Browse kinase structures

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetailsFile
Aak1 (AAK1)NAKOther7lvhAn-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse13820
Aak1 (AAK1)NAKOther7lviAA(2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamideMouse13822
Aak1 (AAK1)NAKOther7lviAB(2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamideMouse13821
Aak1 (AAK1)NAKOther7rj6AA5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineMouse14132
Aak1 (AAK1)NAKOther7rj6AB5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineMouse14131
Aak1 (AAK1)NAKOther7rj7AA2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrileMouse14128
Aak1 (AAK1)NAKOther7rj7AB2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrileMouse14129
Aak1 (AAK1)NAKOther7rj8AAn-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse14130
Aak1 (AAK1)NAKOther7rj8ABn-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse14127
AAK1NAKOther4wsqAAk-252aHuman3834
AAK1NAKOther4wsqABk-252aHuman3836
AAK1NAKOther4wsqBAk-252aHuman3833
AAK1NAKOther4wsqBBk-252aHuman3835
AAK1NAKOther5l4qAA~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6679
AAK1NAKOther5l4qAB~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6677
AAK1NAKOther5l4qBA~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6680
AAK1NAKOther5l4qBB~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6678
AAK1NAKOther5te0Amethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman7156
AAK1NAKOther8gmcA5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman14843
AAK1NAKOther8gmdA(5p)-3-({(8r)-5-[(4-aminopiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-[2-(propan-2-yl)-2h-tetrazol-5-yl]phenolHuman14844
Abl1 (ABL1)AblTK1fpuAn-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamideMouse5728
Abl1 (ABL1)AblTK1fpuBn-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamideMouse5705
Abl1 (ABL1)AblTK1iepA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5703
Abl1 (ABL1)AblTK1iepB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5727
Abl1 (ABL1)AblTK1m52A6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-oneMouse5720
Abl1 (ABL1)AblTK1m52B6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-oneMouse5715
Abl1 (ABL1)AblTK1opjA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5732
Abl1 (ABL1)AblTK1opjB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5736
Abl1 (ABL1)AblTK1opkA6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneMouse5709
Abl1 (ABL1)AblTK2hznA1-[4-(pyridin-4-yloxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaMouse5701
Abl1 (ABL1)AblTK2qohA5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamideMouse5707
Abl1 (ABL1)AblTK2qohB5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamideMouse5716
Abl1 (ABL1)AblTK2z60A5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamideMouse5735
Abl1 (ABL1)AblTK3dk3AA2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5726
Abl1 (ABL1)AblTK3dk3AB2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5729
Abl1 (ABL1)AblTK3dk3BA2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5712
Abl1 (ABL1)AblTK3dk3BB2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5737
Abl1 (ABL1)AblTK3dk6A2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5725
Abl1 (ABL1)AblTK3dk6B2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5718
Abl1 (ABL1)AblTK3dk7A2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5704
Abl1 (ABL1)AblTK3dk7B2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamideMouse5714
Abl1 (ABL1)AblTK3ik3A3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideMouse5731
Abl1 (ABL1)AblTK3ik3B3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideMouse5739
Abl1 (ABL1)AblTK3k5vAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5734
Abl1 (ABL1)AblTK3k5vAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5723
Abl1 (ABL1)AblTK3k5vBA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5710
Abl1 (ABL1)AblTK3k5vBB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5722
Abl1 (ABL1)AblTK3kf4An-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amineMouse5717
Abl1 (ABL1)AblTK3kf4Bn-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amineMouse5741
Abl1 (ABL1)AblTK3kfaA3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamideMouse5742
Abl1 (ABL1)AblTK3kfaB3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamideMouse5740
Abl1 (ABL1)AblTK3ms9AA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5733
Abl1 (ABL1)AblTK3ms9AB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5708
Abl1 (ABL1)AblTK3ms9BA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5713
Abl1 (ABL1)AblTK3ms9BB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5706
Abl1 (ABL1)AblTK3mssA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5724
Abl1 (ABL1)AblTK3mssB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5730
Abl1 (ABL1)AblTK3mssC4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5719
Abl1 (ABL1)AblTK3mssD4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse5702
Abl1 (ABL1)AblTK3oxzA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideMouse5721
Abl1 (ABL1)AblTK3oy3A5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamideMouse5711
Abl1 (ABL1)AblTK3oy3B5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamideMouse5738
Abl1 (ABL1)AblTK6hd4AA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10645
Abl1 (ABL1)AblTK6hd4AB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10647
Abl1 (ABL1)AblTK6hd4BA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10648
Abl1 (ABL1)AblTK6hd4BB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10646
Abl1 (ABL1)AblTK6hd6AA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10609
Abl1 (ABL1)AblTK6hd6AB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10608
Abl1 (ABL1)AblTK6hd6BA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10611
Abl1 (ABL1)AblTK6hd6BB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideMouse10610
ABL1AblTK1oplA6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1104
ABL1AblTK1oplB6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1086
ABL1AblTK2e2bAn-[3-(4,5'-bipyrimidin-2-ylamino)-4-methylphenyl]-4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-3-(trifluoromethyl)benzamideHuman1054
ABL1AblTK2e2bBn-[3-(4,5'-bipyrimidin-2-ylamino)-4-methylphenyl]-4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-3-(trifluoromethyl)benzamideHuman1065
ABL1AblTK2f4jAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman1090
ABL1AblTK2fo0A6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1073
ABL1AblTK2g1tA-Human1045
ABL1AblTK2g1tB-Human1105
ABL1AblTK2g1tC-Human1064
ABL1AblTK2g1tD-Human1096
ABL1AblTK2g2fA-Human1097
ABL1AblTK2g2fBphosphothiophosphoric acid-adenylate esterHuman1079
ABL1AblTK2g2hA6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1106
ABL1AblTK2g2hB6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1089
ABL1AblTK2g2iAadenosine-5'-diphosphateHuman1111
ABL1AblTK2g2iBadenosine-5'-diphosphateHuman1075
ABL1AblTK2gqgAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1060
ABL1AblTK2gqgABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1053
ABL1AblTK2gqgBAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1084
ABL1AblTK2gqgBBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1082
ABL1AblTK2hiwA7-amino-1-methyl-3-(2-methyl-5-{[3-(trifluoromethyl)benzoyl]amino}phenyl)-2-oxo-2,3-dihydropyrimido[4,5-d]pyrimidin-1-iumHuman1069
ABL1AblTK2hiwB7-amino-1-methyl-3-(2-methyl-5-{[3-(trifluoromethyl)benzoyl]amino}phenyl)-2-oxo-2,3-dihydropyrimido[4,5-d]pyrimidin-1-iumHuman1110
ABL1AblTK2hyyA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1092
ABL1AblTK2hyyB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1078
ABL1AblTK2hyyC4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1048
ABL1AblTK2hyyD4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1068
ABL1AblTK2hz0AA2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamideHuman1052
ABL1AblTK2hz0AB2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamideHuman1083
ABL1AblTK2hz0BA2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamideHuman1095
ABL1AblTK2hz0BB2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamideHuman1109
ABL1AblTK2hz4A-Human1059
ABL1AblTK2hz4B1,2,3,4-tetrahydrogen-staurosporineHuman1058
ABL1AblTK2hz4C-Human1067
ABL1AblTK2hziAA6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1102
ABL1AblTK2hziAB6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1087
ABL1AblTK2hziBA6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1108
ABL1AblTK2hziBB6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman1055
ABL1AblTK2v7aAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman1088
ABL1AblTK2v7aBn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman1072
ABL1AblTK3cs9AAnilotinibHuman1080
ABL1AblTK3cs9ABnilotinibHuman1107
ABL1AblTK3cs9BAnilotinibHuman1050
ABL1AblTK3cs9BBnilotinibHuman1112
ABL1AblTK3cs9CAnilotinibHuman1046
ABL1AblTK3cs9CBnilotinibHuman1093
ABL1AblTK3cs9DAnilotinibHuman1077
ABL1AblTK3cs9DBnilotinibHuman1066
ABL1AblTK3pyyAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1049
ABL1AblTK3pyyAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1071
ABL1AblTK3pyyBA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1062
ABL1AblTK3pyyBB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1098
ABL1AblTK3qriAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1051
ABL1AblTK3qriAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1047
ABL1AblTK3qriBA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1103
ABL1AblTK3qriBB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1076
ABL1AblTK3qrjAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1085
ABL1AblTK3qrjAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1099
ABL1AblTK3qrjBA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1101
ABL1AblTK3qrjBB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman1070
ABL1AblTK3qrkA(3s)-6-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acidHuman1056
ABL1AblTK3ue4A4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman1057
ABL1AblTK3ue4B4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman1074
ABL1AblTK4twpAaxitinibHuman1091
ABL1AblTK4twpBaxitinibHuman1081
ABL1AblTK4wa9AaxitinibHuman1061
ABL1AblTK4wa9BaxitinibHuman1063
ABL1AblTK4xeyAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1094
ABL1AblTK4xeyBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman1100
ABL1AblTK4yc8A2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-n-(4-phenoxyphenyl)-1,3-thiazole-5-carboxamideHuman6419
ABL1AblTK4yc8B2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-n-(4-phenoxyphenyl)-1,3-thiazole-5-carboxamideHuman6420
ABL1AblTK4zogAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman7043
ABL1AblTK4zogBcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman7042
ABL1AblTK5hu9AA4-[(4-methylpiperazin-1-yl)methyl]-n-(4-methyl-3-{[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]oxy}phenyl)-3-(trifluoromethyl)benzamideHuman6754
ABL1AblTK5hu9AB4-[(4-methylpiperazin-1-yl)methyl]-n-(4-methyl-3-{[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]oxy}phenyl)-3-(trifluoromethyl)benzamideHuman6755
ABL1AblTK5mo4AAnilotinibHuman7527
ABL1AblTK5mo4ABnilotinibHuman7526
ABL1AblTK6bl8AApurvalanol bHuman9699
ABL1AblTK6bl8ABpurvalanol bHuman9698
ABL1AblTK6bl8BApurvalanol bHuman9701
ABL1AblTK6bl8BBpurvalanol bHuman9700
ABL1AblTK6npeAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10946
ABL1AblTK6npeAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10943
ABL1AblTK6npeBA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10947
ABL1AblTK6npeBB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10945
ABL1AblTK6npuA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10942
ABL1AblTK6npuB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10944
ABL1AblTK6npvAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10948
ABL1AblTK6npvAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10951
ABL1AblTK6npvBA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10949
ABL1AblTK6npvBB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman10950
ABL1AblTK6xr6A1-Human12905
ABL1AblTK6xr6A10-Human12901
ABL1AblTK6xr6A11-Human12872
ABL1AblTK6xr6A12-Human12871
ABL1AblTK6xr6A13-Human12869
ABL1AblTK6xr6A14-Human12873
ABL1AblTK6xr6A15-Human12862
ABL1AblTK6xr6A16-Human12902
ABL1AblTK6xr6A17-Human12874
ABL1AblTK6xr6A18-Human12912
ABL1AblTK6xr6A19-Human12892
ABL1AblTK6xr6A2-Human12878
ABL1AblTK6xr6A20-Human12861
ABL1AblTK6xr6A3-Human12908
ABL1AblTK6xr6A4-Human12898
ABL1AblTK6xr6A5-Human12858
ABL1AblTK6xr6A6-Human12896
ABL1AblTK6xr6A7-Human12881
ABL1AblTK6xr6A8-Human12906
ABL1AblTK6xr6A9-Human12885
ABL1AblTK6xr7A1-Human12867
ABL1AblTK6xr7A10-Human12903
ABL1AblTK6xr7A11-Human12866
ABL1AblTK6xr7A12-Human12860
ABL1AblTK6xr7A13-Human12910
ABL1AblTK6xr7A14-Human12865
ABL1AblTK6xr7A15-Human12913
ABL1AblTK6xr7A16-Human12859
ABL1AblTK6xr7A17-Human12870
ABL1AblTK6xr7A18-Human12909
ABL1AblTK6xr7A19-Human12879
ABL1AblTK6xr7A2-Human12883
ABL1AblTK6xr7A20-Human12914
ABL1AblTK6xr7A3-Human12900
ABL1AblTK6xr7A4-Human12894
ABL1AblTK6xr7A5-Human12857
ABL1AblTK6xr7A6-Human12897
ABL1AblTK6xr7A7-Human12907
ABL1AblTK6xr7A8-Human12863
ABL1AblTK6xr7A9-Human12915
ABL1AblTK6xrgA1-Human12890
ABL1AblTK6xrgA10-Human12889
ABL1AblTK6xrgA11-Human12877
ABL1AblTK6xrgA12-Human12882
ABL1AblTK6xrgA13-Human12904
ABL1AblTK6xrgA14-Human12875
ABL1AblTK6xrgA15-Human12911
ABL1AblTK6xrgA16-Human12887
ABL1AblTK6xrgA17-Human12916
ABL1AblTK6xrgA18-Human12880
ABL1AblTK6xrgA19-Human12886
ABL1AblTK6xrgA2-Human12895
ABL1AblTK6xrgA20-Human12888
ABL1AblTK6xrgA3-Human12893
ABL1AblTK6xrgA4-Human12899
ABL1AblTK6xrgA5-Human12884
ABL1AblTK6xrgA6-Human12876
ABL1AblTK6xrgA7-Human12868
ABL1AblTK6xrgA8-Human12864
ABL1AblTK6xrgA9-Human12891
ABL1AblTK7cc2A[4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methyl-phenyl]boronic acidHuman13620
ABL1AblTK7dt2A[4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methanoyl-5-methoxy-phenyl]boronic acidHuman13621
ABL1AblTK7n9gAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman14197
ABL1AblTK7w7xA5-[5-(dimethylcarbamoyl)pyridin-3-yl]-3-(5-fluorosulfonyloxy-2-methoxy-phenyl)-1h-pyrrolo[2,3-b]pyridineHuman14196
ABL1AblTK7w7yA5-[3-(5-methanoyl-2-methoxy-4-oxidanyl-phenyl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-~{n},~{n}-dimethyl-pyridine-3-carboxamideHuman14195
ABL1AblTK8h7fA1-[6-(6-methoxyisoquinolin-7-yl)-1,3-benzothiazol-2-yl]-3-(2-oxidanylideneethyl)ureaHuman14632
ABL1AblTK8h7hA5-[3-(6-methoxyisoquinolin-7-yl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-~{n}-methyl-~{n}-prop-2-ynyl-pyridine-3-carboxamideHuman14666
ABL1AblTK8ssnA6,7-dimethoxy-n-(4-phenoxyphenyl)quinazolin-4-amineHuman14878
Abl2 (ABL2)AblTK4xliAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideMouse5689
Abl2 (ABL2)AblTK4xliBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideMouse5690
ABL2AblTK2xynAAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman110
ABL2AblTK2xynABcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman112
ABL2AblTK2xynBAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman111
ABL2AblTK2xynBBcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman113
ABL2AblTK2xynCAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman116
ABL2AblTK2xynCBcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman114
ABL2AblTK3gvuAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman117
ABL2AblTK3gvuAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman109
ABL2AblTK3hmiAA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman115
ABL2AblTK3hmiAB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman118
ACVR1 (ALK2)STKRTKL3h9rA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman1531
ACVR1 (ALK2)STKRTKL3mtfAA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman1513
ACVR1 (ALK2)STKRTKL3mtfAB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman1521
ACVR1 (ALK2)STKRTKL3mtfBA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman1515
ACVR1 (ALK2)STKRTKL3mtfBB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman1530
ACVR1 (ALK2)STKRTKL3oomAA1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanoneHuman1517
ACVR1 (ALK2)STKRTKL3oomAB1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanoneHuman1518
ACVR1 (ALK2)STKRTKL3q4uAA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1527
ACVR1 (ALK2)STKRTKL3q4uAB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1524
ACVR1 (ALK2)STKRTKL3q4uBA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1510
ACVR1 (ALK2)STKRTKL3q4uBB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1523
ACVR1 (ALK2)STKRTKL3q4uCA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1516
ACVR1 (ALK2)STKRTKL3q4uCB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1533
ACVR1 (ALK2)STKRTKL3q4uDA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1520
ACVR1 (ALK2)STKRTKL3q4uDB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1529
ACVR1 (ALK2)STKRTKL4bggAA1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1528
ACVR1 (ALK2)STKRTKL4bggAB1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1508
ACVR1 (ALK2)STKRTKL4bggBA1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1514
ACVR1 (ALK2)STKRTKL4bggBB1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1526
ACVR1 (ALK2)STKRTKL4bggCA1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1511
ACVR1 (ALK2)STKRTKL4bggCB1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1522
ACVR1 (ALK2)STKRTKL4bggDA1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1519
ACVR1 (ALK2)STKRTKL4bggDB1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazineHuman1512
ACVR1 (ALK2)STKRTKL4c02AA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman1525
ACVR1 (ALK2)STKRTKL4c02AB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman1532
ACVR1 (ALK2)STKRTKL4dymA1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman1509
ACVR1 (ALK2)STKRTKL5oxgAA5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8514
ACVR1 (ALK2)STKRTKL5oxgAB5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8518
ACVR1 (ALK2)STKRTKL5oxgBA5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8516
ACVR1 (ALK2)STKRTKL5oxgBB5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8519
ACVR1 (ALK2)STKRTKL5oxgCA5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8517
ACVR1 (ALK2)STKRTKL5oxgCB5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8513
ACVR1 (ALK2)STKRTKL5oxgDA5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8520
ACVR1 (ALK2)STKRTKL5oxgDB5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman8515
ACVR1 (ALK2)STKRTKL5oy6Acyclical inhibitor od36Human8532
ACVR1 (ALK2)STKRTKL5oy6Bcyclical inhibitor od36Human8531
ACVR1 (ALK2)STKRTKL5oy6Ccyclical inhibitor od36Human8529
ACVR1 (ALK2)STKRTKL5oy6Dcyclical inhibitor od36Human8534
ACVR1 (ALK2)STKRTKL5s75AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13714
ACVR1 (ALK2)STKRTKL5s75AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13718
ACVR1 (ALK2)STKRTKL5s76AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13691
ACVR1 (ALK2)STKRTKL5s76AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13672
ACVR1 (ALK2)STKRTKL5s77AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13694
ACVR1 (ALK2)STKRTKL5s77AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13698
ACVR1 (ALK2)STKRTKL5s78AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13716
ACVR1 (ALK2)STKRTKL5s78AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13686
ACVR1 (ALK2)STKRTKL5s79AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13704
ACVR1 (ALK2)STKRTKL5s79AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13708
ACVR1 (ALK2)STKRTKL5s7aAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13683
ACVR1 (ALK2)STKRTKL5s7aAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13644
ACVR1 (ALK2)STKRTKL5s7bAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13650
ACVR1 (ALK2)STKRTKL5s7bAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13719
ACVR1 (ALK2)STKRTKL5s7cAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13689
ACVR1 (ALK2)STKRTKL5s7cAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13690
ACVR1 (ALK2)STKRTKL5s7cAC-Human13702
ACVR1 (ALK2)STKRTKL5s7cAD-Human13680
ACVR1 (ALK2)STKRTKL5s7dAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13730
ACVR1 (ALK2)STKRTKL5s7dAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13668
ACVR1 (ALK2)STKRTKL5s7eAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13715
ACVR1 (ALK2)STKRTKL5s7eAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13643
ACVR1 (ALK2)STKRTKL5s7fAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13671
ACVR1 (ALK2)STKRTKL5s7fAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13737
ACVR1 (ALK2)STKRTKL5s7gAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13713
ACVR1 (ALK2)STKRTKL5s7gAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13717
ACVR1 (ALK2)STKRTKL5s7hAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13682
ACVR1 (ALK2)STKRTKL5s7hAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13660
ACVR1 (ALK2)STKRTKL5s7iAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13699
ACVR1 (ALK2)STKRTKL5s7iAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13663
ACVR1 (ALK2)STKRTKL5s7iAC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13653
ACVR1 (ALK2)STKRTKL5s7jAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13712
ACVR1 (ALK2)STKRTKL5s7jAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13648
ACVR1 (ALK2)STKRTKL5s7kAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13649
ACVR1 (ALK2)STKRTKL5s7kAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13732
ACVR1 (ALK2)STKRTKL5s7lAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13676
ACVR1 (ALK2)STKRTKL5s7lAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13736
ACVR1 (ALK2)STKRTKL5s7lAC-Human13665
ACVR1 (ALK2)STKRTKL5s7mAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13666
ACVR1 (ALK2)STKRTKL5s7mAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13739
ACVR1 (ALK2)STKRTKL5s7mAC-Human13705
ACVR1 (ALK2)STKRTKL5s7nAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13655
ACVR1 (ALK2)STKRTKL5s7nAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13659
ACVR1 (ALK2)STKRTKL5s7oAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13733
ACVR1 (ALK2)STKRTKL5s7oAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13664
ACVR1 (ALK2)STKRTKL5s7oAC-Human13647
ACVR1 (ALK2)STKRTKL5s7pAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13695
ACVR1 (ALK2)STKRTKL5s7pAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13687
ACVR1 (ALK2)STKRTKL5s7qAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13670
ACVR1 (ALK2)STKRTKL5s7qAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13678
ACVR1 (ALK2)STKRTKL5s7rAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13731
ACVR1 (ALK2)STKRTKL5s7rAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13654
ACVR1 (ALK2)STKRTKL5s7sAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13667
ACVR1 (ALK2)STKRTKL5s7sAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13677
ACVR1 (ALK2)STKRTKL5s7sAC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13651
ACVR1 (ALK2)STKRTKL5s7tAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13723
ACVR1 (ALK2)STKRTKL5s7tAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13709
ACVR1 (ALK2)STKRTKL5s7uAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13675
ACVR1 (ALK2)STKRTKL5s7uAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13696
ACVR1 (ALK2)STKRTKL5s7vAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13707
ACVR1 (ALK2)STKRTKL5s7vAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13711
ACVR1 (ALK2)STKRTKL5s7wAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13700
ACVR1 (ALK2)STKRTKL5s7wAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13662
ACVR1 (ALK2)STKRTKL5s7xAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13646
ACVR1 (ALK2)STKRTKL5s7xAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13692
ACVR1 (ALK2)STKRTKL5s7yAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13727
ACVR1 (ALK2)STKRTKL5s7yAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13684
ACVR1 (ALK2)STKRTKL5s7zAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13652
ACVR1 (ALK2)STKRTKL5s7zAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13674
ACVR1 (ALK2)STKRTKL5s80AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13728
ACVR1 (ALK2)STKRTKL5s80AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13669
ACVR1 (ALK2)STKRTKL5s81AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13661
ACVR1 (ALK2)STKRTKL5s81AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13697
ACVR1 (ALK2)STKRTKL5s82AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13681
ACVR1 (ALK2)STKRTKL5s82AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13701
ACVR1 (ALK2)STKRTKL5s83AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13706
ACVR1 (ALK2)STKRTKL5s83AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13685
ACVR1 (ALK2)STKRTKL5s84AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13734
ACVR1 (ALK2)STKRTKL5s84AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13656
ACVR1 (ALK2)STKRTKL5s84AC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13722
ACVR1 (ALK2)STKRTKL5s85AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13710
ACVR1 (ALK2)STKRTKL5s85AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13720
ACVR1 (ALK2)STKRTKL5s85AC4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13679
ACVR1 (ALK2)STKRTKL5s86AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13724
ACVR1 (ALK2)STKRTKL5s86AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13729
ACVR1 (ALK2)STKRTKL5s87AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13738
ACVR1 (ALK2)STKRTKL5s87AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13735
ACVR1 (ALK2)STKRTKL5s88AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13657
ACVR1 (ALK2)STKRTKL5s88AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13703
ACVR1 (ALK2)STKRTKL5s89AA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13673
ACVR1 (ALK2)STKRTKL5s89AB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13688
ACVR1 (ALK2)STKRTKL5s8aAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13725
ACVR1 (ALK2)STKRTKL5s8aAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13693
ACVR1 (ALK2)STKRTKL5s8bAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13726
ACVR1 (ALK2)STKRTKL5s8bAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13721
ACVR1 (ALK2)STKRTKL5s9kAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13645
ACVR1 (ALK2)STKRTKL5s9kAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman13658
ACVR1 (ALK2)STKRTKL6acrAn-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amineHuman10969
ACVR1 (ALK2)STKRTKL6acrBn-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amineHuman10968
ACVR1 (ALK2)STKRTKL6eixAA3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman8530
ACVR1 (ALK2)STKRTKL6eixAB3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenolHuman8533
ACVR1 (ALK2)STKRTKL6gi6A5-methyl-6-quinolin-5-yl-3~{h}-quinazolin-4-oneHuman9919
ACVR1 (ALK2)STKRTKL6ginAA3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHuman9914
ACVR1 (ALK2)STKRTKL6ginAB3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHuman9918
ACVR1 (ALK2)STKRTKL6ginBA3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHuman9920
ACVR1 (ALK2)STKRTKL6ginBB3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-oneHuman9916
ACVR1 (ALK2)STKRTKL6gipAA2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-oneHuman9915
ACVR1 (ALK2)STKRTKL6gipAB2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-oneHuman9917
ACVR1 (ALK2)STKRTKL6i1sAA(4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dioneHuman11603
ACVR1 (ALK2)STKRTKL6i1sAB(4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dioneHuman11604
ACVR1 (ALK2)STKRTKL6juxAA4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amineHuman12161
ACVR1 (ALK2)STKRTKL6juxAB4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amineHuman12160
ACVR1 (ALK2)STKRTKL6srhAA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11632
ACVR1 (ALK2)STKRTKL6srhAB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11630
ACVR1 (ALK2)STKRTKL6srhBA4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11631
ACVR1 (ALK2)STKRTKL6srhBB4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman11633
ACVR1 (ALK2)STKRTKL6szmAA1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHuman11735
ACVR1 (ALK2)STKRTKL6szmAB1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHuman11737
ACVR1 (ALK2)STKRTKL6szmBA1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHuman11734
ACVR1 (ALK2)STKRTKL6szmBB1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazineHuman11736
ACVR1 (ALK2)STKRTKL6t6dAA2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11779
ACVR1 (ALK2)STKRTKL6t6dAB2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11784
ACVR1 (ALK2)STKRTKL6t6dBA2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11781
ACVR1 (ALK2)STKRTKL6t6dBB2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11782
ACVR1 (ALK2)STKRTKL6t6dCA2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11778
ACVR1 (ALK2)STKRTKL6t6dCB2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11780
ACVR1 (ALK2)STKRTKL6t6dDA2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11783
ACVR1 (ALK2)STKRTKL6t6dDB2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamideHuman11785
ACVR1 (ALK2)STKRTKL6t8nAAcyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanoneHuman11831
ACVR1 (ALK2)STKRTKL6t8nABcyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanoneHuman11830
ACVR1 (ALK2)STKRTKL6t8nBAcyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanoneHuman11828
ACVR1 (ALK2)STKRTKL6t8nBBcyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanoneHuman11829
ACVR1 (ALK2)STKRTKL6tn8AA4-[4-[(dimethylamino)methyl]-2,5-dimethoxy-phenyl]-2-methyl-2,7-naphthyridin-1-oneHuman11888
ACVR1 (ALK2)STKRTKL6tn8AB4-[4-[(dimethylamino)methyl]-2,5-dimethoxy-phenyl]-2-methyl-2,7-naphthyridin-1-oneHuman11887
ACVR1 (ALK2)STKRTKL6unqAAphosphoaminophosphonic acid-adenylate esterHuman13783
ACVR1 (ALK2)STKRTKL6unqABphosphoaminophosphonic acid-adenylate esterHuman13784
ACVR1 (ALK2)STKRTKL6unrAphosphoaminophosphonic acid-adenylate esterHuman13785
ACVR1 (ALK2)STKRTKL6unsAA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman13782
ACVR1 (ALK2)STKRTKL6unsAB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman13781
ACVR1 (ALK2)STKRTKL6z36AA4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridineHuman12277
ACVR1 (ALK2)STKRTKL6z36AB4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridineHuman12278
ACVR1 (ALK2)STKRTKL6z36BA4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridineHuman12276
