | 6anl | A | B | tak-715 | Human | 9518 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwt | A | A | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamide | Human | 11248 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwt | A | B | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamide | Human | 11254 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwu | A | A | - | Human | 11247 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwu | A | B | - | Human | 11249 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwv | A | A | - | Human | 11253 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwv | A | B | - | Human | 11250 | |
| MAPK14 (p38a) | MAPK | CMGC | 6m95 | A | | (4-benzylpiperidin-1-yl)[2-methoxy-4-(methylsulfanyl)phenyl]methanone | Human | 11252 | |
| MAPK14 (p38a) | MAPK | CMGC | 6m9l | A | | 3-benzyl-6-[(2,4-difluorophenyl)amino]-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-one | Human | 11255 | |
| MAPK14 (p38a) | MAPK | CMGC | 6ohd | A | A | 3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamide | Human | 11818 | |
| MAPK14 (p38a) | MAPK | CMGC | 6ohd | A | B | 3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamide | Human | 11819 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qdz | A | A | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | 11956 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qdz | A | B | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | 11958 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qe1 | A | | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{r})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | 11957 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qyx | A | | - | Human | 12127 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfi | A | A | ~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamide | Human | 11613 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfi | A | B | ~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamide | Human | 11619 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | A | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | 11614 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | B | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | 11616 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | C | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | 11618 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfk | A | A | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | Human | 11617 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfk | A | B | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | Human | 11620 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfo | A | A | 5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 11615 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfo | A | B | 5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 11621 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | B | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12491 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | B | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12488 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | D | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12486 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | D | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12492 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | F | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12489 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | F | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12490 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | H | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12493 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | H | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12487 | |
| MAPK14 (p38a) | MAPK | CMGC | 6zqs | A | | 2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-one | Human | 12986 | |
| MAPK14 (p38a) | MAPK | CMGC | 6zwp | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 12699 | |
| MAPK14 (p38a) | MAPK | CMGC | 6zwp | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 12698 | |
| MAPK14 (p38a) | MAPK | CMGC | 8a8m | A | | phosphomethylphosphonic acid adenosyl ester | Human | 14289 | |
| MAPK3 (Erk1) | MAPK | CMGC | 2zoq | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 1716 | |
| MAPK3 (Erk1) | MAPK | CMGC | 2zoq | B | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 1712 | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 1714 | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 1713 | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | B | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 1717 | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | B | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 1715 | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | A | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10923 | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | A | B | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10926 | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | B | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10925 | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | B | B | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10924 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | A | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12788 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | A | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12790 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | B | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12792 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | B | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12786 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | C | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12787 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | C | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12784 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | D | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12796 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | D | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12789 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | A | | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | 12791 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | B | | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | 12797 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | C | | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | 12794 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | D | | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | 12795 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yll | A | | ~{n}4-[3-(4-methoxyphenyl)-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]cyclohexane-1,4-diamine | Human | 12793 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yll | B | | - | Human | 12785 | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | A | A | - | Human | 12982 | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | A | B | - | Human | 12981 | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | B | A | - | Human | 12980 | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | B | B | - | Human | 12983 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4b99 | A | | 11-cyclopentyl-2-[[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl-phenyl]amino]-5-methyl-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 388 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic7 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 392 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic7 | D | | phosphoaminophosphonic acid-adenylate ester | Human | 391 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic8 | A | | - | Human | 390 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic8 | B | | - | Human | 389 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsg | A | A | 3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | 6589 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsg | A | B | 3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | 6584 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsj | A | A | 3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | 6588 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsj | A | B | 3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | 6585 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsl | A | | 3-amino-5-[(4-chlorophenyl)amino]-n-[(1s)-1-phenylethyl]-1h-1,2,4-triazole-1-carboxamide | Human | 6586 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byy | A | A | 2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 6591 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byy | A | B | 2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 6587 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byz | A | A | 4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamide | Human | 6590 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byz | A | B | 4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamide | Human | 6592 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5o7i | A | A | 4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamide | Human | 9995 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5o7i | A | B | 4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamide | Human | 9994 | |
| MAPK7 (Erk5) | MAPK | CMGC | 6hkm | A | | [4-(6,7-dimethoxyquinazolin-4-yl)piperidin-1-yl]-[4-(trifluoromethyloxy)phenyl]methanone | Human | 10917 | |
| MAPK7 (Erk5) | MAPK | CMGC | 6hkn | A | A | [2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanone | Human | 10918 | |
| MAPK7 (Erk5) | MAPK | CMGC | 6hkn | A | B | [2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanone | Human | 10919 | |
| MAPK7 (Erk5) | MAPK | CMGC | 7pus | A | A | 4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamide | Human | 14218 | |
| MAPK7 (Erk5) | MAPK | CMGC | 7pus | A | B | 4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamide | Human | 14219 | |
| MAPK8 (JNK1) | MAPK | CMGC | 1ukh | A | | - | Human | 4628 | |
| MAPK8 (JNK1) | MAPK | CMGC | 1uki | A | | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | 4630 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2g01 | A | | 6-chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4h-pyrazolo[3,4-b]quinolin-4-one | Human | 4662 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2g01 | B | | 6-chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4h-pyrazolo[3,4-b]quinolin-4-one | Human | 4641 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2gmx | A | | n-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-bromo-2,5-dimethoxyphenyl)acetamide | Human | 4674 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2gmx | B | | n-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-bromo-2,5-dimethoxyphenyl)acetamide | Human | 4638 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2h96 | A | | 5-cyano-n-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamide | Human | 4655 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2h96 | B | | 5-cyano-n-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamide | Human | 4668 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2no3 | A | | 2-({2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}amino)benzamide | Human | 4640 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2no3 | B | | 2-({2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}amino)benzamide | Human | 4657 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2xrw | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 4675 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2xrw | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 4650 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2xrw | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 4660 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2xs0 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 4629 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3elj | A | A | 2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide | Human | 4658 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3elj | A | B | 2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide | Human | 4636 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3o17 | A | | - | Human | 4670 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3o17 | B | | - | Human | 4667 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3o2m | A | | - | Human | 4676 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3o2m | B | | - | Human | 4649 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3pze | A | | 3-(carbamoylamino)-5-phenylthiophene-2-carboxamide | Human | 4642 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3v3v | A | | 3,5,6,7-tetrahydroxy-2-(3,4-dihydroxyphenyl)-4h-chromen-4-one | Human | 4653 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vud | A | | - | Human | 4664 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vug | A | | - | Human | 4665 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vuh | A | | - | Human | 4663 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vui | A | | - | Human | 4652 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vuk | A | | - | Human | 4659 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vul | A | | - | Human | 4633 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vum | A | | - | Human | 4671 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4awi | A | A | n-(1,1-dioxidotetrahydro-2h-thiopyran-4-yl)-4-[2-(1-methylethyl)-1h-pyrrolo[2,3-b]pyridin-4-yl]benzenesulfonamide | Human | 4661 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4awi | A | B | n-(1,1-dioxidotetrahydro-2h-thiopyran-4-yl)-4-[2-(1-methylethyl)-1h-pyrrolo[2,3-b]pyridin-4-yl]benzenesulfonamide | Human | 4634 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4e73 | A | A | methyl 3-(4-{[(1r,2s,3s,5s,7s)-5-aminotricyclo[3.3.1.1~3,7~]dec-2-yl]carbamoyl}benzyl)-4-oxo-1-phenyl-1,4-dihydro-1,8-naphthyridine-2-carboxylate | Human | 4645 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4e73 | A | B | methyl 3-(4-{[(1r,2s,3s,5s,7s)-5-aminotricyclo[3.3.1.1~3,7~]dec-2-yl]carbamoyl}benzyl)-4-oxo-1-phenyl-1,4-dihydro-1,8-naphthyridine-2-carboxylate | Human | 4669 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4g1w | A | | methyl 7-fluoro-3-{4-[(2-hydroxyethyl)sulfonyl]benzyl}-4-oxo-1-phenyl-1,4-dihydroquinoline-2-carboxylate | Human | 4631 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4hys | A | | trans-4-{[4-(1h-indazol-1-yl)pyrimidin-2-yl]amino}cyclohexanol | Human | 4672 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4hyu | A | | trans-4-[(4-{4-[3-(methylsulfonyl)propoxy]-1h-indazol-1-yl}pyrimidin-2-yl)amino]cyclohexanol | Human | 4632 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4izy | A | | trans-4-[(4-{4-[4-(methylsulfonyl)piperidin-1-yl]-1h-indol-1-yl}pyrimidin-2-yl)amino]cyclohexanol | Human | 4654 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4l7f | A | A | n-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamide | Human | 4639 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4l7f | A | B | n-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamide | Human | 4637 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4l7f | A | C | n-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamide | Human | 4648 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4qtd | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 4651 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4qtd | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 4673 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 4643 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 4646 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 4635 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 4656 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 4644 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 4647 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 4627 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 4666 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | A | A | - | Human | 6452 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | A | B | - | Human | 6448 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | C | A | - | Human | 6449 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | C | B | - | Human | 6447 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | E | A | - | Human | 6451 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | E | B | - | Human | 6454 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | F | A | - | Human | 6450 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | F | B | - | Human | 6453 | |
| MAPK8 (JNK1) | MAPK | CMGC | 5lw1 | B | | adenosine | Human | 9081 | |
| MAPK8 (JNK1) | MAPK | CMGC | 5lw1 | E | | adenosine | Human | 9079 | |
| MAPK8 (JNK1) | MAPK | CMGC | 5lw1 | H | | adenosine | Human | 9080 | |
| MAPK8 (JNK1) | MAPK | CMGC | 6f5e | B | | - | Human | 9078 | |
| MAPK8 (JNK1) | MAPK | CMGC | 6zr5 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 12984 | |
| MAPK8 (JNK1) | MAPK | CMGC | 6zr5 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12985 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8pt8 | A | | - | Human | 15295 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8pt9 | A | | - | Human | 15293 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8pta | A | | - | Human | 15294 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8x5m | A | A | 3-[4-(dimethylamino)butanoylamino]-~{n}-[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide | Human | 15099 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8x5m | A | B | 3-[4-(dimethylamino)butanoylamino]-~{n}-[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide | Human | 15100 | |
| MAPK9 (JNK2) | MAPK | CMGC | 3e7o | A | | n-{3-[5-(1h-1,2,4-triazol-3-yl)-1h-indazol-3-yl]phenyl}furan-2-carboxamide | Human | 1238 | |
| MAPK9 (JNK2) | MAPK | CMGC | 3e7o | B | | n-{3-[5-(1h-1,2,4-triazol-3-yl)-1h-indazol-3-yl]phenyl}furan-2-carboxamide | Human | 1236 | |
| MAPK9 (JNK2) | MAPK | CMGC | 3npc | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 1235 | |
| MAPK9 (JNK2) | MAPK | CMGC | 3npc | B | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 1237 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7cml | A | A | - | Human | 12707 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7cml | A | B | - | Human | 12705 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7cml | B | A | - | Human | 12706 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7cml | B | B | - | Human | 12704 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7n8t | A | A | adenosine monophosphate | Human | 14241 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7n8t | A | B | adenosine monophosphate | Human | 14242 | |
| MAPK9 (JNK2) | MAPK | CMGC | 8elc | A | | 4-(dimethylamino)-n-{4-[(3s)-3-({4-[(8r)-2-phenylpyrazolo[1,5-a]pyridin-3-yl]pyrimidin-2-yl}amino)pyrrolidine-1-carbonyl]phenyl}butanamide | Human | 14816 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1kwp | A | | - | Human | 1280 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1kwp | B | | - | Human | 1296 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1nxk | A | | staurosporine | Human | 1342 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1nxk | B | | staurosporine | Human | 1292 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1nxk | C | | staurosporine | Human | 1312 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1nxk | D | | staurosporine | Human | 1334 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1ny3 | A | | adenosine-5'-diphosphate | Human | 1318 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbo | A | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1333 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | A | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1366 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | B | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1320 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | C | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1344 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | D | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1327 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | E | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1358 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | F | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1335 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | G | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1339 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | H | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1326 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | I | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1364 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | J | | - | Human | 1359 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | K | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1363 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | L | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1283 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2onl | C | | - | Human | 1306 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2onl | D | | - | Human | 1345 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2oza | A | | - | Human | 1310 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2p3g | X | | 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1349 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2pzy | A | | (4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamide | Human | 1314 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2pzy | B | | (4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamide | Human | 1307 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2pzy | C | | staurosporine | Human | 1279 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2pzy | D | | - | Human | 1357 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | A | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1330 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | B | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1332 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | C | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1328 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | D | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1316 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | E | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1315 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | F | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1355 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | G | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1343 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | H | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1325 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | I | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1311 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | J | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1353 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | K | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1360 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | L | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1301 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3fpm | A | | 3-{[(1r)-1-phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dione | Human | 1367 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3fyj | X | | (10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one | Human | 1336 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3fyk | X | | (3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-one | Human | 1297 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | A | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1281 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | B | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1304 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | C | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1350 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | D | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1284 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | E | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1300 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | F | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1362 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | G | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1351 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | H | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1338 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | I | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1305 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | J | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1319 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | K | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1299 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | L | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1365 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3ka0 | A | | 6-{5-[(2-aminopyrimidin-4-yl)amino]-2-hydroxyphenyl}-n-methylidene-1-benzothiophene-2-carboxamide | Human | 1290 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | A | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1289 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | B | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1298 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | C | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1303 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | D | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1288 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | E | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1285 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | F | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1341 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | G | | - | Human | 1356 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | H | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1291 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | I | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1354 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | J | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1347 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | K | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1317 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | L | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1324 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kga | A | A | 6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-one | Human | 9476 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kga | A | B | 6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-one | Human | 9477 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3m2w | A | A | 2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-one | Human | 9474 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3m2w | A | B | 2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-one | Human | 9473 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3m42 | A | | 2-[5-(2-methoxyethoxy)pyridin-3-yl]-8,9,10,11-tetrahydro-7h-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin-7-one | Human | 9475 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | A | | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | 1287 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | B | | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | 1329 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | C | | - | Human | 1368 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | D | | - | Human | 1337 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | E | | - | Human | 1286 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | F | | - | Human | 1321 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | G | | - | Human | 1369 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | H | | - | Human | 1348 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | I | | - | Human | 1294 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | J | | - | Human | 1331 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | K | | - | Human | 1293 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | L | | - | Human | 1295 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2y | A | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1361 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r30 | A | A | 1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acid | Human | 1352 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r30 | A | B | 1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acid | Human | 1309 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | A | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1308 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | B | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1282 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | C | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1346 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | D | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1340 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | E | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1323 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | F | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1313 | |
| MAPKAPK2 | MAPKAPK | CAMK | 4tyh | A | A | - | Human | 1302 | |
| MAPKAPK2 | MAPKAPK | CAMK | 4tyh | A | B | - | Human | 1322 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6t8x | A | | (10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one | Human | 13548 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | A | A | - | Human | 12502 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | A | B | - | Human | 12507 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | C | A | - | Human | 12504 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | C | B | - | Human | 12506 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | E | A | - | Human | 12500 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | E | B | - | Human | 12503 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | G | A | - | Human | 12505 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | G | B | - | Human | 12501 | |
| MAPKAPK2 | MAPKAPK | CAMK | 8xu4 | A | | - | Human | 15173 | |
| MAPKAPK2 | MAPKAPK | CAMK | 8xx1 | A | A | - | Human | 15257 | |
| MAPKAPK2 | MAPKAPK | CAMK | 8xx1 | A | B | - | Human | 15256 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3fhr | A | A | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4590 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3fhr | A | B | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4598 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3fxw | A | A | 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4596 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3fxw | A | B | 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4593 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3r1n | A | A | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | 4589 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3r1n | A | B | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | 4588 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3she | A | A | n-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamide | Human | 4594 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3she | A | B | n-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamide | Human | 4599 | |
| MAPKAPK3 | MAPKAPK | CAMK | 7nrb | A | A | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 14052 | |
| MAPKAPK3 | MAPKAPK | CAMK | 7nrb | A | B | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 14051 | |
| MARK1 | CAMKL | CAMK | 2hak | A | | - | Human | 258 | |
| MARK1 | CAMKL | CAMK | 2hak | B | | - | Human | 259 | |
| MARK1 | CAMKL | CAMK | 2hak | C | | - | Human | 260 | |
| MARK1 | CAMKL | CAMK | 2hak | D | | - | Human | 257 | |
| MARK1 | CAMKL | CAMK | 2hak | E | | - | Human | 255 | |
| MARK1 | CAMKL | CAMK | 2hak | F | | - | Human | 254 | |
| MARK1 | CAMKL | CAMK | 2hak | G | | - | Human | 256 | |
| MARK1 | CAMKL | CAMK | 2hak | H | | - | Human | 261 | |
| MARK1 | CAMKL | CAMK | 6c9d | A | A | - | Human | 10052 | |
| MARK1 | CAMKL | CAMK | 6c9d | A | B | - | Human | 10051 | |
| MARK1 | CAMKL | CAMK | 6c9d | B | A | - | Human | 10049 | |
| MARK1 | CAMKL | CAMK | 6c9d | B | B | - | Human | 10050 | |
| MARK2 | CAMKL | CAMK | 3iec | A | | - | Human | 3045 | |
| MARK2 | CAMKL | CAMK | 3iec | B | | - | Human | 3044 | |
| MARK2 | CAMKL | CAMK | 3iec | C | | - | Human | 3046 | |
| MARK2 | CAMKL | CAMK | 3iec | D | | - | Human | 3043 | |
| MARK2 | CAMKL | CAMK | 5eak | A | | n-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide | Human | 6410 | |
| MARK2 | CAMKL | CAMK | 5eak | B | | n-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide | Human | 6411 | |
| MARK2 | CAMKL | CAMK | 5kz7 | A | | 7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-one | Human | 7967 | |
| MARK2 | CAMKL | CAMK | 5kz7 | B | | 7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-one | Human | 7966 | |
| MARK2 | CAMKL | CAMK | 5kz8 | A | | 5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-one | Human | 7965 | |
| MARK2 | CAMKL | CAMK | 5kz8 | B | | 5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-one | Human | 7968 | |
| MARK2 | CAMKL | CAMK | 8txy | A | | n-[(5p,8r)-5-(2-cyano-5-{[(3r)-1-methylpyrrolidin-3-yl]methoxy}pyridin-4-yl)pyrazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide | Human | 15136 | |
| MARK3 | CAMKL | CAMK | 2qnj | A | | - | Human | 3269 | |
| MARK3 | CAMKL | CAMK | 2qnj | B | | - | Human | 3264 | |
| MARK3 | CAMKL | CAMK | 3fe3 | A | A | - | Human | 3267 | |
| MARK3 | CAMKL | CAMK | 3fe3 | A | B | - | Human | 3266 | |
| MARK3 | CAMKL | CAMK | 3fe3 | B | A | - | Human | 3268 | |
| MARK3 | CAMKL | CAMK | 3fe3 | B | B | - | Human | 3265 | |
| MARK3 | CAMKL | CAMK | 7p1l | A | | 5-bromo-4-n-[2-(1h-imidazol-5-yl)ethyl]-2-n-[3-(morpholin-4-ylmethyl)phenyl]pyrimidine-2,4-diamine | Human | 13799 | |
| MARK4 | CAMKL | CAMK | 5es1 | A | | ~{n}-[(1~{r},6~{r})-6-azanyl-2,2-bis(fluoranyl)cyclohexyl]-5-ethyl-4-[6-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide | Human | 6260 | |
| MARK4 | CAMKL | CAMK | 8xfl | A | | - | Human | 15101 | |
| MASTL | MAST | AGC | 5loh | A | A | staurosporine | Human | 7086 | |
| MASTL | MAST | AGC | 5loh | A | B | staurosporine | Human | 7085 | |
| MASTL | MAST | AGC | 5loh | B | A | staurosporine | Human | 7088 | |
| MASTL | MAST | AGC | 5loh | B | B | staurosporine | Human | 7087 | |
| Melk (MELK) | CAMKL | CAMK | 4bfm | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5798 | |
| Melk (MELK) | CAMKL | CAMK | 4cqg | A | | 1-[6-(3,5-dichloro-4-hydroxyphenyl)-4-({trans-4-[(dimethylamino)methyl]cyclohexyl}amino)-1,5-naphthyridin-3-yl]ethanone | Mouse | 6865 | |
| MELK | CAMKL | CAMK | 4bky | A | A | 3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamide | Human | 2480 | |
| MELK | CAMKL | CAMK | 4bky | A | B | 3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamide | Human | 2490 | |
| MELK | CAMKL | CAMK | 4bkz | A | A | n-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 2505 | |
| MELK | CAMKL | CAMK | 4bkz | A | B | n-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 2484 | |
| MELK | CAMKL | CAMK | 4bl1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2514 | |
| MELK | CAMKL | CAMK | 4bl1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2519 | |
| MELK | CAMKL | CAMK | 4d2p | A | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2513 | |
| MELK | CAMKL | CAMK | 4d2p | A | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2499 | |
| MELK | CAMKL | CAMK | 4d2p | B | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2494 | |
| MELK | CAMKL | CAMK | 4d2p | B | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2498 | |
| MELK | CAMKL | CAMK | 4d2p | C | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2496 | |
| MELK | CAMKL | CAMK | 4d2p | C | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2501 | |
| MELK | CAMKL | CAMK | 4d2p | D | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2486 | |
| MELK | CAMKL | CAMK | 4d2p | D | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2518 | |
| MELK | CAMKL | CAMK | 4d2t | A | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2487 | |
| MELK | CAMKL | CAMK | 4d2t | A | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2489 | |
| MELK | CAMKL | CAMK | 4d2t | B | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2520 | |
| MELK | CAMKL | CAMK | 4d2t | B | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2512 | |
| MELK | CAMKL | CAMK | 4d2t | C | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2491 | |
| MELK | CAMKL | CAMK | 4d2t | C | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2526 | |
| MELK | CAMKL | CAMK | 4d2t | D | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2530 | |
| MELK | CAMKL | CAMK | 4d2t | D | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2511 | |
| MELK | CAMKL | CAMK | 4d2v | A | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2493 | |
| MELK | CAMKL | CAMK | 4d2v | A | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2522 | |
| MELK | CAMKL | CAMK | 4d2v | B | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2483 | |
| MELK | CAMKL | CAMK | 4d2v | B | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2507 | |
| MELK | CAMKL | CAMK | 4d2v | C | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2529 | |
| MELK | CAMKL | CAMK | 4d2v | C | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2492 | |
| MELK | CAMKL | CAMK | 4d2v | D | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2502 | |
| MELK | CAMKL | CAMK | 4d2v | D | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2506 | |
| MELK | CAMKL | CAMK | 4d2w | A | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2515 | |
| MELK | CAMKL | CAMK | 4d2w | A | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2509 | |
| MELK | CAMKL | CAMK | 4d2w | B | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2500 | |
| MELK | CAMKL | CAMK | 4d2w | B | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2482 | |
| MELK | CAMKL | CAMK | 4d2w | C | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2527 | |
| MELK | CAMKL | CAMK | 4d2w | C | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2503 | |
| MELK | CAMKL | CAMK | 4d2w | D | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2481 | |
| MELK | CAMKL | CAMK | 4d2w | D | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2495 | |
| MELK | CAMKL | CAMK | 4ixp | A | | - | Human | 2528 | |
| MELK | CAMKL | CAMK | 4ump | A | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2497 | |
| MELK | CAMKL | CAMK | 4ump | A | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2485 | |
| MELK | CAMKL | CAMK | 4ump | B | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2524 | |
| MELK | CAMKL | CAMK | 4ump | B | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2504 | |
| MELK | CAMKL | CAMK | 4ump | C | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2479 | |
| MELK | CAMKL | CAMK | 4ump | C | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2508 | |
| MELK | CAMKL | CAMK | 4ump | D | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2516 | |
| MELK | CAMKL | CAMK | 4ump | D | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2525 | |
| MELK | CAMKL | CAMK | 4umq | A | A | 3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminium | Human | 2488 | |
| MELK | CAMKL | CAMK | 4umq | A | B | 3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminium | Human | 2523 | |
| MELK | CAMKL | CAMK | 4umr | A | | 4-fluoro-n-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamide | Human | 2521 | |
| MELK | CAMKL | CAMK | 4umt | A | | 1-(4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}-2-methoxybenzyl)piperazinediium | Human | 2510 | |
| MELK | CAMKL | CAMK | 4umu | A | | (2-ethoxy-4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}phenyl)methanaminium | Human | 2517 | |
| MELK | CAMKL | CAMK | 5ih8 | A | | n-[(pyridin-2-yl)methyl]-4-[4-(pyridin-4-yl)-1h-pyrazol-1-yl]benzamide | Human | 6661 | |
| MELK | CAMKL | CAMK | 5ih9 | A | A | 1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazine | Human | 6659 | |
| MELK | CAMKL | CAMK | 5ih9 | A | B | 1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazine | Human | 6657 | |
| MELK | CAMKL | CAMK | 5iha | A | A | 1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazine | Human | 6663 | |
| MELK | CAMKL | CAMK | 5iha | A | B | 1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazine | Human | 6658 | |
| MELK | CAMKL | CAMK | 5ihc | A | A | 4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridine | Human | 6660 | |
| MELK | CAMKL | CAMK | 5ihc | A | B | 4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridine | Human | 6662 | |
| MELK | CAMKL | CAMK | 5k00 | A | A | 4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamide | Human | 7497 | |
| MELK | CAMKL | CAMK | 5k00 | A | B | 4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamide | Human | 7498 | |
| MELK | CAMKL | CAMK | 5m5a | A | A | k-252a | Human | 8735 | |
| MELK | CAMKL | CAMK | 5m5a | A | B | k-252a | Human | 8733 | |
| MELK | CAMKL | CAMK | 5maf | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 8732 | |
| MELK | CAMKL | CAMK | 5mag | A | A | pf-3758309 | Human | 8736 | |
| MELK | CAMKL | CAMK | 5mag | A | B | pf-3758309 | Human | 8731 | |
| MELK | CAMKL | CAMK | 5mah | A | A | ~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide | Human | 8729 | |
| MELK | CAMKL | CAMK | 5mah | A | B | ~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide | Human | 8734 | |
| MELK | CAMKL | CAMK | 5mai | A | A | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 8728 | |
| MELK | CAMKL | CAMK | 5mai | A | B | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 8730 | |
| MELK | CAMKL | CAMK | 5tvt | A | | 9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3-methyl-3,4-dihydropyrimido[5,4-c][1,5]naphthyridin-2(1h)-one | Human | 8667 | |
| MELK | CAMKL | CAMK | 5twl | A | | 9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3,4-dihydropyrimido[5,4-c]quinolin-2(1h)-one | Human | 8668 | |
| MELK | CAMKL | CAMK | 5twu | A | | - | Human | 8670 | |
| MELK | CAMKL | CAMK | 5twu | B | | - | Human | 8672 | |
| MELK | CAMKL | CAMK | 5twy | A | | 2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 8671 | |
| MELK | CAMKL | CAMK | 5twy | B | | 2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 8669 | |
| MELK | CAMKL | CAMK | 5twz | A | | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 8675 | |
| MELK | CAMKL | CAMK | 5tx3 | A | | 7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-one | Human | 8673 | |
| MELK | CAMKL | CAMK | 5tx3 | B | | 7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-one | Human | 8674 | |
| MELK | CAMKL | CAMK | 6gvx | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11137 | |
| MELK | CAMKL | CAMK | 6gvx | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11139 | |
| MELK | CAMKL | CAMK | 6gvx | B | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11136 | |
| MELK | CAMKL | CAMK | 6gvx | B | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11138 | |
| MELK | CAMKL | CAMK | 6vxr | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 12645 | |
| MELK | CAMKL | CAMK | 6vxr | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 12644 | |
| MERTK (MER) | Axl | TK | 2p0c | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 286 | |
| MERTK (MER) | Axl | TK | 2p0c | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 287 | |
| MERTK (MER) | Axl | TK | 2p0c | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 271 | |
| MERTK (MER) | Axl | TK | 2p0c | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 280 | |
| MERTK (MER) | Axl | TK | 3bpr | A | A | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 278 | |
| MERTK (MER) | Axl | TK | 3bpr | A | B | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 263 | |
| MERTK (MER) | Axl | TK | 3bpr | B | A | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 281 | |
| MERTK (MER) | Axl | TK | 3bpr | B | B | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 275 | |
| MERTK (MER) | Axl | TK | 3bpr | C | A | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 284 | |
| MERTK (MER) | Axl | TK | 3bpr | C | B | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 276 | |
| MERTK (MER) | Axl | TK | 3bpr | D | A | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 279 | |
| MERTK (MER) | Axl | TK | 3bpr | D | B | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 282 | |
| MERTK (MER) | Axl | TK | 3brb | A | A | adenosine-5'-diphosphate | Human | 266 | |
| MERTK (MER) | Axl | TK | 3brb | A | B | adenosine-5'-diphosphate | Human | 273 | |
| MERTK (MER) | Axl | TK | 3brb | B | A | adenosine-5'-diphosphate | Human | 267 | |
| MERTK (MER) | Axl | TK | 3brb | B | B | adenosine-5'-diphosphate | Human | 274 | |
| MERTK (MER) | Axl | TK | 3tcp | A | | 1-[(trans-4-aminocyclohexyl)methyl]-n-butyl-3-(4-fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-6-amine | Human | 272 | |
| MERTK (MER) | Axl | TK | 3tcp | B | | 1-[(trans-4-aminocyclohexyl)methyl]-n-butyl-3-(4-fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-6-amine | Human | 285 | |
| MERTK (MER) | Axl | TK | 4m3q | A | | trans-4-{[2-(butylamino)-5-(pyridin-2-yl)pyrimidin-4-yl]amino}cyclohexanol | Human | 283 | |
| MERTK (MER) | Axl | TK | 4m3q | B | | trans-4-{[2-(butylamino)-5-(pyridin-2-yl)pyrimidin-4-yl]amino}cyclohexanol | Human | 269 | |
| MERTK (MER) | Axl | TK | 4mh7 | A | | n-butyl-2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-methylpyrimidine-5-carboxamide | Human | 262 | |
| MERTK (MER) | Axl | TK | 4mh7 | B | | - | Human | 265 | |
| MERTK (MER) | Axl | TK | 4mha | A | A | 2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-(4-sulfamoylbenzyl)pyrimidine-5-carboxamide | Human | 264 | |
| MERTK (MER) | Axl | TK | 4mha | A | B | 2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-(4-sulfamoylbenzyl)pyrimidine-5-carboxamide | Human | 277 | |
| MERTK (MER) | Axl | TK | 4mha | B | A | 2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-(4-sulfamoylbenzyl)pyrimidine-5-carboxamide | Human | 268 | |
| MERTK (MER) | Axl | TK | 4mha | B | B | 2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-(4-sulfamoylbenzyl)pyrimidine-5-carboxamide | Human | 270 | |
| MERTK (MER) | Axl | TK | 5k0k | A | A | 15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-one | Human | 7345 | |
| MERTK (MER) | Axl | TK | 5k0k | A | B | 15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-one | Human | 7347 | |
| MERTK (MER) | Axl | TK | 5k0k | B | A | 15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-one | Human | 7348 | |
| MERTK (MER) | Axl | TK | 5k0k | B | B | 15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-one | Human | 7346 | |
| MERTK (MER) | Axl | TK | 5k0x | A | A | (7s)-7-amino-n-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamide | Human | 7433 | |
| MERTK (MER) | Axl | TK | 5k0x | A | B | (7s)-7-amino-n-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamide | Human | 7432 | |
| MERTK (MER) | Axl | TK | 5k0x | B | A | (7s)-7-amino-n-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamide | Human | 7434 | |
| MERTK (MER) | Axl | TK | 5k0x | B | B | (7s)-7-amino-n-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamide | Human | 7431 | |
| MERTK (MER) | Axl | TK | 5tc0 | A | | n-(2-{4-[(2s)-4-(methylsulfonyl)morpholin-2-yl]-1,3-thiazol-2-yl}phenyl)-1h-imidazole-2-carboxamide | Human | 7383 | |
| MERTK (MER) | Axl | TK | 5tc0 | B | | - | Human | 7381 | |
| MERTK (MER) | Axl | TK | 5td2 | A | A | n-[2-{4-[(2s)-4-(methylsulfonyl)morpholin-2-yl]-1,3-thiazol-2-yl}-4-(morpholin-4-yl)phenyl]-1h-imidazole-2-carboxamide | Human | 7384 | |
| MERTK (MER) | Axl | TK | 5td2 | A | B | n-[2-{4-[(2s)-4-(methylsulfonyl)morpholin-2-yl]-1,3-thiazol-2-yl}-4-(morpholin-4-yl)phenyl]-1h-imidazole-2-carboxamide | Human | 7380 | |
| MERTK (MER) | Axl | TK | 5td2 | B | A | - | Human | 7385 | |
| MERTK (MER) | Axl | TK | 5td2 | B | B | - | Human | 7382 | |
| MERTK (MER) | Axl | TK | 5u6c | A | A | (10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 8251 | |
| MERTK (MER) | Axl | TK | 5u6c | A | B | (10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 8253 | |
| MERTK (MER) | Axl | TK | 5u6c | B | A | (10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 8250 | |
| MERTK (MER) | Axl | TK | 5u6c | B | B | (10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-one | Human | 8252 | |
| MERTK (MER) | Axl | TK | 6mep | A | | cis-4-[(2-[(4-{[4-(1,3-dioxolan-2-yl)pyridin-2-yl]ethynyl}phenyl)amino]-5-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}pyrimidin-4-yl)amino]cyclohexan-1-ol | Human | 11602 | |
| MERTK (MER) | Axl | TK | 6mep | B | | cis-4-[(2-[(4-{[4-(1,3-dioxolan-2-yl)pyridin-2-yl]ethynyl}phenyl)amino]-5-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}pyrimidin-4-yl)amino]cyclohexan-1-ol | Human | 11601 | |
| MERTK (MER) | Axl | TK | 7aax | A | A | ~{n}-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluoranyl-phenyl]-4-ethoxy-1-(4-fluoranyl-2-methyl-phenyl)pyrazole-3-carboxamide | Human | 12938 | |
| MERTK (MER) | Axl | TK | 7aax | A | B | ~{n}-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluoranyl-phenyl]-4-ethoxy-1-(4-fluoranyl-2-methyl-phenyl)pyrazole-3-carboxamide | Human | 12941 | |
| MERTK (MER) | Axl | TK | 7aay | A | A | n-(3-fluoro-4-{[1-methyl-6-(1h-pyrazol-4-yl)-1h-indazol-5-yl]oxy}phenyl)-1-(4-fluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 12940 | |
| MERTK (MER) | Axl | TK | 7aay | A | B | n-(3-fluoro-4-{[1-methyl-6-(1h-pyrazol-4-yl)-1h-indazol-5-yl]oxy}phenyl)-1-(4-fluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 12935 | |
| MERTK (MER) | Axl | TK | 7aaz | A | A | 2-azanyl-~{n}-[(1~{s},2~{s})-2-[[4-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]phenyl]methoxy]cyclopentyl]-5-(1-methylpyrazol-4-yl)pyridine-3-carboxamide | Human | 12962 | |
| MERTK (MER) | Axl | TK | 7aaz | A | B | 2-azanyl-~{n}-[(1~{s},2~{s})-2-[[4-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]phenyl]methoxy]cyclopentyl]-5-(1-methylpyrazol-4-yl)pyridine-3-carboxamide | Human | 12964 | |
| MERTK (MER) | Axl | TK | 7ab0 | A | A | - | Human | 12937 | |
| MERTK (MER) | Axl | TK | 7ab0 | A | B | - | Human | 12939 | |
| MERTK (MER) | Axl | TK | 7ab1 | A | | 6-ethyl-3-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-5-(oxan-4-ylamino)pyrazine-2-carboxamide | Human | 12933 | |
| MERTK (MER) | Axl | TK | 7ab2 | A | A | 4-[2-(butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | Human | 12934 | |
| MERTK (MER) | Axl | TK | 7ab2 | A | B | 4-[2-(butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | Human | 12936 | |
| MERTK (MER) | Axl | TK | 7avx | A | | 1-(4-fluorophenyl)-n-[3-fluoro-4-[(3-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)oxy]phenyl]-2,3-dimethyl-5-oxopyrazole-4-carboxamide | Human | 13372 | |
| MERTK (MER) | Axl | TK | 7avx | B | | 1-(4-fluorophenyl)-n-[3-fluoro-4-[(3-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)oxy]phenyl]-2,3-dimethyl-5-oxopyrazole-4-carboxamide | Human | 13375 | |
| MERTK (MER) | Axl | TK | 7avy | A | | n-(2-(2-cyclopropylethoxy)pyrimidin-5-yl)-7-methoxy-6-(piperidin-4-ylmethoxy)quinazolin-4-amine | Human | 13369 | |
| MERTK (MER) | Axl | TK | 7avz | A | | (r)-n2-(4-(cyclopropylmethoxy)-3,5-difluorophenyl)-5-(3-methylpiperazin-1-yl)-n4-(tetrahydro-2h-pyran-4-yl)pyrimidine-2,4-diamine | Human | 13370 | |
| MERTK (MER) | Axl | TK | 7aw0 | A | | 2-(cyclopentyloxy)-9-(2,6-difluorobenzyl)-n-methyl-9h-purin-6-amine | Human | 13373 | |
| MERTK (MER) | Axl | TK | 7aw1 | A | | n-(6-(4-(3-(4-((5,6-dihydroimidazo[1,2-a]pyrazin-7(8h)-yl)methyl)-3-(trifluoromethyl)phenyl)ureido)phenoxy)pyrimidin-4-yl)cyclopropanecarboxamide | Human | 13366 | |
| MERTK (MER) | Axl | TK | 7aw2 | A | | 5-(2'-chloro-[1,1'-biphenyl]-4-yl)-n-(imidazo[1,2-a]pyridin-6-ylmethyl)-n-methyl-1,3,4-oxadiazol-2-amine | Human | 13377 | |
| MERTK (MER) | Axl | TK | 7aw3 | A | | 2-(1-((5-chloro-1h-pyrrolo[2,3-b]pyridine-3-carboxamido)methyl)-2-azabicyclo[2.1.1]hexan-2-yl)-n-methyl-4-(trifluoromethyl)thiazole-5-carboxamide | Human | 13367 | |
| MERTK (MER) | Axl | TK | 7aw4 | A | A | 3-methyl-5-(4-methyl-1,2,3-thiadiazol-5-yl)-n-((r)-1-(((r)-3-(methylamino)-3-oxo-1-(4-(trifluoromethyl)phenyl)propyl)amino)-1-oxo-4-phenylbutan-2-yl)isoxazole-4-carboxamide | Human | 13374 | |
| MERTK (MER) | Axl | TK | 7aw4 | A | B | 3-methyl-5-(4-methyl-1,2,3-thiadiazol-5-yl)-n-((r)-1-(((r)-3-(methylamino)-3-oxo-1-(4-(trifluoromethyl)phenyl)propyl)amino)-1-oxo-4-phenylbutan-2-yl)isoxazole-4-carboxamide | Human | 13371 | |
| MERTK (MER) | Axl | TK | 7aw4 | B | A | 3-methyl-5-(4-methyl-1,2,3-thiadiazol-5-yl)-n-((r)-1-(((r)-3-(methylamino)-3-oxo-1-(4-(trifluoromethyl)phenyl)propyl)amino)-1-oxo-4-phenylbutan-2-yl)isoxazole-4-carboxamide | Human | 13376 | |
| MERTK (MER) | Axl | TK | 7aw4 | B | B | 3-methyl-5-(4-methyl-1,2,3-thiadiazol-5-yl)-n-((r)-1-(((r)-3-(methylamino)-3-oxo-1-(4-(trifluoromethyl)phenyl)propyl)amino)-1-oxo-4-phenylbutan-2-yl)isoxazole-4-carboxamide | Human | 13368 | |
| MERTK (MER) | Axl | TK | 7cqe | A | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 12963 | |
| MERTK (MER) | Axl | TK | 7cqe | C | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 12965 | |
| MERTK (MER) | Axl | TK | 7dxl | A | | 3-[4-[6-chloranyl-5-[[(3r)-pyrrolidin-3-yl]amino]-1h-indazol-3-yl]pyrazol-1-yl]benzenecarbonitrile | Human | 13941 | |
| MERTK (MER) | Axl | TK | 7m5z | A | A | 2-(butylamino)-n-[1-(3-fluoropropyl)piperidin-4-yl]-4-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyrimidine-5-carboxamide | Human | 13919 | |
| MERTK (MER) | Axl | TK | 7m5z | A | B | 2-(butylamino)-n-[1-(3-fluoropropyl)piperidin-4-yl]-4-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyrimidine-5-carboxamide | Human | 13920 | |
| MERTK (MER) | Axl | TK | 7oam | A | | - | Human | 13556 | |
| MERTK (MER) | Axl | TK | 7ols | A | | 5-[4-(1,5-dimethylpyrazol-4-yl)-2-methyl-phenyl]-~{n}-(imidazo[1,2-a]pyridin-6-ylmethyl)-~{n}-methyl-1,3,4-oxadiazol-2-amine | Human | 13899 | |
| MERTK (MER) | Axl | TK | 7olv | A | | 4-[4-[5-[imidazo[1,2-a]pyridin-6-ylmethyl(methyl)amino]-1,3,4-oxadiazol-2-yl]-3-methyl-phenyl]-2,5-dimethyl-pyrazole-3-carbonitrile | Human | 13898 | |
| MERTK (MER) | Axl | TK | 7olx | A | | ~{n}-[[3-[4-[(dimethylamino)methyl]phenyl]imidazo[1,2-a]pyridin-6-yl]methyl]-~{n}-methyl-5-[3-methyl-5-(1,3,5-trimethylpyrazol-4-yl)pyridin-2-yl]-1,3,4-oxadiazol-2-amine | Human | 13897 | |
| MERTK (MER) | Axl | TK | 7xhy | A | | ~{n}-[4-(2-azanyl-3-chloranyl-pyridin-4-yl)oxy-3-fluoranyl-phenyl]-5-(4-fluorophenyl)-4-oxidanylidene-1~{h}-pyridine-3-carboxamide | Human | 14517 | |
| MET | Met | TK | 1r0p | A | | k-252a | Human | 2991 | |
| MET | Met | TK | 1r1w | A | | - | Human | 3014 | |
| MET | Met | TK | 2g15 | A | | - | Human | 2983 | |
| MET | Met | TK | 2rfn | A | | 2-benzyl-5-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-3-methylpyrimidin-4(3h)-one | Human | 3022 | |
| MET | Met | TK | 2rfn | B | | 2-benzyl-5-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-3-methylpyrimidin-4(3h)-one | Human | 2961 | |
| MET | Met | TK | 2rfs | A | | n-(3-chlorophenyl)-n-methyl-2-oxo-3-[(3,4,5-trimethyl-1h-pyrrol-2-yl)methyl]-2h-indole-5-sulfonamide | Human | 2974 | |
| MET | Met | TK | 2wd1 | A | A | 1-[(2-nitrophenyl)sulfonyl]-1h-pyrrolo[3,2-b]pyridine-6-carboxamide | Human | 3032 | |
| MET | Met | TK | 2wd1 | A | B | 1-[(2-nitrophenyl)sulfonyl]-1h-pyrrolo[3,2-b]pyridine-6-carboxamide | Human | 2976 | |
| MET | Met | TK | 2wgj | A | | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 3009 | |
| MET | Met | TK | 2wkm | A | | (3z)-5-[(2,6-dichlorobenzyl)sulfonyl]-3-[(3,5-dimethyl-4-{[(2s)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]carbonyl}-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3021 | |
| MET | Met | TK | 3a4p | A | | (2e)-3-{6-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]quinolin-3-yl}-n-methylprop-2-enamide | Human | 3005 | |
| MET | Met | TK | 3c1x | A | | n-{[4-({5-[(4-aminopiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}oxy)-3-fluorophenyl]carbamoyl}-2-(4-fluorophenyl)acetamide | Human | 3020 | |
| MET | Met | TK | 3ccn | A | | 4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methyl]phenol | Human | 2971 | |
| MET | Met | TK | 3cd8 | A | A | 7-methoxy-4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy]quinoline | Human | 3008 | |
| MET | Met | TK | 3cd8 | A | B | 7-methoxy-4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy]quinoline | Human | 2995 | |
| MET | Met | TK | 3ce3 | A | | 1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 6769 | |
| MET | Met | TK | 3cth | A | | n-({4-[(2-aminopyridin-4-yl)oxy]-3-fluorophenyl}carbamoyl)-2-(4-fluorophenyl)acetamide | Human | 6768 | |
| MET | Met | TK | 3ctj | A | A | 2-(4-fluorophenyl)-n-{[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]carbamoyl}acetamide | Human | 6767 | |
| MET | Met | TK | 3ctj | A | B | 2-(4-fluorophenyl)-n-{[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]carbamoyl}acetamide | Human | 6766 | |
| MET | Met | TK | 3dkc | A | A | adenosine-5'-triphosphate | Human | 2997 | |
| MET | Met | TK | 3dkc | A | B | adenosine-5'-triphosphate | Human | 2952 | |
| MET | Met | TK | 3dkf | A | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 3030 | |
| MET | Met | TK | 3dkf | A | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 3029 | |
| MET | Met | TK | 3dkf | A | C | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 2984 | |
| MET | Met | TK | 3dkg | A | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 2993 | |
| MET | Met | TK | 3dkg | A | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 3019 | |
| MET | Met | TK | 3dkg | A | C | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 3006 | |
| MET | Met | TK | 3efj | A | | 2-benzyl-5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-3-methylpyrimidin-4(3h)-one | Human | 3015 | |
| MET | Met | TK | 3efj | B | | 2-benzyl-5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-3-methylpyrimidin-4(3h)-one | Human | 2957 | |
| MET | Met | TK | 3efk | A | | 5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-2-[(4-fluorophenyl)amino]-3-methylpyrimidin-4(3h)-one | Human | 3018 | |
| MET | Met | TK | 3efk | B | | 5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-2-[(4-fluorophenyl)amino]-3-methylpyrimidin-4(3h)-one | Human | 2988 | |
| MET | Met | TK | 3f66 | A | A | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | 2989 | |
| MET | Met | TK | 3f66 | A | B | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | 3027 | |
| MET | Met | TK | 3f66 | A | C | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | 3011 | |
| MET | Met | TK | 3f66 | A | D | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | 3026 | |
| MET | Met | TK | 3f66 | B | A | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | 3034 | |
| MET | Met | TK | 3f66 | B | B | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | 2992 | |
| MET | Met | TK | 3f66 | B | C | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | 2966 | |
| MET | Met | TK | 3f66 | B | D | 3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenol | Human | 3000 | |
| MET | Met | TK | 3f82 | A | | n-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorophenyl}-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 2977 | |
| MET | Met | TK | 3i5n | A | | 7-methoxy-n-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methyl]-1,5-naphthyridin-4-amine | Human | 3013 | |
| MET | Met | TK | 3l8v | A | | 2-({4-[(2-aminopyridin-4-yl)oxy]-3-fluorophenyl}amino)-n-(2,4-difluorophenyl)pyridine-3-carboxamide | Human | 2978 | |
| MET | Met | TK | 3lq8 | A | A | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 2998 | |
| MET | Met | TK | 3lq8 | A | B | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 2964 | |
| MET | Met | TK | 3q6u | A | A | - | Human | 2954 | |
| MET | Met | TK | 3q6u | A | B | - | Human | 2962 | |
| MET | Met | TK | 3q6w | A | | 3-{5-oxo-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-5h-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl}-n-(pyridin-2-ylmethyl)propanamide | Human | 2969 | |
| MET | Met | TK | 3qti | A | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | 2994 | |
| MET | Met | TK | 3qti | A | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | 3028 | |
| MET | Met | TK | 3qti | B | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | 3017 | |
| MET | Met | TK | 3qti | B | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | 3024 | |
| MET | Met | TK | 3r7o | A | | n-[(2r)-1,4-dioxan-2-ylmethyl]-n-methyl-n'-{5-oxo-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-5h-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl}sulfuric diamide | Human | 3038 | |
| MET | Met | TK | 3rhk | A | | 1-[(3r,4r)-4-(1h-indol-3-yl)-2,5-dioxopyrrolidin-3-yl]pyrrolo[3,2,1-ij]quinolinium | Human | 2979 | |
| MET | Met | TK | 3rhk | B | | 1-[(3r,4r)-4-(1h-indol-3-yl)-2,5-dioxopyrrolidin-3-yl]pyrrolo[3,2,1-ij]quinolinium | Human | 2959 | |
| MET | Met | TK | 3u6h | A | A | n-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamide | Human | 2996 | |
| MET | Met | TK | 3u6h | A | B | n-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamide | Human | 2965 | |
| MET | Met | TK | 3u6i | A | | n-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-1-[(2r)-2-hydroxypropyl]-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamide | Human | 2967 | |
| MET | Met | TK | 3vw8 | A | | n-({4-[(6,7-dimethoxyquinolin-4-yl)oxy]phenyl}carbamothioyl)-2-phenylacetamide | Human | 2985 | |
| MET | Met | TK | 3zbx | A | | 6-[[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinoline | Human | 3036 | |
| MET | Met | TK | 3zc5 | A | | 6-{(1s)-1-[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]ethyl}quinoline | Human | 3003 | |
| MET | Met | TK | 3zcl | A | | (s)-3-(1-(1h-pyrrolo(2,3-b)pyridin-3-yl)ethyl)-n-isopropyl-(1,2,4)triazolo(4,3-b)pyridazin-6-amine | Human | 2990 | |
| MET | Met | TK | 3zxz | A | | 2-{4-[1-(quinolin-6-ylmethyl)-1h-[1,2,3]triazolo[4,5-b]pyrazin-6-yl]-1h-pyrazol-1-yl}ethanol | Human | 2999 | |