ACVR1 (ALK2)STKRTKL6z36BB4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridineHuman12275
ACVR1 (ALK2)STKRTKL6zgcAn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman12638
ACVR1 (ALK2)STKRTKL6zgcBn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman12641
ACVR1 (ALK2)STKRTKL6zgcCn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman12640
ACVR1 (ALK2)STKRTKL6zgcDn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman12639
ACVR1 (ALK2)STKRTKL7a21AA4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman12777
ACVR1 (ALK2)STKRTKL7a21AB4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman12779
ACVR1 (ALK2)STKRTKL7a21BA4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman12776
ACVR1 (ALK2)STKRTKL7a21BB4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridineHuman12778
ACVR1 (ALK2)STKRTKL7c3gAA~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amineHuman13389
ACVR1 (ALK2)STKRTKL7c3gAB~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amineHuman13390
ACVR1 (ALK2)STKRTKL7c3gBA~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amineHuman13392
ACVR1 (ALK2)STKRTKL7c3gBB~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amineHuman13391
ACVR1 (ALK2)STKRTKL7nnsBAmomelotinibHuman13465
ACVR1 (ALK2)STKRTKL7nnsBBmomelotinibHuman13464
ACVR1 (ALK2)STKRTKL8c7wAA6-methyl-9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,7-dihydropyrido[4,3-d][2]benzazepineHuman14608
ACVR1 (ALK2)STKRTKL8c7wAB6-methyl-9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,7-dihydropyrido[4,3-d][2]benzazepineHuman14609
ACVR1 (ALK2)STKRTKL8c7zAA9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1]benzoxepino[5,4-c]pyridineHuman14605
ACVR1 (ALK2)STKRTKL8c7zAB9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1]benzoxepino[5,4-c]pyridineHuman14604
ACVR2A (ACTR2)STKRTKL3q4tAA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2682
ACVR2A (ACTR2)STKRTKL3q4tAB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2686
ACVR2A (ACTR2)STKRTKL3q4tBA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2680
ACVR2A (ACTR2)STKRTKL3q4tBB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman2684
ACVR2A (ACTR2)STKRTKL3socAA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2675
ACVR2A (ACTR2)STKRTKL3socAB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2676
ACVR2A (ACTR2)STKRTKL3socBA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2677
ACVR2A (ACTR2)STKRTKL3socBB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2685
ACVR2A (ACTR2)STKRTKL4asxAA7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-oneHuman2678
ACVR2A (ACTR2)STKRTKL4asxAB7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-oneHuman2681
ACVR2A (ACTR2)STKRTKL4asxBA7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-oneHuman2683
ACVR2A (ACTR2)STKRTKL4asxBB7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-oneHuman2679
ACVR2B (ACTR2B)STKRTKL2qluAadenineHuman2940
ACVRL1 (ALK1)STKRTKL3my0A4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1266
ACVRL1 (ALK1)STKRTKL3my0B4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1273
ACVRL1 (ALK1)STKRTKL3my0C4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1269
ACVRL1 (ALK1)STKRTKL3my0D4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1258
ACVRL1 (ALK1)STKRTKL3my0E4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1263
ACVRL1 (ALK1)STKRTKL3my0F4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1276
ACVRL1 (ALK1)STKRTKL3my0G4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1272
ACVRL1 (ALK1)STKRTKL3my0H4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1260
ACVRL1 (ALK1)STKRTKL3my0I4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1261
ACVRL1 (ALK1)STKRTKL3my0J4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1277
ACVRL1 (ALK1)STKRTKL3my0K4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1267
ACVRL1 (ALK1)STKRTKL3my0L4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1265
ACVRL1 (ALK1)STKRTKL3my0M4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1268
ACVRL1 (ALK1)STKRTKL3my0N4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1257
ACVRL1 (ALK1)STKRTKL3my0O4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1262
ACVRL1 (ALK1)STKRTKL3my0P4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1270
ACVRL1 (ALK1)STKRTKL3my0Q4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1274
ACVRL1 (ALK1)STKRTKL3my0R4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1256
ACVRL1 (ALK1)STKRTKL3my0S4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1259
ACVRL1 (ALK1)STKRTKL3my0T4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1264
ACVRL1 (ALK1)STKRTKL3my0U4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1278
ACVRL1 (ALK1)STKRTKL3my0V4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1271
ACVRL1 (ALK1)STKRTKL3my0W4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1255
ACVRL1 (ALK1)STKRTKL3my0X4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1275
AKT1AktAGC3cquAAn-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6764
AKT1AktAGC3cquABn-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6762
AKT1AktAGC3cqwAA5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridineHuman6763
AKT1AktAGC3cqwAB5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridineHuman6765
AKT1AktAGC3mv5AA(3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amineHuman2537
AKT1AktAGC3mv5AB(3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amineHuman2532
AKT1AktAGC3mvhAAn-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamideHuman2538
AKT1AktAGC3mvhABn-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamideHuman2531
AKT1AktAGC3o96A-Human2545
AKT1AktAGC3ocbA(2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amineHuman2548
AKT1AktAGC3ocbB(2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amineHuman2534
AKT1AktAGC3ow4A(2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amineHuman2547
AKT1AktAGC3ow4B(2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amineHuman2533
AKT1AktAGC3qkkAn-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(2r)-6-hydroxy-4-oxo-3,4-dihydro-1'h-spiro[chromene-2,3'-piperidin]-1'-yl]propyl}-2,6-dimethylbenzenesulfonamideHuman2535
AKT1AktAGC3qklAn-{(2s)-3-[(3s)-8',9'-dihydro-1h,3'h-spiro[piperidine-3,7'-pyrano[3,2-e]indazol]-1-yl]-2-hydroxypropyl}-n-(2-ethoxyethyl)-2,6-dimethylbenzenesulfonamideHuman2544
AKT1AktAGC3qkmAn-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(5r)-2-(quinazolin-4-yl)-2,7-diazaspiro[4.5]dec-7-yl]propyl}-2,6-dimethylbenzenesulfonamideHuman2546
AKT1AktAGC4ejnA-Human2542
AKT1AktAGC4ekkAphosphoaminophosphonic acid-adenylate esterHuman2541
AKT1AktAGC4ekkBphosphoaminophosphonic acid-adenylate esterHuman2539
AKT1AktAGC4eklA(2s)-2-(4-chlorophenyl)-1-{4-[(5r,7r)-7-hydroxy-5-methyl-6,7-dihydro-5h-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl}-3-(propan-2-ylamino)propan-1-oneHuman2540
AKT1AktAGC4gv1AA4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamideHuman2543
AKT1AktAGC4gv1AB4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamideHuman2536
AKT1AktAGC5kcvA3-[3-[4-(1-azanylcyclobutyl)phenyl]-5-phenyl-imidazo[4,5-b]pyridin-2-yl]pyridin-2-amineHuman6708
AKT1AktAGC6buuAA-Human10432
AKT1AktAGC6buuAB-Human10433
AKT1AktAGC6buuAC-Human10438
AKT1AktAGC6buuBA-Human10430
AKT1AktAGC6buuBB-Human10439
AKT1AktAGC6buuBC-Human10428
AKT1AktAGC6ccyAA(5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-oneHuman9868
AKT1AktAGC6ccyAB(5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-oneHuman9869
AKT1AktAGC6hhfAborussertibHuman10970
AKT1AktAGC6hhgA~{n}-[2-chloranyl-5-[[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]carbamoylamino]phenyl]propanamideHuman10916
AKT1AktAGC6hhhA~{n}-[4-[4-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperazin-1-yl]phenyl]propanamideHuman10915
AKT1AktAGC6hhiA~{n}-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]-3-(propanoylamino)benzamideHuman10913
AKT1AktAGC6hhjA~{n}-[1-methyl-2-oxidanylidene-3-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]benzimidazol-5-yl]propanamideHuman10914
AKT1AktAGC6npzAA-Human10880
AKT1AktAGC6npzAB-Human10882
AKT1AktAGC6npzBA-Human10881
AKT1AktAGC6npzBB-Human10879
AKT1AktAGC6s9wAA~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamideHuman11748
AKT1AktAGC6s9wAB~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamideHuman11747
AKT1AktAGC6s9xA~{n}-[3-[1-[[4-[5-[(4-hydroxyphenyl)methyl]-6-oxidanylidene-2-phenyl-1~{h}-pyrazin-3-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamideHuman11746
AKT1AktAGC7apjA-Human13854
AKT1AktAGC7nh4AA~{n}-[3-[1-[[4-[5-(hydroxymethyl)-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamideHuman13865
AKT1AktAGC7nh4AB~{n}-[3-[1-[[4-[5-(hydroxymethyl)-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamideHuman13866
AKT1AktAGC7nh5AA~{n}-methyl-6-[4-[[4-[2-oxidanylidene-6-(propanoylamino)-3~{h}-benzimidazol-1-yl]piperidin-1-yl]methyl]phenyl]-5-phenyl-pyridine-3-carboxamideHuman13867
AKT1AktAGC7nh5AB~{n}-methyl-6-[4-[[4-[2-oxidanylidene-6-(propanoylamino)-3~{h}-benzimidazol-1-yl]piperidin-1-yl]methyl]phenyl]-5-phenyl-pyridine-3-carboxamideHuman13868
AKT2AktAGC1gzkA-Human1916
AKT2AktAGC1gznA-Human1915
AKT2AktAGC1gzoA-Human1914
AKT2AktAGC1mrvA-Human1917
AKT2AktAGC1mryA-Human1907
AKT2AktAGC1o6kAphosphoaminophosphonic acid-adenylate esterHuman1923
AKT2AktAGC1o6lAphosphoaminophosphonic acid-adenylate esterHuman1906
AKT2AktAGC2jdoAisoquinoline-5-sulfonic acid (2-(2-(4-chlorobenzyloxy)ethylamino)ethyl)amideHuman1922
AKT2AktAGC2jdrA(2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amineHuman1918
AKT2AktAGC2uw9A4-(4-chlorophenyl)-4-[4-(1h-pyrazol-4-yl)phenyl]piperidineHuman1919
AKT2AktAGC2x39A4-amino-n-(4-chlorobenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamideHuman1913
AKT2AktAGC2xh5A4-(4-tert-butylbenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-aminiumHuman1924
AKT2AktAGC3d0eA4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-olHuman1912
AKT2AktAGC3d0eB4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-olHuman1920
AKT2AktAGC3e87AAn-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamideHuman1910
AKT2AktAGC3e87ABn-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamideHuman1911
AKT2AktAGC3e87BAn-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamideHuman1909
AKT2AktAGC3e87BBn-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamideHuman1903
AKT2AktAGC3e88A4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1908
AKT2AktAGC3e88B4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1905
AKT2AktAGC3e8dAA4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1921
AKT2AktAGC3e8dAB4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1926
AKT2AktAGC3e8dBA4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1925
AKT2AktAGC3e8dBB4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-olHuman1904
AKT2AktAGC8q61AA6-[4-(1-azanyl-3-methyl-3-oxidanyl-cyclobutyl)phenyl]-7-phenyl-1-propyl-pyrido[2,3-b][1,4]oxazin-2-oneHuman14978
AKT2AktAGC8q61AB6-[4-(1-azanyl-3-methyl-3-oxidanyl-cyclobutyl)phenyl]-7-phenyl-1-propyl-pyrido[2,3-b][1,4]oxazin-2-oneHuman14979
ALKALKTK2xb7A5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHuman5365
ALKALKTK2xbaA5-[(2r)-2-hydroxy-2-phenylacetyl]-3-({[4-(4-methylpiperazin-1-yl)phenyl]carbonyl}amino)-1,6-dihydropyrrolo[3,4-c]pyrazol-5-ium Human5408
ALKALKTK2xp2A3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman5394
ALKALKTK2yfxA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman5402
ALKALKTK2yhvA-Human5384
ALKALKTK2yjrAA-Human5399
ALKALKTK2yjrAB-Human5380
ALKALKTK2yjsA-Human5373
ALKALKTK3aoxAA9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrileHuman5387
ALKALKTK3aoxAB9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrileHuman5370
ALKALKTK3l9pAA-Human5363
ALKALKTK3l9pAB-Human5375
ALKALKTK3lcsAAstaurosporineHuman5381
ALKALKTK3lcsABstaurosporineHuman5376
ALKALKTK3lctAAadenosine-5'-diphosphateHuman5393
ALKALKTK3lctABadenosine-5'-diphosphateHuman5400
ALKALKTK4anlA-Human5385
ALKALKTK4anqA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman5368
ALKALKTK4ansA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman5374
ALKALKTK4ccbA3-[(1r)-1-[5-fluoranyl-2-(1,2,3-triazol-2-yl)phenyl]ethoxy]-5-(3-methyl-1h-pyrazol-4-yl)pyridin-2-amineHuman5390
ALKALKTK4ccuA2-(5-(6-amino-5-((r)-1-(5-fluoro-2-(2h-1,2,3-triazol-2-yl)phenyl)ethoxy)pyridin-3-yl)-4-methylthiazol-2-yl)propan-2-olHuman5396
ALKALKTK4cd0A(2r)-2-[5-(6-amino-5-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diolHuman5407
ALKALKTK4cliA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman5405
ALKALKTK4cljA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman5369
ALKALKTK4cmoA2-[(1r)-1-{[3-amino-6-(2-methoxypyridin-3-yl)pyrazin-2-yl]oxy}ethyl]-4-fluoro-n-methylbenzamideHuman5391
ALKALKTK4cmtA3-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}-5-[3-(methylsulfonyl)phenyl]pyridin-2-amineHuman5371
ALKALKTK4cmuA(10r)-7-amino-12-fluoro-1,3,10,16-tetramethyl-16,17-dihydro-1h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman5398
ALKALKTK4cnhA3-[(1r)-1-(5-fluoro-2-methoxyphenyl)ethoxy]-5-(1-methyl-1h-1,2,3-triazol-5-yl)pyridin-2-amineHuman5388
ALKALKTK4cnhB3-[(1r)-1-(5-fluoro-2-methoxyphenyl)ethoxy]-5-(1-methyl-1h-1,2,3-triazol-5-yl)pyridin-2-amineHuman5378
ALKALKTK4ctbA(5r)-8-amino-3-fluoro-5,19-dimethyl-20-oxo-5,18,19,20-tetrahydro-11,7-(azeno)pyrido[2',1':2,3]imidazo[4,5-h][2,5,11]benzoxadiazacyclotetradecine-14-carbonitrileHuman5395
ALKALKTK4ctcA(10r)-7-amino-3-cyclopropyl-12-fluoro-1,10,16-trimethyl-16,17-dihydro-1h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman5364
ALKALKTK4dceA(3s)-n-(4-methylbenzyl)-1-{2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}piperidine-3-carboxamideHuman5379
ALKALKTK4dceB(3s)-n-(4-methylbenzyl)-1-{2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}piperidine-3-carboxamideHuman5372
ALKALKTK4fnwA-Human5403
ALKALKTK4fnxA-Human5366
ALKALKTK4fnyAn-(4-chlorophenyl)-5-[(6,7-dimethoxyquinolin-4-yl)oxy]-1,3-benzoxazol-2-amineHuman5367
ALKALKTK4fnzA(3s)-n-[3-(trifluoromethoxy)benzyl]-1-{2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}piperidine-3-carboxamideHuman5397
ALKALKTK4fobAn-{1-[cis-4-(hydroxymethyl)cyclohexyl]-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl}-3-(prop-2-en-1-ylsulfamoyl)benzamideHuman5377
ALKALKTK4focAmethyl cis-4-[2-(benzoylamino)-6-(piperidin-1-ylmethyl)-1h-benzimidazol-1-yl]cyclohexanecarboxylateHuman5392
ALKALKTK4fodAA4-fluoro-n-{(2e)-6-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-1-[cis-4-(propan-2-ylcarbamoyl)cyclohexyl]-1,3-dihydro-2h-benzimidazol-2-ylidene}benzamideHuman5383
ALKALKTK4fodAB4-fluoro-n-{(2e)-6-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-1-[cis-4-(propan-2-ylcarbamoyl)cyclohexyl]-1,3-dihydro-2h-benzimidazol-2-ylidene}benzamideHuman5404
ALKALKTK4joaAA3-[1-(2,5-difluorobenzyl)-1h-pyrazol-4-yl]-5-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman5389
ALKALKTK4mkcAA5-chloro-n~2~-[5-methyl-4-(piperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]pyrimidine-2,4-diamineHuman5401
ALKALKTK4mkcAB5-chloro-n~2~-[5-methyl-4-(piperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]pyrimidine-2,4-diamineHuman5386
ALKALKTK4tt7AA-Human5406
ALKALKTK4tt7AB-Human5382
ALKALKTK4z55AAn~6~-[5-methyl-4-(1-methylpiperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]-2h-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman6393
ALKALKTK4z55ABn~6~-[5-methyl-4-(1-methylpiperidin-4-yl)-2-(propan-2-yloxy)phenyl]-n~4~-[2-(propan-2-ylsulfonyl)phenyl]-2h-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman6392
ALKALKTK5a9uAA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6692
ALKALKTK5a9uAB(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6685
ALKALKTK5aa8AA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6688
ALKALKTK5aa8AB(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6684
ALKALKTK5aa9AA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6682
ALKALKTK5aa9AB(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman6687
ALKALKTK5aaaAA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6691
ALKALKTK5aaaAB3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6683
ALKALKTK5aabAA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6689
ALKALKTK5aabAB3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6681
ALKALKTK5aacAA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6690
ALKALKTK5aacAB3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman6686
ALKALKTK5ftoAAentrectinibHuman6520
ALKALKTK5ftoABentrectinibHuman6521
ALKALKTK5ftqAAn-[5-(3,5-difluorobenzyl)-1h-indazol-3-yl]-2-[(4-hydroxycyclohexyl)amino]-4-(4-methylpiperazin-1-yl) benzamideHuman6519
ALKALKTK5ftqABn-[5-(3,5-difluorobenzyl)-1h-indazol-3-yl]-2-[(4-hydroxycyclohexyl)amino]-4-(4-methylpiperazin-1-yl) benzamideHuman6518
ALKALKTK5imxA5-chloro-n~2~-{5-methyl-4-(1-methylpiperidin-4-yl)-2-[(propan-2-yl)oxy]phenyl}-n~4~-{1-methyl-3-[(propan-2-yl)sulfonyl]-1h-pyrazol-4-yl}pyrimidine-2,4-diamineHuman6604
ALKALKTK5iugAAn-[3-(4-{[(5-tert-butyl-1,2-oxazol-3-yl)carbamoyl]amino}-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamideHuman6640
ALKALKTK5iugABn-[3-(4-{[(5-tert-butyl-1,2-oxazol-3-yl)carbamoyl]amino}-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamideHuman6639
ALKALKTK5iuhA4-[(4-methylpiperazin-1-yl)methyl]-n-{3-[3-methyl-4-({[5-(propan-2-yl)-1,2-oxazol-3-yl]carbamoyl}amino)phenyl]-1h-pyrazol-5-yl}benzamideHuman6638
ALKALKTK5iuiAAn-[3-(4-amino-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamideHuman6641
ALKALKTK5iuiABn-[3-(4-amino-3-methylphenyl)-1h-pyrazol-5-yl]-4-[(4-methylpiperazin-1-yl)methyl]benzamideHuman6642
ALKALKTK5kz0A2-[(1~{r})-1-[2-azanyl-5-(1,3-dimethylpyrazol-4-yl)pyridin-3-yl]oxyethyl]-4-fluoranyl-~{n},~{n}-dimethyl-benzamideHuman6970
ALKALKTK6cdtA-Human11263
ALKALKTK6e0rAAn-[(1s)-1-(5-fluoropyridin-2-yl)ethyl]-1-(5-methyl-1h-pyrazol-3-yl)-3-[(oxetan-3-yl)sulfonyl]-1h-pyrrolo[2,3-b]pyridin-6-amineHuman11268
ALKALKTK6e0rABn-[(1s)-1-(5-fluoropyridin-2-yl)ethyl]-1-(5-methyl-1h-pyrazol-3-yl)-3-[(oxetan-3-yl)sulfonyl]-1h-pyrrolo[2,3-b]pyridin-6-amineHuman11266
ALKALKTK6ebwAA[6-{[(1s)-1-(5-fluoropyridin-2-yl)ethyl]amino}-1-(5-methyl-1h-pyrazol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl](morpholin-4-yl)methanoneHuman11269
ALKALKTK6ebwAB[6-{[(1s)-1-(5-fluoropyridin-2-yl)ethyl]amino}-1-(5-methyl-1h-pyrazol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl](morpholin-4-yl)methanoneHuman11264
ALKALKTK6edlAAn-[(1s)-1-(2,4-difluorophenyl)ethyl]-3-(5-methyl-1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-6-amineHuman11267
ALKALKTK6edlABn-[(1s)-1-(2,4-difluorophenyl)ethyl]-3-(5-methyl-1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-6-amineHuman11265
ALKALKTK6mx8AA5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamineHuman10798
ALKALKTK6mx8AB5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamineHuman10799
ALKALKTK7bttAA2-(dimethylamino)-1-[5-methoxy-6-[[4-[(2-propan-2-ylsulfonylphenyl)amino]-5h-pyrrolo[3,2-d]pyrimidin-2-yl]amino]-2,3-dihydroindol-1-yl]ethanoneHuman13484
ALKALKTK7bttAB2-(dimethylamino)-1-[5-methoxy-6-[[4-[(2-propan-2-ylsulfonylphenyl)amino]-5h-pyrrolo[3,2-d]pyrimidin-2-yl]amino]-2,3-dihydroindol-1-yl]ethanoneHuman13483
ALKALKTK7jy4A1-{(1s,2s)-1-(2,4-difluorophenyl)-2-[2-(3-methyl-1h-pyrazol-5-yl)-4-(trifluoromethyl)phenoxy]cyclopropyl}methanamineHuman13240
ALKALKTK7jyrAA4-{[(1r,2r)-2-(2,4-difluorophenyl)cyclopropyl]oxy}-3-(5-methyl-1h-pyrazol-3-yl)benzonitrileHuman13243
ALKALKTK7jyrAB4-{[(1r,2r)-2-(2,4-difluorophenyl)cyclopropyl]oxy}-3-(5-methyl-1h-pyrazol-3-yl)benzonitrileHuman13241
ALKALKTK7jysAA3-(3-chlorophenyl)-5-methyl-1h-pyrazoleHuman13244
ALKALKTK7jysAB3-(3-chlorophenyl)-5-methyl-1h-pyrazoleHuman13239
ALKALKTK7jytAA3-(3-methyl-1h-pyrazol-5-yl)pyridineHuman13238
ALKALKTK7jytAB3-(3-methyl-1h-pyrazol-5-yl)pyridineHuman13242
ALKALKTK7r7kA4-(6-amino-5-{(1r)-1-[5-fluoro-2-(2h-1,2,3-triazol-2-yl)phenyl]ethoxy}pyridin-3-yl)-2,3-dihydro-1h-isoindol-1-oneHuman14267
ALKALKTK7r7rA(2r)-2-[5-(6-amino-5-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diolHuman14266
ALKALKTK8arjAA3-(dimethylamino)-1-[3-[4-(4-methylpiperazin-1-yl)phenyl]-9~{h}-pyrido[2,3-b]indol-6-yl]prop-2-en-1-oneHuman14366
ALKALKTK8arjAB3-(dimethylamino)-1-[3-[4-(4-methylpiperazin-1-yl)phenyl]-9~{h}-pyrido[2,3-b]indol-6-yl]prop-2-en-1-oneHuman14367
ANTXR1 (DNAPK)PIKKAtypical5luqA-Human9321
ANTXR1 (DNAPK)PIKKAtypical5luqB-Human9319
ANTXR1 (DNAPK)PIKKAtypical5w1rA-Human9320
ANTXR1 (DNAPK)PIKKAtypical5y3rC-Human9318
ANTXR1 (DNAPK)PIKKAtypical6zfpA-Human12926
ANTXR1 (DNAPK)PIKKAtypical6zh2A-Human12927
ANTXR1 (DNAPK)PIKKAtypical6zh4A-Human12930
ANTXR1 (DNAPK)PIKKAtypical6zh6A-Human12929
ANTXR1 (DNAPK)PIKKAtypical6zh8A-Human12925
ANTXR1 (DNAPK)PIKKAtypical6zhaA-Human12931
ANTXR1 (DNAPK)PIKKAtypical6zheA-Human12928
ANTXR1 (DNAPK)PIKKAtypical6zheF-Human12932
ANTXR1 (DNAPK)PIKKAtypical7k0yAA-Human13213
ANTXR1 (DNAPK)PIKKAtypical7k0yAB-Human13214
ANTXR1 (DNAPK)PIKKAtypical7k10A-Human13217
ANTXR1 (DNAPK)PIKKAtypical7k11A-Human13208
ANTXR1 (DNAPK)PIKKAtypical7k17A-Human13215
ANTXR1 (DNAPK)PIKKAtypical7k17B-Human13212
ANTXR1 (DNAPK)PIKKAtypical7k19A-Human13216
ANTXR1 (DNAPK)PIKKAtypical7k1bA-Human13218
ANTXR1 (DNAPK)PIKKAtypical7k1jA-Human13209
ANTXR1 (DNAPK)PIKKAtypical7k1kA-Human13211
ANTXR1 (DNAPK)PIKKAtypical7k1nA-Human13210
ANTXR1 (DNAPK)PIKKAtypical7lt3Cadenosine-5'-diphosphateHuman13500
ANTXR1 (DNAPK)PIKKAtypical7lt3Ladenosine-5'-diphosphateHuman13501
ANTXR1 (DNAPK)PIKKAtypical7nfcA-Human13852
ANTXR1 (DNAPK)PIKKAtypical7nfeA-Human13851
ANTXR1 (DNAPK)PIKKAtypical7otmA8-(dibenzo[b,d]thiophen-4-yl)-2-(morpholin-4-yl)-4h-chromen-4-oneHuman14061
ANTXR1 (DNAPK)PIKKAtypical7otpAphosphothiophosphoric acid-adenylate esterHuman14054
ANTXR1 (DNAPK)PIKKAtypical7otvA(1s,6br,9as,11r,11br)-9a,11b-dimethyl-1-[(methyloxy)methyl]-3,6,9-trioxo-1,6,6b,7,8,9,9a,10,11,11b-decahydro-3h-furo[4,3,2-de]indeno[4,5-h][2]benzopyran-11-yl acetateHuman14063
ANTXR1 (DNAPK)PIKKAtypical7otwA7-methyl-2-[(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(oxan-4-yl)purin-8-oneHuman14056
ANTXR1 (DNAPK)PIKKAtypical7otyA(~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanolHuman14057
ANTXR1 (DNAPK)PIKKAtypical7sglAAadenosine-5'-triphosphateHuman14059
ANTXR1 (DNAPK)PIKKAtypical7sglABadenosine-5'-triphosphateHuman14062
ANTXR1 (DNAPK)PIKKAtypical7su3AAadenosine-5'-triphosphateHuman14058
ANTXR1 (DNAPK)PIKKAtypical7su3ABadenosine-5'-triphosphateHuman14053
ANTXR1 (DNAPK)PIKKAtypical7sudAAadenosine-5'-triphosphateHuman14055
ANTXR1 (DNAPK)PIKKAtypical7sudABadenosine-5'-triphosphateHuman14060
ANTXR1 (DNAPK)PIKKAtypical7tyrAA-Human14322
ANTXR1 (DNAPK)PIKKAtypical7tyrAB-Human14321
ANTXR1 (DNAPK)PIKKAtypical7z87AA(~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanolHuman14592
ANTXR1 (DNAPK)PIKKAtypical7z87AB(~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanolHuman14593
ANTXR1 (DNAPK)PIKKAtypical7z88A(~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanolHuman14594
ANTXR1 (DNAPK)PIKKAtypical8bh3A-Human14768
ANTXR1 (DNAPK)PIKKAtypical8bhvA-Human14769
ANTXR1 (DNAPK)PIKKAtypical8bhyA-Human14770
ANTXR1 (DNAPK)PIKKAtypical8ezbCadenosine-5'-triphosphateHuman14798
ATMPIKKAtypical5np0A-Human9267
ATMPIKKAtypical5np0B-Human9266
ATMPIKKAtypical5np1A-Human9268
ATMPIKKAtypical6k9kA-Human11897
ATMPIKKAtypical6k9lA-Human11896
ATMPIKKAtypical6k9lB-Human11895
ATMPIKKAtypical7ni4A8-(1,3-dimethylpyrazol-4-yl)-1-(3-fluoranyl-5-methoxy-pyridin-4-yl)-7-methoxy-3-methyl-imidazo[4,5-c]quinolin-2-oneHuman13864
ATMPIKKAtypical7ni5A2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-oneHuman13863
ATMPIKKAtypical7ni6Aphosphothiophosphoric acid-adenylate esterHuman13862
ATMPIKKAtypical7sicAphosphoaminophosphonic acid-adenylate esterHuman14101
ATMPIKKAtypical7sidAphosphoaminophosphonic acid-adenylate esterHuman14102
ATMPIKKAtypical8oxmBphosphoaminophosphonic acid-adenylate esterHuman14992
ATMPIKKAtypical8oxoBphosphoaminophosphonic acid-adenylate esterHuman14993
ATMPIKKAtypical8oxpAphosphoaminophosphonic acid-adenylate esterHuman14991
ATMPIKKAtypical8oxqAphosphoaminophosphonic acid-adenylate esterHuman14990
ATRPIKKAtypical5yz0A-Human9523
ATRPIKKAtypical5yz0B-Human9524
Aurka (AurA)AUROther3d14AA1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouse5781
Aurka (AurA)AUROther3d14AB1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouse5775
Aurka (AurA)AUROther3d15AA1-(3-chlorophenyl)-3-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}ureaMouse5777
Aurka (AurA)AUROther3d2iA1-(5-{2-[(1-methyl-1h-pyrazolo[4,3-d]pyrimidin-7-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouse5782
Aurka (AurA)AUROther3d2kA(7-{[2-(2-{[(3-chlorophenyl)carbamoyl]amino}-1,3-thiazol-5-yl)ethyl]amino}-1h-pyrazolo[4,3-d]pyrimidin-1-yl)acetic acidMouse5776
Aurka (AurA)AUROther3dajAn-butyl-3-{[6-(9h-purin-6-ylamino)hexanoyl]amino}benzamideMouse5779
Aurka (AurA)AUROther3dj5A3-({3-[(6-amino-5-bromopyrimidin-4-yl)sulfanyl]propanoyl}amino)-4-methoxy-n-phenylbenzamideMouse5783
Aurka (AurA)AUROther3dj6A4-methoxy-n-phenyl-3-({3-[(1h-pyrrolo[2,3-b]pyridin-5-ylmethyl)sulfanyl]propanoyl}amino)benzamideMouse5778
Aurka (AurA)AUROther3dj7AA1-(5-{2-[(6-amino-5-bromopyrimidin-4-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouse5780
AURKA (AurA)AurOther1mq4Aadenosine-5'-diphosphateHuman1977
AURKA (AurA)AurOther1muoAadenosineHuman2062
AURKA (AurA)AurOther1ol5Aadenosine-5'-diphosphateHuman2080
AURKA (AurA)AurOther1ol6Aadenosine-5'-triphosphateHuman2081
AURKA (AurA)AurOther1ol7Aadenosine-5'-diphosphateHuman2014
AURKA (AurA)AurOther2bmcA(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2015
AURKA (AurA)AurOther2bmcB(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2008
AURKA (AurA)AurOther2bmcC(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2060
AURKA (AurA)AurOther2bmcD(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman1984
AURKA (AurA)AurOther2bmcE(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2069
AURKA (AurA)AurOther2bmcF(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman1993
AURKA (AurA)AurOther2c6dAAphosphoaminophosphonic acid-adenylate esterHuman2019
AURKA (AurA)AurOther2c6dABphosphoaminophosphonic acid-adenylate esterHuman1981
AURKA (AurA)AurOther2c6eAn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHuman1989
AURKA (AurA)AurOther2c6eBn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHuman2046
AURKA (AurA)AurOther2dwbAphosphoaminophosphonic acid-adenylate esterHuman2035
AURKA (AurA)AurOther2j4zA4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHuman2053
AURKA (AurA)AurOther2j4zB4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHuman1990
AURKA (AurA)AurOther2j50An-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman2001
AURKA (AurA)AurOther2j50Bn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman2050
AURKA (AurA)AurOther2np8An-{3-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]phenyl}cyclopropanecarboxamideHuman2075
AURKA (AurA)AurOther2w1cA4-{[2-(4-{[(4-fluorophenyl)carbonyl]amino}-1h-pyrazol-3-yl)-1h-benzimidazol-6-yl]methyl}morpholin-4-iumHuman2027
AURKA (AurA)AurOther2w1dA2-(1h-pyrazol-3-yl)-1h-benzimidazoleHuman2011
AURKA (AurA)AurOther2w1eA4-[(2-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-3-yl}-1h-benzimidazol-5-yl)methyl]morpholin-4-iumHuman2038
AURKA (AurA)AurOther2w1fAn-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamideHuman2055
AURKA (AurA)AurOther2w1gA2-{4-[(cyclopropylcarbamoyl)amino]-1h-pyrazol-3-yl}-6-(morpholin-4-ium-4-ylmethyl)-1h-3,1-benzimidazol-3-iumHuman1962
AURKA (AurA)AurOther2wqeAadenosine-5'-diphosphateHuman2071
AURKA (AurA)AurOther2wtvAA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2056
AURKA (AurA)AurOther2wtvAB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman1997
AURKA (AurA)AurOther2wtvBA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2037
AURKA (AurA)AurOther2wtvBB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2057
AURKA (AurA)AurOther2wtvCA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2017
AURKA (AurA)AurOther2wtvCB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2016
AURKA (AurA)AurOther2wtvDA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2078
AURKA (AurA)AurOther2wtvDB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2076
AURKA (AurA)AurOther2wtwA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman1956
AURKA (AurA)AurOther2x6dAA6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridineHuman1978
AURKA (AurA)AurOther2x6dAB6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridineHuman1975
AURKA (AurA)AurOther2x6eA6-bromo-7-{4-[(5-methylisoxazol-3-yl)methyl]piperazin-1-yl}-2-[4-(4-methylpiperazin-1-yl)phenyl]-1h-imidazo[4,5-b]pyridineHuman2079
AURKA (AurA)AurOther2x81A4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman1966
AURKA (AurA)AurOther2xneA3-chloro-n-(4-morpholin-4-ylphenyl)-6-pyridin-3-ylimidazo[1,2-a]pyrazin-8-amineHuman7221
AURKA (AurA)AurOther2xngAAn-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamideHuman1994
AURKA (AurA)AurOther2xngABn-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamideHuman2083
AURKA (AurA)AurOther2xruA3-({[4-(4-methylpiperazin-1-yl)phenyl]carbonyl}amino)-n-[(1r)-1-phenylpropyl]-1h-thieno[3,2-c]pyrazole-5-carboxamideHuman1954
AURKA (AurA)AurOther3cohA8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-oneHuman1963
AURKA (AurA)AurOther3cohB8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-oneHuman2024
AURKA (AurA)AurOther3e5aAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman2006
AURKA (AurA)AurOther3efwA1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHuman2010
AURKA (AurA)AurOther3efwB1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHuman2074
AURKA (AurA)AurOther3fdnAn-[3-(acetylamino)phenyl]-5-{(2e)-2-[(4-methoxyphenyl)methylidene]hydrazino}-3-methyl-1h-pyrazole-4-carboxamideHuman1973
AURKA (AurA)AurOther3h0yA2-chloro-n-[4-({5-fluoro-2-[(4-hydroxyphenyl)amino]pyrimidin-4-yl}amino)phenyl]benzamideHuman1965
AURKA (AurA)AurOther3h0zA4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHuman1970
AURKA (AurA)AurOther3h0zB4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHuman1986
AURKA (AurA)AurOther3h0zC4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHuman2063
AURKA (AurA)AurOther3h10A9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHuman2009
AURKA (AurA)AurOther3h10B9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHuman1988
AURKA (AurA)AurOther3h10D9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHuman2059
AURKA (AurA)AurOther3ha6An~2~-(3,4-dimethoxyphenyl)-n~4~-[2-(2-fluorophenyl)ethyl]-n~6~-quinolin-6-yl-1,3,5-triazine-2,4,6-triamineHuman2048