| MET | Met | TK | 3zze | A | | (2s)-n'-[(3r)-4-chloro-7-methyl-2-oxo-2,3-dihydro-1h-indol-3-yl]-2-(4-hydroxyphenyl)propanehydrazide | Human | 2980 | |
| MET | Met | TK | 4aoi | A | | 4-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-6-yl]benzenecarbonitrile | Human | 2958 | |
| MET | Met | TK | 4ap7 | A | | 4-[[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]phenol | Human | 3035 | |
| MET | Met | TK | 4deg | A | | 7-methoxy-n-{[6-(3-methyl-1,2-thiazol-5-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]methyl}-1,5-naphthyridin-4-amine | Human | 2981 | |
| MET | Met | TK | 4deh | A | | 5-phenyl-3-(quinolin-6-ylmethyl)-3,5,6,7-tetrahydro-4h-[1,2,3]triazolo[4,5-c]pyridin-4-one | Human | 2963 | |
| MET | Met | TK | 4dei | A | | 3-{(1s)-1-[3-(2-methoxyethoxy)quinolin-6-yl]ethyl}-5-(3-methyl-1,2-thiazol-5-yl)-3,5-dihydro-4h-[1,2,3]triazolo[4,5-c]pyridin-4-one | Human | 3016 | |
| MET | Met | TK | 4eev | A | A | n-(3-fluoro-4-{[1-methyl-6-(1h-pyrazol-4-yl)-1h-indazol-5-yl]oxy}phenyl)-1-(4-fluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 3012 | |
| MET | Met | TK | 4eev | A | B | n-(3-fluoro-4-{[1-methyl-6-(1h-pyrazol-4-yl)-1h-indazol-5-yl]oxy}phenyl)-1-(4-fluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 3023 | |
| MET | Met | TK | 4gg5 | A | A | 3-(4-methylpiperazin-1-yl)-n-(3-nitrobenzyl)-7-(trifluoromethyl)quinolin-5-amine | Human | 2956 | |
| MET | Met | TK | 4gg5 | A | B | 3-(4-methylpiperazin-1-yl)-n-(3-nitrobenzyl)-7-(trifluoromethyl)quinolin-5-amine | Human | 2953 | |
| MET | Met | TK | 4gg7 | A | A | n-(3-nitrobenzyl)-6-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine | Human | 3002 | |
| MET | Met | TK | 4gg7 | A | B | n-(3-nitrobenzyl)-6-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine | Human | 2987 | |
| MET | Met | TK | 4iwd | A | | 1-{5-oxo-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-5h-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl}-n-(pyridin-2-ylmethyl)methanesulfonamide | Human | 2975 | |
| MET | Met | TK | 4knb | A | A | 7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amine | Human | 2960 | |
| MET | Met | TK | 4knb | A | B | 7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amine | Human | 3037 | |
| MET | Met | TK | 4knb | B | A | 7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amine | Human | 3007 | |
| MET | Met | TK | 4knb | B | B | 7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amine | Human | 2970 | |
| MET | Met | TK | 4knb | C | A | 7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amine | Human | 2955 | |
| MET | Met | TK | 4knb | C | B | 7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amine | Human | 3001 | |
| MET | Met | TK | 4knb | D | A | 7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amine | Human | 3010 | |
| MET | Met | TK | 4knb | D | B | 7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amine | Human | 2968 | |
| MET | Met | TK | 4mxc | A | A | n-(3-fluoro-4-{[2-({3-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 3033 | |
| MET | Met | TK | 4mxc | A | B | n-(3-fluoro-4-{[2-({3-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 3025 | |
| MET | Met | TK | 4r1v | A | A | 3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrile | Human | 3004 | |
| MET | Met | TK | 4r1v | A | B | 3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrile | Human | 2972 | |
| MET | Met | TK | 4r1y | A | | 3-(diethylamino)propyl (3-{[5-(3,4-dimethoxyphenyl)-2-oxo-2h-1,3,4-thiadiazin-3(6h)-yl]methyl}phenyl)carbamate | Human | 2973 | |
| MET | Met | TK | 4xmo | A | | 6-{(1r)-1-fluoro-1-[8-fluoro-6-(3-methyl-1,2-oxazol-5-yl)[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl}-3-methoxyquinoline | Human | 3031 | |
| MET | Met | TK | 4xyf | A | A | 6-{(1s)-1-[8-fluoro-6-(3-methyl-1,2-oxazol-5-yl)[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl}-3-(2-methoxyethoxy)quinoline | Human | 2986 | |
| MET | Met | TK | 4xyf | A | B | 6-{(1s)-1-[8-fluoro-6-(3-methyl-1,2-oxazol-5-yl)[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl}-3-(2-methoxyethoxy)quinoline | Human | 2982 | |
| MET | Met | TK | 5dg5 | A | A | n-(2,5-difluoro-4-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 7037 | |
| MET | Met | TK | 5dg5 | A | B | n-(2,5-difluoro-4-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 7034 | |
| MET | Met | TK | 5dg5 | B | A | n-(2,5-difluoro-4-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 7035 | |
| MET | Met | TK | 5dg5 | B | B | n-(2,5-difluoro-4-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 7036 | |
| MET | Met | TK | 5eob | A | A | 6-[bis(fluoranyl)-[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinoline | Human | 7100 | |
| MET | Met | TK | 5eob | A | B | 6-[bis(fluoranyl)-[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinoline | Human | 7101 | |
| MET | Met | TK | 5eyc | A | A | 6-[(1~{r})-1-[8-fluoranyl-6-(3-methyl-1,2-oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl]-1,6-naphthyridin-5-one | Human | 6401 | |
| MET | Met | TK | 5eyc | A | B | 6-[(1~{r})-1-[8-fluoranyl-6-(3-methyl-1,2-oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl]-1,6-naphthyridin-5-one | Human | 6400 | |
| MET | Met | TK | 5eyd | A | A | 6-[(1~{r})-1-[8-fluoranyl-6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl]-3-(2-methoxyethoxy)-1,6-naphthyridin-5-one | Human | 6402 | |
| MET | Met | TK | 5eyd | A | B | 6-[(1~{r})-1-[8-fluoranyl-6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl]-3-(2-methoxyethoxy)-1,6-naphthyridin-5-one | Human | 6399 | |
| MET | Met | TK | 5hlw | A | | 1-[2-(1-ethylpiperidin-4-yl)ethyl]-3-(6-{[6-(thiophen-2-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1,3-benzothiazol-2-yl)urea | Human | 7275 | |
| MET | Met | TK | 5hni | X | | methyl (6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1h-benzimidazol-2-yl)carbamate | Human | 7280 | |
| MET | Met | TK | 5hni | Y | | methyl (6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1h-benzimidazol-2-yl)carbamate | Human | 7278 | |
| MET | Met | TK | 5ho6 | A | | 1-(6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1,3-benzothiazol-2-yl)-3-[2-(morpholin-4-yl)ethyl]urea | Human | 7277 | |
| MET | Met | TK | 5hoa | A | | 1-(6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1,3-benzothiazol-2-yl)-3-[2-(morpholin-4-yl)ethyl]urea | Human | 7279 | |
| MET | Met | TK | 5hor | A | | 1-(6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1,3-benzothiazol-2-yl)-3-[2-(morpholin-4-yl)ethyl]urea | Human | 7276 | |
| MET | Met | TK | 5hti | A | A | n-[3-fluoro-4-({7-[2-(morpholin-4-yl)ethoxy]-1,6-naphthyridin-4-yl}oxy)phenyl]-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 8010 | |
| MET | Met | TK | 5hti | A | B | n-[3-fluoro-4-({7-[2-(morpholin-4-yl)ethoxy]-1,6-naphthyridin-4-yl}oxy)phenyl]-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 8009 | |
| MET | Met | TK | 5t3q | A | | n-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-1-(2-hydroxy-2-methylpropyl)-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamide | Human | 7413 | |
| MET | Met | TK | 5uab | A | A | n-{6-[([1,2,4]triazolo[4,3-a]pyridin-3-yl)sulfanyl]imidazo[1,2-b]pyridazin-2-yl}cyclopropanecarboxamide | Human | 7961 | |
| MET | Met | TK | 5uab | A | B | n-{6-[([1,2,4]triazolo[4,3-a]pyridin-3-yl)sulfanyl]imidazo[1,2-b]pyridazin-2-yl}cyclopropanecarboxamide | Human | 7964 | |
| MET | Met | TK | 5uad | A | | n-(6-{[6-(1-methyl-1h-pyrazol-4-yl)-1h-benzotriazol-1-yl]methyl}imidazo[1,2-b]pyridazin-2-yl)cyclopropanecarboxamide | Human | 7963 | |
| MET | Met | TK | 5ya5 | A | A | 2-[3-(4-methoxybenzyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1h-indole | Human | 10040 | |
| MET | Met | TK | 5ya5 | A | B | 2-[3-(4-methoxybenzyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1h-indole | Human | 10039 | |
| MET | Met | TK | 6sd9 | A | | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 11531 | |
| MET | Met | TK | 6sdc | A | A | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 11532 | |
| MET | Met | TK | 6sdc | A | B | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 11534 | |
| MET | Met | TK | 6sdd | A | | n-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorophenyl}-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 11533 | |
| MET | Met | TK | 6sde | A | | volitinib | Human | 11535 | |
| MET | Met | TK | 6ubw | A | | n-(6-{difluoro[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-a]pyridin-3-yl]methyl}imidazo[1,2-b]pyridazin-2-yl)cyclopropanecarboxamide | Human | 11979 | |
| MET | Met | TK | 7b3q | A | A | 1-(phenylmethyl)-5~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 13177 | |
| MET | Met | TK | 7b3q | A | B | 1-(phenylmethyl)-5~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 13182 | |
| MET | Met | TK | 7b3t | A | A | 3-(phenylmethyl)-1~{h}-pyrrolo[2,3-b]pyridine | Human | 13183 | |
| MET | Met | TK | 7b3t | A | B | 3-(phenylmethyl)-1~{h}-pyrrolo[2,3-b]pyridine | Human | 13191 | |
| MET | Met | TK | 7b3v | A | A | 3-(3-methyl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)-1~{h}-pyrrolo[3,4-b]pyrrol-6-one | Human | 13188 | |
| MET | Met | TK | 7b3v | A | B | 3-(3-methyl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)-1~{h}-pyrrolo[3,4-b]pyrrol-6-one | Human | 13194 | |
| MET | Met | TK | 7b3w | A | A | 3-(6-fluoranyl-1~{h}-indazol-4-yl)-4,5-dihydro-1~{h}-pyrrolo[3,4-b]pyrrol-6-one | Human | 13180 | |
| MET | Met | TK | 7b3w | A | B | 3-(6-fluoranyl-1~{h}-indazol-4-yl)-4,5-dihydro-1~{h}-pyrrolo[3,4-b]pyrrol-6-one | Human | 13178 | |
| MET | Met | TK | 7b3z | A | A | 3-[3-(phenylmethyl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-4,5-dihydro-1~{h}-pyrrolo[3,4-b]pyrrol-6-one | Human | 13181 | |
| MET | Met | TK | 7b3z | A | B | 3-[3-(phenylmethyl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-4,5-dihydro-1~{h}-pyrrolo[3,4-b]pyrrol-6-one | Human | 13186 | |
| MET | Met | TK | 7b40 | A | | 3-(phenylmethyl)-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridine | Human | 13192 | |
| MET | Met | TK | 7b41 | A | A | 3-[(2-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridine | Human | 13184 | |
| MET | Met | TK | 7b41 | A | B | 3-[(2-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridine | Human | 13193 | |
| MET | Met | TK | 7b42 | A | | 3-[(3-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridine | Human | 13190 | |
| MET | Met | TK | 7b43 | A | | 3-[(4-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridine | Human | 13189 | |
| MET | Met | TK | 7b43 | B | | 3-[(4-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridine | Human | 13187 | |
| MET | Met | TK | 7b44 | A | A | 5-methoxy-1~{h}-indazole | Human | 13185 | |
| MET | Met | TK | 7b44 | A | B | 5-methoxy-1~{h}-indazole | Human | 13179 | |
| MET | Met | TK | 7v3r | A | A | ~{n}1'-[3-fluoranyl-4-(2-phenylazanylpyrimidin-4-yl)oxy-phenyl]-~{n}1-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 14328 | |
| MET | Met | TK | 7v3r | A | B | ~{n}1'-[3-fluoranyl-4-(2-phenylazanylpyrimidin-4-yl)oxy-phenyl]-~{n}1-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 14330 | |
| MET | Met | TK | 7v3s | A | A | ~{n}1'-[3-fluoranyl-4-(10~{h}-pyrido[3,2-b][1,4]benzoxazin-4-yloxy)phenyl]-~{n}1-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 14329 | |
| MET | Met | TK | 7v3s | A | B | ~{n}1'-[3-fluoranyl-4-(10~{h}-pyrido[3,2-b][1,4]benzoxazin-4-yloxy)phenyl]-~{n}1-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 14327 | |
| MET | Met | TK | 7y4t | A | | 2-[2-[3-(1-methylpyrazol-4-yl)quinolin-6-yl]ethyl]-6-(3-nitrophenyl)pyridazin-3-one | Human | 14548 | |
| MET | Met | TK | 7y4u | A | | ~{n}-methyl-4-[1-[2-[3-(1-methylpyrazol-4-yl)quinolin-6-yl]ethyl]-6-oxidanylidene-pyridazin-3-yl]-2-(trifluoromethyl)benzamide | Human | 14550 | |
| MET | Met | TK | 8an8 | A | | 3-[bis(fluoranyl)methyl]-~{n}-methyl-~{n}-[(1~{r})-8-methyl-5-(3-methyl-1~{h}-indazol-6-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]pyridine-2-carboxamide | Human | 14355 | |
| MET | Met | TK | 8ans | A | | 3-[bis(fluoranyl)methyl]-~{n}-methyl-~{n}-[(1~{r})-8-methyl-5-(3-methyl-1~{h}-indazol-6-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]pyridine-2-carboxamide | Human | 14356 | |
| MET | Met | TK | 8au3 | A | | 3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrile | Human | 14982 | |
| MET | Met | TK | 8au5 | A | | 3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrile | Human | 14983 | |
| MET | Met | TK | 8aw1 | A | A | 3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrile | Human | 14981 | |
| MET | Met | TK | 8aw1 | A | B | 3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrile | Human | 14980 | |
| MET | Met | TK | 8gvj | A | | (1^4z,5^2e)-6^3-(trifluoromethyl)-5^1,5^6-dihydro-1^1h-8-aza-2(3,6)-quinolina-5(1,3)-pyridazina-1(4,1)-pyrazola-6(1,4)-benzenacyclododecaphane-5^6,7-dione | Human | 14549 | |
| MET | Met | TK | 8k78 | A | A | - | Human | 15352 | |
| MET | Met | TK | 8k78 | A | B | - | Human | 15351 | |
| MET | Met | TK | 8ouu | A | A | 5-(3-ethynyl-5-fluoranyl-1h-indazol-7-yl)-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dione | Human | 14821 | |
| MET | Met | TK | 8ouu | A | B | 5-(3-ethynyl-5-fluoranyl-1h-indazol-7-yl)-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dione | Human | 14824 | |
| MET | Met | TK | 8ouv | A | A | 5-(1h-indazol-7-yl)-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dione | Human | 14820 | |
| MET | Met | TK | 8ouv | A | B | 5-(1h-indazol-7-yl)-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dione | Human | 14823 | |
| MET | Met | TK | 8ov7 | A | | 5-[3,5-bis(fluoranyl)phenyl]-1-[(1s)-1-[3-(1h-imidazol-5-yl)phenyl]ethyl]pyrimidine-2,4-dione | Human | 14817 | |
| MET | Met | TK | 8ovz | A | | 1-[(1s)-1-[3-(1h-imidazol-4-yl)phenyl]ethyl]-5-(1h-indazol-7-yl)pyrimidine-2,4-dione | Human | 14822 | |
| MET | Met | TK | 8ow3 | A | | 5-[3,5-bis(fluoranyl)phenyl]-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dione | Human | 14818 | |
| MET | Met | TK | 8owg | A | | 5-[3,5-bis(fluoranyl)phenyl]-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dione | Human | 14819 | |
| MET | Met | TK | 9c1r | A | A | n-(2,5-difluoro-4-{[(1s,3s)-3-(1-methyl-1h-pyrazol-3-yl)cyclobutyl][(8r)-pyrazolo[1,5-a]pyrazin-4-yl]amino}phenyl)-2-(5-fluoropyridin-2-yl)-3-oxo-2,3-dihydropyridazine-4-carboxamide | Human | 15368 | |
| MET | Met | TK | 9c1r | A | B | n-(2,5-difluoro-4-{[(1s,3s)-3-(1-methyl-1h-pyrazol-3-yl)cyclobutyl][(8r)-pyrazolo[1,5-a]pyrazin-4-yl]amino}phenyl)-2-(5-fluoropyridin-2-yl)-3-oxo-2,3-dihydropyridazine-4-carboxamide | Human | 15369 | |
| MKNK1 (MNK1) | MAPKAPK | CAMK | 2hw6 | A | | - | Human | 2084 | |
| MKNK1 (MNK1) | MAPKAPK | CAMK | 2hw6 | B | | - | Human | 2085 | |
| MKNK1 (MNK1) | MAPKAPK | CAMK | 5wvd | A | | 1-methyl-n-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamide | Human | 9464 | |
| MKNK1 (MNK1) | MAPKAPK | CAMK | 5wvd | B | | 1-methyl-n-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamide | Human | 9465 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 2ac3 | A | | - | Human | 765 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 2ac5 | A | A | - | Human | 763 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 2ac5 | A | B | - | Human | 766 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 2hw7 | A | | staurosporine | Human | 764 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cj5 | A | | 3-(pyridin-3-yl)imidazo[1,2-a]pyridine-8-carboxamide | Human | 9886 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cje | A | | 4-[(9h-purin-6-yl)amino]benzamide | Human | 9884 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cjh | A | | 3-phenyl-5-(pyridin-4-yl)-1h-indazole | Human | 9885 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cjw | A | | 3-(pyridin-4-yl)imidazo[1,2-b]pyridazine | Human | 9879 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cjy | A | | 5-[(7h-purin-6-yl)amino]-1h-isoindol-1-one | Human | 9881 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6ck3 | A | | (3r)-3-methyl-5-[(pyrimidin-4-yl)amino]-2,3-dihydro-1h-isoindol-1-one | Human | 9883 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6ck6 | A | | 6'-[(6-aminopyrimidin-4-yl)amino]-8'-methyl-2'h-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione | Human | 9880 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cki | A | | 3,3-dimethyl-6-[(pyrimidin-4-yl)amino]-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione | Human | 9882 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6jlr | A | | 4-[5-(1-methylpyrazol-4-yl)pyridin-3-yl]benzamide | Human | 11968 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 8p9b | A | | 4-[6-(4-morpholin-4-ylcarbonylphenyl)imidazo[1,2-a]pyridin-3-yl]benzenecarbonitrile | Human | 15296 | |
| Mlkl (MLKL) | TKL-Unique | TKL | 4btf | A | | - | Mouse | 5816 | |
| Mlkl (MLKL) | TKL-Unique | TKL | 4m68 | A | A | - | Mouse | 5820 | |
| Mlkl (MLKL) | TKL-Unique | TKL | 4m68 | A | B | - | Mouse | 5819 | |
| Mlkl (MLKL) | TKL-Unique | TKL | 4m69 | B | A | - | Mouse | 5818 | |
| Mlkl (MLKL) | TKL-Unique | TKL | 4m69 | B | B | - | Mouse | 5817 | |
| MLKL | TKL-Unique | TKL | 4m67 | A | | - | Human | 3048 | |
| MLKL | TKL-Unique | TKL | 4mwi | A | A | - | Human | 3047 | |
| MLKL | TKL-Unique | TKL | 4mwi | A | B | - | Human | 3049 | |
| MLKL | TKL-Unique | TKL | 5knj | A | | 1-[4-[methyl-[2-[(3-sulfamoylphenyl)amino]pyrimidin-4-yl]amino]phenyl]-3-[4-(trifluoromethyloxy)phenyl]urea | Human | 7270 | |
| MLKL | TKL-Unique | TKL | 5knj | B | | 1-[4-[methyl-[2-[(3-sulfamoylphenyl)amino]pyrimidin-4-yl]amino]phenyl]-3-[4-(trifluoromethyloxy)phenyl]urea | Human | 7268 | |
| MLKL | TKL-Unique | TKL | 5ko1 | A | A | [(1~{r})-2-[(4-fluorophenyl)amino]-2-oxidanylidene-1-phenyl-ethyl] 3-azanylpyrazine-2-carboxylate | Human | 7269 | |
| MLKL | TKL-Unique | TKL | 5ko1 | A | B | [(1~{r})-2-[(4-fluorophenyl)amino]-2-oxidanylidene-1-phenyl-ethyl] 3-azanylpyrazine-2-carboxylate | Human | 7271 | |
| MLKL | TKL-Unique | TKL | 6bwk | A | | - | Human | 10038 | |
| MLKL | TKL-Unique | TKL | 6lk5 | A | | - | Human | 13094 | |
| MLKL | TKL-Unique | TKL | 6lk6 | A | | - | Human | 13095 | |
| MLKL | TKL-Unique | TKL | 6o5z | A | | - | Human | 12782 | |
| MLKL | TKL-Unique | TKL | 6o5z | B | | 1-[2-fluoranyl-5-(trifluoromethyl)phenyl]-3-[4-[methyl-[2-[(3-sulfamoylphenyl)amino]pyrimidin-4-yl]amino]phenyl]urea | Human | 12783 | |
| MLKL | TKL-Unique | TKL | 7jw7 | A | | - | Human | 13395 | |
| MLKL | TKL-Unique | TKL | 7jxu | A | | - | Human | 13394 | |
| MLKL | TKL-Unique | TKL | 7jxu | B | | - | Human | 13396 | |
| MLKL | TKL-Unique | TKL | 7mon | A | | n-[4-({2-[(cyclopropanecarbonyl)amino]pyridin-4-yl}oxy)-3-fluorophenyl]-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 13980 | |
| MLKL | TKL-Unique | TKL | 8slz | A | | - | Human | 14988 | |
| MST1R (RON) | Met | TK | 3pls | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 1492 | |
| MST1R (RON) | Met | TK | 3pls | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 1491 | |
| MST1R (RON) | Met | TK | 8zkd | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15347 | |
| MST1R (RON) | Met | TK | 8zkd | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15346 | |
| MTOR (FRAP) | PIKK | Atypical | 3jbz | A | | adenosine-5'-diphosphate | Human | 9113 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsn | A | | - | Human | 9114 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsn | B | | - | Human | 9115 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsp | A | | phosphothiophosphoric acid-adenylate ester | Human | 9106 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsp | B | | phosphothiophosphoric acid-adenylate ester | Human | 9107 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsv | A | | adenosine-5'-diphosphate | Human | 9109 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsv | B | | adenosine-5'-diphosphate | Human | 9100 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsx | A | | 9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-one | Human | 9112 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsx | B | | 9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-one | Human | 9111 | |
| MTOR (FRAP) | PIKK | Atypical | 4jt5 | A | | 2-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-1h-indol-5-ol | Human | 9116 | |
| MTOR (FRAP) | PIKK | Atypical | 4jt5 | B | | 2-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-1h-indol-5-ol | Human | 9104 | |
| MTOR (FRAP) | PIKK | Atypical | 4jt6 | A | | 3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenol | Human | 9103 | |
| MTOR (FRAP) | PIKK | Atypical | 4jt6 | B | | 3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenol | Human | 9102 | |
| MTOR (FRAP) | PIKK | Atypical | 5flc | B | A | - | Human | 9105 | |
| MTOR (FRAP) | PIKK | Atypical | 5flc | B | B | - | Human | 9108 | |
| MTOR (FRAP) | PIKK | Atypical | 5flc | F | A | - | Human | 9101 | |
| MTOR (FRAP) | PIKK | Atypical | 5flc | F | B | - | Human | 9117 | |
| MTOR (FRAP) | PIKK | Atypical | 5h64 | a | | - | Human | 9110 | |
| MTOR (FRAP) | PIKK | Atypical | 5h64 | A | | - | Human | 9099 | |
| MTOR (FRAP) | PIKK | Atypical | 5wbu | A | | - | Human | 9407 | |
| MTOR (FRAP) | PIKK | Atypical | 5wbu | B | | - | Human | 9405 | |
| MTOR (FRAP) | PIKK | Atypical | 5wby | A | | - | Human | 9404 | |
| MTOR (FRAP) | PIKK | Atypical | 5wby | B | | - | Human | 9406 | |
| MTOR (FRAP) | PIKK | Atypical | 5zcs | A | | - | Human | 9748 | |
| MTOR (FRAP) | PIKK | Atypical | 5zcs | B | | - | Human | 9749 | |
| MTOR (FRAP) | PIKK | Atypical | 6sb0 | A | | - | Human | 11727 | |
| MTOR (FRAP) | PIKK | Atypical | 6sb0 | B | | - | Human | 11725 | |
| MTOR (FRAP) | PIKK | Atypical | 6sb2 | A | | - | Human | 11724 | |
| MTOR (FRAP) | PIKK | Atypical | 6sb2 | B | | - | Human | 11726 | |
| MTOR (FRAP) | PIKK | Atypical | 6zwm | A | | phosphothiophosphoric acid-adenylate ester | Human | 12989 | |
| MTOR (FRAP) | PIKK | Atypical | 6zwm | B | | phosphothiophosphoric acid-adenylate ester | Human | 12988 | |
| MTOR (FRAP) | PIKK | Atypical | 6zwo | B | | phosphothiophosphoric acid-adenylate ester | Human | 12987 | |
| MTOR (FRAP) | PIKK | Atypical | 7pe7 | A | | - | Human | 13901 | |
| MTOR (FRAP) | PIKK | Atypical | 7pe8 | A | | - | Human | 13870 | |
| MTOR (FRAP) | PIKK | Atypical | 7pe9 | A | | - | Human | 13871 | |
| MTOR (FRAP) | PIKK | Atypical | 7pea | A | | - | Human | 13873 | |
| MTOR (FRAP) | PIKK | Atypical | 7peb | A | | - | Human | 13869 | |
| MTOR (FRAP) | PIKK | Atypical | 7pec | A | | - | Human | 13872 | |
| MTOR (FRAP) | PIKK | Atypical | 7tzo | A | | - | Human | 14575 | |
| MTOR (FRAP) | PIKK | Atypical | 7uxc | A | | - | Human | 14525 | |
| MTOR (FRAP) | PIKK | Atypical | 8era | A | | 1-[6-{[(3m)-4-amino-3-(2-amino-1,3-benzoxazol-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-3,4-dihydroisoquinolin-2(1h)-yl]-3-hydroxypropan-1-one | Human | 14569 | |
| MTOR (FRAP) | PIKK | Atypical | 9f44 | A | | - | Human | 15316 | |
| MTOR (FRAP) | PIKK | Atypical | 9f45 | A | | - | Human | 15315 | |
| MYLK4 (SgK085) | MLCK | CAMK | 2x4f | A | A | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | 4865 | |
| MYLK4 (SgK085) | MLCK | CAMK | 2x4f | A | B | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | 4867 | |
| MYLK4 (SgK085) | MLCK | CAMK | 2x4f | B | A | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | 4866 | |
| MYLK4 (SgK085) | MLCK | CAMK | 2x4f | B | B | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | 4868 | |
| NEK1 | NEK | Other | 4apc | A | A | - | Human | 1215 | |
| NEK1 | NEK | Other | 4apc | A | B | - | Human | 1208 | |
| NEK1 | NEK | Other | 4apc | B | A | - | Human | 1212 | |
| NEK1 | NEK | Other | 4apc | B | B | - | Human | 1210 | |
| NEK1 | NEK | Other | 4b9d | A | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 1211 | |
| NEK1 | NEK | Other | 4b9d | A | B | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 1213 | |
| NEK1 | NEK | Other | 4b9d | B | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 1214 | |
| NEK1 | NEK | Other | 4b9d | B | B | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 1209 | |
| NEK2 | NEK | Other | 2jav | A | A | 5-[(z)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 332 | |
| NEK2 | NEK | Other | 2jav | A | B | 5-[(z)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 323 | |
| NEK2 | NEK | Other | 2w5a | A | A | adenosine-5'-diphosphate | Human | 302 | |
| NEK2 | NEK | Other | 2w5a | A | B | adenosine-5'-diphosphate | Human | 317 | |
| NEK2 | NEK | Other | 2w5b | A | A | phosphothiophosphoric acid-adenylate ester | Human | 320 | |
| NEK2 | NEK | Other | 2w5b | A | B | phosphothiophosphoric acid-adenylate ester | Human | 305 | |
| NEK2 | NEK | Other | 2w5h | A | A | - | Human | 327 | |
| NEK2 | NEK | Other | 2w5h | A | B | - | Human | 310 | |
| NEK2 | NEK | Other | 2wqo | A | | 4-[2-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]benzoic acid | Human | 331 | |
| NEK2 | NEK | Other | 2xk3 | A | A | 4-[3-amino-6-(3-ethylthiophen-2-yl)pyrazin-2-yl]cyclohexane-1-carboxylic acid | Human | 309 | |
| NEK2 | NEK | Other | 2xk3 | A | B | 4-[3-amino-6-(3-ethylthiophen-2-yl)pyrazin-2-yl]cyclohexane-1-carboxylic acid | Human | 329 | |
| NEK2 | NEK | Other | 2xk4 | A | A | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acid | Human | 314 | |
| NEK2 | NEK | Other | 2xk4 | A | B | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acid | Human | 316 | |
| NEK2 | NEK | Other | 2xk4 | A | C | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acid | Human | 304 | |
| NEK2 | NEK | Other | 2xk6 | A | | cis-4-[3-amino-6-(3-cyclopropylthiophen-2-yl)pyrazin-2-yl]cyclohexanecarboxylic acid | Human | 301 | |
| NEK2 | NEK | Other | 2xk7 | A | A | (3r,4r)-1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-3-ethylpiperidine-4-carboxylic acid | Human | 326 | |
| NEK2 | NEK | Other | 2xk7 | A | B | (3r,4r)-1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-3-ethylpiperidine-4-carboxylic acid | Human | 318 | |
| NEK2 | NEK | Other | 2xk8 | A | | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methoxybenzoic acid | Human | 300 | |
| NEK2 | NEK | Other | 2xkc | A | A | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methylbenzoic acid | Human | 321 | |
| NEK2 | NEK | Other | 2xkc | A | B | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methylbenzoic acid | Human | 307 | |
| NEK2 | NEK | Other | 2xkd | A | A | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]benzoic acid | Human | 330 | |
| NEK2 | NEK | Other | 2xkd | A | B | 4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]benzoic acid | Human | 298 | |
| NEK2 | NEK | Other | 2xke | A | | 1-[3-amino-6-(3-methoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acid | Human | 299 | |
| NEK2 | NEK | Other | 2xkf | A | A | 1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acid | Human | 315 | |
| NEK2 | NEK | Other | 2xkf | A | B | 1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acid | Human | 311 | |
| NEK2 | NEK | Other | 2xnm | A | A | 5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamide | Human | 306 | |
| NEK2 | NEK | Other | 2xnm | A | B | 5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamide | Human | 324 | |
| NEK2 | NEK | Other | 2xnn | A | A | 5-(1h-benzimidazol-1-yl)-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamide | Human | 303 | |
| NEK2 | NEK | Other | 2xnn | A | B | 5-(1h-benzimidazol-1-yl)-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamide | Human | 308 | |
| NEK2 | NEK | Other | 2xno | A | A | 5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{[2-(trifluoromethyl)benzyl]oxy}thiophene-2-carboxamide | Human | 319 | |
| NEK2 | NEK | Other | 2xno | A | B | 5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{[2-(trifluoromethyl)benzyl]oxy}thiophene-2-carboxamide | Human | 313 | |
| NEK2 | NEK | Other | 2xnp | A | A | 4-{5-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamide | Human | 328 | |
| NEK2 | NEK | Other | 2xnp | A | B | 4-{5-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamide | Human | 322 | |
| NEK2 | NEK | Other | 4a4x | A | | 4-(2-amino-5-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridin-3-yl)-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamide | Human | 325 | |
| NEK2 | NEK | Other | 4afe | A | | 4-(2-amino-5-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridin-3-yl)-2-{[(1r,2z)-4,4,4-trifluoro-1-methylbut-2-en-1-yl]oxy}benzamide | Human | 312 | |
| NEK2 | NEK | Other | 5m51 | A | | 3-[[6-(cyclohexylmethoxy)-9~{h}-purin-2-yl]amino]benzamide | Human | 7157 | |
| NEK2 | NEK | Other | 5m53 | A | A | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n},~{n}-dimethyl-benzamide | Human | 7159 | |
| NEK2 | NEK | Other | 5m53 | A | B | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n},~{n}-dimethyl-benzamide | Human | 7161 | |
| NEK2 | NEK | Other | 5m55 | A | A | 6-[(~{z})-2-(diethylamino)ethenyl]-~{n}-phenyl-7~{h}-purin-2-amine | Human | 7140 | |
| NEK2 | NEK | Other | 5m55 | A | B | 6-[(~{z})-2-(diethylamino)ethenyl]-~{n}-phenyl-7~{h}-purin-2-amine | Human | 7139 | |
| NEK2 | NEK | Other | 5m57 | A | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 7272 | |
| NEK2 | NEK | Other | 6sgd | A | A | 4-[(6-ethenyl-7~{h}-purin-2-yl)amino]benzenesulfonamide | Human | 12373 | |
| NEK2 | NEK | Other | 6sgd | A | B | 4-[(6-ethenyl-7~{h}-purin-2-yl)amino]benzenesulfonamide | Human | 12375 | |
| NEK2 | NEK | Other | 6sgh | A | A | 2-[4-[(6-ethenyl-9~{h}-purin-2-yl)amino]phenyl]ethanamide | Human | 12374 | |
| NEK2 | NEK | Other | 6sgh | A | B | 2-[4-[(6-ethenyl-9~{h}-purin-2-yl)amino]phenyl]ethanamide | Human | 12372 | |
| NEK2 | NEK | Other | 6sgi | A | A | 4-[(6-ethyl-7~{h}-purin-2-yl)amino]benzenesulfonamide | Human | 12378 | |
| NEK2 | NEK | Other | 6sgi | A | B | 4-[(6-ethyl-7~{h}-purin-2-yl)amino]benzenesulfonamide | Human | 12380 | |
| NEK2 | NEK | Other | 6sgk | A | | 2-phenylazanyl-9~{h}-purine-6-carbonitrile | Human | 12377 | |
| NEK2 | NEK | Other | 6sk9 | A | A | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamide | Human | 12376 | |
| NEK2 | NEK | Other | 6sk9 | A | B | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamide | Human | 12379 | |
| NEK7 | NEK | Other | 2wqm | A | A | - | Human | 3854 | |
| NEK7 | NEK | Other | 2wqm | A | B | - | Human | 3857 | |
| NEK7 | NEK | Other | 2wqn | A | A | adenosine-5'-diphosphate | Human | 3855 | |
| NEK7 | NEK | Other | 2wqn | A | B | adenosine-5'-diphosphate | Human | 3856 | |
| NEK7 | NEK | Other | 5de2 | A | A | - | Human | 6246 | |
| NEK7 | NEK | Other | 5de2 | A | B | - | Human | 6244 | |
| NEK7 | NEK | Other | 5de2 | B | A | - | Human | 6245 | |
| NEK7 | NEK | Other | 5de2 | B | B | - | Human | 6247 | |
| NEK7 | NEK | Other | 6npy | B | A | - | Human | 11338 | |
| NEK7 | NEK | Other | 6npy | B | B | - | Human | 11337 | |
| NEK7 | NEK | Other | 6s73 | A | | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamide | Human | 12357 | |
| NEK7 | NEK | Other | 6s73 | B | | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamide | Human | 12353 | |
| NEK7 | NEK | Other | 6s73 | C | | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamide | Human | 12362 | |
| NEK7 | NEK | Other | 6s73 | D | | - | Human | 12355 | |
| NEK7 | NEK | Other | 6s75 | A | | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamide | Human | 12356 | |
| NEK7 | NEK | Other | 6s75 | B | | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamide | Human | 12358 | |
| NEK7 | NEK | Other | 6s75 | C | | 3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamide | Human | 12360 | |
| NEK7 | NEK | Other | 6s75 | D | | - | Human | 12359 | |
| NEK7 | NEK | Other | 6s76 | A | | - | Human | 12351 | |
| NEK7 | NEK | Other | 6s76 | B | | - | Human | 12354 | |
| NEK7 | NEK | Other | 6s76 | C | | - | Human | 12352 | |
| NEK7 | NEK | Other | 6s76 | D | | - | Human | 12361 | |
| NEK7 | NEK | Other | 8sxn | A | | - | Human | 15246 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | A | A | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3602 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | A | B | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3610 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | B | A | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3607 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | B | B | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3604 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | C | A | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3617 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | C | B | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3621 | |
| NTRK1 (TRKA) | Trk | TK | 4f0i | A | | - | Human | 3603 | |
| NTRK1 (TRKA) | Trk | TK | 4f0i | B | | - | Human | 3605 | |
| NTRK1 (TRKA) | Trk | TK | 4gt5 | A | A | - | Human | 3616 | |
| NTRK1 (TRKA) | Trk | TK | 4gt5 | A | B | - | Human | 3609 | |
| NTRK1 (TRKA) | Trk | TK | 4pmm | A | A | n-(3-cyclopropyl-1-phenyl-1h-pyrazol-5-yl)-2-{4-[3-methoxy-4-(4-methyl-1h-imidazol-1-yl)phenyl]-1h-1,2,3-triazol-1-yl}acetamide | Human | 3618 | |
| NTRK1 (TRKA) | Trk | TK | 4pmm | A | B | n-(3-cyclopropyl-1-phenyl-1h-pyrazol-5-yl)-2-{4-[3-methoxy-4-(4-methyl-1h-imidazol-1-yl)phenyl]-1h-1,2,3-triazol-1-yl}acetamide | Human | 3619 | |
| NTRK1 (TRKA) | Trk | TK | 4pmp | A | A | 1-cyclopropyl-1-[3-(1,3-thiazol-2-yl)benzyl]-3-[4-(trifluoromethoxy)phenyl]urea | Human | 3613 | |
| NTRK1 (TRKA) | Trk | TK | 4pmp | A | B | 1-cyclopropyl-1-[3-(1,3-thiazol-2-yl)benzyl]-3-[4-(trifluoromethoxy)phenyl]urea | Human | 3608 | |
| NTRK1 (TRKA) | Trk | TK | 4pms | A | A | 4-(naphthalen-1-yl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1h-pyrrolo[3,2-c]pyridine-2-carboxylic acid | Human | 3606 | |
| NTRK1 (TRKA) | Trk | TK | 4pms | A | B | 4-(naphthalen-1-yl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1h-pyrrolo[3,2-c]pyridine-2-carboxylic acid | Human | 3601 | |
| NTRK1 (TRKA) | Trk | TK | 4pmt | A | A | n~4~-[4-(morpholin-4-yl)phenyl]-n~6~-(pyridin-3-ylmethyl)pyrido[3,2-d]pyrimidine-4,6-diamine | Human | 3614 | |
| NTRK1 (TRKA) | Trk | TK | 4pmt | A | B | n~4~-[4-(morpholin-4-yl)phenyl]-n~6~-(pyridin-3-ylmethyl)pyrido[3,2-d]pyrimidine-4,6-diamine | Human | 3612 | |
| NTRK1 (TRKA) | Trk | TK | 4yne | A | A | 6-[(2r)-2-(3-fluorophenyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)imidazo[1,2-b]pyridazine | Human | 3620 | |
| NTRK1 (TRKA) | Trk | TK | 4yne | A | B | 6-[(2r)-2-(3-fluorophenyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)imidazo[1,2-b]pyridazine | Human | 3611 | |
| NTRK1 (TRKA) | Trk | TK | 4yps | A | | 4-{6-[(3r)-3-(3-fluorophenyl)morpholin-4-yl]imidazo[1,2-b]pyridazin-3-yl}benzonitrile | Human | 3615 | |
| NTRK1 (TRKA) | Trk | TK | 5h3q | A | A | 1-[(3s,4r)-4-[3,4-bis(fluoranyl)phenyl]-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(5-ethoxy-4-methyl-2-phenyl-pyrazol-3-yl)urea | Human | 7461 | |
| NTRK1 (TRKA) | Trk | TK | 5h3q | A | B | 1-[(3s,4r)-4-[3,4-bis(fluoranyl)phenyl]-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(5-ethoxy-4-methyl-2-phenyl-pyrazol-3-yl)urea | Human | 7460 | |
| NTRK1 (TRKA) | Trk | TK | 5i8a | A | A | (6r)-3-(methylsulfanyl)-6-phenyl-1-(1h-pyrazol-3-yl)-6,7-dihydrothieno[3,4-c]pyridin-4(5h)-one | Human | 8311 | |
| NTRK1 (TRKA) | Trk | TK | 5i8a | A | B | (6r)-3-(methylsulfanyl)-6-phenyl-1-(1h-pyrazol-3-yl)-6,7-dihydrothieno[3,4-c]pyridin-4(5h)-one | Human | 8312 | |
| NTRK1 (TRKA) | Trk | TK | 5jfs | A | A | n-{4-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-2-yl}-n'-(2,4-difluorophenyl)urea | Human | 7506 | |
| NTRK1 (TRKA) | Trk | TK | 5jfs | A | B | n-{4-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-2-yl}-n'-(2,4-difluorophenyl)urea | Human | 7502 | |
| NTRK1 (TRKA) | Trk | TK | 5jfv | A | A | n-{5-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}-2-(4-chlorophenyl)acetamide | Human | 7504 | |
| NTRK1 (TRKA) | Trk | TK | 5jfv | A | B | n-{5-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}-2-(4-chlorophenyl)acetamide | Human | 7503 | |
| NTRK1 (TRKA) | Trk | TK | 5jfw | A | A | 2-(4-cyanophenyl)-n-{5-[7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}acetamide | Human | 7500 | |
| NTRK1 (TRKA) | Trk | TK | 5jfw | A | B | 2-(4-cyanophenyl)-n-{5-[7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}acetamide | Human | 7505 | |
| NTRK1 (TRKA) | Trk | TK | 5jfx | A | | n-{5-[2-amino-7-(1-hydroxy-2-methylpropan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}-2-(5-chloropyridin-2-yl)acetamide | Human | 7501 | |
| NTRK1 (TRKA) | Trk | TK | 5kmi | A | | 1-(9~{h}-fluoren-9-yl)-3-(2-methyl-4-phenyl-pyrimidin-5-yl)urea | Human | 7330 | |
| NTRK1 (TRKA) | Trk | TK | 5kmj | A | A | ~{n}-(pyridin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)ethanamide | Human | 7334 | |
| NTRK1 (TRKA) | Trk | TK | 5kmj | A | B | ~{n}-(pyridin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)ethanamide | Human | 7335 | |
| NTRK1 (TRKA) | Trk | TK | 5kmk | A | | 2-fluoranyl-~{n}-[2-(4-fluorophenyl)-6-methyl-pyridin-3-yl]-4-(trifluoromethyl)benzamide | Human | 7336 | |
| NTRK1 (TRKA) | Trk | TK | 5kml | A | | 1-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-3-[[2-(trifluoromethyl)phenyl]methyl]urea | Human | 7333 | |
| NTRK1 (TRKA) | Trk | TK | 5kmm | A | | 1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-naphthalen-1-yl-urea | Human | 7331 | |
| NTRK1 (TRKA) | Trk | TK | 5kmn | A | | 1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-[[2-(trifluoromethyl)phenyl]methyl]urea | Human | 7332 | |
| NTRK1 (TRKA) | Trk | TK | 5kmo | A | | 1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-pyridin-2-yl-urea | Human | 7329 | |
| NTRK1 (TRKA) | Trk | TK | 5kvt | A | A | entrectinib | Human | 9450 | |
| NTRK1 (TRKA) | Trk | TK | 5kvt | A | B | entrectinib | Human | 9451 | |
| NTRK1 (TRKA) | Trk | TK | 5wr7 | A | | n-tert-butyl-2-[2-[6,6-dimethyl-8-(methylsulfonylamino)-11-oxidanylidene-naphtho[2,3-b][1]benzofuran-3-yl]ethynyl]-6-methyl-pyridine-4-carboxamide | Human | 8737 | |
| NTRK1 (TRKA) | Trk | TK | 6d1y | A | A | 2,4-dichloro-n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)benzamide | Human | 9873 | |
| NTRK1 (TRKA) | Trk | TK | 6d1y | A | B | 2,4-dichloro-n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)benzamide | Human | 9871 | |
| NTRK1 (TRKA) | Trk | TK | 6d1z | A | A | 5-{[5-(6-aminopyridin-2-yl)-2-chlorobenzene-1-carbonyl]amino}-1-phenyl-1h-pyrazole-3-carboxamide | Human | 9874 | |
| NTRK1 (TRKA) | Trk | TK | 6d1z | A | B | 5-{[5-(6-aminopyridin-2-yl)-2-chlorobenzene-1-carbonyl]amino}-1-phenyl-1h-pyrazole-3-carboxamide | Human | 9870 | |
| NTRK1 (TRKA) | Trk | TK | 6d20 | A | | 5-{[2,4-dichloro-5-(pyridin-2-yl)benzene-1-carbonyl]amino}-n-(2-hydroxy-2-methylpropyl)-1-phenyl-1h-pyrazole-3-carboxamide | Human | 9875 | |
| NTRK1 (TRKA) | Trk | TK | 6d22 | A | | - | Human | 9872 | |
| NTRK1 (TRKA) | Trk | TK | 6dkb | A | | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamide | Human | 10057 | |
| NTRK1 (TRKA) | Trk | TK | 6dkg | A | A | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-4-(2-hydroxy-2-methylpropoxy)benzamide | Human | 10059 | |
| NTRK1 (TRKA) | Trk | TK | 6dkg | A | B | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-4-(2-hydroxy-2-methylpropoxy)benzamide | Human | 10063 | |
| NTRK1 (TRKA) | Trk | TK | 6dki | A | A | 6-amino-5-{[(3s)-4,4-difluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}pyrrolidin-3-yl]oxy}-n-methylpyridine-3-carboxamide | Human | 10060 | |
| NTRK1 (TRKA) | Trk | TK | 6dki | A | B | 6-amino-5-{[(3s)-4,4-difluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}pyrrolidin-3-yl]oxy}-n-methylpyridine-3-carboxamide | Human | 10061 | |
| NTRK1 (TRKA) | Trk | TK | 6dkw | A | A | 5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamide | Human | 10056 | |
| NTRK1 (TRKA) | Trk | TK | 6dkw | A | B | 5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamide | Human | 10058 | |
| NTRK1 (TRKA) | Trk | TK | 6dkw | B | A | 5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamide | Human | 10062 | |
| NTRK1 (TRKA) | Trk | TK | 6dkw | B | B | 5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamide | Human | 10064 | |
| NTRK1 (TRKA) | Trk | TK | 6iqn | A | | 4-[[4-azanyl-3-(4-cyclohexylpiperazin-1-yl)-9,10-bis(oxidanylidene)anthracen-1-yl]amino]benzoic acid | Human | 11951 | |
| NTRK1 (TRKA) | Trk | TK | 6iqn | B | | 4-[[4-azanyl-3-(4-cyclohexylpiperazin-1-yl)-9,10-bis(oxidanylidene)anthracen-1-yl]amino]benzoic acid | Human | 11950 | |
| NTRK1 (TRKA) | Trk | TK | 6j5l | A | A | n-{2-[({3-[6-(piperazin-1-yl)pyridin-3-yl]-1h-indazol-5-yl}amino)methyl]phenyl}methanesulfonamide | Human | 11436 | |
| NTRK1 (TRKA) | Trk | TK | 6j5l | A | B | n-{2-[({3-[6-(piperazin-1-yl)pyridin-3-yl]-1h-indazol-5-yl}amino)methyl]phenyl}methanesulfonamide | Human | 11435 | |
| NTRK1 (TRKA) | Trk | TK | 6j5l | A | C | n-{2-[({3-[6-(piperazin-1-yl)pyridin-3-yl]-1h-indazol-5-yl}amino)methyl]phenyl}methanesulfonamide | Human | 11437 | |
| NTRK1 (TRKA) | Trk | TK | 6npt | A | | 4-tert-butyl-n-(1,3-diphenyl-1h-pyrazol-5-yl)benzamide | Human | 11172 | |
| NTRK1 (TRKA) | Trk | TK | 6nsp | A | A | n-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)-2-(3-oxo-2,3-dihydro-4h-1,4-benzothiazin-4-yl)acetamide | Human | 11173 | |
| NTRK1 (TRKA) | Trk | TK | 6nsp | A | B | n-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)-2-(3-oxo-2,3-dihydro-4h-1,4-benzothiazin-4-yl)acetamide | Human | 11175 | |
| NTRK1 (TRKA) | Trk | TK | 6nss | A | A | n-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)-2-(10h-phenoxazin-10-yl)acetamide | Human | 11174 | |
| NTRK1 (TRKA) | Trk | TK | 6nss | A | B | n-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)-2-(10h-phenoxazin-10-yl)acetamide | Human | 11176 | |
| NTRK1 (TRKA) | Trk | TK | 6pl1 | A | A | n-(5-{[(7-methyl-4-oxo-4h-pyrido[1,2-a]pyrimidin-2-yl)methyl]sulfanyl}-1,3,4-thiadiazol-2-yl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | 11722 | |
| NTRK1 (TRKA) | Trk | TK | 6pl1 | A | B | n-(5-{[(7-methyl-4-oxo-4h-pyrido[1,2-a]pyrimidin-2-yl)methyl]sulfanyl}-1,3,4-thiadiazol-2-yl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | 11723 | |
| NTRK1 (TRKA) | Trk | TK | 6pl2 | A | | n-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-2-{[1-(4-hydroxyphenyl)-1h-tetrazol-5-yl]sulfanyl}acetamide | Human | 11598 | |
| NTRK1 (TRKA) | Trk | TK | 6pl3 | A | A | 2-[(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)amino]-2-oxoethyl 4-(1h-tetrazol-1-yl)benzoate | Human | 11599 | |
| NTRK1 (TRKA) | Trk | TK | 6pl3 | A | B | 2-[(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)amino]-2-oxoethyl 4-(1h-tetrazol-1-yl)benzoate | Human | 11600 | |
| NTRK1 (TRKA) | Trk | TK | 6pl4 | A | A | n-{[5-(methoxymethyl)-2-(trifluoromethoxy)phenyl]methyl}-n'-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)urea | Human | 12463 | |
| NTRK1 (TRKA) | Trk | TK | 6pl4 | A | B | n-{[5-(methoxymethyl)-2-(trifluoromethoxy)phenyl]methyl}-n'-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)urea | Human | 12464 | |
| NTRK1 (TRKA) | Trk | TK | 6pma | A | | n-[2-chloro-5-(trifluoromethyl)phenyl]-2-[1-(4-methoxyphenyl)-4-oxo-1,4-dihydro-5h-pyrazolo[3,4-d]pyrimidin-5-yl]acetamide | Human | 12006 | |
| NTRK1 (TRKA) | Trk | TK | 6pmb | A | | 2-[5,7-dimethyl-2-(pyridin-3-yl)[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 12001 | |
| NTRK1 (TRKA) | Trk | TK | 6pmc | A | | n-(6-{[(5-chloro-2-methoxyphenyl)carbamoyl]amino}-1,3-benzothiazol-2-yl)benzamide | Human | 12002 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | A | A | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12004 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | A | B | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12005 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | B | A | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12007 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | B | B | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12000 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | C | A | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 11999 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | C | B | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12003 | |
| NTRK1 (TRKA) | Trk | TK | 7vkm | A | A | - | Human | 13946 | |
| NTRK1 (TRKA) | Trk | TK | 7vkm | A | B | - | Human | 13942 | |
| NTRK1 (TRKA) | Trk | TK | 7vkn | A | A | repotrectinib | Human | 13945 | |
| NTRK1 (TRKA) | Trk | TK | 7vkn | A | B | repotrectinib | Human | 13944 | |
| NTRK1 (TRKA) | Trk | TK | 7vko | A | | repotrectinib | Human | 13943 | |
| NTRK1 (TRKA) | Trk | TK | 7xaf | A | | 4^6,14-dimethyl-n-(3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-10-oxo-5-oxa-11,14-diaza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclo-tetradecaphan-2-yne-45-carboxamide | Human | 14232 | |
| NTRK1 (TRKA) | Trk | TK | 7xbi | A | A | 4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]-~{n}-[3-(1-methylpyrazol-4-yl)-1~{h}-indazol-5-yl]-2-(trifluoromethyl)benzamide | Human | 14687 | |
| NTRK1 (TRKA) | Trk | TK | 7xbi | A | B | 4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]-~{n}-[3-(1-methylpyrazol-4-yl)-1~{h}-indazol-5-yl]-2-(trifluoromethyl)benzamide | Human | 14686 | |
| NTRK1 (TRKA) | Trk | TK | 8j5w | A | | n-(3-cyclopropyl-5-((4-methylpiperazin-1-yl)methyl)phenyl)-4^6-methyl-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamide | Human | 14985 | |
| NTRK1 (TRKA) | Trk | TK | 8j5x | A | | n-(3-cyclopropyl-5-((4-methylpiperazin-1-yl)methyl)phenyl)-4^6-methyl-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamide | Human | 14987 | |
| NTRK1 (TRKA) | Trk | TK | 8j61 | A | | 4^6-methyl-n-(3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamide | Human | 14986 | |
| NTRK1 (TRKA) | Trk | TK | 8j63 | A | | 4^6-methyl-n-(3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-11-oxo-5-oxa-10,14-diaza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamide | Human | 14984 | |
| NTRK2 (TRKB) | Trk | TK | 4asz | A | | - | Human | 3599 | |
| NTRK2 (TRKB) | Trk | TK | 4at3 | A | | (5z)-5-(carbamoylimino)-3-[(5r)-6,7,8,9-tetrahydro-5h-benzo[7]annulen-5-ylsulfanyl]-2,5-dihydroisothiazole-4-carboxamide | Human | 3600 | |
| NTRK2 (TRKB) | Trk | TK | 4at4 | A | | 1-[4-(4-aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea | Human | 3598 | |
| NTRK2 (TRKB) | Trk | TK | 4at5 | A | | 5-{3-methoxy-4-[(4-methoxybenzyl)oxy]benzyl}pyrimidine-2,4-diamine | Human | 3597 | |
| NTRK3 (TRKC) | Trk | TK | 3v5q | A | | 1-(3-{[(3z)-2-oxo-3-(1h-pyrrol-2-ylmethylidene)-2,3-dihydro-1h-indol-6-yl]amino}phenyl)-3-[3-(trifluoromethyl)phenyl]urea | Human | 102 | |
| NTRK3 (TRKC) | Trk | TK | 3v5q | B | | 1-(3-{[(3z)-2-oxo-3-(1h-pyrrol-2-ylmethylidene)-2,3-dihydro-1h-indol-6-yl]amino}phenyl)-3-[3-(trifluoromethyl)phenyl]urea | Human | 97 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | A | A | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 101 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | A | B | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 98 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | B | A | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 100 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | B | B | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 99 | |
| NTRK3 (TRKC) | Trk | TK | 6kzc | A | | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-2-methyl-~{n}-[3-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]benzamide | Human | 11696 | |
| NTRK3 (TRKC) | Trk | TK | 6kzd | A | | 3-[2-[6-(4-aminophenyl)imidazo[1,2-a]pyrazin-3-yl]ethynyl]-2-methyl-~{n}-[3-(4-methylpiperazin-1-yl)-5-propan-2-yl-phenyl]benzamide | Human | 11697 | |
| OXSR1 (OSR1) | STE20 | STE | 2vwi | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 4842 | |
| OXSR1 (OSR1) | STE20 | STE | 2vwi | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 4839 | |
| OXSR1 (OSR1) | STE20 | STE | 2vwi | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 4843 | |
| OXSR1 (OSR1) | STE20 | STE | 2vwi | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 4836 | |
| OXSR1 (OSR1) | STE20 | STE | 2vwi | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 4838 | |
| OXSR1 (OSR1) | STE20 | STE | 2vwi | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 4844 | |
| OXSR1 (OSR1) | STE20 | STE | 2vwi | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 4835 | |
| OXSR1 (OSR1) | STE20 | STE | 2vwi | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 4833 | |
| OXSR1 (OSR1) | STE20 | STE | 3dak | A | | phosphoaminophosphonic acid-adenylate ester | Human | 4834 | |
| OXSR1 (OSR1) | STE20 | STE | 3dak | B | | phosphoaminophosphonic acid-adenylate ester | Human | 4841 | |
| OXSR1 (OSR1) | STE20 | STE | 3dak | C | | phosphoaminophosphonic acid-adenylate ester | Human | 4837 | |
| OXSR1 (OSR1) | STE20 | STE | 3dak | D | | phosphoaminophosphonic acid-adenylate ester | Human | 4840 | |
| PAK1 | STE20 | STE | 1f3m | C | | - | Human | 161 | |
| PAK1 | STE20 | STE | 1f3m | D | | - | Human | 158 | |
| PAK1 | STE20 | STE | 1yhv | A | | - | Human | 177 | |
| PAK1 | STE20 | STE | 1yhw | A | | - | Human | 160 | |
| PAK1 | STE20 | STE | 2hy8 | 1 | | (5s,6r,7r,9r)-12-hydroxy-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9-tetrahydro-5h,14h-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-one | Human | 172 | |
| PAK1 | STE20 | STE | 3fxz | A | A | octahedral ru-pyridocarbazole | Human | 7198 | |
| PAK1 | STE20 | STE | 3fxz | A | B | octahedral ru-pyridocarbazole | Human | 7200 | |
| PAK1 | STE20 | STE | 3fy0 | A | | ruthenium pyridocarbazole | Human | 7202 | |
| PAK1 | STE20 | STE | 3q4z | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 166 | |
| PAK1 | STE20 | STE | 3q4z | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 174 | |
| PAK1 | STE20 | STE | 3q4z | B | A | - | Human | 144 | |
| PAK1 | STE20 | STE | 3q4z | B | B | - | Human | 183 | |
| PAK1 | STE20 | STE | 3q52 | A | | - | Human | 146 | |
| PAK1 | STE20 | STE | 3q53 | A | | adenosine-5'-triphosphate | Human | 165 | |
| PAK1 | STE20 | STE | 4daw | A | A | [1,3-dioxo-6-(pyridin-2-yl-kappan)-2,3-dihydro-1h-isoindol-5-yl-kappac~5~][(thioxomethylidene)azanido-kappan](1,4,7-trithionane-kappa~3~s~1~,s~4~,s~7~)ruthenium | Human | 7201 | |
| PAK1 | STE20 | STE | 4daw | A | B | [1,3-dioxo-6-(pyridin-2-yl-kappan)-2,3-dihydro-1h-isoindol-5-yl-kappac~5~][(thioxomethylidene)azanido-kappan](1,4,7-trithionane-kappa~3~s~1~,s~4~,s~7~)ruthenium | Human | 7199 | |
| PAK1 | STE20 | STE | 4eqc | A | A | 6-[2-chloro-4-(1,3-thiazol-5-yl)phenyl]-8-ethyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 180 | |
| PAK1 | STE20 | STE | 4eqc | A | B | 6-[2-chloro-4-(1,3-thiazol-5-yl)phenyl]-8-ethyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 147 | |
| PAK1 | STE20 | STE | 4o0r | A | | pf-3758309 | Human | 171 | |
| PAK1 | STE20 | STE | 4o0r | B | | - | Human | 145 | |
| PAK1 | STE20 | STE | 4o0t | A | | 1-({1-(2-aminopyrimidin-4-yl)-2-[(2-methoxyethyl)amino]-1h-benzimidazol-6-yl}ethynyl)cyclohexanol | Human | 143 | |
| PAK1 | STE20 | STE | 4o0t | B | | - | Human | 141 | |
| PAK1 | STE20 | STE | 4p90 | A | | [2-chloro-5-(hydroxymethyl)phenyl]{5-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl}methanone | Human | 164 | |
| PAK1 | STE20 | STE | 4p90 | B | | [2-chloro-5-(hydroxymethyl)phenyl]{5-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl}methanone | Human | 151 | |
| PAK1 | STE20 | STE | 4zji | A | A | 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine | Human | 159 | |
| PAK1 | STE20 | STE | 4zji | A | B | 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine | Human | 175 | |
| PAK1 | STE20 | STE | 4zji | B | A | 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine | Human | 168 | |
| PAK1 | STE20 | STE | 4zji | B | B | 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine | Human | 185 | |
| PAK1 | STE20 | STE | 4zji | C | A | 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine | Human | 167 | |
| PAK1 | STE20 | STE | 4zji | C | B | 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine | Human | 152 | |
| PAK1 | STE20 | STE | 4zji | D | A | 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine | Human | 139 | |
| PAK1 | STE20 | STE | 4zji | D | B | 2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepine | Human | 150 | |
| PAK1 | STE20 | STE | 4zjj | A | A | (s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamide | Human | 157 | |
| PAK1 | STE20 | STE | 4zjj | A | B | (s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamide | Human | 153 | |
| PAK1 | STE20 | STE | 4zjj | B | A | (s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamide | Human | 176 | |
| PAK1 | STE20 | STE | 4zjj | B | B | (s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamide | Human | 137 | |
| PAK1 | STE20 | STE | 4zjj | C | A | (s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamide | Human | 182 | |
| PAK1 | STE20 | STE | 4zjj | C | B | (s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamide | Human | 178 | |
| PAK1 | STE20 | STE | 4zjj | D | A | (s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamide | Human | 169 | |
| PAK1 | STE20 | STE | 4zjj | D | B | (s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamide | Human | 162 | |
| PAK1 | STE20 | STE | 4zlo | A | A | 2,8-difluoro-11-(4-methylpiperazin-1-yl)-5h-dibenzo[b,e][1,4]diazepine | Human | 142 | |
| PAK1 | STE20 | STE | 4zlo | A | B | 2,8-difluoro-11-(4-methylpiperazin-1-yl)-5h-dibenzo[b,e][1,4]diazepine | Human | 181 | |
| PAK1 | STE20 | STE | 4zlo | B | A | - | Human | 188 | |
| PAK1 | STE20 | STE | 4zlo | B | B | - | Human | 170 | |
| PAK1 | STE20 | STE | 4zy4 | A | | 2-(4-aminopiperidin-1-yl)-n-(5-cyclopropyl-1h-pyrazol-3-yl)thieno[3,2-d]pyrimidin-4-amine | Human | 187 | |
| PAK1 | STE20 | STE | 4zy4 | B | | 2-(4-aminopiperidin-1-yl)-n-(5-cyclopropyl-1h-pyrazol-3-yl)thieno[3,2-d]pyrimidin-4-amine | Human | 154 | |
| PAK1 | STE20 | STE | 4zy5 | A | | n~2~-[(trans-4-aminocyclohexyl)methyl]-n~4~-(3-cyclopropyl-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 155 | |
| PAK1 | STE20 | STE | 4zy5 | B | | n~2~-[(trans-4-aminocyclohexyl)methyl]-n~4~-(3-cyclopropyl-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 163 | |
| PAK1 | STE20 | STE | 4zy6 | A | A | n~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine | Human | 138 | |
| PAK1 | STE20 | STE | 4zy6 | A | B | n~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine | Human | 173 | |
| PAK1 | STE20 | STE | 4zy6 | B | A | n~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine | Human | 156 | |
| PAK1 | STE20 | STE | 4zy6 | B | B | n~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine | Human | 184 | |
| PAK1 | STE20 | STE | 5dew | A | | 8-[(trans-4-aminocyclohexyl)methyl]-6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-2-(ethylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 7408 | |
| PAK1 | STE20 | STE | 5dew | B | | 8-[(trans-4-aminocyclohexyl)methyl]-6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-2-(ethylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 7409 | |
| PAK1 | STE20 | STE | 5dey | A | | 8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6364 | |
| PAK1 | STE20 | STE | 5dey | B | | 8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6365 | |
| PAK1 | STE20 | STE | 5dfp | A | A | 6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-8-ethyl-2-{[2-(1-methylpiperidin-4-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6366 | |
| PAK1 | STE20 | STE | 5dfp | A | B | 6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-8-ethyl-2-{[2-(1-methylpiperidin-4-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6363 | |
| PAK1 | STE20 | STE | 5ime | A | | 8-(3-aminopropyl)-6-[2-chloro-4-(3-methyl-2-oxopyrazin-1(2h)-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6644 | |
| PAK1 | STE20 | STE | 5ime | B | | 8-(3-aminopropyl)-6-[2-chloro-4-(3-methyl-2-oxopyrazin-1(2h)-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6643 | |
| PAK1 | STE20 | STE | 5kbq | A | | [4-methyl-3-[methyl-[2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]pyrimidin-4-yl]amino]phenyl]methanol | Human | 7081 | |
| PAK1 | STE20 | STE | 5kbq | B | | - | Human | 7082 | |
| PAK1 | STE20 | STE | 5kbr | A | | (4-chlorophenyl)-[5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]methanone | Human | 7080 | |
| PAK1 | STE20 | STE | 5kbr | B | | (4-chlorophenyl)-[5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]methanone | Human | 7079 | |
| PAK1 | STE20 | STE | 6b16 | A | | n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)-n~2~-[(1s)-1-(1h-pyrrolo[3,2-b]pyridin-5-yl)ethyl]pyrimidine-2,4-diamine | Human | 8574 | |
| PAK1 | STE20 | STE | 6b16 | B | | n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)-n~2~-[(1s)-1-(1h-pyrrolo[3,2-b]pyridin-5-yl)ethyl]pyrimidine-2,4-diamine | Human | 8575 | |
| PAK1 | STE20 | STE | 7vto | A | A | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 14483 | |
| PAK1 | STE20 | STE | 7vto | A | B | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 14484 | |
| PAK1 | STE20 | STE | 8x5z | A | A | - | Human | 15049 | |
| PAK1 | STE20 | STE | 8x5z | A | B | - | Human | 15048 | |
| PAK3 | STE20 | STE | 6fd3 | A | A | adenosine-5'-diphosphate | Human | 9462 | |
| PAK3 | STE20 | STE | 6fd3 | A | B | adenosine-5'-diphosphate | Human | 9463 | |
| PAK4 | STE20 | STE | 2bva | A | | - | Human | 1394 | |
| PAK4 | STE20 | STE | 2bva | B | | - | Human | 1407 | |
| PAK4 | STE20 | STE | 2cdz | A | A | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 1378 | |
| PAK4 | STE20 | STE | 2cdz | A | B | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 1374 | |
| PAK4 | STE20 | STE | 2j0i | A | A | - | Human | 1391 | |
| PAK4 | STE20 | STE | 2j0i | A | B | - | Human | 1377 | |
| PAK4 | STE20 | STE | 2q0n | A | A | - | Human | 1393 | |
| PAK4 | STE20 | STE | 2q0n | A | B | - | Human | 1401 | |
| PAK4 | STE20 | STE | 2x4z | A | | pf-3758309 | Human | 1387 | |
| PAK4 | STE20 | STE | 4app | A | A | n-[6,6-dimethyl-5-[(2s)-4-methyl-2-(phenylmethyl)piperazin-1-yl]carbonyl-2,4-dihydropyrrolo[3,4-c]pyrazol-3-yl]-3-phenoxy-benzamide | Human | 1385 | |
| PAK4 | STE20 | STE | 4app | A | B | n-[6,6-dimethyl-5-[(2s)-4-methyl-2-(phenylmethyl)piperazin-1-yl]carbonyl-2,4-dihydropyrrolo[3,4-c]pyrazol-3-yl]-3-phenoxy-benzamide | Human | 1390 | |
| PAK4 | STE20 | STE | 4fie | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1405 | |
| PAK4 | STE20 | STE | 4fie | B | | phosphoaminophosphonic acid-adenylate ester | Human | 1372 | |
| PAK4 | STE20 | STE | 4fif | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 1395 | |
| PAK4 | STE20 | STE | 4fif | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 1370 | |
| PAK4 | STE20 | STE | 4fif | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 1381 | |
| PAK4 | STE20 | STE | 4fif | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 1379 | |
| PAK4 | STE20 | STE | 4fig | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1392 | |
| PAK4 | STE20 | STE | 4fig | B | | phosphoaminophosphonic acid-adenylate ester | Human | 1373 | |
| PAK4 | STE20 | STE | 4fih | A | A | - | Human | 1399 | |
| PAK4 | STE20 | STE | 4fih | A | B | - | Human | 1402 | |
| PAK4 | STE20 | STE | 4fii | A | A | - | Human | 1383 | |
| PAK4 | STE20 | STE | 4fii | A | B | - | Human | 1396 | |
| PAK4 | STE20 | STE | 4fij | A | | - | Human | 1408 | |
| PAK4 | STE20 | STE | 4jdh | A | A | - | Human | 1371 | |
| PAK4 | STE20 | STE | 4jdh | A | B | - | Human | 1406 | |
| PAK4 | STE20 | STE | 4jdi | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 1403 | |
| PAK4 | STE20 | STE | 4jdi | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 1380 | |
| PAK4 | STE20 | STE | 4jdj | A | A | - | Human | 1400 | |
| PAK4 | STE20 | STE | 4jdj | A | B | - | Human | 1397 | |
| PAK4 | STE20 | STE | 4jdk | A | A | - | Human | 1375 | |
| PAK4 | STE20 | STE | 4jdk | A | B | - | Human | 1398 | |
| PAK4 | STE20 | STE | 4l67 | A | | - | Human | 1376 | |
| PAK4 | STE20 | STE | 4njd | A | A | n-(1h-indazol-5-yl)-n'-[2-(1h-indol-3-yl)ethyl]-6-methoxy-1,3,5-triazine-2,4-diamine | Human | 1382 | |
| PAK4 | STE20 | STE | 4njd | A | B | n-(1h-indazol-5-yl)-n'-[2-(1h-indol-3-yl)ethyl]-6-methoxy-1,3,5-triazine-2,4-diamine | Human | 1384 | |
| PAK4 | STE20 | STE | 4o0v | A | | 1-({1-(2-aminopyrimidin-4-yl)-2-[(2-methoxyethyl)amino]-1h-benzimidazol-6-yl}ethynyl)cyclohexanol | Human | 1386 | |
| PAK4 | STE20 | STE | 4o0x | A | | 1-{[1-(4-amino-1,3,5-triazin-2-yl)-2-methyl-1h-benzimidazol-6-yl]ethynyl}cyclohexanol | Human | 1404 | |
| PAK4 | STE20 | STE | 4o0y | A | | 4-[1-(4-amino-1,3,5-triazin-2-yl)-2-(ethylamino)-1h-benzimidazol-6-yl]-2-methylbut-3-yn-2-ol | Human | 1388 | |
| PAK4 | STE20 | STE | 4xbr | A | | adenosine-5'-triphosphate | Human | 6257 | |
| PAK4 | STE20 | STE | 4xbu | A | | - | Human | 6256 | |
| PAK4 | STE20 | STE | 5bms | A | | n~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamine | Human | 1389 | |
| PAK4 | STE20 | STE | 5i0b | A | | 6-bromo-2-[1-methyl-3-(propan-2-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridine | Human | 7315 | |
| PAK4 | STE20 | STE | 5upk | B | | phosphoaminophosphonic acid-adenylate ester | Human | 9435 | |
| PAK4 | STE20 | STE | 5upl | A | | - | Human | 9436 | |
| PAK4 | STE20 | STE | 5ved | A | | staurosporine | Human | 8570 | |
| PAK4 | STE20 | STE | 5vee | A | | 6-(2,4-dichlorophenyl)-8-ethyl-2-{[3-fluoro-4-(piperazin-1-yl)phenyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 8572 | |
| PAK4 | STE20 | STE | 5vef | A | A | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 8569 | |
| PAK4 | STE20 | STE | 5vef | A | B | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 8571 | |
| PAK4 | STE20 | STE | 5xva | A | | [6-chloranyl-4-[(5-methyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl]-[(3r)-3-methylpiperazin-1-yl]methanone | Human | 9550 | |
| PAK4 | STE20 | STE | 5xvf | A | | 2-(4-azanylpiperidin-1-yl)-6-chloranyl-n-(1-methylimidazol-4-yl)quinazolin-4-amine | Human | 9549 | |
| PAK4 | STE20 | STE | 5xvg | A | | [6-chloranyl-4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl]-[(3r)-3-methylpiperazin-1-yl]methanone | Human | 9551 | |
| PAK4 | STE20 | STE | 5zjw | A | A | (3z)-n-[(1s)-2-hydroxy-1-phenylethyl]-3-[(1h-imidazol-2-yl)(phenyl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 10999 | |
| PAK4 | STE20 | STE | 5zjw | A | B | (3z)-n-[(1s)-2-hydroxy-1-phenylethyl]-3-[(1h-imidazol-2-yl)(phenyl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 11000 | |
| PAK4 | STE20 | STE | 6wlx | A | A | - | Human | 12399 | |
| PAK4 | STE20 | STE | 6wlx | A | B | - | Human | 12400 | |
| PAK4 | STE20 | STE | 6wly | A | A | - | Human | 12397 | |
| PAK4 | STE20 | STE | 6wly | A | B | - | Human | 12396 | |
| PAK4 | STE20 | STE | 6wly | A | C | - | Human | 12398 | |