AURKA (AurA)AurOther3k5uA2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanolHuman2031
AURKA (AurA)AurOther3lauAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]butanamideHuman1971
AURKA (AurA)AurOther3m11A1-(4-{2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHuman2036
AURKA (AurA)AurOther3mygA2-{ethyl[(5-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}isothiazol-3-yl)methyl]amino}-2-methylpropan-1-olHuman2065
AURKA (AurA)AurOther3nrmAn-(3-methylisothiazol-5-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-amineHuman2052
AURKA (AurA)AurOther3o50An-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHuman1958
AURKA (AurA)AurOther3o50Bn-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHuman2067
AURKA (AurA)AurOther3o51An-[4-({3-[5-fluoro-2-(methylideneamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-2-(phenylamino)benzamideHuman1974
AURKA (AurA)AurOther3p9jA4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-oneHuman2003
AURKA (AurA)AurOther3qbnA5-chloro-n~4~-cyclopropyl-n~2~-[4-(2-methoxyethoxy)phenyl]pyrimidine-2,4-diamineHuman2032
AURKA (AurA)AurOther3r21AAn-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHuman1991
AURKA (AurA)AurOther3r21ABn-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHuman2033
AURKA (AurA)AurOther3r22An-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHuman2034
AURKA (AurA)AurOther3unzA4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1972
AURKA (AurA)AurOther3unzB4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2049
AURKA (AurA)AurOther3uo4A4-{[4-(biphenyl-2-ylamino)pyrimidin-2-yl]amino}benzoic acidHuman1976
AURKA (AurA)AurOther3uo5A4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acidHuman2045
AURKA (AurA)AurOther3uo6A4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1985
AURKA (AurA)AurOther3uo6B4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1960
AURKA (AurA)AurOther3uodA4-[(4-{[2-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzoic acidHuman1980
AURKA (AurA)AurOther3uohA4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2077
AURKA (AurA)AurOther3uohB4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2000
AURKA (AurA)AurOther3uojA4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2042
AURKA (AurA)AurOther3uojB4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1979
AURKA (AurA)AurOther3uokA4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acidHuman2054
AURKA (AurA)AurOther3uokB4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acidHuman2047
AURKA (AurA)AurOther3uolAn~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamineHuman2004
AURKA (AurA)AurOther3uolBn~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamineHuman2051
AURKA (AurA)AurOther3up2A4-[(4-{[2-(trifluoromethoxy)phenyl]amino}pyrimidin-2-yl)amino]benzoic acidHuman2005
AURKA (AurA)AurOther3up7A2-({2-[(4-carboxyphenyl)amino]pyrimidin-4-yl}amino)benzoic acidHuman2025
AURKA (AurA)AurOther3vapA3-(1-{2-[(3-fluoropyridinium-4-yl)amino]-2-oxoethyl}-1h-pyrazol-4-yl)-6-methyl-8-[(3-{[(1r,3r)-3-methylpiperidinium-1-yl]methyl}-1,2-thiazol-5-yl)amino]imidazo[1,2-a]pyrazin-1-iumHuman2029
AURKA (AurA)AurOther3w10A1-(3-methoxyphenyl)-n-(5-methyl-1h-pyrazol-3-yl)isoquinolin-3-amineHuman2068
AURKA (AurA)AurOther3w16A4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-oneHuman2012
AURKA (AurA)AurOther3w18A2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamideHuman1961
AURKA (AurA)AurOther3w18B2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamideHuman1967
AURKA (AurA)AurOther3w2cA2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman2066
AURKA (AurA)AurOther3w2cC2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman2021
AURKA (AurA)AurOther3w2cE2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman1953
AURKA (AurA)AurOther3w2cG2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman2026
AURKA (AurA)AurOther4b0gAA6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridineHuman2082
AURKA (AurA)AurOther4b0gAB6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridineHuman2070
AURKA (AurA)AurOther4bn1AAadenosine-5'-diphosphateHuman1955
AURKA (AurA)AurOther4bn1ABadenosine-5'-diphosphateHuman1983
AURKA (AurA)AurOther4byiA(s)-n-((1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)methyl)acetamideHuman1992
AURKA (AurA)AurOther4byjA(s)-n-(1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)acetamideHuman1969
AURKA (AurA)AurOther4c3pAphosphomethylphosphonic acid adenylate esterHuman2018
AURKA (AurA)AurOther4c3pDphosphomethylphosphonic acid adenylate esterHuman2030
AURKA (AurA)AurOther4c3rAphosphomethylphosphonic acid adenylate esterHuman2058
AURKA (AurA)AurOther4cegAadenosine-5'-diphosphateHuman2073
AURKA (AurA)AurOther4deaA4,4'-(pyrimidine-2,4-diyldiimino)dibenzoic acidHuman2064
AURKA (AurA)AurOther4debA4-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzamideHuman1996
AURKA (AurA)AurOther4dedA2-({2-[(4-carbamoylphenyl)amino]pyrimidin-4-yl}amino)benzamideHuman2043
AURKA (AurA)AurOther4deeAadenosine-5'-diphosphateHuman1952
AURKA (AurA)AurOther4dhfA7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman1964
AURKA (AurA)AurOther4dhfB7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman1982
AURKA (AurA)AurOther4j8mA1-[4-[[4-[(5-cyclopentyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHuman2020
AURKA (AurA)AurOther4j8nA-Human2028
AURKA (AurA)AurOther4j8nB-Human2061
AURKA (AurA)AurOther4j8nC-Human2007
AURKA (AurA)AurOther4j8nD-Human1995
AURKA (AurA)AurOther4jaiAn-{4-[(6-oxo-5,6-dihydrobenzo[c][1,8]naphthyridin-1-yl)amino]phenyl}benzamideHuman1999
AURKA (AurA)AurOther4jajAbenzo[c][1,8]naphthyridin-6(5h)-oneHuman2040
AURKA (AurA)AurOther4jboA1-(4-{2-[(6-{4-[2-(dimethylamino)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHuman2072
AURKA (AurA)AurOther4jbpA1-(4-{2-[(6-{4-[2-(4-hydroxypiperidin-1-yl)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHuman2041
AURKA (AurA)AurOther4jbqAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman1957
AURKA (AurA)AurOther4o0sAadenosineHuman2039
AURKA (AurA)AurOther4o0uAadenosineHuman2022
AURKA (AurA)AurOther4o0wAadenosineHuman1959
AURKA (AurA)AurOther4prjAn-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman2023
AURKA (AurA)AurOther4uynAethyl (9s)-9-[5-(1h-benzimidazol-2-ylsulfanyl)furan-2-yl]-8-hydroxy-5,6,7,9-tetrahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHuman2002
AURKA (AurA)AurOther4uzdAethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHuman2013
AURKA (AurA)AurOther4uzdBethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHuman1968
AURKA (AurA)AurOther4uzhA(4s)-4-(2-fluorophenyl)-2,4,6,7,8,9-hexahydro-5h-pyrazolo[3,4-b][1,7]naphthyridin-5-oneHuman1998
AURKA (AurA)AurOther4zs0A5-hydroxy-1'h-1,2'-bibenzimidazol-2(3h)-oneHuman6801
AURKA (AurA)AurOther4ztqA(2z,5z)-2-[(4-ethylphenyl)imino]-3-(2-methoxyethyl)-5-(pyridin-4-ylmethylidene)-1,3-thiazolidin-4-oneHuman6804
AURKA (AurA)AurOther4ztrA6-({4-[(z)-{(2z)-2-[(4-ethylphenyl)imino]-3-methyl-4-oxo-1,3-thiazolidin-5-ylidene}methyl]pyridin-2-yl}amino)pyridine-3-carboxylic acidHuman6817
AURKA (AurA)AurOther4ztsA(2z,5z)-2-[(4-ethylphenyl)imino]-3-methyl-5-[(2-{[4-(1h-tetrazol-5-yl)phenyl]amino}pyridin-4-yl)methylidene]-1,3-thiazolidin-4-oneHuman6814
AURKA (AurA)AurOther5aadA7-(1-benzyl-1h-pyrazol-4-yl)-6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridineHuman6011
AURKA (AurA)AurOther5aaeA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-5-methylisoxazoleHuman6012
AURKA (AurA)AurOther5aafA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-n,n-dimethylbenzamideHuman6013
AURKA (AurA)AurOther5aagA[3-[[4-[6-chloranyl-2-(1,3-dimethylpyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl]pyrazol-1-yl]methyl]phenyl]-(4-methylpiperazin-1-yl)methanoneHuman6010
AURKA (AurA)AurOther5dn3AAadenosine-5'-triphosphateHuman6802
AURKA (AurA)AurOther5dn3ABadenosine-5'-triphosphateHuman6818
AURKA (AurA)AurOther5dnrAAadenosine-5'-triphosphateHuman6810
AURKA (AurA)AurOther5dnrABadenosine-5'-triphosphateHuman6809
AURKA (AurA)AurOther5dosAadenosine-5'-triphosphateHuman6807
AURKA (AurA)AurOther5dpvAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6808
AURKA (AurA)AurOther5dpvAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6826
AURKA (AurA)AurOther5dr2Aadenosine-5'-triphosphateHuman6825
AURKA (AurA)AurOther5dr6AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6811
AURKA (AurA)AurOther5dr6AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6805
AURKA (AurA)AurOther5dr9A4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6821
AURKA (AurA)AurOther5drdAadenosine-5'-triphosphateHuman6823
AURKA (AurA)AurOther5dt0AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6806
AURKA (AurA)AurOther5dt0AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6803
AURKA (AurA)AurOther5dt3Aadenosine-5'-triphosphateHuman6816
AURKA (AurA)AurOther5dt4Aadenosine-5'-triphosphateHuman6815
AURKA (AurA)AurOther5ew9AA4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHuman6359
AURKA (AurA)AurOther5ew9AB4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHuman6360
AURKA (AurA)AurOther5g15AAphosphomethylphosphonic acid adenylate esterHuman9737
AURKA (AurA)AurOther5g15ABphosphomethylphosphonic acid adenylate esterHuman9739
AURKA (AurA)AurOther5g1xAAadenosine-5'-diphosphateHuman7267
AURKA (AurA)AurOther5g1xABadenosine-5'-diphosphateHuman7266
AURKA (AurA)AurOther5l8jAAadenosine-5'-diphosphateHuman6820
AURKA (AurA)AurOther5l8jABadenosine-5'-diphosphateHuman6812
AURKA (AurA)AurOther5l8kAAadenosine-5'-diphosphateHuman6819
AURKA (AurA)AurOther5l8kABadenosine-5'-diphosphateHuman6813
AURKA (AurA)AurOther5l8lAAadenosine-5'-diphosphateHuman6822
AURKA (AurA)AurOther5l8lABadenosine-5'-diphosphateHuman6824
AURKA (AurA)AurOther5lxmAAadenosine-5'-diphosphateHuman7142
AURKA (AurA)AurOther5lxmABadenosine-5'-diphosphateHuman7141
AURKA (AurA)AurOther5objAadenosine-5'-triphosphateHuman8305
AURKA (AurA)AurOther5obrA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8304
AURKA (AurA)AurOther5odtAAadenosine-5'-diphosphateHuman9738
AURKA (AurA)AurOther5odtABadenosine-5'-diphosphateHuman9736
AURKA (AurA)AurOther5oneAA4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamideHuman8371
AURKA (AurA)AurOther5oneAB4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamideHuman8370
AURKA (AurA)AurOther5orlAadenosine-5'-diphosphateHuman8642
AURKA (AurA)AurOther5ornAadenosine-5'-diphosphateHuman8649
AURKA (AurA)AurOther5oroAadenosine-5'-diphosphateHuman8641
AURKA (AurA)AurOther5orpAadenosine-5'-diphosphateHuman8648
AURKA (AurA)AurOther5orrAadenosine-5'-diphosphateHuman8636
AURKA (AurA)AurOther5orsAadenosine-5'-diphosphateHuman8646
AURKA (AurA)AurOther5ortAadenosine-5'-diphosphateHuman8638
AURKA (AurA)AurOther5orvAadenosine-5'-diphosphateHuman8643
AURKA (AurA)AurOther5orwAadenosine-5'-diphosphateHuman8631
AURKA (AurA)AurOther5orxAadenosine-5'-diphosphateHuman8644
AURKA (AurA)AurOther5oryAadenosine-5'-diphosphateHuman8627
AURKA (AurA)AurOther5orzAAadenosine-5'-diphosphateHuman8639
AURKA (AurA)AurOther5orzABadenosine-5'-diphosphateHuman8650
AURKA (AurA)AurOther5os0Aadenosine-5'-diphosphateHuman8632
AURKA (AurA)AurOther5os1AAadenosine-5'-diphosphateHuman8628
AURKA (AurA)AurOther5os1ABadenosine-5'-diphosphateHuman8630
AURKA (AurA)AurOther5os2AAadenosine-5'-diphosphateHuman8635
AURKA (AurA)AurOther5os2ABadenosine-5'-diphosphateHuman8633
AURKA (AurA)AurOther5os3Aadenosine-5'-diphosphateHuman8637
AURKA (AurA)AurOther5os4Aadenosine-5'-diphosphateHuman8652
AURKA (AurA)AurOther5os5AAadenosine-5'-diphosphateHuman8647
AURKA (AurA)AurOther5os5ABadenosine-5'-diphosphateHuman8629
AURKA (AurA)AurOther5os6Aadenosine-5'-diphosphateHuman8651
AURKA (AurA)AurOther5osdAadenosine-5'-diphosphateHuman8634
AURKA (AurA)AurOther5oseAadenosine-5'-diphosphateHuman8645
AURKA (AurA)AurOther5osfAadenosine-5'-diphosphateHuman8640
AURKA (AurA)AurOther5zanA7-(4-methylpiperazin-1-yl)-n-(5-methyl-1h-pyrazol-3-yl)-2-[(e)-2-phenylethenyl]quinazolin-4-amineHuman10898
AURKA (AurA)AurOther6c2rAA(2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acidHuman10864
AURKA (AurA)AurOther6c2rAB(2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acidHuman10865
AURKA (AurA)AurOther6c2tAA(2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acidHuman10866
AURKA (AurA)AurOther6c2tAB(2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acidHuman10863
AURKA (AurA)AurOther6c83Aphosphomethylphosphonic acid adenylate esterHuman10934
AURKA (AurA)AurOther6c83Bphosphomethylphosphonic acid adenylate esterHuman10935
AURKA (AurA)AurOther6cpeAA-Human10036
AURKA (AurA)AurOther6cpeAB-Human10035
AURKA (AurA)AurOther6cpfAphosphomethylphosphonic acid adenylate esterHuman10033
AURKA (AurA)AurOther6cpgA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10032
AURKA (AurA)AurOther6cpgD1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10034
AURKA (AurA)AurOther6graA1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)ureaHuman11130
AURKA (AurA)AurOther6hjjAA~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamideHuman10410
AURKA (AurA)AurOther6hjjAB~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamideHuman10412
AURKA (AurA)AurOther6hjkA(~{e})-~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-but-2-enamideHuman10411
AURKA (AurA)AurOther6i2uA-Human11652
AURKA (AurA)AurOther6r49Aadenosine-5'-diphosphateHuman11131
AURKA (AurA)AurOther6r4aAadenosine-5'-diphosphateHuman11134
AURKA (AurA)AurOther6r4bABadenosine-5'-diphosphateHuman11133
AURKA (AurA)AurOther6r4cAadenosine-5'-diphosphateHuman11135
AURKA (AurA)AurOther6r4dAadenosine-5'-diphosphateHuman11132
AURKA (AurA)AurOther6vpgAAphosphoaminophosphonic acid-adenylate esterHuman12659
AURKA (AurA)AurOther6vpgABphosphoaminophosphonic acid-adenylate esterHuman12667
AURKA (AurA)AurOther6vphAAdithiane diolHuman12666
AURKA (AurA)AurOther6vphABdithiane diolHuman12655
AURKA (AurA)AurOther6vpiAAphosphoaminophosphonic acid-adenylate esterHuman12656
AURKA (AurA)AurOther6vpiABphosphoaminophosphonic acid-adenylate esterHuman12669
AURKA (AurA)AurOther6vpjAAphosphoaminophosphonic acid-adenylate esterHuman12657
AURKA (AurA)AurOther6vpjABphosphoaminophosphonic acid-adenylate esterHuman12654
AURKA (AurA)AurOther6vplAAphosphoaminophosphonic acid-adenylate esterHuman12662
AURKA (AurA)AurOther6vplABphosphoaminophosphonic acid-adenylate esterHuman12670
AURKA (AurA)AurOther6vplBAphosphoaminophosphonic acid-adenylate esterHuman12664
AURKA (AurA)AurOther6vplBBphosphoaminophosphonic acid-adenylate esterHuman12668
AURKA (AurA)AurOther6vpmAAadenosine monophosphateHuman12661
AURKA (AurA)AurOther6vpmABadenosine monophosphateHuman12658
AURKA (AurA)AurOther6vpmBAadenosine monophosphateHuman12660
AURKA (AurA)AurOther6vpmBBadenosine monophosphateHuman12663
AURKA (AurA)AurOther6xkaA-Human12665
AURKA (AurA)AurOther6z4yAA6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12306
AURKA (AurA)AurOther6z4yAB6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12307
AURKA (AurA)AurOther7ayhA7-[2-[(4-methoxyphenyl)amino]pyrimidin-4-yl]-1,3,4,5-tetrahydro-1-benzazepin-2-oneHuman13228
AURKA (AurA)AurOther7ayiA7-(2-phenylazanylpyrimidin-4-yl)-1,3,4,5-tetrahydro-1-benzazepin-2-oneHuman13229
AURKA (AurA)AurOther7ficAA6-[(5-cyclopropyl-1~{h}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{n}-prop-2-ynyl-pyrimidine-4-carboxamideHuman14234
AURKA (AurA)AurOther7ficAB6-[(5-cyclopropyl-1~{h}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{n}-prop-2-ynyl-pyrimidine-4-carboxamideHuman14233
AURKA (AurA)AurOther7o2vA1-[[3,4-bis(fluoranyl)phenyl]methyl]-~{n}-[(1~{r})-2-[[(3~{e})-3-(1~{h}-imidazol-5-ylmethylidene)-2-oxidanylidene-1~{h}-indol-5-yl]amino]-2-oxidanylidene-1-phenyl-ethyl]-6-methyl-2-oxidanylidene-pyridine-3-carboxamideHuman13947
AURKA (AurA)AurOther7ztlAAadenosine-5'-diphosphateHuman14582
AURKA (AurA)AurOther7ztlABadenosine-5'-diphosphateHuman14581
AURKA (AurA)AurOther8c14AAadenosine-5'-diphosphateHuman15143
AURKA (AurA)AurOther8c14ABadenosine-5'-diphosphateHuman15150
AURKA (AurA)AurOther8c15AAadenosine-5'-diphosphateHuman15141
AURKA (AurA)AurOther8c15ABadenosine-5'-diphosphateHuman15151
AURKA (AurA)AurOther8c1dAAadenosine-5'-diphosphateHuman15152
AURKA (AurA)AurOther8c1dABadenosine-5'-diphosphateHuman15138
AURKA (AurA)AurOther8c1eAadenosine-5'-triphosphateHuman15145
AURKA (AurA)AurOther8c1fAAadenosine-5'-diphosphateHuman15140
AURKA (AurA)AurOther8c1fABadenosine-5'-diphosphateHuman15149
AURKA (AurA)AurOther8c1gAadenosine-5'-diphosphateHuman15148
AURKA (AurA)AurOther8c1hAAadenosine-5'-diphosphateHuman15147
AURKA (AurA)AurOther8c1hABadenosine-5'-diphosphateHuman15142
AURKA (AurA)AurOther8c1iAAadenosine-5'-diphosphateHuman15144
AURKA (AurA)AurOther8c1iABadenosine-5'-diphosphateHuman15139
AURKA (AurA)AurOther8c1kAadenosine-5'-diphosphateHuman15146
AURKA (AurA)AurOther8c1mAadenosine-5'-diphosphateHuman15137
AURKA (AurA)AurOther8guwAadenosine-5'-diphosphateHuman14753
AURKA (AurA)AurOther8jmxA5-(4-morpholin-4-yl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2-oxidanyl-benzaldehydeHuman14864
AURKA (AurA)AurOther8ssoAAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14866
AURKA (AurA)AurOther8ssoABn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14867
AURKA (AurA)AurOther8ssoACn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14863
AURKA (AurA)AurOther8sspAAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14868
AURKA (AurA)AurOther8sspABn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14865
AURKB (AurB)AurOther4af3Acyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman407
AURKC (AurC)AurOther6gr8AA1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)ureaHuman11122
AURKC (AurC)AurOther6gr8AB1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)ureaHuman11125
AURKC (AurC)AurOther6gr9AAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman11123
AURKC (AurC)AurOther6gr9ABcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman11124
AXLAxlTK5u6bA(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8258
AXLAxlTK5u6bB(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8260
AXLAxlTK5u6bC(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8257
AXLAxlTK5u6bD(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8259
BMP2K (BIKE)NAKOther4w9wAA5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman3274
BMP2K (BIKE)NAKOther4w9wAB5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman3272
BMP2K (BIKE)NAKOther4w9xAbaricitinibHuman3273
BMP2K (BIKE)NAKOther5i3oAn-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamideHuman6437
BMP2K (BIKE)NAKOther5i3oBn-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamideHuman6434
BMP2K (BIKE)NAKOther5i3rAn-[6-(3-{[(cyclopropylmethyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]cyclopropanecarboxamideHuman6435
BMP2K (BIKE)NAKOther5i3rBn-[6-(3-{[(cyclopropylmethyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]cyclopropanecarboxamideHuman6436
BMP2K (BIKE)NAKOther5ikwAn-(6-{3-[(cyclopropylsulfonyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamideHuman6709
BMPR1BSTKRTKL3mdyAA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1502
BMPR1BSTKRTKL3mdyAB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1501
BMPR1BSTKRTKL3mdyCA4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1503
BMPR1BSTKRTKL3mdyCB4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineHuman1500
BMPR2STKRTKL3g2fAAadenosine-5'-diphosphateHuman6870
BMPR2STKRTKL3g2fABadenosine-5'-diphosphateHuman6868
BMPR2STKRTKL3g2fBAadenosine-5'-diphosphateHuman6867
BMPR2STKRTKL3g2fBBadenosine-5'-diphosphateHuman6869
BMPR2STKRTKL6unpAAadenosine-5'-diphosphateHuman13795
BMPR2STKRTKL6unpABadenosine-5'-diphosphateHuman13794
BMXTecTK3sxrAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman3482
BMXTecTK3sxrBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman3481
BMXTecTK3sxsA1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamineHuman3483
BMXTecTK6i99A~{n}-[2-methyl-5-[8-[4-(methylsulfonylamino)phenyl]-2-oxidanylidene-benzo[h][1,6]naphthyridin-1-yl]phenyl]-3-oxidanyl-propanamideHuman12348
BMXTecTK6i99B~{n}-[2-methyl-5-[8-[4-(methylsulfonylamino)phenyl]-2-oxidanylidene-benzo[h][1,6]naphthyridin-1-yl]phenyl]-3-oxidanyl-propanamideHuman12349
BMXTecTK8x2aAA4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamideHuman15131
BMXTecTK8x2aAB4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamideHuman15130
BRAFRAFTKL1uwhA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3127
BRAFRAFTKL1uwhB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3109
BRAFRAFTKL1uwjA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3135
BRAFRAFTKL1uwjB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3105
BRAFRAFTKL2fb8A(1z)-5-(2-{4-[2-(dimethylamino)ethoxy]phenyl}-5-pyridin-4-yl-1h-imidazol-4-yl)indan-1-one oximeHuman3062
BRAFRAFTKL2fb8B(1z)-5-(2-{4-[2-(dimethylamino)ethoxy]phenyl}-5-pyridin-4-yl-1h-imidazol-4-yl)indan-1-one oximeHuman3086
BRAFRAFTKL3c4cAn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamideHuman3115
BRAFRAFTKL3c4cBn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamideHuman3063
BRAFRAFTKL3d4qA(1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oximeHuman3095
BRAFRAFTKL3d4qB(1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oximeHuman3060
BRAFRAFTKL3idpAn~1~-(4-chlorophenyl)-6-methyl-n~5~-[3-(7h-purin-6-yl)pyridin-2-yl]isoquinoline-1,5-diamineHuman3077
BRAFRAFTKL3idpBn~1~-(4-chlorophenyl)-6-methyl-n~5~-[3-(7h-purin-6-yl)pyridin-2-yl]isoquinoline-1,5-diamineHuman3121
BRAFRAFTKL3ii5An-[3-(3-{4-[(dimethylamino)methyl]phenyl}pyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-3-(trifluoromethyl)benzamideHuman3116
BRAFRAFTKL3ii5Bn-[3-(3-{4-[(dimethylamino)methyl]phenyl}pyrazolo[1,5-a]pyrimidin-7-yl)phenyl]-3-(trifluoromethyl)benzamideHuman3076
BRAFRAFTKL3og7An-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman3113
BRAFRAFTKL3og7B-Human3140
BRAFRAFTKL3ppjAmethyl 3-{[(5s)-1-(hydroxyamino)-5h-inden-5-yl]amino}furo[2,3-c]pyridine-2-carboxylateHuman3091
BRAFRAFTKL3ppjBmethyl 3-{[(5s)-1-(hydroxyamino)-5h-inden-5-yl]amino}furo[2,3-c]pyridine-2-carboxylateHuman3087
BRAFRAFTKL3ppkA3-[(5-hydroxynaphthalen-2-yl)amino]-n-(pyrimidin-4-yl)furo[2,3-c]pyridine-2-carboxamideHuman3106
BRAFRAFTKL3ppkB3-[(5-hydroxynaphthalen-2-yl)amino]-n-(pyrimidin-4-yl)furo[2,3-c]pyridine-2-carboxamideHuman3092
BRAFRAFTKL3prfA2-chloro-5-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}phenolHuman3129
BRAFRAFTKL3prfB2-chloro-5-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}phenolHuman3139
BRAFRAFTKL3priA3-(4-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}-1h-indazol-3-yl)propan-1-olHuman3093
BRAFRAFTKL3priB3-(4-{[2-(pyrimidin-2-yl)furo[2,3-c]pyridin-3-yl]amino}-1h-indazol-3-yl)propan-1-olHuman3103
BRAFRAFTKL3psbAethyl 3-{[1-(hydroxyamino)-2h-inden-5-yl]amino}thieno[2,3-c]pyridine-2-carboxylateHuman3111
BRAFRAFTKL3psbBethyl 3-{[1-(hydroxyamino)-2h-inden-5-yl]amino}thieno[2,3-c]pyridine-2-carboxylateHuman3125
BRAFRAFTKL3psdA6-[1-(piperidin-4-yl)-3-(pyridin-4-yl)-1h-pyrazol-4-yl]indeno[1,2-c]pyrazoleHuman3142
BRAFRAFTKL3psdB6-[1-(piperidin-4-yl)-3-(pyridin-4-yl)-1h-pyrazol-4-yl]indeno[1,2-c]pyrazoleHuman3083
BRAFRAFTKL3q4cA[(1,2,3,4,5,6-eta)-(1s,2r,3r,4r,5s,6s)-1-carboxycyclohexane-1,2,3,4,5,6-hexayl](chloro)(3-methyl-5,7-dioxo-6,7-dihydro-5h-pyrido[2,3-a]pyrrolo[3,4-c]carbazol-12-ide-kappa~2~n~1~,n~12~)ruthenium(1+)Human7251
BRAFRAFTKL3q4cB-Human7250
BRAFRAFTKL3q96A(2s)-n-[3-(2-aminopropan-2-yl)-5-(trifluoromethyl)phenyl]-7-[(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-4-yl)oxy]-1,2,3,4-tetrahydronaphthalene-2-carboxamideHuman3072
BRAFRAFTKL3q96B(2s)-n-[3-(2-aminopropan-2-yl)-5-(trifluoromethyl)phenyl]-7-[(7-oxo-5,6,7,8-tetrahydro-1,8-naphthyridin-4-yl)oxy]-1,2,3,4-tetrahydronaphthalene-2-carboxamideHuman3089
BRAFRAFTKL3skcA2,6-difluoro-n-[(5s)-3-methoxy-5h-pyrazolo[3,4-b]pyridin-5-yl]-3-[(phenylsulfonyl)amino]benzamideHuman3100
BRAFRAFTKL3skcB2,6-difluoro-n-[(5s)-3-methoxy-5h-pyrazolo[3,4-b]pyridin-5-yl]-3-[(phenylsulfonyl)amino]benzamideHuman3128
BRAFRAFTKL3tv4An-(6-amino-5-bromopyridin-3-yl)-2,6-difluoro-3-[(propylsulfonyl)amino]benzamideHuman3054
BRAFRAFTKL3tv4Bn-(6-amino-5-bromopyridin-3-yl)-2,6-difluoro-3-[(propylsulfonyl)amino]benzamideHuman3133
BRAFRAFTKL3tv6A2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)-3-[(propylsulfonyl)amino]benzamideHuman3080
BRAFRAFTKL3tv6B2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)-3-[(propylsulfonyl)amino]benzamideHuman3136
BRAFRAFTKL4cqeAn-{4-[2-(1-cyclopropylpiperidin-4-yl)-4-(3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)-1,3-thiazol-5-yl]pyridin-2-yl}acetamideHuman3088
BRAFRAFTKL4cqeBn-{4-[2-(1-cyclopropylpiperidin-4-yl)-4-(3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)-1,3-thiazol-5-yl]pyridin-2-yl}acetamideHuman3107
BRAFRAFTKL4dbnA2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamideHuman3052
BRAFRAFTKL4dbnB2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamideHuman3070
BRAFRAFTKL4e26A5-chloro-7-[(r)-furan-2-yl(pyridin-2-ylamino)methyl]quinolin-8-olHuman3108
BRAFRAFTKL4e26B5-chloro-7-[(r)-furan-2-yl(pyridin-2-ylamino)methyl]quinolin-8-olHuman3102
BRAFRAFTKL4e4xAn-(2,4-difluoro-3-{2-[(3-hydroxypropyl)amino]-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl}phenyl)propane-1-sulfonamideHuman3051
BRAFRAFTKL4e4xBn-(2,4-difluoro-3-{2-[(3-hydroxypropyl)amino]-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl}phenyl)propane-1-sulfonamideHuman3104
BRAFRAFTKL4eheA4-amino-n-{2,6-difluoro-3-[(propylsulfonyl)amino]phenyl}thieno[3,2-d]pyrimidine-7-carboxamideHuman3112
BRAFRAFTKL4eheB4-amino-n-{2,6-difluoro-3-[(propylsulfonyl)amino]phenyl}thieno[3,2-d]pyrimidine-7-carboxamideHuman3082
BRAFRAFTKL4ehgAn-{2,4-difluoro-3-[({6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}carbamoyl)amino]phenyl}propane-1-sulfonamideHuman3064
BRAFRAFTKL4ehgBn-{2,4-difluoro-3-[({6-[(2-hydroxyethyl)amino]pyrimidin-4-yl}carbamoyl)amino]phenyl}propane-1-sulfonamideHuman3078
BRAFRAFTKL4fc0A2-chloro-3-[(2-cyanopropan-2-yl)oxy]-n-{5-[{2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}(methyl)amino]-2-fluorophenyl}benzamideHuman3131
BRAFRAFTKL4fc0B2-chloro-3-[(2-cyanopropan-2-yl)oxy]-n-{5-[{2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}(methyl)amino]-2-fluorophenyl}benzamideHuman3069
BRAFRAFTKL4fk3An-{2,4-difluoro-3-[(5-pyridin-3-yl-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]phenyl}ethanesulfonamideHuman3118
BRAFRAFTKL4fk3B-Human3068
BRAFRAFTKL4g9cA3-{[3-(2-cyanopropan-2-yl)benzoyl]amino}-2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)benzamideHuman3084
BRAFRAFTKL4g9cB3-{[3-(2-cyanopropan-2-yl)benzoyl]amino}-2,6-difluoro-n-(3-methoxy-2h-pyrazolo[3,4-b]pyridin-5-yl)benzamideHuman3067
BRAFRAFTKL4g9rA3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman3130
BRAFRAFTKL4g9rB3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman3101
BRAFRAFTKL4h58AAn-(4-{[(2-methoxyethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)quinazolin-2-amineHuman3137
BRAFRAFTKL4h58ABn-(4-{[(2-methoxyethyl)amino]methyl}phenyl)-6-(pyridin-4-yl)quinazolin-2-amineHuman3110
BRAFRAFTKL4h58BA-Human3097
BRAFRAFTKL4h58BB-Human3120
BRAFRAFTKL4h58CA-Human3056
BRAFRAFTKL4h58CB-Human3114
BRAFRAFTKL4jvgA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman3134
BRAFRAFTKL4jvgB1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman3085
BRAFRAFTKL4jvgC1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman3050
BRAFRAFTKL4jvgD1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman3059
BRAFRAFTKL4kspAn-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]acetyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamideHuman3081
BRAFRAFTKL4kspBn-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]acetyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamideHuman3066
BRAFRAFTKL4ksqAn-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamideHuman3065
BRAFRAFTKL4ksqBn-{7-cyano-6-[4-fluoro-3-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]-1,3-benzothiazol-2-yl}cyclopropanecarboxamideHuman3055
BRAFRAFTKL4mbjA2,6-difluoro-n-(1h-imidazo[4,5-b]pyridin-6-yl)-3-[(propylsulfonyl)amino]benzamideHuman3090
BRAFRAFTKL4mbjB2,6-difluoro-n-(1h-imidazo[4,5-b]pyridin-6-yl)-3-[(propylsulfonyl)amino]benzamideHuman3057
BRAFRAFTKL4mneBA-Human3075
BRAFRAFTKL4mneBB-Human3061
BRAFRAFTKL4mneCA-Human3122
BRAFRAFTKL4mneCB-Human3058
BRAFRAFTKL4mneFA-Human3099
BRAFRAFTKL4mneFB-Human3117
BRAFRAFTKL4mneGA-Human3071
BRAFRAFTKL4mneGB-Human3073
BRAFRAFTKL4mnfAA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman3096
BRAFRAFTKL4mnfAB2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman3141
BRAFRAFTKL4mnfBA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman3124
BRAFRAFTKL4mnfBB2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman3098
BRAFRAFTKL4pp7An-{2,4-difluoro-3-[methyl(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamideHuman3094
BRAFRAFTKL4pp7Bn-{2,4-difluoro-3-[methyl(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamideHuman3126
BRAFRAFTKL4r5yA5-({(1r,1as,6br)-1-[5-(trifluoromethyl)-1h-benzimidazol-2-yl]-1a,6b-dihydro-1h-cyclopropa[b][1]benzofuran-5-yl}oxy)-3,4-dihydro-1,8-naphthyridin-2(1h)-oneHuman6414
BRAFRAFTKL4r5yB5-({(1r,1as,6br)-1-[5-(trifluoromethyl)-1h-benzimidazol-2-yl]-1a,6b-dihydro-1h-cyclopropa[b][1]benzofuran-5-yl}oxy)-3,4-dihydro-1,8-naphthyridin-2(1h)-oneHuman6413
BRAFRAFTKL4rzvAn-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6944
BRAFRAFTKL4rzvBn-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6941
BRAFRAFTKL4rzwA3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6939
BRAFRAFTKL4rzwB3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6942
BRAFRAFTKL4wo5An-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamideHuman3079
BRAFRAFTKL4wo5Bn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}propane-1-sulfonamideHuman3143
BRAFRAFTKL4xv1An'-(3-{[5-(2-cyclopropylpyrimidin-5-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)-n-ethyl-n-methylsulfuric diamideHuman6214
BRAFRAFTKL4xv1B-Human6216
BRAFRAFTKL4xv2AdabrafenibHuman6213
BRAFRAFTKL4xv2BdabrafenibHuman6219
BRAFRAFTKL4xv3An'-{3-[5-(2-aminopyrimidin-4-yl)-2-tert-butyl-1,3-thiazol-4-yl]-2-fluorophenyl}-n-ethyl-n-methylsulfuric diamideHuman6217
BRAFRAFTKL4xv3B-Human6218
BRAFRAFTKL4xv9AAn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}-4-(trifluoromethyl)benzenesulfonamideHuman6220
BRAFRAFTKL4xv9ABn-{3-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-difluorophenyl}-4-(trifluoromethyl)benzenesulfonamideHuman6215
BRAFRAFTKL4yhtA3-[(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6442
BRAFRAFTKL4yhtB3-[(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6443
BRAFRAFTKL5c9cAA1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman3123
BRAFRAFTKL5c9cAB1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman3074
BRAFRAFTKL5c9cBA1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman3138
BRAFRAFTKL5c9cBB1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman3119
BRAFRAFTKL5cswAdabrafenibHuman6433
BRAFRAFTKL5cswBdabrafenibHuman6431
BRAFRAFTKL5csxAn-(3-{5-[(1-ethylpiperidin-4-yl)(methyl)amino]-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-1-yl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6432
BRAFRAFTKL5ct7A1-methyl-5-({2-[5-(trifluoromethyl)-1h-imidazol-2-yl]pyridin-4-yl}oxy)-n-[4-(trifluoromethyl)phenyl]-1h-benzimidazol-2-amineHuman6032
BRAFRAFTKL5ct7B1-methyl-5-({2-[5-(trifluoromethyl)-1h-imidazol-2-yl]pyridin-4-yl}oxy)-n-[4-(trifluoromethyl)phenyl]-1h-benzimidazol-2-amineHuman6033
BRAFRAFTKL5fd2A6-[2-[[3-(dimethylsulfamoylamino)-2,6-bis(fluoranyl)phenyl]amino]pyridin-3-yl]-7~{h}-purineHuman6603
BRAFRAFTKL5fd2B6-[2-[[3-(dimethylsulfamoylamino)-2,6-bis(fluoranyl)phenyl]amino]pyridin-3-yl]-7~{h}-purineHuman6602
BRAFRAFTKL5hi2A4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman6515
BRAFRAFTKL5hidAA3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6506
BRAFRAFTKL5hidAB3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6512
BRAFRAFTKL5hidBA3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6511
BRAFRAFTKL5hidBB3-(2-cyanopropan-2-yl)-n-{4-methyl-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}benzamideHuman6517
BRAFRAFTKL5hieAAdabrafenibHuman6516
BRAFRAFTKL5hieABdabrafenibHuman6508
BRAFRAFTKL5hieBAdabrafenibHuman6509
BRAFRAFTKL5hieBBdabrafenibHuman6505
BRAFRAFTKL5hieCAdabrafenibHuman6513
BRAFRAFTKL5hieCBdabrafenibHuman6507
BRAFRAFTKL5hieDAdabrafenibHuman6510
BRAFRAFTKL5hieDBdabrafenibHuman6514
BRAFRAFTKL5itaAn-{2-cyano-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamideHuman6940
BRAFRAFTKL5itaBn-{2-cyano-3-[(3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]phenyl}propane-1-sulfonamideHuman6943
BRAFRAFTKL5jrqA(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)[5-(4-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methanoneHuman7061
BRAFRAFTKL5jrqB(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)[5-(4-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methanoneHuman7054
BRAFRAFTKL5jsmAA-Human7056
BRAFRAFTKL5jsmAB-Human7058
BRAFRAFTKL5jsmBAn,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide)Human7060
BRAFRAFTKL5jsmBBn,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide)Human7062
BRAFRAFTKL5jsmCAn,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide)Human7059
BRAFRAFTKL5jsmCBn,n'-{ethane-1,2-diylbis[oxyethane-2,1-diyloxy-4,1-phenylene-1h-pyrrolo[2,3-b]pyridine-5,3-diylcarbonyl(2,4-difluoro-3,1-phenylene)]}di(propane-1-sulfonamide)Human7063
BRAFRAFTKL5jsmDA-Human7055
BRAFRAFTKL5jsmDB-Human7053
BRAFRAFTKL5jt2A2,2'-oxybis[n-({4-[3-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorobenzene-1-carbonyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]phenyl}methyl)acetamide]Human7065
BRAFRAFTKL5jt2B-Human7057
BRAFRAFTKL5jt2C2,2'-oxybis[n-({4-[3-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorobenzene-1-carbonyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]phenyl}methyl)acetamide]Human7064
BRAFRAFTKL5jt2D-Human7066
BRAFRAFTKL5valAn-(3-tert-butylphenyl)-4-methyl-3-[6-(morpholin-4-yl)pyrimidin-4-yl]benzamideHuman8190
BRAFRAFTKL5valBn-(3-tert-butylphenyl)-4-methyl-3-[6-(morpholin-4-yl)pyrimidin-4-yl]benzamideHuman8188
BRAFRAFTKL5vamAAn-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamideHuman8185
BRAFRAFTKL5vamABn-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamideHuman8189
BRAFRAFTKL5vamBAn-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamideHuman8186
BRAFRAFTKL5vamBBn-{2-methyl-5'-(morpholin-4-yl)-6'-[(oxan-4-yl)oxy][3,3'-bipyridin]-5-yl}-3-(trifluoromethyl)benzamideHuman8187
BRAFRAFTKL6b8uA~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8679
BRAFRAFTKL6b8uB~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8678
BRAFRAFTKL6cadA1-(propan-2-yl)-3-({3-[3-(trifluoromethyl)phenyl]isoquinolin-8-yl}ethynyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9576
BRAFRAFTKL6cadB1-(propan-2-yl)-3-({3-[3-(trifluoromethyl)phenyl]isoquinolin-8-yl}ethynyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9575
BRAFRAFTKL6n0pAAn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman11597
BRAFRAFTKL6n0pABn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman11596
BRAFRAFTKL6n0pBAn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman11594
BRAFRAFTKL6n0pBBn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman11595
BRAFRAFTKL6n0qAAn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHuman11771
BRAFRAFTKL6n0qABn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHuman11768
BRAFRAFTKL6n0qBAn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHuman11770
BRAFRAFTKL6n0qBBn-[4-methyl-3-(1-methyl-2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)phenyl]-3-(trifluoromethyl)benzamideHuman11769
BRAFRAFTKL6nsqA5-[(4-amino-1-ethyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-n-(4-chlorophenyl)-6-methylisoquinolin-1-amineHuman11328
BRAFRAFTKL6nsqB5-[(4-amino-1-ethyl-1h-pyrazolo[3,4-d]pyrimidin-3-yl)ethynyl]-n-(4-chlorophenyl)-6-methylisoquinolin-1-amineHuman11329
BRAFRAFTKL6nybAphosphothiophosphoric acid-adenylate esterHuman11708
BRAFRAFTKL6p3dA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman12809
BRAFRAFTKL6p7gA3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHuman12810
BRAFRAFTKL6p7gB3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHuman12806
BRAFRAFTKL6p7gC3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHuman12807
BRAFRAFTKL6p7gD3-[(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-n-[4-({[2-(morpholin-4-yl)ethyl]amino}methyl)-3-(trifluoromethyl)phenyl]benzamideHuman12808
BRAFRAFTKL6pp9AAphosphoaminophosphonic acid-adenylate esterHuman11711
BRAFRAFTKL6pp9ABphosphoaminophosphonic acid-adenylate esterHuman11709
BRAFRAFTKL6q0jAA-Human11704
BRAFRAFTKL6q0jAB-Human11701
BRAFRAFTKL6q0jBA-Human11703
BRAFRAFTKL6q0jBB-Human11712
BRAFRAFTKL6q0kA-Human11706
BRAFRAFTKL6q0kB-Human11710
BRAFRAFTKL6q0tAA-Human11705
BRAFRAFTKL6q0tAB-Human11707
BRAFRAFTKL6q0tBA-Human11702
BRAFRAFTKL6q0tBB-Human11700
BRAFRAFTKL6u2gBphosphomethylphosphonic acid adenylate esterHuman11567
BRAFRAFTKL6u2hCA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman11568
BRAFRAFTKL6u2hDA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman11569
BRAFRAFTKL6uanB-Human11641
BRAFRAFTKL6uanC-Human11642
BRAFRAFTKL6uuoA1-[4-{[1-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-5-yl](methyl)amino}pyridin-1(4h)-yl]ethan-1-oneHuman12347
BRAFRAFTKL6uuoB1-[4-{[1-(3-{[dihydroxy(propyl)-lambda~4~-sulfanyl]amino}-2,6-difluorophenyl)-3-(pyrimidin-5-yl)-1h-pyrrolo[3,2-b]pyridin-5-yl](methyl)amino}pyridin-1(4h)-yl]ethan-1-oneHuman12346
BRAFRAFTKL6v2uAdabrafenibHuman13034
BRAFRAFTKL6v2uBdabrafenibHuman13031
BRAFRAFTKL6v2wAAphosphoaminophosphonic acid-adenylate esterHuman13026
BRAFRAFTKL6v2wABphosphoaminophosphonic acid-adenylate esterHuman13032
BRAFRAFTKL6v34A6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamideHuman13200
BRAFRAFTKL6v34B6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamideHuman13199
BRAFRAFTKL6xagCA-Human12922
BRAFRAFTKL6xagDA-Human12921
BRAFRAFTKL6xfpAA4-amino-n-{1-[(3-chloro-2-fluorophenyl)amino]-6-methylisoquinolin-5-yl}thieno[3,2-d]pyrimidine-7-carboxamideHuman13403
BRAFRAFTKL6xfpAB4-amino-n-{1-[(3-chloro-2-fluorophenyl)amino]-6-methylisoquinolin-5-yl}thieno[3,2-d]pyrimidine-7-carboxamideHuman13404
BRAFRAFTKL6xloA3-(2-cyanopropan-2-yl)-n-[2-fluoro-4-methyl-5-(7-methyl-8-oxo-7,8-dihydropyrido[2,3-d]pyridazin-3-yl)phenyl]benzamideHuman13618
BRAFRAFTKL7k0vAAn-(3,3-dimethylbutyl)-n'-{2-fluoro-5-[(5-fluoro-3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]-4-methylphenyl}ureaHuman13617
BRAFRAFTKL7k0vABn-(3,3-dimethylbutyl)-n'-{2-fluoro-5-[(5-fluoro-3-methyl-4-oxo-3,4-dihydroquinazolin-6-yl)amino]-4-methylphenyl}ureaHuman13616
BRAFRAFTKL7m0tAphosphoaminophosphonic acid-adenylate esterHuman13525
BRAFRAFTKL7m0uAphosphoaminophosphonic acid-adenylate esterHuman13527
BRAFRAFTKL7m0vAAphosphoaminophosphonic acid-adenylate esterHuman13526
BRAFRAFTKL7m0vABphosphoaminophosphonic acid-adenylate esterHuman13522
BRAFRAFTKL7m0wAphosphoaminophosphonic acid-adenylate esterHuman13528
BRAFRAFTKL7m0xAAphosphoaminophosphonic acid-adenylate esterHuman13524
BRAFRAFTKL7m0xABphosphoaminophosphonic acid-adenylate esterHuman13523
BRAFRAFTKL7m0yAphosphoaminophosphonic acid-adenylate esterHuman13520
BRAFRAFTKL7m0zAphosphoaminophosphonic acid-adenylate esterHuman13521
BRAFRAFTKL7mfdA-Human14077
BRAFRAFTKL7mfeA-Human14078
BRAFRAFTKL7p3vA~{n}-[3-[5-(2-azanylpyrimidin-4-yl)-2-[(3~{s})-morpholin-3-yl]-1,3-thiazol-4-yl]-2-fluoranyl-phenyl]-2,5-bis(fluoranyl)benzenesulfonamideHuman13961
BRAFRAFTKL7shvAA2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman14482
BRAFRAFTKL7shvAB2-{4-[(1e)-1-(hydroxyimino)-2,3-dihydro-1h-inden-5-yl]-3-(pyridin-4-yl)-1h-pyrazol-1-yl}ethanolHuman14481
BRAFRAFTKL8c7xAA~{n}-[3-[(5-chloranyl-1~{h}-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-bis(fluoranyl)phenyl]-3-(2-cyanopropan-2-yl)benzamideHuman14630
BRAFRAFTKL8c7xAB~{n}-[3-[(5-chloranyl-1~{h}-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-bis(fluoranyl)phenyl]-3-(2-cyanopropan-2-yl)benzamideHuman14627
BRAFRAFTKL8c7yAA~{n}-[3-[(5-chloranyl-1~{h}-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-bis(fluoranyl)phenyl]-3-(2-cyanopropan-2-yl)benzamideHuman14629
BRAFRAFTKL8c7yAB~{n}-[3-[(5-chloranyl-1~{h}-pyrrolo[2,3-b]pyridin-3-yl)carbonyl]-2,4-bis(fluoranyl)phenyl]-3-(2-cyanopropan-2-yl)benzamideHuman14628
BRAFRAFTKL8dgsAAphosphothiophosphoric acid-adenylate esterHuman14831
BRAFRAFTKL8dgsABphosphothiophosphoric acid-adenylate esterHuman14829
BRAFRAFTKL8dgtAAphosphothiophosphoric acid-adenylate esterHuman14832
BRAFRAFTKL8dgtABphosphothiophosphoric acid-adenylate esterHuman14830
BRAFRAFTKL8f7oAA6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamideHuman14704
BRAFRAFTKL8f7oAB6-amino-5-chloro-n-[(1r)-1-(5-{[5-chloro-4-(trifluoromethyl)pyridin-2-yl]carbamoyl}-1,3-thiazol-2-yl)ethyl]pyrimidine-4-carboxamideHuman14703
BRAFRAFTKL8f7pAAn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman14705
BRAFRAFTKL8f7pABn-{3-[2-(2-hydroxyethoxy)-6-(morpholin-4-yl)pyridin-4-yl]-4-methylphenyl}-2-(trifluoromethyl)pyridine-4-carboxamideHuman14702
BRAFRAFTKL8qqgAA(3~{s})-~{n}-[4-methyl-3-[2-morpholin-4-yl-6-[[(2~{r})-1-oxidanylpropan-2-yl]amino]pyridin-4-yl]phenyl]-3-[2,2,2-tris(fluoranyl)ethyl]pyrrolidine-1-carboxamideHuman15178
BRAFRAFTKL8qqgAB(3~{s})-~{n}-[4-methyl-3-[2-morpholin-4-yl-6-[[(2~{r})-1-oxidanylpropan-2-yl]amino]pyridin-4-yl]phenyl]-3-[2,2,2-tris(fluoranyl)ethyl]pyrrolidine-1-carboxamideHuman15179
Brsk2 (BRSK2)CAMKLCAMK4ynzA-Mouse6293
Brsk2 (BRSK2)CAMKLCAMK4ynzB-Mouse6291
Brsk2 (BRSK2)CAMKLCAMK4yomB-Mouse6292
Btk (BTK)TecTK4xi2A-Mouse5815
Btk (BTK)TecTK6mnyAA5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamideMouse11307
Btk (BTK)TecTK6mnyAB5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamideMouse11308
Btk (BTK)TecTK6mnyBA-Mouse11306
Btk (BTK)TecTK6mnyBB-Mouse11309
Btk (BTK)TecTK8fd9AAacalabrutinibMouse14836
Btk (BTK)TecTK8fd9ABacalabrutinibMouse14835
Btk (BTK)TecTK8ff0A6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-oneMouse14834
Btk (BTK)TecTK8gmbA2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-oneMouse14999
Btk (BTK)TecTK8s93AA2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-oneMouse14997
Btk (BTK)TecTK8s93AB2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-oneMouse14996
Btk (BTK)TecTK8s9fAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideMouse14998
BTKTecTK1k2pA-Human2918
BTKTecTK1k2pB-Human2919
BTKTecTK3genAA4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentaneHuman2928
BTKTecTK3genAB4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentaneHuman2900
BTKTecTK3k54AAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman2932
BTKTecTK3k54ABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman2906
BTKTecTK3ocsA4-tert-butyl-n-[2-methyl-3-(4-methyl-6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-5-oxo-4,5-dihydropyrazin-2-yl)phenyl]benzamideHuman2907
BTKTecTK3octAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman2899
BTKTecTK3octABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman2908
BTKTecTK3p08A-Human2905
BTKTecTK3p08B-Human2894
BTKTecTK3pixA7-(4-methylpiperazin-1-yl)-4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-(propan-2-yl)phthalazin-1(2h)-oneHuman2927
BTKTecTK3piyA6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-oneHuman2909
BTKTecTK3pizA[5-amino-1-(2-methylphenyl)-1h-pyrazol-4-yl]{3-[1-(methylsulfonyl)piperidin-4-yl]phenyl}methanoneHuman2922
BTKTecTK3pj1A3-(2,6-dichlorophenyl)-7-({4-[2-(diethylamino)ethoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman2904
BTKTecTK3pj2A2-({4-[2-(diethylamino)ethoxy]phenyl}amino)-6-(4-fluorophenoxy)-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman2911
BTKTecTK3pj3A2-methyl-n-(2-phenyl-3h-imidazo[4,5-b]pyridin-6-yl)-5-{[(2e)-3-phenylprop-2-enoyl]amino}benzamideHuman2910
BTKTecTK4nwmAA4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamideHuman2930
BTKTecTK4nwmAB4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamideHuman2917
BTKTecTK4nwmBA4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamideHuman2898
BTKTecTK4nwmBB4-tert-butyl-n-[2-methyl-3-(6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-7h-purin-2-yl)phenyl]benzamideHuman2903
BTKTecTK4ot5A4-tert-butyl-n-{3-[8-({4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}amino)imidazo[1,2-a]pyrazin-6-yl]phenyl}benzamideHuman2913
BTKTecTK4ot6A4-(methylsulfonyl)-n-[3-(8-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}imidazo[1,2-a]pyrazin-6-yl)phenyl]benzamideHuman2931
BTKTecTK4otfAAn-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman2901
BTKTecTK4otfABn-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman2921
BTKTecTK4otqA1-{5-[3-(7-tert-butyl-4-oxoquinazolin-3(4h)-yl)-2-methylphenyl]-1-methyl-2-oxo-1,2-dihydropyridin-3-yl}-3-methylureaHuman2895
BTKTecTK4otrA6-cyclopropyl-2-[3-(5-{[5-(4-ethylpiperazin-1-yl)pyridin-2-yl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-(hydroxymethyl)phenyl]-8-fluoroisoquinolin-1(2h)-oneHuman2896
BTKTecTK4rfyAA6-(dimethylamino)-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]-3,4-dihydroisoquinolin-1(2h)-oneHuman2935
BTKTecTK4rfyAB6-(dimethylamino)-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]-3,4-dihydroisoquinolin-1(2h)-oneHuman2933
BTKTecTK4rfzA6-(dimethylamino)-8-fluoro-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholin-4-ylcarbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]isoquinolin-1(2h)-oneHuman2925
BTKTecTK4rg0A2-{8-fluoro-2-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]-1-oxo-1,2,3,4-tetrahydroisoquinolin-6-yl}-2-methylpropanenitrileHuman2929
BTKTecTK4rx5AAn-(6-fluoro-2-methyl-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl)-1-benzothiophene-2-carboxamideHuman6259
BTKTecTK4rx5ABn-(6-fluoro-2-methyl-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl)-1-benzothiophene-2-carboxamideHuman6258
BTKTecTK4yhfAA(2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrileHuman2916
BTKTecTK4yhfAB(2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrileHuman2902
BTKTecTK4yhfBA(2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrileHuman2897
BTKTecTK4yhfBB(2s)-2-({(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}carbonyl)-4,4-dimethylpentanenitrileHuman2912
BTKTecTK4z3vAA4-amino-8-(5-methyl-1h-indazol-6-yl)cinnoline-3-carboxamideHuman2934
BTKTecTK4z3vAB4-amino-8-(5-methyl-1h-indazol-6-yl)cinnoline-3-carboxamideHuman2914
BTKTecTK4zlyAA4-aminocinnoline-3-carboxamideHuman2926
BTKTecTK4zlyAB4-aminocinnoline-3-carboxamideHuman2920
BTKTecTK4zlyAC4-aminocinnoline-3-carboxamideHuman2915
BTKTecTK4zlzAA4-amino-8-(4-methylpyridin-3-yl)cinnoline-3-carboxamideHuman2923
BTKTecTK4zlzAB4-amino-8-(4-methylpyridin-3-yl)cinnoline-3-carboxamideHuman2924
BTKTecTK5bpyA6-{(3r)-3-[(4-tert-butylbenzoyl)amino]piperidin-1-yl}-2-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}pyridine-3-carboxamideHuman6095
BTKTecTK5bpyB6-{(3r)-3-[(4-tert-butylbenzoyl)amino]piperidin-1-yl}-2-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}pyridine-3-carboxamideHuman6094
BTKTecTK5bq0AA4-(2-chlorophenyl)-7-[(4-methylpiperazin-1-yl)carbonyl]-9h-carbazole-1-carboxamideHuman6871
BTKTecTK5bq0AB4-(2-chlorophenyl)-7-[(4-methylpiperazin-1-yl)carbonyl]-9h-carbazole-1-carboxamideHuman6872
BTKTecTK5fbnCA4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6381
BTKTecTK5fbnCB4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6382
BTKTecTK5fbnDA4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6384
BTKTecTK5fbnDB4-[8-azanyl-3-[(3~{r})-1-(3-methyloxetan-3-yl)carbonylpiperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6383
BTKTecTK5fboAA4-[8-azanyl-3-[(3~{r},6~{s})-1-cyclopropylcarbonyl-6-methyl-piperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoranyl-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6455
BTKTecTK5fboAB4-[8-azanyl-3-[(3~{r},6~{s})-1-cyclopropylcarbonyl-6-methyl-piperidin-3-yl]imidazo[1,5-a]pyrazin-1-yl]-3-fluoranyl-~{n}-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman6456
BTKTecTK5j87AAn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8002
BTKTecTK5j87ABn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8003
BTKTecTK5j87BAn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8005
BTKTecTK5j87BBn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8007
BTKTecTK5j87CAn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8004
BTKTecTK5j87CBn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8006
BTKTecTK5j87DAn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8008
BTKTecTK5j87DBn-[3-(5-{[3-(acryloylamino)-4-(morpholine-4-carbonyl)phenyl]amino}-1-methyl-6-oxo-1,6-dihydropyridin-3-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman8001
BTKTecTK5jrsA4-[2-fluoro-3-(4-oxoquinazolin-3(4h)-yl)phenyl]-7-(2-hydroxypropan-2-yl)-9h-carbazole-1-carboxamideHuman7032
BTKTecTK5jrsB4-[2-fluoro-3-(4-oxoquinazolin-3(4h)-yl)phenyl]-7-(2-hydroxypropan-2-yl)-9h-carbazole-1-carboxamideHuman7033
BTKTecTK5kupAA6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-6-oxidanylidene-5-(pyrimidin-4-ylamino)pyridin-3-yl]pyridin-2-yl]phthalazin-1-oneHuman7051
BTKTecTK5kupAB6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-6-oxidanylidene-5-(pyrimidin-4-ylamino)pyridin-3-yl]pyridin-2-yl]phthalazin-1-oneHuman7052
BTKTecTK5p9fAAn-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman7632
BTKTecTK5p9fABn-{3-[6-({4-[(2r)-1,4-dimethyl-3-oxopiperazin-2-yl]phenyl}amino)-4-methyl-5-oxo-4,5-dihydropyrazin-2-yl]-2-methylphenyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman7629
BTKTecTK5p9gAA6-cyclopropyl-8-fluoranyl-2-[2-(hydroxymethyl)-3-[1-methyl-5-[[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridin-3-yl]phenyl]isoquinolin-1-oneHuman7635
BTKTecTK5p9gAB6-cyclopropyl-8-fluoranyl-2-[2-(hydroxymethyl)-3-[1-methyl-5-[[5-(4-methylpiperazin-1-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridin-3-yl]phenyl]isoquinolin-1-oneHuman7644
BTKTecTK5p9hAA6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-5-[[5-(1-methylpiperidin-4-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridazin-3-yl]pyridin-2-yl]phthalazin-1-oneHuman7631
BTKTecTK5p9hAB6-~{tert}-butyl-8-fluoranyl-2-[3-(hydroxymethyl)-4-[1-methyl-5-[[5-(1-methylpiperidin-4-yl)pyridin-2-yl]amino]-6-oxidanylidene-pyridazin-3-yl]pyridin-2-yl]phthalazin-1-oneHuman7643
BTKTecTK5p9iAA1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman7627
BTKTecTK5p9iAB1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman7642
BTKTecTK5p9iAC1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman7638
BTKTecTK5p9jAA1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman7637
BTKTecTK5p9jAB1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman7628
BTKTecTK5p9jAC1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman7640
BTKTecTK5p9kAA4-[4-[[5-fluoranyl-4-[[3-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]phenoxy]-~{n}-methyl-pyridine-2-carboxamideHuman7633
BTKTecTK5p9kAB4-[4-[[5-fluoranyl-4-[[3-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]phenoxy]-~{n}-methyl-pyridine-2-carboxamideHuman7636
BTKTecTK5p9kAC4-[4-[[5-fluoranyl-4-[[3-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]phenoxy]-~{n}-methyl-pyridine-2-carboxamideHuman7626
BTKTecTK5p9lAA~{n}-[3-[[5-fluoranyl-2-[[4-(2-methoxyethoxy)phenyl]amino]pyrimidin-4-yl]amino]phenyl]propanamideHuman7625
BTKTecTK5p9lAB~{n}-[3-[[5-fluoranyl-2-[[4-(2-methoxyethoxy)phenyl]amino]pyrimidin-4-yl]amino]phenyl]propanamideHuman7630
BTKTecTK5p9mAA6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-oneHuman7634
BTKTecTK5p9mAB6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-oneHuman7639
BTKTecTK5p9mAC6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-oneHuman7641
BTKTecTK5t18AA6-fluoro-5-(r)-(3-(s)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4h)-yl)-2-methylphenyl)-2-(s)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamideHuman7508
BTKTecTK5t18AB6-fluoro-5-(r)-(3-(s)-(8-fluoro-1-methyl-2,4-dioxo-1,2-dihydroquinazolin-3(4h)-yl)-2-methylphenyl)-2-(s)-(2-hydroxypropan-2-yl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamideHuman7507
BTKTecTK5u9dAA(r)-n-methyl-2-(3-((quinoxalin-6-ylamino)methyl)furan-2-carbonyl)-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamideHuman7393
BTKTecTK5u9dAB(r)-n-methyl-2-(3-((quinoxalin-6-ylamino)methyl)furan-2-carbonyl)-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamideHuman7392
BTKTecTK5vfiAA2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-oneHuman9602
BTKTecTK5vfiAB2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-oneHuman9601
BTKTecTK5vgoAA2-(2-methoxyethoxy)ethanolHuman8218
BTKTecTK5vgoAB2-(2-methoxyethoxy)ethanolHuman8219
BTKTecTK5xyzAAn-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamideHuman9929
BTKTecTK5xyzABn-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamideHuman9932
BTKTecTK5xyzBAn-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamideHuman9931
BTKTecTK5xyzBBn-[3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-1h-1,2,4-triazol-3-yl)phenyl]propanamideHuman9930
BTKTecTK5zz4An-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10479
BTKTecTK5zz4Bn-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10468
BTKTecTK5zz4Cn-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10464
BTKTecTK5zz4Dn-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10478
BTKTecTK5zz4En-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10470
BTKTecTK5zz4Fn-[3-(4-amino-6-{[4-(morpholine-4-carbonyl)phenyl]amino}-1,3,5-triazin-2-yl)-2-methylphenyl]-4-tert-butylbenzamideHuman10469
BTKTecTK6auaAAn-{3-[(2r)-6-{[3-amino-4-(morpholine-4-carbonyl)phenyl]amino}-5-oxo-2,5-dihydropyrazin-2-yl]-2-methylphenyl}-4-(piperidin-1-yl)benzamideHuman10472
BTKTecTK6auaABn-{3-[(2r)-6-{[3-amino-4-(morpholine-4-carbonyl)phenyl]amino}-5-oxo-2,5-dihydropyrazin-2-yl]-2-methylphenyl}-4-(piperidin-1-yl)benzamideHuman10473
BTKTecTK6aubAA4-tert-butyl-n-[2-methyl-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]benzamideHuman10466
BTKTecTK6aubAB4-tert-butyl-n-[2-methyl-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridin-3-yl)phenyl]benzamideHuman10475
BTKTecTK6bikAA4-tert-butyl-n-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridazin-3-yl)phenyl]benzamideHuman10680
BTKTecTK6bikAB4-tert-butyl-n-[2-(hydroxymethyl)-3-(1-methyl-5-{[5-(morpholine-4-carbonyl)pyridin-2-yl]amino}-6-oxo-1,6-dihydropyridazin-3-yl)phenyl]benzamideHuman10678
BTKTecTK6bkeAAn-[2-(2-hydroxyethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamideHuman10681
BTKTecTK6bkeABn-[2-(2-hydroxyethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamideHuman10683
BTKTecTK6bkhAAn-[2-(hydroxymethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamideHuman10682
BTKTecTK6bkhABn-[2-(hydroxymethyl)-3-{5-[(5-methyl-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}phenyl]-1-benzothiophene-2-carboxamideHuman10677
BTKTecTK6bkwAAn-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-1-methyl-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman10686
BTKTecTK6bkwABn-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-1-methyl-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman10679
BTKTecTK6blnAAn-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman10685
BTKTecTK6blnABn-(3-{5-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-oxo-1,6-dihydropyridazin-3-yl}-2,6-difluorophenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamideHuman10684
BTKTecTK6di0AA6-(cyclohexylamino)pyridine-3-carboxamideHuman10629
BTKTecTK6di0AB6-(cyclohexylamino)pyridine-3-carboxamideHuman10626
BTKTecTK6di0AC6-(cyclohexylamino)pyridine-3-carboxamideHuman10628
BTKTecTK6di1AA4-amino-2-[(3s)-3-(propanoylamino)pyrrolidin-1-yl]pyrimidine-5-carboxamideHuman10630
BTKTecTK6di1AB4-amino-2-[(3s)-3-(propanoylamino)pyrrolidin-1-yl]pyrimidine-5-carboxamideHuman10627
BTKTecTK6di3A6-[(3s)-3-(acryloylamino)pyrrolidin-1-yl]-2-(4-phenoxyphenoxy)pyridine-3-carboxamideHuman10474
BTKTecTK6di5AA2-(4-phenoxyphenoxy)-6-[(1s,4s)-5-propanoyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyridine-3-carboxamideHuman10471
BTKTecTK6di5AB2-(4-phenoxyphenoxy)-6-[(1s,4s)-5-propanoyl-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyridine-3-carboxamideHuman10481
BTKTecTK6di9AA6-[(3s)-3-(acryloylamino)pyrrolidin-1-yl]-2-{[4-(tert-butylcarbamoyl)phenyl]amino}pyridine-3-carboxamideHuman10465
BTKTecTK6di9AB6-[(3s)-3-(acryloylamino)pyrrolidin-1-yl]-2-{[4-(tert-butylcarbamoyl)phenyl]amino}pyridine-3-carboxamideHuman10476
BTKTecTK6e4fAA1,5-anhydro-2-{[5-(2-chloro-4-phenoxybenzene-1-carbonyl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-2,3,4-trideoxy-d-erythro-hexitolHuman10477
BTKTecTK6e4fAB1,5-anhydro-2-{[5-(2-chloro-4-phenoxybenzene-1-carbonyl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}-2,3,4-trideoxy-d-erythro-hexitolHuman10480
BTKTecTK6ep9An-[2-methyl-3-[4-methyl-6-[4-(4-methylpiperazine-1-carbonyl)anilino]-5-oxo-pyrazin-2-yl]phenyl]-4-(1-piperidyl)benzamideHuman10467
BTKTecTK6hrpA6-~{tert}-butyl-8-fluoranyl-2-[2-(hydroxymethyl)-3-[1-methyl-5-[(5-morpholin-4-ylcarbonylpyridin-2-yl)amino]-6-oxidanylidene-pyridazin-3-yl]phenyl]phthalazin-1-oneHuman10971
BTKTecTK6hrtA(9~{s})-12-(6-~{tert}-butyl-8-fluoranyl-1-oxidanylidene-phthalazin-2-yl)-6-methyl-4-[(5-morpholin-4-ylcarbonylpyridin-2-yl)amino]-9-oxidanyl-6-azatricyclo[9.4.0.0^{2,7}]pentadeca-1(15),2(7),3,11,13-pentaen-5-oneHuman10972
BTKTecTK6j6mAA(7s)-2-(4-phenoxyphenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11767
BTKTecTK6j6mAB(7s)-2-(4-phenoxyphenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11766
BTKTecTK6n9pAAn-(3-{[2-amino-3-(4-phenoxyphenyl)pyridin-4-yl]oxy}phenyl)propanamideHuman10886
BTKTecTK6n9pABn-(3-{[2-amino-3-(4-phenoxyphenyl)pyridin-4-yl]oxy}phenyl)propanamideHuman10887
BTKTecTK6n9pACn-(3-{[2-amino-3-(4-phenoxyphenyl)pyridin-4-yl]oxy}phenyl)propanamideHuman10888
BTKTecTK6nfhAA8-(2,3-dihydro-1h-inden-5-yl)-2-({4-[(2s)-3-(dimethylamino)-2-hydroxypropoxy]phenyl}amino)-5,8-dihydropteridine-6,7-dioneHuman10964
BTKTecTK6nfhAB8-(2,3-dihydro-1h-inden-5-yl)-2-({4-[(2s)-3-(dimethylamino)-2-hydroxypropoxy]phenyl}amino)-5,8-dihydropteridine-6,7-dioneHuman10965
BTKTecTK6nfiAAn-(3-{[(2,6-dimethylphenyl)methyl]amino}-7-methoxyindeno[1,2-c]pyrazol-6-yl)methanesulfonamideHuman10962
BTKTecTK6nfiABn-(3-{[(2,6-dimethylphenyl)methyl]amino}-7-methoxyindeno[1,2-c]pyrazol-6-yl)methanesulfonamideHuman10963
BTKTecTK6nzmAAn-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}ureaHuman11144
BTKTecTK6nzmABn-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}ureaHuman11143
BTKTecTK6nzmDAn-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}ureaHuman11141
BTKTecTK6nzmDBn-[2-fluoro-6-(pyrrolidin-1-yl)phenyl]-n'-{3-[(2r)-1-(2-hydroxyethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-2-yl]phenyl}ureaHuman11142
BTKTecTK6o8iAA4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamideHuman11002
BTKTecTK6o8iAB4-[(3s)-3-{[(2e)-but-2-enoyl]amino}piperidin-1-yl]-5-fluoro-2,3-dimethyl-1h-indole-7-carboxamideHuman11001
BTKTecTK6omuAA1-[4-({[6-amino-5-(4-phenoxyphenyl)pyrimidin-4-yl]amino}methyl)piperidin-1-yl]prop-2-en-1-oneHuman11529
BTKTecTK6omuAB1-[4-({[6-amino-5-(4-phenoxyphenyl)pyrimidin-4-yl]amino}methyl)piperidin-1-yl]prop-2-en-1-oneHuman11530
BTKTecTK6omuAC-Human11528
BTKTecTK6s90A4-~{tert}-butyl-~{n}-[2-methyl-3-[6-[4-(4-methylpiperazin-1-yl)carbonylphenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]benzamideHuman11636
BTKTecTK6s90B4-~{tert}-butyl-~{n}-[2-methyl-3-[6-[4-(4-methylpiperazin-1-yl)carbonylphenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]phenyl]benzamideHuman11635
BTKTecTK6tfpA~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12024
BTKTecTK6tfpB~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12020
BTKTecTK6tfpC~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12023
BTKTecTK6tfpD~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12021
BTKTecTK6tfpE~{n}-[3-[6-azanyl-5-[2-[methyl(propanoyl)amino]ethoxy]pyrimidin-4-yl]-5-fluoranyl-2-methyl-phenyl]-4-cyclopropyl-2-fluoranyl-benzamideHuman12022
BTKTecTK6vxqAAn-{[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]methyl}benzamideHuman13100
BTKTecTK6vxqABn-{[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]methyl}benzamideHuman13101
BTKTecTK6w06AA4-~{tert}-butyl-~{n}-[[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]methyl]benzamideHuman13099
BTKTecTK6w06AB4-~{tert}-butyl-~{n}-[[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]methyl]benzamideHuman13098
BTKTecTK6w07AA~{n}-[[2-methyl-4-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]phenyl]methyl]-3-propan-2-yloxy-azetidine-1-carboxamideHuman13096
BTKTecTK6w07AB~{n}-[[2-methyl-4-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]phenyl]methyl]-3-propan-2-yloxy-azetidine-1-carboxamideHuman13102
BTKTecTK6w07AC~{n}-[[2-methyl-4-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]phenyl]methyl]-3-propan-2-yloxy-azetidine-1-carboxamideHuman13097
BTKTecTK6w7oA[5-({[(3s)-2-(n-methyl-l-alanyl-3-methyl-l-valyl)-3-{[(1r)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl}-1,2,3,4-tetrahydroisoquinolin-7-yl]oxy}methyl)pyrazin-2-yl]methyl (3r)-3-{5-amino-4-carbamoyl-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazol-1-yl}piperidine-1-carboxylateHuman13195