| PAK4 | STE20 | STE | 7cmb | A | | 1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indole-3-carboxamide | Human | 13818 | |
| PAK4 | STE20 | STE | 7cp3 | A | | [(3r)-3-azanylpiperidin-1-yl]-[1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]methanone | Human | 13849 | |
| PAK4 | STE20 | STE | 7cp4 | A | | [1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]-[(3s)-3-methylpiperazin-1-yl]methanone | Human | 13850 | |
| PAK4 | STE20 | STE | 7s46 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14495 | |
| PAK4 | STE20 | STE | 7s47 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 14493 | |
| PAK4 | STE20 | STE | 7s47 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 14494 | |
| PAK4 | STE20 | STE | 7s48 | A | A | - | Human | 14492 | |
| PAK4 | STE20 | STE | 7s48 | A | B | - | Human | 14491 | |
| PAK4 | STE20 | STE | 8ahg | A | A | ~{n}-methyl-3-propan-2-yl-1~{h}-pyrazolo[3,4-c]pyridine-4-carboxamide | Human | 14370 | |
| PAK4 | STE20 | STE | 8ahg | A | B | ~{n}-methyl-3-propan-2-yl-1~{h}-pyrazolo[3,4-c]pyridine-4-carboxamide | Human | 14368 | |
| PAK4 | STE20 | STE | 8ahh | A | A | 5-cyano-~{n}-methyl-pyrazolo[1,5-a]pyridine-3-carboxamide | Human | 14372 | |
| PAK4 | STE20 | STE | 8ahh | A | B | 5-cyano-~{n}-methyl-pyrazolo[1,5-a]pyridine-3-carboxamide | Human | 14371 | |
| PAK4 | STE20 | STE | 8ahi | A | | ~{n}-methyl-1,3-benzothiazole-6-carboxamide | Human | 14369 | |
| PAK4 | STE20 | STE | 8yhk | A | | - | Human | 15260 | |
| PAK5 | STE20 | STE | 2f57 | A | A | - | Human | 200 | |
| PAK5 | STE20 | STE | 2f57 | A | B | - | Human | 202 | |
| PAK5 | STE20 | STE | 2f57 | B | A | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 199 | |
| PAK5 | STE20 | STE | 2f57 | B | B | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 201 | |
| PAK5 | STE20 | STE | 8c12 | A | A | - | Human | 14952 | |
| PAK5 | STE20 | STE | 8c12 | A | B | - | Human | 14953 | |
| PAK6 | STE20 | STE | 2c30 | A | A | - | Human | 4679 | |
| PAK6 | STE20 | STE | 2c30 | A | B | - | Human | 4678 | |
| PAK6 | STE20 | STE | 4ks7 | A | A | pf-3758309 | Human | 4682 | |
| PAK6 | STE20 | STE | 4ks7 | A | B | pf-3758309 | Human | 4681 | |
| PAK6 | STE20 | STE | 4ks8 | A | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 4683 | |
| PAK6 | STE20 | STE | 4ks8 | A | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 4680 | |
| PASK | CAMKL | CAMK | 3dls | A | | adenosine-5'-diphosphate | Human | 3382 | |
| PASK | CAMKL | CAMK | 3dls | B | | adenosine-5'-diphosphate | Human | 3381 | |
| PASK | CAMKL | CAMK | 3dls | C | | adenosine-5'-diphosphate | Human | 3377 | |
| PASK | CAMKL | CAMK | 3dls | D | | adenosine-5'-diphosphate | Human | 3378 | |
| PASK | CAMKL | CAMK | 3dls | E | | adenosine-5'-diphosphate | Human | 3379 | |
| PASK | CAMKL | CAMK | 3dls | F | | adenosine-5'-diphosphate | Human | 3380 | |
| PBK | TOPK | Other | 5j0a | A | | - | Human | 7083 | |
| PBK | TOPK | Other | 5j0a | B | | - | Human | 7084 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 5grn | A | A | n-[2-(dimethylamino)ethyl]-n-[[4-[[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methyl]pyridine-3-carboxamide | Human | 9479 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 5grn | A | B | n-[2-(dimethylamino)ethyl]-n-[[4-[[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methyl]pyridine-3-carboxamide | Human | 9478 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 5k5x | A | | - | Human | 6962 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 6a32 | A | | - | Human | 11327 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 6joi | A | | 1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amine | Human | 12102 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 6joj | A | | 1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amine | Human | 12104 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 6jok | A | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 12105 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 6jol | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 12103 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 8pqh | A | | (1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15107 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 8pqi | A | A | (1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15109 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 8pqi | A | B | (1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamine | Human | 15104 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 8pqj | A | A | - | Human | 15106 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 8pqj | A | B | - | Human | 15105 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 8pqk | A | A | - | Human | 15110 | |
| PDGFRA (PDGFRa) | PDGFR | TK | 8pqk | A | B | - | Human | 15108 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1h1w | A | A | adenosine-5'-triphosphate | Human | 3186 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1h1w | A | B | adenosine-5'-triphosphate | Human | 3194 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1oky | A | A | staurosporine | Human | 3164 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1oky | A | B | staurosporine | Human | 3195 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1okz | A | | 7-hydroxystaurosporine | Human | 3209 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu3 | A | A | (9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dione | Human | 3180 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu3 | A | B | (9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dione | Human | 3248 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu7 | A | | 3-(1h-indol-3-yl)-4-(1-{2-[(2s)-1-methylpyrrolidinyl]ethyl}-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3224 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu8 | A | A | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3239 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu8 | A | B | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3237 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu9 | A | A | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 6800 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu9 | A | B | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 6799 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uvr | A | | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3193 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1z5m | A | | n-(3-{[5-bromo-2-({3-[(pyrrolidin-1-ylcarbonyl)amino]phenyl}amino)pyrimidin-4-yl]amino}propyl)-2,2-dimethylmalonamide | Human | 3152 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2biy | A | A | adenosine-5'-triphosphate | Human | 3232 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2biy | A | B | adenosine-5'-triphosphate | Human | 3169 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2pe0 | A | | 5-hydroxy-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-2-one | Human | 3206 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2pe1 | A | | 1-{2-oxo-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-5-yl}urea | Human | 3167 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2pe2 | A | | 3-[5-({5-[(aminocarbonyl)amino]-2-oxo-2h-indol-3-yl}methyl)-1h-pyrrol-3-yl]-n-(2-piperidin-1-ylethyl)benzamide | Human | 3163 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2r7b | A | | 10,11-dimethoxy-4-methyldibenzo[c,f]-2,7-naphthyridine-3,6-diamine | Human | 3215 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2xch | A | | 8-(cyclohexa-2,5-dien-1-ylideneamino)-1-(piperidin-4-ylmethyl)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 3220 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2xck | A | | 1-methyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-n-[(2-methylpyridin-4-yl)methyl]-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 3201 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3h9o | A | | 2-(1h-imidazol-1-yl)-9-methoxy-8-(2-methoxyethoxy)benzo[c][2,7]naphthyridin-4-amine | Human | 3226 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3hrc | A | A | adenosine-5'-triphosphate | Human | 3172 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3hrc | A | B | adenosine-5'-triphosphate | Human | 3223 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3hrf | A | A | adenosine-5'-triphosphate | Human | 3170 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3hrf | A | B | adenosine-5'-triphosphate | Human | 3247 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3ion | A | | 2-(5-{[(2s)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amine | Human | 3218 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3iop | A | | 2-(5-{[(2r)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amine | Human | 3204 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nax | A | | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 3200 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nay | A | | 4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-one | Human | 3231 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nay | B | | 4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-one | Human | 3203 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nun | A | A | 6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amine | Human | 3183 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nun | A | B | 6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amine | Human | 3216 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nus | A | A | 1h-indazol-3-amine | Human | 3233 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nus | A | B | 1h-indazol-3-amine | Human | 3185 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nuu | A | A | 3,4-dihydroisoquinolin-1(2h)-one | Human | 3214 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nuu | A | B | 3,4-dihydroisoquinolin-1(2h)-one | Human | 3159 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nuy | A | A | quinazolin-4(1h)-one | Human | 3236 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nuy | A | B | quinazolin-4(1h)-one | Human | 3242 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | A | | - | Human | 3235 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | B | | - | Human | 3178 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | C | | - | Human | 3245 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | D | | - | Human | 3210 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | E | | - | Human | 3202 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | F | | - | Human | 3228 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | G | | - | Human | 3189 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | H | | - | Human | 3177 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | A | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3197 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | A | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3181 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | B | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3160 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | B | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3198 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | C | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3150 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | C | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3243 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | D | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3192 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | D | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3184 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3otu | A | | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3217 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3pwy | A | | n-[2-({6-[(2-sulfanylethyl)amino]pyrimidin-4-yl}amino)ethyl]propanamide | Human | 3155 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | A | A | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 9254 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | A | B | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 9253 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | B | A | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 9255 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | B | B | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 9256 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcq | A | A | 6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamine | Human | 3205 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcq | A | B | 6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamine | Human | 3166 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcs | A | A | 6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amine | Human | 3179 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcs | A | B | 6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amine | Human | 3157 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcx | A | A | 6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amine | Human | 3187 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcx | A | B | 6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amine | Human | 3249 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcy | A | A | (2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamide | Human | 3151 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcy | A | B | (2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamide | Human | 3161 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd0 | A | A | (3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamide | Human | 3196 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd0 | A | B | (3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamide | Human | 3162 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd3 | A | A | tert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamate | Human | 3188 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd3 | A | B | tert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamate | Human | 3171 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd4 | A | A | tert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamate | Human | 3225 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd4 | A | B | tert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamate | Human | 3190 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3rcj | A | | 3-(1-benzyl-1h-1,2,3-triazol-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 3154 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3rwp | A | A | [4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanone | Human | 3208 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3rwp | A | B | [4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanone | Human | 3199 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3rwq | A | | [4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[2-(pyridin-3-yl)ethyl]amino}pyrazin-2-yl)methanone | Human | 3213 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3sc1 | A | | 6-[2-(hydroxymethyl)phenyl]isoquinolin-1(2h)-one | Human | 3173 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4a06 | A | A | adenosine-5'-triphosphate | Human | 3207 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4a06 | A | B | adenosine-5'-triphosphate | Human | 3227 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4a07 | A | A | adenosine-5'-triphosphate | Human | 3234 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4a07 | A | B | adenosine-5'-triphosphate | Human | 3238 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4aw0 | A | A | adenosine-5'-triphosphate | Human | 3176 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4aw0 | A | B | adenosine-5'-triphosphate | Human | 3241 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4aw1 | A | A | adenosine-5'-triphosphate | Human | 3229 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4aw1 | A | B | adenosine-5'-triphosphate | Human | 3221 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4ct1 | A | A | adenosine-5'-triphosphate | Human | 3158 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4ct1 | A | B | adenosine-5'-triphosphate | Human | 3168 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4ct2 | A | A | adenosine-5'-triphosphate | Human | 3153 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4ct2 | A | B | adenosine-5'-triphosphate | Human | 3230 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqk | A | A | adenosine-5'-triphosphate | Human | 3175 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqk | A | B | adenosine-5'-triphosphate | Human | 3156 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqk | A | C | adenosine-5'-triphosphate | Human | 3211 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqv | A | A | adenosine-5'-triphosphate | Human | 3219 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqv | A | B | adenosine-5'-triphosphate | Human | 3182 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqv | A | C | adenosine-5'-triphosphate | Human | 3222 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rrv | A | A | adenosine-5'-triphosphate | Human | 3244 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rrv | A | B | adenosine-5'-triphosphate | Human | 3212 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rrv | A | C | adenosine-5'-triphosphate | Human | 3191 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4xx9 | A | A | adenosine-5'-triphosphate | Human | 6193 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4xx9 | A | B | adenosine-5'-triphosphate | Human | 6192 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ack | A | A | adenosine-5'-triphosphate | Human | 6191 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ack | A | B | adenosine-5'-triphosphate | Human | 6194 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5hkm | A | | 4-ethyl-6-[5-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-2-amine | Human | 6670 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5hng | A | | 6-methoxy-2-(1h-pyrazol-5-yl)-1h-benzimidazole | Human | 6675 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ho7 | A | A | 5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamide | Human | 6673 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ho7 | A | B | 5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamide | Human | 6671 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ho8 | A | A | 4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 6674 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ho8 | A | B | 4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 6672 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvl | A | A | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | 7106 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvl | A | B | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | 7110 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvm | A | A | adenine | Human | 7112 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvm | A | B | adenine | Human | 7103 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvm | A | C | adenine | Human | 7138 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvn | A | A | adenosine | Human | 7105 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvn | A | B | adenosine | Human | 7109 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvo | A | A | adenosine-5'-triphosphate | Human | 7104 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvo | A | B | adenosine-5'-triphosphate | Human | 7114 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvp | A | | adenosine-5'-triphosphate | Human | 7102 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvp | B | | adenosine-5'-triphosphate | Human | 7113 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvp | C | | adenosine-5'-triphosphate | Human | 7111 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvp | D | | adenosine-5'-triphosphate | Human | 7108 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5mrd | A | A | adenosine-5'-triphosphate | Human | 7395 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5mrd | A | B | adenosine-5'-triphosphate | Human | 7394 | |
| PDPK1 (PDK1) | PDK1 | AGC | 8dqt | A | | - | Human | 14812 | |
| PEAK1 (SgK269) | NKF3 | Other | 6bhc | A | A | - | Human | 9068 | |
| PEAK1 (SgK269) | NKF3 | Other | 6bhc | A | B | - | Human | 9067 | |
| PHKG1 (PHKg1) | PHK | CAMK | 8jfl | B | | - | Human | 15265 | |
| PHKG1 (PHKg1) | PHK | CAMK | 8xyb | C | | - | Human | 15264 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | A | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1894 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | A | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1893 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | B | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1897 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | B | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1895 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | C | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1896 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | C | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1900 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | D | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1898 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | D | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1899 | |
| PI4K2A | PIK | Atypical | 4hnd | A | | adenosine-5'-diphosphate | Human | 9265 | |
| PI4K2A | PIK | Atypical | 4hnd | B | | adenosine-5'-diphosphate | Human | 9261 | |
| PI4K2A | PIK | Atypical | 4hne | A | | adenosine-5'-diphosphate | Human | 9262 | |
| PI4K2A | PIK | Atypical | 4hne | B | | adenosine-5'-diphosphate | Human | 9263 | |
| PI4K2A | PIK | Atypical | 4pla | A | | adenosine-5'-triphosphate | Human | 9259 | |
| PI4K2A | PIK | Atypical | 4yc4 | A | | [(1s,3s,4s)-3-(6-amino-9h-purin-9-yl)bicyclo[2.2.1]hept-1-yl]methanol | Human | 9258 | |
| PI4K2A | PIK | Atypical | 5eut | A | | - | Human | 9264 | |
| PI4K2A | PIK | Atypical | 5i0n | A | A | adenosine-5'-triphosphate | Human | 9260 | |
| PI4K2A | PIK | Atypical | 5i0n | A | B | adenosine-5'-triphosphate | Human | 9257 | |
| PI4K2B | PIK | Atypical | 4wtv | A | A | adenosine-5'-triphosphate | Human | 9095 | |
| PI4K2B | PIK | Atypical | 4wtv | A | B | adenosine-5'-triphosphate | Human | 9098 | |
| PI4K2B | PIK | Atypical | 4wtv | B | A | adenosine-5'-triphosphate | Human | 9097 | |
| PI4K2B | PIK | Atypical | 4wtv | B | B | adenosine-5'-triphosphate | Human | 9096 | |
| PI4K2B | PIK | Atypical | 8a5x | A | | 4-azanyl-7-[3-(hydroxymethyl)phenyl]quinazoline-6-carboxamide | Human | 14384 | |
| PI4KA | PIK | Atypical | 6bq1 | A | | 5-{2-amino-1-[4-(morpholin-4-yl)phenyl]-1h-benzimidazol-6-yl}-n-(2-fluorophenyl)-2-methoxypyridine-3-sulfonamide | Human | 9070 | |
| PI4KA | PIK | Atypical | 6bq1 | E | | 5-{2-amino-1-[4-(morpholin-4-yl)phenyl]-1h-benzimidazol-6-yl}-n-(2-fluorophenyl)-2-methoxypyridine-3-sulfonamide | Human | 9069 | |
| PI4KB | PIK | Atypical | 4d0l | A | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9152 | |
| PI4KB | PIK | Atypical | 4d0l | C | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9143 | |
| PI4KB | PIK | Atypical | 4d0l | E | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9139 | |
| PI4KB | PIK | Atypical | 4d0m | A | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9136 | |
| PI4KB | PIK | Atypical | 4d0m | c | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9148 | |
| PI4KB | PIK | Atypical | 4d0m | C | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9153 | |
| PI4KB | PIK | Atypical | 4d0m | g | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9146 | |
| PI4KB | PIK | Atypical | 4d0m | G | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9134 | |
| PI4KB | PIK | Atypical | 4d0m | I | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9151 | |
| PI4KB | PIK | Atypical | 4d0m | M | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9138 | |
| PI4KB | PIK | Atypical | 4d0m | O | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9154 | |
| PI4KB | PIK | Atypical | 4d0m | Q | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9145 | |
| PI4KB | PIK | Atypical | 4d0m | S | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9142 | |
| PI4KB | PIK | Atypical | 4d0m | W | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9155 | |
| PI4KB | PIK | Atypical | 4d0m | Y | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9133 | |
| PI4KB | PIK | Atypical | 4wae | A | | adenosine-5'-triphosphate | Human | 9144 | |
| PI4KB | PIK | Atypical | 4wag | A | | 6-chloro-3-(3,4-dimethoxyphenyl)-2-methylimidazo[1,2-b]pyridazin-8-amine | Human | 9137 | |
| PI4KB | PIK | Atypical | 5c46 | E | | - | Human | 9141 | |
| PI4KB | PIK | Atypical | 5c4g | E | | n~2~-[7-(3,4-dimethoxyphenyl)quinoxalin-2-yl]-n-methylglycinamide | Human | 9135 | |
| PI4KB | PIK | Atypical | 5euq | E | | ~{n}-[5-[3-[[(4-hydroxyphenyl)amino]-bis(oxidanyl)-$l^{4}-sulfanyl]-4-methoxy-phenyl]-4-methyl-1,3-thiazol-2-yl]cyclopentanecarboxamide | Human | 9132 | |
| PI4KB | PIK | Atypical | 5fbl | A | | ~{n}-[2-[[6-chloranyl-3-(4-methoxy-3-morpholin-4-ylsulfonyl-phenyl)-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamide | Human | 9150 | |
| PI4KB | PIK | Atypical | 5fbq | A | | ~{n}-[2-[[6-chloranyl-3-[3-[4-(hydroxymethyl)piperidin-1-yl]sulfonyl-4-methoxy-phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamide | Human | 9131 | |
| PI4KB | PIK | Atypical | 5fbr | A | | ~{n}-[2-[[3-[3-[(4-azanylcyclohexyl)sulfamoyl]-4-methoxy-phenyl]-6-chloranyl-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamide | Human | 9140 | |
| PI4KB | PIK | Atypical | 5fbv | A | | ~{n}-[2-[[6-chloranyl-3-[3-(2-hydroxyethylsulfamoyl)-4-methoxy-phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamide | Human | 9147 | |
| PI4KB | PIK | Atypical | 5fbw | A | | ~{n}-[2-[[6-chloranyl-3-[4-methoxy-3-[[(2~{r})-1-oxidanylbutan-2-yl]sulfamoyl]phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamide | Human | 9149 | |
| PI4KB | PIK | Atypical | 6gl3 | A | | (3~{s})-4-(6-azanyl-1-methyl-pyrazolo[3,4-d]pyrimidin-4-yl)-~{n}-(4-methoxy-2-methyl-phenyl)-3-methyl-piperazine-1-carboxamide | Human | 10442 | |
| PI4KB | PIK | Atypical | 6gl3 | B | | - | Human | 10443 | |
| PI4KB | PIK | Atypical | 8q6f | A | A | 3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidine | Human | 15018 | |
| PI4KB | PIK | Atypical | 8q6f | A | B | 3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidine | Human | 15013 | |
| PI4KB | PIK | Atypical | 8q6f | A | C | 3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidine | Human | 15011 | |
| PI4KB | PIK | Atypical | 8q6g | A | A | 3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidine | Human | 15014 | |
| PI4KB | PIK | Atypical | 8q6g | A | B | 3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidine | Human | 15012 | |
| PI4KB | PIK | Atypical | 8q6g | A | C | 3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidine | Human | 15016 | |
| PI4KB | PIK | Atypical | 8q6h | A | A | 3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidine | Human | 15015 | |
| PI4KB | PIK | Atypical | 8q6h | A | B | 3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidine | Human | 15017 | |
| PI4KB | PIK | Atypical | 8vof | A | | methyl 2-chloro-5-(methyl{(8r)-3-[4-(methylcarbamoyl)phenyl]pyrazolo[1,5-a]pyridine-5-carbonyl}amino)benzoate | Human | 15377 | |
| Pik3c2a | PIP | Atypical | 7bi2 | A | A | 9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-one | Mouse | 14153 | |
| Pik3c2a | PIP | Atypical | 7bi2 | A | B | 9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-one | Mouse | 14151 | |
| Pik3c2a | PIP | Atypical | 7bi4 | A | A | - | Mouse | 14155 | |
| Pik3c2a | PIP | Atypical | 7bi4 | A | B | - | Mouse | 14156 | |
| Pik3c2a | PIP | Atypical | 7bi6 | A | A | adenosine-5'-triphosphate | Mouse | 14154 | |
| Pik3c2a | PIP | Atypical | 7bi6 | A | B | adenosine-5'-triphosphate | Mouse | 14149 | |
| Pik3c2a | PIP | Atypical | 7bi9 | A | A | n-(2,3-dihydro-7,8-dimethoxyimidazo[1,2-c] quinazolin-5-yl)nicotinamide | Mouse | 14150 | |
| Pik3c2a | PIP | Atypical | 7bi9 | A | B | n-(2,3-dihydro-7,8-dimethoxyimidazo[1,2-c] quinazolin-5-yl)nicotinamide | Mouse | 14152 | |
| Pik3c2a | PIP | Atypical | 7z74 | A | A | ~{n}-[4-(3-hydroxyphenyl)-1,3-thiazol-2-yl]-2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-ethanamide | Mouse | 14360 | |
| Pik3c2a | PIP | Atypical | 7z74 | A | B | ~{n}-[4-(3-hydroxyphenyl)-1,3-thiazol-2-yl]-2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-ethanamide | Mouse | 14357 | |
| Pik3c2a | PIP | Atypical | 7z75 | A | | ~{n}-[4-[3-(methylsulfonylamino)phenyl]-1,3-thiazol-2-yl]-2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-ethanamide | Mouse | 14359 | |
| Pik3c2a | PIP | Atypical | 8a9i | A | A | 2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-~{n}-(1,3-thiazol-2-yl)ethanamide | Mouse | 14361 | |
| Pik3c2a | PIP | Atypical | 8a9i | A | B | 2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-~{n}-(1,3-thiazol-2-yl)ethanamide | Mouse | 14358 | |
| PIK3C3 | PIK | Atypical | 3ihy | A | | - | Human | 9341 | |
| PIK3C3 | PIK | Atypical | 3ihy | B | | - | Human | 9336 | |
| PIK3C3 | PIK | Atypical | 3ihy | C | | - | Human | 9331 | |
| PIK3C3 | PIK | Atypical | 3ihy | D | | - | Human | 9337 | |
| PIK3C3 | PIK | Atypical | 3ihy | E | | - | Human | 9344 | |
| PIK3C3 | PIK | Atypical | 3ls8 | A | A | - | Human | 9340 | |
| PIK3C3 | PIK | Atypical | 3ls8 | A | B | - | Human | 9348 | |
| PIK3C3 | PIK | Atypical | 3ls8 | B | A | - | Human | 9333 | |
| PIK3C3 | PIK | Atypical | 3ls8 | B | B | - | Human | 9339 | |
| PIK3C3 | PIK | Atypical | 4oys | A | | (8s)-9-[(5-chloranylpyridin-3-yl)methyl]-2-[(3r)-3-methylmorpholin-4-yl]-8-(trifluoromethyl)-6,7,8,9a-tetrahydro-3h-pyrimido[1,2-a]pyrimidin-4-one | Human | 9327 | |
| PIK3C3 | PIK | Atypical | 4ph4 | B | A | - | Human | 9326 | |
| PIK3C3 | PIK | Atypical | 4ph4 | B | B | - | Human | 9330 | |
| PIK3C3 | PIK | Atypical | 4uwf | A | | - | Human | 9328 | |
| PIK3C3 | PIK | Atypical | 4uwg | A | A | - | Human | 9347 | |
| PIK3C3 | PIK | Atypical | 4uwg | A | B | - | Human | 9350 | |
| PIK3C3 | PIK | Atypical | 4uwh | A | A | - | Human | 9346 | |
| PIK3C3 | PIK | Atypical | 4uwh | A | B | - | Human | 9334 | |
| PIK3C3 | PIK | Atypical | 4uwk | A | A | - | Human | 9342 | |
| PIK3C3 | PIK | Atypical | 4uwk | A | B | - | Human | 9335 | |
| PIK3C3 | PIK | Atypical | 4uwl | A | | - | Human | 9332 | |
| PIK3C3 | PIK | Atypical | 5anl | A | | (8s)-2-(morpholin-4-yl)-9-[2-(propan-2-yloxy)ethyl]-8-(trifluoromethyl)-6,7,8,9-tetrahydro-4h-pyrimido[1,2-a]pyrimidin-4-one | Human | 9349 | |
| PIK3C3 | PIK | Atypical | 5enn | A | A | 1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-ol | Human | 9343 | |
| PIK3C3 | PIK | Atypical | 5enn | A | B | 1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-ol | Human | 9338 | |
| PIK3C3 | PIK | Atypical | 5enn | B | A | 1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-ol | Human | 9345 | |
| PIK3C3 | PIK | Atypical | 5enn | B | B | 1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-ol | Human | 9329 | |
| PIK3C3 | PIK | Atypical | 6i3u | A | | 2-morpholin-4-yl-6-[7-[(2~{r})-1-morpholin-4-ylpropan-2-yl]oxy-9~{h}-thioxanthen-4-yl]pyran-4-one | Human | 11292 | |
| PIK3C3 | PIK | Atypical | 6ykg | A | | 4-morpholin-4-yl-6-[(2~{r})-2-(phenylmethyl)pyrrolidin-1-yl]-1~{h}-pyridin-2-one | Human | 13509 | |
| PIK3C3 | PIK | Atypical | 7bl1 | B | | - | Human | 13361 | |
| PIK3C3 | PIK | Atypical | 7rsj | A | A | n-{4-[(7r,8r)-4-oxo-7-(propan-2-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]pyridin-2-yl}cyclopropanecarboxamide | Human | 13983 | |
| PIK3C3 | PIK | Atypical | 7rsj | A | B | n-{4-[(7r,8r)-4-oxo-7-(propan-2-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]pyridin-2-yl}cyclopropanecarboxamide | Human | 13982 | |
| PIK3C3 | PIK | Atypical | 7rsp | A | A | (7r,8r)-2-[(3r)-3-methylmorpholin-4-yl]-7-(propan-2-yl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5h)-one | Human | 13981 | |
| PIK3C3 | PIK | Atypical | 7rsp | A | B | (7r,8r)-2-[(3r)-3-methylmorpholin-4-yl]-7-(propan-2-yl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5h)-one | Human | 13986 | |
| PIK3C3 | PIK | Atypical | 7rsv | A | A | (5as,8ar,9s)-2-[(3r)-3-methylmorpholin-4-yl]-5,5a,6,7,8,8a-hexahydro-4h-cyclopenta[e]pyrazolo[1,5-a]pyrazin-4-one | Human | 13985 | |
| PIK3C3 | PIK | Atypical | 7rsv | A | B | (5as,8ar,9s)-2-[(3r)-3-methylmorpholin-4-yl]-5,5a,6,7,8,8a-hexahydro-4h-cyclopenta[e]pyrazolo[1,5-a]pyrazin-4-one | Human | 13984 | |
| PIK3C3 | PIK | Atypical | 8sor | A | | - | Human | 14803 | |
| Pik3ca (p110a) | PIK | Atypical | 4a55 | A | | pik-108 | Mouse | 9403 | |
| PIK3CA (p110a) | PIK | Atypical | 2rd0 | A | | - | Human | 9287 | |
| PIK3CA (p110a) | PIK | Atypical | 3hhm | A | | (1s,6br,9as,11r,11br)-9a,11b-dimethyl-1-[(methyloxy)methyl]-3,6,9-trioxo-1,6,6b,7,8,9,9a,10,11,11b-decahydro-3h-furo[4,3,2-de]indeno[4,5-h][2]benzopyran-11-yl acetate | Human | 9275 | |
| PIK3CA (p110a) | PIK | Atypical | 3hiz | A | | - | Human | 9311 | |
| PIK3CA (p110a) | PIK | Atypical | 3zim | A | | 1-[4-[[2-(1h-indazol-4-yl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidin-6-yl]methyl]piperazin-1-yl]-6-methyl-hept-5-ene-1,4-dione | Human | 9294 | |
| PIK3CA (p110a) | PIK | Atypical | 4jps | A | A | (2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamide | Human | 9317 | |
| PIK3CA (p110a) | PIK | Atypical | 4jps | A | B | (2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamide | Human | 9314 | |
| PIK3CA (p110a) | PIK | Atypical | 4l1b | A | | - | Human | 9292 | |
| PIK3CA (p110a) | PIK | Atypical | 4l23 | A | | 3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenol | Human | 9290 | |
| PIK3CA (p110a) | PIK | Atypical | 4l2y | A | | 3-amino-5-[4-(morpholin-4-yl)pyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl]phenol | Human | 9276 | |
| PIK3CA (p110a) | PIK | Atypical | 4ovu | A | A | - | Human | 9291 | |
| PIK3CA (p110a) | PIK | Atypical | 4ovu | A | B | - | Human | 9271 | |
| PIK3CA (p110a) | PIK | Atypical | 4ovv | A | | - | Human | 9307 | |
| PIK3CA (p110a) | PIK | Atypical | 4tuu | A | | - | Human | 9281 | |
| PIK3CA (p110a) | PIK | Atypical | 4tv3 | A | | 2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9278 | |
| PIK3CA (p110a) | PIK | Atypical | 4waf | A | A | n,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamide | Human | 9288 | |
| PIK3CA (p110a) | PIK | Atypical | 4waf | A | B | n,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamide | Human | 9272 | |
| PIK3CA (p110a) | PIK | Atypical | 4ykn | A | A | 3-(6-methoxypyridin-3-yl)-5-[({4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl}amino)methyl]benzoic acid | Human | 9283 | |
| PIK3CA (p110a) | PIK | Atypical | 4ykn | A | B | 3-(6-methoxypyridin-3-yl)-5-[({4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl}amino)methyl]benzoic acid | Human | 9315 | |
| PIK3CA (p110a) | PIK | Atypical | 4zop | A | A | (2s,3r)-n~1~-(8-tert-butyl-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-2-yl)-3-methylpyrrolidine-1,2-dicarboxamide | Human | 9298 | |
| PIK3CA (p110a) | PIK | Atypical | 4zop | A | B | (2s,3r)-n~1~-(8-tert-butyl-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-2-yl)-3-methylpyrrolidine-1,2-dicarboxamide | Human | 9312 | |
| PIK3CA (p110a) | PIK | Atypical | 5dxh | A | | methyl {2-[4-(2-chlorophenyl)-4h-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl}carbamate | Human | 9310 | |
| PIK3CA (p110a) | PIK | Atypical | 5dxh | D | | methyl {2-[4-(2-chlorophenyl)-4h-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl}carbamate | Human | 9300 | |
| PIK3CA (p110a) | PIK | Atypical | 5dxt | A | | (2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamide | Human | 9299 | |
| PIK3CA (p110a) | PIK | Atypical | 5fi4 | A | A | ~{n}-[6-[5-azanyl-6-[(2~{s})-1,1,1-tris(fluoranyl)propan-2-yl]oxy-pyrazin-2-yl]imidazo[1,2-a]pyridin-2-yl]ethanamide | Human | 9302 | |
| PIK3CA (p110a) | PIK | Atypical | 5fi4 | A | B | ~{n}-[6-[5-azanyl-6-[(2~{s})-1,1,1-tris(fluoranyl)propan-2-yl]oxy-pyrazin-2-yl]imidazo[1,2-a]pyridin-2-yl]ethanamide | Human | 9309 | |
| PIK3CA (p110a) | PIK | Atypical | 5itd | A | | 5-{4-[3-(4-acetylpiperazine-1-carbonyl)phenyl]quinazolin-6-yl}-2-methoxypyridine-3-carbonitrile | Human | 9313 | |
| PIK3CA (p110a) | PIK | Atypical | 5sw8 | A | | - | Human | 9274 | |
| PIK3CA (p110a) | PIK | Atypical | 5swg | A | | - | Human | 9306 | |
| PIK3CA (p110a) | PIK | Atypical | 5swo | A | | - | Human | 9303 | |
| PIK3CA (p110a) | PIK | Atypical | 5swp | A | | - | Human | 9293 | |
| PIK3CA (p110a) | PIK | Atypical | 5swr | A | | - | Human | 9279 | |
| PIK3CA (p110a) | PIK | Atypical | 5swt | A | | - | Human | 9273 | |
| PIK3CA (p110a) | PIK | Atypical | 5sx8 | A | | - | Human | 9269 | |
| PIK3CA (p110a) | PIK | Atypical | 5sx9 | A | | - | Human | 9305 | |
| PIK3CA (p110a) | PIK | Atypical | 5sxa | A | | - | Human | 9285 | |
| PIK3CA (p110a) | PIK | Atypical | 5sxb | A | | - | Human | 9282 | |
| PIK3CA (p110a) | PIK | Atypical | 5sxc | A | | - | Human | 9297 | |
| PIK3CA (p110a) | PIK | Atypical | 5sxd | A | | - | Human | 9304 | |
| PIK3CA (p110a) | PIK | Atypical | 5sxe | A | | - | Human | 9280 | |
| PIK3CA (p110a) | PIK | Atypical | 5sxf | A | | - | Human | 9284 | |
| PIK3CA (p110a) | PIK | Atypical | 5sxi | A | | - | Human | 9270 | |
| PIK3CA (p110a) | PIK | Atypical | 5sxj | A | | - | Human | 9301 | |
| PIK3CA (p110a) | PIK | Atypical | 5sxk | A | | - | Human | 9296 | |
| PIK3CA (p110a) | PIK | Atypical | 5ubr | A | | 1-[4-(3-{4-amino-5-[1-(oxan-4-yl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)piperazin-1-yl]ethan-1-one | Human | 9289 | |
| PIK3CA (p110a) | PIK | Atypical | 5uk8 | A | A | (r)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1h-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholine | Human | 9295 | |
| PIK3CA (p110a) | PIK | Atypical | 5uk8 | A | B | (r)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1h-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholine | Human | 9286 | |
| PIK3CA (p110a) | PIK | Atypical | 5ukj | A | | n,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamide | Human | 9277 | |
| PIK3CA (p110a) | PIK | Atypical | 5ul1 | A | A | 3-amino-6-(4-{[(2s)-1-(dimethylamino)propan-2-yl]sulfonyl}phenyl)-n-phenylpyrazine-2-carboxamide | Human | 9316 | |
| PIK3CA (p110a) | PIK | Atypical | 5ul1 | A | B | 3-amino-6-(4-{[(2s)-1-(dimethylamino)propan-2-yl]sulfonyl}phenyl)-n-phenylpyrazine-2-carboxamide | Human | 9308 | |
| PIK3CA (p110a) | PIK | Atypical | 5xgh | A | | 3-[(4-fluorophenyl)methylamino]-5-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenol | Human | 9864 | |
| PIK3CA (p110a) | PIK | Atypical | 5xgi | A | | 3-azanyl-5-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenol | Human | 9865 | |
| PIK3CA (p110a) | PIK | Atypical | 5xgj | A | | 3-(4-morpholin-4-ylfuro[3,2-d]pyrimidin-2-yl)-5-[(phenylmethyl)amino]phenol | Human | 9863 | |
| PIK3CA (p110a) | PIK | Atypical | 6gvf | A | A | 5-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amine | Human | 11659 | |
| PIK3CA (p110a) | PIK | Atypical | 6gvf | A | B | 5-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amine | Human | 11658 | |
| PIK3CA (p110a) | PIK | Atypical | 6gvg | A | | 5-(6-azanyl-4-methyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amine | Human | 11655 | |
| PIK3CA (p110a) | PIK | Atypical | 6gvh | A | A | 5-(6-azanyl-4-chloranyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amine | Human | 11657 | |
| PIK3CA (p110a) | PIK | Atypical | 6gvh | A | B | 5-(6-azanyl-4-chloranyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amine | Human | 11653 | |
| PIK3CA (p110a) | PIK | Atypical | 6gvi | A | A | 3-(2-azanyl-1,3-benzoxazol-5-yl)-1-propan-2-yl-pyrazolo[3,4-d]pyrimidine-4,6-diamine | Human | 11656 | |
| PIK3CA (p110a) | PIK | Atypical | 6gvi | A | B | 3-(2-azanyl-1,3-benzoxazol-5-yl)-1-propan-2-yl-pyrazolo[3,4-d]pyrimidine-4,6-diamine | Human | 11654 | |
| PIK3CA (p110a) | PIK | Atypical | 6nct | A | | - | Human | 11221 | |
| PIK3CA (p110a) | PIK | Atypical | 6oac | A | | 4-(difluoromethyl)-5-{4-[(3s)-3-methylmorpholin-4-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}pyridin-2-amine | Human | 11381 | |
| PIK3CA (p110a) | PIK | Atypical | 6pys | A | A | (3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-one | Human | 11575 | |
| PIK3CA (p110a) | PIK | Atypical | 6pys | A | B | (3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-one | Human | 11576 | |
| PIK3CA (p110a) | PIK | Atypical | 7jiu | A | A | (3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-one | Human | 13760 | |
| PIK3CA (p110a) | PIK | Atypical | 7jiu | A | B | (3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-one | Human | 13761 | |
| PIK3CA (p110a) | PIK | Atypical | 7k6m | A | A | 2,2-difluoroethyl (3s)-3-{[2'-amino-5-fluoro-2-(morpholin-4-yl)[4,5'-bipyrimidin]-6-yl]amino}-3-(hydroxymethyl)pyrrolidine-1-carboxylate | Human | 13225 | |
| PIK3CA (p110a) | PIK | Atypical | 7k6m | A | B | 2,2-difluoroethyl (3s)-3-{[2'-amino-5-fluoro-2-(morpholin-4-yl)[4,5'-bipyrimidin]-6-yl]amino}-3-(hydroxymethyl)pyrrolidine-1-carboxylate | Human | 13227 | |
| PIK3CA (p110a) | PIK | Atypical | 7k6n | A | A | tert-butyl (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-3-methylpyrrolidine-1-carboxylate | Human | 13226 | |
| PIK3CA (p110a) | PIK | Atypical | 7k6n | A | B | tert-butyl (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-3-methylpyrrolidine-1-carboxylate | Human | 13224 | |
| PIK3CA (p110a) | PIK | Atypical | 7k6o | A | A | (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-n-methylpyrrolidine-1-sulfonamide | Human | 13207 | |
| PIK3CA (p110a) | PIK | Atypical | 7k6o | A | B | (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-n-methylpyrrolidine-1-sulfonamide | Human | 13206 | |
| PIK3CA (p110a) | PIK | Atypical | 7k71 | A | | 2-(morpholin-4-yl)[4,5'-bipyrimidin]-2'-amine | Human | 13219 | |
| PIK3CA (p110a) | PIK | Atypical | 7mlk | A | A | 4-[6-(3,4,5-trimethoxyanilino)pyrazin-2-yl]benzamide | Human | 14216 | |
| PIK3CA (p110a) | PIK | Atypical | 7mlk | A | B | 4-[6-(3,4,5-trimethoxyanilino)pyrazin-2-yl]benzamide | Human | 14217 | |
| PIK3CA (p110a) | PIK | Atypical | 7myn | A | A | - | Human | 13963 | |
| PIK3CA (p110a) | PIK | Atypical | 7myn | A | B | - | Human | 13964 | |
| PIK3CA (p110a) | PIK | Atypical | 7myo | B | A | - | Human | 13962 | |
| PIK3CA (p110a) | PIK | Atypical | 7myo | B | B | - | Human | 13965 | |
| PIK3CA (p110a) | PIK | Atypical | 7pg5 | A | A | - | Human | 14346 | |
| PIK3CA (p110a) | PIK | Atypical | 7pg5 | A | B | - | Human | 14347 | |
| PIK3CA (p110a) | PIK | Atypical | 7pg6 | A | A | (2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamide | Human | 14348 | |
| PIK3CA (p110a) | PIK | Atypical | 7pg6 | A | B | (2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamide | Human | 14349 | |
| PIK3CA (p110a) | PIK | Atypical | 7r9v | A | | n-[2-(4-{4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethyl]-1-(prop-2-enoyl)piperidine-4-carboxamide | Human | 14178 | |
| PIK3CA (p110a) | PIK | Atypical | 7r9y | A | | n-[2-(4-{4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethyl]-n-methyl-1-(prop-2-enoyl)piperidine-4-carboxamide | Human | 14179 | |
| PIK3CA (p110a) | PIK | Atypical | 7tz7 | A | A | (4s,5r)-3-[2'-amino-2-(morpholin-4-yl)-4'-(trifluoromethyl)[4,5'-bipyrimidin]-6-yl]-4-(hydroxymethyl)-5-methyl-1,3-oxazolidin-2-one | Human | 14223 | |
| PIK3CA (p110a) | PIK | Atypical | 7tz7 | A | B | (4s,5r)-3-[2'-amino-2-(morpholin-4-yl)-4'-(trifluoromethyl)[4,5'-bipyrimidin]-6-yl]-4-(hydroxymethyl)-5-methyl-1,3-oxazolidin-2-one | Human | 14222 | |
| PIK3CA (p110a) | PIK | Atypical | 8am0 | A | | (2r)-2-[[2-[(4s)-4-[bis(fluoranyl)methyl]-2-oxidanylidene-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl]amino]propanamide | Human | 15083 | |
| PIK3CA (p110a) | PIK | Atypical | 8bfu | A | | - | Human | 14613 | |
| PIK3CA (p110a) | PIK | Atypical | 8dcp | A | A | - | Human | 14380 | |
| PIK3CA (p110a) | PIK | Atypical | 8dcp | A | B | - | Human | 14376 | |
| PIK3CA (p110a) | PIK | Atypical | 8dcx | A | | - | Human | 14377 | |
| PIK3CA (p110a) | PIK | Atypical | 8dd4 | A | A | - | Human | 14378 | |
| PIK3CA (p110a) | PIK | Atypical | 8dd4 | A | B | - | Human | 14379 | |
| PIK3CA (p110a) | PIK | Atypical | 8dd8 | A | | - | Human | 14375 | |
| PIK3CA (p110a) | PIK | Atypical | 8exl | A | A | 2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamide | Human | 14537 | |
| PIK3CA (p110a) | PIK | Atypical | 8exl | A | B | 2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamide | Human | 14536 | |
| PIK3CA (p110a) | PIK | Atypical | 8exo | A | A | 1-{(4s,11am)-2-[(4r)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-prolinamide | Human | 14541 | |
| PIK3CA (p110a) | PIK | Atypical | 8exo | A | B | 1-{(4s,11am)-2-[(4r)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-prolinamide | Human | 14534 | |
| PIK3CA (p110a) | PIK | Atypical | 8exu | A | A | (2s)-2-cyclopropyl-2-({(4s,11am)-2-[(4s)-2-oxo-4-(trifluoromethyl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}amino)acetamide | Human | 14539 | |
| PIK3CA (p110a) | PIK | Atypical | 8exu | A | B | (2s)-2-cyclopropyl-2-({(4s,11am)-2-[(4s)-2-oxo-4-(trifluoromethyl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}amino)acetamide | Human | 14544 | |
| PIK3CA (p110a) | PIK | Atypical | 8exv | A | A | n~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamide | Human | 14542 | |
| PIK3CA (p110a) | PIK | Atypical | 8exv | A | B | n~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamide | Human | 14538 | |
| PIK3CA (p110a) | PIK | Atypical | 8gua | A | | (2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamide | Human | 14540 | |
| PIK3CA (p110a) | PIK | Atypical | 8gub | A | | (2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamide | Human | 14543 | |
| PIK3CA (p110a) | PIK | Atypical | 8gud | A | A | (2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamide | Human | 14535 | |
| PIK3CA (p110a) | PIK | Atypical | 8ilr | A | B | n-[(2s)-1-(ethylamino)-1-oxidanylidene-3-[4-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamide | Human | 14973 | |
| PIK3CA (p110a) | PIK | Atypical | 8ils | A | B | n-[(2r)-1-(ethylamino)-1-oxidanylidene-3-[4-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamide | Human | 14968 | |
| PIK3CA (p110a) | PIK | Atypical | 8ilv | A | | n-[(2r)-1-(ethylamino)-1-oxidanylidene-3-[3-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamide | Human | 14974 | |
| PIK3CA (p110a) | PIK | Atypical | 8ow2 | A | A | - | Human | 14765 | |
| PIK3CA (p110a) | PIK | Atypical | 8ow2 | A | B | - | Human | 14764 | |
| PIK3CA (p110a) | PIK | Atypical | 8sbc | A | A | (2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(pyridin-2-yl)-1h-imidazo[4,5-b]pyridine | Human | 14841 | |
| PIK3CA (p110a) | PIK | Atypical | 8sbc | A | B | (2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(pyridin-2-yl)-1h-imidazo[4,5-b]pyridine | Human | 14842 | |
| PIK3CA (p110a) | PIK | Atypical | 8sbj | A | A | (2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(1h-pyrazol-3-yl)-3h-imidazo[4,5-b]pyridine | Human | 14839 | |
| PIK3CA (p110a) | PIK | Atypical | 8sbj | A | B | (2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(1h-pyrazol-3-yl)-3h-imidazo[4,5-b]pyridine | Human | 14840 | |
| PIK3CA (p110a) | PIK | Atypical | 8tdu | A | A | n~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamide | Human | 14967 | |
| PIK3CA (p110a) | PIK | Atypical | 8tdu | A | B | n~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamide | Human | 14969 | |
| PIK3CA (p110a) | PIK | Atypical | 8tgd | A | A | n~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamide | Human | 14972 | |
| PIK3CA (p110a) | PIK | Atypical | 8tgd | A | B | n~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamide | Human | 14970 | |
| PIK3CA (p110a) | PIK | Atypical | 8ts7 | A | | - | Human | 15088 | |
| PIK3CA (p110a) | PIK | Atypical | 8ts8 | A | | - | Human | 15086 | |
| PIK3CA (p110a) | PIK | Atypical | 8ts9 | A | | - | Human | 15089 | |
| PIK3CA (p110a) | PIK | Atypical | 8tsa | A | | - | Human | 15087 | |
| PIK3CA (p110a) | PIK | Atypical | 8tsb | A | | - | Human | 15085 | |
| PIK3CA (p110a) | PIK | Atypical | 8tsc | A | | - | Human | 15084 | |
| PIK3CA (p110a) | PIK | Atypical | 8tsd | A | | - | Human | 15090 | |
| PIK3CA (p110a) | PIK | Atypical | 8tu6 | A | | - | Human | 14971 | |
| PIK3CA (p110a) | PIK | Atypical | 8twy | A | | n-[4-[5-(1,2,4-oxadiazol-3-yl)thiophen-2-yl]pyridin-2-yl]cyclopropanecarboxamide | Human | 15392 | |
| PIK3CA (p110a) | PIK | Atypical | 8v8h | A | | (2s)-n~1~-[(4p)-2-tert-butyl-4'-methyl[4,5'-bi-1,3-thiazol]-2'-yl]pyrrolidine-1,2-dicarboxamide | Human | 15249 | |
| PIK3CA (p110a) | PIK | Atypical | 8v8i | A | | (2s)-n~1~-[(4p)-2-tert-butyl-4'-methyl[4,5'-bi-1,3-thiazol]-2'-yl]pyrrolidine-1,2-dicarboxamide | Human | 15248 | |
| PIK3CA (p110a) | PIK | Atypical | 8v8j | A | | (2s)-n~1~-[(4p)-2-tert-butyl-4'-methyl[4,5'-bi-1,3-thiazol]-2'-yl]pyrrolidine-1,2-dicarboxamide | Human | 15251 | |
| PIK3CA (p110a) | PIK | Atypical | 8v8u | A | | (2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamide | Human | 15250 | |
| PIK3CA (p110a) | PIK | Atypical | 8v8v | A | | (2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamide | Human | 15252 | |
| PIK3CA (p110a) | PIK | Atypical | 8w9a | A | | - | Human | 15274 | |
| PIK3CA (p110a) | PIK | Atypical | 8w9b | A | | - | Human | 15273 | |
| Pik3cb (p110b) | PIK | Atypical | 2y3a | A | | 2-(1h-indazol-4-yl)-6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-yl-thieno[3,2-d]pyrimidine | Mouse | 9402 | |
| Pik3cb (p110b) | PIK | Atypical | 4bfr | A | | 2-[2-(2-methyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-6-morpholin-4-yl-3h-pyrimidin-4-one | Mouse | 9400 | |
| Pik3cb (p110b) | PIK | Atypical | 4bfr | B | | 2-[2-(2-methyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-6-morpholin-4-yl-3h-pyrimidin-4-one | Mouse | 9401 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxf | A | A | 2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-one | Mouse | 9355 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxf | A | B | 2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-one | Mouse | 9352 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxg | A | | 2-{[4-amino-3-(3-fluoro-5-hydroxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-one | Mouse | 9395 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxh | A | | 2-{[4-amino-3-(3-fluoro-4-hydroxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-one | Mouse | 9387 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxi | A | | 2-{[4-amino-3-(3-hydroxyprop-1-yn-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-one | Mouse | 9373 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxj | A | | n-[6-(4-amino-1-{[2-(4-methylpiperazin-1-yl)quinolin-3-yl]methyl}-1h-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Mouse | 9375 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxk | A | | 3-(2-amino-1,3-benzothiazol-6-yl)-1-{[2-(4-methylpiperazin-1-yl)quinolin-3-yl]methyl}-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Mouse | 9382 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxl | A | A | 2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-1h-benzimidazole | Mouse | 9376 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxl | A | B | 2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-1h-benzimidazole | Mouse | 9389 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxm | A | | 1-(1-methylethyl)-3-(pyridin-3-ylethynyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Mouse | 9359 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxn | A | | 3-{[4-amino-1-(1-methylethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]ethynyl}phenol | Mouse | 9365 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxo | A | A | n-(3-{[(1z)-3,5-dimethoxycyclohexa-2,4-dien-1-ylidene]amino}quinoxalin-2-yl)-4-fluorobenzenesulfonamide | Mouse | 9381 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxo | A | B | n-(3-{[(1z)-3,5-dimethoxycyclohexa-2,4-dien-1-ylidene]amino}quinoxalin-2-yl)-4-fluorobenzenesulfonamide | Mouse | 9361 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxp | A | | 2-(1h-indazol-4-yl)-6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-yl-thieno[3,2-d]pyrimidine | Mouse | 9366 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxq | A | | 2-{[3-(2-methoxyphenyl)-4-oxo-3,4,5,6,7,8-hexahydroquinazolin-2-yl]sulfanyl}-n-quinoxalin-6-ylacetamide | Mouse | 9393 | |
| Pik3cd (p110d) | PIK | Atypical | 2wxr | A | | - | Mouse | 9385 | |
| Pik3cd (p110d) | PIK | Atypical | 2x38 | A | A | 2-[(6-amino-9h-purin-9-yl)methyl]-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-one | Mouse | 9369 | |
| Pik3cd (p110d) | PIK | Atypical | 2x38 | A | B | 2-[(6-amino-9h-purin-9-yl)methyl]-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-one | Mouse | 9380 | |
| Pik3cd (p110d) | PIK | Atypical | 4ajw | A | | 2-[(1-methyl-1h-benzimidazol-2-yl)methyl]-6-morpholin-4-ylpyrimidin-4(3h)-one | Mouse | 9364 | |
| Pik3cd (p110d) | PIK | Atypical | 4ajw | B | | 2-[(1-methyl-1h-benzimidazol-2-yl)methyl]-6-morpholin-4-ylpyrimidin-4(3h)-one | Mouse | 9360 | |
| Pik3cd (p110d) | PIK | Atypical | 4v0i | A | | 2-[2-(2-methyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-6-morpholin-4-yl-3h-pyrimidin-4-one | Mouse | 9399 | |
| Pik3cd (p110d) | PIK | Atypical | 4v0i | B | | 2-[2-(2-methyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-6-morpholin-4-yl-3h-pyrimidin-4-one | Mouse | 9384 | |
| Pik3cd (p110d) | PIK | Atypical | 4xe0 | A | | 5-fluoro-3-phenyl-2-[(1s)-1-(7h-purin-6-ylamino)propyl]quinazolin-4(3h)-one | Mouse | 9368 | |
| Pik3cd (p110d) | PIK | Atypical | 5ae8 | A | | 6-(1h-indol-4-yl)-4-(5-{[4-(1-methylethyl)-1-piperazinyl]methyl}-1,3-oxazol-2-yl)-1h-indazole | Mouse | 9390 | |
| Pik3cd (p110d) | PIK | Atypical | 5ae9 | A | | n-[5-[4-(5-{[(2r,6s)-2,6-dimethyl-4-morpholinyl]methyl}-1,3-oxazol-2-yl)-1h-indazol-6-yl]-2-(methyloxy)-3-pyridinyl]methanesulfonamide | Mouse | 9372 | |
| Pik3cd (p110d) | PIK | Atypical | 5i4u | A | | 2,4-diamino-6-{[(1s)-1-(5-chloro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethyl]amino}pyrimidine-5-carbonitrile | Mouse | 9391 | |
| Pik3cd (p110d) | PIK | Atypical | 5i6u | A | | 2-[(1s)-1-({6-amino-5-[(1h-pyrazol-4-yl)ethynyl]pyrimidin-4-yl}amino)ethyl]-5-chloro-3-phenylquinazolin-4(3h)-one | Mouse | 9370 | |
| Pik3cd (p110d) | PIK | Atypical | 5is5 | A | | 5-{4-[3-(4-acetylpiperazine-1-carbonyl)phenyl]quinazolin-6-yl}-2-methoxypyridine-3-carbonitrile | Mouse | 9356 | |
| Pik3cd (p110d) | PIK | Atypical | 5l72 | A | | n-[6-(5-methanesulfonamido-6-methoxypyridin-3-yl)-1,3-dihydro-2-benzofuran-4-yl]-2-(morpholin-4-yl)acetamide | Mouse | 9386 | |
| Pik3cd (p110d) | PIK | Atypical | 5ncy | A | A | 4-azanyl-6-[[(1~{s})-1-(3-methyl-5-oxidanylidene-6-phenyl-[1,3]thiazolo[3,2-a]pyridin-7-yl)ethyl]amino]pyrimidine-5-carbonitrile | Mouse | 9379 | |
| Pik3cd (p110d) | PIK | Atypical | 5ncy | A | B | 4-azanyl-6-[[(1~{s})-1-(3-methyl-5-oxidanylidene-6-phenyl-[1,3]thiazolo[3,2-a]pyridin-7-yl)ethyl]amino]pyrimidine-5-carbonitrile | Mouse | 9357 | |
| Pik3cd (p110d) | PIK | Atypical | 5ncz | A | A | 4-azanyl-6-[[(1~{s})-1-[6-[3-[(dimethylamino)methyl]phenyl]-3-methyl-5-oxidanylidene-[1,3]thiazolo[3,2-a]pyridin-7-yl]ethyl]amino]pyrimidine-5-carbonitrile | Mouse | 9396 | |
| Pik3cd (p110d) | PIK | Atypical | 5ncz | A | B | 4-azanyl-6-[[(1~{s})-1-[6-[3-[(dimethylamino)methyl]phenyl]-3-methyl-5-oxidanylidene-[1,3]thiazolo[3,2-a]pyridin-7-yl]ethyl]amino]pyrimidine-5-carbonitrile | Mouse | 9388 | |
| Pik3cd (p110d) | PIK | Atypical | 5ngb | A | | 3-[[4-(2-morpholin-4-yl-4-oxidanylidene-3~{h}-quinolin-8-yl)-1,2,3-triazol-1-yl]methyl]benzoic acid | Mouse | 9353 | |
| Pik3cd (p110d) | PIK | Atypical | 5o83 | A | | leniolisib | Mouse | 9351 | |
| Pik3cd (p110d) | PIK | Atypical | 5t27 | A | | 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{s})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine | Mouse | 9383 | |
| Pik3cd (p110d) | PIK | Atypical | 5t28 | A | | 3-(benzotriazol-1-yl)-5-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-amine | Mouse | 9398 | |
| Pik3cd (p110d) | PIK | Atypical | 5t2b | A | | 5-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]-3-(1~{h}-pyrazol-4-yl)pyrazin-2-amine | Mouse | 9374 | |
| Pik3cd (p110d) | PIK | Atypical | 5t2d | A | | 4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]-~{n},~{n}-dimethyl-pyrazole-1-sulfonamide | Mouse | 9397 | |
| Pik3cd (p110d) | PIK | Atypical | 5t2g | A | | 4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-1-carboxamide | Mouse | 9363 | |
| Pik3cd (p110d) | PIK | Atypical | 5t2i | A | A | 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-4-carboxamide | Mouse | 9358 | |
| Pik3cd (p110d) | PIK | Atypical | 5t2i | A | B | 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-4-carboxamide | Mouse | 9367 | |
| Pik3cd (p110d) | PIK | Atypical | 5t2l | A | A | 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-3-carboxamide | Mouse | 9378 | |
| Pik3cd (p110d) | PIK | Atypical | 5t2l | A | B | 1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-3-carboxamide | Mouse | 9394 | |
| Pik3cd (p110d) | PIK | Atypical | 5t2m | A | | 4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]benzamide | Mouse | 9371 | |
| Pik3cd (p110d) | PIK | Atypical | 5t7f | A | | 2,4-bis(azanyl)-6-[[(1~{s})-1-[5-chloranyl-3-(5-fluoranyl-4-methyl-pyridin-3-yl)-4-oxidanylidene-quinazolin-2-yl]ethyl]amino]pyrimidine-5-carbonitrile | Mouse | 9362 | |
| Pik3cd (p110d) | PIK | Atypical | 5t7f | B | | 2,4-bis(azanyl)-6-[[(1~{s})-1-[5-chloranyl-3-(5-fluoranyl-4-methyl-pyridin-3-yl)-4-oxidanylidene-quinazolin-2-yl]ethyl]amino]pyrimidine-5-carbonitrile | Mouse | 9354 | |
| Pik3cd (p110d) | PIK | Atypical | 5t8i | A | A | 2,4-diamino-6-{[(s)-[5-chloro-8-fluoro-4-oxo-3-(pyridin-3-yl)-3,4-dihydroquinazolin-2-yl](cyclopropyl)methyl]amino}pyrimidine-5-carbonitrile | Mouse | 9392 | |
| Pik3cd (p110d) | PIK | Atypical | 5t8i | A | B | 2,4-diamino-6-{[(s)-[5-chloro-8-fluoro-4-oxo-3-(pyridin-3-yl)-3,4-dihydroquinazolin-2-yl](cyclopropyl)methyl]amino}pyrimidine-5-carbonitrile | Mouse | 9377 | |
| Pik3cd (p110d) | PIK | Atypical | 6dgt | A | | 4-[1-(5,8-difluoroquinolin-4-yl)-2-methyl-4-(4h-1,2,4-triazol-3-yl)-1h-benzimidazol-6-yl]-3-fluoropyridin-2-amine | Mouse | 10603 | |
| Pik3cd (p110d) | PIK | Atypical | 6eyz | A | | 2-methoxy-5-[4-[5-[(4-propan-2-ylpiperazin-1-yl)methyl]-1,3-oxazol-2-yl]-2~{h}-indazol-6-yl]pyridine-3-carboxylic acid | Mouse | 9426 | |
| Pik3cd (p110d) | PIK | Atypical | 6ez6 | A | | methyl 2-methoxy-5-[4-[5-[(4-propan-2-ylpiperazin-1-yl)methyl]-1,3-oxazol-2-yl]-2~{h}-indazol-6-yl]pyridine-3-carboxylate | Mouse | 9460 | |
| Pik3cd (p110d) | PIK | Atypical | 6ftn | A | A | ~{n}-[5-[2-[(1~{s})-1-cyclopropylethyl]-7-methyl-1-oxidanylidene-3~{h}-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamide | Mouse | 10010 | |
| Pik3cd (p110d) | PIK | Atypical | 6ftn | A | B | ~{n}-[5-[2-[(1~{s})-1-cyclopropylethyl]-7-methyl-1-oxidanylidene-3~{h}-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamide | Mouse | 10011 | |
| Pik3cd (p110d) | PIK | Atypical | 6gy0 | A | | ~{n}-[4-methyl-5-(1-oxidanylidene-7-sulfamoyl-isoindol-5-yl)-1,3-thiazol-2-yl]ethanamide | Mouse | 11298 | |
| Pik3cd (p110d) | PIK | Atypical | 6hi1 | A | | 3-(6-morpholin-4-ylpyridin-2-yl)phenol | Mouse | 11624 | |
| Pik3cd (p110d) | PIK | Atypical | 6hi2 | A | | 3-[6-[(1~{s},6~{r})-3-oxabicyclo[4.1.0]heptan-6-yl]pyridin-2-yl]phenol | Mouse | 11623 | |
| Pik3cd (p110d) | PIK | Atypical | 6hi9 | A | A | 3-[6-(oxan-4-yl)pyridin-2-yl]phenol | Mouse | 11625 | |
| Pik3cd (p110d) | PIK | Atypical | 6hi9 | A | B | 3-[6-(oxan-4-yl)pyridin-2-yl]phenol | Mouse | 11622 | |
| Pik3cd (p110d) | PIK | Atypical | 6mul | A | A | 1-{1-[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]piperidin-4-yl}-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-one | Mouse | 11300 | |
| Pik3cd (p110d) | PIK | Atypical | 6mul | A | B | 1-{1-[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]piperidin-4-yl}-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-one | Mouse | 11297 | |
| Pik3cd (p110d) | PIK | Atypical | 6mul | B | A | 1-{1-[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]piperidin-4-yl}-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-one | Mouse | 11301 | |
| Pik3cd (p110d) | PIK | Atypical | 6mul | B | B | 1-{1-[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]piperidin-4-yl}-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-one | Mouse | 11293 | |
| Pik3cd (p110d) | PIK | Atypical | 6mum | A | A | [(3s)-3-{[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]oxy}pyrrolidin-1-yl](oxan-4-yl)methanone | Mouse | 11294 | |
| Pik3cd (p110d) | PIK | Atypical | 6mum | A | B | [(3s)-3-{[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]oxy}pyrrolidin-1-yl](oxan-4-yl)methanone | Mouse | 11296 | |
| Pik3cd (p110d) | PIK | Atypical | 6mum | B | A | [(3s)-3-{[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]oxy}pyrrolidin-1-yl](oxan-4-yl)methanone | Mouse | 11299 | |
| Pik3cd (p110d) | PIK | Atypical | 6mum | B | B | [(3s)-3-{[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]oxy}pyrrolidin-1-yl](oxan-4-yl)methanone | Mouse | 11295 | |
| Pik3cd (p110d) | PIK | Atypical | 6q6y | A | | ~{n}-(2-chloranyl-5-phenyl-pyridin-3-yl)benzenesulfonamide | Mouse | 10826 | |
| Pik3cd (p110d) | PIK | Atypical | 6q73 | A | | ~{n}-[2-chloranyl-5-(3,6-dihydro-2~{h}-pyran-4-yl)pyridin-3-yl]methanesulfonamide | Mouse | 10825 | |
| Pik3cd (p110d) | PIK | Atypical | 6q74 | A | | ~{n}-[5-(3,6-dihydro-2~{h}-pyran-4-yl)-2-methoxy-pyridin-3-yl]-2-methyl-1-(phenylmethyl)imidazole-4-sulfonamide | Mouse | 10824 | |
| Pik3cd (p110d) | PIK | Atypical | 6tnr | A | A | ~{n}-[2-methoxy-5-[7-[2-[4-(2-oxidanylpropan-2-yl)piperidin-1-yl]ethoxy]-1,3-dihydro-2-benzofuran-5-yl]pyridin-3-yl]methanesulfonamide | Mouse | 11911 | |
| Pik3cd (p110d) | PIK | Atypical | 6tnr | A | B | ~{n}-[2-methoxy-5-[7-[2-[4-(2-oxidanylpropan-2-yl)piperidin-1-yl]ethoxy]-1,3-dihydro-2-benzofuran-5-yl]pyridin-3-yl]methanesulfonamide | Mouse | 11910 | |
| Pik3cd (p110d) | PIK | Atypical | 6tns | A | | 2-methoxy-~{n}-[2-methoxy-5-[7-[[(2~{r})-4-(oxetan-3-yl)morpholin-2-yl]methoxy]-1,3-dihydro-2-benzofuran-5-yl]pyridin-3-yl]ethanesulfonamide | Mouse | 11909 | |
| Pik3cd (p110d) | PIK | Atypical | 6zaa | A | | 4-[6-methoxy-5-(methylsulfamoyl)pyridin-3-yl]-~{n}-(1-methylpiperidin-4-yl)-2,3-dihydro-1,4-benzoxazine-6-carboxamide | Mouse | 12635 | |