BTKTecTK6w7oB[5-({[(3s)-2-(n-methyl-l-alanyl-3-methyl-l-valyl)-3-{[(1r)-1,2,3,4-tetrahydronaphthalen-1-yl]carbamoyl}-1,2,3,4-tetrahydroisoquinolin-7-yl]oxy}methyl)pyrazin-2-yl]methyl (3r)-3-{5-amino-4-carbamoyl-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazol-1-yl}piperidine-1-carboxylateHuman13196
BTKTecTK6w8iA-Human12990
BTKTecTK6w8iB-Human12991
BTKTecTK6x3nAA4-{8-amino-3-[(6r,8as)-3-oxohexahydro-3h-[1,3]oxazolo[3,4-a]pyridin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12514
BTKTecTK6x3nAB4-{8-amino-3-[(6r,8as)-3-oxohexahydro-3h-[1,3]oxazolo[3,4-a]pyridin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12510
BTKTecTK6x3oAA4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12513
BTKTecTK6x3oAB4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12512
BTKTecTK6x3oBA4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12508
BTKTecTK6x3oBB4-{8-amino-3-[(6r,8as)-3-oxo-3,5,6,7,8,8a-hexahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-methoxy-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12511
BTKTecTK6x3pAA4-{8-amino-3-[(6r,8as)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(cyclopropyloxy)-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12516
BTKTecTK6x3pAB4-{8-amino-3-[(6r,8as)-3-oxooctahydroindolizin-6-yl]imidazo[1,5-a]pyrazin-1-yl}-3-(cyclopropyloxy)-n-[4-(trifluoromethyl)pyridin-2-yl]benzamideHuman12517
BTKTecTK6xe4AA(1s,2s)-n-[2'-(6-tert-butyl-8-fluoro-1-oxophthalazin-2(1h)-yl)-3'-(hydroxymethyl)-1-methyl-6-oxo[1,6-dihydro[3,4'-bipyridine]]-5-yl]-2-fluorocyclopropane-1-carboxamideHuman12515
BTKTecTK6xe4AB(1s,2s)-n-[2'-(6-tert-butyl-8-fluoro-1-oxophthalazin-2(1h)-yl)-3'-(hydroxymethyl)-1-methyl-6-oxo[1,6-dihydro[3,4'-bipyridine]]-5-yl]-2-fluorocyclopropane-1-carboxamideHuman12509
BTKTecTK7kxlAA3-tert-butyl-n-({2-fluoro-4-[2-(1-methyl-1h-pyrazol-4-yl)-1h-imidazo[4,5-b]pyridin-7-yl]phenyl}methyl)-1,2,4-oxadiazole-5-carboxamideHuman13563
BTKTecTK7kxlAB3-tert-butyl-n-({2-fluoro-4-[2-(1-methyl-1h-pyrazol-4-yl)-1h-imidazo[4,5-b]pyridin-7-yl]phenyl}methyl)-1,2,4-oxadiazole-5-carboxamideHuman13561
BTKTecTK7kxlAC3-tert-butyl-n-({2-fluoro-4-[2-(1-methyl-1h-pyrazol-4-yl)-1h-imidazo[4,5-b]pyridin-7-yl]phenyl}methyl)-1,2,4-oxadiazole-5-carboxamideHuman13576
BTKTecTK7kxmAA4-tert-butyl-n-(2-methyl-3-{2-[4-(morpholine-4-carbonyl)phenyl]-1h-imidazo[4,5-b]pyridin-7-yl}phenyl)benzamideHuman13569
BTKTecTK7kxmAB4-tert-butyl-n-(2-methyl-3-{2-[4-(morpholine-4-carbonyl)phenyl]-1h-imidazo[4,5-b]pyridin-7-yl}phenyl)benzamideHuman13564
BTKTecTK7kxmAC4-tert-butyl-n-(2-methyl-3-{2-[4-(morpholine-4-carbonyl)phenyl]-1h-imidazo[4,5-b]pyridin-7-yl}phenyl)benzamideHuman13567
BTKTecTK7kxnAA3-tert-butyl-n-[(1s)-6-{2-[5-methyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamideHuman13574
BTKTecTK7kxnAB3-tert-butyl-n-[(1s)-6-{2-[5-methyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamideHuman13571
BTKTecTK7kxnAC3-tert-butyl-n-[(1s)-6-{2-[5-methyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamideHuman13570
BTKTecTK7kxoAA3-tert-butyl-n-[(1r)-6-{2-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamideHuman13573
BTKTecTK7kxoAB3-tert-butyl-n-[(1r)-6-{2-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamideHuman13568
BTKTecTK7kxoAC3-tert-butyl-n-[(1r)-6-{2-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamideHuman13572
BTKTecTK7kxpAA3-tert-butyl-n-[(1s)-6-{2-[3-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamideHuman13575
BTKTecTK7kxpAB3-tert-butyl-n-[(1s)-6-{2-[3-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridin-7-yl}-1,2,3,4-tetrahydronaphthalen-1-yl]-1,2,4-oxadiazole-5-carboxamideHuman13566
BTKTecTK7kxqAA3-tert-butyl-n-[(5r)-2-{2-[3,5-dimethyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-6,7,8,9-tetrahydro-5h-benzo[7]annulen-5-yl]-1,2,4-oxadiazole-5-carboxamideHuman13562
BTKTecTK7kxqAB3-tert-butyl-n-[(5r)-2-{2-[3,5-dimethyl-1-(propan-2-yl)-1h-pyrazol-4-yl]-3h-imidazo[4,5-b]pyridin-7-yl}-6,7,8,9-tetrahydro-5h-benzo[7]annulen-5-yl]-1,2,4-oxadiazole-5-carboxamideHuman13565
BTKTecTK7l5oAA(2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrileHuman14272
BTKTecTK7l5oAB(2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrileHuman14271
BTKTecTK7l5oAC(2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrileHuman14268
BTKTecTK7l5pAA(2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrileHuman14269
BTKTecTK7l5pAB(2e)-2-{(3r)-3-[4-amino-3-(2-fluoro-4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidine-1-carbonyl}-4-methyl-4-[4-(oxetan-3-yl)piperazin-1-yl]pent-2-enenitrileHuman14270
BTKTecTK7ltyAA~{n}-[(5~{r})-2-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-6,7,8,9-tetrahydro-5~{h}-benzo[7]annulen-5-yl]-3-propan-2-yloxy-azetidine-1-carboxamideHuman14065
BTKTecTK7ltyAB~{n}-[(5~{r})-2-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-6,7,8,9-tetrahydro-5~{h}-benzo[7]annulen-5-yl]-3-propan-2-yloxy-azetidine-1-carboxamideHuman14069
BTKTecTK7ltyAC~{n}-[(5~{r})-2-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-6,7,8,9-tetrahydro-5~{h}-benzo[7]annulen-5-yl]-3-propan-2-yloxy-azetidine-1-carboxamideHuman14068
BTKTecTK7ltyAD~{n}-[(5~{r})-2-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-6,7,8,9-tetrahydro-5~{h}-benzo[7]annulen-5-yl]-3-propan-2-yloxy-azetidine-1-carboxamideHuman14064
BTKTecTK7ltzAA1-~{tert}-butyl-~{n}-[(5~{r})-8-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-2-(oxetan-3-yl)-1,3,4,5-tetrahydro-2-benzazepin-5-yl]-1,2,3-triazole-4-carboxamideHuman14067
BTKTecTK7ltzAB1-~{tert}-butyl-~{n}-[(5~{r})-8-[2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]-2-(oxetan-3-yl)-1,3,4,5-tetrahydro-2-benzazepin-5-yl]-1,2,3-triazole-4-carboxamideHuman14066
BTKTecTK7n4qAA(2r)-2-(3-chloro-5-fluoroanilino)-2-cyclopropyl-n-[(3r)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]acetamideHuman14227
BTKTecTK7n4qAB(2r)-2-(3-chloro-5-fluoroanilino)-2-cyclopropyl-n-[(3r)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]acetamideHuman14224
BTKTecTK7n4rAAn-{2-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]ethyl}-n~2~-phenylglycinamideHuman14226
BTKTecTK7n4rABn-{2-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]ethyl}-n~2~-phenylglycinamideHuman14228
BTKTecTK7n4rACn-{2-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]ethyl}-n~2~-phenylglycinamideHuman14225
BTKTecTK7n4sA(3r,3'r)-3-anilino-1'-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)[1,3'-bipiperidin]-2-oneHuman14229
BTKTecTK7n5oAA5-(1h-benzimidazol-2-yl)-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman13896
BTKTecTK7n5oAB5-(1h-benzimidazol-2-yl)-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman13891
BTKTecTK7n5rAA5-phenyl-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman13895
BTKTecTK7n5rAB5-phenyl-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman13890
BTKTecTK7n5xAA5-(1-ethoxyisoquinolin-3-yl)-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman13893
BTKTecTK7n5xAB5-(1-ethoxyisoquinolin-3-yl)-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman13889
BTKTecTK7n5yAA5-(1-{[(3s)-1-propanoylpyrrolidin-3-yl]oxy}isoquinolin-3-yl)-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman13894
BTKTecTK7n5yAB5-(1-{[(3s)-1-propanoylpyrrolidin-3-yl]oxy}isoquinolin-3-yl)-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman13892
BTKTecTK7r60AA2-(4-phenoxyphenoxy)-5-[(3r)-1-(prop-2-enoyl)piperidin-3-yl]pyridine-3-carboxamideHuman13937
BTKTecTK7r60AB2-(4-phenoxyphenoxy)-5-[(3r)-1-(prop-2-enoyl)piperidin-3-yl]pyridine-3-carboxamideHuman13939
BTKTecTK7r61AA5-{(3s)-1-[(z)-iminomethyl]piperidin-3-yl}-2-(4-phenoxyphenoxy)pyridine-3-carboxamideHuman13938
BTKTecTK7r61AB5-{(3s)-1-[(z)-iminomethyl]piperidin-3-yl}-2-(4-phenoxyphenoxy)pyridine-3-carboxamideHuman13936
BTKTecTK7r61AC5-{(3s)-1-[(z)-iminomethyl]piperidin-3-yl}-2-(4-phenoxyphenoxy)pyridine-3-carboxamideHuman13940
BTKTecTK7yc9AA(7~{s})-2-(4-bromanyl-3,5-dimethoxy-phenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamideHuman14746
BTKTecTK7yc9AB(7~{s})-2-(4-bromanyl-3,5-dimethoxy-phenyl)-7-(1-propanoylpiperidin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamideHuman14745
BTKTecTK8e2mAA(5p)-5-[4-methyl-6-(2-methylpropyl)pyridin-3-yl]-4-oxo-n-[(1r,2s)-2-propanamidocyclopentyl]-4,5-dihydro-3h-1-thia-3,5,8-triazaacenaphthylene-2-carboxamideHuman14552
BTKTecTK8e2mAB(5p)-5-[4-methyl-6-(2-methylpropyl)pyridin-3-yl]-4-oxo-n-[(1r,2s)-2-propanamidocyclopentyl]-4,5-dihydro-3h-1-thia-3,5,8-triazaacenaphthylene-2-carboxamideHuman14553
BTKTecTK8e2mAC(5p)-5-[4-methyl-6-(2-methylpropyl)pyridin-3-yl]-4-oxo-n-[(1r,2s)-2-propanamidocyclopentyl]-4,5-dihydro-3h-1-thia-3,5,8-triazaacenaphthylene-2-carboxamideHuman14551
BTKTecTK8ejbAA5-[(3r)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamideHuman14614
BTKTecTK8ejbAB5-[(3r)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamideHuman14615
BTKTecTK8flgAAn~2~-(3-chlorophenyl)-n-[(3r)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]glycinamideHuman14641
BTKTecTK8flgABn~2~-(3-chlorophenyl)-n-[(3r)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-3-yl]glycinamideHuman14634
BTKTecTK8flhAA2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]azepan-1-yl}ethan-1-oneHuman14637
BTKTecTK8flhAB2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]azepan-1-yl}ethan-1-oneHuman14638
BTKTecTK8flhAC2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]azepan-1-yl}ethan-1-oneHuman14639
BTKTecTK8fllAApirtobrutinibHuman14636
BTKTecTK8fllABpirtobrutinibHuman14640
BTKTecTK8flnAApirtobrutinibHuman14642
BTKTecTK8flnABpirtobrutinibHuman14635
BTKTecTK8flnACpirtobrutinibHuman14633
BTKTecTK8flvAA2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}ethan-1-oneHuman14698
BTKTecTK8flvAB2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}ethan-1-oneHuman14699
BTKTecTK8flvAC2-(3,5-dichloroanilino)-1-{(3r)-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}ethan-1-oneHuman14697
BTKTecTK8gc7AA5-(piperidin-1-yl)-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamideHuman15196
BTKTecTK8gc7AB5-(piperidin-1-yl)-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamideHuman15197
BTKTecTK8gc8AA5-(piperidin-1-yl)-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamideHuman15195
BTKTecTK8gc8AB5-(piperidin-1-yl)-3-[4-(piperidin-4-yl)anilino]pyrazine-2-carboxamideHuman15192
BTKTecTK8u2dAA(3r)-2-[n-(1h-indazole-5-carbonyl)-3-methyl-d-phenylalanyl]-n-methyl-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamideHuman15199
BTKTecTK8u2dAB(3r)-2-[n-(1h-indazole-5-carbonyl)-3-methyl-d-phenylalanyl]-n-methyl-2,3,4,9-tetrahydro-1h-pyrido[3,4-b]indole-3-carboxamideHuman15193
BTKTecTK8u2eAA(2s)-6-fluoro-5-[(3s)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-2-(4-methylpiperazine-1-carbonyl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamideHuman15198
BTKTecTK8u2eAB(2s)-6-fluoro-5-[(3s)-3-(3-methyl-2-oxoimidazolidin-1-yl)piperidin-1-yl]-2-(4-methylpiperazine-1-carbonyl)-2,3,4,9-tetrahydro-1h-carbazole-8-carboxamideHuman15194
BUB1BUBOther4qpmAadenosine-5'-diphosphateHuman1843
BUB1BUBOther4qpmBadenosine-5'-diphosphateHuman1844
BUB1BUBOther4r8qAadenosine-5'-diphosphateHuman1842
BUB1BUBOther5dmzAadenosine-5'-diphosphateHuman6287
BUB1BUBOther5dmzBadenosine-5'-diphosphateHuman6286
BUB1BUBOther6f7bAA2-[3,5-bis(fluoranyl)-4-[[3-[5-methoxy-4-[(3-methoxypyridin-4-yl)amino]pyrimidin-2-yl]indazol-1-yl]methyl]phenoxy]ethanolHuman10808
BUB1BUBOther6f7bAB2-[3,5-bis(fluoranyl)-4-[[3-[5-methoxy-4-[(3-methoxypyridin-4-yl)amino]pyrimidin-2-yl]indazol-1-yl]methyl]phenoxy]ethanolHuman10807
BUB1B (BUBR1)BUBOther6tljS-Human11992
CAMK1 (CaMK1a)CAMK1CAMK4fg7Aadenosine-5'-triphosphateHuman4848
CAMK1 (CaMK1a)CAMK1CAMK4fg8Aadenosine-5'-triphosphateHuman4850
CAMK1 (CaMK1a)CAMK1CAMK4fg8Badenosine-5'-triphosphateHuman4849
CAMK1 (CaMK1a)CAMK1CAMK4fg9Aadenosine-5'-triphosphateHuman4846
CAMK1 (CaMK1a)CAMK1CAMK4fg9Badenosine-5'-triphosphateHuman4845
CAMK1 (CaMK1a)CAMK1CAMK4fgbA-Human4847
CAMK1D (CaMK1d)CAMK1CAMK2jc6AAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4829
CAMK1D (CaMK1d)CAMK1CAMK2jc6ABn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4830
CAMK1D (CaMK1d)CAMK1CAMK2jc6CAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4832
CAMK1D (CaMK1d)CAMK1CAMK2jc6CBn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4831
CAMK1D (CaMK1d)CAMK1CAMK6qp5AA-Human12028
CAMK1D (CaMK1d)CAMK1CAMK6qp5AB-Human12029
CAMK1D (CaMK1d)CAMK1CAMK6t28AA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamideHuman13202
CAMK1D (CaMK1d)CAMK1CAMK6t28AB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamideHuman13205
CAMK1D (CaMK1d)CAMK1CAMK6t29AA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamideHuman13204
CAMK1D (CaMK1d)CAMK1CAMK6t29AB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamideHuman13203
CAMK1D (CaMK1d)CAMK1CAMK6t6fAA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11939
CAMK1D (CaMK1d)CAMK1CAMK6t6fAB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11940
CAMK1D (CaMK1d)CAMK1CAMK6t6fBA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11941
CAMK1D (CaMK1d)CAMK1CAMK6t6fBB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11942
CAMK1D (CaMK1d)CAMK1CAMK8bfmApyrazolo[5,1-a]phthalazin-6-amineHuman14516
CAMK1D (CaMK1d)CAMK1CAMK8bfsAA3~{h}-pyrrolo[2,3-c]isoquinolin-5-amineHuman14506
CAMK1D (CaMK1d)CAMK1CAMK8bfsAB3~{h}-pyrrolo[2,3-c]isoquinolin-5-amineHuman14505
CAMK1G (CaMK1g)CAMK1CAMK2jamAA5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1218
CAMK1G (CaMK1g)CAMK1CAMK2jamAB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1221
CAMK1G (CaMK1g)CAMK1CAMK2jamBA5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1220
CAMK1G (CaMK1g)CAMK1CAMK2jamBB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1219
Camk2a (CaMK2a)CAMK2CAMK7b55AA-Mouse14244
Camk2a (CaMK2a)CAMK2CAMK7b55AB-Mouse14247
Camk2a (CaMK2a)CAMK2CAMK7b56AA-Mouse14245
Camk2a (CaMK2a)CAMK2CAMK7b56AB-Mouse14249
Camk2a (CaMK2a)CAMK2CAMK7b57AA-Mouse14246
Camk2a (CaMK2a)CAMK2CAMK7b57AB-Mouse14248
CAMK2A (CaMK2a)CAMK2CAMK2vz6AA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2472
CAMK2A (CaMK2a)CAMK2CAMK2vz6AB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2471
CAMK2A (CaMK2a)CAMK2CAMK2vz6BA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2474
CAMK2A (CaMK2a)CAMK2CAMK2vz6BB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2470
CAMK2A (CaMK2a)CAMK2CAMK3soaA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman2473
CAMK2A (CaMK2a)CAMK2CAMK6vzkA4'-hydroxycinnamic acidHuman12165
CAMK2A (CaMK2a)CAMK2CAMK6w4oO-Human12485
CAMK2A (CaMK2a)CAMK2CAMK6w4pH-Human12484
CAMK2A (CaMK2a)CAMK2CAMK6x5gAA-Human13061
CAMK2A (CaMK2a)CAMK2CAMK6x5gAB-Human13068
CAMK2A (CaMK2a)CAMK2CAMK6x5qA-Human13056
CAMK2A (CaMK2a)CAMK2CAMK7kl0Amethyl 6-o-(heptylcarbamoyl)-beta-l-altropyranosideHuman13111
CAMK2A (CaMK2a)CAMK2CAMK7kl0Bmethyl 6-o-(heptylcarbamoyl)-beta-l-altropyranosideHuman13114
CAMK2A (CaMK2a)CAMK2CAMK7kl1Aadenosine-5'-triphosphateHuman13059
CAMK2A (CaMK2a)CAMK2CAMK7kl1Badenosine-5'-triphosphateHuman13062
CAMK2A (CaMK2a)CAMK2CAMK7kl2A-Human13064
CAMK2A (CaMK2a)CAMK2CAMK7uiqA-Human14175
CAMK2A (CaMK2a)CAMK2CAMK7uirAadenosine-5'-triphosphateHuman14173
CAMK2A (CaMK2a)CAMK2CAMK7uisA-Human14174
CAMK2A (CaMK2a)CAMK2CAMK7ujpAadenosine-5'-diphosphateHuman14193
CAMK2A (CaMK2a)CAMK2CAMK7ujqAmethyl 6-o-(heptylcarbamoyl)-beta-l-altropyranosideHuman14189
CAMK2A (CaMK2a)CAMK2CAMK7ujrA-Human14191
CAMK2A (CaMK2a)CAMK2CAMK7ujsAadenosine-5'-diphosphateHuman14190
CAMK2A (CaMK2a)CAMK2CAMK7ujtAadenosine-5'-triphosphateHuman14192
CAMK2B (CaMK2b)CAMK2CAMK3bhhA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1507
CAMK2B (CaMK2b)CAMK2CAMK3bhhB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1506
CAMK2B (CaMK2b)CAMK2CAMK3bhhC-Human1505
CAMK2B (CaMK2b)CAMK2CAMK3bhhD-Human1504
Camk2d (CaMK2d)CAMK2CAMK6babAAn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8694
Camk2d (CaMK2d)CAMK2CAMK6babABn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8691
Camk2d (CaMK2d)CAMK2CAMK6babBAn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8690
Camk2d (CaMK2d)CAMK2CAMK6babBBn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8693
Camk2d (CaMK2d)CAMK2CAMK6babCAn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8697
Camk2d (CaMK2d)CAMK2CAMK6babCBn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8692
Camk2d (CaMK2d)CAMK2CAMK6babDAn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8695
Camk2d (CaMK2d)CAMK2CAMK6babDBn-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideMouse8696
CAMK2D (CaMK2d)CAMK2CAMK2vn9A[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2140
CAMK2D (CaMK2d)CAMK2CAMK2vn9B[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2139
CAMK2D (CaMK2d)CAMK2CAMK2welAA(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2138
CAMK2D (CaMK2d)CAMK2CAMK2welAB(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2137
CAMK2D (CaMK2d)CAMK2CAMK2welAC(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2136
CAMK2D (CaMK2d)CAMK2CAMK5vloAn-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideHuman8348
CAMK2D (CaMK2d)CAMK2CAMK5vloBn-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideHuman8347
CAMK2D (CaMK2d)CAMK2CAMK6aywAn-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman8666
CAMK2D (CaMK2d)CAMK2CAMK6aywBn-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman8665
CAMK2G (CaMK2g)CAMK2CAMK2v7oAA-Human7239
CAMK2G (CaMK2g)CAMK2CAMK2v7oAB-Human7238
CAMK4 (CaMK4)CAMK1CAMK2w4oA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman2687
CAMKK1 (CaMKK1)CAMKKOther6ccfAn-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamideHuman9712
CAMKK1 (CaMKK1)CAMKKOther6ccfBn-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamideHuman9717
CAMKK1 (CaMKK1)CAMKKOther6cd6AA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9716
CAMKK1 (CaMKK1)CAMKKOther6cd6AB2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9714
CAMKK1 (CaMKK1)CAMKKOther6cd6BA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9709
CAMKK1 (CaMKK1)CAMKKOther6cd6BB2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9713
CAMKK1 (CaMKK1)CAMKKOther6cd6CA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9711
CAMKK1 (CaMKK1)CAMKKOther6cd6CB2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9715
CAMKK1 (CaMKK1)CAMKKOther6cd6DA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9710
CAMKK1 (CaMKK1)CAMKKOther6cd6DB2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9708
CAMKK2 (CaMKK2)CAMKKOther2zv2A7-oxo-7h-benzimidazo[2,1-a]benz[de]isoquinoline-3-carboxylic acidHuman406
CAMKK2 (CaMKK2)CAMKKOther5uy6A2-cyclopentyl-4-(5-phenylfuro[2,3-b]pyridin-3-yl)benzoic acidHuman7982
CAMKK2 (CaMKK2)CAMKKOther5uyjAA2-cyclopentyl-4-(7-methoxyquinolin-4-yl)benzoic acidHuman7560
CAMKK2 (CaMKK2)CAMKKOther5uyjAB2-cyclopentyl-4-(7-methoxyquinolin-4-yl)benzoic acidHuman7559
CAMKK2 (CaMKK2)CAMKKOther5vt1A4-({5-[(3-hydroxy-4-methylphenyl)amino]-4-oxo-4h-1,2,6-thiadiazin-3-yl}amino)benzamideHuman7591
CAMKK2 (CaMKK2)CAMKKOther5yv8AA1-amino-4-hydroxy-9,10-dioxo-9,10-dihydroanthracene-2-carboxylic acidHuman10753
CAMKK2 (CaMKK2)CAMKKOther5yv8AB1-amino-4-hydroxy-9,10-dioxo-9,10-dihydroanthracene-2-carboxylic acidHuman10755
CAMKK2 (CaMKK2)CAMKKOther5yv9A5-chloro-2-methoxy-4[(1z)-3-(4-methoxyphenyl)-3-oxoprop-1-en-1-yl]aminobenzoic acidHuman10752
CAMKK2 (CaMKK2)CAMKKOther5yvaA3-(1h-tetrazol-5-yl)-10lambda~6~-thioxanthene-9,10,10-trioneHuman10750
CAMKK2 (CaMKK2)CAMKKOther5yvbA(3z)-5-chloro-3-[(1-methyl-1h-pyrazol-4-yl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman10751
CAMKK2 (CaMKK2)CAMKKOther5yvcA3-{2,4-dimethyl-5-[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-1h-pyrrol-3-yl}propanoic acidHuman10754
CAMKK2 (CaMKK2)CAMKKOther6bkuA2-cyclopentyl-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman8687
CAMKK2 (CaMKK2)CAMKKOther6bleAA1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amineHuman8688
CAMKK2 (CaMKK2)CAMKKOther6bleAB1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amineHuman8689
CAMKK2 (CaMKK2)CAMKKOther6bqlA2-({5-chloro-2-[(2-methoxy-4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}amino)-n-methylbenzamideHuman9061
CAMKK2 (CaMKK2)CAMKKOther6bqpA1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amineHuman9064
CAMKK2 (CaMKK2)CAMKKOther6bqqA4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman9063
CAMKK2 (CaMKK2)CAMKKOther6brcA5-chloro-n~2~-{4-[4-(dimethylamino)piperidin-1-yl]-2-methoxyphenyl}-n~4~-[2-(dimethylphosphoryl)phenyl]pyrimidine-2,4-diamineHuman9062
CAMKK2 (CaMKK2)CAMKKOther6brcB5-chloro-n~2~-{4-[4-(dimethylamino)piperidin-1-yl]-2-methoxyphenyl}-n~4~-[2-(dimethylphosphoryl)phenyl]pyrimidine-2,4-diamineHuman9060
CAMKK2 (CaMKK2)CAMKKOther6cmjAA2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9784
CAMKK2 (CaMKK2)CAMKKOther6cmjAB2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9783
CAMKK2 (CaMKK2)CAMKKOther6cmjBA2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9786
CAMKK2 (CaMKK2)CAMKKOther6cmjBB2-(2-methylpropyl)-4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman9785
CAMKK2 (CaMKK2)CAMKKOther8tucAA(4m)-2-cyclopentyl-4-(7-ethoxyquinazolin-4-yl)benzoic acidHuman15005
CAMKK2 (CaMKK2)CAMKKOther8tucAB(4m)-2-cyclopentyl-4-(7-ethoxyquinazolin-4-yl)benzoic acidHuman15004
CASKCASKCAMK3c0gAA[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3828
CASKCASKCAMK3c0gAB[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3827
CASKCASKCAMK3c0gBA[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3824
CASKCASKCAMK3c0gBB[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3826
CASKCASKCAMK3c0hAadenosine monophosphateHuman3825
CASKCASKCAMK3c0hBadenosine monophosphateHuman3817
CASKCASKCAMK3c0iAA[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3830
CASKCASKCAMK3c0iAB[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3819
CASKCASKCAMK3mfrAAphosphoaminophosphonic acid-adenylate esterHuman3822
CASKCASKCAMK3mfrABphosphoaminophosphonic acid-adenylate esterHuman3831
CASKCASKCAMK3mfsAAphosphoaminophosphonic acid-adenylate esterHuman3818
CASKCASKCAMK3mfsABphosphoaminophosphonic acid-adenylate esterHuman3829
CASKCASKCAMK3mftAA-Human3823
CASKCASKCAMK3mftAB-Human3821
CASKCASKCAMK3mfuAAphosphoaminophosphonic acid-adenylate esterHuman3816
CASKCASKCAMK3mfuABphosphoaminophosphonic acid-adenylate esterHuman3832
CASKCASKCAMK3tacA-Human3820
CASKCASKCAMK6kmhA-Human12672
CASKCASKCAMK6kmhB-Human12671
CASKCASKCAMK7oaiAA4-(cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-n-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideHuman13584
CASKCASKCAMK7oaiAB4-(cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-n-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideHuman13583
CASKCASKCAMK7oajAA4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-n-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamideHuman13582
CASKCASKCAMK7oajAB4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-n-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamideHuman13581
CASKCASKCAMK7oakA2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclopentylamino)-n-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideHuman13585
CASKCASKCAMK7oalA2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclohexylamino)-n-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideHuman13586
CDC42BPB (MRCKb)DMPKAGC3qfvA2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamideHuman4860
CDC42BPB (MRCKb)DMPKAGC3qfvB2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamideHuman4857
CDC42BPB (MRCKb)DMPKAGC3tkuA5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman4862
CDC42BPB (MRCKb)DMPKAGC3tkuB5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman4859
CDC42BPB (MRCKb)DMPKAGC4uakAAadenosine-5'-diphosphateHuman4864
CDC42BPB (MRCKb)DMPKAGC4uakABadenosine-5'-diphosphateHuman4863
CDC42BPB (MRCKb)DMPKAGC4ualAA4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamideHuman4861
CDC42BPB (MRCKb)DMPKAGC4ualAB4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamideHuman4858
CDC42BPB (MRCKb)DMPKAGC5oteA2-[4-[(6~{s})-1,8-diazaspiro[5.5]undecan-8-yl]-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]-1,3-thiazoleHuman9578
CDC42BPB (MRCKb)DMPKAGC5otfA(6~{s})-8-(3-pyrimidin-4-yl-1~{h}-pyrrolo[2,3-b]pyridin-4-yl)-1,8-diazaspiro[5.5]undecaneHuman9577
CDC7CDC7Other4f99Aadenosine-5'-diphosphateHuman4824
CDC7CDC7Other4f9aAadenosine-5'-diphosphateHuman4825
CDC7CDC7Other4f9aCadenosine-5'-diphosphateHuman4826
CDC7CDC7Other4f9bA2-(pyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4828
CDC7CDC7Other4f9bC2-(pyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4827
CDC7CDC7Other4f9cA8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman4823
CDC7CDC7Other6ya6AA8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman13844
CDC7CDC7Other6ya6AB8-chloro-2-[(2s)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman13841
CDC7CDC7Other6ya7AAadenosine-5'-diphosphateHuman13845
CDC7CDC7Other6ya7ABadenosine-5'-diphosphateHuman13842
CDC7CDC7Other6ya8AAadenosine-5'-diphosphateHuman13846
CDC7CDC7Other6ya8ABadenosine-5'-diphosphateHuman13843
CDK1 (CDC2)CDKCMGC4y72AA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4610
CDK1 (CDC2)CDKCMGC4y72AB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4609
CDK1 (CDC2)CDKCMGC4yc3AA-Human6555
CDK1 (CDC2)CDKCMGC4yc3AB-Human6554
CDK1 (CDC2)CDKCMGC4yc6AA-Human4607
CDK1 (CDC2)CDKCMGC4yc6AB-Human4616
CDK1 (CDC2)CDKCMGC4yc6CA-Human4608
CDK1 (CDC2)CDKCMGC4yc6CB-Human4611
CDK1 (CDC2)CDKCMGC4yc6EA-Human4612
CDK1 (CDC2)CDKCMGC4yc6EB-Human4614
CDK1 (CDC2)CDKCMGC4yc6GA-Human4613
CDK1 (CDC2)CDKCMGC4yc6GB-Human4615
CDK1 (CDC2)CDKCMGC5hq0AA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman6422
CDK1 (CDC2)CDKCMGC5hq0AB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman6421
CDK1 (CDC2)CDKCMGC5lqfAAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7364
CDK1 (CDC2)CDKCMGC5lqfABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7366
CDK1 (CDC2)CDKCMGC5lqfDAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7365
CDK1 (CDC2)CDKCMGC5lqfDBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7367
CDK1 (CDC2)CDKCMGC6gu2AA2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10780
CDK1 (CDC2)CDKCMGC6gu2AB2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10776
CDK1 (CDC2)CDKCMGC6gu3A4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10778
CDK1 (CDC2)CDKCMGC6gu4A~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10777
CDK1 (CDC2)CDKCMGC6gu6A3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman10774
CDK1 (CDC2)CDKCMGC6gu7A4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10781
CDK1 (CDC2)CDKCMGC6gu7C-Human10775
CDK1 (CDC2)CDKCMGC6gu7E-Human10782
CDK1 (CDC2)CDKCMGC6gu7G-Human10779
CDK1 (CDC2)CDKCMGC7nj0B-Human13827
CDK12 (CRK7)CDKCMGC4cxaAphosphoaminophosphonic acid-adenylate esterHuman4856
CDK12 (CRK7)CDKCMGC4cxaC-Human4853
CDK12 (CRK7)CDKCMGC4nstAadenosine-5'-diphosphateHuman4852
CDK12 (CRK7)CDKCMGC4nstCadenosine-5'-diphosphateHuman4851
CDK12 (CRK7)CDKCMGC4un0C-Human4854
CDK12 (CRK7)CDKCMGC4un0D-Human4855
CDK12 (CRK7)CDKCMGC5acbCn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman6701
CDK12 (CRK7)CDKCMGC5acbDn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman6702
CDK12 (CRK7)CDKCMGC6b3eA2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-olHuman9452
CDK12 (CRK7)CDKCMGC6b3eC2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-olHuman9453
CDK12 (CRK7)CDKCMGC6ckxAn-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamideHuman10578
CDK12 (CRK7)CDKCMGC6ckxCn-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamideHuman10579
CDK12 (CRK7)CDKCMGC6td3B(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12371
CDK12 (CRK7)CDKCMGC6td3E(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12369
CDK12 (CRK7)CDKCMGC6td3H(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12370
CDK12 (CRK7)CDKCMGC7nxkA(e)-n-[4-[(1r,3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]cyclohexyl]oxyphenyl]-4-(dimethylamino)but-2-enamideHuman13547
CDK12 (CRK7)CDKCMGC8bu1B(2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-olHuman14930
CDK12 (CRK7)CDKCMGC8bu2B~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-propan-2-yl-purin-6-amineHuman14918
CDK12 (CRK7)CDKCMGC8bu3B2-morpholin-4-yl-9-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]purin-6-amineHuman14931
CDK12 (CRK7)CDKCMGC8bu4B(2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-olHuman14910
CDK12 (CRK7)CDKCMGC8bu5B~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman14926
CDK12 (CRK7)CDKCMGC8bu6B~{n}-(1~{h}-benzimidazol-2-ylmethyl)-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman14921
CDK12 (CRK7)CDKCMGC8bu7B-Human14913
CDK12 (CRK7)CDKCMGC8bu9Br-roscovitineHuman14914
CDK12 (CRK7)CDKCMGC8buaB(2~{r})-~{n}-(1~{h}-benzimidazol-2-yl)-2-(3-oxidanylidene-1~{h}-isoindol-2-yl)propanamideHuman14932
CDK12 (CRK7)CDKCMGC8bubB~{n}-(5-methyl-2,3-dihydro-1,3-thiazol-2-yl)-3-(5-methylfuran-2-yl)carbonyl-1,3-thiazolidine-4-carboxamideHuman14928
CDK12 (CRK7)CDKCMGC8bucB2-(1~{h}-benzimidazol-2-ylsulfanyl)-~{n}-(5-chloranylpyridin-2-yl)ethanamideHuman14909
CDK12 (CRK7)CDKCMGC8budB~{n}-(5-bromanylpyridin-2-yl)-3-(4-oxidanylidenequinazolin-3-yl)propanamideHuman14929
CDK12 (CRK7)CDKCMGC8bueB~{n}-(1~{h}-benzimidazol-2-yl)-1-(2-methoxy-5-methyl-phenyl)-5-oxidanylidene-pyrrolidine-3-carboxamideHuman14912
CDK12 (CRK7)CDKCMGC8bufB2-(6,7-dihydro-4~{h}-thieno[3,2-c]pyridin-5-ylmethyl)-6,7-dimethoxy-3~{h}-quinazolin-4-oneHuman14919
CDK12 (CRK7)CDKCMGC8bugB2-[2-[(6-methylpyridin-2-yl)amino]-1,3-thiazol-4-yl]-~{n}-(5-methyl-1,3-thiazol-2-yl)ethanamideHuman14935
CDK12 (CRK7)CDKCMGC8buhB6-[[[2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-9-propan-2-yl-purin-6-yl]amino]methyl]-3-pyridin-2-yl-1~{h}-pyridin-2-oneHuman14922
CDK12 (CRK7)CDKCMGC8buiB(2~{r})-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)amino]purin-2-yl]amino]butan-1-olHuman14925
CDK12 (CRK7)CDKCMGC8bujB(2~{r})-2-[[6-(octylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14933
CDK12 (CRK7)CDKCMGC8bukB(2~{r})-2-[[6-(naphthalen-2-ylmethylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14927
CDK12 (CRK7)CDKCMGC8bulB(2~{r})-2-[[6-(3-phenylpropylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14911
CDK12 (CRK7)CDKCMGC8bumB(2r)-2-[[6-(5-naphthalen-1-ylpentylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14924
CDK12 (CRK7)CDKCMGC8bunB(2~{r})-2-[[6-[(4-phenylphenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14916
CDK12 (CRK7)CDKCMGC8buoB(2~{r})-2-[[6-[(3-fluoranyl-4-pyridin-2-yl-phenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14934
CDK12 (CRK7)CDKCMGC8bupB(2~{r})-2-[[6-[3-(3-methylphenyl)propylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14923
CDK12 (CRK7)CDKCMGC8buqB(2~{r})-2-[[6-[[1-(3-chlorophenyl)pyrazol-3-yl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14917
CDK12 (CRK7)CDKCMGC8burBA~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamideHuman14915