| Pik3cd (p110d) | PIK | Atypical | 6zac | A | A | ~{n}-[5-[6-[(dimethylamino)methyl]-2,3-dihydro-1,4-benzoxazin-4-yl]-2-methoxy-pyridin-3-yl]methanesulfonamide | Mouse | 12633 | |
| Pik3cd (p110d) | PIK | Atypical | 6zac | A | B | ~{n}-[5-[6-[(dimethylamino)methyl]-2,3-dihydro-1,4-benzoxazin-4-yl]-2-methoxy-pyridin-3-yl]methanesulfonamide | Mouse | 12634 | |
| Pik3cd (p110d) | PIK | Atypical | 6zad | A | | methoxymethyloxathiatetraazatetracyclodocosahexaenedione | Mouse | 12653 | |
| Pik3cd (p110d) | PIK | Atypical | 7oi4 | A | A | n-[5-[2-[(1s)-1-cyclopropylethyl]-7-[[4-[(dimethylamino)methyl]phenyl]sulfamoyl]-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamide | Mouse | 13800 | |
| Pik3cd (p110d) | PIK | Atypical | 7oi4 | A | B | n-[5-[2-[(1s)-1-cyclopropylethyl]-7-[[4-[(dimethylamino)methyl]phenyl]sulfamoyl]-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamide | Mouse | 13805 | |
| Pik3cd (p110d) | PIK | Atypical | 7oij | A | A | 6-[[5-[2-[(1s)-1-cyclopropylethyl]-7-(methylsulfamoyl)-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]amino]-n-[3-(dimethylamino)propyl]pyridine-2-carboxamide | Mouse | 13801 | |
| Pik3cd (p110d) | PIK | Atypical | 7oij | A | B | 6-[[5-[2-[(1s)-1-cyclopropylethyl]-7-(methylsulfamoyl)-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]amino]-n-[3-(dimethylamino)propyl]pyridine-2-carboxamide | Mouse | 13807 | |
| Pik3cd (p110d) | PIK | Atypical | 7oil | A | A | 2-[(1s)-1-cyclopropylethyl]-5-[4-methyl-2-[[6-(2-oxidanylidenepyrrolidin-1-yl)pyridin-2-yl]amino]-1,3-thiazol-5-yl]-7-methylsulfonyl-3h-isoindol-1-one | Mouse | 13804 | |
| Pik3cd (p110d) | PIK | Atypical | 7oil | A | B | 2-[(1s)-1-cyclopropylethyl]-5-[4-methyl-2-[[6-(2-oxidanylidenepyrrolidin-1-yl)pyridin-2-yl]amino]-1,3-thiazol-5-yl]-7-methylsulfonyl-3h-isoindol-1-one | Mouse | 13806 | |
| Pik3cd (p110d) | PIK | Atypical | 7ois | A | A | n-[5-[2-[(1s)-1-cyclopropylethyl]-7-[(3-methylsulfonylphenyl)sulfamoyl]-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamide | Mouse | 13803 | |
| Pik3cd (p110d) | PIK | Atypical | 7ois | A | B | n-[5-[2-[(1s)-1-cyclopropylethyl]-7-[(3-methylsulfonylphenyl)sulfamoyl]-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamide | Mouse | 13802 | |
| Pik3cd (p110d) | PIK | Atypical | 7pop | A | | 5-[3,6-dihydro-2h-pyran-4-yl]-2-methoxy-n-[2-methylpyridin-4-yl]pyridine-3-sulfonamide | Mouse | 13917 | |
| Pik3cd (p110d) | PIK | Atypical | 7por | A | | ~{n}-[2-[2-fluoranyl-4-[(4-propan-2-ylpiperazin-1-yl)methyl]phenyl]pyridin-4-yl]-2-methoxy-5-morpholin-4-yl-pyridine-3-sulfonamide | Mouse | 13915 | |
| Pik3cd (p110d) | PIK | Atypical | 7pos | A | | 5-(3,6-dihydro-2~{h}-pyran-4-yl)-2-methoxy-~{n}-[5-[3-(4-propan-2-ylpiperazin-1-yl)prop-1-ynyl]pyridin-3-yl]pyridine-3-sulfonamide | Mouse | 13918 | |
| Pik3cd (p110d) | PIK | Atypical | 7pot | A | | n-[5-(3,6-dihydro-2h-pyran-4-yl)-2-methoxy-pyridin-3-yl]benzenesulfonamide | Mouse | 13916 | |
| Pik3cd (p110d) | PIK | Atypical | 7r26 | A | | 5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amine | Mouse | 14231 | |
| Pik3cd (p110d) | PIK | Atypical | 7r2b | A | | (4~{s})-3-[6-[2-azanyl-4-(trifluoromethyl)pyrimidin-5-yl]-2-morpholin-4-yl-pyrimidin-4-yl]-4-methyl-1,3-oxazolidin-2-one | Mouse | 14230 | |
| PIK3CD (p110d) | PIK | Atypical | 5dxu | A | | (2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamide | Human | 9091 | |
| PIK3CD (p110d) | PIK | Atypical | 5m6u | A | | 4-azanyl-6-[[(1~{s})-1-(4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]pyrimidine-5-carbonitrile | Human | 9094 | |
| PIK3CD (p110d) | PIK | Atypical | 5t8f | A | | 2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamide | Human | 9093 | |
| PIK3CD (p110d) | PIK | Atypical | 5ubt | A | | 1-[4-(3-{4-amino-5-[1-(oxan-4-yl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)piperazin-1-yl]ethan-1-one | Human | 9092 | |
| PIK3CD (p110d) | PIK | Atypical | 5vlr | A | | 4-acetyl-1-(3-{4-amino-5-[1-(2,2,2-trifluoroethyl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)-3,3-dimethylpiperazin-2-one | Human | 9090 | |
| PIK3CD (p110d) | PIK | Atypical | 6g6w | A | A | ~{n}-[3-[4-[[(1~{s})-1-(5-methyl-4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-5-oxidanyl-phenyl]methanesulfonamide | Human | 10673 | |
| PIK3CD (p110d) | PIK | Atypical | 6g6w | A | B | ~{n}-[3-[4-[[(1~{s})-1-(5-methyl-4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-5-oxidanyl-phenyl]methanesulfonamide | Human | 10674 | |
| PIK3CD (p110d) | PIK | Atypical | 6oco | A | | 4-[(1s,4s)-5-(3-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carbonitrile | Human | 11865 | |
| PIK3CD (p110d) | PIK | Atypical | 6ocu | A | | 5-{(3r)-3-methyl-4-[(1r,2r)-2-methylcyclopropane-1-carbonyl]piperazin-1-yl}-3-(1-methyl-1h-pyrazol-4-yl)pyrazine-2-carbonitrile | Human | 11864 | |
| PIK3CD (p110d) | PIK | Atypical | 6pyr | A | A | (3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-one | Human | 11547 | |
| PIK3CD (p110d) | PIK | Atypical | 6pyr | A | B | (3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-one | Human | 11546 | |
| PIK3CD (p110d) | PIK | Atypical | 6pyu | A | | (3s)-1'-(cyclopropanecarbonyl)-5-(quinoxalin-6-yl)spiro[indole-3,2'-pyrrolidin]-2(1h)-one | Human | 11548 | |
| PIK3CD (p110d) | PIK | Atypical | 7jis | A | | (3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-one | Human | 13201 | |
| PIK3CD (p110d) | PIK | Atypical | 7lm2 | A | | cyclopropyl[(3s)-3-{[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]amino}pyrrolidin-1-yl]methanone | Human | 13532 | |
| PIK3CD (p110d) | PIK | Atypical | 7lq1 | A | | n-(5-(6-(2-((2s,6r)-2,6-dimethylmorpholino)pyridin-4-yl)-1-oxoisoindolin-4-yl)-2-methoxypyridin-3-yl)methanesulfonamide | Human | 14106 | |
| PIK3CD (p110d) | PIK | Atypical | 8bcy | A | A | 9-[2-(3,4-dichlorophenyl)ethyl]-2-(3-hydroxyphenyl)-8-oxidanylidene-7~{h}-purine-6-carboxamide | Human | 14735 | |
| PIK3CD (p110d) | PIK | Atypical | 8bcy | A | B | 9-[2-(3,4-dichlorophenyl)ethyl]-2-(3-hydroxyphenyl)-8-oxidanylidene-7~{h}-purine-6-carboxamide | Human | 14734 | |
| PIK3CG (p110g) | PIK | Atypical | 1e8y | A | | - | Human | 9248 | |
| PIK3CG (p110g) | PIK | Atypical | 1e8z | A | | staurosporine | Human | 9228 | |
| PIK3CG (p110g) | PIK | Atypical | 1he8 | A | | - | Human | 9201 | |
| PIK3CG (p110g) | PIK | Atypical | 2a4z | A | | (5e)-5-[(2,2-difluoro-1,3-benzodioxol-5-yl)methylene]-1,3-thiazolidine-2,4-dione | Human | 9180 | |
| PIK3CG (p110g) | PIK | Atypical | 2a5u | A | | (5e)-5-(quinoxalin-6-ylmethylene)-1,3-thiazolidine-2,4-dione | Human | 9183 | |
| PIK3CG (p110g) | PIK | Atypical | 2chw | A | | 2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-one | Human | 9182 | |
| PIK3CG (p110g) | PIK | Atypical | 2chx | A | | n-(2,3-dihydro-7,8-dimethoxyimidazo[1,2-c] quinazolin-5-yl)nicotinamide | Human | 9247 | |
| PIK3CG (p110g) | PIK | Atypical | 2chz | A | | n-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamide | Human | 9251 | |
| PIK3CG (p110g) | PIK | Atypical | 2v4l | A | | 3-[4-amino-1-(1-methylethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]phenol | Human | 9237 | |
| PIK3CG (p110g) | PIK | Atypical | 3apc | A | | 5-(7-methanesulfonyl-2-morpholin-4-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamine | Human | 9231 | |
| PIK3CG (p110g) | PIK | Atypical | 3apd | A | | 5-(2-morpholin-4-yl-7-pyridin-3-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamine | Human | 9205 | |
| PIK3CG (p110g) | PIK | Atypical | 3apf | A | | 3-[7-(1h-benzimidazol-5-yl)-2-(morpholin-4-yl)-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl]phenol | Human | 9250 | |
| PIK3CG (p110g) | PIK | Atypical | 3csf | A | | - | Human | 9215 | |
| PIK3CG (p110g) | PIK | Atypical | 3cst | A | | methylated ruthenium pyridocarbazole | Human | 9220 | |
| PIK3CG (p110g) | PIK | Atypical | 3dbs | A | | 2-(1h-indazol-4-yl)-6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-yl-thieno[3,2-d]pyrimidine | Human | 9230 | |
| PIK3CG (p110g) | PIK | Atypical | 3dpd | A | | 5,5-dimethyl-2-morpholin-4-yl-5,6-dihydro-1,3-benzothiazol-7(4h)-one | Human | 9159 | |
| PIK3CG (p110g) | PIK | Atypical | 3ene | A | | 1-methyl-3-naphthalen-2-yl-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 9188 | |
| PIK3CG (p110g) | PIK | Atypical | 3ibe | A | | 1-(4-{4-morpholin-4-yl-1-[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-6-yl}phenyl)-3-pyridin-4-ylurea | Human | 9171 | |
| PIK3CG (p110g) | PIK | Atypical | 3l08 | A | A | 2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamide | Human | 9217 | |
| PIK3CG (p110g) | PIK | Atypical | 3l08 | A | B | 2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamide | Human | 9164 | |
| PIK3CG (p110g) | PIK | Atypical | 3l13 | A | | [3-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenyl]methanol | Human | 9167 | |
| PIK3CG (p110g) | PIK | Atypical | 3l16 | A | | 5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyridin-2-amine | Human | 9233 | |
| PIK3CG (p110g) | PIK | Atypical | 3l17 | A | | 4-methyl-5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyrimidin-2-amine | Human | 9185 | |
| PIK3CG (p110g) | PIK | Atypical | 3l54 | A | | 6-(1h-pyrazolo[3,4-b]pyridin-5-yl)-4-pyridin-4-ylquinoline | Human | 9197 | |
| PIK3CG (p110g) | PIK | Atypical | 3lj3 | A | | (2z)-4,6-dihydroxy-2-{[1-methyl-4-(4-methylpiperazin-1-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methylidene}-1-benzofuran-3(2h)-one | Human | 9214 | |
| PIK3CG (p110g) | PIK | Atypical | 3mjw | A | | (2z)-4,6-dihydroxy-2-[(8-methoxy-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)methylidene]-1-benzofuran-3(2h)-one | Human | 9229 | |
| PIK3CG (p110g) | PIK | Atypical | 3ml8 | A | | 8-cyclopentyl-6-[3-(hydroxymethyl)phenyl]-4-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9192 | |
| PIK3CG (p110g) | PIK | Atypical | 3ml9 | A | | 2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9187 | |
| PIK3CG (p110g) | PIK | Atypical | 3nzs | A | | 6-(1,1-dioxidothiomorpholin-4-yl)-n-(3-methoxyphenyl)-1-methyl-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 9179 | |
| PIK3CG (p110g) | PIK | Atypical | 3nzu | A | | 6-(2h-indazol-4-yl)-1-methyl-n-[3-(methylsulfonyl)propyl]-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 9177 | |
| PIK3CG (p110g) | PIK | Atypical | 3oaw | A | | 2-amino-4-methyl-8-(1-methylethyl)-6-(1h-pyrazol-4-yl)pteridin-7(8h)-one | Human | 9240 | |
| PIK3CG (p110g) | PIK | Atypical | 3p2b | A | A | 3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenol | Human | 9169 | |
| PIK3CG (p110g) | PIK | Atypical | 3p2b | A | B | 3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenol | Human | 9165 | |
| PIK3CG (p110g) | PIK | Atypical | 3pre | A | | 2-amino-8-(trans-4-methoxycyclohexyl)-4-methyl-6-(1h-pyrazol-3-yl)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9198 | |
| PIK3CG (p110g) | PIK | Atypical | 3prz | A | | 4-amino-2-methyl-n-(1h-pyrazol-3-yl)quinazoline-8-carboxamide | Human | 9210 | |
| PIK3CG (p110g) | PIK | Atypical | 3ps6 | A | | 4-amino-n-(6-methoxypyridin-3-yl)-2-methylquinazoline-8-carboxamide | Human | 9170 | |
| PIK3CG (p110g) | PIK | Atypical | 3qaq | A | | [(4-{2-[(3-hydroxyphenyl)amino]-1h-benzimidazol-1-yl}-1,3,5-triazin-2-yl)amino]acetonitrile | Human | 9211 | |
| PIK3CG (p110g) | PIK | Atypical | 3qar | A | | 1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-3-yl)-1h-benzimidazol-2-amine | Human | 9178 | |
| PIK3CG (p110g) | PIK | Atypical | 3qjz | A | | n-{6-[2-(methylsulfanyl)pyrimidin-4-yl]-1,3-benzothiazol-2-yl}acetamide | Human | 9181 | |
| PIK3CG (p110g) | PIK | Atypical | 3qk0 | A | | n-[6-(6-chloro-5-{[(4-fluorophenyl)sulfonyl]amino}pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Human | 9213 | |
| PIK3CG (p110g) | PIK | Atypical | 3r7q | A | | n-(2-chlorophenyl)-n-methyl-4h-thieno[3,2-c]chromene-2-carboxamide | Human | 9227 | |
| PIK3CG (p110g) | PIK | Atypical | 3r7r | A | | 8-(acetylamino)-n-(2-chlorophenyl)-n-methyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2-carboxamide | Human | 9168 | |
| PIK3CG (p110g) | PIK | Atypical | 3s2a | A | | n-{2-chloro-5-[4-(morpholin-4-yl)quinolin-6-yl]pyridin-3-yl}-4-fluorobenzenesulfonamide | Human | 9158 | |
| PIK3CG (p110g) | PIK | Atypical | 3sd5 | A | | 5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amine | Human | 9243 | |
| PIK3CG (p110g) | PIK | Atypical | 3t8m | A | | n~2~-{2-chloro-4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-n~2~,n~8~-dimethyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2,8-dicarboxamide | Human | 9186 | |
| PIK3CG (p110g) | PIK | Atypical | 3tjp | A | | n~6~-(3,4-dimethoxyphenyl)-2-(morpholin-4-yl)-4,5'-bipyrimidine-2',6-diamine | Human | 9234 | |
| PIK3CG (p110g) | PIK | Atypical | 3tl5 | A | | (2s)-1-(4-{[2-(2-aminopyrimidin-5-yl)-7-methyl-4-(morpholin-4-yl)thieno[3,2-d]pyrimidin-6-yl]methyl}piperazin-1-yl)-2-hydroxypropan-1-one | Human | 9160 | |
| PIK3CG (p110g) | PIK | Atypical | 3zvv | A | | 5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-amine | Human | 9172 | |
| PIK3CG (p110g) | PIK | Atypical | 3zw3 | A | | n-{6-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]imidazo[1,2-a]pyridin-2-yl}acetamide | Human | 9207 | |
| PIK3CG (p110g) | PIK | Atypical | 4anu | A | | 3-amino-n-methyl-6-[3-(1h-tetrazol-5-yl)phenyl]pyrazine-2-carboxamide | Human | 9162 | |
| PIK3CG (p110g) | PIK | Atypical | 4anv | A | A | 2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazine | Human | 9195 | |
| PIK3CG (p110g) | PIK | Atypical | 4anv | A | B | 2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazine | Human | 9166 | |
| PIK3CG (p110g) | PIK | Atypical | 4anw | A | A | 3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamide | Human | 9174 | |
| PIK3CG (p110g) | PIK | Atypical | 4anw | A | B | 3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamide | Human | 9175 | |
| PIK3CG (p110g) | PIK | Atypical | 4anx | A | | 5-{3-[(4-{3-[4-(1-methylethyl)phenyl]pyrazin-2-yl}piperazin-1-yl)sulfonyl]phenyl}pyrimidin-2-amine | Human | 9252 | |
| PIK3CG (p110g) | PIK | Atypical | 4aof | A | | n-[6-(5-methylsulfonylpyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]ethanamide | Human | 9245 | |
| PIK3CG (p110g) | PIK | Atypical | 4dk5 | A | | 4-(2-[(6-methoxypyridin-3-yl)amino]-5-{[4-(methylsulfonyl)piperazin-1-yl]methyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amine | Human | 9232 | |
| PIK3CG (p110g) | PIK | Atypical | 4ezj | A | | 2-(1-{[2-(5-fluoro-1h-indol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-ol | Human | 9222 | |
| PIK3CG (p110g) | PIK | Atypical | 4ezk | A | | 2-(1-{[2-(2h-indazol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-ol | Human | 9176 | |
| PIK3CG (p110g) | PIK | Atypical | 4ezl | A | | 2-(1-{[2-(2-aminopyrimidin-5-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-ol | Human | 9235 | |
| PIK3CG (p110g) | PIK | Atypical | 4f1s | A | | n-(5-{[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-(tetrahydro-2h-pyran-4-yl)pyridin-2-yl]amino}-2-chloropyridin-3-yl)methanesulfonamide | Human | 9221 | |
| PIK3CG (p110g) | PIK | Atypical | 4fa6 | A | | 2-amino-8-cyclopentyl-4-methyl-6-(1h-pyrazol-4-yl)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9191 | |
| PIK3CG (p110g) | PIK | Atypical | 4fad | A | | 2-amino-6-(5-fluoro-6-methoxypyridin-3-yl)-4-methyl-8-(pyrrolidin-1-yl)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 9202 | |
| PIK3CG (p110g) | PIK | Atypical | 4fhj | A | | 3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-5-yl)imidazo[1,2-a]pyridin-2-amine | Human | 9209 | |
| PIK3CG (p110g) | PIK | Atypical | 4fhk | A | | 3-[2-methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]-n-(1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-2-amine | Human | 9204 | |
| PIK3CG (p110g) | PIK | Atypical | 4fjy | A | | 4-[3,3-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1h-indol-1-yl]-7-fluoro-3-methyl-2-(pyridin-3-yl)quinoline | Human | 9249 | |
| PIK3CG (p110g) | PIK | Atypical | 4fjz | A | | 1'-[7-fluoro-3-methyl-2-(pyridin-2-yl)quinolin-4-yl]-6'-(morpholin-4-yl)-1',2,2',3,5,6-hexahydrospiro[pyran-4,3'-pyrrolo[3,2-b]pyridine] | Human | 9173 | |
| PIK3CG (p110g) | PIK | Atypical | 4flh | A | | 4-(2-[(5-fluoro-6-methoxypyridin-3-yl)amino]-5-{(1r)-1-[4-(methylsulfonyl)piperazin-1-yl]ethyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amine | Human | 9212 | |
| PIK3CG (p110g) | PIK | Atypical | 4ful | A | | 4-({4-[3-(piperidin-1-ylcarbonyl)phenyl]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 9242 | |
| PIK3CG (p110g) | PIK | Atypical | 4g11 | A | | 2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyrimidin-2-yl]-n-phenylacetamide | Human | 9223 | |
| PIK3CG (p110g) | PIK | Atypical | 4gb9 | A | | 2-[1-({2-[2-(dimethylamino)-1h-benzimidazol-1-yl]-9-methyl-6-(morpholin-4-yl)-9h-purin-8-yl}methyl)piperidin-4-yl]propan-2-ol | Human | 9218 | |
| PIK3CG (p110g) | PIK | Atypical | 4hle | A | | 2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepine-8-carboxamide | Human | 9219 | |
| PIK3CG (p110g) | PIK | Atypical | 4hvb | A | | 1-{1-[(2s)-2-hydroxypropanoyl]piperidin-4-yl}-3-methyl-8-(6-methylpyridin-3-yl)-1,3-dihydro-2h-imidazo[4,5-c][1,5]naphthyridin-2-one | Human | 9225 | |
| PIK3CG (p110g) | PIK | Atypical | 4j6i | A | | 2-methyl-1-(4-{2-[1-(2,2,2-trifluoroethyl)-1h-1,2,4-triazol-5-yl]-4,5-dihydro[1]benzoxepino[5,4-d][1,3]thiazol-8-yl}-1h-pyrazol-1-yl)propan-2-ol | Human | 9189 | |
| PIK3CG (p110g) | PIK | Atypical | 4kz0 | A | | methyl 2-(acetylamino)-1,3-benzothiazole-6-carboxylate | Human | 9161 | |
| PIK3CG (p110g) | PIK | Atypical | 4kzc | A | | n-{6-[6-amino-5-(trifluoromethyl)pyridin-3-yl]imidazo[1,2-a]pyridin-2-yl}acetamide | Human | 9224 | |
| PIK3CG (p110g) | PIK | Atypical | 4ps3 | A | | 1-[6-(5-methoxypyridin-3-yl)-1,3-benzothiazol-2-yl]-3-[2-(1-propyl-1h-imidazol-4-yl)ethyl]urea | Human | 9193 | |
| PIK3CG (p110g) | PIK | Atypical | 4ps7 | A | | n-[6-(pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Human | 9163 | |
| PIK3CG (p110g) | PIK | Atypical | 4ps8 | A | | n-[6-(5,6-dimethoxypyridin-3-yl)-1,3-benzothiazol-2-yl]acetamide | Human | 9184 | |
| PIK3CG (p110g) | PIK | Atypical | 4urk | A | | 2-[[(1r)-1-(7-methyl-2-morpholin-4-yl-4-oxidanylidene-pyrido[1,2-a]pyrimidin-9-yl)ethyl]amino]benzoic acid | Human | 9196 | |
| PIK3CG (p110g) | PIK | Atypical | 4wwn | A | | n-{(1s)-1-[7-fluoro-2-(pyridin-2-yl)quinolin-3-yl]ethyl}-9h-purin-6-amine | Human | 9226 | |
| PIK3CG (p110g) | PIK | Atypical | 4wwo | A | | n-{(1s)-1-[8-chloro-2-(3-fluorophenyl)quinolin-3-yl]ethyl}-9h-purin-6-amine | Human | 9190 | |
| PIK3CG (p110g) | PIK | Atypical | 4wwp | A | | n-{(1s)-1-[8-chloro-2-(2-methylpyridin-3-yl)quinolin-3-yl]ethyl}-9h-purin-6-amine | Human | 9200 | |
| PIK3CG (p110g) | PIK | Atypical | 4xx5 | A | | n-[5-(5-methoxypyridin-3-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamide | Human | 9236 | |
| PIK3CG (p110g) | PIK | Atypical | 4xz4 | A | | n-[5-(6-methoxypyrazin-2-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamide | Human | 9194 | |
| PIK3CG (p110g) | PIK | Atypical | 5eds | A | | 4-azanyl-6-[[(1~{s})-1-[6-fluoranyl-1-(3-methylsulfonylphenyl)benzimidazol-2-yl]ethyl]amino]pyrimidine-5-carbonitrile | Human | 9208 | |
| PIK3CG (p110g) | PIK | Atypical | 5g2n | A | | 2-azanyl-~{n}-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]pyrimidine-5-carboxamide | Human | 9206 | |
| PIK3CG (p110g) | PIK | Atypical | 5g55 | A | | 6-cyano-4-[[(1r)-1-(4-methylphenyl)ethyl]amino]quinoline-3-carboxamide | Human | 9199 | |
| PIK3CG (p110g) | PIK | Atypical | 5jha | A | | [1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)pyrimidin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanol | Human | 9246 | |
| PIK3CG (p110g) | PIK | Atypical | 5jhb | A | | [1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanol | Human | 9238 | |
| PIK3CG (p110g) | PIK | Atypical | 5kae | A | | 4-azanyl-6-[[(1~{s})-1-(6-fluoranyl-3-phenyl-4-piperazin-1-ylcarbonyl-quinolin-2-yl)ethyl]amino]pyrimidine-5-carbonitrile | Human | 9241 | |
| PIK3CG (p110g) | PIK | Atypical | 5oq4 | A | A | 5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | 9244 | |
| PIK3CG (p110g) | PIK | Atypical | 5oq4 | A | B | 5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | 9203 | |
| PIK3CG (p110g) | PIK | Atypical | 5t23 | A | | 3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{s})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amine | Human | 9157 | |
| PIK3CG (p110g) | PIK | Atypical | 6aud | A | A | 10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine | Human | 9239 | |
| PIK3CG (p110g) | PIK | Atypical | 6aud | A | B | 10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine | Human | 9216 | |
| PIK3CG (p110g) | PIK | Atypical | 6c1s | A | | {4-[2-(5,6-dimethoxypyridin-3-yl)-5-oxo-5,7-dihydro-6h-pyrrolo[3,4-b]pyridin-6-yl]-1h-pyrazol-1-yl}acetonitrile | Human | 10037 | |
| PIK3CG (p110g) | PIK | Atypical | 6fh5 | A | | 3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-one | Human | 10883 | |
| PIK3CG (p110g) | PIK | Atypical | 6gq7 | A | | 3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-one | Human | 10009 | |
| PIK3CG (p110g) | PIK | Atypical | 6t3b | A | | 2-[(4-methoxy-2-methyl-phenyl)amino]-7-methyl-9-(4-oxidanylcyclohexyl)purin-8-one | Human | 11906 | |
| PIK3CG (p110g) | PIK | Atypical | 6t3c | A | | 7-methyl-2-[(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(oxan-4-yl)purin-8-one | Human | 11907 | |
| PIK3CG (p110g) | PIK | Atypical | 6xrl | A | | 2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 12774 | |
| PIK3CG (p110g) | PIK | Atypical | 6xrm | A | | 5-[2-amino-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-2-[(1s)-1-cyclopropylethyl]-7-(trifluoromethyl)-2,3-dihydro-1h-isoindol-1-one | Human | 12775 | |
| PIK3CG (p110g) | PIK | Atypical | 6xrn | A | | 2-amino-5-{2-[(1s)-1-cyclopropylethyl]-7-methyl-1-oxo-2,3-dihydro-1h-isoindol-5-yl}-n-(trans-3-hydroxycyclobutyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 13954 | |
| PIK3CG (p110g) | PIK | Atypical | 7jwe | A | | gedatolisib | Human | 13412 | |
| PIK3CG (p110g) | PIK | Atypical | 7jwz | A | | 2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 13410 | |
| PIK3CG (p110g) | PIK | Atypical | 7jx0 | A | | n~3~-{[5-(4-acetylphenyl)-4-methyl-1,3-thiazol-2-yl]carbamoyl}-n-tert-butyl-beta-alaninamide | Human | 13411 | |
| PIK3CG (p110g) | PIK | Atypical | 7kke | A | | n-[2-(3,3-dimethylbutoxy)ethyl]-n'-{4-methyl-5-[(pyridin-4-yl)ethynyl]-1,3-thiazol-2-yl}urea | Human | 13433 | |
| PIK3CG (p110g) | PIK | Atypical | 7mez | A | | - | Human | 13798 | |
| PIK3CG (p110g) | PIK | Atypical | 7z61 | A | | 9-[(3~{r},4~{r})-4-fluoranylpyrrolidin-3-yl]-7-methyl-2-[(7-methylquinolin-6-yl)amino]purin-8-one | Human | 14286 | |
| PIK3CG (p110g) | PIK | Atypical | 8dp0 | A | | - | Human | 14838 | |
| PIK3CG (p110g) | PIK | Atypical | 8sc8 | A | A | n-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide | Human | 15289 | |
| PIK3CG (p110g) | PIK | Atypical | 8sc8 | A | B | n-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide | Human | 15291 | |
| PIK3CG (p110g) | PIK | Atypical | 8sc8 | A | C | n-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamide | Human | 15290 | |
| PIK3R4 | VPS15 | Other | 7bl1 | C | | - | Human | 13360 | |
| PIK3R4 | VPS15 | Other | 8sor | D | | - | Human | 14802 | |
| PIM1 | PIM | CAMK | 1xqz | A | | - | Human | 2361 | |
| PIM1 | PIM | CAMK | 1xr1 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2406 | |
| PIM1 | PIM | CAMK | 1xws | A | A | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2343 | |
| PIM1 | PIM | CAMK | 1xws | A | B | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2441 | |
| PIM1 | PIM | CAMK | 1yhs | A | | staurosporine | Human | 2444 | |
| PIM1 | PIM | CAMK | 1yi3 | A | | 2-morpholin-4-yl-7-phenyl-4h-chromen-4-one | Human | 2398 | |
| PIM1 | PIM | CAMK | 1yi4 | A | | adenosine | Human | 2403 | |
| PIM1 | PIM | CAMK | 1ywv | A | A | - | Human | 2430 | |
| PIM1 | PIM | CAMK | 1ywv | A | B | - | Human | 2397 | |
| PIM1 | PIM | CAMK | 1yxs | A | A | - | Human | 2417 | |
| PIM1 | PIM | CAMK | 1yxs | A | B | - | Human | 2461 | |
| PIM1 | PIM | CAMK | 1yxt | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2425 | |
| PIM1 | PIM | CAMK | 1yxt | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2319 | |
| PIM1 | PIM | CAMK | 1yxu | A | | adenosine monophosphate | Human | 2438 | |
| PIM1 | PIM | CAMK | 1yxu | B | | adenosine monophosphate | Human | 2410 | |
| PIM1 | PIM | CAMK | 1yxu | C | | adenosine monophosphate | Human | 2408 | |
| PIM1 | PIM | CAMK | 1yxu | D | | adenosine monophosphate | Human | 2332 | |
| PIM1 | PIM | CAMK | 1yxv | A | A | 3,4-dihydroxy-1-methylquinolin-2(1h)-one | Human | 2367 | |
| PIM1 | PIM | CAMK | 1yxv | A | B | 3,4-dihydroxy-1-methylquinolin-2(1h)-one | Human | 2366 | |
| PIM1 | PIM | CAMK | 1yxx | A | A | (3e)-3-[(4-hydroxyphenyl)imino]-1h-indol-2(3h)-one | Human | 2351 | |
| PIM1 | PIM | CAMK | 1yxx | A | B | (3e)-3-[(4-hydroxyphenyl)imino]-1h-indol-2(3h)-one | Human | 2437 | |
| PIM1 | PIM | CAMK | 2bik | B | A | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2341 | |
| PIM1 | PIM | CAMK | 2bik | B | B | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2463 | |
| PIM1 | PIM | CAMK | 2bil | B | | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2449 | |
| PIM1 | PIM | CAMK | 2bzh | B | A | ruthenium-pyridocarbazole-1 | Human | 7230 | |
| PIM1 | PIM | CAMK | 2bzh | B | B | ruthenium-pyridocarbazole-1 | Human | 7234 | |
| PIM1 | PIM | CAMK | 2bzi | B | A | - | Human | 7225 | |
| PIM1 | PIM | CAMK | 2bzi | B | B | - | Human | 7233 | |
| PIM1 | PIM | CAMK | 2bzj | A | A | ruthenium-pyridocarbazole-3 | Human | 7224 | |
| PIM1 | PIM | CAMK | 2bzj | A | B | ruthenium-pyridocarbazole-3 | Human | 7228 | |
| PIM1 | PIM | CAMK | 2bzk | B | | phosphoaminophosphonic acid-adenylate ester | Human | 2330 | |
| PIM1 | PIM | CAMK | 2c3i | B | A | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 2348 | |
| PIM1 | PIM | CAMK | 2c3i | B | B | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 2374 | |
| PIM1 | PIM | CAMK | 2j2i | B | A | (9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dione | Human | 2318 | |
| PIM1 | PIM | CAMK | 2j2i | B | B | (9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dione | Human | 2434 | |
| PIM1 | PIM | CAMK | 2o3p | A | A | 3,5,7,3',4'-pentahydroxyflavone | Human | 2320 | |
| PIM1 | PIM | CAMK | 2o3p | A | B | 3,5,7,3',4'-pentahydroxyflavone | Human | 2409 | |
| PIM1 | PIM | CAMK | 2o63 | A | | 3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)-4h-chromen-4-one | Human | 2453 | |
| PIM1 | PIM | CAMK | 2o64 | A | | 3,5,6,7-tetrahydroxy-2-(3,4-dihydroxyphenyl)-4h-chromen-4-one | Human | 2421 | |
| PIM1 | PIM | CAMK | 2o65 | A | | 5,7-dihydroxy-2-(3,4,5-trihydroxyphenyl)-4h-chromen-4-one | Human | 2324 | |
| PIM1 | PIM | CAMK | 2obj | A | | 6-(5-bromo-2-hydroxyphenyl)-2-oxo-4-phenyl-1,2-dihydropyridine-3-carbonitrile | Human | 2336 | |
| PIM1 | PIM | CAMK | 2oi4 | X | A | - | Human | 7236 | |
| PIM1 | PIM | CAMK | 2oi4 | X | B | - | Human | 7226 | |
| PIM1 | PIM | CAMK | 2xix | A | A | 3,5-diamino-1h-[1,2,4]triazole | Human | 2468 | |
| PIM1 | PIM | CAMK | 2xix | A | B | 3,5-diamino-1h-[1,2,4]triazole | Human | 2433 | |
| PIM1 | PIM | CAMK | 2xiy | A | A | 2-hydroxymethyl-benzoimidazole | Human | 2415 | |
| PIM1 | PIM | CAMK | 2xiy | A | B | 2-hydroxymethyl-benzoimidazole | Human | 2363 | |
| PIM1 | PIM | CAMK | 2xiz | A | A | (e)-pyridin-4-yl-acrylic acid | Human | 2436 | |
| PIM1 | PIM | CAMK | 2xiz | A | B | (e)-pyridin-4-yl-acrylic acid | Human | 2373 | |
| PIM1 | PIM | CAMK | 2xj0 | A | A | (e)-3-(2-amino-pyridine-5yl)-acrylic acid | Human | 2435 | |
| PIM1 | PIM | CAMK | 2xj0 | A | B | (e)-3-(2-amino-pyridine-5yl)-acrylic acid | Human | 2395 | |
| PIM1 | PIM | CAMK | 2xj1 | A | A | (2e)-3-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}phenyl)prop-2-enoic acid | Human | 2469 | |
| PIM1 | PIM | CAMK | 2xj1 | A | B | (2e)-3-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}phenyl)prop-2-enoic acid | Human | 2422 | |
| PIM1 | PIM | CAMK | 2xj2 | A | A | (2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acid | Human | 2334 | |
| PIM1 | PIM | CAMK | 2xj2 | A | B | (2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acid | Human | 2418 | |
| PIM1 | PIM | CAMK | 3a99 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2322 | |
| PIM1 | PIM | CAMK | 3bgp | A | | 4-[3-(4-chlorophenyl)-2,1-benzisoxazol-5-yl]pyrimidin-2-amine | Human | 2359 | |
| PIM1 | PIM | CAMK | 3bgq | A | | n-cyclohexyl-3-[3-(trifluoromethyl)phenyl][1,2,4]triazolo[4,3-b]pyridazin-6-amine | Human | 2465 | |
| PIM1 | PIM | CAMK | 3bgz | A | | 2,3-diphenyl-1h-indole-7-carboxylic acid | Human | 2462 | |
| PIM1 | PIM | CAMK | 3bwf | A | A | - | Human | 7231 | |
| PIM1 | PIM | CAMK | 3bwf | A | B | - | Human | 7235 | |
| PIM1 | PIM | CAMK | 3c4e | A | | n-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amine | Human | 2413 | |
| PIM1 | PIM | CAMK | 3c4e | B | | n-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amine | Human | 2423 | |
| PIM1 | PIM | CAMK | 3c4e | C | | n-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amine | Human | 2440 | |
| PIM1 | PIM | CAMK | 3c4e | D | | n-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amine | Human | 2378 | |
| PIM1 | PIM | CAMK | 3cxw | A | A | (4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 2464 | |
| PIM1 | PIM | CAMK | 3cxw | A | B | (4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 2392 | |
| PIM1 | PIM | CAMK | 3cy2 | A | A | (4r)-7-chloro-9-methyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 2333 | |
| PIM1 | PIM | CAMK | 3cy2 | A | B | (4r)-7-chloro-9-methyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 2459 | |
| PIM1 | PIM | CAMK | 3cy3 | A | | (2s)-1,3-benzothiazol-2-yl{2-[(2-pyridin-3-ylethyl)amino]pyrimidin-4-yl}ethanenitrile | Human | 2443 | |
| PIM1 | PIM | CAMK | 3dcv | A | | 4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-one | Human | 2372 | |
| PIM1 | PIM | CAMK | 3f2a | A | | (2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acid | Human | 2460 | |
| PIM1 | PIM | CAMK | 3jpv | A | | 1,10-dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde | Human | 2431 | |
| PIM1 | PIM | CAMK | 3jxw | A | | 8-[(e)-2-cyclopropylethenyl]-2-[(dimethylamino)methyl][1]benzothieno[3,2-d]pyrimidin-4(3h)-one | Human | 2393 | |
| PIM1 | PIM | CAMK | 3jy0 | A | A | 8-chloro-2-{[(3s)-3-hydroxypyrrolidin-1-yl]methyl}[1]benzothieno[3,2-d]pyrimidin-4(3h)-one | Human | 2405 | |
| PIM1 | PIM | CAMK | 3jya | A | A | 6,9-dichloro[1]benzothieno[3,2-d]pyrimidin-4(3h)-one | Human | 2371 | |
| PIM1 | PIM | CAMK | 3ma3 | A | A | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 2368 | |
| PIM1 | PIM | CAMK | 3ma3 | A | B | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 2347 | |
| PIM1 | PIM | CAMK | 3qf9 | A | A | 6-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}naphthalene-1-carboxamide | Human | 2329 | |
| PIM1 | PIM | CAMK | 3qf9 | A | B | 6-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}naphthalene-1-carboxamide | Human | 2331 | |
| PIM1 | PIM | CAMK | 3r00 | A | | 5-bromo-1-benzofuran-2-carboxylic acid | Human | 2467 | |
| PIM1 | PIM | CAMK | 3r01 | A | | 5-bromo-7-methoxy-1-benzofuran-2-carboxylic acid | Human | 2407 | |
| PIM1 | PIM | CAMK | 3r02 | A | A | 7-[(cis-4-aminocyclohexyl)amino]-5-bromo-1-benzofuran-2-carboxylic acid | Human | 2420 | |
| PIM1 | PIM | CAMK | 3r02 | A | B | 7-[(cis-4-aminocyclohexyl)amino]-5-bromo-1-benzofuran-2-carboxylic acid | Human | 2338 | |
| PIM1 | PIM | CAMK | 3r04 | A | A | 5-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}-1-benzofuran-2-carboxylic acid | Human | 2353 | |
| PIM1 | PIM | CAMK | 3r04 | A | B | 5-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}-1-benzofuran-2-carboxylic acid | Human | 2335 | |
| PIM1 | PIM | CAMK | 3t9i | A | | 2-methoxy-4-(3-phenyl-2h-pyrazolo[3,4-b]pyridin-6-yl)phenol | Human | 2450 | |
| PIM1 | PIM | CAMK | 3uix | A | A | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | 2456 | |
| PIM1 | PIM | CAMK | 3uix | A | B | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | 2387 | |
| PIM1 | PIM | CAMK | 3umw | A | A | (2z)-2-(1h-indazol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3(2h)-one | Human | 2411 | |
| PIM1 | PIM | CAMK | 3umw | A | B | (2z)-2-(1h-indazol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3(2h)-one | Human | 2414 | |
| PIM1 | PIM | CAMK | 3umx | A | A | (2z)-7-(azepan-1-ylmethyl)-6-hydroxy-2-(1h-indol-3-ylmethylidene)-1-benzofuran-3(2h)-one | Human | 2432 | |
| PIM1 | PIM | CAMK | 3umx | A | B | (2z)-7-(azepan-1-ylmethyl)-6-hydroxy-2-(1h-indol-3-ylmethylidene)-1-benzofuran-3(2h)-one | Human | 2375 | |
| PIM1 | PIM | CAMK | 3vbq | A | A | 5-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}benzyl)-2h-1lambda~4~,3-thiazole-2,4(3h)-dione | Human | 2354 | |
| PIM1 | PIM | CAMK | 3vbq | A | B | 5-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}benzyl)-2h-1lambda~4~,3-thiazole-2,4(3h)-dione | Human | 2454 | |
| PIM1 | PIM | CAMK | 3vbt | A | | 4-chloro-2-(1h-pyrazol-3-yl)phenol | Human | 2349 | |
| PIM1 | PIM | CAMK | 3vbv | A | | 8-hydroxyquinoline-2-carboxamide | Human | 2399 | |
| PIM1 | PIM | CAMK | 3vbw | A | | 1,3-dioxo-2,3-dihydro-1h-indene-2-carbonitrile | Human | 2390 | |
| PIM1 | PIM | CAMK | 3vbx | A | A | 6-bromo-4-hydroxy-2h-chromen-2-one | Human | 2427 | |
| PIM1 | PIM | CAMK | 3vbx | A | B | 6-bromo-4-hydroxy-2h-chromen-2-one | Human | 2448 | |
| PIM1 | PIM | CAMK | 3vby | A | | furan-2-yl(1h-indol-3-yl)methanone | Human | 2466 | |
| PIM1 | PIM | CAMK | 3vc4 | A | | (5z)-5-[3-(trifluoromethyl)benzylidene]-1,3-thiazolidine-2,4-dione | Human | 2356 | |
| PIM1 | PIM | CAMK | 3we8 | A | A | cyclopentadienyl(carbon monoxide)(7-oxo-7,10-dihydro-1,8-phenanthrolin-10-yl-kappa~2~c~10~,n~1~)ruthenium | Human | 7237 | |
| PIM1 | PIM | CAMK | 3we8 | A | B | cyclopentadienyl(carbon monoxide)(7-oxo-7,10-dihydro-1,8-phenanthrolin-10-yl-kappa~2~c~10~,n~1~)ruthenium | Human | 7232 | |
| PIM1 | PIM | CAMK | 4a7c | A | | n-(piperidin-4-ylmethyl)-3-[3-(trifluoromethyloxy)phenyl]-[1,2,3]triazolo[4,5-b]pyridin-5-amine | Human | 2321 | |
| PIM1 | PIM | CAMK | 4alu | A | A | 8-bromo-2-(2-chlorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 2452 | |
| PIM1 | PIM | CAMK | 4alu | A | B | 8-bromo-2-(2-chlorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 2384 | |
| PIM1 | PIM | CAMK | 4alv | A | A | 8-bromo-2-{2-chloro-4-[(piperidin-4-ylmethyl)amino]phenyl}[1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 2323 | |
| PIM1 | PIM | CAMK | 4alv | A | B | 8-bromo-2-{2-chloro-4-[(piperidin-4-ylmethyl)amino]phenyl}[1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 2396 | |
| PIM1 | PIM | CAMK | 4alw | A | A | 8-bromanyl-2-[(4-methylpiperazin-1-yl)methyl]-3h-[1]benzofuro[3,2-d]pyrimidin-4-one | Human | 2419 | |
| PIM1 | PIM | CAMK | 4alw | A | B | 8-bromanyl-2-[(4-methylpiperazin-1-yl)methyl]-3h-[1]benzofuro[3,2-d]pyrimidin-4-one | Human | 2350 | |
| PIM1 | PIM | CAMK | 4as0 | A | A | phtalimide-ruthenium complex | Human | 7227 | |
| PIM1 | PIM | CAMK | 4as0 | A | B | phtalimide-ruthenium complex | Human | 7229 | |
| PIM1 | PIM | CAMK | 4bzn | A | | n-(2,2-dimethylpropyl)-2-[1-oxo-7-(thiophen-3-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamide | Human | 2402 | |
| PIM1 | PIM | CAMK | 4bzo | A | | n-[(1s)-2-amino-1-phenylethyl]-2-[(4s)-7-(2-fluoro-4-pyridinyl)-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamide | Human | 2339 | |
| PIM1 | PIM | CAMK | 4dtk | A | A | (5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dione | Human | 2344 | |
| PIM1 | PIM | CAMK | 4dtk | A | B | (5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dione | Human | 2451 | |
| PIM1 | PIM | CAMK | 4enx | A | | (2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-nitrobenzylidene)-1,3-thiazolidin-4-one | Human | 2352 | |
| PIM1 | PIM | CAMK | 4eny | A | A | (2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-one | Human | 2342 | |
| PIM1 | PIM | CAMK | 4eny | A | B | (2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-one | Human | 2424 | |
| PIM1 | PIM | CAMK | 4gw8 | A | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 2428 | |
| PIM1 | PIM | CAMK | 4gw8 | A | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 2391 | |
| PIM1 | PIM | CAMK | 4i41 | A | | 1,4-dihydroxy-5,8-bis({2-[(2-hydroxyethyl)amino]ethyl}amino)-9,10-anthracenedione | Human | 2326 | |
| PIM1 | PIM | CAMK | 4iaa | A | | 10-{2-[(2r)-1-methylpiperidin-2-yl]ethyl}-2-(methylsulfanyl)-10h-phenothiazine | Human | 2325 | |
| PIM1 | PIM | CAMK | 4jx3 | A | | - | Human | 2380 | |
| PIM1 | PIM | CAMK | 4jx7 | A | | 2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6h)-one | Human | 2340 | |
| PIM1 | PIM | CAMK | 4k0y | A | A | n-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2455 | |
| PIM1 | PIM | CAMK | 4k0y | A | B | n-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2445 | |
| PIM1 | PIM | CAMK | 4k18 | A | | 5-(4-cyanobenzyl)-n-(4-fluorophenyl)-7-hydroxypyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2377 | |
| PIM1 | PIM | CAMK | 4k1b | A | | n-[5-(2-fluorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-5-({[(3r,4r)-3-fluoropiperidin-4-yl]methyl}amino)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2362 | |
| PIM1 | PIM | CAMK | 4ll5 | A | A | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | 2365 | |
| PIM1 | PIM | CAMK | 4ll5 | A | B | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | 2382 | |
| PIM1 | PIM | CAMK | 4lm5 | A | A | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | 2400 | |
| PIM1 | PIM | CAMK | 4lm5 | A | B | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | 2327 | |
| PIM1 | PIM | CAMK | 4lmu | A | A | 3,5,7,3',4'-pentahydroxyflavone | Human | 2376 | |
| PIM1 | PIM | CAMK | 4lmu | A | B | 3,5,7,3',4'-pentahydroxyflavone | Human | 2404 | |
| PIM1 | PIM | CAMK | 4mbi | A | | n,n-dimethyl-n'-[3-(1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]ethane-1,2-diamine | Human | 2447 | |
| PIM1 | PIM | CAMK | 4mbl | A | | (1r,2r)-n-[3-(naphthalen-2-yl)pyrazolo[1,5-a]pyrimidin-5-yl]cyclohexane-1,2-diamine | Human | 2381 | |
| PIM1 | PIM | CAMK | 4mta | A | | 2-methyl-5-phenylfuran-3-carboxylic acid | Human | 2370 | |
| PIM1 | PIM | CAMK | 4n6y | A | | 2-(acetylamino)-n-[2-(piperidin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 2383 | |
| PIM1 | PIM | CAMK | 4n6z | A | | 3-amino-n-{4-[(3s)-3-aminopiperidin-1-yl]pyridin-3-yl}pyrazine-2-carboxamide | Human | 2442 | |
| PIM1 | PIM | CAMK | 4n70 | A | A | n-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | Human | 2388 | |
| PIM1 | PIM | CAMK | 4n70 | A | B | n-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | Human | 2357 | |
| PIM1 | PIM | CAMK | 4rbl | A | | 1,4,5,8-tetrahydroxyanthracene-9,10-dione | Human | 2385 | |
| PIM1 | PIM | CAMK | 4rc2 | A | | 1-amino-5,8-dihydroxy-4-({2-[(2-hydroxyethyl)amino]ethyl}amino)anthracene-9,10-dione | Human | 2346 | |
| PIM1 | PIM | CAMK | 4rc3 | A | | 1,4-dihydroxy-5,8-bis{[2-(2-hydroxyethoxy)ethyl]amino}anthracene-9,10-dione | Human | 2412 | |
| PIM1 | PIM | CAMK | 4rc4 | A | | 1,4-bis[(2-aminoethyl)amino]-5,8-dihydroxyanthracene-9,10-dione | Human | 2369 | |
| PIM1 | PIM | CAMK | 4rpv | A | | (3s)-1-{6-[5-(2,6-difluorophenyl)-2h-indazol-3-yl]pyrazin-2-yl}piperidin-3-amine | Human | 2364 | |
| PIM1 | PIM | CAMK | 4ty1 | A | | n-tert-butyl-5-[3-(4-cyclopropylpyrimidin-2-yl)-1h-indol-5-yl]-1,3,4-oxadiazol-2-amine | Human | 2394 | |
| PIM1 | PIM | CAMK | 4wrs | A | | 3-{6-[(4r)-6-azaspiro[2.5]oct-4-yloxy]pyrazin-2-yl}-5-(2,6-difluorophenyl)-1h-indazole | Human | 2439 | |
| PIM1 | PIM | CAMK | 4wsy | A | | 5-[3-(quinolin-3-yl)-2h-indazol-5-yl]-1,3-thiazol-2-amine | Human | 2429 | |
| PIM1 | PIM | CAMK | 4wt6 | A | | 6-[5-(5-amino-1,3,4-thiadiazol-2-yl)-1h-indol-3-yl]-n-cyclopentylpyridin-2-amine | Human | 2386 | |
| PIM1 | PIM | CAMK | 4xh6 | A | | 5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4h-chromen-4-one | Human | 5975 | |
| PIM1 | PIM | CAMK | 4xhk | B | A | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | 2446 | |
| PIM1 | PIM | CAMK | 4xhk | B | B | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | 2355 | |
| PIM1 | PIM | CAMK | 5c1q | B | | 3-methoxy[1]benzothieno[2,3-c]quinolin-6(5h)-one | Human | 6288 | |
| PIM1 | PIM | CAMK | 5dgz | A | | (2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amine | Human | 6209 | |
| PIM1 | PIM | CAMK | 5dhj | A | A | 3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridine | Human | 6212 | |
| PIM1 | PIM | CAMK | 5dhj | A | B | 3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridine | Human | 6211 | |
| PIM1 | PIM | CAMK | 5dia | A | | (1s,3s)-n-{6-[5-(pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridin-3-yl]pyridin-2-yl}cyclohexane-1,3-diamine | Human | 6210 | |
| PIM1 | PIM | CAMK | 5dwr | A | | n-{4-[(1r,3s,5s)-3-amino-5-methylcyclohexyl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | Human | 6238 | |
| PIM1 | PIM | CAMK | 5eol | A | | macrocyclic quinoxaline-pyrrolodihydropiperidinone | Human | 6601 | |
| PIM1 | PIM | CAMK | 5iis | A | | 3-amino-n-(2'-amino-6'-methyl[4,4'-bipyridin]-3-yl)-6-(2-fluorophenyl)pyridine-2-carboxamide | Human | 6504 | |
| PIM1 | PIM | CAMK | 5ipj | A | | 2-(tert-butylamino)-3-methyl-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-one | Human | 6703 | |
| PIM1 | PIM | CAMK | 5kcx | A | A | 4-chloranyl-1-methyl-2-[4-(4-methylpiperazin-1-yl)phenyl]pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 8247 | |
| PIM1 | PIM | CAMK | 5kcx | A | B | 4-chloranyl-1-methyl-2-[4-(4-methylpiperazin-1-yl)phenyl]pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 8248 | |
| PIM1 | PIM | CAMK | 5kgd | A | | 2-pyridin-3-yl-1~{h}-benzimidazole | Human | 8309 | |
| PIM1 | PIM | CAMK | 5kge | A | | 5-(3,4-dichlorophenyl)-1~{h}-pyrazol-3-amine | Human | 8310 | |
| PIM1 | PIM | CAMK | 5kgg | A | | 2-(5-chloranyl-1~{h}-indol-3-yl)ethanamine | Human | 8308 | |
| PIM1 | PIM | CAMK | 5kgi | A | | 2-[3,4-bis(chloranyl)phenoxy]ethanamine | Human | 8306 | |
| PIM1 | PIM | CAMK | 5kgk | A | | 3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amine | Human | 8307 | |
| PIM1 | PIM | CAMK | 5kzi | A | | ~{n}-[4-[(3~{s})-3-azanylpiperidin-1-yl]pyridin-3-yl]-2-[2,6-bis(fluoranyl)phenyl]imidazo[1,5-b]pyridazin-7-amine | Human | 7195 | |
| PIM1 | PIM | CAMK | 5mzl | A | A | ~{n}-quinolin-5-ylpyridine-3-carboxamide | Human | 9562 | |
| PIM1 | PIM | CAMK | 5mzl | A | B | ~{n}-quinolin-5-ylpyridine-3-carboxamide | Human | 9563 | |
| PIM1 | PIM | CAMK | 5n4n | A | A | 3,4-dimethyl-5-(1~{h}-1,2,4-triazol-3-yl)thiophene-2-carbonitrile | Human | 9579 | |
| PIM1 | PIM | CAMK | 5n4n | A | B | 3,4-dimethyl-5-(1~{h}-1,2,4-triazol-3-yl)thiophene-2-carbonitrile | Human | 9595 | |
| PIM1 | PIM | CAMK | 5n4o | A | A | (~{e})-3-(4-methylphenyl)prop-2-enoic acid | Human | 9580 | |
| PIM1 | PIM | CAMK | 5n4o | A | B | (~{e})-3-(4-methylphenyl)prop-2-enoic acid | Human | 9582 | |
| PIM1 | PIM | CAMK | 5n4r | A | A | 2-(azepan-1-yl)-1-(1~{h}-indol-3-yl)propan-1-one | Human | 9584 | |
| PIM1 | PIM | CAMK | 5n4r | A | B | 2-(azepan-1-yl)-1-(1~{h}-indol-3-yl)propan-1-one | Human | 9583 | |
| PIM1 | PIM | CAMK | 5n4u | A | A | 5-(2-azanyl-1,3-thiazol-4-yl)-1,3-dihydrobenzimidazol-2-one | Human | 9588 | |
| PIM1 | PIM | CAMK | 5n4u | A | B | 5-(2-azanyl-1,3-thiazol-4-yl)-1,3-dihydrobenzimidazol-2-one | Human | 9590 | |
| PIM1 | PIM | CAMK | 5n4v | A | A | 2-cyclopropyl-4,5-dimethyl-thieno[2,3-d]pyrimidine-6-carboxylic acid | Human | 9592 | |
| PIM1 | PIM | CAMK | 5n4v | A | B | 2-cyclopropyl-4,5-dimethyl-thieno[2,3-d]pyrimidine-6-carboxylic acid | Human | 9594 | |
| PIM1 | PIM | CAMK | 5n4x | A | A | 4,5-bis(bromanyl)thiophene-2-carbohydrazide | Human | 9600 | |
| PIM1 | PIM | CAMK | 5n4x | A | B | 4,5-bis(bromanyl)thiophene-2-carbohydrazide | Human | 9593 | |
| PIM1 | PIM | CAMK | 5n4y | A | A | 2,5-dihydro-1~{h}-isothiochromeno[4,3-c]pyrazol-3-one | Human | 9589 | |
| PIM1 | PIM | CAMK | 5n4y | A | B | 2,5-dihydro-1~{h}-isothiochromeno[4,3-c]pyrazol-3-one | Human | 9597 | |
| PIM1 | PIM | CAMK | 5n4z | A | A | (~{e})-4-(4-hydroxyphenyl)but-3-en-2-one | Human | 9587 | |
| PIM1 | PIM | CAMK | 5n4z | A | B | (~{e})-4-(4-hydroxyphenyl)but-3-en-2-one | Human | 9599 | |
| PIM1 | PIM | CAMK | 5n50 | A | A | 2-(4-chlorophenyl)sulfanylethanehydrazide | Human | 9585 | |
| PIM1 | PIM | CAMK | 5n50 | A | B | 2-(4-chlorophenyl)sulfanylethanehydrazide | Human | 9598 | |
| PIM1 | PIM | CAMK | 5n51 | A | A | 3,4-bis(bromanyl)thiophene-2-carboxylic acid | Human | 9596 | |
| PIM1 | PIM | CAMK | 5n51 | A | B | 3,4-bis(bromanyl)thiophene-2-carboxylic acid | Human | 9591 | |
| PIM1 | PIM | CAMK | 5n52 | A | A | (~{e})-3-(2,3-dimethoxyphenyl)prop-2-enoic acid | Human | 9581 | |
| PIM1 | PIM | CAMK | 5n52 | A | B | (~{e})-3-(2,3-dimethoxyphenyl)prop-2-enoic acid | Human | 9586 | |
| PIM1 | PIM | CAMK | 5n5l | A | A | 5-bromanyl-1~{h}-indole-3-carboxylic acid | Human | 9703 | |
| PIM1 | PIM | CAMK | 5n5l | A | B | 5-bromanyl-1~{h}-indole-3-carboxylic acid | Human | 9704 | |
| PIM1 | PIM | CAMK | 5n5m | A | A | ~{n}-(isoquinolin-5-ylmethyl)-~{n}-methyl-2-[(3~{r})-pyrrolidin-3-yl]benzamide | Human | 9702 | |
| PIM1 | PIM | CAMK | 5n5m | A | B | ~{n}-(isoquinolin-5-ylmethyl)-~{n}-methyl-2-[(3~{r})-pyrrolidin-3-yl]benzamide | Human | 9705 | |
| PIM1 | PIM | CAMK | 5ndt | A | A | 3-(2-thiophen-2-ylethenyl)-1~{h}-quinoxalin-2-one | Human | 9907 | |
| PIM1 | PIM | CAMK | 5ndt | A | B | 3-(2-thiophen-2-ylethenyl)-1~{h}-quinoxalin-2-one | Human | 9906 | |
| PIM1 | PIM | CAMK | 5o11 | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 8656 | |
| PIM1 | PIM | CAMK | 5o11 | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 8657 | |
| PIM1 | PIM | CAMK | 5o12 | A | | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 8654 | |
| PIM1 | PIM | CAMK | 5o13 | A | A | (3~{e})-5-chloranyl-3-[[5-[3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl]furan-2-yl]methylidene]-1~{h}-indol-2-one | Human | 8653 | |
| PIM1 | PIM | CAMK | 5o13 | A | B | (3~{e})-5-chloranyl-3-[[5-[3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl]furan-2-yl]methylidene]-1~{h}-indol-2-one | Human | 8655 | |
| PIM1 | PIM | CAMK | 5tel | A | A | 4-chloro-2-{5,6-dimethoxy-1-[2-(4-methylpiperazin-1-yl)ethyl]-1h-indol-3-yl}-1h-pyrrolo[2,3-b]pyridine | Human | 8564 | |
| PIM1 | PIM | CAMK | 5tel | A | B | 4-chloro-2-{5,6-dimethoxy-1-[2-(4-methylpiperazin-1-yl)ethyl]-1h-indol-3-yl}-1h-pyrrolo[2,3-b]pyridine | Human | 8562 | |
| PIM1 | PIM | CAMK | 5tex | A | | (4-{4-chloro-1-methyl-2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)methanol | Human | 8566 | |
| PIM1 | PIM | CAMK | 5toe | A | | 2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrile | Human | 8563 | |
| PIM1 | PIM | CAMK | 5tur | A | | 1-methyl-2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrile | Human | 8565 | |
| PIM1 | PIM | CAMK | 5v80 | A | | 1-methyl-4-{3-[6-(piperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[3,4-c]pyridin-5-yl}piperazin-2-one | Human | 9828 | |
| PIM1 | PIM | CAMK | 5v82 | A | | 1-{6-[(3r)-4,4-difluoropiperidin-3-yl]pyridin-2-yl}-6-(6-methylpyrazin-2-yl)-1h-pyrazolo[4,3-c]pyridine | Human | 7581 | |
| PIM1 | PIM | CAMK | 5vua | B | A | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9074 | |
| PIM1 | PIM | CAMK | 5vua | B | B | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9077 | |
| PIM1 | PIM | CAMK | 5vub | B | A | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9073 | |
| PIM1 | PIM | CAMK | 5vub | B | B | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9076 | |
| PIM1 | PIM | CAMK | 5vub | B | C | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9072 | |
| PIM1 | PIM | CAMK | 5vuc | B | A | (2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-one | Human | 9071 | |
| PIM1 | PIM | CAMK | 5vuc | B | B | (2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-one | Human | 9075 | |
| PIM1 | PIM | CAMK | 6ayd | A | A | n-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamide | Human | 9442 | |
| PIM1 | PIM | CAMK | 6ayd | A | B | n-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamide | Human | 9443 | |
| PIM1 | PIM | CAMK | 6bsk | A | | 4-{6-[6-(propan-2-ylamino)-1h-indazol-1-yl]pyrazin-2-yl}benzoic acid | Human | 9758 | |
| PIM1 | PIM | CAMK | 6kzi | A | | 4-(2-chloro-10h-phenoxazin-10-yl)-n,n-diethylbutan-1-amine | Human | 12019 | |
| PIM1 | PIM | CAMK | 6l11 | A | | 5-(2-chloranylphenoxazin-10-yl)-~{n},~{n}-diethyl-pentan-1-amine | Human | 12336 | |
| PIM1 | PIM | CAMK | 6l12 | A | | 4-[(2-chloranylphenoxazin-10-yl)methyl]cyclohexan-1-amine | Human | 12340 | |
| PIM1 | PIM | CAMK | 6l13 | A | | 2-chloranyl-10-(2-piperidin-4-ylethyl)phenoxazine | Human | 12337 | |
| PIM1 | PIM | CAMK | 6l14 | A | | 2-chloranyl-10-[3-[(3~{s})-piperidin-3-yl]propyl]phenoxazine | Human | 12338 | |
| PIM1 | PIM | CAMK | 6l15 | A | | 7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazine | Human | 12339 | |
| PIM1 | PIM | CAMK | 6l16 | A | | 2-[4-[2-(7-chloranylpyrido[3,4-b][1,4]benzoxazin-5-yl)ethyl]piperidin-1-yl]ethanamine | Human | 12335 | |
| PIM1 | PIM | CAMK | 6l17 | A | | 7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazin-8-amine | Human | 12740 | |
| PIM1 | PIM | CAMK | 6mt0 | A | | 3-(1-methylcyclopropyl)-2-[(1-methylcyclopropyl)amino]-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-one | Human | 10850 | |
| PIM1 | PIM | CAMK | 6no8 | A | | 5-amino-n-{5-[(4s)-4-aminoazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide | Human | 11832 | |
| PIM1 | PIM | CAMK | 6no9 | A | | 5-amino-n-{5-[(4r,5r)-4-amino-5-fluoroazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide | Human | 10936 | |
| PIM1 | PIM | CAMK | 6pcw | A | | 4-[5-(cyclopropylcarbamoyl)thiophen-2-yl]-1-benzothiophene-2-carboxamide | Human | 11455 | |
| PIM1 | PIM | CAMK | 6pdi | A | | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11459 | |
| PIM1 | PIM | CAMK | 6pdn | A | A | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acid | Human | 11456 | |
| PIM1 | PIM | CAMK | 6pdn | A | B | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acid | Human | 11458 | |
| PIM1 | PIM | CAMK | 6pdo | A | A | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamide | Human | 11461 | |
| PIM1 | PIM | CAMK | 6pdo | A | B | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamide | Human | 11460 | |
| PIM1 | PIM | CAMK | 6pdp | A | A | 5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamide | Human | 11454 | |
| PIM1 | PIM | CAMK | 6pdp | A | B | 5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamide | Human | 11457 | |
| PIM1 | PIM | CAMK | 6qxk | B | A | 2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-one | Human | 11035 | |
| PIM1 | PIM | CAMK | 6qxk | B | B | 2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-one | Human | 11036 | |
| PIM1 | PIM | CAMK | 6vru | A | A | 3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 13127 | |
| PIM1 | PIM | CAMK | 6vru | A | B | 3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 13128 | |
| PIM1 | PIM | CAMK | 6vrv | A | | 4-chloro-1-{(1s)-1-[(3s)-3-fluoropyrrolidin-3-yl]ethyl}-3-methyl-1h-pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 13129 | |
| PIM1 | PIM | CAMK | 6ykd | A | A | ~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamide | Human | 12402 | |
| PIM1 | PIM | CAMK | 6ykd | A | B | ~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamide | Human | 12401 | |
| PIM1 | PIM | CAMK | 7oov | A | | ~{n}-[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-azanyl-5-[[$l^{1}-azanyl($l^{2}-azanylidene)methyl]-$l^{2}-azanyl]-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]-9-oxidanylidene-9-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]nonanamide | Human | 13824 | |
| PIM1 | PIM | CAMK | 7oow | A | | - | Human | 13826 | |
| PIM1 | PIM | CAMK | 7oox | A | A | - | Human | 13825 | |
| PIM1 | PIM | CAMK | 7oox | A | B | - | Human | 13823 | |
| PIM1 | PIM | CAMK | 7qb2 | A | | 4-[(e)-(6-azanyl-1-methyl-2-oxidanylidene-indol-3-ylidene)methyl]benzoic acid | Human | 14518 | |
| PIM1 | PIM | CAMK | 7qfm | A | A | 4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | 14561 | |
| PIM1 | PIM | CAMK | 7qfm | A | B | 4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | 14560 | |
| PIM1 | PIM | CAMK | 7vsy | A | | - | Human | 15098 | |
| PIM1 | PIM | CAMK | 7xsv | A | A | 8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaene | Human | 14287 | |
| PIM1 | PIM | CAMK | 7xsv | A | B | 8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaene | Human | 14288 | |
| PIM1 | PIM | CAMK | 7z6u | A | A | 4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | 14602 | |
| PIM1 | PIM | CAMK | 7z6u | A | B | 4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | 14600 | |
| PIM1 | PIM | CAMK | 7zun | A | | (4~{s})-4-(2-azanylethyl)-6-phenyl-7-[3-(trifluoromethyloxy)phenyl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1-ol | Human | 14383 | |
| PIM1 | PIM | CAMK | 8afr | A | A | 4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acid | Human | 14603 | |
| PIM1 | PIM | CAMK | 8afr | A | B | 4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acid | Human | 14601 | |
| PIM1 | PIM | CAMK | 8r10 | A | A | (z)-4-(4-hydroxystyryl)benzoic acid | Human | 15214 | |
| PIM1 | PIM | CAMK | 8r10 | A | B | (z)-4-(4-hydroxystyryl)benzoic acid | Human | 15209 | |
| PIM1 | PIM | CAMK | 8r18 | A | A | (e)-4-(4-hydroxystyryl)benzoic acid | Human | 15213 | |
| PIM1 | PIM | CAMK | 8r18 | A | B | (e)-4-(4-hydroxystyryl)benzoic acid | Human | 15208 | |
| PIM1 | PIM | CAMK | 8r1n | A | | 4-(4-hydroxyphenethyl)benzoic acid | Human | 15215 | |
| PIM1 | PIM | CAMK | 8r1p | A | | 4-(4-aminostyryl)benzoic acid | Human | 15210 | |
| PIM1 | PIM | CAMK | 8r1t | A | A | 4-(4-aminophenethyl)benzoic acid | Human | 15212 | |
| PIM1 | PIM | CAMK | 8r1t | A | B | 4-(4-aminophenethyl)benzoic acid | Human | 15211 | |
| PIM2 | PIM | CAMK | 2iwi | A | | ruthenium-pyridocarbazole-1 | Human | 7217 | |
| PIM2 | PIM | CAMK | 2iwi | B | | ruthenium-pyridocarbazole-1 | Human | 7216 | |
| PIM2 | PIM | CAMK | 4x7q | A | | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | 1415 | |
| PIM2 | PIM | CAMK | 4x7q | B | | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | 1416 | |
| PKMYT1 (MYT1) | WEE | Other | 3p1a | A | A | - | Human | 1216 | |
| PKMYT1 (MYT1) | WEE | Other | 3p1a | A | B | - | Human | 1217 | |
| PKMYT1 (MYT1) | WEE | Other | 5vcv | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 8339 | |
| PKMYT1 (MYT1) | WEE | Other | 5vcw | A | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamide | Human | 8335 | |
| PKMYT1 (MYT1) | WEE | Other | 5vcw | B | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamide | Human | 8346 | |
| PKMYT1 (MYT1) | WEE | Other | 5vcx | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 8341 | |
| PKMYT1 (MYT1) | WEE | Other | 5vcy | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 8345 | |
| PKMYT1 (MYT1) | WEE | Other | 5vcy | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 8338 | |
| PKMYT1 (MYT1) | WEE | Other | 5vcz | A | A | 4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 8342 | |
| PKMYT1 (MYT1) | WEE | Other | 5vcz | A | B | 4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 8336 | |
| PKMYT1 (MYT1) | WEE | Other | 5vd0 | A | | 1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 8344 | |
| PKMYT1 (MYT1) | WEE | Other | 5vd1 | A | A | n,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 8337 | |
| PKMYT1 (MYT1) | WEE | Other | 5vd1 | A | B | n,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 8340 | |
| PKMYT1 (MYT1) | WEE | Other | 5vd3 | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 8343 | |
| PKMYT1 (MYT1) | WEE | Other | 8d6c | A | | (1p)-2-amino-6-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 14296 | |
| PKMYT1 (MYT1) | WEE | Other | 8d6d | A | | (1p)-2-amino-5-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 14294 | |
| PKMYT1 (MYT1) | WEE | Other | 8d6e | A | A | (1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamide | Human | 14295 | |
| PKMYT1 (MYT1) | WEE | Other | 8d6e | A | B | (1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamide | Human | 14293 | |
| PKMYT1 (MYT1) | WEE | Other | 8d6f | A | | (1m)-2-amino-1-(5-hydroxy-2-methylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 14297 | |
| PKMYT1 (MYT1) | WEE | Other | 8wjy | A | A | [6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanone | Human | 15008 | |
| PKMYT1 (MYT1) | WEE | Other | 8wjy | A | B | [6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanone | Human | 15007 | |
| PKN1 | PKN | AGC | 4otd | A | A | - | Human | 545 | |
| PKN1 | PKN | AGC | 4otd | A | B | - | Human | 546 | |
| PKN1 | PKN | AGC | 4otg | A | A | lestaurtinib | Human | 548 | |
| PKN1 | PKN | AGC | 4otg | A | B | lestaurtinib | Human | 549 | |
| PKN1 | PKN | AGC | 4oth | A | A | - | Human | 7203 | |
| PKN1 | PKN | AGC | 4oth | A | B | - | Human | 7204 | |
| PKN1 | PKN | AGC | 4oti | A | A | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 551 | |
| PKN1 | PKN | AGC | 4oti | A | B | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 547 | |
| PKN2 | PKN | AGC | 4crs | A | | phosphothiophosphoric acid-adenylate ester | Human | 535 | |
| PLK1 | PLK | Other | 2ou7 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 4956 | |
| PLK1 | PLK | Other | 2ou7 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 4973 | |
| PLK1 | PLK | Other | 2owb | A | A | 4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamide | Human | 4974 | |
| PLK1 | PLK | Other | 2owb | A | B | 4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamide | Human | 4958 | |
| PLK1 | PLK | Other | 2rku | A | A | 4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 4969 | |
| PLK1 | PLK | Other | 2rku | A | B | 4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 4966 | |
| PLK1 | PLK | Other | 2v5q | A | A | - | Human | 4970 | |
| PLK1 | PLK | Other | 2v5q | A | B | - | Human | 4960 | |
| PLK1 | PLK | Other | 2v5q | B | A | - | Human | 4959 | |
| PLK1 | PLK | Other | 2v5q | B | B | - | Human | 4961 | |
| PLK1 | PLK | Other | 2yac | A | | 1-(2-hydroxyethyl)-8-[[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)phenyl]amino]-4,5-dihydropyrimido[5,4-g]indazole-3-carboxamide | Human | 4957 | |
| PLK1 | PLK | Other | 3fc2 | A | A | n-{trans-4-[4-(cyclopropylmethyl)piperazin-1-yl]cyclohexyl}-4-{[(7r)-7-ethyl-5-methyl-8-(1-methylethyl)-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxybenzamide | Human | 4964 | |
| PLK1 | PLK | Other | 3fc2 | A | B | n-{trans-4-[4-(cyclopropylmethyl)piperazin-1-yl]cyclohexyl}-4-{[(7r)-7-ethyl-5-methyl-8-(1-methylethyl)-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxybenzamide | Human | 4967 | |
| PLK1 | PLK | Other | 3kb7 | A | | 8-{[2-methoxy-5-(4-methylpiperazin-1-yl)phenyl]amino}-1-methyl-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4962 | |
| PLK1 | PLK | Other | 3thb | A | | 9-chloro-2-({5-[3-(dimethylamino)propyl]-2-methylpyridin-3-yl}amino)-5,7-dihydro-6h-pyrimido[5,4-d][1]benzazepine-6-thione | Human | 4968 | |
| PLK1 | PLK | Other | 4a4l | A | | 1-methyl-5-(2-{[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)phenyl]amino}pyrimidin-4-yl)-1h-pyrrole-3-carboxamide | Human | 4971 | |
| PLK1 | PLK | Other | 4a4o | A | | 1-methyl-2-(2-{[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)phenyl]amino}pyrimidin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4965 | |
| PLK1 | PLK | Other | 4j52 | A | A | 4-{[(7r)-9-cyclopentyl-7-ethenyl-7-fluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl]amino}-3-methoxy-n-(4-methylpiperazin-1-yl)benzamide | Human | 4955 | |
| PLK1 | PLK | Other | 4j52 | A | B | 4-{[(7r)-9-cyclopentyl-7-ethenyl-7-fluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl]amino}-3-methoxy-n-(4-methylpiperazin-1-yl)benzamide | Human | 4976 | |
| PLK1 | PLK | Other | 4j53 | A | A | 4-[(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-2-fluoro-5-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 4975 | |
| PLK1 | PLK | Other | 4j53 | A | B | 4-[(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-2-fluoro-5-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 4972 | |
| PLK1 | PLK | Other | 4j53 | A | C | 4-[(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-2-fluoro-5-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 4963 | |
| PLK1 | PLK | Other | 5ta6 | A | A | 4-{[(6r)-7-cyano-5-cyclopentyl-6-ethyl-5,6-dihydroimidazo[1,5-f]pteridin-3-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 7465 | |
| PLK1 | PLK | Other | 5ta6 | A | B | 4-{[(6r)-7-cyano-5-cyclopentyl-6-ethyl-5,6-dihydroimidazo[1,5-f]pteridin-3-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 7462 | |
| PLK1 | PLK | Other | 5ta6 | A | C | 4-{[(6r)-7-cyano-5-cyclopentyl-6-ethyl-5,6-dihydroimidazo[1,5-f]pteridin-3-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 7463 | |
| PLK1 | PLK | Other | 5ta8 | A | A | 4-[(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 7464 | |
| PLK1 | PLK | Other | 8bjt | A | | 1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 14712 | |
| PLK1 | PLK | Other | 8x72 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15097 | |
| PLK2 | PLK | Other | 4i5m | A | | 4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamide | Human | 5557 | |
| PLK2 | PLK | Other | 4i5p | A | A | (7r)-8-cyclopentyl-7-ethyl-5-methyl-2-(1h-pyrrol-2-yl)-7,8-dihydropteridin-6(5h)-one | Human | 5559 | |
| PLK2 | PLK | Other | 4i5p | A | B | (7r)-8-cyclopentyl-7-ethyl-5-methyl-2-(1h-pyrrol-2-yl)-7,8-dihydropteridin-6(5h)-one | Human | 5560 | |
| PLK2 | PLK | Other | 4i6b | A | A | (7r)-8-cyclopentyl-7-ethyl-5-methyl-7,8-dihydropteridin-6(5h)-one | Human | 5565 | |
| PLK2 | PLK | Other | 4i6b | A | B | (7r)-8-cyclopentyl-7-ethyl-5-methyl-7,8-dihydropteridin-6(5h)-one | Human | 5562 | |
| PLK2 | PLK | Other | 4i6f | A | A | (7r)-8-cyclopentyl-7-ethyl-5-methyl-2-(2-phenyl-1h-imidazol-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 5564 | |
| PLK2 | PLK | Other | 4i6f | A | B | (7r)-8-cyclopentyl-7-ethyl-5-methyl-2-(2-phenyl-1h-imidazol-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 5563 | |
| PLK2 | PLK | Other | 4i6h | A | A | (7r)-8-cyclopentyl-7-ethyl-5-methyl-2-[2-(1,3-thiazol-4-yl)-1h-imidazol-1-yl]-7,8-dihydropteridin-6(5h)-one | Human | 5558 | |
| PLK2 | PLK | Other | 4i6h | A | B | (7r)-8-cyclopentyl-7-ethyl-5-methyl-2-[2-(1,3-thiazol-4-yl)-1h-imidazol-1-yl]-7,8-dihydropteridin-6(5h)-one | Human | 5561 | |
| PLK3 | PLK | Other | 4b6l | A | | 4-[[(4r)-5-cyclopentyl-4-ethyl-3a,4-dihydro-3h-[1,2,4]triazolo[4,3-f]pteridin-7-yl]amino]-n-cyclopropyl-3-methoxy-benzamide | Human | 3797 | |