CDK12 (CRK7)CDKCMGC8burBB~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamideHuman14920
CDK12 (CRK7)CDKCMGC8busB1,3-dimethyl-5-[[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]methyl]pyrazole-4-sulfonamideHuman14908
CDK12 (CRK7)CDKCMGC8butB2-[[6-[[4-(2-hydroxyethyloxy)phenyl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14936
CDK12 (CRK7)CDKCMGC8p81AA~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman15062
CDK12 (CRK7)CDKCMGC8p81AB~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman15061
CDK13 (CHED)CDKCMGC5efqAadenosine-5'-diphosphateHuman6323
CDK13 (CHED)CDKCMGC5efqCadenosine-5'-diphosphateHuman6324
CDK13 (CHED)CDKCMGC7nxjAn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman13544
CDK16 (PCTAIRE1)CDKCMGC3mtlAA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human1701
CDK16 (PCTAIRE1)CDKCMGC3mtlAB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human1702
CDK16 (PCTAIRE1)CDKCMGC5g6vA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman7273
CDK16 (PCTAIRE1)CDKCMGC5g6vB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman7274
CDK2CDKCMGC1aq1AstaurosporineHuman4267
CDK2CDKCMGC1b38Aadenosine-5'-triphosphateHuman4483
CDK2CDKCMGC1b39Aadenosine-5'-triphosphateHuman4407
CDK2CDKCMGC1buhA-Human4178
CDK2CDKCMGC1ckpAApurvalanol bHuman4066
CDK2CDKCMGC1ckpABpurvalanol bHuman4214
CDK2CDKCMGC1di8A4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman4577
CDK2CDKCMGC1dm2AA4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHuman4104
CDK2CDKCMGC1dm2AB4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHuman4024
CDK2CDKCMGC1e1vA6-o-cyclohexylmethyl guanineHuman3886
CDK2CDKCMGC1e1xA6-cyclohexylmethyloxy-5-nitroso-pyrimidine-2,4-diamineHuman4114
CDK2CDKCMGC1e9hA2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHuman4302
CDK2CDKCMGC1e9hC2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHuman4570
CDK2CDKCMGC1f5qAA-Human4194
CDK2CDKCMGC1f5qAB-Human4517
CDK2CDKCMGC1f5qCA-Human4281
CDK2CDKCMGC1f5qCB-Human3952
CDK2CDKCMGC1finAadenosine-5'-triphosphateHuman4367
CDK2CDKCMGC1finCadenosine-5'-triphosphateHuman4479
CDK2CDKCMGC1fq1Badenosine-5'-triphosphateHuman4266
CDK2CDKCMGC1fvtA4-(5-bromo-2-oxo-2h-indol-3-ylazo)-benzenesulfonamideHuman4480
CDK2CDKCMGC1fvvA4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman4065
CDK2CDKCMGC1fvvC4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman4461
CDK2CDKCMGC1g5sA2-[trans-(4-aminocyclohexyl)amino]-6-(benzyl-amino)-9-cyclopentylpurineHuman3888
CDK2CDKCMGC1gihA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHuman3922
CDK2CDKCMGC1giiA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHuman4448
CDK2CDKCMGC1gijA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-(5-pyrrolidin-2-yl-1h-pyrazol-3-yl)-ureaHuman4542
CDK2CDKCMGC1gy3Aadenosine-5'-triphosphateHuman3978
CDK2CDKCMGC1gy3Cadenosine-5'-triphosphateHuman4445
CDK2CDKCMGC1gz8AA1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHuman3981
CDK2CDKCMGC1gz8AB1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHuman3956
CDK2CDKCMGC1h00AA(2s)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4484
CDK2CDKCMGC1h00AB(2r)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4428
CDK2CDKCMGC1h01AA(2r)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman3974
CDK2CDKCMGC1h01AB(2s)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4561
CDK2CDKCMGC1h07AA((2-bromo-4-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHuman3918
CDK2CDKCMGC1h07AB((2-bromo-4-methylphenyl){6-[(4-{[(2s)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHuman3908
CDK2CDKCMGC1h08AA(2r)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHuman4220
CDK2CDKCMGC1h08AB(2s)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHuman4411
CDK2CDKCMGC1h0vAA5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHuman4368
CDK2CDKCMGC1h0vAB5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHuman3933
CDK2CDKCMGC1h0wAA1-amino-6-cyclohex-3-enylmethyloxypurineHuman3987
CDK2CDKCMGC1h0wAB1-amino-6-cyclohex-3-enylmethyloxypurineHuman4016
CDK2CDKCMGC1h1pA6-o-cyclohexylmethyl guanineHuman4309
CDK2CDKCMGC1h1pC6-o-cyclohexylmethyl guanineHuman4581
CDK2CDKCMGC1h1qA2-anilino-6-cyclohexylmethoxypurineHuman4195
CDK2CDKCMGC1h1qC2-anilino-6-cyclohexylmethoxypurineHuman4053
CDK2CDKCMGC1h1rAA6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman3906
CDK2CDKCMGC1h1rAB6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman4494
CDK2CDKCMGC1h1rCA6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman3920
CDK2CDKCMGC1h1rCB6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman4081
CDK2CDKCMGC1h1sAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4400
CDK2CDKCMGC1h1sCo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4572
CDK2CDKCMGC1h24A-Human4199
CDK2CDKCMGC1h24C-Human4296
CDK2CDKCMGC1h25A-Human4273
CDK2CDKCMGC1h25C-Human4112
CDK2CDKCMGC1h26A-Human4122
CDK2CDKCMGC1h26C-Human4179
CDK2CDKCMGC1h27A-Human4116
CDK2CDKCMGC1h27C-Human4030
CDK2CDKCMGC1h28A-Human4169
CDK2CDKCMGC1h28C-Human4351
CDK2CDKCMGC1hckAAadenosine-5'-triphosphateHuman3878
CDK2CDKCMGC1hckABadenosine-5'-triphosphateHuman4416
CDK2CDKCMGC1hclAA-Human4545
CDK2CDKCMGC1hclAB-Human4540
CDK2CDKCMGC1jstAadenosine-5'-triphosphateHuman4455
CDK2CDKCMGC1jstCadenosine-5'-triphosphateHuman4356
CDK2CDKCMGC1jsuA-Human4146
CDK2CDKCMGC1jsvA4-[(6-amino-4-pyrimidinyl)amino]benzenesulfonamideHuman4171
CDK2CDKCMGC1jvpP13-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazoleHuman3919
CDK2CDKCMGC1jvpP23-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazoleHuman4097
CDK2CDKCMGC1ke5An-methyl-4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4376
CDK2CDKCMGC1ke6An-methyl-{4-[2-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)hydrazino]phenyl}methanesulfonamideHuman4219
CDK2CDKCMGC1ke7A3-{[(2,2-dioxido-1,3-dihydro-2-benzothien-5-yl)amino]methylene}-5-(1,3-oxazol-5-yl)-1,3-dihydro-2h-indol-2-oneHuman4295
CDK2CDKCMGC1ke8A4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}-n-(1,3-thiazol-2-yl)benzenesulfonamideHuman4048
CDK2CDKCMGC1ke9A3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4250
CDK2CDKCMGC1oguAA4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3965
CDK2CDKCMGC1oguAB4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3935
CDK2CDKCMGC1oguCA4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3964
CDK2CDKCMGC1oguCB4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman4560
CDK2CDKCMGC1oi9AA6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4033
CDK2CDKCMGC1oi9AB6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4492
CDK2CDKCMGC1oi9CA6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4571
CDK2CDKCMGC1oi9CB6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4036
CDK2CDKCMGC1oiqAn-[4-(2-methylimidazo[1,2-a]pyridin-3-yl)-2-pyrimidinyl]acetamideHuman4379
CDK2CDKCMGC1oirA1-(dimethylamino)-3-(4-{{4-(2-methylimidazo[1,2-a]pyridin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4389
CDK2CDKCMGC1oitA4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]benzenesulfonamideHuman4025
CDK2CDKCMGC1oiuAA3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4110
CDK2CDKCMGC1oiuAB3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4556
CDK2CDKCMGC1oiuCA3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4524
CDK2CDKCMGC1oiuCB3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4049
CDK2CDKCMGC1oiyAA4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4225
CDK2CDKCMGC1oiyAB4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman3945
CDK2CDKCMGC1oiyCA4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4465
CDK2CDKCMGC1oiyCB4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4245
CDK2CDKCMGC1okvA-Human3921
CDK2CDKCMGC1okvC-Human4093
CDK2CDKCMGC1okwA-Human4314
CDK2CDKCMGC1okwC-Human3896
CDK2CDKCMGC1ol1A-Human4429
CDK2CDKCMGC1ol1C-Human3951
CDK2CDKCMGC1ol2A-Human4305
CDK2CDKCMGC1ol2C-Human4497
CDK2CDKCMGC1p2aA5-[(2-aminoethyl)amino]-6-fluoro-3-(1h-pyrrol-2-yl)benzo[cd]indol-2(1h)-oneHuman4422
CDK2CDKCMGC1p5eA4,5,6,7-tetrabromobenzotriazoleHuman4090
CDK2CDKCMGC1p5eC4,5,6,7-tetrabromobenzotriazoleHuman4434
CDK2CDKCMGC1pf8A(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3861
CDK2CDKCMGC1pkdA7-hydroxystaurosporineHuman4170
CDK2CDKCMGC1pkdC7-hydroxystaurosporineHuman3973
CDK2CDKCMGC1pw2A-Human4432
CDK2CDKCMGC1pxiAA4-(2,5-dichlorothien-3-yl)pyrimidin-2-amineHuman4381
CDK2CDKCMGC1pxiAB-Human3924
CDK2CDKCMGC1pxjAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman3927
CDK2CDKCMGC1pxjAB-Human3911
CDK2CDKCMGC1pxkAAn-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n'-hydroxyimidoformamideHuman3915
CDK2CDKCMGC1pxkAB-Human3980
CDK2CDKCMGC1pxlAA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4233
CDK2CDKCMGC1pxlAB-Human4074
CDK2CDKCMGC1pxmAA3-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-ylamino]-phenolHuman3944
CDK2CDKCMGC1pxmAB-Human3936
CDK2CDKCMGC1pxnAA4-[4-(4-methyl-2-methylamino-thiazol-5-yl)-pyrimidin-2-ylamino]-phenolHuman4383
CDK2CDKCMGC1pxnAB-Human4172
CDK2CDKCMGC1pxoAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4512
CDK2CDKCMGC1pxoAB-Human3860
CDK2CDKCMGC1pxoAC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4546
CDK2CDKCMGC1pxoAD[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4167
CDK2CDKCMGC1pxpAAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4316
CDK2CDKCMGC1pxpAB-Human3943
CDK2CDKCMGC1pyeA[2-amino-6-(2,6-difluoro-benzoyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl-methanoneHuman4284
CDK2CDKCMGC1qmzAadenosine-5'-triphosphateHuman4242
CDK2CDKCMGC1qmzCadenosine-5'-triphosphateHuman4527
CDK2CDKCMGC1r78AA4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman4253
CDK2CDKCMGC1r78AB4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman4249
CDK2CDKCMGC1urcAA-Human4334
CDK2CDKCMGC1urcAB-Human4010
CDK2CDKCMGC1urcCA-Human4006
CDK2CDKCMGC1urcCB-Human3937
CDK2CDKCMGC1urwAA2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]-Human4054
CDK2CDKCMGC1urwAB2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]-Human4196
CDK2CDKCMGC1v1kAA(2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-olHuman4189
CDK2CDKCMGC1v1kAB(2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-olHuman3928
CDK2CDKCMGC1vywAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamideHuman3992
CDK2CDKCMGC1vywCn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamideHuman4133
CDK2CDKCMGC1vyzAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzamideHuman4325
CDK2CDKCMGC1w0xCAolomoucineHuman4537
CDK2CDKCMGC1w0xCBolomoucineHuman4478
CDK2CDKCMGC1w8cAA6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHuman4332
CDK2CDKCMGC1w8cAB6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHuman4197
CDK2CDKCMGC1w98A-Human4013
CDK2CDKCMGC1wccAA2-amino-6-chloropyrazineHuman4394
CDK2CDKCMGC1wccAB2-amino-6-chloropyrazineHuman3897
CDK2CDKCMGC1y8yA(5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-(4-methanesulfonylphenyl)amineHuman3914
CDK2CDKCMGC1y91A4-[5-(trans-4-aminocyclohexylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-7-ylamino]-n,n-dimethylbenzenesulfonamideHuman4505
CDK2CDKCMGC1ykrA4-{[6-(2,6-dichlorobenzoyl)imidazo[1,2-a]pyridin-2-yl]amino}benzenesulfonamideHuman4578
CDK2CDKCMGC2a0cXA2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHuman4157
CDK2CDKCMGC2a0cXB2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHuman3868
CDK2CDKCMGC2a4lAr-roscovitineHuman4238
CDK2CDKCMGC2b52A1-(3-(2,4-dimethylthiazol-5-yl)-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)-3-(4-methylpiperazin-1-yl)ureaHuman3997
CDK2CDKCMGC2b53A6-(3-aminophenyl)-n-(tert-butyl)-2-(trifluoromethyl)quinazolin-4-amineHuman3875
CDK2CDKCMGC2b54A6-(3,4-dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4(5h)-oneHuman4292
CDK2CDKCMGC2b55A2-(4-(aminomethyl)piperidin-1-yl)-n-(3_cyclohexyl-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)acetamideHuman4216
CDK2CDKCMGC2bheA(2z)-5'-bromo-2,3'-biindole-2',3(1h,1'h)-dione ammoniateHuman4184
CDK2CDKCMGC2bhhA(2e,3s)-3-hydroxy-5'-[(4-hydroxypiperidin-1-yl)sulfonyl]-3-methyl-1,3-dihydro-2,3'-biindol-2'(1'h)-oneHuman4417
CDK2CDKCMGC2bkzA1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHuman3942
CDK2CDKCMGC2bkzC1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHuman4555
CDK2CDKCMGC2bpmA(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHuman4042
CDK2CDKCMGC2bpmC(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHuman4128
CDK2CDKCMGC2btrAn-(5-isopropyl-thiazol-2-yl)-2-pyridin-3-yl-acetamideHuman3998
CDK2CDKCMGC2btsA4-[(5-isopropyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4443
CDK2CDKCMGC2c4gA(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHuman4088
CDK2CDKCMGC2c4gC(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHuman4453
CDK2CDKCMGC2c5nAAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4063
CDK2CDKCMGC2c5nABn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4223
CDK2CDKCMGC2c5nCAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4161
CDK2CDKCMGC2c5nCBn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman3903
CDK2CDKCMGC2c5oAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4388
CDK2CDKCMGC2c5oAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4440
CDK2CDKCMGC2c5oCA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4414
CDK2CDKCMGC2c5oCB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4050
CDK2CDKCMGC2c5vAA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4012
CDK2CDKCMGC2c5vAB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4338
CDK2CDKCMGC2c5vCA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4384
CDK2CDKCMGC2c5vCB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4209
CDK2CDKCMGC2c5xAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4312
CDK2CDKCMGC2c5xABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman3892
CDK2CDKCMGC2c5xCAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4466
CDK2CDKCMGC2c5xCBhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4418
CDK2CDKCMGC2c5yAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman6785
CDK2CDKCMGC2c5yABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman6777
CDK2CDKCMGC2c68A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydropyrazolo[1,5-a]pyrimidin-7-amineHuman6776
CDK2CDKCMGC2c69A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-7-amineHuman6775
CDK2CDKCMGC2c6iA4-{[5-(cyclohexylmethoxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6774
CDK2CDKCMGC2c6kA4-{[5-(cyclohexylamino)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6773
CDK2CDKCMGC2c6lA4-({5-[(4-aminocyclohexyl)amino][1,2,4]triazolo[1,5-a]pyrimidin-7-yl}amino)benzenesulfonamideHuman6779
CDK2CDKCMGC2c6mA4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6782
CDK2CDKCMGC2c6oAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman6783
CDK2CDKCMGC2c6tA4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman4371
CDK2CDKCMGC2c6tC4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman3994
CDK2CDKCMGC2cchAAadenosine-5'-triphosphateHuman4303
CDK2CDKCMGC2cchABadenosine-5'-triphosphateHuman4553
CDK2CDKCMGC2cchAC-Human4566
CDK2CDKCMGC2cchCAadenosine-5'-triphosphateHuman3932
CDK2CDKCMGC2cchCBadenosine-5'-triphosphateHuman4000
CDK2CDKCMGC2cchCC-Human4431
CDK2CDKCMGC2cciAadenosine-5'-triphosphateHuman4373
CDK2CDKCMGC2cciCadenosine-5'-triphosphateHuman4532
CDK2CDKCMGC2cjmAadenosine-5'-triphosphateHuman4406
CDK2CDKCMGC2cjmCadenosine-5'-triphosphateHuman4126
CDK2CDKCMGC2clxAA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3909
CDK2CDKCMGC2clxAB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3880
CDK2CDKCMGC2ds1A(13r,15s)-13-methyl-16-oxa-8,9,12,22,24-pentaazahexacyclo[15.6.2.16,9.1,12,15.0,2,7.0,21,25]heptacosa-1(24),2,4,6,17(25),18,20-heptaene-23,26-dioneHuman4513
CDK2CDKCMGC2duvA2-(3,4-dihydroxyphenyl)-8-(1,1-dioxidoisothiazolidin-2-yl)-3-hydroxy-6-methyl-4h-chromen-4-oneHuman4193
CDK2CDKCMGC2exmAn-(3-methylbut-2-en-1-yl)-9h-purin-6-amineHuman4055
CDK2CDKCMGC2fvdA(4-amino-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrimidin-5-yl)(2,3-difluoro-6-methoxyphenyl)methanoneHuman4408
CDK2CDKCMGC2g9xA3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-olHuman3883
CDK2CDKCMGC2g9xC3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-olHuman4082
CDK2CDKCMGC2i40AA5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4363
CDK2CDKCMGC2i40AB5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4470
CDK2CDKCMGC2i40CA5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4222
CDK2CDKCMGC2i40CB5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4043
CDK2CDKCMGC2iw6A[(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrileHuman4019
CDK2CDKCMGC2iw6C[(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrileHuman4108
CDK2CDKCMGC2iw8AAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4142
CDK2CDKCMGC2iw8ABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4377
CDK2CDKCMGC2iw8CAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4294
CDK2CDKCMGC2iw8CBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4350
CDK2CDKCMGC2iw9AAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4174
CDK2CDKCMGC2iw9ABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3955
CDK2CDKCMGC2iw9CAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4218
CDK2CDKCMGC2iw9CBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3858
CDK2CDKCMGC2j9mAA6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxideHuman4154
CDK2CDKCMGC2j9mAB6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxideHuman4246
CDK2CDKCMGC2jgzA-Human4117
CDK2CDKCMGC2r3fAA5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4175
CDK2CDKCMGC2r3fAB5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4291
CDK2CDKCMGC2r3gAA6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman4276
CDK2CDKCMGC2r3gAB6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman3923
CDK2CDKCMGC2r3hAA3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman4152
CDK2CDKCMGC2r3hAB3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman3970
CDK2CDKCMGC2r3iAA5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4135
CDK2CDKCMGC2r3iAB5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4059
CDK2CDKCMGC2r3iAC-Human4317
CDK2CDKCMGC2r3jAA3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4185
CDK2CDKCMGC2r3jAB3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4544
CDK2CDKCMGC2r3kAA3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman3953
CDK2CDKCMGC2r3kAB3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman3876
CDK2CDKCMGC2r3kAC3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman4022
CDK2CDKCMGC2r3lAA3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4200
CDK2CDKCMGC2r3lAB3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4085
CDK2CDKCMGC2r3lAC3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4496
CDK2CDKCMGC2r3mAAn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHuman4286
CDK2CDKCMGC2r3mABn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHuman4576
CDK2CDKCMGC2r3nAA3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4101
CDK2CDKCMGC2r3nAB3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4046
CDK2CDKCMGC2r3oAA(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4147
CDK2CDKCMGC2r3oAB(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4354
CDK2CDKCMGC2r3oAC(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4229
CDK2CDKCMGC2r3pAA5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHuman4176
CDK2CDKCMGC2r3pAB5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHuman4392
CDK2CDKCMGC2r3qAA3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman4038
CDK2CDKCMGC2r3qAB3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman4459
CDK2CDKCMGC2r3qAC3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman3976
CDK2CDKCMGC2r3rAA3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4040
CDK2CDKCMGC2r3rAB3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4215
CDK2CDKCMGC2r64An-[5-(1,1-dioxidoisothiazolidin-2-yl)-1h-indazol-3-yl]-2-(4-piperidin-1-ylphenyl)acetamideHuman4425
CDK2CDKCMGC2uueA4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHuman4515
CDK2CDKCMGC2uueC4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHuman4321
CDK2CDKCMGC2uzbAC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4099
CDK2CDKCMGC2uzbAD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman3866
CDK2CDKCMGC2uzbCC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4045
CDK2CDKCMGC2uzbCD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4502
CDK2CDKCMGC2uzdA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3877
CDK2CDKCMGC2uzdC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3900
CDK2CDKCMGC2uzeA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHuman3949
CDK2CDKCMGC2uzeC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHuman4071
CDK2CDKCMGC2uzlA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHuman3917
CDK2CDKCMGC2uzlC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHuman4106
CDK2CDKCMGC2uznA4-{5-[(1z)-1-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)ethyl]-2-furyl}benzenesulfonamideHuman4064
CDK2CDKCMGC2uzoA4-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3862
CDK2CDKCMGC2v0dA2-imino-5-(1-pyridin-2-yl-meth-(e)-ylidene)-1,3-thiazolidin-4-oneHuman4327
CDK2CDKCMGC2v22A-Human4077
CDK2CDKCMGC2v22C-Human4255
CDK2CDKCMGC2vtaA1h-indazoleHuman4118
CDK2CDKCMGC2vthA5-hydroxynaphthalene-1-sulfonamideHuman4274
CDK2CDKCMGC2vtiAn-(4-sulfamoylphenyl)-1h-indazole-3-carboxamideHuman4177
CDK2CDKCMGC2vtjA4-[(6-chloropyrazin-2-yl)amino]benzenesulfonamideHuman3959
CDK2CDKCMGC2vtlAn-phenyl-1h-pyrazole-3-carboxamideHuman3870
CDK2CDKCMGC2vtmApyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4283
CDK2CDKCMGC2vtnA4-(acetylamino)-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4027
CDK2CDKCMGC2vtoAAn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHuman4421
CDK2CDKCMGC2vtoABn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHuman3946
CDK2CDKCMGC2vtpAA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4511
CDK2CDKCMGC2vtpAB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4401
CDK2CDKCMGC2vtqA{[(2,6-difluorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman3891
CDK2CDKCMGC2vtrAA5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4391
CDK2CDKCMGC2vtrAB5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman3907
CDK2CDKCMGC2vtsA5-[(4-aminocyclohexyl)amino]-7-(propan-2-ylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4300
CDK2CDKCMGC2vttA4-{[(2,6-difluorophenyl)carbonyl]amino}-n-[(3s)-piperidin-3-yl]-1h-pyrazole-3-carboxamideHuman4100
CDK2CDKCMGC2vu3AA4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman4582
CDK2CDKCMGC2vu3AB4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman3884
CDK2CDKCMGC2vv9AA2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHuman3989
CDK2CDKCMGC2vv9AB2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHuman3881
CDK2CDKCMGC2w05AAn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHuman4547
CDK2CDKCMGC2w05ABn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHuman4256
CDK2CDKCMGC2w06A4-{[4-(1-cyclopropyl-2-methyl-1h-imidazol-5-yl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman3982
CDK2CDKCMGC2w17AAn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman3968
CDK2CDKCMGC2w17ABn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman4165
CDK2CDKCMGC2w1hAn-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamideHuman4228
CDK2CDKCMGC2wevAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4067
CDK2CDKCMGC2wevAB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4580
CDK2CDKCMGC2wevAC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4007
CDK2CDKCMGC2wevCA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4503
CDK2CDKCMGC2wevCB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman3859
CDK2CDKCMGC2wevCC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4288
CDK2CDKCMGC2wfyAA-Human4324
CDK2CDKCMGC2wfyAB-Human4426
CDK2CDKCMGC2wfyCA-Human4329
CDK2CDKCMGC2wfyCB-Human4096
CDK2CDKCMGC2whbAA-Human4471
CDK2CDKCMGC2whbAB-Human4457
CDK2CDKCMGC2whbCA-Human4132
CDK2CDKCMGC2whbCB-Human4352
CDK2CDKCMGC2wihAn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4163
CDK2CDKCMGC2wihCn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4119
CDK2CDKCMGC2wipA1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHuman4520
CDK2CDKCMGC2wipC1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHuman4190
CDK2CDKCMGC2wmaA-Human4435
CDK2CDKCMGC2wmaC-Human4410
CDK2CDKCMGC2wmbA-Human4060
CDK2CDKCMGC2wmbC-Human4474
CDK2CDKCMGC2wpaAn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHuman4399
CDK2CDKCMGC2wpaCn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHuman4162
CDK2CDKCMGC2wxvAn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4318
CDK2CDKCMGC2wxvCn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4504
CDK2CDKCMGC2x1nAA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4579
CDK2CDKCMGC2x1nAB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4078
CDK2CDKCMGC2x1nCA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman3991
CDK2CDKCMGC2x1nCB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4062
CDK2CDKCMGC2xmyAA4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHuman4526
CDK2CDKCMGC2xmyAB4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHuman3985
CDK2CDKCMGC2xnbAA3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHuman4217
CDK2CDKCMGC2xnbAB3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHuman4034
CDK2CDKCMGC3bhtAA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman3950
CDK2CDKCMGC3bhtAB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4491
CDK2CDKCMGC3bhtCA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4151
CDK2CDKCMGC3bhtCB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman3889
CDK2CDKCMGC3bhuAA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4105
CDK2CDKCMGC3bhuAB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4446
CDK2CDKCMGC3bhuCA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4087
CDK2CDKCMGC3bhuCB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4464
CDK2CDKCMGC3bhvAA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4531
CDK2CDKCMGC3bhvAB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4001
CDK2CDKCMGC3bhvCA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4353
CDK2CDKCMGC3bhvCB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4529
CDK2CDKCMGC3ddpAA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6781
CDK2CDKCMGC3ddpAB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6780
CDK2CDKCMGC3ddpCA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6784
CDK2CDKCMGC3ddpCB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6778
CDK2CDKCMGC3ddqAAr-roscovitineHuman4477
CDK2CDKCMGC3ddqABr-roscovitineHuman4269
CDK2CDKCMGC3ddqCAr-roscovitineHuman4364
CDK2CDKCMGC3ddqCBr-roscovitineHuman4289
CDK2CDKCMGC3dogAA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4541
CDK2CDKCMGC3dogAB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4365
CDK2CDKCMGC3dogCA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4382
CDK2CDKCMGC3dogCB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4121
CDK2CDKCMGC3eidAA(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4386
CDK2CDKCMGC3eidAB(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4424
CDK2CDKCMGC3eidCA-Human4072
CDK2CDKCMGC3eidCB-Human4467
CDK2CDKCMGC3ej1An-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHuman4168
CDK2CDKCMGC3ej1Cn-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHuman4092
CDK2CDKCMGC3eocA5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman4390
CDK2CDKCMGC3eocC5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman3969
CDK2CDKCMGC3ezrA3-methoxy-4-{3-[4-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman4475
CDK2CDKCMGC3ezvA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman4083
CDK2CDKCMGC3f5xA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman3882
CDK2CDKCMGC3f5xC4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman3894
CDK2CDKCMGC3fz1A(3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-oneHuman4335
CDK2CDKCMGC3ig7An-{1-[cis-3-(acetylamino)cyclobutyl]-1h-imidazol-4-yl}-2-(4-methoxyphenyl)acetamideHuman4021
CDK2CDKCMGC3iggAn-[1-(cis-3-hydroxycyclobutyl)-1h-imidazol-4-yl]-2-(4-methoxyphenyl)acetamideHuman4360
CDK2CDKCMGC3le6A5-(2-chlorophenyl)-3-methyl-7-nitropyrazolo[3,4-b][1,4]benzodiazepineHuman4125
CDK2CDKCMGC3lfnAn-[6-(4-hydroxyphenyl)-5-phenyl-1h-indazol-3-yl]butanamideHuman4330
CDK2CDKCMGC3lfqAn-(6,7-difluoro-5-phenyl-1h-indazol-3-yl)butanamideHuman4320
CDK2CDKCMGC3lfsAn-(6-chloro-5-phenyl-1h-indazol-3-yl)butanamideHuman4069
CDK2CDKCMGC3my5AA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4554
CDK2CDKCMGC3my5AB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3887
CDK2CDKCMGC3my5AC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3910
CDK2CDKCMGC3my5CA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4473
CDK2CDKCMGC3my5CB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4003
CDK2CDKCMGC3my5CC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3929
CDK2CDKCMGC3ns9A(2s,3s)-3-{[7-(benzylamino)-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-5-yl]amino}butane-1,2,4-triolHuman4575
CDK2CDKCMGC3pj8AA(2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-olHuman4375
CDK2CDKCMGC3pj8AB(2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-olHuman4454
CDK2CDKCMGC3pxfAA8-anilino-1-naphthalene sulfonateHuman4047
CDK2CDKCMGC3pxfAB8-anilino-1-naphthalene sulfonateHuman4301
CDK2CDKCMGC3pxqA8-anilino-1-naphthalene sulfonateHuman3947
CDK2CDKCMGC3pxrAA-Human3941
CDK2CDKCMGC3pxrAB-Human4173
CDK2CDKCMGC3pxyAA2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenolHuman4057
CDK2CDKCMGC3pxyAB2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenolHuman3904
CDK2CDKCMGC3pxzA8-anilino-1-naphthalene sulfonateHuman4251
CDK2CDKCMGC3py0AA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3995
CDK2CDKCMGC3py0AB(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3869
CDK2CDKCMGC3py1AA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman4361
CDK2CDKCMGC3py1AB(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman4444
CDK2CDKCMGC3qhrAadenosine-5'-diphosphateHuman4458
CDK2CDKCMGC3qhrCadenosine-5'-diphosphateHuman3879
CDK2CDKCMGC3qhwAAadenosine-5'-diphosphateHuman4346
CDK2CDKCMGC3qhwABadenosine-5'-diphosphateHuman4156
CDK2CDKCMGC3qhwCAadenosine-5'-diphosphateHuman4129
CDK2CDKCMGC3qhwCBadenosine-5'-diphosphateHuman4143
CDK2CDKCMGC3ql8AA3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrileHuman3916
CDK2CDKCMGC3ql8AB3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrileHuman4306
CDK2CDKCMGC3qqfAA5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4211
CDK2CDKCMGC3qqfAB5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4287
CDK2CDKCMGC3qqgAA4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4130
CDK2CDKCMGC3qqgAB4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4310
CDK2CDKCMGC3qqhAA2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenolHuman4393
CDK2CDKCMGC3qqhAB2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenolHuman4533
CDK2CDKCMGC3qqjAA2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4113
CDK2CDKCMGC3qqjAB2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4204
CDK2CDKCMGC3qqkAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4568
CDK2CDKCMGC3qqkAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4514
CDK2CDKCMGC3qqlAA(5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4341
CDK2CDKCMGC3qqlAB(5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4378
CDK2CDKCMGC3qrtAA(5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4586
CDK2CDKCMGC3qrtAB(5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4536
CDK2CDKCMGC3qruAA(5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4237
CDK2CDKCMGC3qruAB(5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4516
CDK2CDKCMGC3qtqAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4210
CDK2CDKCMGC3qtqAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4103
CDK2CDKCMGC3qtrAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman3874
CDK2CDKCMGC3qtrAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4243
CDK2CDKCMGC3qtsAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanoneHuman4275
CDK2CDKCMGC3qtsAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanoneHuman4564
CDK2CDKCMGC3qtuAA4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4009
CDK2CDKCMGC3qtuAB4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4323
CDK2CDKCMGC3qtwAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4397
CDK2CDKCMGC3qtwAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman3890
CDK2CDKCMGC3qtxAA4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4339
CDK2CDKCMGC3qtxAB4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4419
CDK2CDKCMGC3qtzAA4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4109
CDK2CDKCMGC3qtzAB4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4337
CDK2CDKCMGC3qu0AA4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4427
CDK2CDKCMGC3qu0AB4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4558
CDK2CDKCMGC3qwjAA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamideHuman4265
CDK2CDKCMGC3qwjAB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamideHuman4182
CDK2CDKCMGC3qwkAA4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4091
CDK2CDKCMGC3qwkAB4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4155
CDK2CDKCMGC3qx2AA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamideHuman4031
CDK2CDKCMGC3qx2AB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamideHuman4297
CDK2CDKCMGC3qx4AA4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4409
CDK2CDKCMGC3qx4AB4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3990
CDK2CDKCMGC3qxoA5-nitro-2-[(4-sulfamoylbenzyl)amino]benzamideHuman4282
CDK2CDKCMGC3qxpAA4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4343
CDK2CDKCMGC3qxpAB4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4482
CDK2CDKCMGC3qzfA2-(4,6-diamino-1,3,5-triazin-2-yl)benzene-1,4-diolHuman4569
CDK2CDKCMGC3qzgAA2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenolHuman4144
CDK2CDKCMGC3qzgAB2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenolHuman4347
CDK2CDKCMGC3qzhA4-methoxy-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3954
CDK2CDKCMGC3qziAA4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamideHuman4094
CDK2CDKCMGC3qziAB4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamideHuman4500
CDK2CDKCMGC3r1qAA4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4224
CDK2CDKCMGC3r1qAB4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4507
CDK2CDKCMGC3r1sAA2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4263
CDK2CDKCMGC3r1sAB2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4358
CDK2CDKCMGC3r1yAA2-[(pyridin-3-ylmethyl)amino]benzamideHuman4319
CDK2CDKCMGC3r1yAB2-[(pyridin-3-ylmethyl)amino]benzamideHuman4405
CDK2CDKCMGC3r28AA4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamideHuman4052
CDK2CDKCMGC3r28AB4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamideHuman4293
CDK2CDKCMGC3r6xAA4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4398
CDK2CDKCMGC3r6xAB4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4107
CDK2CDKCMGC3r71AA4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3962
CDK2CDKCMGC3r71AB4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4345
CDK2CDKCMGC3r73AA4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4187
CDK2CDKCMGC3r73AB4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3899
CDK2CDKCMGC3r7eAA5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamideHuman4159
CDK2CDKCMGC3r7eAB5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamideHuman4447
CDK2CDKCMGC3r7iAA4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acidHuman4450
CDK2CDKCMGC3r7iAB4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acidHuman4070
CDK2CDKCMGC3r7uAA2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamideHuman4510
CDK2CDKCMGC3r7uAB2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamideHuman4023
CDK2CDKCMGC3r7vAA5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamideHuman4380
CDK2CDKCMGC3r7vAB5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamideHuman4183
CDK2CDKCMGC3r7yAA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamideHuman4476
CDK2CDKCMGC3r7yAB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamideHuman3975
CDK2CDKCMGC3r83AA4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4234
CDK2CDKCMGC3r83AB4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4543
CDK2CDKCMGC3r8lAA(5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4186
CDK2CDKCMGC3r8lAB(5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4523
CDK2CDKCMGC3r8mAA1h-indazole-3-carbohydrazideHuman4111
CDK2CDKCMGC3r8mAB1h-indazole-3-carbohydrazideHuman4451
CDK2CDKCMGC3r8pAA(5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4232
CDK2CDKCMGC3r8pAB(5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4538
CDK2CDKCMGC3r8uAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman3926
CDK2CDKCMGC3r8uAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman3864
CDK2CDKCMGC3r8vAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3938
CDK2CDKCMGC3r8vAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman4191
CDK2CDKCMGC3r8zAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanoneHuman4137
CDK2CDKCMGC3r8zAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanoneHuman4140
CDK2CDKCMGC3r9dAA4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4562
CDK2CDKCMGC3r9dAB4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4565
CDK2CDKCMGC3r9hAA4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman3958
CDK2CDKCMGC3r9hAB4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4336
CDK2CDKCMGC3r9nAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3885
CDK2CDKCMGC3r9nAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3867
CDK2CDKCMGC3r9oA4-amino-n-(3,5-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4279
CDK2CDKCMGC3rahAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman4438
CDK2CDKCMGC3rahAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman4206
CDK2CDKCMGC3raiAA4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4441
CDK2CDKCMGC3raiAB4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4002
CDK2CDKCMGC3rakAA4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4574
CDK2CDKCMGC3rakAB4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4331
CDK2CDKCMGC3ralAA4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4017
CDK2CDKCMGC3ralAB4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3984
CDK2CDKCMGC3rjcAA{4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanoneHuman4032
CDK2CDKCMGC3rjcAB{4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanoneHuman4469
CDK2CDKCMGC3rk5A4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzoic acidHuman4160
CDK2CDKCMGC3rk7A4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzamideHuman4236
CDK2CDKCMGC3rk9AA[4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4158
CDK2CDKCMGC3rk9AB[4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4259
CDK2CDKCMGC3rkbAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4460
CDK2CDKCMGC3rkbAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4039
CDK2CDKCMGC3rm6AA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamideHuman4262
CDK2CDKCMGC3rm6AB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamideHuman4357
CDK2CDKCMGC3rm7AA2-[(4-hydroxybenzyl)amino]-5-nitrobenzamideHuman3893
CDK2CDKCMGC3rm7AB2-[(4-hydroxybenzyl)amino]-5-nitrobenzamideHuman4499
CDK2CDKCMGC3rmfAA4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3873
CDK2CDKCMGC3rmfAB4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4014
CDK2CDKCMGC3rniAA3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman3993
CDK2CDKCMGC3rniAB3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4420
CDK2CDKCMGC3royAA4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4131
CDK2CDKCMGC3royAB4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4239
CDK2CDKCMGC3rpoAA4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acidHuman3966
CDK2CDKCMGC3rpoAB4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acidHuman4098
CDK2CDKCMGC3rprAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanoneHuman4452
CDK2CDKCMGC3rprAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanoneHuman4241
CDK2CDKCMGC3rpvAA4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4348
CDK2CDKCMGC3rpvAB4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4372
CDK2CDKCMGC3rpyAA4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4261
CDK2CDKCMGC3rpyAB4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4519
CDK2CDKCMGC3rzbAA4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamideHuman4264
CDK2CDKCMGC3rzbAB4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamideHuman4395
CDK2CDKCMGC3s00AA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHuman4208
CDK2CDKCMGC3s00AB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHuman4248
CDK2CDKCMGC3s0oAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHuman3898
CDK2CDKCMGC3s0oAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHuman4123
CDK2CDKCMGC3s1hAA4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4068
CDK2CDKCMGC3s1hAB4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4226
CDK2CDKCMGC3s2pA(3s,4s)-1-{3-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-4-hydroxyphenyl}pyrrolidine-3,4-diolHuman4404
CDK2CDKCMGC3sqqAA4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4231
CDK2CDKCMGC3sqqAB4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3925
CDK2CDKCMGC3sw4AAn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHuman4076
CDK2CDKCMGC3sw4ABn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHuman4439
CDK2CDKCMGC3sw7AAn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHuman4198
CDK2CDKCMGC3sw7ABn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHuman4584
CDK2CDKCMGC3ti1AAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4201
CDK2CDKCMGC3ti1ABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4213
CDK2CDKCMGC3tiyAA2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHuman4413
CDK2CDKCMGC3tiyAB2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHuman4488
CDK2CDKCMGC3tizA1-{(e)-[(4-hydroxyphenyl)imino]methyl}naphthalen-2-olHuman4136
CDK2CDKCMGC3tnwAA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman4254
CDK2CDKCMGC3tnwAB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3948
CDK2CDKCMGC3tnwCA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3940
CDK2CDKCMGC3tnwCB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman4493
CDK2CDKCMGC3uliAA1-(aminomethyl)-n-(3-{[6-bromo-2-(4-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-7-yl]amino}propyl)cyclopropanecarboxamideHuman4115
CDK2CDKCMGC3unjA4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acidHuman4498
CDK2CDKCMGC3unkA4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman4374
CDK2CDKCMGC3wblAn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman3895
CDK2CDKCMGC4acmAA3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman4247
CDK2CDKCMGC4acmAB3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman3983
CDK2CDKCMGC4bckAA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4095
CDK2CDKCMGC4bckAB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman3960
CDK2CDKCMGC4bckAC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4433
CDK2CDKCMGC4bckAD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4563
CDK2CDKCMGC4bckCA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4268
CDK2CDKCMGC4bckCB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4506
CDK2CDKCMGC4bckCC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4029
CDK2CDKCMGC4bckCD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4080
CDK2CDKCMGC4bcmAA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4290
CDK2CDKCMGC4bcmAB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4203
CDK2CDKCMGC4bcmCA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4227
CDK2CDKCMGC4bcmCB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4124
CDK2CDKCMGC4bcnAA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4084
CDK2CDKCMGC4bcnAB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4298
CDK2CDKCMGC4bcnCA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4436
CDK2CDKCMGC4bcnCB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4150
CDK2CDKCMGC4bcoAA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman3988
CDK2CDKCMGC4bcoAB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4051
CDK2CDKCMGC4bcoCA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4333
CDK2CDKCMGC4bcoCB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4018
CDK2CDKCMGC4bcpAA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4552
CDK2CDKCMGC4bcpAB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4304
CDK2CDKCMGC4bcpCA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman3872
CDK2CDKCMGC4bcpCB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4501
CDK2CDKCMGC4bcqAA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4396
CDK2CDKCMGC4bcqAB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4415
CDK2CDKCMGC4bcqCA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman3996
CDK2CDKCMGC4bcqCB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4120
CDK2CDKCMGC4bghAA4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHuman4073
CDK2CDKCMGC4bghAB4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHuman4509
CDK2CDKCMGC4bzdAA6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHuman3865
CDK2CDKCMGC4bzdAB6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHuman4490
CDK2CDKCMGC4cfmAA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4207
CDK2CDKCMGC4cfmAB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman3986
CDK2CDKCMGC4cfmCA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4260
CDK2CDKCMGC4cfmCB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4005
CDK2CDKCMGC4cfnAA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4285
CDK2CDKCMGC4cfnAB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4437
CDK2CDKCMGC4cfnCA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4355
CDK2CDKCMGC4cfnCB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4567
CDK2CDKCMGC4cfuAA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman3905
CDK2CDKCMGC4cfuAB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman4308
CDK2CDKCMGC4cfuCA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman3967
CDK2CDKCMGC4cfuCB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman4539
CDK2CDKCMGC4cfvAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman4180
CDK2CDKCMGC4cfvAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman4328
CDK2CDKCMGC4cfvCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman3999
CDK2CDKCMGC4cfvCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman3979
CDK2CDKCMGC4cfwAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4280
CDK2CDKCMGC4cfwAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4557
CDK2CDKCMGC4cfwAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4141
CDK2CDKCMGC4cfwCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4549
CDK2CDKCMGC4cfwCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4508
CDK2CDKCMGC4cfwCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4102
CDK2CDKCMGC4cfxAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4485
CDK2CDKCMGC4cfxAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4086
CDK2CDKCMGC4cfxAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman3963
CDK2CDKCMGC4cfxCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4166
CDK2CDKCMGC4cfxCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4257
CDK2CDKCMGC4cfxCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4442
CDK2CDKCMGC4d1xA(4s)-2-(6-hydroxy-1,3-benzothiazol-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHuman4344
CDK2CDKCMGC4d1zA(4s)-2-(8-hydroxyquinolin-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHuman4486
CDK2CDKCMGC4ek3AA-Human3971
CDK2CDKCMGC4ek3AB-Human4202
CDK2CDKCMGC4ek4AA4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman4212
CDK2CDKCMGC4ek4AB4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman3957
CDK2CDKCMGC4ek4AC4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman4369
CDK2CDKCMGC4ek5AAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHuman4037
CDK2CDKCMGC4ek5ABn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHuman4145
CDK2CDKCMGC4ek6AAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHuman4359
CDK2CDKCMGC4ek6ABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHuman4056
CDK2CDKCMGC4ek8AA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amineHuman4079
CDK2CDKCMGC4ek8AB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amineHuman3871
CDK2CDKCMGC4eoiAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4307
CDK2CDKCMGC4eoiAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4342
CDK2CDKCMGC4eoiCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4522
CDK2CDKCMGC4eoiCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4011
CDK2CDKCMGC4eojAAadenosine-5'-triphosphateHuman4271
CDK2CDKCMGC4eojABadenosine-5'-triphosphateHuman4015
CDK2CDKCMGC4eojCAadenosine-5'-triphosphateHuman4041
CDK2CDKCMGC4eojCBadenosine-5'-triphosphateHuman4311
CDK2CDKCMGC4eokAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3913
CDK2CDKCMGC4eokCo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4385
CDK2CDKCMGC4eolAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4089
CDK2CDKCMGC4eolAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4270
CDK2CDKCMGC4eolCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4235
CDK2CDKCMGC4eolCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4521
CDK2CDKCMGC4eomAAadenosine-5'-triphosphateHuman4528
CDK2CDKCMGC4eomABadenosine-5'-triphosphateHuman4472
CDK2CDKCMGC4eomCAadenosine-5'-triphosphateHuman4481
CDK2CDKCMGC4eomCBadenosine-5'-triphosphateHuman4423
CDK2CDKCMGC4eonAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman3902
CDK2CDKCMGC4eonAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4326
CDK2CDKCMGC4eonCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4153
CDK2CDKCMGC4eonCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4192
CDK2CDKCMGC4eooAAadenosine-5'-triphosphateHuman4403
CDK2CDKCMGC4eooABadenosine-5'-triphosphateHuman4278
CDK2CDKCMGC4eooCAadenosine-5'-triphosphateHuman4188
CDK2CDKCMGC4eooCBadenosine-5'-triphosphateHuman4139
CDK2CDKCMGC4eopAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4258
CDK2CDKCMGC4eopAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4044
CDK2CDKCMGC4eopCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4061
CDK2CDKCMGC4eopCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4463
CDK2CDKCMGC4eoqAAadenosine-5'-triphosphateHuman4402
CDK2CDKCMGC4eoqABadenosine-5'-triphosphateHuman4230
CDK2CDKCMGC4eoqCAadenosine-5'-triphosphateHuman4004
CDK2CDKCMGC4eoqCBadenosine-5'-triphosphateHuman3912
CDK2CDKCMGC4eorAAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4205
CDK2CDKCMGC4eorABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3934
CDK2CDKCMGC4eorCAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4221
CDK2CDKCMGC4eorCBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4487
CDK2CDKCMGC4eosAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4340
CDK2CDKCMGC4eosAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4028
CDK2CDKCMGC4eosCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4008
CDK2CDKCMGC4eosCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4181
CDK2CDKCMGC4erwAstaurosporineHuman4370
CDK2CDKCMGC4ez3A4-[(e)-(6-hydroxy-2-oxo-1,2-dihydropyridin-3-yl)diazenyl]benzenesulfonamideHuman4551
CDK2CDKCMGC4ez7AstaurosporineHuman4240
CDK2CDKCMGC4fkgAA4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acidHuman4020
CDK2CDKCMGC4fkgAB4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acidHuman4559
CDK2CDKCMGC4fkiAAn-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamideHuman4430
CDK2CDKCMGC4fkiABn-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamideHuman4272
CDK2CDKCMGC4fkjAAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHuman4387
CDK2CDKCMGC4fkjABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHuman4164
CDK2CDKCMGC4fklAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4583
CDK2CDKCMGC4fklAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4134
CDK2CDKCMGC4fkoAA2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHuman4449
CDK2CDKCMGC4fkoAB2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHuman4534
CDK2CDKCMGC4fkpAA3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4035
CDK2CDKCMGC4fkpAB3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4313
CDK2CDKCMGC4fkpAC3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4468
CDK2CDKCMGC4fkqAA4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHuman3972
CDK2CDKCMGC4fkqAB4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHuman4026
CDK2CDKCMGC4fkrAA(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman4149
CDK2CDKCMGC4fkrAB(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman4535
CDK2CDKCMGC4fksAAn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4412
CDK2CDKCMGC4fksABn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4489
CDK2CDKCMGC4fksACn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4315
CDK2CDKCMGC4fktAAn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4548
CDK2CDKCMGC4fktABn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4322
CDK2CDKCMGC4fkuAA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman3863
CDK2CDKCMGC4fkuAB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4573
CDK2CDKCMGC4fkvAA(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHuman4299
CDK2CDKCMGC4fkvAB(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHuman3939
CDK2CDKCMGC4fkwAA2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHuman4252
CDK2CDKCMGC4fkwAB2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHuman4277
CDK2CDKCMGC4fx3AA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4518
CDK2CDKCMGC4fx3AB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman3931
CDK2CDKCMGC4fx3CA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4349
CDK2CDKCMGC4fx3CB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4495
CDK2CDKCMGC4gcjAA4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4138
CDK2CDKCMGC4gcjAB4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4362
CDK2CDKCMGC4i3zAadenosine-5'-diphosphateHuman4148
CDK2CDKCMGC4i3zCadenosine-5'-diphosphateHuman3961
CDK2CDKCMGC4ii5AAadenosine-5'-diphosphateHuman3930
CDK2CDKCMGC4ii5ABadenosine-5'-diphosphateHuman4456
CDK2CDKCMGC4ii5CAadenosine-5'-diphosphateHuman4530
CDK2CDKCMGC4ii5CBadenosine-5'-diphosphateHuman4462
CDK2CDKCMGC4kd1AA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman4585
CDK2CDKCMGC4kd1AB3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman4525
CDK2CDKCMGC4lynA(2s)-n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)-2-phenylpropanamideHuman4550
CDK2CDKCMGC4nj3AA6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman4075
CDK2CDKCMGC4nj3AB6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman4366
CDK2CDKCMGC4rj3AA1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4244
CDK2CDKCMGC4rj3AB1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4127
CDK2CDKCMGC5a14AA1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHuman3977
CDK2CDKCMGC5a14AB1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHuman3901
CDK2CDKCMGC5andA2-imidazol-1-yl-1h-benzimidazoleHuman6543
CDK2CDKCMGC5aneA6-methoxy-9h-purineHuman6542
CDK2CDKCMGC5angA7-hydroxy-4-(morpholinomethyl)chromen-2-oneHuman6540
CDK2CDKCMGC5aniA6-chloro-9h-purineHuman6539
CDK2CDKCMGC5anjAn-(9h-purin-6-yl)thiophene-2-carboxamideHuman6541
CDK2CDKCMGC5ankA2,4,6-trioxo-1-phenyl-hexahydropyrimidine-5-carboxamideHuman6538
CDK2CDKCMGC5anoA-Human6537
CDK2CDKCMGC5cyiAA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6052
CDK2CDKCMGC5cyiAB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6054
CDK2CDKCMGC5cyiCA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6055
CDK2CDKCMGC5cyiCB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6053
CDK2CDKCMGC5d1jAn-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamideHuman4058
CDK2CDKCMGC5fp5A4-fluorobenzoic acidHuman6285
CDK2CDKCMGC5fp6AA3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHuman6302
CDK2CDKCMGC5fp6AB3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHuman6301
CDK2CDKCMGC5ievAAroniciclibHuman6567
CDK2CDKCMGC5ievABroniciclibHuman6570
CDK2CDKCMGC5iexAA(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHuman6565
CDK2CDKCMGC5iexAB(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHuman6572
CDK2CDKCMGC5ieyAA4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHuman6566
CDK2CDKCMGC5ieyAB4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHuman6573
CDK2CDKCMGC5if1AA-Human6568
CDK2CDKCMGC5if1AB-Human6569
CDK2CDKCMGC5if1CA-Human6564
CDK2CDKCMGC5if1CB-Human6571
CDK2CDKCMGC5jq5A(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman7416
CDK2CDKCMGC5jq8A(3s,4s)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman7417
CDK2CDKCMGC5k4jAA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6751
CDK2CDKCMGC5k4jAB1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6750
CDK2CDKCMGC5l2wA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman6993
CDK2CDKCMGC5lmkAA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7399
CDK2CDKCMGC5lmkAB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7398
CDK2CDKCMGC5lmkCA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7396
CDK2CDKCMGC5lmkCB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7397
CDK2CDKCMGC5mhqAA(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHuman9409
CDK2CDKCMGC5mhqAB(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHuman9408
CDK2CDKCMGC5nevA4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHuman8020
CDK2CDKCMGC5nevC4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHuman8019
CDK2CDKCMGC5oo0AA-Human9744
CDK2CDKCMGC5oo0AC-Human9745
CDK2CDKCMGC5oo1A~{n}-(4-pyrimidin-2-ylphenyl)propanamideHuman10566
CDK2CDKCMGC5oo3AA1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHuman10569
CDK2CDKCMGC5oo3AB1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHuman10568
CDK2CDKCMGC5osjAA-Human9743
CDK2CDKCMGC5osjAB-Human9742
CDK2CDKCMGC5osmAAmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHuman9741
CDK2CDKCMGC5osmABmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHuman9740
CDK2CDKCMGC5uq1A-Human8220
CDK2CDKCMGC5uq1C-Human8223
CDK2CDKCMGC5uq2A-Human8221
CDK2CDKCMGC5uq3A-Human8222
CDK2CDKCMGC6athAA-Human10567
CDK2CDKCMGC6athAB-Human10570
CDK2CDKCMGC6gubA2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10764
CDK2CDKCMGC6gubC2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10763
CDK2CDKCMGC6gucA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman10767
CDK2CDKCMGC6gucC(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman10766
CDK2CDKCMGC6gueA4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10771
CDK2CDKCMGC6gueC4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10772
CDK2CDKCMGC6gufAn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman10770
CDK2CDKCMGC6gufCn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman10762
CDK2CDKCMGC6guhAA4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10765
CDK2CDKCMGC6guhAB4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10769
CDK2CDKCMGC6gukAA~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10773
CDK2CDKCMGC6gukAB~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10768
CDK2CDKCMGC6gvaAA5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman11206
CDK2CDKCMGC6gvaAB5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman11204
CDK2CDKCMGC6inlA2,2'-{[6-{[(4-methoxyphenyl)methyl]amino}-9-(propan-2-yl)-9h-purin-2-yl]azanediyl}di(ethan-1-ol)Human11794
CDK2CDKCMGC6jgmA4-{[6-(cyclohexylmethoxy)-7h-purin-2-yl]amino}-n,n-diethylbenzamideHuman12008
CDK2CDKCMGC6oqiA5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4s)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12648
CDK2CDKCMGC6p3wAA-Human11515
CDK2CDKCMGC6p3wAB-Human11517
CDK2CDKCMGC6p3wCA-Human11514
CDK2CDKCMGC6p3wCB-Human11516
CDK2CDKCMGC6q3bAA4-iodopyrazoleHuman11177
CDK2CDKCMGC6q3bAB4-iodopyrazoleHuman11208
CDK2CDKCMGC6q3cAA4-bromo-1h-pyrazoleHuman11191
CDK2CDKCMGC6q3cAB4-bromo-1h-pyrazoleHuman11203
CDK2CDKCMGC6q3cAC-Human11178
CDK2CDKCMGC6q3fAA-Human11181
CDK2CDKCMGC6q3fAB-Human11187
CDK2CDKCMGC6q48AA4-iodanyl-3~{h}-pyridin-2-oneHuman11192
CDK2CDKCMGC6q48AB4-iodanyl-3~{h}-pyridin-2-oneHuman11218
CDK2CDKCMGC6q48AC4-iodanyl-3~{h}-pyridin-2-oneHuman11196
CDK2CDKCMGC6q49AA-Human11185
CDK2CDKCMGC6q49AB-Human11220
CDK2CDKCMGC6q49AC-Human11193
CDK2CDKCMGC6q4aAA5-iodanylpyrimidineHuman11195
CDK2CDKCMGC6q4aAB5-iodanylpyrimidineHuman11200
CDK2CDKCMGC6q4aAC5-iodanylpyrimidineHuman11216
CDK2CDKCMGC6q4bAA5-bromanylpyrimidineHuman11198
CDK2CDKCMGC6q4bAB5-bromanylpyrimidineHuman11210
CDK2CDKCMGC6q4bAC5-bromanylpyrimidineHuman11180
CDK2CDKCMGC6q4cAA4-bromanyl-1,8-naphthyridineHuman11182
CDK2CDKCMGC6q4cAB4-bromanyl-1,8-naphthyridineHuman11207
CDK2CDKCMGC6q4cAC4-bromanyl-1,8-naphthyridineHuman11201
CDK2CDKCMGC6q4dAA2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11184
CDK2CDKCMGC6q4dAB2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11215
CDK2CDKCMGC6q4dAC2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11188
CDK2CDKCMGC6q4eAA6-iodanyl-7~{h}-purin-2-amineHuman11199