| PLK4 | PLK | Other | 3cok | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 1814 | |
| PLK4 | PLK | Other | 3cok | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 1818 | |
| PLK4 | PLK | Other | 3cok | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 1815 | |
| PLK4 | PLK | Other | 3cok | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 1817 | |
| PLK4 | PLK | Other | 4jxf | A | | (1r,2s)-2-{3-[(e)-2-{4-[(dimethylamino)methyl]phenyl}ethenyl]-2h-indazol-6-yl}-5'-methoxyspiro[cyclopropane-1,3'-indol]-2'(1'h)-one | Human | 1816 | |
| PLK4 | PLK | Other | 4yur | A | | 2-({2-fluoro-4-[(2-fluoro-3-nitrobenzyl)sulfonyl]phenyl}sulfanyl)-5-methoxy-n-(3-methyl-1h-pyrazol-5-yl)-6-(morpholin-4-yl)pyrimidin-4-amine | Human | 1813 | |
| Pomk (SGK196) | Other-Unique | Other | 5gz8 | A | | - | Mouse | 8033 | |
| Pomk (SGK196) | Other-Unique | Other | 5gz9 | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 8034 | |
| PRAG1 (SgK223) | NKF3 | Other | 5ve6 | A | | - | Human | 8573 | |
| Prkaa1 (AMPKa1) | CAMKL | CAMK | 5ufu | A | | staurosporine | Mouse | 7590 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4red | A | | - | Human | 122 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4red | B | | - | Human | 123 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4rer | A | | staurosporine | Human | 121 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4rew | A | | staurosporine | Human | 124 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9f | A | | staurosporine | Human | 10716 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9g | A | | staurosporine | Human | 10715 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9h | A | | staurosporine | Human | 10714 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9j | A | | staurosporine | Human | 10717 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jhg | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 13816 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jhh | A | | - | Human | 13817 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jij | B | | - | Human | 13819 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7m74 | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 14017 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 2h6d | A | A | - | Human | 196 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 2h6d | A | B | - | Human | 194 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 2yza | A | | - | Human | 189 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 3aqv | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 193 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cfe | A | | staurosporine | Human | 195 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cfe | C | | staurosporine | Human | 192 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cff | A | | staurosporine | Human | 191 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cff | C | | staurosporine | Human | 190 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | A | A | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6425 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | A | B | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6429 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | C | A | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6427 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | C | B | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6423 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | A | A | staurosporine | Human | 6424 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | A | B | staurosporine | Human | 6428 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | C | A | staurosporine | Human | 6430 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | C | B | staurosporine | Human | 6426 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5iso | A | | staurosporine | Human | 7981 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5iso | C | | staurosporine | Human | 7980 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | A | A | staurosporine | Human | 9848 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | A | B | staurosporine | Human | 9849 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | C | A | staurosporine | Human | 9847 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | C | B | staurosporine | Human | 9850 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b2e | A | | staurosporine | Human | 9851 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6bx6 | A | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 9878 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6bx6 | A | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 9877 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 7myj | A | | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 14273 | |
| Prkaca (PKACa) | PKA | AGC | 1apm | E | A | - | Mouse | 5972 | |
| Prkaca (PKACa) | PKA | AGC | 1apm | E | B | - | Mouse | 5949 | |
| Prkaca (PKACa) | PKA | AGC | 1atp | E | | adenosine-5'-triphosphate | Mouse | 5902 | |
| Prkaca (PKACa) | PKA | AGC | 1bkx | A | | adenosine-5'-monophosphate | Mouse | 5957 | |
| Prkaca (PKACa) | PKA | AGC | 1bx6 | A | | balanol | Mouse | 5955 | |
| Prkaca (PKACa) | PKA | AGC | 1fmo | E | | adenosine | Mouse | 5932 | |
| Prkaca (PKACa) | PKA | AGC | 1j3h | A | | - | Mouse | 5926 | |
| Prkaca (PKACa) | PKA | AGC | 1j3h | B | | - | Mouse | 5873 | |
| Prkaca (PKACa) | PKA | AGC | 1jbp | E | | adenosine-5'-diphosphate | Mouse | 5914 | |
| Prkaca (PKACa) | PKA | AGC | 1jlu | E | | - | Mouse | 5924 | |
| Prkaca (PKACa) | PKA | AGC | 1l3r | E | | adenosine-5'-diphosphate | Mouse | 5950 | |
| Prkaca (PKACa) | PKA | AGC | 1rdq | E | A | adenosine-5'-diphosphate | Mouse | 5964 | |
| Prkaca (PKACa) | PKA | AGC | 1rdq | E | B | adenosine-5'-triphosphate | Mouse | 5927 | |
| Prkaca (PKACa) | PKA | AGC | 1re8 | A | | 3-[(4-hydroxybenzoyl)amino]azepan-4-yl 4-(2-hydroxybenzoyl)benzoate | Mouse | 5923 | |
| Prkaca (PKACa) | PKA | AGC | 1rej | A | | 3-[(4-hydroxybenzoyl)amino]azepan-4-yl 4-hydroxybenzoate | Mouse | 5931 | |
| Prkaca (PKACa) | PKA | AGC | 1rek | A | | 3-[(3-sec-butyl-4-hydroxybenzoyl)amino]azepan-4-yl 4-(2-hydroxy-5-methoxybenzoyl)benzoate | Mouse | 5969 | |
| Prkaca (PKACa) | PKA | AGC | 1syk | A | | - | Mouse | 5891 | |
| Prkaca (PKACa) | PKA | AGC | 1syk | B | | - | Mouse | 5948 | |
| Prkaca (PKACa) | PKA | AGC | 2cpk | E | | - | Mouse | 5959 | |
| Prkaca (PKACa) | PKA | AGC | 2erz | E | | 1-(1-hydroxy-5-isoquinolinesulfonyl)homopiperazine | Mouse | 5895 | |
| Prkaca (PKACa) | PKA | AGC | 2qcs | A | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 5945 | |
| Prkaca (PKACa) | PKA | AGC | 2qcs | A | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 5956 | |
| Prkaca (PKACa) | PKA | AGC | 2qur | A | | - | Mouse | 5896 | |
| Prkaca (PKACa) | PKA | AGC | 2qvs | E | | - | Mouse | 5922 | |
| Prkaca (PKACa) | PKA | AGC | 3fhi | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5951 | |
| Prkaca (PKACa) | PKA | AGC | 3fjq | E | | adenosine-5'-triphosphate | Mouse | 5875 | |
| Prkaca (PKACa) | PKA | AGC | 3idb | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5939 | |
| Prkaca (PKACa) | PKA | AGC | 3idc | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5933 | |
| Prkaca (PKACa) | PKA | AGC | 3j4q | D | A | - | Mouse | 5888 | |
| Prkaca (PKACa) | PKA | AGC | 3j4q | D | B | - | Mouse | 5943 | |
| Prkaca (PKACa) | PKA | AGC | 3j4q | E | A | - | Mouse | 5937 | |
| Prkaca (PKACa) | PKA | AGC | 3j4q | E | B | - | Mouse | 5913 | |
| Prkaca (PKACa) | PKA | AGC | 3j4r | D | A | - | Mouse | 5928 | |
| Prkaca (PKACa) | PKA | AGC | 3j4r | D | B | - | Mouse | 5967 | |
| Prkaca (PKACa) | PKA | AGC | 3j4r | E | A | - | Mouse | 5877 | |
| Prkaca (PKACa) | PKA | AGC | 3j4r | E | B | - | Mouse | 5940 | |
| Prkaca (PKACa) | PKA | AGC | 3o7l | B | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5908 | |
| Prkaca (PKACa) | PKA | AGC | 3o7l | D | | - | Mouse | 5958 | |
| Prkaca (PKACa) | PKA | AGC | 3ow3 | A | | (2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amine | Mouse | 5941 | |
| Prkaca (PKACa) | PKA | AGC | 3pvb | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5880 | |
| Prkaca (PKACa) | PKA | AGC | 3qal | E | | adenosine-5'-triphosphate | Mouse | 5921 | |
| Prkaca (PKACa) | PKA | AGC | 3qam | E | | adenosine-5'-triphosphate | Mouse | 5906 | |
| Prkaca (PKACa) | PKA | AGC | 3tnp | C | | - | Mouse | 5889 | |
| Prkaca (PKACa) | PKA | AGC | 3tnp | F | | - | Mouse | 5893 | |
| Prkaca (PKACa) | PKA | AGC | 3x2u | A | A | adenosine-5'-triphosphate | Mouse | 6294 | |
| Prkaca (PKACa) | PKA | AGC | 3x2u | A | B | adenosine-5'-triphosphate | Mouse | 6298 | |
| Prkaca (PKACa) | PKA | AGC | 3x2v | A | A | adenosine-5'-triphosphate | Mouse | 6299 | |
| Prkaca (PKACa) | PKA | AGC | 3x2v | A | B | adenosine-5'-triphosphate | Mouse | 6297 | |
| Prkaca (PKACa) | PKA | AGC | 3x2w | A | A | adenosine-5'-triphosphate | Mouse | 6296 | |
| Prkaca (PKACa) | PKA | AGC | 3x2w | A | B | adenosine-5'-triphosphate | Mouse | 6295 | |
| Prkaca (PKACa) | PKA | AGC | 4dfx | E | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 5925 | |
| Prkaca (PKACa) | PKA | AGC | 4dfx | E | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 5885 | |
| Prkaca (PKACa) | PKA | AGC | 4dfy | A | | - | Mouse | 5886 | |
| Prkaca (PKACa) | PKA | AGC | 4dfy | E | | - | Mouse | 5960 | |
| Prkaca (PKACa) | PKA | AGC | 4dfz | E | A | - | Mouse | 5874 | |
| Prkaca (PKACa) | PKA | AGC | 4dfz | E | B | - | Mouse | 5966 | |
| Prkaca (PKACa) | PKA | AGC | 4dfz | E | C | - | Mouse | 5971 | |
| Prkaca (PKACa) | PKA | AGC | 4dg0 | E | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 5929 | |
| Prkaca (PKACa) | PKA | AGC | 4dg0 | E | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 5892 | |
| Prkaca (PKACa) | PKA | AGC | 4dg2 | E | A | - | Mouse | 5952 | |
| Prkaca (PKACa) | PKA | AGC | 4dg2 | E | B | - | Mouse | 5962 | |
| Prkaca (PKACa) | PKA | AGC | 4dg3 | E | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5898 | |
| Prkaca (PKACa) | PKA | AGC | 4dh1 | A | | adenosine-5'-triphosphate | Mouse | 5907 | |
| Prkaca (PKACa) | PKA | AGC | 4dh3 | A | | adenosine-5'-triphosphate | Mouse | 5965 | |
| Prkaca (PKACa) | PKA | AGC | 4dh5 | A | | adenosine-5'-diphosphate | Mouse | 5917 | |
| Prkaca (PKACa) | PKA | AGC | 4dh7 | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5934 | |
| Prkaca (PKACa) | PKA | AGC | 4dh8 | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5904 | |
| Prkaca (PKACa) | PKA | AGC | 4din | A | | adenosine-5'-triphosphate | Mouse | 5919 | |
| Prkaca (PKACa) | PKA | AGC | 4hpt | E | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 5899 | |
| Prkaca (PKACa) | PKA | AGC | 4hpt | E | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 5884 | |
| Prkaca (PKACa) | PKA | AGC | 4hpu | E | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 5963 | |
| Prkaca (PKACa) | PKA | AGC | 4hpu | E | B | - | Mouse | 5882 | |
| Prkaca (PKACa) | PKA | AGC | 4iac | A | | phosphomethylphosphonic acid adenylate ester | Mouse | 5936 | |
| Prkaca (PKACa) | PKA | AGC | 4iad | A | | adenosine-5'-diphosphate | Mouse | 5883 | |
| Prkaca (PKACa) | PKA | AGC | 4iaf | A | | adenosine-5'-diphosphate | Mouse | 5876 | |
| Prkaca (PKACa) | PKA | AGC | 4iai | A | A | adenosine-5'-diphosphate | Mouse | 5881 | |
| Prkaca (PKACa) | PKA | AGC | 4iai | A | B | adenosine-5'-diphosphate | Mouse | 5901 | |
| Prkaca (PKACa) | PKA | AGC | 4iai | A | C | adenosine-5'-diphosphate | Mouse | 5912 | |
| Prkaca (PKACa) | PKA | AGC | 4iak | A | A | adenosine-5'-diphosphate | Mouse | 5903 | |
| Prkaca (PKACa) | PKA | AGC | 4iak | A | B | adenosine-5'-diphosphate | Mouse | 5918 | |
| Prkaca (PKACa) | PKA | AGC | 4iay | A | | adenosine-5'-diphosphate | Mouse | 5911 | |
| Prkaca (PKACa) | PKA | AGC | 4iaz | A | A | adenosine-5'-diphosphate | Mouse | 5900 | |
| Prkaca (PKACa) | PKA | AGC | 4iaz | A | B | adenosine-5'-diphosphate | Mouse | 5938 | |
| Prkaca (PKACa) | PKA | AGC | 4ib0 | A | A | adenosine-5'-diphosphate | Mouse | 5947 | |
| Prkaca (PKACa) | PKA | AGC | 4ib0 | A | B | adenosine-5'-diphosphate | Mouse | 5910 | |
| Prkaca (PKACa) | PKA | AGC | 4ib1 | A | A | adenosine-5'-diphosphate | Mouse | 5968 | |
| Prkaca (PKACa) | PKA | AGC | 4ib1 | A | B | adenosine-5'-diphosphate | Mouse | 5961 | |
| Prkaca (PKACa) | PKA | AGC | 4ib3 | A | | adenosine-5'-diphosphate | Mouse | 5944 | |
| Prkaca (PKACa) | PKA | AGC | 4nts | A | | - | Mouse | 5920 | |
| Prkaca (PKACa) | PKA | AGC | 4nts | B | | - | Mouse | 5879 | |
| Prkaca (PKACa) | PKA | AGC | 4ntt | A | | adenosine-5'-diphosphate | Mouse | 5942 | |
| Prkaca (PKACa) | PKA | AGC | 4ntt | B | | adenosine-5'-diphosphate | Mouse | 5905 | |
| Prkaca (PKACa) | PKA | AGC | 4o21 | A | A | adenosine-5'-diphosphate | Mouse | 5954 | |
| Prkaca (PKACa) | PKA | AGC | 4o21 | A | B | adenosine-5'-diphosphate | Mouse | 5909 | |
| Prkaca (PKACa) | PKA | AGC | 4o22 | A | A | - | Mouse | 5953 | |
| Prkaca (PKACa) | PKA | AGC | 4o22 | A | B | - | Mouse | 5970 | |
| Prkaca (PKACa) | PKA | AGC | 4wbb | B | | - | Mouse | 5930 | |
| Prkaca (PKACa) | PKA | AGC | 4x6q | C | | - | Mouse | 5916 | |
| Prkaca (PKACa) | PKA | AGC | 4x6r | A | A | adenosine-5'-triphosphate | Mouse | 5897 | |
| Prkaca (PKACa) | PKA | AGC | 4x6r | A | B | adenosine-5'-triphosphate | Mouse | 5887 | |
| Prkaca (PKACa) | PKA | AGC | 4xw4 | A | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 5946 | |
| Prkaca (PKACa) | PKA | AGC | 4xw4 | A | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 5935 | |
| Prkaca (PKACa) | PKA | AGC | 4xw5 | A | A | adenosine-5'-triphosphate | Mouse | 5890 | |
| Prkaca (PKACa) | PKA | AGC | 4xw5 | A | B | adenosine-5'-triphosphate | Mouse | 5894 | |
| Prkaca (PKACa) | PKA | AGC | 4xw6 | A | A | adenosine-5'-diphosphate | Mouse | 5878 | |
| Prkaca (PKACa) | PKA | AGC | 4xw6 | A | B | adenosine-5'-diphosphate | Mouse | 5915 | |
| Prkaca (PKACa) | PKA | AGC | 5jr7 | A | | adenosine-5'-diphosphate | Mouse | 7509 | |
| Prkaca (PKACa) | PKA | AGC | 5jr7 | C | | adenosine-5'-diphosphate | Mouse | 7510 | |
| Prkaca (PKACa) | PKA | AGC | 5x3f | B | | - | Mouse | 8191 | |
| Prkaca (PKACa) | PKA | AGC | 6e21 | A | A | adenosine-5'-diphosphate | Mouse | 11316 | |
| Prkaca (PKACa) | PKA | AGC | 6e21 | A | B | adenosine-5'-diphosphate | Mouse | 11323 | |
| Prkaca (PKACa) | PKA | AGC | 6mm5 | E | A | - | Mouse | 11319 | |
| Prkaca (PKACa) | PKA | AGC | 6mm5 | E | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 11315 | |
| Prkaca (PKACa) | PKA | AGC | 6mm6 | C | A | - | Mouse | 11326 | |
| Prkaca (PKACa) | PKA | AGC | 6mm6 | C | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 11310 | |
| Prkaca (PKACa) | PKA | AGC | 6mm6 | C | C | phosphoaminophosphonic acid-adenylate ester | Mouse | 11321 | |
| Prkaca (PKACa) | PKA | AGC | 6mm6 | E | A | - | Mouse | 11311 | |
| Prkaca (PKACa) | PKA | AGC | 6mm6 | E | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 11314 | |
| Prkaca (PKACa) | PKA | AGC | 6mm6 | E | C | phosphoaminophosphonic acid-adenylate ester | Mouse | 11320 | |
| Prkaca (PKACa) | PKA | AGC | 6mm7 | A | A | - | Mouse | 11325 | |
| Prkaca (PKACa) | PKA | AGC | 6mm7 | A | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 11322 | |
| Prkaca (PKACa) | PKA | AGC | 6mm7 | D | A | - | Mouse | 11312 | |
| Prkaca (PKACa) | PKA | AGC | 6mm7 | D | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 11318 | |
| Prkaca (PKACa) | PKA | AGC | 6mm8 | C | A | - | Mouse | 11317 | |
| Prkaca (PKACa) | PKA | AGC | 6mm8 | C | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 11324 | |
| Prkaca (PKACa) | PKA | AGC | 6mm8 | C | C | phosphoaminophosphonic acid-adenylate ester | Mouse | 11313 | |
| Prkaca (PKACa) | PKA | AGC | 7e0z | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 14205 | |
| Prkaca (PKACa) | PKA | AGC | 7e11 | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 14206 | |
| PRKACA (PKACa) | PKA | AGC | 2gu8 | A | | n-[(1s)-2-amino-1-(2,4-dichlorobenzyl)ethyl]-5-[2-(methylamino)pyrimidin-4-yl]thiophene-2-carboxamide | Human | 5295 | |
| PRKACA (PKACa) | PKA | AGC | 3agl | A | | (10r,20r,23r)-1-[(2s,3s,4r,5r)-5-(6-amino-9h-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]-20,23-bis(3-carbamimidamidopropyl)-10-methyl-1,8,11,18,21-pentaoxo-2,9,12,19,22-pentaazatetracosan-24-amide | Human | 5267 | |
| PRKACA (PKACa) | PKA | AGC | 3agl | B | | (10r,20r,23r)-1-[(2s,3s,4r,5r)-5-(6-amino-9h-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]-20,23-bis(3-carbamimidamidopropyl)-10-methyl-1,8,11,18,21-pentaoxo-2,9,12,19,22-pentaazatetracosan-24-amide | Human | 5283 | |
| PRKACA (PKACa) | PKA | AGC | 3agm | A | | - | Human | 5282 | |
| PRKACA (PKACa) | PKA | AGC | 3ama | A | | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 5284 | |
| PRKACA (PKACa) | PKA | AGC | 3amb | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 5276 | |
| PRKACA (PKACa) | PKA | AGC | 3l9l | A | | 5-[2-({(2s)-2-amino-3-[4-(trifluoromethyl)phenyl]propyl}amino)-1,3-thiazol-5-yl]-1,3-dihydro-2h-indol-2-one | Human | 5305 | |
| PRKACA (PKACa) | PKA | AGC | 3l9l | B | | 5-[2-({(2s)-2-amino-3-[4-(trifluoromethyl)phenyl]propyl}amino)-1,3-thiazol-5-yl]-1,3-dihydro-2h-indol-2-one | Human | 5302 | |
| PRKACA (PKACa) | PKA | AGC | 3l9m | A | | (2s)-n~1~-[5-(3-methyl-1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamine | Human | 5270 | |
| PRKACA (PKACa) | PKA | AGC | 3l9m | B | | (2s)-n~1~-[5-(3-methyl-1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamine | Human | 5278 | |
| PRKACA (PKACa) | PKA | AGC | 3l9n | A | | (2s)-n~1~-[5-(1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamine | Human | 5292 | |
| PRKACA (PKACa) | PKA | AGC | 3mvj | A | | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 5289 | |
| PRKACA (PKACa) | PKA | AGC | 3mvj | B | | - | Human | 5288 | |
| PRKACA (PKACa) | PKA | AGC | 3mvj | E | | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 5291 | |
| PRKACA (PKACa) | PKA | AGC | 3nx8 | A | A | - | Human | 5277 | |
| PRKACA (PKACa) | PKA | AGC | 3nx8 | A | B | - | Human | 5294 | |
| PRKACA (PKACa) | PKA | AGC | 3oog | A | A | 1-(4-hydroxy-3-methylphenyl)ethanone | Human | 5281 | |
| PRKACA (PKACa) | PKA | AGC | 3oog | A | B | 1-(4-hydroxy-3-methylphenyl)ethanone | Human | 5272 | |
| PRKACA (PKACa) | PKA | AGC | 3ovv | A | A | n'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5266 | |
| PRKACA (PKACa) | PKA | AGC | 3ovv | A | B | n'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5269 | |
| PRKACA (PKACa) | PKA | AGC | 3owp | A | A | (2s)-2-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylethanehydrazide | Human | 5273 | |
| PRKACA (PKACa) | PKA | AGC | 3owp | A | B | (2s)-2-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylethanehydrazide | Human | 5296 | |
| PRKACA (PKACa) | PKA | AGC | 3oxt | A | | (2s)-2-amino-n'-[(1e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-phenylethanehydrazide | Human | 5268 | |
| PRKACA (PKACa) | PKA | AGC | 3p0m | A | A | (2r)-4-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylbutanehydrazide | Human | 5297 | |
| PRKACA (PKACa) | PKA | AGC | 3p0m | A | B | (2r)-4-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylbutanehydrazide | Human | 5279 | |
| PRKACA (PKACa) | PKA | AGC | 3poo | A | A | n'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5300 | |
| PRKACA (PKACa) | PKA | AGC | 3poo | A | B | n'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5285 | |
| PRKACA (PKACa) | PKA | AGC | 3vqh | A | A | n-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamide | Human | 5271 | |
| PRKACA (PKACa) | PKA | AGC | 3vqh | A | B | n-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamide | Human | 5275 | |
| PRKACA (PKACa) | PKA | AGC | 4ae6 | A | A | - | Human | 5274 | |
| PRKACA (PKACa) | PKA | AGC | 4ae6 | A | B | - | Human | 5301 | |
| PRKACA (PKACa) | PKA | AGC | 4ae6 | B | A | - | Human | 5290 | |
| PRKACA (PKACa) | PKA | AGC | 4ae6 | B | B | - | Human | 5298 | |
| PRKACA (PKACa) | PKA | AGC | 4ae9 | A | A | - | Human | 5265 | |
| PRKACA (PKACa) | PKA | AGC | 4ae9 | A | B | - | Human | 5307 | |
| PRKACA (PKACa) | PKA | AGC | 4ae9 | B | A | - | Human | 5299 | |
| PRKACA (PKACa) | PKA | AGC | 4ae9 | B | B | - | Human | 5286 | |
| PRKACA (PKACa) | PKA | AGC | 4uj1 | A | | 7-[(3s,4r)-4-(3-chlorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6548 | |
| PRKACA (PKACa) | PKA | AGC | 4uj2 | A | A | 7-[(3s,4r)-4-(3-iodanylphenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6550 | |
| PRKACA (PKACa) | PKA | AGC | 4uj2 | A | B | 7-[(3s,4r)-4-(3-iodanylphenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6551 | |
| PRKACA (PKACa) | PKA | AGC | 4uj9 | A | | 7-[(3s,4r)-4-[4-(trifluoromethyl)phenyl]carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6544 | |
| PRKACA (PKACa) | PKA | AGC | 4uja | A | A | 7-{(3s,4r)-4-[(5-bromothiophen-2-yl)carbonyl]pyrrolidin-3-yl}quinazolin-4(3h)-one | Human | 6549 | |
| PRKACA (PKACa) | PKA | AGC | 4uja | A | B | 7-{(3s,4r)-4-[(5-bromothiophen-2-yl)carbonyl]pyrrolidin-3-yl}quinazolin-4(3h)-one | Human | 6547 | |
| PRKACA (PKACa) | PKA | AGC | 4ujb | A | A | 7-[(3s,4r)-4-(3-fluorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6546 | |
| PRKACA (PKACa) | PKA | AGC | 4ujb | A | B | 7-[(3s,4r)-4-(3-fluorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6545 | |
| PRKACA (PKACa) | PKA | AGC | 4wb5 | A | A | adenosine-5'-triphosphate | Human | 5280 | |
| PRKACA (PKACa) | PKA | AGC | 4wb5 | A | B | adenosine-5'-triphosphate | Human | 5306 | |
| PRKACA (PKACa) | PKA | AGC | 4wb6 | A | | adenosine-5'-triphosphate | Human | 5303 | |
| PRKACA (PKACa) | PKA | AGC | 4wb6 | B | | adenosine-5'-triphosphate | Human | 5293 | |
| PRKACA (PKACa) | PKA | AGC | 4wb7 | A | A | adenosine-5'-triphosphate | Human | 6876 | |
| PRKACA (PKACa) | PKA | AGC | 4wb7 | A | B | adenosine-5'-triphosphate | Human | 6878 | |
| PRKACA (PKACa) | PKA | AGC | 4wb7 | B | A | adenosine-5'-triphosphate | Human | 6875 | |
| PRKACA (PKACa) | PKA | AGC | 4wb7 | B | B | adenosine-5'-triphosphate | Human | 6877 | |
| PRKACA (PKACa) | PKA | AGC | 4wb8 | A | A | adenosine-5'-triphosphate | Human | 5304 | |
| PRKACA (PKACa) | PKA | AGC | 4wb8 | A | B | adenosine-5'-triphosphate | Human | 5287 | |
| PRKACA (PKACa) | PKA | AGC | 5bx6 | A | A | 4-chlorophthalazin-1(2h)-one | Human | 7075 | |
| PRKACA (PKACa) | PKA | AGC | 5bx6 | A | B | 4-chlorophthalazin-1(2h)-one | Human | 7078 | |
| PRKACA (PKACa) | PKA | AGC | 5bx7 | A | A | 1-benzothiophen-3-ylmethanol | Human | 7076 | |
| PRKACA (PKACa) | PKA | AGC | 5bx7 | A | B | 1-benzothiophen-3-ylmethanol | Human | 7077 | |
| PRKACA (PKACa) | PKA | AGC | 5izf | A | | - | Human | 6854 | |
| PRKACA (PKACa) | PKA | AGC | 5izj | A | A | - | Human | 6857 | |
| PRKACA (PKACa) | PKA | AGC | 5izj | A | B | - | Human | 6855 | |
| PRKACA (PKACa) | PKA | AGC | 5izj | B | A | - | Human | 6851 | |
| PRKACA (PKACa) | PKA | AGC | 5izj | B | B | - | Human | 6858 | |
| PRKACA (PKACa) | PKA | AGC | 5j5x | A | A | - | Human | 6853 | |
| PRKACA (PKACa) | PKA | AGC | 5j5x | A | B | - | Human | 6856 | |
| PRKACA (PKACa) | PKA | AGC | 5j5x | A | C | - | Human | 6852 | |
| PRKACA (PKACa) | PKA | AGC | 5n23 | A | A | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 9747 | |
| PRKACA (PKACa) | PKA | AGC | 5n23 | A | B | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 9746 | |
| PRKACA (PKACa) | PKA | AGC | 5uzk | A | A | 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(1h-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Human | 9726 | |
| PRKACA (PKACa) | PKA | AGC | 6byr | A | | adenosine-5'-triphosphate | Human | 11256 | |
| PRKACA (PKACa) | PKA | AGC | 6byr | C | | adenosine-5'-triphosphate | Human | 11258 | |
| PRKACA (PKACa) | PKA | AGC | 6bys | A | | - | Human | 11259 | |
| PRKACA (PKACa) | PKA | AGC | 6bys | C | | - | Human | 11257 | |
| PRKACA (PKACa) | PKA | AGC | 6bys | E | | - | Human | 11262 | |
| PRKACA (PKACa) | PKA | AGC | 6bys | G | | - | Human | 11260 | |
| PRKACA (PKACa) | PKA | AGC | 6c0u | A | | n-[(3r,4r)-4-{[4-(2-fluoro-3-methoxy-6-propoxybenzene-1-carbonyl)benzene-1-carbonyl]amino}pyrrolidin-3-yl]-1h-indazole-5-carboxamide | Human | 9974 | |
| PRKACA (PKACa) | PKA | AGC | 6frx | A | | ~{n}-[3-[(5-chloranyl-2-phenylazanyl-pyrimidin-4-yl)amino]phenyl]prop-2-enamide | Human | 11261 | |
| PRKACA (PKACa) | PKA | AGC | 6no7 | A | | - | Human | 11465 | |
| PRKACA (PKACa) | PKA | AGC | 6no7 | C | | - | Human | 11466 | |
| PRKACA (PKACa) | PKA | AGC | 6no7 | E | | adenosine-5'-triphosphate | Human | 11463 | |
| PRKACA (PKACa) | PKA | AGC | 6no7 | G | | adenosine-5'-triphosphate | Human | 11464 | |
| PRKACA (PKACa) | PKA | AGC | 6qj7 | A | A | ~{n}'-[(2~{s})-2-[3,5-bis(fluoranyl)phenyl]-2-oxidanyl-ethanoyl]-2-ethyl-3-methyl-4-oxidanyl-benzohydrazide | Human | 11990 | |
| PRKACA (PKACa) | PKA | AGC | 6qj7 | A | B | ~{n}'-[(2~{s})-2-[3,5-bis(fluoranyl)phenyl]-2-oxidanyl-ethanoyl]-2-ethyl-3-methyl-4-oxidanyl-benzohydrazide | Human | 11991 | |
| PRKACA (PKACa) | PKA | AGC | 6wjf | A | | - | Human | 13008 | |
| PRKACA (PKACa) | PKA | AGC | 6wjf | B | | - | Human | 13009 | |
| PRKACA (PKACa) | PKA | AGC | 6wjg | A | | - | Human | 13006 | |
| PRKACA (PKACa) | PKA | AGC | 6wjg | B | | - | Human | 13007 | |
| PRKACA (PKACa) | PKA | AGC | 7y1g | A | A | 1-chloranyl-~{n}-[(~{s})-(3-chloranyl-4-cyano-phenyl)-[(2~{r},4~{s})-4-oxidanylpyrrolidin-2-yl]methyl]-7-methoxy-isoquinoline-6-carboxamide | Human | 14422 | |
| PRKACA (PKACa) | PKA | AGC | 7y1g | A | B | 1-chloranyl-~{n}-[(~{s})-(3-chloranyl-4-cyano-phenyl)-[(2~{r},4~{s})-4-oxidanylpyrrolidin-2-yl]methyl]-7-methoxy-isoquinoline-6-carboxamide | Human | 14423 | |
| PRKACA (PKACa) | PKA | AGC | 8fe2 | A | | 6-[(6m)-6-(1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-9h-purine | Human | 14889 | |
| PRKACA (PKACa) | PKA | AGC | 8fe5 | A | | 6-[(6p)-6-(1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-7,9-dihydro-8h-purin-8-one | Human | 14888 | |
| PRKACA (PKACa) | PKA | AGC | 8fec | A | | 6-[(6p)-6-(4-bromo-1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-7h-purine | Human | 14890 | |
| PRKACA (PKACa) | PKA | AGC | 8x5l | A | | (2s)-2-(4-chlorophenyl)-2-hydroxy-2-[4-(1h-pyrazol-4-yl)phenyl]ethanaminium | Human | 15111 | |
| PRKCA (PKCa) | PKC | AGC | 3iw4 | A | | 3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dione | Human | 3041 | |
| PRKCA (PKCa) | PKC | AGC | 3iw4 | B | | 3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dione | Human | 3039 | |
| PRKCA (PKCa) | PKC | AGC | 3iw4 | C | | 3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dione | Human | 3042 | |
| PRKCA (PKCa) | PKC | AGC | 4ra4 | A | | (1r)-9-[(3s,4s)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 3040 | |
| PRKCA (PKCa) | PKC | AGC | 8u37 | A | A | (6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamide | Human | 15159 | |
| PRKCA (PKCa) | PKC | AGC | 8u37 | A | B | (6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamide | Human | 15162 | |
| PRKCA (PKCa) | PKC | AGC | 8uak | A | A | (6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamide | Human | 15161 | |
| PRKCA (PKCa) | PKC | AGC | 8uak | A | B | (6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamide | Human | 15160 | |
| PRKCB (PKCb) | PKC | AGC | 2i0e | A | | 3-{1-[3-(dimethylamino)propyl]-2-methyl-1h-indol-3-yl}-4-(2-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2550 | |
| PRKCB (PKCb) | PKC | AGC | 2i0e | B | | 3-{1-[3-(dimethylamino)propyl]-2-methyl-1h-indol-3-yl}-4-(2-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2549 | |
| PRKCH (PKCh) | PKC | AGC | 3txo | A | | 2-methyl-n~1~-[3-(pyridin-4-yl)-2,6-naphthyridin-1-yl]propane-1,2-diamine | Human | 2316 | |
| PRKCH (PKCh) | PKC | AGC | 8fp1 | A | | (3p)-3-[6-chloro-4-(9-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | 14694 | |
| PRKCH (PKCh) | PKC | AGC | 8fp3 | A | A | (3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | Human | 14696 | |
| PRKCH (PKCh) | PKC | AGC | 8fp3 | A | B | (3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | Human | 14695 | |
| Prkci (PKCi) | PKC | AGC | 4dc2 | A | A | adenine | Mouse | 5830 | |
| Prkci (PKCi) | PKC | AGC | 4dc2 | A | B | adenine | Mouse | 5829 | |
| PRKCI (PKCi) | PKC | AGC | 1zrz | A | | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3354 | |
| PRKCI (PKCi) | PKC | AGC | 3a8w | A | | adenosine-5'-triphosphate | Human | 3353 | |
| PRKCI (PKCi) | PKC | AGC | 3a8w | B | | adenosine-5'-triphosphate | Human | 3346 | |
| PRKCI (PKCi) | PKC | AGC | 3a8x | A | | - | Human | 3351 | |
| PRKCI (PKCi) | PKC | AGC | 3a8x | B | | - | Human | 3348 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | A | A | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3349 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | A | B | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3350 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | B | A | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3356 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | B | B | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3347 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | C | A | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3355 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | C | B | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3352 | |
| PRKCI (PKCi) | PKC | AGC | 5li1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 7072 | |
| PRKCI (PKCi) | PKC | AGC | 5li1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 7067 | |
| PRKCI (PKCi) | PKC | AGC | 5li9 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 7068 | |
| PRKCI (PKCi) | PKC | AGC | 5li9 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 7074 | |
| PRKCI (PKCi) | PKC | AGC | 5lih | A | A | adenosine-5'-diphosphate | Human | 7071 | |
| PRKCI (PKCi) | PKC | AGC | 5lih | A | B | adenosine-5'-diphosphate | Human | 7070 | |
| PRKCI (PKCi) | PKC | AGC | 5lih | B | A | adenosine-5'-diphosphate | Human | 7069 | |
| PRKCI (PKCi) | PKC | AGC | 5lih | B | B | adenosine-5'-diphosphate | Human | 7073 | |
| PRKCI (PKCi) | PKC | AGC | 6ilz | A | | 2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamide | Human | 11358 | |
| PRKCI (PKCi) | PKC | AGC | 6ilz | C | | 2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamide | Human | 11357 | |
| PRKCI (PKCi) | PKC | AGC | 6ilz | E | | 2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamide | Human | 11356 | |
| PRKCI (PKCi) | PKC | AGC | 6ilz | G | | 2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamide | Human | 11355 | |
| PRKCQ (PKCt) | PKC | AGC | 1xjd | A | | staurosporine | Human | 5357 | |
| PRKCQ (PKCt) | PKC | AGC | 2jed | A | | 3-(8-dimethylaminomethyl-6,7,8,9-tetrahydro-pyrido[1,2-a]indol-10-yl)-4-(1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 5352 | |
| PRKCQ (PKCt) | PKC | AGC | 2jed | B | | 3-(8-dimethylaminomethyl-6,7,8,9-tetrahydro-pyrido[1,2-a]indol-10-yl)-4-(1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 5358 | |
| PRKCQ (PKCt) | PKC | AGC | 4q9z | A | A | (1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5356 | |
| PRKCQ (PKCt) | PKC | AGC | 4q9z | A | B | (1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5353 | |
| PRKCQ (PKCt) | PKC | AGC | 4q9z | B | A | (1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5355 | |
| PRKCQ (PKCt) | PKC | AGC | 4q9z | B | B | (1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5362 | |
| PRKCQ (PKCt) | PKC | AGC | 4ra5 | A | A | (1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5354 | |
| PRKCQ (PKCt) | PKC | AGC | 4ra5 | A | B | (1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5359 | |
| PRKCQ (PKCt) | PKC | AGC | 4ra5 | B | A | (1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5361 | |
| PRKCQ (PKCt) | PKC | AGC | 4ra5 | B | B | (1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5360 | |
| PRKCQ (PKCt) | PKC | AGC | 5f9e | A | A | 2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-one | Human | 6630 | |
| PRKCQ (PKCt) | PKC | AGC | 5f9e | A | B | 2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-one | Human | 6629 | |
| PRKCQ (PKCt) | PKC | AGC | 5f9e | B | A | 2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-one | Human | 6631 | |
| PRKCQ (PKCt) | PKC | AGC | 5f9e | B | B | 2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-one | Human | 6628 | |
| PRKG1 (PKG1) | PKG | AGC | 6bdl | A | A | - | Human | 10641 | |
| PRKG1 (PKG1) | PKG | AGC | 6bdl | A | B | - | Human | 10644 | |
| PRKG1 (PKG1) | PKG | AGC | 6bdl | B | A | - | Human | 10643 | |
| PRKG1 (PKG1) | PKG | AGC | 6bdl | B | B | - | Human | 10642 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 10670 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 10667 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 10668 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 10666 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 10669 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 10672 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 10671 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 10665 | |
| PRKG1 (PKG1) | PKG | AGC | 6c0t | A | | n-[(3r,4r)-4-{[4-(2-fluoro-3-methoxy-6-propoxybenzene-1-carbonyl)benzene-1-carbonyl]amino}pyrrolidin-3-yl]-1h-indazole-5-carboxamide | Human | 9975 | |
| PRKG1 (PKG1) | PKG | AGC | 7lv3 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14343 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4t | A | A | adenosine-5'-triphosphate | Human | 14791 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4t | A | B | adenosine-5'-triphosphate | Human | 14795 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4u | A | A | - | Human | 14788 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4u | A | B | - | Human | 14789 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4v | A | A | - | Human | 14790 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4v | A | B | - | Human | 14792 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4w | A | A | - | Human | 14794 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4w | A | B | - | Human | 14793 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ian | A | | - | Human | 5543 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ian | B | | - | Human | 5546 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ifc | A | A | adenosine-5'-diphosphate | Human | 5538 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ifc | A | B | adenosine-5'-diphosphate | Human | 5544 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ifc | B | A | adenosine-5'-diphosphate | Human | 5542 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ifc | B | B | adenosine-5'-diphosphate | Human | 5540 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4iir | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5545 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4iir | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5539 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4iir | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 5536 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4iir | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 5537 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ijp | A | A | 4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 5547 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ijp | A | B | 4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 5535 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ijp | B | A | 4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 5541 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ijp | B | B | 4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 5534 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6cnh | A | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 9776 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6cnh | A | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 9775 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | A | A | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11585 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | A | B | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11577 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | B | A | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11583 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | B | B | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11581 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | C | A | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11578 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | C | B | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11586 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | D | A | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11580 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | D | B | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11579 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pk6 | A | A | 4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11582 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pk6 | A | B | 4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11584 | |
| PRPF4B (PRP4) | DYRK | CMGC | 8h6e | H | | - | Human | 15282 | |
| PRPF4B (PRP4) | DYRK | CMGC | 8h6j | H | A | - | Human | 15281 | |
| PRPF4B (PRP4) | DYRK | CMGC | 8h6j | H | B | - | Human | 15283 | |
| PTK2 (FAK) | FAK | TK | 1mp8 | A | | adenosine-5'-diphosphate | Human | 217 | |
| PTK2 (FAK) | FAK | TK | 2etm | A | | 7-pyridin-2-yl-n-(3,4,5-trimethoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-2-amine | Human | 246 | |
| PTK2 (FAK) | FAK | TK | 2etm | B | | 7-pyridin-2-yl-n-(3,4,5-trimethoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-2-amine | Human | 225 | |
| PTK2 (FAK) | FAK | TK | 2ijm | A | A | adenosine-5'-triphosphate | Human | 215 | |
| PTK2 (FAK) | FAK | TK | 2ijm | A | B | adenosine-5'-triphosphate | Human | 243 | |
| PTK2 (FAK) | FAK | TK | 2ijm | B | A | adenosine-5'-diphosphate | Human | 220 | |
| PTK2 (FAK) | FAK | TK | 2ijm | B | B | adenosine-5'-diphosphate | Human | 249 | |
| PTK2 (FAK) | FAK | TK | 3bz3 | A | A | n-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamide | Human | 228 | |
| PTK2 (FAK) | FAK | TK | 3bz3 | A | B | n-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamide | Human | 227 | |
| PTK2 (FAK) | FAK | TK | 3pxk | A | | 6-(4,4-dimethylpent-2-yn-1-yl)-1lambda~4~-pyrrolo[2,3-d][1,3]thiazole | Human | 241 | |
| PTK2 (FAK) | FAK | TK | 3pxk | B | | 6-(4,4-dimethylpent-2-yn-1-yl)-1lambda~4~-pyrrolo[2,3-d][1,3]thiazole | Human | 236 | |
| PTK2 (FAK) | FAK | TK | 4ebv | A | A | - | Human | 237 | |
| PTK2 (FAK) | FAK | TK | 4ebv | A | B | - | Human | 231 | |
| PTK2 (FAK) | FAK | TK | 4ebv | A | C | - | Human | 224 | |
| PTK2 (FAK) | FAK | TK | 4ebw | A | A | - | Human | 218 | |
| PTK2 (FAK) | FAK | TK | 4ebw | A | B | - | Human | 219 | |
| PTK2 (FAK) | FAK | TK | 4ebw | A | C | - | Human | 235 | |
| PTK2 (FAK) | FAK | TK | 4gu6 | A | A | n-(3-{[(5-cyano-2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)amino]methyl}pyridin-2-yl)-n-methylmethanesulfonamide | Human | 252 | |
| PTK2 (FAK) | FAK | TK | 4gu6 | A | B | n-(3-{[(5-cyano-2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)amino]methyl}pyridin-2-yl)-n-methylmethanesulfonamide | Human | 226 | |
| PTK2 (FAK) | FAK | TK | 4gu6 | B | A | n-(3-{[(5-cyano-2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)amino]methyl}pyridin-2-yl)-n-methylmethanesulfonamide | Human | 240 | |
| PTK2 (FAK) | FAK | TK | 4gu6 | B | B | n-(3-{[(5-cyano-2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)amino]methyl}pyridin-2-yl)-n-methylmethanesulfonamide | Human | 223 | |
| PTK2 (FAK) | FAK | TK | 4gu9 | A | | n-(2-fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 222 | |
| PTK2 (FAK) | FAK | TK | 4gu9 | B | | n-(2-fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 221 | |
| PTK2 (FAK) | FAK | TK | 4i4e | A | A | [4-(2-hydroxyethyl)piperidin-1-yl][4-(5-methyl-4,4-dioxido-1,5-dihydropyrazolo[4,3-c][2,1]benzothiazin-8-yl)phenyl]methanone | Human | 245 | |
| PTK2 (FAK) | FAK | TK | 4i4e | A | B | [4-(2-hydroxyethyl)piperidin-1-yl][4-(5-methyl-4,4-dioxido-1,5-dihydropyrazolo[4,3-c][2,1]benzothiazin-8-yl)phenyl]methanone | Human | 216 | |
| PTK2 (FAK) | FAK | TK | 4i4e | A | C | [4-(2-hydroxyethyl)piperidin-1-yl][4-(5-methyl-4,4-dioxido-1,5-dihydropyrazolo[4,3-c][2,1]benzothiazin-8-yl)phenyl]methanone | Human | 234 | |
| PTK2 (FAK) | FAK | TK | 4i4f | A | A | - | Human | 238 | |
| PTK2 (FAK) | FAK | TK | 4i4f | A | B | - | Human | 251 | |
| PTK2 (FAK) | FAK | TK | 4i4f | A | C | - | Human | 232 | |
| PTK2 (FAK) | FAK | TK | 4k8a | A | | 3-bromo-5-(2h-tetrazol-5-yl)pyridine | Human | 244 | |
| PTK2 (FAK) | FAK | TK | 4k8a | B | | 3-bromo-5-(2h-tetrazol-5-yl)pyridine | Human | 239 | |
| PTK2 (FAK) | FAK | TK | 4k9y | A | A | 1-[4-(6-amino-9h-purin-9-yl)phenyl]-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 230 | |
| PTK2 (FAK) | FAK | TK | 4k9y | A | B | 1-[4-(6-amino-9h-purin-9-yl)phenyl]-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 233 | |
| PTK2 (FAK) | FAK | TK | 4k9y | A | C | 1-[4-(6-amino-9h-purin-9-yl)phenyl]-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 229 | |
| PTK2 (FAK) | FAK | TK | 4kab | A | | 3-methyl-1,5-dihydropyrazolo[4,3-c]pyrazole | Human | 242 | |
| PTK2 (FAK) | FAK | TK | 4kab | B | | 3-methyl-1,5-dihydropyrazolo[4,3-c]pyrazole | Human | 250 | |
| PTK2 (FAK) | FAK | TK | 4kao | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(pyridin-3-yl)phenyl]urea | Human | 248 | |
| PTK2 (FAK) | FAK | TK | 4kao | B | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(pyridin-3-yl)phenyl]urea | Human | 253 | |
| PTK2 (FAK) | FAK | TK | 4q9s | A | | 3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 247 | |
| PTK2 (FAK) | FAK | TK | 6i8z | A | | 3-methoxy-~{n}-(1-methylpiperidin-1-ium-4-yl)-4-[[4-[(3-oxidanylidene-1,2-dihydroinden-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide | Human | 10904 | |
| PTK2 (FAK) | FAK | TK | 6yoj | A | A | 6-[[4-[(3-methylsulfonylphenyl)methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3,4-dihydro-1~{h}-quinolin-2-one | Human | 13319 | |
| PTK2 (FAK) | FAK | TK | 6yoj | A | B | 6-[[4-[(3-methylsulfonylphenyl)methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3,4-dihydro-1~{h}-quinolin-2-one | Human | 13316 | |
| PTK2 (FAK) | FAK | TK | 6yq1 | A | A | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13332 | |
| PTK2 (FAK) | FAK | TK | 6yq1 | A | B | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13327 | |
| PTK2 (FAK) | FAK | TK | 6yq1 | B | A | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13317 | |
| PTK2 (FAK) | FAK | TK | 6yq1 | B | B | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13312 | |
| PTK2 (FAK) | FAK | TK | 6yq1 | C | A | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13315 | |
| PTK2 (FAK) | FAK | TK | 6yq1 | C | B | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13324 | |
| PTK2 (FAK) | FAK | TK | 6yq1 | D | A | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13330 | |
| PTK2 (FAK) | FAK | TK | 6yq1 | D | B | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13333 | |
| PTK2 (FAK) | FAK | TK | 6yr9 | A | A | n-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamide | Human | 13325 | |
| PTK2 (FAK) | FAK | TK | 6yr9 | A | B | n-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamide | Human | 13313 | |
| PTK2 (FAK) | FAK | TK | 6yr9 | B | A | n-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamide | Human | 13326 | |
| PTK2 (FAK) | FAK | TK | 6yr9 | B | B | n-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamide | Human | 13328 | |
| PTK2 (FAK) | FAK | TK | 6yr9 | C | A | n-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamide | Human | 13311 | |
| PTK2 (FAK) | FAK | TK | 6yr9 | C | B | n-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamide | Human | 13334 | |
| PTK2 (FAK) | FAK | TK | 6yr9 | D | A | n-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamide | Human | 13321 | |
| PTK2 (FAK) | FAK | TK | 6yr9 | D | B | n-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamide | Human | 13314 | |
| PTK2 (FAK) | FAK | TK | 6yt6 | B | A | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-1,3-dihydroindol-5-yl)amino]pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13271 | |
| PTK2 (FAK) | FAK | TK | 6yt6 | B | B | ~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-1,3-dihydroindol-5-yl)amino]pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamide | Human | 13272 | |
| PTK2 (FAK) | FAK | TK | 6yvs | A | A | 5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-one | Human | 13323 | |
| PTK2 (FAK) | FAK | TK | 6yvs | A | B | 5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-one | Human | 13310 | |
| PTK2 (FAK) | FAK | TK | 6yvs | B | A | 5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-one | Human | 13335 | |
| PTK2 (FAK) | FAK | TK | 6yvs | B | B | 5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-one | Human | 13331 | |
| PTK2 (FAK) | FAK | TK | 6yvs | C | A | 5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-one | Human | 13320 | |
| PTK2 (FAK) | FAK | TK | 6yvs | C | B | 5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-one | Human | 13307 | |
| PTK2 (FAK) | FAK | TK | 6yvs | D | A | 5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-one | Human | 13318 | |
| PTK2 (FAK) | FAK | TK | 6yvs | D | B | 5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-one | Human | 13309 | |
| PTK2 (FAK) | FAK | TK | 6yvy | A | A | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13275 | |
| PTK2 (FAK) | FAK | TK | 6yvy | A | B | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13270 | |
| PTK2 (FAK) | FAK | TK | 6yvy | B | A | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13276 | |
| PTK2 (FAK) | FAK | TK | 6yvy | B | B | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13267 | |
| PTK2 (FAK) | FAK | TK | 6yvy | C | A | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13269 | |
| PTK2 (FAK) | FAK | TK | 6yvy | C | B | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13268 | |
| PTK2 (FAK) | FAK | TK | 6yvy | D | A | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13273 | |
| PTK2 (FAK) | FAK | TK | 6yvy | D | B | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 13274 | |
| PTK2 (FAK) | FAK | TK | 6yxv | A | | ~{n}-methyl-~{n}-[3-[(~{e})-[2-phenylazanyl-5-(trifluoromethyl)pyrimidin-4-yl]iminomethyl]pyridin-2-yl]methanesulfonamide | Human | 13336 | |
| PTK2 (FAK) | FAK | TK | 6yxv | B | | ~{n}-methyl-~{n}-[3-[(~{e})-[2-phenylazanyl-5-(trifluoromethyl)pyrimidin-4-yl]iminomethyl]pyridin-2-yl]methanesulfonamide | Human | 13329 | |
| PTK2 (FAK) | FAK | TK | 6yxv | C | | ~{n}-methyl-~{n}-[3-[(~{e})-[2-phenylazanyl-5-(trifluoromethyl)pyrimidin-4-yl]iminomethyl]pyridin-2-yl]methanesulfonamide | Human | 13322 | |
| PTK2 (FAK) | FAK | TK | 6yxv | D | | ~{n}-methyl-~{n}-[3-[(~{e})-[2-phenylazanyl-5-(trifluoromethyl)pyrimidin-4-yl]iminomethyl]pyridin-2-yl]methanesulfonamide | Human | 13308 | |
| PTK2 (FAK) | FAK | TK | 7pi4 | D | A | - | Human | 13913 | |
| PTK2 (FAK) | FAK | TK | 7pi4 | D | B | - | Human | 13914 | |
| PTK2B (PYK2) | FAK | TK | 3cc6 | A | A | - | Human | 93 | |
| PTK2B (PYK2) | FAK | TK | 3cc6 | A | B | - | Human | 92 | |
| PTK2B (PYK2) | FAK | TK | 3et7 | A | | 5-{[4-{[2-(pyrrolidin-1-ylsulfonyl)benzyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,3-dihydro-2h-indol-2-one | Human | 90 | |
| PTK2B (PYK2) | FAK | TK | 3fzo | A | | - | Human | 95 | |
| PTK2B (PYK2) | FAK | TK | 3fzp | A | | phosphothiophosphoric acid-adenylate ester | Human | 88 | |
| PTK2B (PYK2) | FAK | TK | 3fzr | A | | n-methyl-n-{2-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]phenyl}methanesulfonamide | Human | 87 | |
| PTK2B (PYK2) | FAK | TK | 3fzs | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 94 | |
| PTK2B (PYK2) | FAK | TK | 3fzt | A | | 1-[5-tert-butyl-2-(4-methylphenyl)-1,2-dihydro-3h-pyrazol-3-ylidene]-3-{3-[(pyridin-3-yloxy)methyl]-1h-pyrazol-5-yl}urea | Human | 86 | |
| PTK2B (PYK2) | FAK | TK | 3h3c | A | | 4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 96 | |
| PTK2B (PYK2) | FAK | TK | 4h1j | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(4-methoxy-2-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 91 | |
| PTK2B (PYK2) | FAK | TK | 4h1m | A | | 7-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)-n-(propan-2-yl)-1h-indole-2-carboxamide | Human | 89 | |
| PTK2B (PYK2) | FAK | TK | 5to8 | A | | 25-(methylsulfonyl)-8-(trifluoromethyl)-5,17,18,21,22,23,24,25-octahydro-12h-7,11-(azeno)-16,13-(metheno)pyrido[3,2-i]pyrrolo[1,2-q][1,3,7,11,17]pentaazacyclohenicosin-20(6h)-one | Human | 7316 | |
| PTK2B (PYK2) | FAK | TK | 5tob | A | | n-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamide | Human | 8686 | |
| PTK2B (PYK2) | FAK | TK | 8xox | A | A | n-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamide | Human | 15171 | |
| PTK2B (PYK2) | FAK | TK | 8xox | A | B | n-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamide | Human | 15172 | |
| PTK2B (PYK2) | FAK | TK | 8ygx | A | A | - | Human | 15245 | |
| PTK2B (PYK2) | FAK | TK | 8ygx | A | B | - | Human | 15244 | |
| PTK6 (BRK) | Src | TK | 5d7v | A | A | - | Human | 6953 | |
| PTK6 (BRK) | Src | TK | 5d7v | A | B | - | Human | 6950 | |
| PTK6 (BRK) | Src | TK | 5d7v | B | A | - | Human | 6955 | |
| PTK6 (BRK) | Src | TK | 5d7v | B | B | - | Human | 6951 | |
| PTK6 (BRK) | Src | TK | 5d7v | C | A | - | Human | 6949 | |
| PTK6 (BRK) | Src | TK | 5d7v | C | B | - | Human | 6954 | |
| PTK6 (BRK) | Src | TK | 5d7v | D | A | - | Human | 6948 | |
| PTK6 (BRK) | Src | TK | 5d7v | D | B | - | Human | 6952 | |
| PTK6 (BRK) | Src | TK | 5da3 | A | A | (2-chloro-4-{[6-cyclopropyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanone | Human | 6989 | |
| PTK6 (BRK) | Src | TK | 5da3 | A | B | (2-chloro-4-{[6-cyclopropyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanone | Human | 6988 | |
| PTK6 (BRK) | Src | TK | 5h2u | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7338 | |
| PTK6 (BRK) | Src | TK | 5h2u | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7343 | |
| PTK6 (BRK) | Src | TK | 5h2u | B | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7339 | |
| PTK6 (BRK) | Src | TK | 5h2u | B | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7337 | |
| PTK6 (BRK) | Src | TK | 5h2u | C | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7341 | |
| PTK6 (BRK) | Src | TK | 5h2u | C | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7342 | |
| PTK6 (BRK) | Src | TK | 5h2u | D | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7344 | |
| PTK6 (BRK) | Src | TK | 5h2u | D | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7340 | |
| PTK6 (BRK) | Src | TK | 6cz2 | A | A | - | Human | 10030 | |
| PTK6 (BRK) | Src | TK | 6cz2 | A | B | - | Human | 10031 | |
| PTK6 (BRK) | Src | TK | 6cz3 | A | A | (3-fluoro-4-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanone | Human | 10001 | |
| PTK6 (BRK) | Src | TK | 6cz3 | A | B | (3-fluoro-4-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanone | Human | 9999 | |
| PTK6 (BRK) | Src | TK | 6cz4 | A | A | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamide | Human | 9998 | |
| PTK6 (BRK) | Src | TK | 6cz4 | A | B | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamide | Human | 10000 | |
| PTK7 (CCK4) | CCK4 | TK | 6vg3 | A | | - | Human | 12292 | |
| PTK7 (CCK4) | CCK4 | TK | 6vg3 | B | | - | Human | 12293 | |
| PTK7 (CCK4) | CCK4 | TK | 6vg3 | C | | - | Human | 12291 | |
| RAF1 | RAF | TKL | 3omv | A | | (1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oxime | Human | 937 | |
| RAF1 | RAF | TKL | 3omv | B | | (1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oxime | Human | 936 | |
| RAF1 | RAF | TKL | 8chf | A | | 2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanol | Human | 15220 | |
| RAF1 | RAF | TKL | 8cpd | A | | - | Human | 15221 | |
| RAF1 | RAF | TKL | 8gae | D | | - | Human | 14715 | |
| RAF1 | RAF | TKL | 8gft | D | | - | Human | 14725 | |
| RAF1 | RAF | TKL | 8u1l | C | | - | Human | 15219 | |
| RET | Ret | TK | 2ivs | A | A | (3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxide | Human | 3372 | |
| RET | Ret | TK | 2ivs | A | B | (3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxide | Human | 3369 | |
| RET | Ret | TK | 2ivs | B | A | (3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxide | Human | 3357 | |
| RET | Ret | TK | 2ivs | B | B | (3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxide | Human | 3374 | |
| RET | Ret | TK | 2ivt | A | A | adenosine monophosphate | Human | 3361 | |
| RET | Ret | TK | 2ivt | A | B | adenosine monophosphate | Human | 3365 | |
| RET | Ret | TK | 2ivu | A | | 4-bromo-2-fluoro-n-[(4e)-6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4(1h)-ylidene]aniline | Human | 3364 | |
| RET | Ret | TK | 2ivv | A | | 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 3373 | |
| RET | Ret | TK | 2x2k | A | A | (3z)-5-amino-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3360 | |
| RET | Ret | TK | 2x2k | A | B | (3z)-5-amino-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3358 | |
| RET | Ret | TK | 2x2l | A | A | (3z)-5-amino-3-[(4-methoxyphenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3363 | |
| RET | Ret | TK | 2x2l | A | B | (3z)-5-amino-3-[(4-methoxyphenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3371 | |
| RET | Ret | TK | 2x2l | A | C | (3z)-5-amino-3-[(4-methoxyphenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3367 | |
| RET | Ret | TK | 2x2m | A | | (3z)-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3366 | |
| RET | Ret | TK | 2x2m | B | | (3z)-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 3375 | |
| RET | Ret | TK | 4cki | A | A | adenosine | Human | 3362 | |
| RET | Ret | TK | 4cki | A | B | adenosine | Human | 3370 | |
| RET | Ret | TK | 4cki | A | C | adenosine | Human | 3368 | |
| RET | Ret | TK | 4ckj | A | A | adenosine | Human | 3359 | |
| RET | Ret | TK | 4ckj | A | B | adenosine | Human | 3376 | |
| RET | Ret | TK | 5amn | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 6412 | |
| RET | Ret | TK | 5fm2 | A | | 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 7328 | |
| RET | Ret | TK | 5fm3 | A | | 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 7327 | |
| RET | Ret | TK | 6fek | A | A | adenosine | Human | 9604 | |
| RET | Ret | TK | 6fek | A | B | adenosine | Human | 9603 | |
| RET | Ret | TK | 6i82 | A | A | ~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamine | Human | 12050 | |
| RET | Ret | TK | 6i82 | A | B | ~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamine | Human | 12054 | |
| RET | Ret | TK | 6i82 | B | A | ~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamine | Human | 12052 | |
| RET | Ret | TK | 6i82 | B | B | ~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamine | Human | 12053 | |
| RET | Ret | TK | 6i83 | A | | 4-[5-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]benzamide | Human | 12051 | |
| RET | Ret | TK | 6ne7 | A | A | adenosine monophosphate | Human | 11149 | |
| RET | Ret | TK | 6ne7 | A | B | adenosine monophosphate | Human | 11148 | |
| RET | Ret | TK | 6ne7 | A | C | adenosine monophosphate | Human | 11152 | |
| RET | Ret | TK | 6nec | A | A | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11151 | |
| RET | Ret | TK | 6nec | A | B | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11150 | |
| RET | Ret | TK | 6nec | C | A | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11147 | |
| RET | Ret | TK | 6nec | C | B | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 11153 | |
| RET | Ret | TK | 6nja | A | A | adenine | Human | 11146 | |
| RET | Ret | TK | 6nja | A | B | adenine | Human | 11145 | |
| RET | Ret | TK | 6vhg | A | A | 3-(3,4-dimethoxyphenyl)-n~5~-(1-methylpiperidin-4-yl)-6-phenylpyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 11997 | |
| RET | Ret | TK | 6vhg | A | B | 3-(3,4-dimethoxyphenyl)-n~5~-(1-methylpiperidin-4-yl)-6-phenylpyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 11998 | |
| RET | Ret | TK | 7du8 | A | A | selpercatinib | Human | 14096 | |
| RET | Ret | TK | 7du8 | A | B | selpercatinib | Human | 14095 | |
| RET | Ret | TK | 7du9 | A | A | pralsetinib | Human | 14050 | |
| RET | Ret | TK | 7du9 | A | B | pralsetinib | Human | 14047 | |
| RET | Ret | TK | 7dua | A | A | 4-azanyl-7-(1-methylcyclopropyl)-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamide | Human | 14048 | |
| RET | Ret | TK | 7dua | A | B | 4-azanyl-7-(1-methylcyclopropyl)-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamide | Human | 14049 | |
| RET | Ret | TK | 7dua | A | C | 4-azanyl-7-(1-methylcyclopropyl)-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamide | Human | 14046 | |
| RET | Ret | TK | 7ju5 | A | A | pralsetinib | Human | 13106 | |
| RET | Ret | TK | 7ju5 | A | B | pralsetinib | Human | 13109 | |
| RET | Ret | TK | 7ju5 | B | A | pralsetinib | Human | 13105 | |
| RET | Ret | TK | 7ju5 | B | B | pralsetinib | Human | 13108 | |
| RET | Ret | TK | 7ju6 | A | A | selpercatinib | Human | 13103 | |
| RET | Ret | TK | 7ju6 | A | B | selpercatinib | Human | 13107 | |
| RET | Ret | TK | 7ju6 | B | A | selpercatinib | Human | 13110 | |
| RET | Ret | TK | 7ju6 | B | B | selpercatinib | Human | 13104 | |
| RET | Ret | TK | 7nzn | A | | 2-[4-[[4-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]-6-[(3-methyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]-~{n}-(3-fluorophenyl)ethanamide | Human | 14105 | |
| RET | Ret | TK | 7run | A | | 1-(4-{(1s,3s)-3-[4-amino-5-(3-amino-4-chlorophenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl}piperazin-1-yl)ethan-1-one | Human | 14072 | |
| RIOK1 | RIO | Atypical | 4otp | A | | adenosine-5'-diphosphate | Human | 9156 | |
| RIOK1 | RIO | Atypical | 6g5i | z | | - | Human | 10004 | |
| RIOK1 | RIO | Atypical | 6zv6 | I | A | - | Human | 13546 | |
| RIOK1 | RIO | Atypical | 6zv6 | I | B | - | Human | 13545 | |
| RIOK1 | RIO | Atypical | 6zxd | z | | - | Human | 13013 | |
| RIOK1 | RIO | Atypical | 6zxe | z | | - | Human | 13011 | |
| RIOK1 | RIO | Atypical | 6zxf | z | | adenosine-5'-triphosphate | Human | 13010 | |
| RIOK1 | RIO | Atypical | 6zxg | z | | adenosine-5'-triphosphate | Human | 13012 | |
| RIOK1 | RIO | Atypical | 6zxh | z | | adenosine-5'-triphosphate | Human | 13073 | |
| RIOK2 | RIO | Atypical | 6fdm | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 10875 | |
| RIOK2 | RIO | Atypical | 6fdm | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 10877 | |
| RIOK2 | RIO | Atypical | 6fdm | B | A | - | Human | 10869 | |
| RIOK2 | RIO | Atypical | 6fdm | B | B | - | Human | 10871 | |
| RIOK2 | RIO | Atypical | 6fdm | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 10874 | |
| RIOK2 | RIO | Atypical | 6fdm | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 10876 | |
| RIOK2 | RIO | Atypical | 6fdm | D | A | - | Human | 10868 | |
| RIOK2 | RIO | Atypical | 6fdm | D | B | - | Human | 10872 | |
| RIOK2 | RIO | Atypical | 6fdn | A | | - | Human | 10873 | |
| RIOK2 | RIO | Atypical | 6fdn | B | | - | Human | 10867 | |
| RIOK2 | RIO | Atypical | 6fdo | A | | - | Human | 10878 | |
| RIOK2 | RIO | Atypical | 6fdo | B | | - | Human | 10870 | |
| RIOK2 | RIO | Atypical | 6g18 | v | | - | Human | 9986 | |
| RIOK2 | RIO | Atypical | 6g51 | v | | - | Human | 9985 | |
| RIOK2 | RIO | Atypical | 6hk6 | A | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10638 | |
| RIOK2 | RIO | Atypical | 6hk6 | B | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10636 | |
| RIOK2 | RIO | Atypical | 6hk6 | C | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10639 | |
| RIOK2 | RIO | Atypical | 6hk6 | D | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10634 | |
| RIOK2 | RIO | Atypical | 6hk6 | E | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10633 | |
| RIOK2 | RIO | Atypical | 6hk6 | F | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10637 | |
| RIOK2 | RIO | Atypical | 6hk6 | G | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10640 | |
| RIOK2 | RIO | Atypical | 6hk6 | H | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10632 | |
| RIOK2 | RIO | Atypical | 6hk6 | I | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10631 | |
| RIOK2 | RIO | Atypical | 6hk6 | J | | 2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamide | Human | 10635 | |
| RIOK2 | RIO | Atypical | 7vbt | A | | 8-(6-methoxypyridin-3-yl)-1-[4-piperazin-1-yl-3-(trifluoromethyl)phenyl]-5h-[1,2,3]triazolo[4,5-c]quinolin-4-one | Human | 14274 | |
| RIPK1 | RIPK | TKL | 4ith | A | A | (5r)-5-[(7-chloro-1h-indol-3-yl)methyl]-3-methylimidazolidine-2,4-dione | Human | 566 | |
| RIPK1 | RIPK | TKL | 4ith | A | B | (5r)-5-[(7-chloro-1h-indol-3-yl)methyl]-3-methylimidazolidine-2,4-dione | Human | 567 | |
| RIPK1 | RIPK | TKL | 4ith | B | A | (5r)-5-[(7-chloro-1h-indol-3-yl)methyl]-3-methylimidazolidine-2,4-dione | Human | 564 | |
| RIPK1 | RIPK | TKL | 4ith | B | B | (5r)-5-[(7-chloro-1h-indol-3-yl)methyl]-3-methylimidazolidine-2,4-dione | Human | 571 | |
| RIPK1 | RIPK | TKL | 4iti | A | A | 1-{(3s,3as)-3-[3-fluoro-4-(trifluoromethoxy)phenyl]-8-methoxy-3,3a,4,5-tetrahydro-2h-benzo[g]indazol-2-yl}-2-hydroxyethanone | Human | 570 | |
| RIPK1 | RIPK | TKL | 4iti | A | B | 1-{(3s,3as)-3-[3-fluoro-4-(trifluoromethoxy)phenyl]-8-methoxy-3,3a,4,5-tetrahydro-2h-benzo[g]indazol-2-yl}-2-hydroxyethanone | Human | 563 | |
| RIPK1 | RIPK | TKL | 4iti | B | A | 1-{(3s,3as)-3-[3-fluoro-4-(trifluoromethoxy)phenyl]-8-methoxy-3,3a,4,5-tetrahydro-2h-benzo[g]indazol-2-yl}-2-hydroxyethanone | Human | 562 | |
| RIPK1 | RIPK | TKL | 4iti | B | B | 1-{(3s,3as)-3-[3-fluoro-4-(trifluoromethoxy)phenyl]-8-methoxy-3,3a,4,5-tetrahydro-2h-benzo[g]indazol-2-yl}-2-hydroxyethanone | Human | 569 | |
| RIPK1 | RIPK | TKL | 4itj | A | A | n-[(1s)-1-(2-chloro-6-fluorophenyl)ethyl]-5-cyano-1-methyl-1h-pyrrole-2-carboxamide | Human | 575 | |
| RIPK1 | RIPK | TKL | 4itj | A | B | n-[(1s)-1-(2-chloro-6-fluorophenyl)ethyl]-5-cyano-1-methyl-1h-pyrrole-2-carboxamide | Human | 572 | |
| RIPK1 | RIPK | TKL | 4itj | B | A | n-[(1s)-1-(2-chloro-6-fluorophenyl)ethyl]-5-cyano-1-methyl-1h-pyrrole-2-carboxamide | Human | 565 | |
| RIPK1 | RIPK | TKL | 4itj | B | B | n-[(1s)-1-(2-chloro-6-fluorophenyl)ethyl]-5-cyano-1-methyl-1h-pyrrole-2-carboxamide | Human | 574 | |
| RIPK1 | RIPK | TKL | 4neu | A | A | 1-[4-(1-aminoisoquinolin-5-yl)phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)urea | Human | 576 | |
| RIPK1 | RIPK | TKL | 4neu | A | B | 1-[4-(1-aminoisoquinolin-5-yl)phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)urea | Human | 561 | |
| RIPK1 | RIPK | TKL | 4neu | B | A | 1-[4-(1-aminoisoquinolin-5-yl)phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)urea | Human | 568 | |
| RIPK1 | RIPK | TKL | 4neu | B | B | 1-[4-(1-aminoisoquinolin-5-yl)phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)urea | Human | 573 | |
| RIPK1 | RIPK | TKL | 5hx6 | A | | 5-benzyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-1,2-oxazole-3-carboxamide | Human | 6417 | |
| RIPK1 | RIPK | TKL | 5hx6 | B | | 5-benzyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-1,2-oxazole-3-carboxamide | Human | 6418 | |
| RIPK1 | RIPK | TKL | 5tx5 | A | A | gsk2982772 | Human | 8214 | |
| RIPK1 | RIPK | TKL | 5tx5 | A | B | gsk2982772 | Human | 8217 | |
| RIPK1 | RIPK | TKL | 5tx5 | B | A | gsk2982772 | Human | 8216 | |
| RIPK1 | RIPK | TKL | 5tx5 | B | B | gsk2982772 | Human | 8215 | |
| RIPK1 | RIPK | TKL | 6c3e | A | A | 2-benzyl-5-nitro-1h-benzimidazole | Human | 9750 | |
| RIPK1 | RIPK | TKL | 6c3e | A | B | 2-benzyl-5-nitro-1h-benzimidazole | Human | 9751 | |
| RIPK1 | RIPK | TKL | 6c3e | B | A | 2-benzyl-5-nitro-1h-benzimidazole | Human | 9755 | |
| RIPK1 | RIPK | TKL | 6c3e | B | B | 2-benzyl-5-nitro-1h-benzimidazole | Human | 9757 | |
| RIPK1 | RIPK | TKL | 6c4d | A | | (3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrile | Human | 9754 | |
| RIPK1 | RIPK | TKL | 6c4d | B | | (3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrile | Human | 9752 | |
| RIPK1 | RIPK | TKL | 6c4d | C | | (3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrile | Human | 9756 | |
| RIPK1 | RIPK | TKL | 6c4d | D | | (3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrile | Human | 9753 | |
| RIPK1 | RIPK | TKL | 6hho | A | | 6-[4-[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]carbonylpiperidin-1-yl]pyrimidine-4-carbonitrile | Human | 10783 | |
| RIPK1 | RIPK | TKL | 6hho | B | | 6-[4-[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]carbonylpiperidin-1-yl]pyrimidine-4-carbonitrile | Human | 10784 | |
| RIPK1 | RIPK | TKL | 6nw2 | A | A | (5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 11040 | |
| RIPK1 | RIPK | TKL | 6nw2 | A | B | (5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 11041 | |
| RIPK1 | RIPK | TKL | 6nw2 | B | A | (5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 11039 | |
| RIPK1 | RIPK | TKL | 6nw2 | B | B | (5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 11043 | |
| RIPK1 | RIPK | TKL | 6nyh | A | | (5s)-n-[(3s)-7-methoxy-1-methyl-2-oxo-2,3,4,5-tetrahydro-1h-pyrido[3,4-b]azepin-3-yl]-5-phenyl-6,7-dihydro-5h-pyrrolo[1,2-b][1,2,4]triazole-2-carboxamide | Human | 11057 | |
| RIPK1 | RIPK | TKL | 6nyh | B | | (5s)-n-[(3s)-7-methoxy-1-methyl-2-oxo-2,3,4,5-tetrahydro-1h-pyrido[3,4-b]azepin-3-yl]-5-phenyl-6,7-dihydro-5h-pyrrolo[1,2-b][1,2,4]triazole-2-carboxamide | Human | 11056 | |
| RIPK1 | RIPK | TKL | 6ocq | A | A | 1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one | Human | 11046 | |
| RIPK1 | RIPK | TKL | 6ocq | A | B | 1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one | Human | 11047 | |
| RIPK1 | RIPK | TKL | 6ocq | B | A | 1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one | Human | 11048 | |
| RIPK1 | RIPK | TKL | 6ocq | B | B | 1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-one | Human | 11045 | |
| RIPK1 | RIPK | TKL | 6r5f | A | | [(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanone | Human | 11038 | |
| RIPK1 | RIPK | TKL | 6r5f | B | | [(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanone | Human | 11044 | |
| RIPK1 | RIPK | TKL | 6r5f | C | | [(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanone | Human | 11042 | |
| RIPK1 | RIPK | TKL | 6r5f | D | | [(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanone | Human | 11037 | |
| RIPK1 | RIPK | TKL | 6rln | A | | ~{n}-[(3~{s})-7,9-bis(fluoranyl)-2-oxidanylidene-1,3,4,5-tetrahydro-1-benzazepin-3-yl]-3-(phenylmethyl)-1~{h}-1,2,4-triazole-5-carboxamide | Human | 11383 | |
| RIPK1 | RIPK | TKL | 6rln | B | | ~{n}-[(3~{s})-7,9-bis(fluoranyl)-2-oxidanylidene-1,3,4,5-tetrahydro-1-benzazepin-3-yl]-3-(phenylmethyl)-1~{h}-1,2,4-triazole-5-carboxamide | Human | 11382 | |
| RIPK1 | RIPK | TKL | 7fcz | A | | n-[(3s)-7-(2-cyclopropylethynyl)-5-methyl-4-oxidanylidene-2,3-dihydro-1,5-benzoxazepin-3-yl]-5-(phenylmethyl)-4h-1,2,4-triazole-3-carboxamide | Human | 14071 | |
| RIPK1 | RIPK | TKL | 7fd0 | A | | n-[(3s)-5-methyl-7-[2-(oxan-4-yl)ethynyl]-4-oxidanylidene-2,3-dihydro-1,5-benzoxazepin-3-yl]-5-(phenylmethyl)-4h-1,2,4-triazole-3-carboxamide | Human | 14070 | |
| RIPK1 | RIPK | TKL | 7xmk | A | | 5-[2-(cyclopropylcarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-7-yl]-n-[(1s)-1-(3-fluorophenyl)ethyl]-1-methyl-indole-3-carboxamide | Human | 14716 | |
| RIPK1 | RIPK | TKL | 7ydx | A | A | 1-methyl-5-[2-(2-methylpropanoylamino)-[1,2,4]triazolo[1,5-a]pyridin-7-yl]-n-[(1s)-1-phenylethyl]indole-3-carboxamide | Human | 14711 | |
| RIPK1 | RIPK | TKL | 7ydx | A | B | 1-methyl-5-[2-(2-methylpropanoylamino)-[1,2,4]triazolo[1,5-a]pyridin-7-yl]-n-[(1s)-1-phenylethyl]indole-3-carboxamide | Human | 14710 | |
| RIPK1 | RIPK | TKL | 8i2n | A | | ~{n}-methyl-1-[4-[[[1-methyl-5-(phenylmethyl)pyrazol-3-yl]carbonylamino]methyl]phenyl]benzimidazole-5-carboxamide | Human | 15186 | |
| RIPK2 | RIPK | TKL | 4c8b | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 1254 | |
| RIPK2 | RIPK | TKL | 4c8b | B | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 1253 | |
| RIPK2 | RIPK | TKL | 5ar2 | A | A | - | Human | 6183 | |
| RIPK2 | RIPK | TKL | 5ar2 | A | B | - | Human | 6173 | |
| RIPK2 | RIPK | TKL | 5ar2 | B | A | - | Human | 6185 | |
| RIPK2 | RIPK | TKL | 5ar2 | B | B | - | Human | 6181 | |
| RIPK2 | RIPK | TKL | 5ar3 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 6184 | |
| RIPK2 | RIPK | TKL | 5ar3 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 6186 | |
| RIPK2 | RIPK | TKL | 5ar3 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 6177 | |
| RIPK2 | RIPK | TKL | 5ar3 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 6190 | |
| RIPK2 | RIPK | TKL | 5ar4 | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 6180 | |
| RIPK2 | RIPK | TKL | 5ar4 | B | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 6187 | |
| RIPK2 | RIPK | TKL | 5ar5 | A | A | 2-(2-(4-chlorophenyl)-1h-imidazol-5-yl)-n,1-bis(2-methoxyethyl)-1h-benzo[d]imidazole-5-carboxamide | Human | 6189 | |
| RIPK2 | RIPK | TKL | 5ar5 | A | B | 2-(2-(4-chlorophenyl)-1h-imidazol-5-yl)-n,1-bis(2-methoxyethyl)-1h-benzo[d]imidazole-5-carboxamide | Human | 6175 | |
| RIPK2 | RIPK | TKL | 5ar5 | B | A | 2-(2-(4-chlorophenyl)-1h-imidazol-5-yl)-n,1-bis(2-methoxyethyl)-1h-benzo[d]imidazole-5-carboxamide | Human | 6171 | |
| RIPK2 | RIPK | TKL | 5ar5 | B | B | 2-(2-(4-chlorophenyl)-1h-imidazol-5-yl)-n,1-bis(2-methoxyethyl)-1h-benzo[d]imidazole-5-carboxamide | Human | 6172 | |
| RIPK2 | RIPK | TKL | 5ar7 | A | A | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-pyridin-4-yloxyphenyl)urea | Human | 6174 | |
| RIPK2 | RIPK | TKL | 5ar7 | A | B | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-pyridin-4-yloxyphenyl)urea | Human | 6182 | |
| RIPK2 | RIPK | TKL | 5ar7 | B | A | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-pyridin-4-yloxyphenyl)urea | Human | 6178 | |
| RIPK2 | RIPK | TKL | 5ar7 | B | B | 1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-pyridin-4-yloxyphenyl)urea | Human | 6188 | |
| RIPK2 | RIPK | TKL | 5ar8 | A | | 2,6-bis(fluoranyl)-n-[3-[5-[2-[(3-methylsulfonylphenyl)amino]pyrimidin-4-yl]-2-morpholin-4-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamide | Human | 6176 | |
| RIPK2 | RIPK | TKL | 5ar8 | B | | 2,6-bis(fluoranyl)-n-[3-[5-[2-[(3-methylsulfonylphenyl)amino]pyrimidin-4-yl]-2-morpholin-4-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamide | Human | 6179 | |
| RIPK2 | RIPK | TKL | 5j79 | A | A | 4-methyl-3-{[6-(methylsulfonyl)quinolin-4-yl]amino}phenol | Human | 6634 | |
| RIPK2 | RIPK | TKL | 5j79 | A | B | 4-methyl-3-{[6-(methylsulfonyl)quinolin-4-yl]amino}phenol | Human | 6636 | |
| RIPK2 | RIPK | TKL | 5j79 | B | A | 4-methyl-3-{[6-(methylsulfonyl)quinolin-4-yl]amino}phenol | Human | 6633 | |
| RIPK2 | RIPK | TKL | 5j79 | B | B | 4-methyl-3-{[6-(methylsulfonyl)quinolin-4-yl]amino}phenol | Human | 6635 | |
| RIPK2 | RIPK | TKL | 5j7b | A | | 6-(tert-butylsulfonyl)-n-(5-fluoro-2h-indazol-3-yl)quinolin-4-amine | Human | 6637 | |
| RIPK2 | RIPK | TKL | 5j7b | B | | 6-(tert-butylsulfonyl)-n-(5-fluoro-2h-indazol-3-yl)quinolin-4-amine | Human | 6632 | |
| RIPK2 | RIPK | TKL | 5ng0 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 8054 | |
| RIPK2 | RIPK | TKL | 5ng0 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 8051 | |
| RIPK2 | RIPK | TKL | 5ng0 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 8057 | |
| RIPK2 | RIPK | TKL | 5ng0 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 8055 | |
| RIPK2 | RIPK | TKL | 5ng2 | A | A | staurosporine | Human | 8050 | |
| RIPK2 | RIPK | TKL | 5ng2 | A | B | staurosporine | Human | 8056 | |
| RIPK2 | RIPK | TKL | 5ng2 | B | A | staurosporine | Human | 8053 | |
| RIPK2 | RIPK | TKL | 5ng2 | B | B | staurosporine | Human | 8052 | |
| RIPK2 | RIPK | TKL | 5ng3 | A | | - | Human | 8169 | |
| RIPK2 | RIPK | TKL | 5ng3 | B | | - | Human | 8170 | |
| RIPK2 | RIPK | TKL | 5ng3 | C | | - | Human | 8171 | |
| RIPK2 | RIPK | TKL | 5ng3 | D | | - | Human | 8172 | |
| RIPK2 | RIPK | TKL | 5w5j | A | | n-(2-chlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | Human | 8593 | |
| RIPK2 | RIPK | TKL | 5w5j | B | | n-(2-chlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamide | Human | 8591 | |
| RIPK2 | RIPK | TKL | 5w5o | A | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8579 | |
| RIPK2 | RIPK | TKL | 5w5o | B | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8587 | |
| RIPK2 | RIPK | TKL | 5w5o | C | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8577 | |
| RIPK2 | RIPK | TKL | 5w5o | D | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8576 | |
| RIPK2 | RIPK | TKL | 5w5o | E | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8592 | |
| RIPK2 | RIPK | TKL | 5w5o | F | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8582 | |
| RIPK2 | RIPK | TKL | 5w5o | G | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8580 | |
| RIPK2 | RIPK | TKL | 5w5o | H | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8588 | |
| RIPK2 | RIPK | TKL | 5w5o | I | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8590 | |
| RIPK2 | RIPK | TKL | 5w5o | J | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8586 | |
| RIPK2 | RIPK | TKL | 5w5o | K | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8583 | |
| RIPK2 | RIPK | TKL | 5w5o | L | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8585 | |
| RIPK2 | RIPK | TKL | 5w5o | M | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8589 | |
| RIPK2 | RIPK | TKL | 5w5o | N | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8578 | |
| RIPK2 | RIPK | TKL | 5w5o | O | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8584 | |
| RIPK2 | RIPK | TKL | 5w5o | P | | 4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amine | Human | 8581 | |
| RIPK2 | RIPK | TKL | 6es0 | A | | 2-[2-fluoranyl-4-[[2-fluoranyl-4-[2-(methylcarbamoyl)pyridin-4-yl]oxy-phenyl]carbamoylamino]phenyl]sulfanylethanoic acid | Human | 9574 | |
| RIPK2 | RIPK | TKL | 6es0 | B | | 2-[2-fluoranyl-4-[[2-fluoranyl-4-[2-(methylcarbamoyl)pyridin-4-yl]oxy-phenyl]carbamoylamino]phenyl]sulfanylethanoic acid | Human | 9573 | |
| RIPK2 | RIPK | TKL | 6fu5 | A | | ~{n}-[5-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methoxy-phenyl]propane-1-sulfonamide | Human | 9852 | |
| RIPK2 | RIPK | TKL | 6fu5 | B | | ~{n}-[5-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methoxy-phenyl]propane-1-sulfonamide | Human | 9853 | |
| RIPK2 | RIPK | TKL | 6hmx | A | | 6-~{tert}-butylsulfonyl-~{n}-(3,4-dimethyl-1~{h}-pyrazol-5-yl)-7-methoxy-quinolin-4-amine | Human | 10676 | |
| RIPK2 | RIPK | TKL | 6hmx | B | | 6-~{tert}-butylsulfonyl-~{n}-(3,4-dimethyl-1~{h}-pyrazol-5-yl)-7-methoxy-quinolin-4-amine | Human | 10675 | |
| RIPK2 | RIPK | TKL | 6rn8 | A | | 2-[4-(1,3-benzothiazol-5-ylamino)-6-~{tert}-butylsulfonyl-quinazolin-7-yl]oxyethyl dihydrogen phosphate | Human | 11434 | |
| RIPK2 | RIPK | TKL | 6rn8 | B | | 2-[4-(1,3-benzothiazol-5-ylamino)-6-~{tert}-butylsulfonyl-quinazolin-7-yl]oxyethyl dihydrogen phosphate | Human | 11431 | |
| RIPK2 | RIPK | TKL | 6rna | A | | 2-[4-(1,3-benzothiazol-5-ylamino)-6-~{tert}-butylsulfonyl-quinazolin-7-yl]oxyethanol | Human | 11433 | |
| RIPK2 | RIPK | TKL | 6rna | B | | 2-[4-(1,3-benzothiazol-5-ylamino)-6-~{tert}-butylsulfonyl-quinazolin-7-yl]oxyethanol | Human | 11432 | |
| RIPK2 | RIPK | TKL | 6s1f | A | | ~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamide | Human | 11733 | |
| RIPK2 | RIPK | TKL | 6s1f | B | | ~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamide | Human | 11730 | |
| RIPK2 | RIPK | TKL | 6s1f | C | | ~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamide | Human | 11731 | |
| RIPK2 | RIPK | TKL | 6s1f | D | | ~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamide | Human | 11732 | |
| RIPK2 | RIPK | TKL | 6sze | A | A | 5-amino-1-phenylpyrazole-4-carboxamide | Human | 11759 | |
| RIPK2 | RIPK | TKL | 6sze | A | B | 5-amino-1-phenylpyrazole-4-carboxamide | Human | 11761 | |
| RIPK2 | RIPK | TKL | 6sze | B | A | 5-amino-1-phenylpyrazole-4-carboxamide | Human | 11760 | |
| RIPK2 | RIPK | TKL | 6sze | B | B | 5-amino-1-phenylpyrazole-4-carboxamide | Human | 11758 | |
| RIPK2 | RIPK | TKL | 6szj | A | A | 5-amino-1-~{tert}-butyl-3-(3-methoxyphenyl)pyrazole-4-carboxamide | Human | 11848 | |
| RIPK2 | RIPK | TKL | 6szj | A | B | 5-amino-1-~{tert}-butyl-3-(3-methoxyphenyl)pyrazole-4-carboxamide | Human | 11853 | |
| RIPK2 | RIPK | TKL | 6szj | B | A | 5-amino-1-~{tert}-butyl-3-(3-methoxyphenyl)pyrazole-4-carboxamide | Human | 11846 | |
| RIPK2 | RIPK | TKL | 6szj | B | B | 5-amino-1-~{tert}-butyl-3-(3-methoxyphenyl)pyrazole-4-carboxamide | Human | 11851 | |
| RIPK2 | RIPK | TKL | 6ul8 | A | A | (5s,6s,8r)-2-(1,3-benzothiazol-5-yl)-6-hydroxy-4,5,6,7,8,9-hexahydro-5,8-methanopyrazolo[1,5-a][1,3]diazocine-3-carboxamide | Human | 11847 | |
| RIPK2 | RIPK | TKL | 6ul8 | A | B | (5s,6s,8r)-2-(1,3-benzothiazol-5-yl)-6-hydroxy-4,5,6,7,8,9-hexahydro-5,8-methanopyrazolo[1,5-a][1,3]diazocine-3-carboxamide | Human | 11849 | |
| RIPK2 | RIPK | TKL | 6ul8 | B | A | (5s,6s,8r)-2-(1,3-benzothiazol-5-yl)-6-hydroxy-4,5,6,7,8,9-hexahydro-5,8-methanopyrazolo[1,5-a][1,3]diazocine-3-carboxamide | Human | 11852 | |
| RIPK2 | RIPK | TKL | 6ul8 | B | B | (5s,6s,8r)-2-(1,3-benzothiazol-5-yl)-6-hydroxy-4,5,6,7,8,9-hexahydro-5,8-methanopyrazolo[1,5-a][1,3]diazocine-3-carboxamide | Human | 11850 | |
| RIPK2 | RIPK | TKL | 8aza | B | | - | Human | 14473 | |
| Ripk3 (RIPK3) | RIPK | TKL | 4m66 | A | A | - | Mouse | 5825 | |
| Ripk3 (RIPK3) | RIPK | TKL | 4m66 | A | B | - | Mouse | 5826 | |
| Ripk3 (RIPK3) | RIPK | TKL | 4m66 | B | A | - | Mouse | 5821 | |
| Ripk3 (RIPK3) | RIPK | TKL | 4m66 | B | B | - | Mouse | 5823 | |
| Ripk3 (RIPK3) | RIPK | TKL | 4m69 | A | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 5824 | |
| Ripk3 (RIPK3) | RIPK | TKL | 4m69 | A | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 5822 | |
| Ripk3 (RIPK3) | RIPK | TKL | 6oko | A | A | 1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamide | Mouse | 11438 | |
| Ripk3 (RIPK3) | RIPK | TKL | 6oko | A | B | 1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamide | Mouse | 11439 | |
| Ripk3 (RIPK3) | RIPK | TKL | 6oko | B | A | 1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamide | Mouse | 11440 | |
| Ripk3 (RIPK3) | RIPK | TKL | 6oko | B | B | 1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamide | Mouse | 11441 | |
| RIPK3 | RIPK | TKL | 7mon | B | | n-[4-({2-[(cyclopropanecarbonyl)amino]pyridin-4-yl}oxy)-3-fluorophenyl]-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 13979 | |
| RIPK3 | RIPK | TKL | 7mx3 | A | | 3-(1,3-benzothiazol-5-yl)-7-(1,3-dimethyl-1h-pyrazol-5-yl)thieno[3,2-c]pyridin-4-amine | Human | 13995 | |
| Ripk4 (ANKRD3) | RIPK | TKL | 5wni | A | | adenosine-5'-triphosphate | Mouse | 9889 | |
| Ripk4 (ANKRD3) | RIPK | TKL | 5wnj | A | | lestaurtinib | Mouse | 9893 | |
| Ripk4 (ANKRD3) | RIPK | TKL | 5wnk | A | | 3,3'-(2,4-diaminopteridine-6,7-diyl)diphenol | Mouse | 9892 | |
| Ripk4 (ANKRD3) | RIPK | TKL | 5wnl | A | | staurosporine | Mouse | 9891 | |
| Ripk4 (ANKRD3) | RIPK | TKL | 5wnm | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Mouse | 9890 | |
| RNASEL (RNAseL) | Other-Unique | Other | 4oau | C | | adenosine-5'-diphosphate | Human | 468 | |
| RNASEL (RNAseL) | Other-Unique | Other | 4oav | B | | phosphomethylphosphonic acid adenylate ester | Human | 467 | |
| RNASEL (RNAseL) | Other-Unique | Other | 4oav | D | | phosphomethylphosphonic acid adenylate ester | Human | 466 | |
| ROCK1 | DMPK | AGC | 2esm | A | | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 2726 | |
| ROCK1 | DMPK | AGC | 2esm | B | | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 2714 | |
| ROCK1 | DMPK | AGC | 2etk | A | | 1-(1-hydroxy-5-isoquinolinesulfonyl)homopiperazine | Human | 2707 | |
| ROCK1 | DMPK | AGC | 2etk | B | | 1-(1-hydroxy-5-isoquinolinesulfonyl)homopiperazine | Human | 2723 | |
| ROCK1 | DMPK | AGC | 2etr | A | | (r)-trans-4-(1-aminoethyl)-n-(4-pyridyl) cyclohexanecarboxamide | Human | 2700 | |
| ROCK1 | DMPK | AGC | 2etr | B | | (r)-trans-4-(1-aminoethyl)-n-(4-pyridyl) cyclohexanecarboxamide | Human | 2704 | |
| ROCK1 | DMPK | AGC | 2v55 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2694 | |
| ROCK1 | DMPK | AGC | 2v55 | C | | phosphoaminophosphonic acid-adenylate ester | Human | 2711 | |
| ROCK1 | DMPK | AGC | 3d9v | A | | (s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazine | Human | 2696 | |
| ROCK1 | DMPK | AGC | 3d9v | B | | (s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazine | Human | 2701 | |
| ROCK1 | DMPK | AGC | 3ncz | A | | cis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamide | Human | 2699 | |
| ROCK1 | DMPK | AGC | 3ncz | B | | cis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamide | Human | 2720 | |
| ROCK1 | DMPK | AGC | 3ncz | C | | cis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamide | Human | 2719 | |
| ROCK1 | DMPK | AGC | 3ncz | D | | cis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamide | Human | 2724 | |
| ROCK1 | DMPK | AGC | 3ndm | A | | - | Human | 2695 | |
| ROCK1 | DMPK | AGC | 3ndm | B | | (3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamide | Human | 2698 | |
| ROCK1 | DMPK | AGC | 3ndm | C | | (3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamide | Human | 2722 | |
| ROCK1 | DMPK | AGC | 3ndm | D | | (3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamide | Human | 2705 | |
| ROCK1 | DMPK | AGC | 3tv7 | A | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2697 | |
| ROCK1 | DMPK | AGC | 3tv7 | B | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2703 | |
| ROCK1 | DMPK | AGC | 3tv7 | C | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2717 | |
| ROCK1 | DMPK | AGC | 3tv7 | D | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2725 | |
| ROCK1 | DMPK | AGC | 3twj | A | | 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2710 | |
| ROCK1 | DMPK | AGC | 3twj | B | | - | Human | 2718 | |
| ROCK1 | DMPK | AGC | 3twj | C | | 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2689 | |
| ROCK1 | DMPK | AGC | 3twj | D | | - | Human | 2690 | |
| ROCK1 | DMPK | AGC | 3v8s | A | | 1-(1h-indazol-5-yl)-3-(2-phenylethyl)urea | Human | 2716 | |
| ROCK1 | DMPK | AGC | 3v8s | B | | 1-(1h-indazol-5-yl)-3-(2-phenylethyl)urea | Human | 2709 | |
| ROCK1 | DMPK | AGC | 3v8s | C | | 1-(1h-indazol-5-yl)-3-(2-phenylethyl)urea | Human | 2702 | |
| ROCK1 | DMPK | AGC | 3v8s | D | | 1-(1h-indazol-5-yl)-3-(2-phenylethyl)urea | Human | 2692 | |
| ROCK1 | DMPK | AGC | 4w7p | A | | n~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamine | Human | 2721 | |
| ROCK1 | DMPK | AGC | 4w7p | B | | n~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamine | Human | 2708 | |
| ROCK1 | DMPK | AGC | 4w7p | C | | n~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamine | Human | 2688 | |
| ROCK1 | DMPK | AGC | 4w7p | D | | n~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamine | Human | 2712 | |
| ROCK1 | DMPK | AGC | 4yvc | A | | 2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamide | Human | 2715 | |
| ROCK1 | DMPK | AGC | 4yvc | B | | 2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamide | Human | 2727 | |
| ROCK1 | DMPK | AGC | 4yve | A | | 2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 2693 | |
| ROCK1 | DMPK | AGC | 4yve | B | | 2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 2706 | |
| ROCK1 | DMPK | AGC | 5bml | A | | n-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-{3-[(methylsulfonyl)amino]phenyl}acetamide | Human | 2713 | |
| ROCK1 | DMPK | AGC | 5bml | B | | n-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-{3-[(methylsulfonyl)amino]phenyl}acetamide | Human | 2691 | |
| ROCK1 | DMPK | AGC | 5hvu | A | | 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 7414 | |
| ROCK1 | DMPK | AGC | 5hvu | B | | 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 7415 | |
| ROCK1 | DMPK | AGC | 5kks | A | | 2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8183 | |
| ROCK1 | DMPK | AGC | 5kks | B | | 2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8181 | |
| ROCK1 | DMPK | AGC | 5kkt | A | | 2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8182 | |
| ROCK1 | DMPK | AGC | 5kkt | B | | 2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8184 | |
| ROCK1 | DMPK | AGC | 5uzj | A | | n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide | Human | 9706 | |
| ROCK1 | DMPK | AGC | 5uzj | B | | n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide | Human | 9707 | |
| ROCK1 | DMPK | AGC | 5wne | A | | 3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamide | Human | 10446 | |
| ROCK1 | DMPK | AGC | 5wne | B | | 3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamide | Human | 10453 | |
| ROCK1 | DMPK | AGC | 5wne | C | | 3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamide | Human | 10462 | |
| ROCK1 | DMPK | AGC | 5wne | D | | 3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamide | Human | 10445 | |
| ROCK1 | DMPK | AGC | 5wnf | A | A | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10447 | |
| ROCK1 | DMPK | AGC | 5wnf | A | B | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10444 | |
| ROCK1 | DMPK | AGC | 5wnf | B | A | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10463 | |
| ROCK1 | DMPK | AGC | 5wnf | B | B | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10450 | |
| ROCK1 | DMPK | AGC | 5wnf | C | A | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10455 | |
| ROCK1 | DMPK | AGC | 5wnf | C | B | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10460 | |
| ROCK1 | DMPK | AGC | 5wnf | D | A | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10451 | |
| ROCK1 | DMPK | AGC | 5wnf | D | B | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10452 | |
| ROCK1 | DMPK | AGC | 5wng | A | | (2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamide | Human | 10459 | |
| ROCK1 | DMPK | AGC | 5wng | B | | (2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamide | Human | 10461 | |
| ROCK1 | DMPK | AGC | 5wng | C | | (2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamide | Human | 10458 | |
| ROCK1 | DMPK | AGC | 5wng | D | | (2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamide | Human | 10457 | |
| ROCK1 | DMPK | AGC | 5wnh | A | | (2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide | Human | 10448 | |
| ROCK1 | DMPK | AGC | 5wnh | B | | (2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide | Human | 10449 | |
| ROCK1 | DMPK | AGC | 5wnh | C | | (2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide | Human | 10456 | |
| ROCK1 | DMPK | AGC | 5wnh | D | | (2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide | Human | 10454 | |
| ROCK1 | DMPK | AGC | 6e9w | A | | n-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamide | Human | 10691 | |
| ROCK1 | DMPK | AGC | 6e9w | B | | n-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamide | Human | 10690 | |
| ROCK1 | DMPK | AGC | 7jou | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12768 | |
| ROCK1 | DMPK | AGC | 7s25 | A | A | 2-[3-(methoxymethyl)phenyl]-n-[4-(1h-pyrazol-4-yl)phenyl]acetamide | Human | 14435 | |
| ROCK1 | DMPK | AGC | 7s25 | A | B | 2-[3-(methoxymethyl)phenyl]-n-[4-(1h-pyrazol-4-yl)phenyl]acetamide | Human | 14436 | |
| ROCK1 | DMPK | AGC | 7s26 | A | | 2-[methyl(phenyl)amino]-1-[4-(1h-pyrrolo[2,3-b]pyridin-3-yl)-3,6-dihydropyridin-1(2h)-yl]ethan-1-one | Human | 14437 | |
| ROCK1 | DMPK | AGC | 8zh5 | A | | - | Human | 15364 | |
| ROCK2 | DMPK | AGC | 4l6q | A | | 6-[4-(aminomethyl)-2-fluorophenoxy]-2,1-benzoxaborol-1(3h)-ol | Human | 1811 | |
| ROCK2 | DMPK | AGC | 4l6q | B | | 6-[4-(aminomethyl)-2-fluorophenoxy]-2,1-benzoxaborol-1(3h)-ol | Human | 1810 | |
| ROCK2 | DMPK | AGC | 4wot | A | | methyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoate | Human | 6827 | |
| ROCK2 | DMPK | AGC | 4wot | B | | methyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoate | Human | 6829 | |
| ROCK2 | DMPK | AGC | 4wot | C | | methyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoate | Human | 6828 | |
| ROCK2 | DMPK | AGC | 4wot | D | | methyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoate | Human | 6830 | |
| ROCK2 | DMPK | AGC | 5u7q | A | | - | Human | 7988 | |
| ROCK2 | DMPK | AGC | 5u7q | B | | - | Human | 7990 | |
| ROCK2 | DMPK | AGC | 5u7q | C | | - | Human | 7987 | |
| ROCK2 | DMPK | AGC | 5u7q | D | | - | Human | 7986 | |
| ROCK2 | DMPK | AGC | 5u7r | A | | (1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-one | Human | 7989 | |
| ROCK2 | DMPK | AGC | 5u7r | B | | (1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-one | Human | 7984 | |
| ROCK2 | DMPK | AGC | 5u7r | C | | (1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-one | Human | 7983 | |
| ROCK2 | DMPK | AGC | 5u7r | D | | (1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-one | Human | 7985 | |
| ROCK2 | DMPK | AGC | 6ed6 | A | | n-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamide | Human | 10689 | |
| ROCK2 | DMPK | AGC | 6ed6 | B | | n-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamide | Human | 10688 | |
| ROCK2 | DMPK | AGC | 6p5m | A | A | 6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11920 | |
| ROCK2 | DMPK | AGC | 6p5m | A | B | 6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11915 | |
| ROCK2 | DMPK | AGC | 6p5m | B | A | 6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11921 | |
| ROCK2 | DMPK | AGC | 6p5m | B | B | 6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11924 | |
| ROCK2 | DMPK | AGC | 6p5m | C | A | - | Human | 11917 | |
| ROCK2 | DMPK | AGC | 6p5m | C | B | - | Human | 11916 | |
| ROCK2 | DMPK | AGC | 6p5m | D | A | - | Human | 11925 | |
| ROCK2 | DMPK | AGC | 6p5m | D | B | - | Human | 11922 | |
| ROCK2 | DMPK | AGC | 6p5p | A | | 2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11914 | |
| ROCK2 | DMPK | AGC | 6p5p | B | | 2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11923 | |
| ROCK2 | DMPK | AGC | 6p5p | C | | 2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11919 | |
| ROCK2 | DMPK | AGC | 6p5p | D | | 2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11918 | |
| ROCK2 | DMPK | AGC | 7jnt | A | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12744 | |
| ROCK2 | DMPK | AGC | 7jnt | A | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12754 | |
| ROCK2 | DMPK | AGC | 7jnt | B | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12756 | |
| ROCK2 | DMPK | AGC | 7jnt | B | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12766 | |
| ROCK2 | DMPK | AGC | 7jnt | C | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12752 | |
| ROCK2 | DMPK | AGC | 7jnt | C | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12745 | |
| ROCK2 | DMPK | AGC | 7jnt | D | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12755 | |
| ROCK2 | DMPK | AGC | 7jnt | D | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12750 | |
| ROCK2 | DMPK | AGC | 7jnt | E | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12746 | |
| ROCK2 | DMPK | AGC | 7jnt | E | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12747 | |
| ROCK2 | DMPK | AGC | 7jnt | F | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12749 | |
| ROCK2 | DMPK | AGC | 7jnt | F | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12758 | |
| ROCK2 | DMPK | AGC | 7jnt | G | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12761 | |
| ROCK2 | DMPK | AGC | 7jnt | G | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12767 | |
| ROCK2 | DMPK | AGC | 7jnt | H | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12760 | |
| ROCK2 | DMPK | AGC | 7jnt | H | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12753 | |
| ROCK2 | DMPK | AGC | 7jov | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12757 | |
| ROCK2 | DMPK | AGC | 7jov | B | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12765 | |
| ROCK2 | DMPK | AGC | 7jov | C | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12748 | |
| ROCK2 | DMPK | AGC | 7jov | D | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12764 | |
| ROCK2 | DMPK | AGC | 7jov | E | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12762 | |
| ROCK2 | DMPK | AGC | 7jov | F | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12759 | |
| ROCK2 | DMPK | AGC | 7jov | G | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12763 | |
| ROCK2 | DMPK | AGC | 7jov | H | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12751 | |
| ROCK2 | DMPK | AGC | 7p6n | A | | ~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-yl-piperidine-1-carboxamide | Human | 14314 | |
| ROCK2 | DMPK | AGC | 8gds | A | | 4-{4-[2-(2,3-dihydro-1h-indol-1-yl)-2-oxoethyl]phenyl}phthalazin-1(2h)-one | Human | 14736 | |
| ROR1 | Ror | TK | 6tu9 | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 11944 | |
| ROR1 | Ror | TK | 6tu9 | B | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 11945 | |
| ROR2 | Ror | TK | 3zzw | A | A | - | Human | 410 | |
| ROR2 | Ror | TK | 3zzw | A | B | - | Human | 412 | |
| ROR2 | Ror | TK | 3zzw | B | A | - | Human | 415 | |
| ROR2 | Ror | TK | 3zzw | B | B | - | Human | 411 | |
| ROR2 | Ror | TK | 4gt4 | A | A | - | Human | 414 | |
| ROR2 | Ror | TK | 4gt4 | A | B | - | Human | 409 | |
| ROR2 | Ror | TK | 4gt4 | B | A | - | Human | 413 | |
| ROR2 | Ror | TK | 4gt4 | B | B | - | Human | 408 | |
| ROS1 (ROS) | Sev | TK | 3zbf | A | | 3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amine | Human | 197 | |
| ROS1 (ROS) | Sev | TK | 4uxl | A | | (10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrile | Human | 198 | |
| ROS1 (ROS) | Sev | TK | 7z5w | A | | ~{n}-[6-methyl-2-[(2~{s})-2-[3-(3-methylpyrazin-2-yl)-1,2-oxazol-5-yl]pyrrolidin-1-yl]pyrimidin-4-yl]-1,3-thiazol-2-amine | Human | 14326 | |
| ROS1 (ROS) | Sev | TK | 7z5x | A | | (2r)-2-[5-(6-amino-5-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diol | Human | 14325 | |
| RPS6KA1 (RSK3) | RSK | AGC | 2z7q | A | | phosphomethylphosphonic acid adenylate ester | Human | 2778 | |
| RPS6KA1 (RSK3) | RSK | AGC | 2z7r | A | | staurosporine | Human | 2777 | |
| RPS6KA1 (RSK3) | RSK | AGC | 2z7s | A | | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 2776 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | A | A | - | Human | 6862 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | A | B | - | Human | 6859 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | B | A | - | Human | 6860 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | B | B | - | Human | 6861 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | A | A | - | Human | 5568 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | A | B | - | Human | 5569 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | B | A | - | Human | 5573 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | B | B | - | Human | 5574 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | A | A | - | Human | 5572 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | A | B | - | Human | 5570 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | D | A | - | Human | 5571 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | D | B | - | Human | 5575 | |
| RPS6KA2 (RSK1) | RSK | AGC | 8xov | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15216 | |
| RPS6KA2-b (RSK1-b) | RSKb | CAMK | 8wf4 | A | | - | Human | 15082 | |
| Rps6ka3 (RSK2) | RSK | AGC | 3g51 | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5695 | |
| Rps6ka3 (RSK2) | RSK | AGC | 3ubd | A | A | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4h-chromen-3-yl 3,4-di-o-acetyl-6-deoxy-alpha-l-mannopyranoside | Mouse | 5693 | |
| Rps6ka3 (RSK2) | RSK | AGC | 3ubd | A | B | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4h-chromen-3-yl 3,4-di-o-acetyl-6-deoxy-alpha-l-mannopyranoside | Mouse | 5691 | |
| Rps6ka3 (RSK2) | RSK | AGC | 4el9 | A | | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Mouse | 5692 | |
| Rps6ka3 (RSK2) | RSK | AGC | 4gue | A | A | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Mouse | 5696 | |
| Rps6ka3 (RSK2) | RSK | AGC | 4gue | A | B | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Mouse | 5694 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nus | A | A | 2,6-difluoro-4-{4-[4-(4-methylpiperazin-1-yl)phenyl]pyridin-3-yl}phenol | Human | 133 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nus | A | B | 2,6-difluoro-4-{4-[4-(4-methylpiperazin-1-yl)phenyl]pyridin-3-yl}phenol | Human | 131 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw5 | A | A | 7-(2-fluoro-6-methoxyphenyl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | 134 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw5 | A | B | 7-(2-fluoro-6-methoxyphenyl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | 135 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw6 | A | A | 7-(1h-benzimidazol-7-yl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | 132 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw6 | A | B | 7-(1h-benzimidazol-7-yl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | 136 | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9k | A | | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 5988 | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9k | B | | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 5987 | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9l | A | A | 4,4'-(1h-pyrazole-3,4-diyl)diphenol | Human | 5986 | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9l | A | B | 4,4'-(1h-pyrazole-3,4-diyl)diphenol | Human | 5989 | |
| RPS6KA3 (RSK2) | RSK | AGC | 7opo | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14079 | |
| RPS6KA3 (RSK2) | RSK | AGC | 8eq5 | A | A | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Human | 14713 | |
| RPS6KA3 (RSK2) | RSK | AGC | 8eq5 | A | B | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Human | 14714 | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr7 | A | A | - | Mouse | 5759 | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr7 | A | B | - | Mouse | 5757 | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr8 | A | A | - | Mouse | 5760 | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr8 | A | B | - | Mouse | 5755 | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 4m8t | A | | (2e)-2-cyano-3-[3-(1h-pyrazol-4-yl)phenyl]prop-2-enamide | Mouse | 5756 | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 4mao | A | | (2z)-2-(1h-1,2,4-triazol-1-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]prop-2-enenitrile | Mouse | 5758 | |
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 5o1s | A | | dimethyl fumarate | Mouse | 9976 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4d9t | A | | methyl (2s)-3-{4-amino-7-[(1e)-3-hydroxyprop-1-en-1-yl]-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl}-2-cyanopropanoate | Human | 1493 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4d9u | A | | tert-butyl (2s)-3-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl]-2-cyanopropanoate | Human | 1499 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg6 | A | | (2s)-2-cyano-3-(1h-indazol-5-yl)propanamide | Human | 1495 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg7 | A | A | (2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamide | Human | 1496 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg7 | A | B | (2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamide | Human | 1494 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg8 | A | A | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | 1497 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg8 | A | B | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | 1498 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 8xey | A | | - | Human | 15207 | |
| RPS6KA5 (MSK1) | RSK | AGC | 1vzo | A | A | - | Human | 108 | |
| RPS6KA5 (MSK1) | RSK | AGC | 1vzo | A | B | - | Human | 107 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn5 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 4603 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn5 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 4600 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn6 | A | | - | Human | 4602 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn6 | B | | - | Human | 4601 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up4 | A | A | (5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | 14277 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up4 | A | B | (5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | 14279 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up5 | A | A | (2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrile | Human | 14280 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up5 | A | B | (2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrile | Human | 14278 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up6 | A | A | (e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound form | Human | 14353 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up6 | A | B | (e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound form | Human | 14354 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up7 | A | A | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | 14318 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up7 | A | B | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | 14317 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up8 | A | A | (5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | 14282 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up8 | A | B | (5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | 14281 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g76 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11006 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g76 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 11008 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g77 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11005 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g77 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 11009 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g78 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11010 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g78 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 11007 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a60 | A | | staurosporine | Human | 1852 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a60 | B | | staurosporine | Human | 1856 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a61 | A | | staurosporine | Human | 1846 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a62 | A | | staurosporine | Human | 1867 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3we4 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1860 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf5 | A | A | 4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | 1857 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf5 | A | B | 4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | 1845 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf6 | A | A | 4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | 1864 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf6 | A | B | 4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | 1859 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf7 | A | A | 1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamide | Human | 1854 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf7 | A | B | 1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamide | Human | 1851 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf8 | A | | 2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl 7,8,9,10-tetrahydro-6h-cyclohepta[b]quinoline-11-carboxylate | Human | 1848 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf9 | A | | (2s)-1-oxo-1-[(4-sulfamoylphenyl)amino]propan-2-yl (2s)-2-methyl-1,2,3,4-tetrahydroacridine-9-carboxylate | Human | 1866 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l3j | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1858 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l3l | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1863 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l42 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1865 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l43 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1861 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l44 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1849 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l45 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1850 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l46 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1847 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4rlo | A | | [(amino-kappan)methanethiolato](3-fluoro-9-hydroxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(1,4,7-trithionane-kappa~3~s~1~,s~4~,s~7~)ruthenium | Human | 7218 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4rlo | B | | staurosporine | Human | 7220 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4rlp | A | | [(amino-kappan)methanethiolato](3-fluoro-9-methoxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(n-methyl-1,4,7-trithiecan-9-amine-kappa~3~s~1~,s~4~,s~7~)ruthenium | Human | 7219 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 7n91 | A | | 4-{[(1s)-1-(3-fluorophenyl)-2-(methylamino)ethyl]amino}quinazoline-8-carboxamide | Human | 14284 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 7n93 | A | A | 4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamide | Human | 14285 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 7n93 | A | B | 4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamide | Human | 14283 | |
| RYK | Ryk | TK | 6tua | A | | - | Human | 11943 | |
| SGK1 | SGK | AGC | 2r5t | A | | phosphoaminophosphonic acid-adenylate ester | Human | 6849 | |
| SGK1 | SGK | AGC | 3hdm | A | | 4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 3271 | |
| SGK1 | SGK | AGC | 3hdn | A | | [4-(5-naphthalen-2-yl-1h-pyrrolo[2,3-b]pyridin-3-yl)phenyl]acetic acid | Human | 3270 | |
| SGK1 | SGK | AGC | 7pue | A | | 6-[4-[[2,3-bis(chloranyl)phenyl]sulfonylamino]phenyl]-~{n}-[(3~{r})-pyrrolidin-3-yl]-2~{h}-pyrazolo[3,4-b]pyridine-4-carboxamide | Human | 14012 | |
| SIK3 (QSK) | CAMKL | CAMK | 8oku | A | | ~{n}-ethyl-4-[5-[1-(2-hydroxyethyl)pyrazol-4-yl]benzimidazol-1-yl]-2,6-dimethoxy-benzamide | Human | 15169 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4o | A | | 2-[bis(fluoranyl)methoxy]-4-[6-(2-cyanopropan-2-yl)pyrazolo[1,5-a]pyridin-3-yl]-~{n}-[(1~{r},2~{s})-2-fluoranylcyclopropyl]-6-methoxy-benzamide | Human | 15242 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4q | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 15241 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4u | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 15240 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4v | A | | 1-(2,4-dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]urea | Human | 15243 | |
| SLK | STE20 | STE | 2j51 | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1833 | |
| SLK | STE20 | STE | 2jfl | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1838 | |
| SLK | STE20 | STE | 2jfm | A | A | - | Human | 1836 | |
| SLK | STE20 | STE | 2jfm | A | B | - | Human | 1841 | |
| SLK | STE20 | STE | 2uv2 | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 1834 | |
| SLK | STE20 | STE | 2uv2 | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 1837 | |
| SLK | STE20 | STE | 4usf | A | A | 4-[4-(6-methoxynaphthalen-2-yl)-1h-imidazol-5-yl]pyridine | Human | 1839 | |
| SLK | STE20 | STE | 4usf | A | B | 4-[4-(6-methoxynaphthalen-2-yl)-1h-imidazol-5-yl]pyridine | Human | 1832 | |
| SLK | STE20 | STE | 4usf | B | A | 4-[4-(6-methoxynaphthalen-2-yl)-1h-imidazol-5-yl]pyridine | Human | 1835 | |
| SLK | STE20 | STE | 4usf | B | B | 4-[4-(6-methoxynaphthalen-2-yl)-1h-imidazol-5-yl]pyridine | Human | 1840 | |
| SLK | STE20 | STE | 6hvd | A | A | 3-(1,3-benzothiazol-2-ylamino)-4-(2-methoxyphenyl)pyrrole-2,5-dione | Human | 10625 | |
| SLK | STE20 | STE | 6hvd | A | B | 3-(1,3-benzothiazol-2-ylamino)-4-(2-methoxyphenyl)pyrrole-2,5-dione | Human | 10624 | |
| SLK | STE20 | STE | 8bem | A | A | tivozanib | Human | 14487 | |
| SLK | STE20 | STE | 8bem | A | B | tivozanib | Human | 14486 | |
| SMG1 | PIKK | Atypical | 6l53 | A | | - | Human | 12156 | |
| SMG1 | PIKK | Atypical | 6l54 | A | | - | Human | 12155 | |
| SMG1 | PIKK | Atypical | 6syt | A | | - | Human | 11866 | |
| SMG1 | PIKK | Atypical | 6z3r | A | | phosphoaminophosphonic acid-adenylate ester | Human | 12630 | |
| SMG1 | PIKK | Atypical | 7pw4 | A | | 1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-urea | Human | 14003 | |
| SMG1 | PIKK | Atypical | 7pw5 | A | | 1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-urea | Human | 14002 | |
| SMG1 | PIKK | Atypical | 7pw6 | A | | 1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-urea | Human | 14001 | |
| SMG1 | PIKK | Atypical | 7pw7 | A | | 1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-urea | Human | 14005 | |
| SMG1 | PIKK | Atypical | 7pw8 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14004 | |
| SMG1 | PIKK | Atypical | 7pw9 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14000 | |
| SNRK | CAMKL | CAMK | 5yks | A | | - | Human | 8660 | |
| SNRK | CAMKL | CAMK | 5yks | B | | - | Human | 8661 | |
| Src (SRC) | Src | TK | 6f3f | A | | adenosine-5'-diphosphate | Mouse | 9461 | |
| Src (SRC) | Src | TK | 8xn8 | A | A | adenosine-5'-diphosphate | Mouse | 15182 | |
| Src (SRC) | Src | TK | 8xn8 | A | B | adenosine-5'-diphosphate | Mouse | 15183 | |
| SRC | Src | TK | 1fmk | A | | - | Human | 981 | |
| SRC | Src | TK | 1ksw | A | | n6-benzyl adenosine-5'-diphosphate | Human | 985 | |
| SRC | Src | TK | 1y57 | A | | 4-[(4-methylpiperazin-1-yl)methyl]-n-{3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl}benzamide | Human | 986 | |
| SRC | Src | TK | 1yi6 | A | | - | Human | 967 | |
| SRC | Src | TK | 1yi6 | B | | - | Human | 991 | |
| SRC | Src | TK | 1yoj | A | | - | Human | 984 | |
| SRC | Src | TK | 1yoj | B | | - | Human | 974 | |
| SRC | Src | TK | 1yol | A | | 1-{4-[4-amino-5-(3-methoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl]benzyl}piperidin-4-ol | Human | 968 | |
| SRC | Src | TK | 1yol | B | | 1-{4-[4-amino-5-(3-methoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl]benzyl}piperidin-4-ol | Human | 966 | |
| SRC | Src | TK | 1yom | A | | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 973 | |
| SRC | Src | TK | 1yom | B | | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 987 | |
| SRC | Src | TK | 2bdf | A | | {[(4-{[2-(4-aminocyclohexyl)-9-ethyl-9h-purin-6-yl]amino}phenyl)(hydroxy)phosphoryl]methyl}phosphonic acid | Human | 980 | |
| SRC | Src | TK | 2bdf | B | | {[(4-{[2-(4-aminocyclohexyl)-9-ethyl-9h-purin-6-yl]amino}phenyl)(hydroxy)phosphoryl]methyl}phosphonic acid | Human | 975 | |
| SRC | Src | TK | 2bdj | A | | 3-[2-(2-cyclopentyl-6-{[4-(dimethylphosphoryl)phenyl]amino}-9h-purin-9-yl)ethyl]phenol | Human | 971 | |
| SRC | Src | TK | 2h8h | A | A | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 970 | |
| SRC | Src | TK | 2h8h | A | B | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 992 | |
| SRC | Src | TK | 2src | A | | phosphoaminophosphonic acid-adenylate ester | Human | 979 | |
| SRC | Src | TK | 4k11 | A | A | 1-tert-butyl-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 983 | |
| SRC | Src | TK | 4k11 | A | B | 1-tert-butyl-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 977 | |
| SRC | Src | TK | 4mxo | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 990 | |
| SRC | Src | TK | 4mxo | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 978 | |
| SRC | Src | TK | 4mxx | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 989 | |
| SRC | Src | TK | 4mxx | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 976 | |
| SRC | Src | TK | 4mxy | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 982 | |
| SRC | Src | TK | 4mxy | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 972 | |
| SRC | Src | TK | 4mxz | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 969 | |
| SRC | Src | TK | 4mxz | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 988 | |
| SRC | Src | TK | 6ate | A | | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10920 | |
| SRC | Src | TK | 6e6e | A | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11485 | |
| SRC | Src | TK | 6e6e | A | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11482 | |
| SRC | Src | TK | 6e6e | A | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11491 | |
| SRC | Src | TK | 6e6e | B | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11480 | |
| SRC | Src | TK | 6e6e | B | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11476 | |
| SRC | Src | TK | 6e6e | B | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11484 | |
| SRC | Src | TK | 6e6e | C | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11471 | |
| SRC | Src | TK | 6e6e | C | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11492 | |
| SRC | Src | TK | 6e6e | C | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11488 | |
| SRC | Src | TK | 6e6e | D | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11489 | |
| SRC | Src | TK | 6e6e | D | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11494 | |
| SRC | Src | TK | 6e6e | D | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11473 | |
| SRC | Src | TK | 6e6e | E | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11479 | |
| SRC | Src | TK | 6e6e | E | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11490 | |
| SRC | Src | TK | 6e6e | E | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11478 | |
| SRC | Src | TK | 6e6e | F | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11487 | |
| SRC | Src | TK | 6e6e | F | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11472 | |
| SRC | Src | TK | 6e6e | F | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11486 | |
| SRC | Src | TK | 6e6e | G | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11493 | |
| SRC | Src | TK | 6e6e | G | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11474 | |
| SRC | Src | TK | 6e6e | G | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11477 | |
| SRC | Src | TK | 6e6e | H | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11475 | |
| SRC | Src | TK | 6e6e | H | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11483 | |
| SRC | Src | TK | 6e6e | H | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11481 | |
| SRC | Src | TK | 7ng7 | A | | tert-butyl (4-(4-amino-1-(2-(4-(dimethylamino)piperidin-1-yl)ethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)carbamate | Human | 13900 | |
| SRC | Src | TK | 7ote | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 14240 | |
| SRC | Src | TK | 8haq | A | | 4-[(~{e})-(7-oxidanyl-6~{h}-pyrrolo[2,3-g][1,3]benzothiazol-8-yl)methylideneamino]-~{n}-pyridin-2-yl-benzenesulfonamide | Human | 14883 | |
| SRC | Src | TK | 8jf3 | A | | 2-[4-[4-[bis(oxidanylidene)-$l^5-sulfanyl]oxyphenyl]carbonylpiperazin-1-yl]-6-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-n-prop-2-ynyl-pyrimidine-4-carboxamide | Human | 15226 | |
| SRC | Src | TK | 8jn8 | A | | (2r)-n-cyclopentyl-2-[cyclopropyl(ethanoyl)amino]-2-(4-fluorophenyl)ethanamide | Human | 15312 | |
| SRC | Src | TK | 8jn9 | A | | n-[(1r)-1-[3,5-bis(fluoranyl)phenyl]-2-(cyclopentylamino)-2-oxidanylidene-ethyl]-n-cyclopropyl-prop-2-enamide | Human | 15313 | |
| SRPK1 | SRPK | CMGC | 1wak | A | | - | Human | 120 | |
| SRPK1 | SRPK | CMGC | 1wbp | A | | adenosine-5'-diphosphate | Human | 119 | |
| SRPK1 | SRPK | CMGC | 3beg | A | | phosphoaminophosphonic acid-adenylate ester | Human | 9472 | |
| SRPK1 | SRPK | CMGC | 4wua | A | A | n-[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamide | Human | 9471 | |
| SRPK1 | SRPK | CMGC | 4wua | A | B | n-[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamide | Human | 9469 | |
| SRPK1 | SRPK | CMGC | 5mxx | A | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 9470 | |
| SRPK1 | SRPK | CMGC | 5mxx | A | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 9467 | |
| SRPK1 | SRPK | CMGC | 5my8 | A | A | sphinx31 | Human | 9466 | |
| SRPK1 | SRPK | CMGC | 5my8 | A | B | sphinx31 | Human | 9468 | |
| SRPK1 | SRPK | CMGC | 5xv7 | A | | 9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrile | Human | 9727 | |
| SRPK1 | SRPK | CMGC | 6fad | A | | - | Human | 11638 | |
| SRPK1 | SRPK | CMGC | 6fad | B | | - | Human | 11640 | |
| SRPK1 | SRPK | CMGC | 6fad | C | | - | Human | 11639 | |
| SRPK1 | SRPK | CMGC | 6fad | D | | - | Human | 11637 | |
| SRPK1 | SRPK | CMGC | 7dd1 | A | | - | Human | 13510 | |
| SRPK1 | SRPK | CMGC | 7pqs | A | A | ~{n}-[3-[[[2-(6-chloranyl-7-fluoranyl-1~{h}-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-~{n}-methyl-methanesulfonamide | Human | 14014 | |
| SRPK1 | SRPK | CMGC | 7pqs | A | B | ~{n}-[3-[[[2-(6-chloranyl-7-fluoranyl-1~{h}-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-~{n}-methyl-methanesulfonamide | Human | 14015 | |
| SRPK1 | SRPK | CMGC | 7zks | A | A | n-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamide | Human | 14619 | |
| SRPK1 | SRPK | CMGC | 7zks | A | B | n-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamide | Human | 14618 | |
| SRPK2 | SRPK | CMGC | 2x7g | A | | purvalanol b | Human | 1409 | |
| SRPK2 | SRPK | CMGC | 5myv | A | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7579 | |
| SRPK2 | SRPK | CMGC | 5myv | A | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7575 | |
| SRPK2 | SRPK | CMGC | 5myv | B | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7576 | |
| SRPK2 | SRPK | CMGC | 5myv | B | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7573 | |
| SRPK2 | SRPK | CMGC | 5myv | C | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7580 | |
| SRPK2 | SRPK | CMGC | 5myv | C | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7571 | |
| SRPK2 | SRPK | CMGC | 5myv | D | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7578 | |
| SRPK2 | SRPK | CMGC | 5myv | D | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7572 | |
| SRPK2 | SRPK | CMGC | 7zkx | A | A | n-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamide | Human | 14617 | |
| SRPK2 | SRPK | CMGC | 7zkx | A | B | n-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamide | Human | 14616 | |
| STK10 (LOK) | STE20 | STE | 2j7t | A | A | (3z)-n-(3-chlorophenyl)-3-({3,5-dimethyl-4-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-2-yl}methylene)-n-methyl-2-oxoindoline-5-sulfonamide | Human | 946 | |
| STK10 (LOK) | STE20 | STE | 2j7t | A | B | (3z)-n-(3-chlorophenyl)-3-({3,5-dimethyl-4-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-2-yl}methylene)-n-methyl-2-oxoindoline-5-sulfonamide | Human | 960 | |
| STK10 (LOK) | STE20 | STE | 4aot | A | A | 1-(4-{methyl[2-({4-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]amino}phenyl)-3-{3-[(4-methylpiperazin-1-yl)carbonyl]phenyl}urea | Human | 947 | |
| STK10 (LOK) | STE20 | STE | 4aot | A | B | 1-(4-{methyl[2-({4-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]amino}phenyl)-3-{3-[(4-methylpiperazin-1-yl)carbonyl]phenyl}urea | Human | 944 | |
| STK10 (LOK) | STE20 | STE | 4aot | B | A | 1-(4-{methyl[2-({4-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]amino}phenyl)-3-{3-[(4-methylpiperazin-1-yl)carbonyl]phenyl}urea | Human | 945 | |
| STK10 (LOK) | STE20 | STE | 4aot | B | B | 1-(4-{methyl[2-({4-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]amino}phenyl)-3-{3-[(4-methylpiperazin-1-yl)carbonyl]phenyl}urea | Human | 943 | |
| STK10 (LOK) | STE20 | STE | 4bc6 | A | A | 4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 942 | |
| STK10 (LOK) | STE20 | STE | 4bc6 | A | B | 4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 961 | |
| STK10 (LOK) | STE20 | STE | 4equ | A | A | n-{3-[(3-{4-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}pyridin-2-yl)amino]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | 957 | |
| STK10 (LOK) | STE20 | STE | 4equ | A | B | n-{3-[(3-{4-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}pyridin-2-yl)amino]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | 938 | |
| STK10 (LOK) | STE20 | STE | 4equ | B | A | n-{3-[(3-{4-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}pyridin-2-yl)amino]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | 941 | |
| STK10 (LOK) | STE20 | STE | 4equ | B | B | n-{3-[(3-{4-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}pyridin-2-yl)amino]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | 959 | |
| STK10 (LOK) | STE20 | STE | 4usd | A | A | 4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridine | Human | 953 | |
| STK10 (LOK) | STE20 | STE | 4usd | A | B | 4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridine | Human | 949 | |
| STK10 (LOK) | STE20 | STE | 4usd | B | A | 4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridine | Human | 939 | |
| STK10 (LOK) | STE20 | STE | 4usd | B | B | 4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridine | Human | 956 | |
| STK10 (LOK) | STE20 | STE | 4use | A | A | 4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridine | Human | 952 | |
| STK10 (LOK) | STE20 | STE | 4use | A | B | 4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridine | Human | 951 | |
| STK10 (LOK) | STE20 | STE | 4use | B | A | 4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridine | Human | 958 | |
| STK10 (LOK) | STE20 | STE | 4use | B | B | 4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridine | Human | 954 | |
| STK10 (LOK) | STE20 | STE | 5ajq | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 950 | |
| STK10 (LOK) | STE20 | STE | 5ajq | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 955 | |
| STK10 (LOK) | STE20 | STE | 5ajq | B | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 940 | |
| STK10 (LOK) | STE20 | STE | 5ajq | B | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 948 | |
| STK10 (LOK) | STE20 | STE | 5owq | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 8385 | |
| STK10 (LOK) | STE20 | STE | 5owq | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 8386 | |
| STK10 (LOK) | STE20 | STE | 5owq | B | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 8387 | |
| STK10 (LOK) | STE20 | STE | 5owq | B | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 8389 | |
| STK10 (LOK) | STE20 | STE | 5owr | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 8384 | |
| STK10 (LOK) | STE20 | STE | 5owr | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 8388 | |
| STK10 (LOK) | STE20 | STE | 6eim | A | A | ~{n}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-1~{h}-benzimidazol-2-yl]furan-2-carboxamide | Human | 8626 | |
| STK10 (LOK) | STE20 | STE | 6eim | A | B | ~{n}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-1~{h}-benzimidazol-2-yl]furan-2-carboxamide | Human | 8625 | |
| STK10 (LOK) | STE20 | STE | 6eim | B | A | ~{n}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-1~{h}-benzimidazol-2-yl]furan-2-carboxamide | Human | 8623 | |
| STK10 (LOK) | STE20 | STE | 6eim | B | B | ~{n}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-1~{h}-benzimidazol-2-yl]furan-2-carboxamide | Human | 8624 | |
| STK10 (LOK) | STE20 | STE | 6gtt | A | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 10026 | |
| STK10 (LOK) | STE20 | STE | 6gtt | A | B | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 10025 | |
| STK10 (LOK) | STE20 | STE | 6hxf | A | A | 3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dione | Human | 10656 | |
| STK10 (LOK) | STE20 | STE | 6hxf | A | B | 3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dione | Human | 10654 | |
| STK10 (LOK) | STE20 | STE | 6hxf | B | A | 3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dione | Human | 10651 | |
| STK10 (LOK) | STE20 | STE | 6hxf | B | B | 3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dione | Human | 10652 | |
| STK10 (LOK) | STE20 | STE | 6hxf | C | A | 3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dione | Human | 10649 | |
| STK10 (LOK) | STE20 | STE | 6hxf | C | B | 3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dione | Human | 10655 | |
| STK10 (LOK) | STE20 | STE | 6hxf | D | A | 3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dione | Human | 10650 | |
| STK10 (LOK) | STE20 | STE | 6hxf | D | B | 3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dione | Human | 10653 | |
| STK10 (LOK) | STE20 | STE | 6i2y | A | | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 10787 | |
| STK10 (LOK) | STE20 | STE | 6i2y | B | | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 10788 | |
| STK10 (LOK) | STE20 | STE | 7qgp | A | | 1-[(4-chloranyl-2-methyl-phenyl)methyl]-3-(7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaen-5-yl)urea | Human | 14075 | |
| STK11 (LKB1) | CAMKL | CAMK | 2wtk | C | | phosphoaminophosphonic acid-adenylate ester | Human | 1868 | |
| STK11 (LKB1) | CAMKL | CAMK | 2wtk | F | | phosphoaminophosphonic acid-adenylate ester | Human | 1869 | |
| STK11 (LKB1) | CAMKL | CAMK | 8vsu | B | | adenosine-5'-diphosphate | Human | 15343 | |
| STK16 (MPSK1) | NAK | Other | 2buj | A | | staurosporine | Human | 2229 | |
| STK16 (MPSK1) | NAK | Other | 2buj | B | | staurosporine | Human | 2230 | |
| STK17A (DRAK1) | DAPK | CAMK | 7que | A | | ~{n}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide | Human | 14094 | |
| STK17A (DRAK1) | DAPK | CAMK | 7quf | A | | ~{n}-~{tert}-butyl-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide | Human | 14093 | |
| STK17B (DRAK2) | DAPK | CAMK | 3lm0 | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-5-methylpyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 6796 | |
| STK17B (DRAK2) | DAPK | CAMK | 3lm0 | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-5-methylpyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 6797 | |
| STK17B (DRAK2) | DAPK | CAMK | 3lm5 | A | A | 3,5,7,3',4'-pentahydroxyflavone | Human | 6795 | |
| STK17B (DRAK2) | DAPK | CAMK | 3lm5 | A | B | 3,5,7,3',4'-pentahydroxyflavone | Human | 6798 | |
| STK17B (DRAK2) | DAPK | CAMK | 6qf4 | A | A | adenosine-5'-diphosphate | Human | 11397 | |
| STK17B (DRAK2) | DAPK | CAMK | 6qf4 | A | B | adenosine-5'-diphosphate | Human | 11396 | |
| STK17B (DRAK2) | DAPK | CAMK | 6y6f | A | A | 2-[6-(4-methylsulfanylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12045 | |
| STK17B (DRAK2) | DAPK | CAMK | 6y6f | A | B | 2-[6-(4-methylsulfanylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12042 | |
| STK17B (DRAK2) | DAPK | CAMK | 6y6h | A | A | 2-[6-(1-benzothiophen-2-yl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12043 | |
| STK17B (DRAK2) | DAPK | CAMK | 6y6h | A | B | 2-[6-(1-benzothiophen-2-yl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12044 | |
| STK17B (DRAK2) | DAPK | CAMK | 6zjf | A | A | 2-[6-(4-cyclopropylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12642 | |
| STK17B (DRAK2) | DAPK | CAMK | 6zjf | A | B | 2-[6-(4-cyclopropylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12643 | |
| STK17B (DRAK2) | DAPK | CAMK | 7akg | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 13005 | |
| STK17B (DRAK2) | DAPK | CAMK | 7akg | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 13004 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7c | A | A | adenosine-5'-diphosphate | Human | 14510 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7c | A | B | adenosine-5'-diphosphate | Human | 14508 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7d | A | A | adenosine-5'-triphosphate | Human | 14519 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7d | A | B | adenosine-5'-triphosphate | Human | 14509 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7e | A | A | adenosine-5'-triphosphate | Human | 14520 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7e | A | B | adenosine-5'-triphosphate | Human | 14507 | |
| STK24 (MST3) | STE20 | STE | 3a7f | A | | - | Human | 5596 | |
| STK24 (MST3) | STE20 | STE | 3a7g | A | | - | Human | 5612 | |
| STK24 (MST3) | STE20 | STE | 3a7g | B | | - | Human | 5598 | |
| STK24 (MST3) | STE20 | STE | 3a7h | A | | adenosine-5'-triphosphate | Human | 5600 | |
| STK24 (MST3) | STE20 | STE | 3a7h | B | | adenosine-5'-triphosphate | Human | 5576 | |
| STK24 (MST3) | STE20 | STE | 3a7i | A | | adenine | Human | 5611 | |
| STK24 (MST3) | STE20 | STE | 3a7j | A | | adenosine-5'-diphosphate | Human | 5594 | |
| STK24 (MST3) | STE20 | STE | 3ckw | A | A | - | Human | 5580 | |
| STK24 (MST3) | STE20 | STE | 3ckw | A | B | - | Human | 5601 | |
| STK24 (MST3) | STE20 | STE | 3ckx | A | | staurosporine | Human | 5599 | |
| STK24 (MST3) | STE20 | STE | 3zhp | C | | - | Human | 5593 | |
| STK24 (MST3) | STE20 | STE | 3zhp | D | | - | Human | 5588 | |
| STK24 (MST3) | STE20 | STE | 4o27 | B | | adenosine-5'-diphosphate | Human | 5602 | |
| STK24 (MST3) | STE20 | STE | 4qml | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5605 | |
| STK24 (MST3) | STE20 | STE | 4qmm | A | | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 5583 | |
| STK24 (MST3) | STE20 | STE | 4qmn | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 5587 | |
| STK24 (MST3) | STE20 | STE | 4qmn | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 5604 | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | A | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 5585 | |
| STK24 (MST3) | STE20 | STE | 4qmo | A | B | (8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 5597 | |
| STK24 (MST3) | STE20 | STE | 4qmp | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 5584 | |
| STK24 (MST3) | STE20 | STE | 4qmq | A | A | 1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amine | Human | 5607 | |
| STK24 (MST3) | STE20 | STE | 4qmq | A | B | 1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amine | Human | 5595 | |
| STK24 (MST3) | STE20 | STE | 4qms | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 5590 | |
| STK24 (MST3) | STE20 | STE | 4qms | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 5608 | |
| STK24 (MST3) | STE20 | STE | 4qmt | A | | n-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamide | Human | 5613 | |
| STK24 (MST3) | STE20 | STE | 4qmu | A | A | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 5606 | |
| STK24 (MST3) | STE20 | STE | 4qmu | A | B | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 5603 | |
| STK24 (MST3) | STE20 | STE | 4qmv | A | | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 5581 | |
| STK24 (MST3) | STE20 | STE | 4qmw | A | A | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 5577 | |
| STK24 (MST3) | STE20 | STE | 4qmw | A | B | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 5582 | |
| STK24 (MST3) | STE20 | STE | 4qmx | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 5609 | |
| STK24 (MST3) | STE20 | STE | 4qmy | A | | staurosporine | Human | 5592 | |
| STK24 (MST3) | STE20 | STE | 4qmz | A | | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 5578 | |
| STK24 (MST3) | STE20 | STE | 4qna | A | | 2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 5579 | |
| STK24 (MST3) | STE20 | STE | 4qo9 | A | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 5586 | |
| STK24 (MST3) | STE20 | STE | 4qo9 | B | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 5591 | |
| STK24 (MST3) | STE20 | STE | 4u8z | A | | 3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | 5610 | |
| STK24 (MST3) | STE20 | STE | 4w8d | A | | 5-(1-methyl-1h-pyrazol-4-yl)-4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidine | Human | 5614 | |
| STK24 (MST3) | STE20 | STE | 4w8e | A | | 3-{4-[(2r)-2-(5-methyl-1,2,4-oxadiazol-3-yl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | Human | 5589 | |
| STK24 (MST3) | STE20 | STE | 7b30 | A | | 8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 13047 | |
| STK24 (MST3) | STE20 | STE | 7b31 | A | A | 1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-one | Human | 13045 | |
| STK24 (MST3) | STE20 | STE | 7b31 | A | B | 1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-one | Human | 13050 | |
| STK24 (MST3) | STE20 | STE | 7b32 | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[(2-methoxyphenyl)amino]pyrido[2,3-d]pyrimidin-7-one | Human | 13049 | |
| STK24 (MST3) | STE20 | STE | 7b33 | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[4-[6-[bis(fluoranyl)methyl]pyridin-2-yl]-2-chloranyl-phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 13048 | |
| STK24 (MST3) | STE20 | STE | 7b34 | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranyl-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 13051 | |
| STK24 (MST3) | STE20 | STE | 7b35 | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 13052 | |
| STK24 (MST3) | STE20 | STE | 7b35 | B | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 13046 | |
| STK24 (MST3) | STE20 | STE | 8bzi | A | A | 8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14585 | |
| STK24 (MST3) | STE20 | STE | 8bzi | A | B | 8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14584 | |
| STK24 (MST3) | STE20 | STE | 8bzj | A | A | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14586 | |
| STK24 (MST3) | STE20 | STE | 8bzj | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14583 | |
| STK24 (MST3) | STE20 | STE | 8qlq | A | A | macrocyclic inhibitor | Human | 14873 | |
| STK24 (MST3) | STE20 | STE | 8qlq | A | B | macrocyclic inhibitor | Human | 14870 | |
| STK24 (MST3) | STE20 | STE | 8qlr | A | | 8-(4-azanylbutyl)-2-[1,3-bis(oxidanyl)propan-2-ylamino]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-one | Human | 14875 | |
| STK24 (MST3) | STE20 | STE | 8qls | A | A | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14872 | |
| STK24 (MST3) | STE20 | STE | 8qls | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14876 | |
| STK24 (MST3) | STE20 | STE | 8qls | A | C | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14871 | |
| STK24 (MST3) | STE20 | STE | 8qlt | A | A | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-one | Human | 14874 | |
| STK24 (MST3) | STE20 | STE | 8qlt | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-one | Human | 14869 | |
| STK25 (YSK1) | STE20 | STE | 2xik | A | A | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 463 | |
| STK25 (YSK1) | STE20 | STE | 2xik | A | B | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 465 | |
| STK25 (YSK1) | STE20 | STE | 4nzw | B | | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 464 | |
| STK25 (YSK1) | STE20 | STE | 7z4v | A | A | ~{n}-(5-~{tert}-butyl-1~{h}-pyrazol-3-yl)-4-pyrrolidin-1-ylsulfonyl-benzamide | Human | 14176 | |
| STK25 (YSK1) | STE20 | STE | 7z4v | A | B | ~{n}-(5-~{tert}-butyl-1~{h}-pyrazol-3-yl)-4-pyrrolidin-1-ylsulfonyl-benzamide | Human | 14177 | |
| STK26 (MST4) | STE20 | STE | 3ggf | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 1807 | |
| STK26 (MST4) | STE20 | STE | 3ggf | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 1808 | |
| STK26 (MST4) | STE20 | STE | 3ggf | B | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 1805 | |
| STK26 (MST4) | STE20 | STE | 3ggf | B | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 1804 | |
| STK26 (MST4) | STE20 | STE | 4fza | B | | - | Human | 1806 | |
| STK26 (MST4) | STE20 | STE | 4fzd | B | | - | Human | 1809 | |
| STK26 (MST4) | STE20 | STE | 4fzf | B | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1803 | |
| STK26 (MST4) | STE20 | STE | 7b36 | A | | 8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 13044 | |
| STK26 (MST4) | STE20 | STE | 7b36 | C | | 8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 13043 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | A | A | - | Human | 1442 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | A | B | - | Human | 1438 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | B | A | - | Human | 1433 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | B | B | - | Human | 1427 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | C | A | - | Human | 1432 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | C | B | - | Human | 1440 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | D | A | - | Human | 1435 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | D | B | - | Human | 1434 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | E | A | - | Human | 1439 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | E | B | - | Human | 1441 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | F | A | - | Human | 1431 | |
| STK3 (MST2) | STE20 | STE | 4lg4 | F | B | - | Human | 1436 | |
| STK3 (MST2) | STE20 | STE | 4lgd | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1437 | |
| STK3 (MST2) | STE20 | STE | 4lgd | B | | phosphoaminophosphonic acid-adenylate ester | Human | 1428 | |
| STK3 (MST2) | STE20 | STE | 4lgd | C | | phosphoaminophosphonic acid-adenylate ester | Human | 1429 | |
| STK3 (MST2) | STE20 | STE | 4lgd | D | | phosphoaminophosphonic acid-adenylate ester | Human | 1430 | |
| STK3 (MST2) | STE20 | STE | 5dh3 | A | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 7031 | |
| STK3 (MST2) | STE20 | STE | 5dh3 | A | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 7028 | |
| STK3 (MST2) | STE20 | STE | 5dh3 | B | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 7029 | |
| STK3 (MST2) | STE20 | STE | 5dh3 | B | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 7030 | |
| STK3 (MST2) | STE20 | STE | 6ao5 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 8662 | |
| STK3 (MST2) | STE20 | STE | 8a66 | A | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 14323 | |
| STK3 (MST2) | STE20 | STE | 8a66 | A | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 14324 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | A | A | staurosporine | Human | 4693 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | A | B | staurosporine | Human | 4690 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | B | A | staurosporine | Human | 4692 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | B | B | staurosporine | Human | 4695 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | C | A | staurosporine | Human | 4684 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | C | B | staurosporine | Human | 4694 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | D | A | staurosporine | Human | 4688 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | D | B | staurosporine | Human | 4687 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | E | A | staurosporine | Human | 4689 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | E | B | staurosporine | Human | 4685 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | F | A | staurosporine | Human | 4691 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | F | B | staurosporine | Human | 4686 | |
| STK38 (NDR1) | NDR | AGC | 6bxi | A | | phosphoaminophosphonic acid-adenylate ester | Human | 10326 | |
| STK38 (NDR1) | NDR | AGC | 6bxi | B | | phosphoaminophosphonic acid-adenylate ester | Human | 10325 | |
| Stk39 (STLK3) | STE20 | STE | 5d9h | A | | adenosine-5'-triphosphate | Mouse | 6025 | |
| Stk39 (STLK3) | STE20 | STE | 5d9h | B | | adenosine-5'-triphosphate | Mouse | 6024 | |
| Stk39 (STLK3) | STE20 | STE | 5dbx | A | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 6109 | |
| Stk39 (STLK3) | STE20 | STE | 5dbx | A | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 6107 | |
| Stk39 (STLK3) | STE20 | STE | 5dbx | B | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 6106 | |
| Stk39 (STLK3) | STE20 | STE | 5dbx | B | B | phosphoaminophosphonic acid-adenylate ester | Mouse | 6108 | |
| STK4 (MST1) | STE20 | STE | 3com | A | | - | Human | 2828 | |
| STK4 (MST1) | STE20 | STE | 3com | B | | - | Human | 2829 | |
| STK4 (MST1) | STE20 | STE | 6yat | A | | 4-[5-(3-chlorophenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]morpholine | Human | 12241 | |
| STK4 (MST1) | STE20 | STE | 6yat | B | | 4-[5-(3-chlorophenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]morpholine | Human | 12242 | |
| STK4 (MST1) | STE20 | STE | 8a5j | A | A | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 14290 | |
| STK4 (MST1) | STE20 | STE | 8a5j | A | B | 4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamide | Human | 14291 | |
| STK4 (MST1) | STE20 | STE | 8pav | A | A | 1-[3,5-bis(fluoranyl)-4-[[3-(1,3-thiazol-5-yl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-3-(2-methoxyethyl)urea | Human | 15349 | |
| STK4 (MST1) | STE20 | STE | 8pav | A | B | 1-[3,5-bis(fluoranyl)-4-[[3-(1,3-thiazol-5-yl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-3-(2-methoxyethyl)urea | Human | 15348 | |
| STK4 (MST1) | STE20 | STE | 8paw | A | | 1-[3,5-bis(fluoranyl)-4-[[3-(1-propan-2-ylpyrazol-3-yl)-1~{h}-pyrrolo[2,3-b]pyridin-4-yl]oxy]phenyl]-3-(2-methoxyethyl)urea | Human | 15350 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | A | A | - | Human | 8015 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | A | B | - | Human | 8014 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | B | A | - | Human | 8011 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | B | B | - | Human | 8017 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | C | A | - | Human | 8018 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | C | B | - | Human | 8016 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | D | A | - | Human | 8012 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | D | B | - | Human | 8013 | |
| STRADA (STLK5) | STE20 | STE | 2wtk | B | | phosphoaminophosphonic acid-adenylate ester | Human | 3485 | |
| STRADA (STLK5) | STE20 | STE | 2wtk | E | | phosphoaminophosphonic acid-adenylate ester | Human | 3484 | |
| STRADA (STLK5) | STE20 | STE | 3gni | B | | adenosine-5'-triphosphate | Human | 3486 | |
| STRADA (STLK5) | STE20 | STE | 8vsu | C | | - | Human | 15320 | |
| SYK | Syk | TK | 1xba | A | | - | Human | 1193 | |
| SYK | Syk | TK | 1xbb | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1184 | |
| SYK | Syk | TK | 1xbb | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1196 | |
| SYK | Syk | TK | 1xbc | A | A | staurosporine | Human | 1165 | |
| SYK | Syk | TK | 1xbc | A | B | staurosporine | Human | 1207 | |
| SYK | Syk | TK | 3emg | A | | 2-{2-[(3,5-dimethylphenyl)amino]pyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-methylethyl]-4-methyl-1,3-thiazole-5-carboxamide | Human | 1183 | |
| SYK | Syk | TK | 3fqe | A | | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(3-methylphenyl)amino]pyrimidine-5-carboxamide | Human | 1155 | |
| SYK | Syk | TK | 3fqh | A | | n-(2-hydroxy-1,1-dimethylethyl)-1-methyl-3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indole-5-carboxamide | Human | 1203 | |
| SYK | Syk | TK | 3fqh | B | | n-(2-hydroxy-1,1-dimethylethyl)-1-methyl-3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indole-5-carboxamide | Human | 1171 | |
| SYK | Syk | TK | 3fqs | A | A | 6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-one | Human | 1169 | |
| SYK | Syk | TK | 3fqs | A | B | 6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-one | Human | 1202 | |
| SYK | Syk | TK | 3srv | A | A | 2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamide | Human | 1154 | |
| SYK | Syk | TK | 3srv | A | B | 2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamide | Human | 1162 | |
| SYK | Syk | TK | 3srv | B | A | 2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamide | Human | 1181 | |
| SYK | Syk | TK | 3srv | B | B | 2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamide | Human | 1206 | |
| SYK | Syk | TK | 3tub | A | | 1-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-3-[(1r,2s)-2-phenylcyclopropyl]urea | Human | 1179 | |
| SYK | Syk | TK | 3tuc | A | | 1-benzyl-n-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-2-oxo-1,2-dihydropyridine-3-carboxamide | Human | 1195 | |
| SYK | Syk | TK | 3tud | A | | n-{4-methyl-3-[8-methyl-7-oxo-2-(phenylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]phenyl}-3-(trifluoromethyl)benzamide | Human | 1176 | |
| SYK | Syk | TK | 3vf8 | A | | 3-[5-(5-ethoxy-6-fluoro-1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]-1,1-diethylurea | Human | 1187 | |
| SYK | Syk | TK | 3vf9 | A | | 3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-ol | Human | 1159 | |
| SYK | Syk | TK | 4dfl | A | | 3-amino-6-{3-[(methylsulfonyl)amino]phenyl}-n-(piperidin-4-ylmethyl)pyrazine-2-carboxamide | Human | 1152 | |
| SYK | Syk | TK | 4dfn | A | A | 3-amino-6-[3-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-[(1r,2r,3s,5s,7s)-5-hydroxyadamantan-2-yl]pyrazine-2-carboxamide | Human | 1201 | |
| SYK | Syk | TK | 4dfn | A | B | 3-amino-6-[3-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-[(1r,2r,3s,5s,7s)-5-hydroxyadamantan-2-yl]pyrazine-2-carboxamide | Human | 1199 | |
| SYK | Syk | TK | 4f4p | A | A | n-{6-[3-(piperazin-1-yl)phenyl]pyridin-2-yl}-4-(trifluoromethyl)pyridin-2-amine | Human | 1178 | |
| SYK | Syk | TK | 4f4p | A | B | n-{6-[3-(piperazin-1-yl)phenyl]pyridin-2-yl}-4-(trifluoromethyl)pyridin-2-amine | Human | 1156 | |
| SYK | Syk | TK | 4fl1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 1160 | |
| SYK | Syk | TK | 4fl1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 1167 | |
| SYK | Syk | TK | 4fl2 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1191 | |
| SYK | Syk | TK | 4fl3 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 1170 | |
| SYK | Syk | TK | 4fl3 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 1172 | |
| SYK | Syk | TK | 4fyn | A | A | 3-[8-({4-[ethyl(2-hydroxyethyl)amino]phenyl}amino)imidazo[1,2-a]pyrazin-5-yl]phenol | Human | 1174 | |
| SYK | Syk | TK | 4fyn | A | B | 3-[8-({4-[ethyl(2-hydroxyethyl)amino]phenyl}amino)imidazo[1,2-a]pyrazin-5-yl]phenol | Human | 1197 | |
| SYK | Syk | TK | 4fyo | A | A | 4-{[(3s)-1-{7-[(3,4-dimethoxyphenyl)amino][1,3]thiazolo[5,4-d]pyrimidin-5-yl}pyrrolidin-3-yl]carbamoyl}benzoic acid | Human | 1180 | |
| SYK | Syk | TK | 4fyo | A | B | 4-{[(3s)-1-{7-[(3,4-dimethoxyphenyl)amino][1,3]thiazolo[5,4-d]pyrimidin-5-yl}pyrrolidin-3-yl]carbamoyl}benzoic acid | Human | 1205 | |
| SYK | Syk | TK | 4fz6 | A | A | n-{6-[(2s)-2-methylpyrrolidin-1-yl]pyridin-2-yl}-6-phenylimidazo[1,2-b]pyridazin-8-amine | Human | 1173 | |
| SYK | Syk | TK | 4fz6 | A | B | n-{6-[(2s)-2-methylpyrrolidin-1-yl]pyridin-2-yl}-6-phenylimidazo[1,2-b]pyridazin-8-amine | Human | 1185 | |
| SYK | Syk | TK | 4fz7 | A | A | 6-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(6-ethylpyridin-2-yl)amino]pyridazine-3-carboxamide | Human | 1186 | |
| SYK | Syk | TK | 4fz7 | A | B | 6-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(6-ethylpyridin-2-yl)amino]pyridazine-3-carboxamide | Human | 1177 | |
| SYK | Syk | TK | 4gfg | A | | 6-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(5,6-dimethylpyridin-2-yl)amino]pyridazine-3-carboxamide | Human | 1188 | |
| SYK | Syk | TK | 4i0r | A | A | n-(propan-2-yl)-2-(3,4,5-trimethoxyphenyl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 1192 | |
| SYK | Syk | TK | 4i0r | A | B | n-(propan-2-yl)-2-(3,4,5-trimethoxyphenyl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 1175 | |
| SYK | Syk | TK | 4i0s | A | A | 2-(6-chloro-1-methyl-1h-indazol-3-yl)-n-(propan-2-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 1157 | |
| SYK | Syk | TK | 4i0s | A | B | 2-(6-chloro-1-methyl-1h-indazol-3-yl)-n-(propan-2-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 1166 | |
| SYK | Syk | TK | 4i0t | A | A | n-tert-butyl-2-(5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-1-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 1198 | |
| SYK | Syk | TK | 4i0t | A | B | n-tert-butyl-2-(5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-1-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamide | Human | 1164 | |
| SYK | Syk | TK | 4puz | A | | 6-(1h-indazol-6-yl)-n-[4-(morpholin-4-yl)phenyl]imidazo[1,2-a]pyrazin-8-amine | Human | 1163 | |
| SYK | Syk | TK | 4puz | B | | 6-(1h-indazol-6-yl)-n-[4-(morpholin-4-yl)phenyl]imidazo[1,2-a]pyrazin-8-amine | Human | 1153 | |
| SYK | Syk | TK | 4pv0 | A | | 4-[(3-{8-[(3,4-dimethoxyphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzoyl)amino]benzoic acid | Human | 1161 | |
| SYK | Syk | TK | 4px6 | A | A | 7-{[(1r,2s)-2-aminocyclohexyl]amino}-5-(1h-indol-7-ylamino)pyrido[4,3-d]pyrimidin-4(3h)-one | Human | 1200 | |
| SYK | Syk | TK | 4px6 | A | B | 7-{[(1r,2s)-2-aminocyclohexyl]amino}-5-(1h-indol-7-ylamino)pyrido[4,3-d]pyrimidin-4(3h)-one | Human | 1204 | |
| SYK | Syk | TK | 4rss | A | A | 1-[(3-methyl-1-{2-[(1,2,3-trimethyl-1h-indol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6169 | |
| SYK | Syk | TK | 4rss | A | B | 1-[(3-methyl-1-{2-[(1,2,3-trimethyl-1h-indol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6170 | |
| SYK | Syk | TK | 4rx7 | A | A | 3-{[(1r,2s)-2-aminocyclohexyl]amino}-5-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}-1,2,4-triazine-6-carboxamide | Human | 1189 | |
| SYK | Syk | TK | 4rx7 | A | B | 3-{[(1r,2s)-2-aminocyclohexyl]amino}-5-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}-1,2,4-triazine-6-carboxamide | Human | 1182 | |
| SYK | Syk | TK | 4rx8 | A | A | 3-{[(1r,2s)-2-aminocyclohexyl]amino}-5-(1h-indol-7-ylamino)-1,2,4-triazine-6-carboxamide | Human | 1158 | |
| SYK | Syk | TK | 4rx8 | A | B | 3-{[(1r,2s)-2-aminocyclohexyl]amino}-5-(1h-indol-7-ylamino)-1,2,4-triazine-6-carboxamide | Human | 1168 | |
| SYK | Syk | TK | 4rx9 | A | A | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamide | Human | 1190 | |
| SYK | Syk | TK | 4rx9 | A | B | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamide | Human | 1194 | |
| SYK | Syk | TK | 4wnm | A | | n~3~-(tetrahydro-2h-pyran-4-yl)-n~6~-[5-(tetrahydro-2h-pyran-4-ylmethyl)[1,2,4]triazolo[1,5-a]pyridin-2-yl]-1h-indazole-3,6-diamine | Human | 6358 | |
| SYK | Syk | TK | 4xg2 | A | | - | Human | 6309 | |
| SYK | Syk | TK | 4xg3 | A | | 4-{[5-fluoro-4-(3-{[(3r)-3-hydroxypyrrolidin-1-yl]methyl}-4-methyl-1h-pyrrol-1-yl)pyrimidin-2-yl]amino}-2,6-dimethylphenyl methanesulfonate | Human | 6308 | |
| SYK | Syk | TK | 4xg3 | B | | 4-{[5-fluoro-4-(3-{[(3r)-3-hydroxypyrrolidin-1-yl]methyl}-4-methyl-1h-pyrrol-1-yl)pyrimidin-2-yl]amino}-2,6-dimethylphenyl methanesulfonate | Human | 6314 | |
| SYK | Syk | TK | 4xg4 | A | | (3r)-1-{[1-(5-fluoro-2-{[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]amino}pyrimidin-4-yl)-4-methyl-1h-pyrrol-3-yl]methyl}pyrrolidin-3-ol | Human | 6319 | |
| SYK | Syk | TK | 4xg6 | A | | 1-[(1-{2-[(3,5-dimethylphenyl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6312 | |
| SYK | Syk | TK | 4xg7 | A | A | 1-[(3-methyl-1-{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6316 | |
| SYK | Syk | TK | 4xg7 | A | B | 1-[(3-methyl-1-{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6318 | |
| SYK | Syk | TK | 4xg8 | A | | 1-[(1-{2-[(3-chloro-1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6317 | |
| SYK | Syk | TK | 4xg8 | C | | 1-[(1-{2-[(3-chloro-1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6310 | |
| SYK | Syk | TK | 4xg9 | A | | 1-[(1-{2-[(3-chloro-1,2-dimethyl-1h-indol-5-yl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6311 | |
| SYK | Syk | TK | 4xg9 | B | | 1-[(1-{2-[(3-chloro-1,2-dimethyl-1h-indol-5-yl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-ol | Human | 6315 | |
| SYK | Syk | TK | 4yjo | A | A | 5-chloro-n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6120 | |
| SYK | Syk | TK | 4yjo | A | B | 5-chloro-n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6119 | |
| SYK | Syk | TK | 4yjp | A | | 2-[{2-[(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)amino]pyrimidin-4-yl}(1h-indazol-4-yl)amino]ethanol | Human | 6115 | |
| SYK | Syk | TK | 4yjq | A | A | 3-[1h-indazol-4-yl(2-{[3-(4-methyl-1,3-oxazol-5-yl)phenyl]amino}pyrimidin-4-yl)amino]propan-1-ol | Human | 6114 | |
| SYK | Syk | TK | 4yjq | A | B | 3-[1h-indazol-4-yl(2-{[3-(4-methyl-1,3-oxazol-5-yl)phenyl]amino}pyrimidin-4-yl)amino]propan-1-ol | Human | 6123 | |
| SYK | Syk | TK | 4yjr | A | A | 3-(1h-indazol-4-yl{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-ol | Human | 6113 | |
| SYK | Syk | TK | 4yjr | A | B | 3-(1h-indazol-4-yl{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-ol | Human | 6116 | |
| SYK | Syk | TK | 4yjr | A | C | 3-(1h-indazol-4-yl{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-ol | Human | 6122 | |
| SYK | Syk | TK | 4yjs | A | | 3-[{2-[(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)amino]pyrimidin-4-yl}(1h-indazol-4-yl)amino]propan-1-ol | Human | 6117 | |
| SYK | Syk | TK | 4yjt | A | A | n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-5-fluoro-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6125 | |
| SYK | Syk | TK | 4yjt | A | B | n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-5-fluoro-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6118 | |
| SYK | Syk | TK | 4yjt | A | C | n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-5-fluoro-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamine | Human | 6124 | |
| SYK | Syk | TK | 4yju | A | A | n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-5-fluoro-n~4~-(1h-indazol-4-yl)-n~4~-methylpyrimidine-2,4-diamine | Human | 6112 | |
| SYK | Syk | TK | 4yju | A | B | n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-5-fluoro-n~4~-(1h-indazol-4-yl)-n~4~-methylpyrimidine-2,4-diamine | Human | 6121 | |
| SYK | Syk | TK | 4yjv | A | A | 3-[6-({4-[ethyl(1h-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1h-indazol-1-yl]propan-1-ol | Human | 6150 | |
| SYK | Syk | TK | 4yjv | A | B | 3-[6-({4-[ethyl(1h-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1h-indazol-1-yl]propan-1-ol | Human | 6148 | |
| SYK | Syk | TK | 4yjv | A | C | 3-[6-({4-[ethyl(1h-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1h-indazol-1-yl]propan-1-ol | Human | 6149 | |
| SYK | Syk | TK | 5c26 | A | | 3-{8-[(3,4-dimethoxyphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzamide | Human | 6131 | |
| SYK | Syk | TK | 5c27 | A | | 3-{8-[(3,4-dimethoxyphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}-n-[4-(methylcarbamoyl)phenyl]benzamide | Human | 6132 | |
| SYK | Syk | TK | 5cxh | A | | (4r)-4-[(1r)-1-{[6-(3,4-dimethoxyphenyl)[1,3]thiazolo[5,4-c]pyridin-4-yl]oxy}ethyl]pyrrolidin-2-one | Human | 6057 | |
| SYK | Syk | TK | 5cxz | A | A | n-{7-[4-(dimethylamino)phenyl]-1,6-naphthyridin-5-yl}propane-1,3-diamine | Human | 6040 | |
| SYK | Syk | TK | 5cxz | A | B | n-{7-[4-(dimethylamino)phenyl]-1,6-naphthyridin-5-yl}propane-1,3-diamine | Human | 6041 | |
| SYK | Syk | TK | 5cy3 | A | A | (5r)-5-[(1r)-1-{[6-(1-methyl-1h-pyrazol-4-yl)-2,1-benzothiazol-4-yl]oxy}ethyl]-1,3-oxazolidin-2-one | Human | 6058 | |
| SYK | Syk | TK | 5cy3 | A | B | (5r)-5-[(1r)-1-{[6-(1-methyl-1h-pyrazol-4-yl)-2,1-benzothiazol-4-yl]oxy}ethyl]-1,3-oxazolidin-2-one | Human | 6056 | |
| SYK | Syk | TK | 5ghv | A | | 1-({1-[2-({3,5-dimethyl-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}amino)pyrimidin-4-yl]-4-methyl-1h-pyrrol-3-yl}methyl)azetidin-3-ol | Human | 6743 | |
| SYK | Syk | TK | 5ghv | B | | 1-({1-[2-({3,5-dimethyl-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}amino)pyrimidin-4-yl]-4-methyl-1h-pyrrol-3-yl}methyl)azetidin-3-ol | Human | 6742 | |
| SYK | Syk | TK | 5lma | A | A | ~{n}'-[7-(4-methylphenyl)pyrido[3,4-b]pyrazin-5-yl]butane-1,4-diamine | Human | 7047 | |
| SYK | Syk | TK | 5lma | A | B | ~{n}'-[7-(4-methylphenyl)pyrido[3,4-b]pyrazin-5-yl]butane-1,4-diamine | Human | 7049 | |
| SYK | Syk | TK | 5lma | A | C | ~{n}'-[7-(4-methylphenyl)pyrido[3,4-b]pyrazin-5-yl]butane-1,4-diamine | Human | 7044 | |
| SYK | Syk | TK | 5lmb | A | A | 7-[6-(dimethylamino)pyridin-3-yl]-~{n}-[[(3~{s})-piperidin-3-yl]methyl]pyrido[3,4-b]pyrazin-5-amine | Human | 7050 | |
| SYK | Syk | TK | 5lmb | A | B | 7-[6-(dimethylamino)pyridin-3-yl]-~{n}-[[(3~{s})-piperidin-3-yl]methyl]pyrido[3,4-b]pyrazin-5-amine | Human | 7046 | |
| SYK | Syk | TK | 5lmb | B | A | 7-[6-(dimethylamino)pyridin-3-yl]-~{n}-[[(3~{s})-piperidin-3-yl]methyl]pyrido[3,4-b]pyrazin-5-amine | Human | 7045 | |
| SYK | Syk | TK | 5lmb | B | B | 7-[6-(dimethylamino)pyridin-3-yl]-~{n}-[[(3~{s})-piperidin-3-yl]methyl]pyrido[3,4-b]pyrazin-5-amine | Human | 7048 | |
| SYK | Syk | TK | 5t68 | A | | n~4~-cyclopropyl-n~2~-(3-methyl-1h-indazol-6-yl)furo[3,2-d]pyrimidine-2,4-diamine | Human | 7119 | |
| SYK | Syk | TK | 5t68 | B | | n~4~-cyclopropyl-n~2~-(3-methyl-1h-indazol-6-yl)furo[3,2-d]pyrimidine-2,4-diamine | Human | 7120 | |
| SYK | Syk | TK | 5tiu | A | A | 5-{[(2s)-2-aminopropyl]amino}-3-(1h-indol-2-yl)pyrazine-2-carboxamide | Human | 7350 | |
| SYK | Syk | TK | 5tiu | A | B | 5-{[(2s)-2-aminopropyl]amino}-3-(1h-indol-2-yl)pyrazine-2-carboxamide | Human | 7349 | |
| SYK | Syk | TK | 5tr6 | A | A | 6-{[(1r,2s)-2-aminocyclohexyl]amino}-7-fluoro-4-(1-methyl-1h-pyrazol-4-yl)-1,2-dihydro-3h-pyrrolo[3,4-c]pyridin-3-one | Human | 7282 | |
| SYK | Syk | TK | 5tr6 | A | B | 6-{[(1r,2s)-2-aminocyclohexyl]amino}-7-fluoro-4-(1-methyl-1h-pyrazol-4-yl)-1,2-dihydro-3h-pyrrolo[3,4-c]pyridin-3-one | Human | 7284 | |
| SYK | Syk | TK | 5tt7 | A | A | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(3-methylphenyl)amino]-6,7-dihydro-5h-pyrrolo[3,4-d]pyrimidin-5-one | Human | 7281 | |
| SYK | Syk | TK | 5tt7 | A | B | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(3-methylphenyl)amino]-6,7-dihydro-5h-pyrrolo[3,4-d]pyrimidin-5-one | Human | 7283 | |
| SYK | Syk | TK | 5y5t | A | | 2-[[(1s,2s)-2-azanylcyclohexyl]amino]-4-[(4-methylsulfonylphenyl)amino]-6h-pyrido[4,3-d]pyrimidin-5-one | Human | 10028 | |
| SYK | Syk | TK | 5y5u | A | | 4-[(1-methylindazol-5-yl)amino]-2-(4-oxidanylpiperidin-1-yl)-8h-pyrido[4,3-d]pyrimidin-5-one | Human | 10027 | |
| SYK | Syk | TK | 5y5u | B | | 4-[(1-methylindazol-5-yl)amino]-2-(4-oxidanylpiperidin-1-yl)-8h-pyrido[4,3-d]pyrimidin-5-one | Human | 10029 | |
| SYK | Syk | TK | 6hm6 | A | A | 2-(4-methylphenyl)-3-(pyridin-2-ylmethoxy)pyridine | Human | 10614 | |
| SYK | Syk | TK | 6hm6 | A | B | 2-(4-methylphenyl)-3-(pyridin-2-ylmethoxy)pyridine | Human | 10613 | |
| SYK | Syk | TK | 6hm7 | A | A | 7-[2-methoxy-6-[(4-methylpyridin-2-yl)methoxy]phenyl]-2,3,4,5-tetrahydro-1~{h}-3-benzazepine | Human | 10612 | |
| SYK | Syk | TK | 6hm7 | A | B | 7-[2-methoxy-6-[(4-methylpyridin-2-yl)methoxy]phenyl]-2,3,4,5-tetrahydro-1~{h}-3-benzazepine | Human | 10615 | |
| SYK | Syk | TK | 6ssb | A | | ~{n}-[4-[5-[(dimethylamino)methyl]-1-methyl-pyrazol-3-yl]pyrimidin-2-yl]-3-methyl-1-(5-methyl-1,3,4-oxadiazol-2-yl)imidazo[1,5-a]pyridin-7-amine | Human | 12817 | |
| SYK | Syk | TK | 6vov | A | | 6-(6-aminopyrazin-2-yl)-n-{4-[4-(oxetan-3-yl)piperazin-1-yl]phenyl}imidazo[1,2-a]pyrazin-8-amine | Human | 12041 | |
| SYK | Syk | TK | 6vov | B | | 6-(6-aminopyrazin-2-yl)-n-{4-[4-(oxetan-3-yl)piperazin-1-yl]phenyl}imidazo[1,2-a]pyrazin-8-amine | Human | 12040 | |
| SYK | Syk | TK | 6zc0 | A | | ~{n},~{n}-dimethyl-1-[1-[2-(1-methylindol-4-yl)-3~{h}-imidazo[4,5-b]pyridin-7-yl]pyrazol-4-yl]methanamine | Human | 13636 | |
| SYK | Syk | TK | 6zcp | A | | 7-[[4-[4-[(dimethylamino)methyl]pyrazol-1-yl]pyrimidin-2-yl]amino]-~{n},3-dimethyl-imidazo[1,5-a]pyridine-1-carboxamide | Human | 13632 | |
| SYK | Syk | TK | 6zcq | A | | 7-[[4-[4-[[(3~{r},4~{r})-3-azanyloxan-4-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]-~{n},3-dimethyl-imidazo[1,5-a]pyridine-1-carboxamide | Human | 13633 | |
| SYK | Syk | TK | 6zcr | A | A | 6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amine | Human | 13630 | |
| SYK | Syk | TK | 6zcr | A | B | 6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amine | Human | 13631 | |
| SYK | Syk | TK | 6zcs | A | A | (3~{r},4~{r})-~{n}4-[1-[2-(1-methylindol-4-yl)-3~{h}-imidazo[4,5-b]pyridin-7-yl]pyrazol-4-yl]oxane-3,4-diamine | Human | 13639 | |
| SYK | Syk | TK | 6zcs | A | B | (3~{r},4~{r})-~{n}4-[1-[2-(1-methylindol-4-yl)-3~{h}-imidazo[4,5-b]pyridin-7-yl]pyrazol-4-yl]oxane-3,4-diamine | Human | 13641 | |
| SYK | Syk | TK | 6zcu | A | A | 6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amine | Human | 13640 | |
| SYK | Syk | TK | 6zcu | A | B | 6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amine | Human | 13635 | |
| SYK | Syk | TK | 6zcx | A | A | ~{n},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{r})-piperidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamide | Human | 13642 | |
| SYK | Syk | TK | 6zcx | A | B | ~{n},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{r})-piperidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamide | Human | 13637 | |
| SYK | Syk | TK | 6zcy | A | A | ~{n},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{r})-pyrrolidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamide | Human | 13634 | |
| SYK | Syk | TK | 6zcy | A | B | ~{n},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{r})-pyrrolidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamide | Human | 13638 | |
| SYK | Syk | TK | 8bi2 | A | | 10,13,23-trimethyl-16-oxa-2,4,8,9,13,19,23,30-octazapentacyclo[19.5.2.1^{3,7}.1^{8,11}.0^{24,28}]triaconta-1(27),3,5,7(30),9,11(29),21,24(28),25-nonaen-20-one | Human | 14779 | |
| SYK | Syk | TK | 8x5k | A | A | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamide | Human | 15103 | |
| SYK | Syk | TK | 8x5k | A | B | 2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamide | Human | 15102 | |
| TAOK3 (TAO3) | STE20 | STE | 6bdn | A | A | adenosine-5'-diphosphate | Human | 11004 | |
| TAOK3 (TAO3) | STE20 | STE | 6bdn | A | B | adenosine-5'-diphosphate | Human | 11003 | |
| Tbk1 (TBK1) | IKK | Other | 4jl9 | A | | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Mouse | 5697 | |
| Tbk1 (TBK1) | IKK | Other | 4jlc | A | | 3-{2,4-dimethyl-5-[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-1h-pyrrol-3-yl}propanoic acid | Mouse | 5698 | |
| Tbk1 (TBK1) | IKK | Other | 6o8c | A | A | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Mouse | 11303 | |
| Tbk1 (TBK1) | IKK | Other | 6o8c | A | B | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Mouse | 11302 | |
| Tbk1 (TBK1) | IKK | Other | 6o8c | B | A | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Mouse | 11305 | |
| Tbk1 (TBK1) | IKK | Other | 6o8c | B | B | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Mouse | 11304 | |
| TBK1 | IKK | Other | 4eut | A | A | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 609 | |
| TBK1 | IKK | Other | 4eut | A | B | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 621 | |
| TBK1 | IKK | Other | 4eut | B | A | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 618 | |
| TBK1 | IKK | Other | 4eut | B | B | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 617 | |
| TBK1 | IKK | Other | 4euu | A | A | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 615 | |
| TBK1 | IKK | Other | 4euu | A | B | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 611 | |
| TBK1 | IKK | Other | 4euu | B | A | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 606 | |
| TBK1 | IKK | Other | 4euu | B | B | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 616 | |
| TBK1 | IKK | Other | 4im0 | A | A | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 610 | |
| TBK1 | IKK | Other | 4im0 | A | B | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 607 | |
| TBK1 | IKK | Other | 4im2 | A | A | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 620 | |
| TBK1 | IKK | Other | 4im2 | A | B | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 613 | |
| TBK1 | IKK | Other | 4im3 | A | A | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 619 | |
| TBK1 | IKK | Other | 4im3 | A | B | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 622 | |
| TBK1 | IKK | Other | 4iw0 | A | | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 608 | |
| TBK1 | IKK | Other | 4iwo | A | | n-{3-[(5-cyclopropyl-2-{[3-(2-oxopyrrolidin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 614 | |
| TBK1 | IKK | Other | 4iwp | A | | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 612 | |
| TBK1 | IKK | Other | 4iwq | A | | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 605 | |
| TBK1 | IKK | Other | 5w5v | A | | 2-amino-7-(1-methylethyl)-5-oxo-5h-chromeno[2,3-b]pyridine-3-carboxylic acid | Human | 10024 | |
| TBK1 | IKK | Other | 6bny | A | | 2-amino-7-(propan-2-yl)-3-(1h-tetrazol-5-yl)-5h-[1]benzopyrano[2,3-b]pyridin-5-one | Human | 10369 | |
| TBK1 | IKK | Other | 6bod | A | | ethyl 2-amino-5-oxo-7-(propan-2-yl)-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylate | Human | 10370 | |
| TBK1 | IKK | Other | 6boe | A | | 2-amino-5-oxo-7-(propan-2-yl)-n-(1h-tetrazol-5-yl)-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxamide | Human | 10371 | |
| TBK1 | IKK | Other | 6cq0 | A | | 2-amino-7-[3-(dimethylamino)propyl]-5-oxo-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acid | Human | 10756 | |
| TBK1 | IKK | Other | 6cq4 | A | | 2-amino-7-(4,4-difluorocyclohexyl)-5-oxo-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acid | Human | 10757 | |
| TBK1 | IKK | Other | 6cq5 | A | | 2-amino-7-(1,1-dioxo-1lambda~6~-thian-4-yl)-5-oxo-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acid | Human | 10758 | |
| TBK1 | IKK | Other | 6nt9 | A | | - | Human | 10940 | |
| TBK1 | IKK | Other | 6nt9 | B | | - | Human | 10941 | |
| TBK1 | IKK | Other | 6o8b | A | | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 11053 | |
| TBK1 | IKK | Other | 6o8b | B | | n-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide | Human | 11054 | |
| TBK1 | IKK | Other | 6rsr | A | | ~{n}-(cyclopropen-1-ylmethyl)-2-[[4-[[4-[3,3,3-tris(fluoranyl)propanoyl]piperazin-1-yl]methyl]pyridin-2-yl]amino]-1~{h}-benzimidazole-5-carboxamide | Human | 11903 | |
| TBK1 | IKK | Other | 6rst | A | | 1-[4-[(1~{r})-1-[2-[[5-[1-(cyclopropylmethyl)pyrazol-4-yl]-1~{h}-benzimidazol-2-yl]amino]pyridin-4-yl]ethyl]piperazin-1-yl]-3,3,3-tris(fluoranyl)propan-1-one | Human | 11902 | |
| TBK1 | IKK | Other | 6rsu | A | | 3,3,3-tris(fluoranyl)-1-[4-[(1~{r})-1-[2-[[(2~{s})-5-(5-propan-2-yloxypyrimidin-4-yl)-2,3-dihydro-1~{h}-benzimidazol-2-yl]amino]pyridin-4-yl]ethyl]piperazin-1-yl]propan-1-one | Human | 12126 | |
| TEK (TIE2) | Tie | TK | 1fvr | A | | - | Human | 5551 | |
| TEK (TIE2) | Tie | TK | 1fvr | B | | - | Human | 5554 | |
| TEK (TIE2) | Tie | TK | 2oo8 | X | | n-{3-[3-(dimethylamino)propyl]-5-(trifluoromethyl)phenyl}-4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]benzamide | Human | 5556 | |
| TEK (TIE2) | Tie | TK | 2osc | A | | n-{4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]phenyl}-3-(trifluoromethyl)benzamide | Human | 5555 | |
| TEK (TIE2) | Tie | TK | 2p4i | A | | 4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)-n-[2-morpholin-4-yl-5-(trifluoromethyl)phenyl]benzamide | Human | 5549 | |
| TEK (TIE2) | Tie | TK | 2p4i | B | | 4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)-n-[2-morpholin-4-yl-5-(trifluoromethyl)phenyl]benzamide | Human | 5550 | |
| TEK (TIE2) | Tie | TK | 2wqb | A | | 2-[3-(cyclohexylmethyl)-5-phenyl-imidazol-4-yl]-[1,3]thiazolo[4,5-e]pyrimidin-7-amine | Human | 5553 | |
| TEK (TIE2) | Tie | TK | 3l8p | A | | 2-methyl-11-(1-methylethyl)-8-[(2s)-tetrahydro-2h-pyran-2-yl]-2,11,12,13-tetrahydro-4h-indazolo[5,4-a]pyrrolo[3,4-c]carbazol-4-one | Human | 5548 | |
| TEK (TIE2) | Tie | TK | 4x3j | A | | 1-[4-(4-amino-5-oxopyrido[2,3-d]pyrimidin-8(5h)-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea | Human | 5552 | |
| TEK (TIE2) | Tie | TK | 6mwe | A | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 10710 | |
| TEK (TIE2) | Tie | TK | 6mwe | A | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 10711 | |
| TEK (TIE2) | Tie | TK | 6mwe | B | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 10712 | |
| TEK (TIE2) | Tie | TK | 6mwe | B | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 10713 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | B | | - | Human | 2133 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | D | | - | Human | 2126 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | F | | - | Human | 2103 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | H | | - | Human | 2099 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | A | | - | Human | 2113 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | B | | - | Human | 2102 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | C | | - | Human | 2117 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | D | | - | Human | 2131 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | E | | - | Human | 2134 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1py5 | A | | 4-(3-pyridin-2-yl-1h-pyrazol-4-yl)quinoline | Human | 2094 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1rw8 | A | | 3-(4-fluorophenyl)-2-(6-methylpyridin-2-yl)-5,6-dihydro-4h-pyrrolo[1,2-b]pyrazole | Human | 2100 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1vjy | A | | 2-[5-(6-methylpyridin-2-yl)-2,3-dihydro-1h-pyrazol-4-yl]-1,5-naphthyridine | Human | 2096 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wot | A | A | 4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amine | Human | 2120 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wot | A | B | 4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amine | Human | 2092 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wou | A | | 4-({4-[(2,6-dimethylpyridin-3-yl)oxy]pyridin-2-yl}amino)benzenesulfonamide | Human | 2125 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | A | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2127 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | B | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2128 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | C | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2104 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | D | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2107 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | E | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2097 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | A | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2118 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | B | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2108 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | C | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2130 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | D | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2132 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | E | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2098 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3gxl | A | | n-1h-indazol-5-yl-2-(6-methylpyridin-2-yl)quinazolin-4-amine | Human | 2116 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3hmm | A | | 2-(6-methylpyridin-2-yl)-n-pyridin-4-ylquinazolin-4-amine | Human | 2111 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | A | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2112 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | B | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2106 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | C | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2093 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | D | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2119 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | E | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2105 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3tzm | A | A | 4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamide | Human | 2095 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3tzm | A | B | 4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamide | Human | 2110 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x0m | A | A | 4-aminopyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2122 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x0m | A | B | 4-aminopyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2121 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2f | A | A | 4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 6207 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2f | A | B | 4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 6208 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2g | A | A | 4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2123 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2g | A | B | 4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2114 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2j | A | A | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2124 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2j | A | B | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2115 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2k | A | A | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2135 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2k | A | B | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2101 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2n | A | A | - | Human | 2129 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2n | A | B | - | Human | 2109 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8s | A | A | - | Human | 6619 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8s | A | B | - | Human | 6609 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8t | A | A | - | Human | 6608 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8t | A | B | - | Human | 6613 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8u | A | | - | Human | 6616 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8w | A | A | staurosporine | Human | 6611 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8w | A | B | staurosporine | Human | 6614 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8x | A | A | staurosporine | Human | 6615 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8x | A | B | staurosporine | Human | 6617 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8z | A | A | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6618 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8z | A | B | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6612 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e90 | A | A | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6610 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e90 | A | B | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6607 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5fri | A | A | n-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamide | Human | 6894 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5fri | A | B | n-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamide | Human | 6893 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qik | A | A | n-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10657 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qik | A | B | n-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10662 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qil | A | A | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10659 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qil | A | B | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10660 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qim | A | A | n-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10658 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qim | A | B | n-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10661 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qtz | A | A | 6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridine | Human | 11965 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qtz | A | B | 6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridine | Human | 11966 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qu0 | A | A | 6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrile | Human | 11967 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qu0 | A | B | 6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrile | Human | 11964 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5usq | A | A | n-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amine | Human | 7558 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5usq | A | B | n-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amine | Human | 7557 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 6b8y | A | A | n-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9553 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 6b8y | A | B | n-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9552 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e8v | A | A | - | Human | 6626 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e8v | A | B | - | Human | 6622 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e8y | A | | staurosporine | Human | 6627 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e91 | A | | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6625 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e92 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 6624 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e92 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 6623 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5qin | A | A | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10664 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5qin | A | B | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10663 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 7dv6 | A | A | 5-[(3s)-5,5-dimethyloxolan-3-yl]-6-methoxy-3-(2-methoxypyridin-4-yl)pyrazolo[1,5-a]pyrimidine | Human | 13629 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 7dv6 | A | B | 5-[(3s)-5,5-dimethyloxolan-3-yl]-6-methoxy-3-(2-methoxypyridin-4-yl)pyrazolo[1,5-a]pyrimidine | Human | 13628 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 8ygz | A | A | - | Human | 15262 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 8ygz | A | B | - | Human | 15263 | |
| TLK2 | TLK | Other | 5o0y | A | | phosphothiophosphoric acid-adenylate ester | Human | 9943 | |
| TNIK | STE20 | STE | 2x7f | A | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1943 | |
| TNIK | STE20 | STE | 2x7f | A | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1951 | |
| TNIK | STE20 | STE | 2x7f | B | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1950 | |
| TNIK | STE20 | STE | 2x7f | B | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1947 | |
| TNIK | STE20 | STE | 2x7f | C | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1942 | |
| TNIK | STE20 | STE | 2x7f | C | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1948 | |
| TNIK | STE20 | STE | 2x7f | D | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1944 | |
| TNIK | STE20 | STE | 2x7f | D | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1945 | |
| TNIK | STE20 | STE | 2x7f | E | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1946 | |
| TNIK | STE20 | STE | 2x7f | E | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 1949 | |
| TNIK | STE20 | STE | 5ax9 | A | | 4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrile | Human | 6887 | |
| TNIK | STE20 | STE | 5ax9 | B | | 4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrile | Human | 6892 | |
| TNIK | STE20 | STE | 5ax9 | C | | 4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrile | Human | 6889 | |
| TNIK | STE20 | STE | 5cwz | A | | - | Human | 6891 | |
| TNIK | STE20 | STE | 5cwz | B | | - | Human | 6890 | |
| TNIK | STE20 | STE | 5cwz | C | | - | Human | 6888 | |
| TNIK | STE20 | STE | 5d7a | A | | cis-4-{[2-(1h-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanol | Human | 6963 | |
| TNIK | STE20 | STE | 5d7a | B | | cis-4-{[2-(1h-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanol | Human | 6964 | |
| TNIK | STE20 | STE | 5d7a | C | | cis-4-{[2-(1h-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanol | Human | 6965 | |
| TNIK | STE20 | STE | 6ra5 | A | | 5-bromanyl-2-(2-fluoranylpyridin-4-yl)-1,7-naphthyridin-8-amine | Human | 12238 | |
| TNIK | STE20 | STE | 6ra5 | B | | - | Human | 12237 | |
| TNIK | STE20 | STE | 6ra7 | A | A | 2-[8-azanyl-2-(2-fluoranylpyridin-4-yl)-1,7-naphthyridin-5-yl]propan-2-ol | Human | 11801 | |
| TNIK | STE20 | STE | 6ra7 | A | B | 2-[8-azanyl-2-(2-fluoranylpyridin-4-yl)-1,7-naphthyridin-5-yl]propan-2-ol | Human | 11800 | |
| TNIK | STE20 | STE | 7xzq | A | | - | Human | 14474 | |
| TNIK | STE20 | STE | 7xzr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 14476 | |
| TNIK | STE20 | STE | 7xzr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 14475 | |
| TNIK | STE20 | STE | 8wm0 | A | A | adenosine | Human | 15232 | |
| TNIK | STE20 | STE | 8wm0 | A | B | adenosine | Human | 15231 | |
| TNIK | STE20 | STE | 8x88 | A | | - | Human | 15060 | |
| TNK2 (ACK) | Ack | TK | 1u46 | A | | - | Human | 3411 | |
| TNK2 (ACK) | Ack | TK | 1u46 | B | | - | Human | 3408 | |
| TNK2 (ACK) | Ack | TK | 1u4d | A | | debromohymenialdisine | Human | 3398 | |
| TNK2 (ACK) | Ack | TK | 1u4d | B | | debromohymenialdisine | Human | 3392 | |
| TNK2 (ACK) | Ack | TK | 1u54 | A | | phosphomethylphosphonic acid adenylate ester | Human | 3409 | |
| TNK2 (ACK) | Ack | TK | 1u54 | B | | phosphomethylphosphonic acid adenylate ester | Human | 3397 | |
| TNK2 (ACK) | Ack | TK | 3eqp | A | | n-(2,6-dimethylphenyl)-4-(2-ethoxyphenoxy)-2-({4-[4-(2-hydroxyethyl)piperazin-1-yl]phenyl}amino)pyrimidine-5-carboxamide | Human | 3403 | |
| TNK2 (ACK) | Ack | TK | 3eqp | B | | n-(2,6-dimethylphenyl)-4-(2-ethoxyphenoxy)-2-({4-[4-(2-hydroxyethyl)piperazin-1-yl]phenyl}amino)pyrimidine-5-carboxamide | Human | 3402 | |
| TNK2 (ACK) | Ack | TK | 3eqr | A | | n~3~-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl)-n~6~-(4-piperazin-1-ylphenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,6-diamine | Human | 3395 | |
| TNK2 (ACK) | Ack | TK | 3eqr | B | | n~3~-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl)-n~6~-(4-piperazin-1-ylphenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,6-diamine | Human | 3406 | |
| TNK2 (ACK) | Ack | TK | 4ewh | A | | 6-{4-[2-(dimethylamino)ethoxy]phenyl}-n-(1,3-dithiolan-2-ylmethyl)-5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 3410 | |
| TNK2 (ACK) | Ack | TK | 4ewh | B | | 6-{4-[2-(dimethylamino)ethoxy]phenyl}-n-(1,3-dithiolan-2-ylmethyl)-5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 3405 | |
| TNK2 (ACK) | Ack | TK | 4hzr | A | A | - | Human | 3394 | |
| TNK2 (ACK) | Ack | TK | 4hzr | A | B | - | Human | 3399 | |
| TNK2 (ACK) | Ack | TK | 4hzr | B | A | - | Human | 3396 | |
| TNK2 (ACK) | Ack | TK | 4hzr | B | B | - | Human | 3391 | |
| TNK2 (ACK) | Ack | TK | 4hzs | A | | - | Human | 3407 | |
| TNK2 (ACK) | Ack | TK | 4hzs | B | | - | Human | 3400 | |
| TNK2 (ACK) | Ack | TK | 4hzs | C | | - | Human | 3393 | |
| TNK2 (ACK) | Ack | TK | 4hzs | D | | - | Human | 3404 | |
| TNK2 (ACK) | Ack | TK | 4id7 | A | | cis-3-[8-amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]cyclobutanol | Human | 3401 | |
| TNK2 (ACK) | Ack | TK | 5zxb | A | A | n-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | 10492 | |
| TNK2 (ACK) | Ack | TK | 5zxb | A | B | n-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | 10494 | |
| TNK2 (ACK) | Ack | TK | 5zxb | B | A | n-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | 10493 | |
| TNK2 (ACK) | Ack | TK | 5zxb | B | B | n-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamide | Human | 10495 | |
| TNK2 (ACK) | Ack | TK | 6vqm | A | | 2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6h-pyrimido[5,4-d][1,3]benzodiazepin-6-one | Human | 13289 | |
| TNK2 (ACK) | Ack | TK | 6vqm | B | | 2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6h-pyrimido[5,4-d][1,3]benzodiazepin-6-one | Human | 13290 | |
| TNK2 (ACK) | Ack | TK | 7kp6 | A | A | 5-chloro-n~2~-[4-(4-methylpiperazin-1-yl)phenyl]-n~4~-{[(2r)-oxolan-2-yl]methyl}pyrimidine-2,4-diamine | Human | 14104 | |
| TNK2 (ACK) | Ack | TK | 7kp6 | A | B | 5-chloro-n~2~-[4-(4-methylpiperazin-1-yl)phenyl]-n~4~-{[(2r)-oxolan-2-yl]methyl}pyrimidine-2,4-diamine | Human | 14103 | |
| TNK2 (ACK) | Ack | TK | 8fe9 | A | | n-[(1s)-1-benzyl-2-[(6-chloro-2-oxo-1h-quinolin-4-yl)methylamino]-2-oxo-ethyl]-4-hydroxy-2-oxo-1h-quinoline-6-carbo | Human | 14676 | |
| TNK2 (ACK) | Ack | TK | 8hmt | A | A | 6-(2-bromophenyl)-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[[(2s)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-7-one | Human | 15009 | |
| TNK2 (ACK) | Ack | TK | 8hmt | A | B | 6-(2-bromophenyl)-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[[(2s)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-7-one | Human | 15010 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | A | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6068 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | A | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6062 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | B | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6065 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | B | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6063 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | C | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6069 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | C | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6067 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | D | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6066 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | D | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6074 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | A | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6059 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | A | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6071 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | B | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6061 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | B | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6060 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | C | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6070 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | C | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6073 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | D | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6072 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | D | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6064 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | A | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9791 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | A | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9800 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | A | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9798 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | B | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9802 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | B | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9794 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | B | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9797 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | C | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9799 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | C | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9793 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | C | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9796 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | D | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9792 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | D | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9801 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | D | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9795 | |
| TNNI3K (HH498) | MLK | TKL | 7mgj | A | | n-methyl-4-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]pyridine-2-carboxamide | Human | 13969 | |
| TNNI3K (HH498) | MLK | TKL | 7mgk | A | A | n-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | 13968 | |
| TNNI3K (HH498) | MLK | TKL | 7mgk | A | B | n-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | 13970 | |
| TP53RK (PRPK) | Bud32 | Other | 6wqx | C | | phosphoaminophosphonic acid-adenylate ester | Human | 13338 | |
| TP53RK (PRPK) | Bud32 | Other | 6wqx | D | | phosphoaminophosphonic acid-adenylate ester | Human | 13339 | |
| TP53RK (PRPK) | Bud32 | Other | 7sza | A | A | 4-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dione | Human | 14597 | |
| TP53RK (PRPK) | Bud32 | Other | 7sza | A | B | 4-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dione | Human | 14599 | |
| TP53RK (PRPK) | Bud32 | Other | 7szb | A | | 5-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dione | Human | 14598 | |
| TP53RK (PRPK) | Bud32 | Other | 7szc | A | | 4-hydroxy-2-[(3r)-3-methyl-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dione | Human | 14559 | |
| TP53RK (PRPK) | Bud32 | Other | 7szd | A | | 2-[(3r)-3-methyl-2,6-dioxopiperidin-3-yl]-1,3-dioxo-2,3-dihydro-1h-isoindole-5-carboxylic acid | Human | 14558 | |
| TRIB1 (Trb1) | Trbl | CAMK | 5cek | A | | - | Human | 6241 | |
| TRIB1 (Trb1) | Trbl | CAMK | 5cem | A | A | - | Human | 6242 | |
| TRIB1 (Trb1) | Trbl | CAMK | 5cem | A | B | - | Human | 6243 | |
| TRIB1 (Trb1) | Trbl | CAMK | 6dc0 | A | A | - | Human | 10622 | |
| TRIB1 (Trb1) | Trbl | CAMK | 6dc0 | A | B | - | Human | 10623 | |
| TRIB1 (Trb1) | Trbl | CAMK | 6dc0 | B | A | - | Human | 10620 | |
| TRIB1 (Trb1) | Trbl | CAMK | 6dc0 | B | B | - | Human | 10621 | |
| TRIB2 (Trb2) | Trbl | CAMK | 7upm | A | | - | Human | 14365 | |
| TRRAP | PIKK | Atypical | 8h7g | A | | - | Human | 14556 | |
| TRRAP | PIKK | Atypical | 8qri | A | | - | Human | 15322 | |
| TRRAP | PIKK | Atypical | 8xvg | A | A | adenosine-5'-diphosphate | Human | 15321 | |
| TRRAP | PIKK | Atypical | 8xvg | A | B | adenosine-5'-diphosphate | Human | 15323 | |
| TTBK1 | TTBK | CK1 | 4btj | A | | adenosine-5'-diphosphate | Human | 769 | |
| TTBK1 | TTBK | CK1 | 4btj | B | | adenosine-5'-triphosphate | Human | 767 | |
| TTBK1 | TTBK | CK1 | 4btk | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 771 | |
| TTBK1 | TTBK | CK1 | 4btm | A | | methyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoate | Human | 772 | |
| TTBK1 | TTBK | CK1 | 4btm | B | | methyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoate | Human | 774 | |
| TTBK1 | TTBK | CK1 | 4nfm | A | | - | Human | 768 | |
| TTBK1 | TTBK | CK1 | 4nfn | A | A | 3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenol | Human | 773 | |
| TTBK1 | TTBK | CK1 | 4nfn | A | B | 3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenol | Human | 770 | |
| TTBK1 | TTBK | CK1 | 7jxx | A | A | 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol | Human | 13579 | |
| TTBK1 | TTBK | CK1 | 7jxx | A | B | 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol | Human | 13578 | |
| TTBK1 | TTBK | CK1 | 7jxy | A | | (3s)-1-[1-(2-aminopyrimidin-4-yl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-methylpent-1-yn-3-ol | Human | 13580 | |
| TTBK1 | TTBK | CK1 | 7q8v | A | | ~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14133 | |
| TTBK1 | TTBK | CK1 | 7q8w | A | A | ~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14134 | |
| TTBK1 | TTBK | CK1 | 7q8w | A | B | ~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14135 | |
| TTBK1 | TTBK | CK1 | 7qhw | A | | ~{n}-[4-(4-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14477 | |
| TTBK1 | TTBK | CK1 | 7zhn | A | A | 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol | Human | 14721 | |
| TTBK1 | TTBK | CK1 | 7zhn | A | B | 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol | Human | 14717 | |
| TTBK1 | TTBK | CK1 | 7zho | A | A | 4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-ol | Human | 14718 | |
| TTBK1 | TTBK | CK1 | 7zho | A | B | 4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-ol | Human | 14722 | |
| TTBK1 | TTBK | CK1 | 7zhp | A | A | 1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-ol | Human | 14724 | |
| TTBK1 | TTBK | CK1 | 7zhp | A | B | 1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-ol | Human | 14719 | |
| TTBK1 | TTBK | CK1 | 7zhq | A | A | (3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-ol | Human | 14720 | |
| TTBK1 | TTBK | CK1 | 7zhq | A | B | (3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-ol | Human | 14723 | |
| TTBK1 | TTBK | CK1 | 8xpz | A | | - | Human | 15163 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12046 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12048 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12049 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12047 | |
| TTBK2 | TTBK | CK1 | 6vrf | A | A | adenosine-5'-diphosphate | Human | 12344 | |
| TTBK2 | TTBK | CK1 | 6vrf | A | B | adenosine-5'-diphosphate | Human | 12343 | |
| TTBK2 | TTBK | CK1 | 6vrf | B | A | adenosine-5'-diphosphate | Human | 12345 | |
| TTBK2 | TTBK | CK1 | 6vrf | B | B | adenosine-5'-diphosphate | Human | 12342 | |
| TTBK2 | TTBK | CK1 | 7q8y | A | A | ~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14141 | |
| TTBK2 | TTBK | CK1 | 7q8y | A | B | ~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14138 | |
| TTBK2 | TTBK | CK1 | 7q8z | A | A | ~{n}-(4-phenoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14142 | |
| TTBK2 | TTBK | CK1 | 7q8z | A | B | ~{n}-(4-phenoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14140 | |
| TTBK2 | TTBK | CK1 | 7q90 | A | A | ~{n}-[4-(4-methoxyphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14139 | |
| TTBK2 | TTBK | CK1 | 7q90 | A | B | ~{n}-[4-(4-methoxyphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14143 | |
| TTK | TTK | Other | 2x9e | A | | n-(2,6-diethylphenyl)-1-methyl-8-({4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(trifluoromethoxy)phenyl}amino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4729 | |
| TTK | TTK | Other | 2zmc | A | | - | Human | 4696 | |
| TTK | TTK | Other | 2zmd | A | | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | 4731 | |
| TTK | TTK | Other | 3cek | A | | - | Human | 4716 | |
| TTK | TTK | Other | 3dbq | A | | - | Human | 4710 | |
| TTK | TTK | Other | 3gfw | A | | 1-(4-(4-(2-(isopropylsulfonyl)phenylamino)-1h-pyrrolo[2,3-b]pyridin-6-ylamino)-3-methoxyphenyl)piperidin-4-ol | Human | 4714 | |
| TTK | TTK | Other | 3h9f | A | A | 9-cyclopentyl-2-(4-(4-hydroxypiperidin-1-yl)-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5h-pyrimido[4,5-b][1,4]diazepin-6(7h)-one | Human | 4701 | |
| TTK | TTK | Other | 3h9f | A | B | 9-cyclopentyl-2-(4-(4-hydroxypiperidin-1-yl)-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5h-pyrimido[4,5-b][1,4]diazepin-6(7h)-one | Human | 4712 | |
| TTK | TTK | Other | 3hmn | A | | adenosine-5'-triphosphate | Human | 4719 | |
| TTK | TTK | Other | 3hmo | A | | staurosporine | Human | 4707 | |
| TTK | TTK | Other | 3hmp | A | | 7-chloro-n-(cyclopropylmethyl)quinazolin-4-amine | Human | 4728 | |
| TTK | TTK | Other | 3vqu | A | | 4-[(4-amino-5-cyano-6-ethoxypyridin-2-yl)amino]benzamide | Human | 4718 | |
| TTK | TTK | Other | 3w1f | A | | 5-[5-ethoxy-6-(1-methyl-1h-pyrazol-4-yl)-1h-indazol-3-yl]-2-methylbenzenesulfonamide | Human | 4722 | |
| TTK | TTK | Other | 3wyx | A | | 6-{[3-(cyanomethoxy)-4-(1-methyl-1h-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrile | Human | 4721 | |
| TTK | TTK | Other | 3wyy | A | | (2e)-3-[4-({4-amino-5-cyano-6-[(3s,5s,7s)-tricyclo[3.3.1.1~3,7~]dec-1-ylamino]pyridin-2-yl}amino)-2-(cyanomethoxy)phenyl]-n-(2-methoxyethyl)prop-2-enamide | Human | 4711 | |
| TTK | TTK | Other | 3wzj | A | | 4-{6-(cyclohexylamino)-8-[(tetrahydro-2h-pyran-4-ylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}-n-cyclopropylbenzamide | Human | 4704 | |
| TTK | TTK | Other | 3wzk | A | | n-cyclopropyl-4-{8-[(thiophen-2-ylmethyl)amino]imidazo[1,2-a]pyrazin-3-yl}benzamide | Human | 4703 | |
| TTK | TTK | Other | 4bhz | A | | thieno[2,3-c][2,6]naphthyridine | Human | 4709 | |
| TTK | TTK | Other | 4bi0 | A | | 5h-pyrimido[5,4-b]indole | Human | 4702 | |
| TTK | TTK | Other | 4bi1 | A | | thieno[3,2-c][2,6]naphthyridine | Human | 4699 | |
| TTK | TTK | Other | 4bi2 | A | | thieno[2,3-c][2,7]naphthyridine | Human | 4700 | |
| TTK | TTK | Other | 4c4e | A | A | n-(3,4-dimethoxyphenyl)-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | 4708 | |
| TTK | TTK | Other | 4c4e | A | B | - | Human | 4726 | |
| TTK | TTK | Other | 4c4f | A | | n-(2-methoxyphenyl)-2-(1,3-oxazol-5-yl)-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | 4715 | |
| TTK | TTK | Other | 4c4g | A | | tert-butyl 6-((2-chloro-4-(dimethylcarbamoyl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | 4697 | |
| TTK | TTK | Other | 4c4h | A | | tert-butyl 6-((2-chloro-4-(dimethylcarbamoyl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | 4725 | |
| TTK | TTK | Other | 4c4i | A | | tert-butyl 6-{[2-chloro-4-(dimethylcarbamoyl)phenyl]amino}-2-(1,3-oxazol-5-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | 4698 | |
| TTK | TTK | Other | 4c4j | A | | tert-butyl 6-{[2-chloro-4-(1-methyl-1h-imidazol-5-yl)phenyl]amino}-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | 4723 | |
| TTK | TTK | Other | 4cv8 | A | | 3-amino-5-(1-methyl-1h-pyrazol-4-yl)pyridin-2(1h)-one | Human | 4706 | |
| TTK | TTK | Other | 4cv9 | A | | 4-(4-methylpiperazin-1-yl)-n-(2-oxo-5-(pyridin-4-yl)-1,2-dihydropyridin-3-yl)benzamide | Human | 4705 | |
| TTK | TTK | Other | 4cva | A | | n-(6-oxo-1,6-dihydro-3,4'-bipyridin-5-yl)-4-(piperidin-1-yl)benzamide | Human | 4713 | |
| TTK | TTK | Other | 4d2s | A | | n-{2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]phenyl}-4-(1h-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 4717 | |
| TTK | TTK | Other | 4js8 | A | | 4-(cyclohexylmethoxy)-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-2h-indazole | Human | 4724 | |
| TTK | TTK | Other | 4jt3 | A | | 2-phenyl-n-[3-(3-sulfamoylphenyl)-2h-indazol-5-yl]acetamide | Human | 4727 | |
| TTK | TTK | Other | 4o6l | A | | n-[(1r)-1-(2-chlorophenyl)propyl]-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1h-indazole-5-carboxamide | Human | 4730 | |
| TTK | TTK | Other | 4o6l | B | | n-[(1r)-1-(2-chlorophenyl)propyl]-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1h-indazole-5-carboxamide | Human | 4720 | |
| TTK | TTK | Other | 4zeg | A | | n-cyclopropyl-2-methyl-4-(7-{[2-(morpholin-4-yl)ethyl]amino}-5-phenoxypyrazolo[1,5-a]pyrimidin-3-yl)benzamide | Human | 6574 | |
| TTK | TTK | Other | 5ap0 | A | | 9-cyclopentyl-2-[[2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-phenyl]amino]-7-methyl-7,9-dihydro-8h-purin-8-one | Human | 6101 | |
| TTK | TTK | Other | 5ap1 | A | | 6-{[3-(cyanomethoxy)-4-(1-methyl-1h-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrile | Human | 6103 | |
| TTK | TTK | Other | 5ap2 | A | | isopropyl 6-((4-(1,2-dimethyl-1h-imidazol-5-yl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | 6105 | |
| TTK | TTK | Other | 5ap3 | A | | 9-cyclopentyl-2-[[2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-phenyl]amino]-7-methyl-7,9-dihydro-8h-purin-8-one | Human | 6099 | |
| TTK | TTK | Other | 5ap4 | A | | 6-{[3-(cyanomethoxy)-4-(1-methyl-1h-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrile | Human | 6097 | |
| TTK | TTK | Other | 5ap5 | A | | tert-butyl 6-((2-chloro-4-(dimethylcarbamoyl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | 6104 | |
| TTK | TTK | Other | 5ap6 | A | A | isopropyl 6-((4-(1,2-dimethyl-1h-imidazol-5-yl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | 6098 | |
| TTK | TTK | Other | 5ap6 | A | B | isopropyl 6-((4-(1,2-dimethyl-1h-imidazol-5-yl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylate | Human | 6102 | |
| TTK | TTK | Other | 5ap7 | A | | n-(2,6-diethylphenyl)-1-methyl-8-({4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(trifluoromethoxy)phenyl}amino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 6100 | |
| TTK | TTK | Other | 5eh0 | A | | n2-(2-methoxy-4-(1-methyl-1h-pyrazol-4-yl)phenyl)-n8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamine | Human | 6850 | |
| TTK | TTK | Other | 5ehl | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 7256 | |
| TTK | TTK | Other | 5eho | A | | ~{n}8-cyclohexyl-~{n}2-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidine-2,8-diamine | Human | 7257 | |
| TTK | TTK | Other | 5ehy | A | | 4-(furan-3-yl)-3-phenyl-2~{h}-pyrazolo[4,3-c]pyridine | Human | 6556 | |
| TTK | TTK | Other | 5ei2 | A | | ~{n}-(2,4-dimethoxyphenyl)-8-(1-methylpyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine | Human | 6559 | |
| TTK | TTK | Other | 5ei6 | A | | ~{n}-(2,4-dimethoxyphenyl)-5-(1-methylpyrazol-4-yl)isoquinolin-3-amine | Human | 6558 | |
| TTK | TTK | Other | 5ei8 | A | | ~{n}-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(1-methylpyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amine | Human | 6557 | |
| TTK | TTK | Other | 5ljj | A | | n~6~-cyclohexyl-n~2~-(4-morpholin-4-ylphenyl)-9h-purine-2,6-diamine | Human | 7092 | |
| TTK | TTK | Other | 5mrb | A | | ~{n}-(2,6-diethylphenyl)-8-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 8270 | |
| TTK | TTK | Other | 5n7v | A | | ~{n}6-cyclohexyl-~{n}2-(2-methyl-4-morpholin-4-yl-phenyl)-7~{h}-purine-2,6-diamine | Human | 7978 | |
| TTK | TTK | Other | 5n84 | A | | ~{n}-cyclopropyl-4-[8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-3-yl]benzamide | Human | 7973 | |
| TTK | TTK | Other | 5n87 | A | | ~{n}-(2,6-diethylphenyl)-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamide | Human | 7977 | |
| TTK | TTK | Other | 5n93 | A | | 4-[[4-azanyl-6-(~{tert}-butylamino)-5-cyano-pyridin-2-yl]amino]benzamide | Human | 7976 | |
| TTK | TTK | Other | 5n9s | A | | (2~{r})-2-(4-fluorophenyl)-~{n}-[4-[2-[(2-methoxy-4-methylsulfonyl-phenyl)amino]-[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl]propanamide | Human | 7979 | |
| TTK | TTK | Other | 5na0 | A | | ~{n}-[3,5-diethyl-1-[2-[2-(2-methoxyethoxy)ethoxy]ethyl]pyrazol-4-yl]-2-[[2-methoxy-4-[4-(2-methoxyethanoyl)piperazin-1-yl]phenyl]amino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamide | Human | 7974 | |
| TTK | TTK | Other | 5nad | A | | bay 1217389 | Human | 7975 | |
| TTK | TTK | Other | 5ntt | A | A | n-(2,6-diethylphenyl)-1-methyl-8-({4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(trifluoromethoxy)phenyl}amino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 8268 | |
| TTK | TTK | Other | 5ntt | A | B | n-(2,6-diethylphenyl)-1-methyl-8-({4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(trifluoromethoxy)phenyl}amino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 8267 | |
| TTK | TTK | Other | 5o91 | A | | ~{n}-(2,6-diethylphenyl)-8-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 8269 | |
| TTK | TTK | Other | 6b4w | A | | 4-{[4-(cyclopentyloxy)-5-(2-methyl-1,3-benzoxazol-6-yl)-7h-pyrrolo[2,3-d]pyrimidin-2-yl]amino}-3-methoxy-n-methylbenzamide | Human | 8616 | |
| TTK | TTK | Other | 6gvj | A | | - | Human | 10847 | |
| TTK | TTK | Other | 6h3k | A | | ~{n}8-(2,2-dimethylpropyl)-~{n}2-[2-ethoxy-4-(4-methyl-1,2,4-triazol-3-yl)phenyl]-6-methyl-pyrido[3,4-d]pyrimidine-2,8-diamine | Human | 10571 | |
| TTK | TTK | Other | 6n6o | A | | 4-({5-chloro-4-[(cis-4-hydroxy-4-methylcyclohexyl)oxy]-7h-pyrrolo[2,3-d]pyrimidin-2-yl}amino)-n,n-dimethyl-3-{[(2r)-1,1,1-trifluoropropan-2-yl]oxy}benzamide | Human | 11240 | |
| TTK | TTK | Other | 6tn9 | A | A | [4-[[6-(3,5-dimethyl-4-oxidanyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]amino]phenyl]-morpholin-4-yl-methanone | Human | 12271 | |
| TTK | TTK | Other | 6tn9 | A | B | [4-[[6-(3,5-dimethyl-4-oxidanyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]amino]phenyl]-morpholin-4-yl-methanone | Human | 12269 | |
| TTK | TTK | Other | 6tnb | A | | (2~{r})-2-(4-fluorophenyl)-~{n}-[4-[2-[(2-methoxy-4-methylsulfonyl-phenyl)amino]-[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl]propanamide | Human | 12267 | |
| TTK | TTK | Other | 6tnc | A | | n-cyclopropyl-4-{8-[(thiophen-2-ylmethyl)amino]imidazo[1,2-a]pyrazin-3-yl}benzamide | Human | 12270 | |
| TTK | TTK | Other | 6tnd | A | A | bay 1217389 | Human | 12268 | |
| TTK | TTK | Other | 6tnd | A | B | bay 1217389 | Human | 12272 | |
| TTK | TTK | Other | 7chm | A | | 4-(cyclohexylamino)-2-[(2-methoxy-4-morpholin-4-ylcarbonyl-phenyl)amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13550 | |
| TTK | TTK | Other | 7chn | A | | 4-(cyclohexylamino)-2-[[2-methoxy-4-(2-oxidanylidenepyrrolidin-1-yl)phenyl]amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13552 | |
| TTK | TTK | Other | 7cht | A | | 2-[[2-methoxy-4-(2-oxidanylidenepyrrolidin-1-yl)phenyl]amino]-4-(oxan-4-ylamino)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13554 | |
| TTK | TTK | Other | 7cil | A | A | 4-(cyclohexylamino)-2-[(1-methylpyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13549 | |
| TTK | TTK | Other | 7cil | A | B | 4-(cyclohexylamino)-2-[(1-methylpyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13555 | |
| TTK | TTK | Other | 7cja | A | | 4-(cyclopentylmethylamino)-2-[[2-methoxy-4-(2-oxidanylidenepyrrolidin-1-yl)phenyl]amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13551 | |
| TTK | TTK | Other | 7clh | A | | 2-[[2-methoxy-4-(2-oxidanylidenepyrrolidin-1-yl)phenyl]amino]-4-(methylamino)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13553 | |
| TTK | TTK | Other | 7lqd | A | | ~{n}-(2,6-diethylphenyl)-2-[[4-(4-methylpiperazin-1-yl)-2-(propanoylamino)phenyl]amino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamide | Human | 14108 | |
| TTN | MLCK | CAMK | 1tki | A | | - | Human | 130 | |
| TTN | MLCK | CAMK | 1tki | B | | - | Human | 126 | |
| TTN | MLCK | CAMK | 4jnw | A | A | - | Human | 127 | |
| TTN | MLCK | CAMK | 4jnw | A | B | - | Human | 129 | |
| TTN | MLCK | CAMK | 4jnw | B | A | - | Human | 125 | |
| TTN | MLCK | CAMK | 4jnw | B | B | - | Human | 128 | |
| TTN | MLCK | CAMK | 6ygn | A | | - | Human | 13488 | |
| TTN | MLCK | CAMK | 6ygn | B | | - | Human | 13487 | |
| Tyk2 (TYK2) | JakA | TK | 4e1z | A | | n-[5-(4-{[(3-chlorophenyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]furan-2-carboxamide | Mouse | 5828 | |
| Tyk2 (TYK2) | JakA | TK | 4e20 | A | | n-[4-(3-amino-1h-indazol-5-yl)phenyl]-3-chlorobenzenesulfonamide | Mouse | 5827 | |
| TYK2 | JakA | TK | 3lxn | A | | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 3337 | |
| TYK2 | JakA | TK | 3lxp | A | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 3340 | |
| TYK2 | JakA | TK | 3nyx | A | A | n-{5-[(7-chloroquinolin-4-yl)sulfanyl]-1,3,4-thiadiazol-2-yl}thiophene-2-carboxamide | Human | 3341 | |
| TYK2 | JakA | TK | 3nyx | A | B | n-{5-[(7-chloroquinolin-4-yl)sulfanyl]-1,3,4-thiadiazol-2-yl}thiophene-2-carboxamide | Human | 3343 | |
| TYK2 | JakA | TK | 3nz0 | A | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 3342 | |
| TYK2 | JakA | TK | 3nz0 | A | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 3335 | |
| TYK2 | JakA | TK | 4gfo | A | A | 2,6-dichloro-n-(2-oxo-2,5-dihydropyridin-4-yl)benzamide | Human | 3336 | |
| TYK2 | JakA | TK | 4gfo | A | B | 2,6-dichloro-n-(2-oxo-2,5-dihydropyridin-4-yl)benzamide | Human | 3338 | |
| TYK2 | JakA | TK | 4gih | A | A | 2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamide | Human | 3339 | |
| TYK2 | JakA | TK | 4gih | A | B | 2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamide | Human | 3332 | |
| TYK2 | JakA | TK | 4gii | A | | 2,6-dichloro-4-cyano-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamide | Human | 3331 | |
| TYK2 | JakA | TK | 4gj2 | A | | 2,6-dichloro-n-[2-({[(1r,2r)-2-fluorocyclopropyl]carbonyl}amino)pyridin-4-yl]benzamide | Human | 3344 | |
| TYK2 | JakA | TK | 4gj3 | A | | 2,6-dichloro-4-cyano-n-[2-({[(1r,2r)-2-fluorocyclopropyl]carbonyl}amino)pyridin-4-yl]benzamide | Human | 3345 | |
| TYK2 | JakA | TK | 4gvj | A | | adenosine-5'-diphosphate | Human | 3334 | |
| TYK2 | JakA | TK | 4py1 | A | | 6-[(2,5-dimethoxyphenyl)sulfanyl]-3-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazine | Human | 3333 | |
| TYK2 | JakA | TK | 5f1z | A | A | 3-azanyl-5-[(2~{s})-3-methylbutan-2-yl]-7-[1-methyl-5-(2-oxidanylpropan-2-yl)pyrazol-3-yl]-1~{h}-pyrazolo[4,3-c]pyridin-4-one | Human | 6356 | |
| TYK2 | JakA | TK | 5f1z | A | B | 3-azanyl-5-[(2~{s})-3-methylbutan-2-yl]-7-[1-methyl-5-(2-oxidanylpropan-2-yl)pyrazol-3-yl]-1~{h}-pyrazolo[4,3-c]pyridin-4-one | Human | 6357 | |
| TYK2 | JakA | TK | 5f20 | A | | 3-azanyl-5-(2-methylphenyl)-7-(1-methylpyrazol-3-yl)-1~{h}-pyrazolo[4,3-c]pyridin-4-one | Human | 6355 | |
| TYK2 | JakA | TK | 5wal | A | A | n-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamide | Human | 8375 | |
| TYK2 | JakA | TK | 5wal | A | B | n-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamide | Human | 8374 | |
| TYK2 | JakA | TK | 6aam | A | | 4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamide | Human | 10489 | |
| TYK2 | JakA | TK | 6dbk | A | | 4-({4-[(1s,4s)-5-(cyanoacetyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyrimidin-2-yl}amino)-n-ethylbenzamide | Human | 10490 | |
| TYK2 | JakA | TK | 6dbm | A | A | [(1s)-2,2-difluorocyclopropyl][(1r,5s)-3-{2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octan-8-yl]methanone | Human | 10491 | |
| TYK2 | JakA | TK | 6dbm | A | B | [(1s)-2,2-difluorocyclopropyl][(1r,5s)-3-{2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octan-8-yl]methanone | Human | 10488 | |
| TYK2 | JakA | TK | 6ova | A | A | 6-({4-[(3s)-3-cyano-3-cyclopropyl-2-oxopyrrolidin-1-yl]pyridin-2-yl}amino)-n,n-dimethylpyridine-3-carboxamide | Human | 11980 | |
| TYK2 | JakA | TK | 6ova | A | B | 6-({4-[(3s)-3-cyano-3-cyclopropyl-2-oxopyrrolidin-1-yl]pyridin-2-yl}amino)-n,n-dimethylpyridine-3-carboxamide | Human | 11981 | |
| TYK2 | JakA | TK | 6vns | A | A | (1r,2r)-2-cyano-n-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropane-1-carboxamide | Human | 12139 | |
| TYK2 | JakA | TK | 6vns | A | B | (1r,2r)-2-cyano-n-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropane-1-carboxamide | Human | 12137 | |
| TYK2 | JakA | TK | 6vnv | A | | (1s,2s)-2-cyano-n-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropane-1-carboxamide | Human | 12138 | |
| TYK2 | JakA | TK | 6vnx | A | | (1s)-2,2-difluoro-n-[(1s,5r,6r)-3-{5-fluoro-2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-6-methyl-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropane-1-carboxamide | Human | 12136 | |
| TYK2 | JakA | TK | 6vny | A | | n-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropanecarboxamide | Human | 12135 | |
| TYK2 | JakA | TK | 6x8f | A | A | [3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrile | Human | 13157 | |
| TYK2 | JakA | TK | 6x8f | A | B | [3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrile | Human | 13159 | |
| TYK2 | JakA | TK | 6x8f | C | A | [3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrile | Human | 13156 | |
| TYK2 | JakA | TK | 6x8f | C | B | [3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrile | Human | 13158 | |
| TYK2 | JakA | TK | 6x8g | A | A | trans-3-(cyanomethyl)-3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}cyclobutane-1-carbonitrile | Human | 12992 | |
| TYK2 | JakA | TK | 6x8g | A | B | trans-3-(cyanomethyl)-3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}cyclobutane-1-carbonitrile | Human | 12993 | |
| TYK2 | JakA | TK | 7uyr | A | A | 2-(4-{[2-(2,6-difluorophenyl)-5-oxo-5h-pyrrolo[3,4-d]pyrimidin-4-yl]amino}phenyl)-n-ethylacetamide | Human | 14338 | |
| TYK2 | JakA | TK | 7uyr | A | B | 2-(4-{[2-(2,6-difluorophenyl)-5-oxo-5h-pyrrolo[3,4-d]pyrimidin-4-yl]amino}phenyl)-n-ethylacetamide | Human | 14335 | |
| TYK2 | JakA | TK | 7uys | A | A | 2-(2,6-difluorophenyl)-4-(4-methoxyanilino)-5h-pyrrolo[3,4-d]pyrimidin-5-one | Human | 14339 | |
| TYK2 | JakA | TK | 7uys | A | B | 2-(2,6-difluorophenyl)-4-(4-methoxyanilino)-5h-pyrrolo[3,4-d]pyrimidin-5-one | Human | 14336 | |
| TYK2 | JakA | TK | 7uyt | A | A | 6-{[(2m)-2-(2-chloro-6-fluorophenyl)-5-oxo-5h-pyrrolo[3,4-b]pyridin-4-yl]amino}-n-ethylpyridine-3-carboxamide | Human | 14342 | |
| TYK2 | JakA | TK | 7uyt | A | B | 6-{[(2m)-2-(2-chloro-6-fluorophenyl)-5-oxo-5h-pyrrolo[3,4-b]pyridin-4-yl]amino}-n-ethylpyridine-3-carboxamide | Human | 14340 | |
| TYK2 | JakA | TK | 7uyu | A | A | 2-(2,6-difluorophenyl)-4-[4-(pyrrolidine-1-carbonyl)anilino]-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 14337 | |
| TYK2 | JakA | TK | 7uyu | A | B | 2-(2,6-difluorophenyl)-4-[4-(pyrrolidine-1-carbonyl)anilino]-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 14341 | |
| TYK2-b | JakB | TK | 3zon | A | | 5-phenyl-2-ureidothiophene-3-carboxamide | Human | 2200 | |
| TYK2-b | JakB | TK | 4oli | A | | 2-chloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamide | Human | 2198 | |
| TYK2-b | JakB | TK | 4wov | A | A | 2-methoxy-n-({6-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]pyridin-2-yl}methyl)acetamide | Human | 2196 | |
| TYK2-b | JakB | TK | 4wov | A | B | 2-methoxy-n-({6-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]pyridin-2-yl}methyl)acetamide | Human | 2199 | |
| TYK2-b | JakB | TK | 4wov | B | A | 2-methoxy-n-({6-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]pyridin-2-yl}methyl)acetamide | Human | 2195 | |
| TYK2-b | JakB | TK | 4wov | B | B | 2-methoxy-n-({6-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]pyridin-2-yl}methyl)acetamide | Human | 2197 | |
| TYK2-b | JakB | TK | 5c01 | A | | unknown ligand | Human | 7222 | |
| TYK2-b | JakB | TK | 5c01 | B | | unknown ligand | Human | 7223 | |
| TYK2-b | JakB | TK | 5c03 | A | A | phosphothiophosphoric acid-adenylate ester | Human | 6043 | |
| TYK2-b | JakB | TK | 5c03 | A | B | phosphothiophosphoric acid-adenylate ester | Human | 6044 | |
| TYK2-b | JakB | TK | 5c03 | B | A | phosphothiophosphoric acid-adenylate ester | Human | 6042 | |
| TYK2-b | JakB | TK | 5c03 | B | B | phosphothiophosphoric acid-adenylate ester | Human | 6045 | |
| TYK2-b | JakB | TK | 5tkd | A | A | 6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide | Human | 7323 | |
| TYK2-b | JakB | TK | 5tkd | A | B | 6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide | Human | 7326 | |
| TYK2-b | JakB | TK | 5tkd | B | A | 6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide | Human | 7325 | |
| TYK2-b | JakB | TK | 5tkd | B | B | 6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide | Human | 7324 | |
| TYK2-b | JakB | TK | 6nsl | A | A | 6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide | Human | 11952 | |
| TYK2-b | JakB | TK | 6nsl | A | B | 6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide | Human | 11954 | |
| TYK2-b | JakB | TK | 6nsl | B | A | 6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide | Human | 11955 | |
| TYK2-b | JakB | TK | 6nsl | B | B | 6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamide | Human | 11953 | |
| TYK2-b | JakB | TK | 6nze | A | A | 4-[(2-carbamoylphenyl)amino]-6-[(5-fluoropyridin-2-yl)amino]-n-methylpyridine-3-carboxamide | Human | 11453 | |
| TYK2-b | JakB | TK | 6nze | A | B | 4-[(2-carbamoylphenyl)amino]-6-[(5-fluoropyridin-2-yl)amino]-n-methylpyridine-3-carboxamide | Human | 11444 | |
| TYK2-b | JakB | TK | 6nze | B | A | 4-[(2-carbamoylphenyl)amino]-6-[(5-fluoropyridin-2-yl)amino]-n-methylpyridine-3-carboxamide | Human | 11448 | |
| TYK2-b | JakB | TK | 6nze | B | B | 4-[(2-carbamoylphenyl)amino]-6-[(5-fluoropyridin-2-yl)amino]-n-methylpyridine-3-carboxamide | Human | 11443 | |
| TYK2-b | JakB | TK | 6nzf | A | A | 6-[(5-fluoropyridin-2-yl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamide | Human | 11446 | |
| TYK2-b | JakB | TK | 6nzf | A | B | 6-[(5-fluoropyridin-2-yl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamide | Human | 11449 | |
| TYK2-b | JakB | TK | 6nzf | B | A | 6-[(5-fluoropyridin-2-yl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamide | Human | 11451 | |
| TYK2-b | JakB | TK | 6nzf | B | B | 6-[(5-fluoropyridin-2-yl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamide | Human | 11445 | |
| TYK2-b | JakB | TK | 6nzh | A | A | 6-[(cyclopropanecarbonyl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamide | Human | 11450 | |
| TYK2-b | JakB | TK | 6nzh | A | B | 6-[(cyclopropanecarbonyl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamide | Human | 11442 | |
| TYK2-b | JakB | TK | 6nzh | B | A | 6-[(cyclopropanecarbonyl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamide | Human | 11447 | |
| TYK2-b | JakB | TK | 6nzh | B | B | 6-[(cyclopropanecarbonyl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamide | Human | 11452 | |
| TYK2-b | JakB | TK | 6nzp | A | A | 6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl]amino}-n-methylpyridazine-3-carboxamide | Human | 11504 | |
| TYK2-b | JakB | TK | 6nzp | A | B | 6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl]amino}-n-methylpyridazine-3-carboxamide | Human | 11501 | |
| TYK2-b | JakB | TK | 6nzp | B | A | 6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl]amino}-n-methylpyridazine-3-carboxamide | Human | 11496 | |
| TYK2-b | JakB | TK | 6nzp | B | B | 6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl]amino}-n-methylpyridazine-3-carboxamide | Human | 11497 | |
| TYK2-b | JakB | TK | 6nzq | A | A | 6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[(2-methoxy-3-{[(pyridin-2-yl)methyl]carbamoyl}phenyl)amino]-n-methylpyridine-3-carboxamide | Human | 11502 | |
| TYK2-b | JakB | TK | 6nzq | A | B | 6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[(2-methoxy-3-{[(pyridin-2-yl)methyl]carbamoyl}phenyl)amino]-n-methylpyridine-3-carboxamide | Human | 11499 | |
| TYK2-b | JakB | TK | 6nzq | B | A | 6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[(2-methoxy-3-{[(pyridin-2-yl)methyl]carbamoyl}phenyl)amino]-n-methylpyridine-3-carboxamide | Human | 11495 | |
| TYK2-b | JakB | TK | 6nzq | B | B | 6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[(2-methoxy-3-{[(pyridin-2-yl)methyl]carbamoyl}phenyl)amino]-n-methylpyridine-3-carboxamide | Human | 11506 | |
| TYK2-b | JakB | TK | 6nzr | A | A | n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}-6-[(pyridin-2-yl)amino]pyridazine-3-carboxamide | Human | 11505 | |
| TYK2-b | JakB | TK | 6nzr | A | B | n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}-6-[(pyridin-2-yl)amino]pyridazine-3-carboxamide | Human | 11503 | |
| TYK2-b | JakB | TK | 6nzr | B | A | n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}-6-[(pyridin-2-yl)amino]pyridazine-3-carboxamide | Human | 11498 | |
| TYK2-b | JakB | TK | 6nzr | B | B | n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}-6-[(pyridin-2-yl)amino]pyridazine-3-carboxamide | Human | 11500 | |
| TYK2-b | JakB | TK | 7ax4 | A | | 2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide | Human | 13499 | |
| TYK2-b | JakB | TK | 7ax4 | B | | 2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide | Human | 13498 | |
| TYK2-b | JakB | TK | 7k7o | A | A | 6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(pyrimidin-2-yl)phenyl]amino}-n-methylpyridazine-3-carboxamide | Human | 13835 | |
| TYK2-b | JakB | TK | 7k7o | A | B | 6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(pyrimidin-2-yl)phenyl]amino}-n-methylpyridazine-3-carboxamide | Human | 13837 | |
| TYK2-b | JakB | TK | 7k7q | A | A | 6-[(cyclopropanecarbonyl)amino]-4-({3-[6-(dimethylcarbamoyl)pyridazin-3-yl]-2-methoxyphenyl}amino)-n-methylpyridazine-3-carboxamide | Human | 13838 | |
| TYK2-b | JakB | TK | 7k7q | A | B | 6-[(cyclopropanecarbonyl)amino]-4-({3-[6-(dimethylcarbamoyl)pyridazin-3-yl]-2-methoxyphenyl}amino)-n-methylpyridazine-3-carboxamide | Human | 13836 | |
| TYK2-b | JakB | TK | 8s98 | A | A | (8s)-n-cyclopropyl-5-[(2-methoxypyridin-3-yl)amino]-7-(methylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 14849 | |
| TYK2-b | JakB | TK | 8s98 | A | B | (8s)-n-cyclopropyl-5-[(2-methoxypyridin-3-yl)amino]-7-(methylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 14846 | |
| TYK2-b | JakB | TK | 8s99 | A | A | (8s)-n-[(1r,2s)-2-fluorocyclopropyl]-5-{[(1m,2'm)-3'-fluoro-2-oxo-2h-[1,2'-bipyridin]-3-yl]amino}-7-(methylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 14847 | |
| TYK2-b | JakB | TK | 8s99 | A | B | (8s)-n-[(1r,2s)-2-fluorocyclopropyl]-5-{[(1m,2'm)-3'-fluoro-2-oxo-2h-[1,2'-bipyridin]-3-yl]amino}-7-(methylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 14850 | |
| TYK2-b | JakB | TK | 8s9a | A | A | (8s)-n-[(1r,2r)-2-methoxycyclobutyl]-7-(methylamino)-5-{[(1p,2'p)-2-oxo-2h-[1,2'-bipyridin]-3-yl]amino}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 14848 | |
| TYK2-b | JakB | TK | 8s9a | A | B | (8s)-n-[(1r,2r)-2-methoxycyclobutyl]-7-(methylamino)-5-{[(1p,2'p)-2-oxo-2h-[1,2'-bipyridin]-3-yl]amino}pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 14851 | |
| TYK2-b | JakB | TK | 8tb5 | A | A | n-{(3p)-3-[3-(dimethylsulfamoyl)phenyl]-1h-pyrrolo[2,3-c]pyridin-5-yl}cyclopropanecarboxamide | Human | 14958 | |
| TYK2-b | JakB | TK | 8tb5 | A | B | n-{(3p)-3-[3-(dimethylsulfamoyl)phenyl]-1h-pyrrolo[2,3-c]pyridin-5-yl}cyclopropanecarboxamide | Human | 14955 | |
| TYK2-b | JakB | TK | 8tb6 | A | A | n-[(3m)-3-{6-[(3r)-3-methoxyoxolan-3-yl]pyridin-2-yl}-1-methyl-1h-pyrrolo[2,3-c]pyridin-5-yl]urea | Human | 14956 | |
| TYK2-b | JakB | TK | 8tb6 | A | B | n-[(3m)-3-{6-[(3r)-3-methoxyoxolan-3-yl]pyridin-2-yl}-1-methyl-1h-pyrrolo[2,3-c]pyridin-5-yl]urea | Human | 14957 | |
| Tyro3 (TYRO3) | Axl | TK | 3qup | A | | (5-fluoro-1h-indol-2-yl)[(3r)-1'-[(3r)-piperidin-3-yl]spiro[indole-3,3'-pyrrolidin]-1(2h)-yl]methanone | Mouse | 5799 | |
| Tyro3 (TYRO3) | Axl | TK | 4feq | A | | 4-(cyclopentylamino)-n-[3-(2-oxopyrrolidin-1-yl)propyl]-2-{[2-(pyridin-4-yl)ethyl]amino}pyrimidine-5-carboxamide | Mouse | 5801 | |
| Tyro3 (TYRO3) | Axl | TK | 4ff8 | A | | 4-(cyclopentylamino)-2-[(2-methoxybenzyl)amino]-n-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | Mouse | 5800 | |
| ULK1 | ULK | Other | 4wno | A | A | n~2~-(4-aminophenyl)-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1881 | |
| ULK1 | ULK | Other | 4wno | A | B | n~2~-(4-aminophenyl)-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1876 | |
| ULK1 | ULK | Other | 4wnp | A | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1878 | |
| ULK1 | ULK | Other | 4wnp | A | B | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1874 | |
| ULK1 | ULK | Other | 4wnp | B | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1872 | |
| ULK1 | ULK | Other | 4wnp | B | B | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1879 | |
| ULK1 | ULK | Other | 4wnp | C | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1877 | |
| ULK1 | ULK | Other | 4wnp | C | B | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1873 | |
| ULK1 | ULK | Other | 4wnp | D | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1875 | |
| ULK1 | ULK | Other | 4wnp | D | B | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 1880 | |
| ULK1 | ULK | Other | 5ci7 | A | A | n-[3-({4-[(3-aminopropyl)amino]-5-iodopyrimidin-2-yl}amino)phenyl]pyrrolidine-1-carboxamide | Human | 5974 | |
| ULK1 | ULK | Other | 5ci7 | A | B | n-[3-({4-[(3-aminopropyl)amino]-5-iodopyrimidin-2-yl}amino)phenyl]pyrrolidine-1-carboxamide | Human | 5973 | |
| ULK1 | ULK | Other | 6mnh | A | A | n-[(2r)-3-methylbutan-2-yl]-1h-benzotriazole-6-carboxamide | Human | 10979 | |
| ULK1 | ULK | Other | 6mnh | A | B | n-[(2r)-3-methylbutan-2-yl]-1h-benzotriazole-6-carboxamide | Human | 10980 | |
| ULK1 | ULK | Other | 6qas | A | A | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 10930 | |
| ULK1 | ULK | Other | 6qas | A | B | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 10931 | |
| ULK1 | ULK | Other | 6qas | B | A | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 10932 | |
| ULK1 | ULK | Other | 6qas | B | B | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 10933 | |
| ULK1 | ULK | Other | 8sv9 | A | A | (4p)-4-[(2p)-2-(1,2,5,6-tetrahydropyridin-3-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n-(2,2,2-trifluoroethyl)thiophene-2-carboxamide | Human | 15222 | |
| ULK1 | ULK | Other | 8sv9 | A | B | (4p)-4-[(2p)-2-(1,2,5,6-tetrahydropyridin-3-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n-(2,2,2-trifluoroethyl)thiophene-2-carboxamide | Human | 15223 | |
| ULK2 | ULK | Other | 6qat | A | | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | 11227 | |
| ULK2 | ULK | Other | 6qat | B | | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | 11226 | |
| ULK2 | ULK | Other | 6qat | C | | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | 11232 | |
| ULK2 | ULK | Other | 6qat | D | | n-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamide | Human | 11230 | |
| ULK2 | ULK | Other | 6qau | A | A | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 11235 | |
| ULK2 | ULK | Other | 6qau | A | B | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 11225 | |
| ULK2 | ULK | Other | 6qau | B | A | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 11222 | |
| ULK2 | ULK | Other | 6qau | B | B | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 11236 | |
| ULK2 | ULK | Other | 6qau | C | A | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 11229 | |
| ULK2 | ULK | Other | 6qau | C | B | n-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamide | Human | 11233 | |
| ULK2 | ULK | Other | 6qav | A | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11231 | |
| ULK2 | ULK | Other | 6qav | A | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11239 | |
| ULK2 | ULK | Other | 6qav | B | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11224 | |
| ULK2 | ULK | Other | 6qav | B | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11237 | |
| ULK2 | ULK | Other | 6qav | C | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11223 | |
| ULK2 | ULK | Other | 6qav | C | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11228 | |
| ULK2 | ULK | Other | 6qav | D | A | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11234 | |
| ULK2 | ULK | Other | 6qav | D | B | ~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamide | Human | 11238 | |
| ULK2 | ULK | Other | 6yid | A | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 12385 | |
| ULK2 | ULK | Other | 6yid | A | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 12382 | |
| ULK2 | ULK | Other | 6yid | B | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 12381 | |
| ULK2 | ULK | Other | 6yid | B | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 12387 | |
| ULK2 | ULK | Other | 6yid | C | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 12384 | |
| ULK2 | ULK | Other | 6yid | C | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 12386 | |
| ULK2 | ULK | Other | 6yid | D | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 12388 | |
| ULK2 | ULK | Other | 6yid | D | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 12383 | |
| ULK3 | ULK | Other | 6fdy | U | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 10389 | |
| ULK3 | ULK | Other | 6fdz | U | | momelotinib | Human | 10390 | |
| ULK4 | ULK | Other | 6tsz | U | | phosphothiophosphoric acid-adenylate ester | Human | 11904 | |
| ULK4 | ULK | Other | 6u5l | A | A | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 11890 | |
| ULK4 | ULK | Other | 6u5l | A | B | n~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamine | Human | 11889 | |
| VRK1 | VRK | CK1 | 2kty | A | 1 | - | Human | 4877 | |
| VRK1 | VRK | CK1 | 2kty | A | 10 | - | Human | 4932 | |
| VRK1 | VRK | CK1 | 2kty | A | 11 | - | Human | 4917 | |
| VRK1 | VRK | CK1 | 2kty | A | 12 | - | Human | 4897 | |
| VRK1 | VRK | CK1 | 2kty | A | 13 | - | Human | 4922 | |
| VRK1 | VRK | CK1 | 2kty | A | 14 | - | Human | 4926 | |
| VRK1 | VRK | CK1 | 2kty | A | 15 | - | Human | 4953 | |
| VRK1 | VRK | CK1 | 2kty | A | 16 | - | Human | 4937 | |
| VRK1 | VRK | CK1 | 2kty | A | 17 | - | Human | 4920 | |
| VRK1 | VRK | CK1 | 2kty | A | 18 | - | Human | 4904 | |
| VRK1 | VRK | CK1 | 2kty | A | 19 | - | Human | 4875 | |
| VRK1 | VRK | CK1 | 2kty | A | 2 | - | Human | 4947 | |
| VRK1 | VRK | CK1 | 2kty | A | 20 | - | Human | 4890 | |
| VRK1 | VRK | CK1 | 2kty | A | 3 | - | Human | 4874 | |
| VRK1 | VRK | CK1 | 2kty | A | 4 | - | Human | 4938 | |
| VRK1 | VRK | CK1 | 2kty | A | 5 | - | Human | 4900 | |
| VRK1 | VRK | CK1 | 2kty | A | 6 | - | Human | 4929 | |
| VRK1 | VRK | CK1 | 2kty | A | 7 | - | Human | 4880 | |
| VRK1 | VRK | CK1 | 2kty | A | 8 | - | Human | 4939 | |
| VRK1 | VRK | CK1 | 2kty | A | 9 | - | Human | 4885 | |
| VRK1 | VRK | CK1 | 2kul | A | 1 | - | Human | 4919 | |
| VRK1 | VRK | CK1 | 2kul | A | 10 | - | Human | 4901 | |
| VRK1 | VRK | CK1 | 2kul | A | 11 | - | Human | 4923 | |
| VRK1 | VRK | CK1 | 2kul | A | 12 | - | Human | 4883 | |
| VRK1 | VRK | CK1 | 2kul | A | 13 | - | Human | 4941 | |
| VRK1 | VRK | CK1 | 2kul | A | 14 | - | Human | 4909 | |
| VRK1 | VRK | CK1 | 2kul | A | 15 | - | Human | 4876 | |
| VRK1 | VRK | CK1 | 2kul | A | 16 | - | Human | 4924 | |
| VRK1 | VRK | CK1 | 2kul | A | 17 | - | Human | 4893 | |
| VRK1 | VRK | CK1 | 2kul | A | 18 | - | Human | 4896 | |
| VRK1 | VRK | CK1 | 2kul | A | 19 | - | Human | 4906 | |
| VRK1 | VRK | CK1 | 2kul | A | 2 | - | Human | 4921 | |
| VRK1 | VRK | CK1 | 2kul | A | 20 | - | Human | 4915 | |
| VRK1 | VRK | CK1 | 2kul | A | 3 | - | Human | 4895 | |
| VRK1 | VRK | CK1 | 2kul | A | 4 | - | Human | 4948 | |
| VRK1 | VRK | CK1 | 2kul | A | 5 | - | Human | 4954 | |
| VRK1 | VRK | CK1 | 2kul | A | 6 | - | Human | 4949 | |
| VRK1 | VRK | CK1 | 2kul | A | 7 | - | Human | 4908 | |
| VRK1 | VRK | CK1 | 2kul | A | 8 | - | Human | 4887 | |
| VRK1 | VRK | CK1 | 2kul | A | 9 | - | Human | 4869 | |
| VRK1 | VRK | CK1 | 2lav | A | 1 | - | Human | 4930 | |
| VRK1 | VRK | CK1 | 2lav | A | 10 | - | Human | 4882 | |
| VRK1 | VRK | CK1 | 2lav | A | 11 | - | Human | 4916 | |
| VRK1 | VRK | CK1 | 2lav | A | 12 | - | Human | 4946 | |
| VRK1 | VRK | CK1 | 2lav | A | 13 | - | Human | 4872 | |
| VRK1 | VRK | CK1 | 2lav | A | 14 | - | Human | 4898 | |
| VRK1 | VRK | CK1 | 2lav | A | 15 | - | Human | 4931 | |
| VRK1 | VRK | CK1 | 2lav | A | 16 | - | Human | 4888 | |
| VRK1 | VRK | CK1 | 2lav | A | 17 | - | Human | 4950 | |
| VRK1 | VRK | CK1 | 2lav | A | 18 | - | Human | 4927 | |
| VRK1 | VRK | CK1 | 2lav | A | 19 | - | Human | 4940 | |
| VRK1 | VRK | CK1 | 2lav | A | 2 | - | Human | 4903 | |
| VRK1 | VRK | CK1 | 2lav | A | 20 | - | Human | 4933 | |
| VRK1 | VRK | CK1 | 2lav | A | 3 | - | Human | 4912 | |
| VRK1 | VRK | CK1 | 2lav | A | 4 | - | Human | 4884 | |
| VRK1 | VRK | CK1 | 2lav | A | 5 | - | Human | 4891 | |
| VRK1 | VRK | CK1 | 2lav | A | 6 | - | Human | 4871 | |
| VRK1 | VRK | CK1 | 2lav | A | 7 | - | Human | 4936 | |
| VRK1 | VRK | CK1 | 2lav | A | 8 | - | Human | 4881 | |
| VRK1 | VRK | CK1 | 2lav | A | 9 | - | Human | 4945 | |
| VRK1 | VRK | CK1 | 2rsv | A | 1 | - | Human | 4910 | |
| VRK1 | VRK | CK1 | 2rsv | A | 10 | - | Human | 4873 | |
| VRK1 | VRK | CK1 | 2rsv | A | 11 | - | Human | 4902 | |
| VRK1 | VRK | CK1 | 2rsv | A | 12 | - | Human | 4952 | |
| VRK1 | VRK | CK1 | 2rsv | A | 13 | - | Human | 4935 | |
| VRK1 | VRK | CK1 | 2rsv | A | 14 | - | Human | 4925 | |
| VRK1 | VRK | CK1 | 2rsv | A | 15 | - | Human | 4911 | |
| VRK1 | VRK | CK1 | 2rsv | A | 16 | - | Human | 4905 | |
| VRK1 | VRK | CK1 | 2rsv | A | 17 | - | Human | 4951 | |
| VRK1 | VRK | CK1 | 2rsv | A | 18 | - | Human | 4934 | |
| VRK1 | VRK | CK1 | 2rsv | A | 2 | - | Human | 4914 | |
| VRK1 | VRK | CK1 | 2rsv | A | 3 | - | Human | 4913 | |
| VRK1 | VRK | CK1 | 2rsv | A | 4 | - | Human | 4907 | |
| VRK1 | VRK | CK1 | 2rsv | A | 5 | - | Human | 4899 | |
| VRK1 | VRK | CK1 | 2rsv | A | 6 | - | Human | 4943 | |
| VRK1 | VRK | CK1 | 2rsv | A | 7 | - | Human | 4889 | |
| VRK1 | VRK | CK1 | 2rsv | A | 8 | - | Human | 4918 | |
| VRK1 | VRK | CK1 | 2rsv | A | 9 | - | Human | 4928 | |
| VRK1 | VRK | CK1 | 3op5 | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4870 | |
| VRK1 | VRK | CK1 | 3op5 | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4942 | |
| VRK1 | VRK | CK1 | 3op5 | B | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4894 | |
| VRK1 | VRK | CK1 | 3op5 | B | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4944 | |
| VRK1 | VRK | CK1 | 3op5 | C | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4886 | |
| VRK1 | VRK | CK1 | 3op5 | C | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4879 | |
| VRK1 | VRK | CK1 | 3op5 | D | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4878 | |
| VRK1 | VRK | CK1 | 3op5 | D | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4892 | |
| VRK1 | VRK | CK1 | 5ukf | A | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8030 | |
| VRK1 | VRK | CK1 | 5ukf | B | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8029 | |
| VRK1 | VRK | CK1 | 5ukf | C | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8027 | |
| VRK1 | VRK | CK1 | 5ukf | D | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8028 | |
| VRK1 | VRK | CK1 | 5uvf | A | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7521 | |
| VRK1 | VRK | CK1 | 5uvf | B | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7523 | |
| VRK1 | VRK | CK1 | 5uvf | C | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7520 | |
| VRK1 | VRK | CK1 | 5uvf | D | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7522 | |
| VRK1 | VRK | CK1 | 6ac9 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 10816 | |
| VRK1 | VRK | CK1 | 6ac9 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 10817 | |
| VRK1 | VRK | CK1 | 6ac9 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 10818 | |
| VRK1 | VRK | CK1 | 6ac9 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 10823 | |
| VRK1 | VRK | CK1 | 6ac9 | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 10822 | |
| VRK1 | VRK | CK1 | 6ac9 | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 10819 | |
| VRK1 | VRK | CK1 | 6ac9 | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 10821 | |
| VRK1 | VRK | CK1 | 6ac9 | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 10820 | |
| VRK1 | VRK | CK1 | 6bp0 | A | A | - | Human | 8744 | |
| VRK1 | VRK | CK1 | 6bp0 | A | B | - | Human | 8738 | |
| VRK1 | VRK | CK1 | 6bp0 | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8740 | |
| VRK1 | VRK | CK1 | 6bp0 | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8741 | |
| VRK1 | VRK | CK1 | 6bp0 | C | A | - | Human | 8743 | |
| VRK1 | VRK | CK1 | 6bp0 | C | B | - | Human | 8742 | |
| VRK1 | VRK | CK1 | 6bp0 | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8745 | |
| VRK1 | VRK | CK1 | 6bp0 | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8739 | |
| VRK1 | VRK | CK1 | 6bru | A | A | - | Human | 9085 | |
| VRK1 | VRK | CK1 | 6bru | A | B | - | Human | 9082 | |
| VRK1 | VRK | CK1 | 6bru | B | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9088 | |
| VRK1 | VRK | CK1 | 6bru | B | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9087 | |
| VRK1 | VRK | CK1 | 6bru | C | A | - | Human | 9089 | |
| VRK1 | VRK | CK1 | 6bru | C | B | - | Human | 9086 | |
| VRK1 | VRK | CK1 | 6bru | D | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9084 | |
| VRK1 | VRK | CK1 | 6bru | D | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9083 | |
| VRK1 | VRK | CK1 | 6btw | A | A | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9418 | |
| VRK1 | VRK | CK1 | 6btw | A | B | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9425 | |
| VRK1 | VRK | CK1 | 6btw | B | A | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9424 | |
| VRK1 | VRK | CK1 | 6btw | B | B | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9411 | |
| VRK1 | VRK | CK1 | 6btw | C | A | - | Human | 9419 | |
| VRK1 | VRK | CK1 | 6btw | C | B | - | Human | 9416 | |
| VRK1 | VRK | CK1 | 6btw | D | A | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9415 | |
| VRK1 | VRK | CK1 | 6btw | D | B | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9420 | |
| VRK1 | VRK | CK1 | 6bu6 | A | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9423 | |
| VRK1 | VRK | CK1 | 6bu6 | A | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9417 | |
| VRK1 | VRK | CK1 | 6bu6 | B | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9421 | |
| VRK1 | VRK | CK1 | 6bu6 | B | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9422 | |
| VRK1 | VRK | CK1 | 6bu6 | C | A | - | Human | 9412 | |
| VRK1 | VRK | CK1 | 6bu6 | C | B | - | Human | 9414 | |
| VRK1 | VRK | CK1 | 6bu6 | D | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9413 | |
| VRK1 | VRK | CK1 | 6bu6 | D | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9410 | |
| VRK1 | VRK | CK1 | 6cfm | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9723 | |
| VRK1 | VRK | CK1 | 6cfm | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9718 | |
| VRK1 | VRK | CK1 | 6cfm | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9724 | |
| VRK1 | VRK | CK1 | 6cfm | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9725 | |
| VRK1 | VRK | CK1 | 6cfm | C | A | - | Human | 9719 | |
| VRK1 | VRK | CK1 | 6cfm | C | B | - | Human | 9720 | |
| VRK1 | VRK | CK1 | 6cfm | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9721 | |
| VRK1 | VRK | CK1 | 6cfm | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9722 | |
| VRK1 | VRK | CK1 | 6cmm | A | A | - | Human | 9763 | |
| VRK1 | VRK | CK1 | 6cmm | A | B | - | Human | 9760 | |
| VRK1 | VRK | CK1 | 6cmm | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9766 | |
| VRK1 | VRK | CK1 | 6cmm | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9761 | |
| VRK1 | VRK | CK1 | 6cmm | C | A | - | Human | 9765 | |
| VRK1 | VRK | CK1 | 6cmm | C | B | - | Human | 9762 | |
| VRK1 | VRK | CK1 | 6cmm | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9764 | |
| VRK1 | VRK | CK1 | 6cmm | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9759 | |
| VRK1 | VRK | CK1 | 6cnx | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9815 | |
| VRK1 | VRK | CK1 | 6cnx | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9810 | |
| VRK1 | VRK | CK1 | 6cnx | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9803 | |
| VRK1 | VRK | CK1 | 6cnx | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9806 | |
| VRK1 | VRK | CK1 | 6cnx | C | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9805 | |
| VRK1 | VRK | CK1 | 6cnx | C | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9804 | |
| VRK1 | VRK | CK1 | 6cnx | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9814 | |
| VRK1 | VRK | CK1 | 6cnx | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9807 | |
| VRK1 | VRK | CK1 | 6cqh | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9774 | |
| VRK1 | VRK | CK1 | 6cqh | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9768 | |
| VRK1 | VRK | CK1 | 6cqh | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9769 | |
| VRK1 | VRK | CK1 | 6cqh | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9770 | |
| VRK1 | VRK | CK1 | 6cqh | C | A | - | Human | 9772 | |
| VRK1 | VRK | CK1 | 6cqh | C | B | - | Human | 9773 | |
| VRK1 | VRK | CK1 | 6cqh | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9771 | |
| VRK1 | VRK | CK1 | 6cqh | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9767 | |
| VRK1 | VRK | CK1 | 6csw | A | A | - | Human | 9818 | |
| VRK1 | VRK | CK1 | 6csw | A | B | - | Human | 9813 | |
| VRK1 | VRK | CK1 | 6csw | B | A | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9812 | |
| VRK1 | VRK | CK1 | 6csw | B | B | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9808 | |
| VRK1 | VRK | CK1 | 6csw | C | A | - | Human | 9816 | |
| VRK1 | VRK | CK1 | 6csw | C | B | - | Human | 9811 | |
| VRK1 | VRK | CK1 | 6csw | D | A | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9817 | |
| VRK1 | VRK | CK1 | 6csw | D | B | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9809 | |
| VRK1 | VRK | CK1 | 6dd4 | A | A | - | Human | 9935 | |
| VRK1 | VRK | CK1 | 6dd4 | A | B | - | Human | 9939 | |
| VRK1 | VRK | CK1 | 6dd4 | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9937 | |
| VRK1 | VRK | CK1 | 6dd4 | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9933 | |
| VRK1 | VRK | CK1 | 6dd4 | C | A | - | Human | 9940 | |
| VRK1 | VRK | CK1 | 6dd4 | C | B | - | Human | 9936 | |
| VRK1 | VRK | CK1 | 6dd4 | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9938 | |
| VRK1 | VRK | CK1 | 6dd4 | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9934 | |
| VRK1 | VRK | CK1 | 6npn | A | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11243 | |
| VRK1 | VRK | CK1 | 6npn | B | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11244 | |
| VRK1 | VRK | CK1 | 6npn | C | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11241 | |
| VRK1 | VRK | CK1 | 6npn | D | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11242 | |
| VRK1 | VRK | CK1 | 6vxu | B | | (7r)-8-(cyclopropylmethyl)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 13362 | |
| VRK1 | VRK | CK1 | 6vzh | A | | - | Human | 12057 | |
| VRK1 | VRK | CK1 | 6vzh | B | | (7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-one | Human | 12056 | |
| VRK1 | VRK | CK1 | 6vzh | C | | - | Human | 12058 | |
| VRK1 | VRK | CK1 | 6vzh | D | | (7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-one | Human | 12055 | |
| VRK1 | VRK | CK1 | 8v42 | A | A | - | Human | 15395 | |
| VRK1 | VRK | CK1 | 8v42 | A | B | - | Human | 15394 | |
| VRK2 | VRK | CK1 | 2v62 | A | A | - | Human | 2628 | |
| VRK2 | VRK | CK1 | 2v62 | A | B | - | Human | 2629 | |
| VRK2 | VRK | CK1 | 2v62 | B | A | - | Human | 2630 | |
| VRK2 | VRK | CK1 | 2v62 | B | B | - | Human | 2631 | |
| VRK2 | VRK | CK1 | 5uu1 | A | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7499 | |
| VRK2 | VRK | CK1 | 6ncg | A | | 4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamide | Human | 10852 | |
| VRK2 | VRK | CK1 | 6ncg | B | | 4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamide | Human | 10851 | |
| VRK2 | VRK | CK1 | 8q1z | A | A | 2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrile | Human | 14899 | |
| VRK2 | VRK | CK1 | 8q1z | A | B | 2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrile | Human | 14898 | |
| VRK3 | VRK | CK1 | 2jii | A | A | - | Human | 2939 | |
| VRK3 | VRK | CK1 | 2jii | A | B | - | Human | 2938 | |
| VRK3 | VRK | CK1 | 2jii | B | A | - | Human | 2936 | |
| VRK3 | VRK | CK1 | 2jii | B | B | - | Human | 2937 | |
| WEE1 (Wee1) | WEE | Other | 1x8b | A | | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 209 | |
| WEE1 (Wee1) | WEE | Other | 2in6 | A | | 3-(9-hydroxy-1,3-dioxo-4-phenyl-2,3-dihydropyrrolo[3,4-c]carbazol-6(1h)-yl)propanoic acid | Human | 207 | |
| WEE1 (Wee1) | WEE | Other | 2io6 | A | | 9-hydroxy-6-(3-hydroxypropyl)-4-(2-methoxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 214 | |
| WEE1 (Wee1) | WEE | Other | 2z2w | A | | n-[4-(2-chlorophenyl)-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-c]carbazol-9-yl]formamide | Human | 203 | |
| WEE1 (Wee1) | WEE | Other | 3bi6 | A | A | 4-(2-chlorophenyl)-9-hydroxy-6-methyl-1,3-dioxo-n-(2-pyrrolidin-1-ylethyl)pyrrolo[3,4-g]carbazole-8-carboxamide | Human | 213 | |
| WEE1 (Wee1) | WEE | Other | 3bi6 | A | B | 4-(2-chlorophenyl)-9-hydroxy-6-methyl-1,3-dioxo-n-(2-pyrrolidin-1-ylethyl)pyrrolo[3,4-g]carbazole-8-carboxamide | Human | 205 | |
| WEE1 (Wee1) | WEE | Other | 3biz | A | A | 4-(2-chlorophenyl)-8-[3-(dimethylamino)propoxy]-9-hydroxy-6-methylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 210 | |
| WEE1 (Wee1) | WEE | Other | 3biz | A | B | 4-(2-chlorophenyl)-8-[3-(dimethylamino)propoxy]-9-hydroxy-6-methylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 204 | |
| WEE1 (Wee1) | WEE | Other | 3cqe | A | A | 8-bromo-4-(2-chlorophenyl)-n-(2-hydroxyethyl)-6-methyl-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-e]indole-7-carboxamide | Human | 206 | |
| WEE1 (Wee1) | WEE | Other | 3cqe | A | B | 8-bromo-4-(2-chlorophenyl)-n-(2-hydroxyethyl)-6-methyl-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-e]indole-7-carboxamide | Human | 211 | |
| WEE1 (Wee1) | WEE | Other | 3cr0 | A | A | 4-(2-chlorophenyl)-8-(2-hydroxyethyl)-6-methylpyrrolo[3,4-e]indole-1,3(2h,6h)-dione | Human | 208 | |
| WEE1 (Wee1) | WEE | Other | 3cr0 | A | B | 4-(2-chlorophenyl)-8-(2-hydroxyethyl)-6-methylpyrrolo[3,4-e]indole-1,3(2h,6h)-dione | Human | 212 | |
| WEE1 (Wee1) | WEE | Other | 5v5y | A | | 1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 8328 | |
| WEE1 (Wee1) | WEE | Other | 5vc3 | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 8329 | |
| WEE1 (Wee1) | WEE | Other | 5vc4 | A | | 4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 8334 | |
| WEE1 (Wee1) | WEE | Other | 5vc5 | A | A | 6-(2,6-dichlorophenyl)-2-({4-[2-(diethylamino)ethoxy]phenyl}amino)-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 8332 | |
| WEE1 (Wee1) | WEE | Other | 5vc5 | A | B | 6-(2,6-dichlorophenyl)-2-({4-[2-(diethylamino)ethoxy]phenyl}amino)-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 8333 | |
| WEE1 (Wee1) | WEE | Other | 5vc6 | A | | n,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 8331 | |
| WEE1 (Wee1) | WEE | Other | 5vd2 | A | | n-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamide | Human | 8330 | |
| WEE1 (Wee1) | WEE | Other | 5vd4 | A | | 6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1-{6-[(1s)-2,2,2-trifluoro-1-hydroxyethyl]pyridin-2-yl}-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 9780 | |
| WEE1 (Wee1) | WEE | Other | 5vd5 | A | | 1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(morpholin-4-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 9778 | |
| WEE1 (Wee1) | WEE | Other | 5vd7 | A | | 6-{[3-fluoro-4-(4-methylpiperazin-1-yl)phenyl]amino}-1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 9782 | |
| WEE1 (Wee1) | WEE | Other | 5vd8 | A | | 6-{[3-chloro-4-(4-methylpiperazin-1-yl)phenyl]amino}-1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 9777 | |
| WEE1 (Wee1) | WEE | Other | 5vd9 | A | | 1-{6-[(1r)-1-hydroxyethyl]pyridin-2-yl}-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 9781 | |
| WEE1 (Wee1) | WEE | Other | 5vda | A | | 1-{6-[(1s)-1-hydroxyethyl]pyridin-2-yl}-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 9779 | |
| WEE1 (Wee1) | WEE | Other | 7n3u | A | | 1-[(7r)-7-ethyl-7-hydroxy-7h-cyclopenta[b]pyridin-2-yl]-6-[4-(4-methylpiperazin-1-yl)anilino]-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 13857 | |
| WEE1 (Wee1) | WEE | Other | 8bju | A | A | 2-(2-methoxyphenyl)-6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1-[6-(2-oxidanylpropan-2-yl)pyridin-2-yl]pyrazolo[3,4-d]pyrimidin-3-one | Human | 14755 | |
| WEE1 (Wee1) | WEE | Other | 8bju | A | B | 2-(2-methoxyphenyl)-6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1-[6-(2-oxidanylpropan-2-yl)pyridin-2-yl]pyrazolo[3,4-d]pyrimidin-3-one | Human | 14754 | |
| WEE2 (Wee1B) | WEE | Other | 5vdk | A | | 1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-one | Human | 8349 | |
| WNK1 (Wnk1) | WNK | Other | 4pwn | A | | - | Human | 1831 | |
| WNK1 (Wnk1) | WNK | Other | 5tf9 | A | | {2-[(4-chlorophenyl)methoxy]phenyl}{5-[2-(methylamino)-1,3-thiazol-4-yl]-2,3-dihydro-1h-indol-1-yl}methanone | Human | 7099 | |
| WNK1 (Wnk1) | WNK | Other | 5tf9 | B | | {2-[(4-chlorophenyl)methoxy]phenyl}{5-[2-(methylamino)-1,3-thiazol-4-yl]-2,3-dihydro-1h-indol-1-yl}methanone | Human | 7098 | |
| WNK1 (Wnk1) | WNK | Other | 5wdy | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 8326 | |
| WNK1 (Wnk1) | WNK | Other | 5wdy | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 8321 | |
| WNK1 (Wnk1) | WNK | Other | 5wdy | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 8323 | |
| WNK1 (Wnk1) | WNK | Other | 5wdy | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 8322 | |
| WNK1 (Wnk1) | WNK | Other | 5we8 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 8324 | |
| WNK1 (Wnk1) | WNK | Other | 5we8 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 8325 | |
| WNK1 (Wnk1) | WNK | Other | 5we8 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 8327 | |
| WNK1 (Wnk1) | WNK | Other | 5we8 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 8320 | |
| WNK3 (Wnk3) | WNK | Other | 5o1v | A | A | - | Human | 8157 | |
| WNK3 (Wnk3) | WNK | Other | 5o1v | A | B | - | Human | 8165 | |
| WNK3 (Wnk3) | WNK | Other | 5o1v | B | A | - | Human | 8152 | |
| WNK3 (Wnk3) | WNK | Other | 5o1v | B | B | - | Human | 8150 | |
| WNK3 (Wnk3) | WNK | Other | 5o21 | A | | - | Human | 8160 | |
| WNK3 (Wnk3) | WNK | Other | 5o21 | B | | - | Human | 8158 | |
| WNK3 (Wnk3) | WNK | Other | 5o23 | A | A | - | Human | 8151 | |
| WNK3 (Wnk3) | WNK | Other | 5o23 | A | B | - | Human | 8155 | |
| WNK3 (Wnk3) | WNK | Other | 5o23 | B | A | - | Human | 8159 | |
| WNK3 (Wnk3) | WNK | Other | 5o23 | B | B | - | Human | 8166 | |
| WNK3 (Wnk3) | WNK | Other | 5o26 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 8164 | |
| WNK3 (Wnk3) | WNK | Other | 5o26 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 8149 | |
| WNK3 (Wnk3) | WNK | Other | 5o26 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 8162 | |
| WNK3 (Wnk3) | WNK | Other | 5o26 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 8156 | |
| WNK3 (Wnk3) | WNK | Other | 5o2b | A | A | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 8163 | |
| WNK3 (Wnk3) | WNK | Other | 5o2b | A | B | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 8153 | |
| WNK3 (Wnk3) | WNK | Other | 5o2b | B | A | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 8154 | |
| WNK3 (Wnk3) | WNK | Other | 5o2b | B | B | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 8161 | |
| WNK3 (Wnk3) | WNK | Other | 5o2c | A | | - | Human | 8148 | |
| WNK3 (Wnk3) | WNK | Other | 8edh | A | | ethyl 1-(5,7-dimethoxy-4-methylquinolin-2-yl)piperidine-4-carboxylate | Human | 14631 | |
| ZAP70 | Syk | TK | 1u59 | A | A | staurosporine | Human | 2734 | |
| ZAP70 | Syk | TK | 1u59 | A | B | staurosporine | Human | 2733 | |
| ZAP70 | Syk | TK | 2ozo | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2735 | |
| ZAP70 | Syk | TK | 4k2r | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2732 | |