CDK2CDKCMGC6q4eAB6-iodanyl-7~{h}-purin-2-amineHuman11205
CDK2CDKCMGC6q4eAC6-iodanyl-7~{h}-purin-2-amineHuman11219
CDK2CDKCMGC6q4fAApyridine-2,6-diamineHuman11202
CDK2CDKCMGC6q4fABpyridine-2,6-diamineHuman11211
CDK2CDKCMGC6q4fACpyridine-2,6-diamineHuman11212
CDK2CDKCMGC6q4gAA2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHuman11214
CDK2CDKCMGC6q4gAB2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHuman11217
CDK2CDKCMGC6q4hAA2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHuman11194
CDK2CDKCMGC6q4hAB2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHuman11190
CDK2CDKCMGC6q4iAA2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHuman11183
CDK2CDKCMGC6q4iAB2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHuman11197
CDK2CDKCMGC6q4jAA2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHuman11209
CDK2CDKCMGC6q4jAB2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHuman11213
CDK2CDKCMGC6q4kAA-Human11179
CDK2CDKCMGC6q4kAB-Human11186
CDK2CDKCMGC6q4kAC-Human11189
CDK2CDKCMGC6rijAA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12623
CDK2CDKCMGC6rijAB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12624
CDK2CDKCMGC6rijCA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12625
CDK2CDKCMGC6rijCB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12622
CDK2CDKCMGC6sg4AA-Human13246
CDK2CDKCMGC6sg4AB-Human13247
CDK2CDKCMGC6sg4CA-Human13248
CDK2CDKCMGC6sg4CB-Human13245
CDK2CDKCMGC6yl1AAmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12497
CDK2CDKCMGC6yl1ABmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12496
CDK2CDKCMGC6yl6AA-Human12498
CDK2CDKCMGC6yl6AB-Human12495
CDK2CDKCMGC6ylkAAmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12499
CDK2CDKCMGC6ylkABmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12494
CDK2CDKCMGC7ackAA8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13451
CDK2CDKCMGC7ackAB8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13453
CDK2CDKCMGC7ackCA8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13450
CDK2CDKCMGC7ackCB8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13452
CDK2CDKCMGC7b5lL-Human13266
CDK2CDKCMGC7b5rL-Human13265
CDK2CDKCMGC7b7sAA7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxideHuman13833
CDK2CDKCMGC7b7sAB7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxideHuman13834
CDK2CDKCMGC7e34A-Human13497
CDK2CDKCMGC7kjsA6-(difluoromethyl)-8-[(1r,2r)-2-hydroxy-2-methylcyclopentyl]-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman13740
CDK2CDKCMGC7m2fAA[(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acidHuman13797
CDK2CDKCMGC7m2fAB[(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acidHuman13796
CDK2CDKCMGC7mkxA2-[(5-bromo-2-{4-[(cyanomethyl)sulfamoyl]anilino}pyrimidin-4-yl)amino]-6-fluorobenzamideHuman14490
CDK2CDKCMGC7nvqAstaurosporineHuman13627
CDK2CDKCMGC7qhlAA5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidineHuman14275
CDK2CDKCMGC7qhlAB5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidineHuman14276
CDK2CDKCMGC7ra5AA4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman13960
CDK2CDKCMGC7ra5AB4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman13959
CDK2CDKCMGC7rweA5-nitro-2-[(3-phenylpropyl)amino]benzoic acidHuman14345
CDK2CDKCMGC7rwfA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHuman14344
CDK2CDKCMGC7rxoAA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acidHuman14352
CDK2CDKCMGC7rxoAB2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acidHuman14351
CDK2CDKCMGC7s4tAA2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHuman14374
CDK2CDKCMGC7s4tAB2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHuman14373
CDK2CDKCMGC7s7aAA2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14427
CDK2CDKCMGC7s7aAB2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14426
CDK2CDKCMGC7s84AA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14424
CDK2CDKCMGC7s84AB2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14432
CDK2CDKCMGC7s85A2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethoxy)benzoic acidHuman14425
CDK2CDKCMGC7s9xAA2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acidHuman14430
CDK2CDKCMGC7s9xAB2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acidHuman14431
CDK2CDKCMGC7sa0AA2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acidHuman14428
CDK2CDKCMGC7sa0AB2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acidHuman14429
CDK2CDKCMGC7ug1AA8-(4-chloroanilino)naphthalene-1-sulfonic acidHuman14700
CDK2CDKCMGC7ug1AB8-(4-chloroanilino)naphthalene-1-sulfonic acidHuman14701
CDK2CDKCMGC7uxiAA-Human14571
CDK2CDKCMGC7uxiAB-Human14572
CDK2CDKCMGC7uxkA-Human14570
CDK2CDKCMGC7vduAA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14136
CDK2CDKCMGC7vduAB[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14137
CDK2CDKCMGC7zpcAA~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamideHuman14606
CDK2CDKCMGC7zpcAB~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamideHuman14607
CDK2CDKCMGC8b54AA~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman14681
CDK2CDKCMGC8b54AB~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman14680
CDK2CDKCMGC8byaA-Human14814
CDK2CDKCMGC8bzoA-Human14815
CDK2CDKCMGC8curAA6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman14693
CDK2CDKCMGC8curAB6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman14692
CDK2CDKCMGC8erdAA(2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanoneHuman14949
CDK2CDKCMGC8erdAB(2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanoneHuman14951
CDK2CDKCMGC8ernAAn,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamideHuman14948
CDK2CDKCMGC8ernABn,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamideHuman14950
CDK2CDKCMGC8fowAA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman14759
CDK2CDKCMGC8fowAB3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman14760
CDK2CDKCMGC8fp0AAr-roscovitineHuman14758
CDK2CDKCMGC8fp0ABr-roscovitineHuman14756
CDK2CDKCMGC8fp5AAadenosine-5'-triphosphateHuman14761
CDK2CDKCMGC8fp5ABadenosine-5'-triphosphateHuman14757
CDK2CDKCMGC8h6pA(7s,10r)-11-oxa-2,4,5,13,17,23-hexaazatetracyclo[17.3.1.1~3,6~.1~7,10~]pentacosa-1(23),3(25),5,19,21-pentaene-12,18-dioneHuman14625
CDK2CDKCMGC8h6tA(1r,3s)-3-{3-[(pyridin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl propan-2-ylcarbamateHuman14626
CDK2CDKCMGC8oy2A(1s,2s,11as)-1-methoxy-1,4,7,10-tetramethyl-2,9-bis(oxidanyl)-2,11a-dihydrobenzo[b][1,4]benzodioxepine-3,6-dioneHuman15078
CDK4CDKCMGC2w96BA-Human3390
CDK4CDKCMGC2w96BB-Human3389
CDK4CDKCMGC2w99B-Human3385
CDK4CDKCMGC2w9fB-Human3386
CDK4CDKCMGC2w9zBA-Human3388
CDK4CDKCMGC2w9zBB-Human3383
CDK4CDKCMGC3g33A-Human3387
CDK4CDKCMGC3g33C-Human3384
CDK4CDKCMGC5fwkK-Human6747
CDK4CDKCMGC5fwlK-Human6748
CDK4CDKCMGC5fwmK-Human6749
CDK4CDKCMGC5fwpK-Human7132
CDK4CDKCMGC6p8eB-Human11891
CDK4CDKCMGC6p8fB-Human11892
CDK4CDKCMGC6p8gB-Human11893
CDK4CDKCMGC6p8hB-Human11894
CDK4CDKCMGC7sj3An-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman14485
CDK5CDKCMGC1h4lA-Human2788
CDK5CDKCMGC1h4lB-Human2779
CDK5CDKCMGC1ungA6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2792
CDK5CDKCMGC1ungB6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2789
CDK5CDKCMGC1unhA(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2780
CDK5CDKCMGC1unhB(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2787
CDK5CDKCMGC1unlAr-roscovitineHuman2785
CDK5CDKCMGC1unlB-Human2790
CDK5CDKCMGC3o0gA-Human2782
CDK5CDKCMGC3o0gB{4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanoneHuman2783
CDK5CDKCMGC4au8AA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2784
CDK5CDKCMGC4au8AB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2786
CDK5CDKCMGC4au8BA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2791
CDK5CDKCMGC4au8BB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2781
CDK5CDKCMGC7vdpA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14145
CDK5CDKCMGC7vdqA2-[[7-[[2-fluoranyl-4-[3-(hydroxymethyl)pyrazol-1-yl]phenyl]amino]-1,6-naphthyridin-2-yl]-(1-methylpiperidin-4-yl)amino]ethanoic acidHuman14144
CDK5CDKCMGC7vdrA(1r)-1-[7-[(2-fluoranyl-4-pyrazol-1-yl-phenyl)amino]-1,6-naphthyridin-2-yl]-1-(1-methylpiperidin-4-yl)ethanolHuman14146
CDK5CDKCMGC7vdsAA5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHuman14148
CDK5CDKCMGC7vdsAB5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHuman14147
CDK6CDKCMGC1bi7A-Human2798
CDK6CDKCMGC1bi8A-Human2796
CDK6CDKCMGC1bi8C-Human2799
CDK6CDKCMGC1blxA-Human2802
CDK6CDKCMGC1g3nA-Human2806
CDK6CDKCMGC1g3nE-Human2805
CDK6CDKCMGC1jowB-Human2793
CDK6CDKCMGC1xo2B3,7,3',4'-tetrahydroxyflavoneHuman2794
CDK6CDKCMGC2eufB6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman2804
CDK6CDKCMGC2f2cB(2s)-2-({6-[(3-amino-5-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHuman2795
CDK6CDKCMGC3nupA4-[3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(1-methylpiperidin-4-yl)pyrimidin-2-amineHuman2797
CDK6CDKCMGC3nuxA4-[5-chloro-3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineHuman2807
CDK6CDKCMGC4auaA1h-benzimidazol-2-yl(1h-pyrrol-2-yl)methanoneHuman2801
CDK6CDKCMGC4ez5A{5-[4-(dimethylamino)piperidin-1-yl]-1h-imidazo[4,5-b]pyridin-2-yl}[2-(isoquinolin-4-yl)pyridin-4-yl]methanoneHuman2800
CDK6CDKCMGC4tthB9-cyclopentyl-n-(5-piperazin-1-ylpyridin-2-yl)pyrido[4,5]pyrrolo[1,2-d]pyrimidin-2-amineHuman2803
CDK6CDKCMGC5l2iA6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6991
CDK6CDKCMGC5l2sAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman6990
CDK6CDKCMGC5l2tA7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman6992
CDK6CDKCMGC6oqlA5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12647
CDK6CDKCMGC6oqoAn-[5-(6-ethyl-2,6-diazaspiro[3.3]heptan-2-yl)pyridin-2-yl]-5-fluoro-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12646
CDK6CDKCMGC8i0mA2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman15164
CDK7CDKCMGC1ua2Aadenosine-5'-triphosphateHuman540
CDK7CDKCMGC1ua2Badenosine-5'-triphosphateHuman541
CDK7CDKCMGC1ua2Cadenosine-5'-triphosphateHuman542
CDK7CDKCMGC1ua2Dadenosine-5'-triphosphateHuman543
CDK7CDKCMGC6o9l8-Human11055
CDK7CDKCMGC6xbzJphosphothiophosphoric acid-adenylate esterHuman12773
CDK7CDKCMGC6xd3Jn-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamideHuman12772
CDK7CDKCMGC7b5oJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13278
CDK7CDKCMGC7b5oJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13279
CDK7CDKCMGC7b5qJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13277
CDK7CDKCMGC7b5qJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13280
CDK7CDKCMGC7nvr8-Human13543
CDK7CDKCMGC8bvwI-Human14733
CDK7CDKCMGC8byqI-Human14732
CDK7CDKCMGC8p4zAA2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHuman14796
CDK7CDKCMGC8p4zAB2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHuman14797
CDK8CDKCMGC3rgfAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3841
CDK8CDKCMGC3rgfAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3846
CDK8CDKCMGC4crlAcortistatin aHuman6096
CDK8CDKCMGC4f6sA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman3848
CDK8CDKCMGC4f6uAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]ureaHuman3849
CDK8CDKCMGC4f6uAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]ureaHuman3844
CDK8CDKCMGC4f6wAn-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-4-[2-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)ethyl]piperazine-1-carboxamideHuman3845
CDK8CDKCMGC4f70A1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[2-(morpholin-4-yl)ethyl]ureaHuman3852
CDK8CDKCMGC4f7jAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)ureaHuman3842
CDK8CDKCMGC4f7jAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)ureaHuman3843
CDK8CDKCMGC4f7lAtert-butyl [3-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)propyl]carbamateHuman3840
CDK8CDKCMGC4f7nA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(5-hydroxypentyl)ureaHuman3847
CDK8CDKCMGC4f7sAAn-(2-phenylethyl)quinazolin-4-amineHuman3850
CDK8CDKCMGC4f7sABn-(2-phenylethyl)quinazolin-4-amineHuman3853
CDK8CDKCMGC4g6lA-Human3851
CDK8CDKCMGC5bnjA8-{3-chloro-5-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]pyridin-4-yl}-2,8-diazaspiro[4.5]decan-1-oneHuman6152
CDK8CDKCMGC5ceiAA4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamideHuman6404
CDK8CDKCMGC5ceiAB4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamideHuman6403
CDK8CDKCMGC5fgkAA8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6391
CDK8CDKCMGC5fgkAB8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6388
CDK8CDKCMGC5hbeAA8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-oneHuman6389
CDK8CDKCMGC5hbeAB8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-oneHuman6386
CDK8CDKCMGC5hbhA5-[5-chloranyl-4-[1-(2-methoxyethyl)-1,8-diazaspiro[4.5]decan-8-yl]pyridin-3-yl]-1-methyl-3~{h}-2,1-benzothiazole 2,2-dioxideHuman6387
CDK8CDKCMGC5hbjAA8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6390
CDK8CDKCMGC5hbjAB8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6385
CDK8CDKCMGC5hnbAA[6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanoneHuman6562
CDK8CDKCMGC5hnbAB[6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanoneHuman6563
CDK8CDKCMGC5hvyAAn-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}ureaHuman6553
CDK8CDKCMGC5hvyABn-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}ureaHuman6552
CDK8CDKCMGC5i5zAn-methyl-8-(1-methyl-2,2-dioxo-2,3-dihydro-1h-2lambda~6~,1-benzothiazol-5-yl)-1,6-naphthyridine-2-carboxamideHuman6536
CDK8CDKCMGC5icpAA[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanoneHuman7318
CDK8CDKCMGC5icpAB[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanoneHuman7321
CDK8CDKCMGC5idnAA[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanoneHuman7322
CDK8CDKCMGC5idnAB[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanoneHuman7319
CDK8CDKCMGC5idpAA(3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanoneHuman7317
CDK8CDKCMGC5idpAB(3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanoneHuman7320
CDK8CDKCMGC5xqxAn-methyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHuman8313
CDK8CDKCMGC5xs2AA3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHuman8315
CDK8CDKCMGC5xs2AB3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHuman8314
CDK8CDKCMGC6qtgA2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]-~{n},~{n}-dimethyl-ethanamideHuman12094
CDK8CDKCMGC6qtjA~{n},~{n}-dimethyl-2-[4-[4-(2,6-naphthyridin-4-yl)phenyl]pyrazol-1-yl]ethanamideHuman12093
CDK8CDKCMGC6r3sAA6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman12140
CDK8CDKCMGC6r3sAB6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman12141
CDK8CDKCMGC6t41A~{n}-[(4-chlorophenyl)methyl]quinazolin-4-amineHuman11908
CDK8CDKCMGC6tpaA1-[4-chloranyl-3-(trifluoromethyl)phenyl]-3-(5-oxidanylidene-6-pyridin-4-yl-pyrido[2,3-b][1,5]benzoxazepin-9-yl)ureaHuman13160
CDK8CDKCMGC6y0aAA6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman13306
CDK8CDKCMGC6y0aAB6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman13305
CDK9CDKCMGC3blhA-Human2251
CDK9CDKCMGC3blqAadenosine-5'-triphosphateHuman2248
CDK9CDKCMGC3blrA2-(2-chloro-phenyl)-5,7-dihydroxy-8-(3-hydroxy-1-methyl-piperidin-4-yl)-4h-benzopyran-4-oneHuman2236
CDK9CDKCMGC3lq5A(2s)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman2253
CDK9CDKCMGC3mi9A-Human2239
CDK9CDKCMGC3miaAphosphoaminophosphonic acid-adenylate esterHuman2242
CDK9CDKCMGC3my1A5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman2249
CDK9CDKCMGC3tn8A4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman2240
CDK9CDKCMGC3tnhA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman2232
CDK9CDKCMGC3tniA-Human2250
CDK9CDKCMGC4bcfA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman2257
CDK9CDKCMGC4bcgA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman2255
CDK9CDKCMGC4bchA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman2246
CDK9CDKCMGC4bciA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman2243
CDK9CDKCMGC4bcjA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman2247
CDK9CDKCMGC4ec8A-Human2244
CDK9CDKCMGC4ec9A-Human2234
CDK9CDKCMGC4imyAAadenosine monophosphateHuman2238
CDK9CDKCMGC4imyABadenosine monophosphateHuman2252
CDK9CDKCMGC4imyCAadenosine monophosphateHuman2237
CDK9CDKCMGC4imyCBadenosine monophosphateHuman2245
CDK9CDKCMGC4imyEAadenosine monophosphateHuman2258
CDK9CDKCMGC4imyEBadenosine monophosphateHuman2256
CDK9CDKCMGC4ogrAadenosineHuman2254
CDK9CDKCMGC4ogrEadenosineHuman2235
CDK9CDKCMGC4ogrIadenosineHuman2241
CDK9CDKCMGC4or5A-Human2233
CDK9CDKCMGC4or5F-Human2231
CDK9CDKCMGC5l1zA-Human7121
CDK9CDKCMGC6cytA-Human10797
CDK9CDKCMGC6gzhA[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHuman10427
CDK9CDKCMGC6w9eAA(4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13859
CDK9CDKCMGC6w9eAB(4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13858
CDK9CDKCMGC6w9eAC(4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13861
CDK9CDKCMGC6w9eAD(4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13860
CDK9CDKCMGC6z45A(1~{s},3~{r})-3-acetamido-~{n}-[5-chloranyl-4-(5,5-dimethyl-4,6-dihydropyrrolo[1,2-b]pyrazol-3-yl)pyridin-2-yl]cyclohexane-1-carboxamideHuman13115
CDK9CDKCMGC7nwkAn-((1r,3r)-3-(7-(4-fluoro-2-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-2-yl)cyclopentyl)acetamideHuman13951
CDK9CDKCMGC8i0lA2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman15170
CDK9CDKCMGC8k5rA(1s,3s)-n3-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamineHuman15081
CDKL1CDKLCMGC4aguAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman761
CDKL1CDKLCMGC4aguBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman760
CDKL1CDKLCMGC4aguCn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman762
CDKL2CDKLCMGC4aaaAA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman964
CDKL2CDKLCMGC4aaaAB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman962
CDKL2CDKLCMGC4bbmA4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diolHuman963
CDKL2CDKLCMGC4bbmB4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diolHuman965
CDKL3CDKLCMGC3zduA[4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4677
CDKL5CDKLCMGC4bgqAA[4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1425
CDKL5CDKLCMGC4bgqAB[4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1426
CDKL5CDKLCMGC8cieA4-[[3,5-bis(fluoranyl)phenyl]carbonylamino]-~{n}-piperidin-4-yl-1~{h}-pyrazole-3-carboxamideHuman14778
CHEK1 (CHK1)CAMKLCAMK1ia8A-Human1656
CHEK1 (CHK1)CAMKLCAMK1nvqA7-hydroxystaurosporineHuman1642
CHEK1 (CHK1)CAMKLCAMK1nvrAstaurosporineHuman1585
CHEK1 (CHK1)CAMKLCAMK1nvsArel-(9r,12s)-9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2h)-dioneHuman1591
CHEK1 (CHK1)CAMKLCAMK1zltA(4z)-4-(2-amino-5-oxo-3,5-dihydro-4h-imidazol-4-ylidene)-2,3-dichloro-4,5,6,7-tetrahydropyrrolo[2,3-c]azepin-8(1h)-oneHuman1596
CHEK1 (CHK1)CAMKLCAMK1zysAn-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamideHuman1655
CHEK1 (CHK1)CAMKLCAMK2aypA(3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-oneHuman1682
CHEK1 (CHK1)CAMKLCAMK2br1AA2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanolHuman1677
CHEK1 (CHK1)CAMKLCAMK2br1AB2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanolHuman1571
CHEK1 (CHK1)CAMKLCAMK2brbA2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanolHuman1582
CHEK1 (CHK1)CAMKLCAMK2brgA(5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-aceticHuman1589
CHEK1 (CHK1)CAMKLCAMK2brhAAn-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycineHuman1694
CHEK1 (CHK1)CAMKLCAMK2brhABn-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycineHuman1654
CHEK1 (CHK1)CAMKLCAMK2brmAA3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-oneHuman1621
CHEK1 (CHK1)CAMKLCAMK2brmAB3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-oneHuman1643
CHEK1 (CHK1)CAMKLCAMK2brnA(2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-olHuman1631
CHEK1 (CHK1)CAMKLCAMK2broA(2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diolHuman1686
CHEK1 (CHK1)CAMKLCAMK2c3jAdebromohymenialdisineHuman1551
CHEK1 (CHK1)CAMKLCAMK2c3kA4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenolHuman1674
CHEK1 (CHK1)CAMKLCAMK2c3lA3-(1h-benzimidazol-2-yl)-1h-indazoleHuman1612
CHEK1 (CHK1)CAMKLCAMK2cguA2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acidHuman1697
CHEK1 (CHK1)CAMKLCAMK2cgvA(2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-olHuman1545
CHEK1 (CHK1)CAMKLCAMK2cgwA4,4'-(1-propyl-1h-1,2,4-triazole-3,5-diyl)bis(2,5-dihydro-1,2,5-oxadiazol-3-amine)Human1683
CHEK1 (CHK1)CAMKLCAMK2cgxA2-[(6-amino-7h-purin-8-yl)thio]acetamideHuman1595
CHEK1 (CHK1)CAMKLCAMK2e9nA3-(4'-hydroxybiphenyl-4-yl)-n-(4-hydroxycyclohexyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamideHuman1690
CHEK1 (CHK1)CAMKLCAMK2e9oA4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHuman1667
CHEK1 (CHK1)CAMKLCAMK2e9pA1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}ureaHuman1618
CHEK1 (CHK1)CAMKLCAMK2e9uA18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-oneHuman1584
CHEK1 (CHK1)CAMKLCAMK2e9vA18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrileHuman1574
CHEK1 (CHK1)CAMKLCAMK2e9vB18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrileHuman1638
CHEK1 (CHK1)CAMKLCAMK2gdoA4-[(3s)-1-azabicyclo[2.2.2]oct-3-ylamino]-3-(1h-benzimidazol-2-yl)-6-chloroquinolin-2(1h)-oneHuman1606
CHEK1 (CHK1)CAMKLCAMK2ghgA5-{5-[(s)-2-amino-3-(1h-indol-3-yl)-propoxyl]-pyridin-3-yl}-3-[1-(1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman1581
CHEK1 (CHK1)CAMKLCAMK2hogA(5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanolHuman1653
CHEK1 (CHK1)CAMKLCAMK2hxlA3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrileHuman1552
CHEK1 (CHK1)CAMKLCAMK2hxqA3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-oneHuman1587
CHEK1 (CHK1)CAMKLCAMK2hy0A3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-pyrazol-4-yl)quinolin-2(1h)-oneHuman1555
CHEK1 (CHK1)CAMKLCAMK2qhmA(3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylateHuman1669
CHEK1 (CHK1)CAMKLCAMK2qhnA5-ethyl-3-methyl-1,5-dihydro-4h-pyrazolo[4,3-c]quinolin-4-oneHuman1675
CHEK1 (CHK1)CAMKLCAMK2r0uA6-(3-aminopropyl)-4-(3-hydroxyphenyl)-9-(1h-pyrazol-4-yl)benzo[h]isoquinolin-1(2h)-oneHuman1632
CHEK1 (CHK1)CAMKLCAMK2wmqAn-(4-oxo-5,6,7,8-tetrahydro-4h-[1,3]thiazolo[5,4-c]azepin-2-yl)acetamideHuman1647
CHEK1 (CHK1)CAMKLCAMK2wmrAA5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-oneHuman1609
CHEK1 (CHK1)CAMKLCAMK2wmrAB5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-oneHuman1604
CHEK1 (CHK1)CAMKLCAMK2wmsA[4-amino-2-(tert-butylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman1657
CHEK1 (CHK1)CAMKLCAMK2wmtAA2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-olHuman1576
CHEK1 (CHK1)CAMKLCAMK2wmtAB2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-olHuman1685
CHEK1 (CHK1)CAMKLCAMK2wmuAA6-morpholin-4-yl-9h-purineHuman1662
CHEK1 (CHK1)CAMKLCAMK2wmuAB6-morpholin-4-yl-9h-purineHuman1578
CHEK1 (CHK1)CAMKLCAMK2wmvA1-[(2s)-4-(7h-purin-6-yl)morpholin-2-yl]methanamineHuman1562
CHEK1 (CHK1)CAMKLCAMK2wmwA1-[(2s)-4-(5-bromo-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamineHuman1594
CHEK1 (CHK1)CAMKLCAMK2wmxA1-[(2s)-4-(5-phenyl-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamineHuman1636
CHEK1 (CHK1)CAMKLCAMK2x8dAA5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1673
CHEK1 (CHK1)CAMKLCAMK2x8dAB5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1620
CHEK1 (CHK1)CAMKLCAMK2x8eA5-methyl-8-pyridin-4-yl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1548
CHEK1 (CHK1)CAMKLCAMK2x8iAA7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1699
CHEK1 (CHK1)CAMKLCAMK2x8iAB7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1558
CHEK1 (CHK1)CAMKLCAMK2xeyA3-(1h-indol-3-yl)-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazineHuman1668
CHEK1 (CHK1)CAMKLCAMK2xezA6-(1h-pyrazol-3-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazineHuman1580
CHEK1 (CHK1)CAMKLCAMK2xf0A3-phenyl-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazineHuman1534
CHEK1 (CHK1)CAMKLCAMK2ydiAA5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamideHuman1684
CHEK1 (CHK1)CAMKLCAMK2ydiAB5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamideHuman1579
CHEK1 (CHK1)CAMKLCAMK2ydjA5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman1649
CHEK1 (CHK1)CAMKLCAMK2ydjB5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman1687
CHEK1 (CHK1)CAMKLCAMK2ydkA2-(carbamoylamino)-5-phenyl-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamideHuman1646
CHEK1 (CHK1)CAMKLCAMK2yerAA5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-oneHuman1611
CHEK1 (CHK1)CAMKLCAMK2yerAB5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-oneHuman1583
CHEK1 (CHK1)CAMKLCAMK2yexAA5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1651
CHEK1 (CHK1)CAMKLCAMK2yexAB5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1567
CHEK1 (CHK1)CAMKLCAMK2ym3AAethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1644
CHEK1 (CHK1)CAMKLCAMK2ym3ABethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1543
CHEK1 (CHK1)CAMKLCAMK2ym4AAethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1572
CHEK1 (CHK1)CAMKLCAMK2ym4ABethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1560
CHEK1 (CHK1)CAMKLCAMK2ym5A(3-{4-[(2s)-2-(aminomethyl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}phenyl)methanolHuman1627
CHEK1 (CHK1)CAMKLCAMK2ym6AA1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamineHuman1563
CHEK1 (CHK1)CAMKLCAMK2ym6AB1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamineHuman1559
CHEK1 (CHK1)CAMKLCAMK2ym7AA5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrileHuman1650
CHEK1 (CHK1)CAMKLCAMK2ym7AB5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrileHuman1645
CHEK1 (CHK1)CAMKLCAMK2ym8A(r)-5-(8-chloroisoquinolin-3-ylamino)-3-(1-(dimethylamino)propan-2-yloxy)pyrazine-2-carbonitrileHuman1588
CHEK1 (CHK1)CAMKLCAMK2ywpA1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)ureaHuman1658
CHEK1 (CHK1)CAMKLCAMK3f9nAA-Human1700
CHEK1 (CHK1)CAMKLCAMK3f9nAB-Human1666
CHEK1 (CHK1)CAMKLCAMK3jvrA-Human1625
CHEK1 (CHK1)CAMKLCAMK3jvsA-Human1630
CHEK1 (CHK1)CAMKLCAMK3nlbA3-methyl-5-[5-(1-methylethyl)-1h-benzimidazol-2-yl]-n-(1-methylpiperidin-4-yl)-1h-pyrazole-4-carboxamideHuman1641
CHEK1 (CHK1)CAMKLCAMK3ot3AA5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amineHuman1696
CHEK1 (CHK1)CAMKLCAMK3ot3AB5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amineHuman1602
CHEK1 (CHK1)CAMKLCAMK3ot8AAn-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amineHuman1569
CHEK1 (CHK1)CAMKLCAMK3ot8ABn-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amineHuman1590
CHEK1 (CHK1)CAMKLCAMK3pa3AA2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamideHuman1691
CHEK1 (CHK1)CAMKLCAMK3pa3AB2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamideHuman1635
CHEK1 (CHK1)CAMKLCAMK3pa4AA2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamideHuman1592
CHEK1 (CHK1)CAMKLCAMK3pa4AB2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamideHuman1566
CHEK1 (CHK1)CAMKLCAMK3pa5AA2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamideHuman1676
CHEK1 (CHK1)CAMKLCAMK3pa5AB2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamideHuman1544
CHEK1 (CHK1)CAMKLCAMK3tkhA1-(morpholin-4-yl)-2-[4-(2-{[5-(pyridin-3-yl)-1,3-thiazol-2-yl]amino}pyridin-4-yl)piperazin-1-yl]ethanoneHuman1665
CHEK1 (CHK1)CAMKLCAMK3tkiAn-(2-aminoethyl)-5-(2-{[4-(morpholin-4-yl)pyridin-2-yl]amino}-1,3-thiazol-5-yl)pyridine-3-carboxamideHuman1599
CHEK1 (CHK1)CAMKLCAMK3u9nA2-(2,3-dihydro-1-benzofuran-5-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman1597
CHEK1 (CHK1)CAMKLCAMK4fsmAA4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenolHuman1570
CHEK1 (CHK1)CAMKLCAMK4fsmAB4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenolHuman1671
CHEK1 (CHK1)CAMKLCAMK4fsnAA4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHuman1542
CHEK1 (CHK1)CAMKLCAMK4fsnAB4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHuman1679
CHEK1 (CHK1)CAMKLCAMK4fsqAA4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-olHuman1688
CHEK1 (CHK1)CAMKLCAMK4fsqAB4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-olHuman1598
CHEK1 (CHK1)CAMKLCAMK4fsrAA6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazoleHuman1629
CHEK1 (CHK1)CAMKLCAMK4fsrAB6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazoleHuman1575
CHEK1 (CHK1)CAMKLCAMK4fstAA4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenolHuman1619
CHEK1 (CHK1)CAMKLCAMK4fstAB4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenolHuman1663
CHEK1 (CHK1)CAMKLCAMK4fsuAA4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrileHuman1539
CHEK1 (CHK1)CAMKLCAMK4fsuAB4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrileHuman1615
CHEK1 (CHK1)CAMKLCAMK4fswAA8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1541
CHEK1 (CHK1)CAMKLCAMK4fswAB8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1623
CHEK1 (CHK1)CAMKLCAMK4fsyAA2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamideHuman1547
CHEK1 (CHK1)CAMKLCAMK4fsyAB2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamideHuman1537
CHEK1 (CHK1)CAMKLCAMK4fszAA(3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acidHuman1553
CHEK1 (CHK1)CAMKLCAMK4fszAB(3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acidHuman1628
CHEK1 (CHK1)CAMKLCAMK4ft0AA2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acidHuman1637
CHEK1 (CHK1)CAMKLCAMK4ft0AB2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acidHuman1693
CHEK1 (CHK1)CAMKLCAMK4ft3AA1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylureaHuman1554
CHEK1 (CHK1)CAMKLCAMK4ft3AB1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylureaHuman1672
CHEK1 (CHK1)CAMKLCAMK4ft5AA1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1617
CHEK1 (CHK1)CAMKLCAMK4ft5AB1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1633
CHEK1 (CHK1)CAMKLCAMK4ft7AA1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1610
CHEK1 (CHK1)CAMKLCAMK4ft7AB1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1557
CHEK1 (CHK1)CAMKLCAMK4ft9AA1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylureaHuman1564
CHEK1 (CHK1)CAMKLCAMK4ft9AB1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylureaHuman1648
CHEK1 (CHK1)CAMKLCAMK4ftaAA6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acidHuman1540
CHEK1 (CHK1)CAMKLCAMK4ftaAB6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acidHuman1660
CHEK1 (CHK1)CAMKLCAMK4ftcAA1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)ureaHuman1593
CHEK1 (CHK1)CAMKLCAMK4ftcAB1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)ureaHuman1680
CHEK1 (CHK1)CAMKLCAMK4ftiAAmethyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylateHuman1577
CHEK1 (CHK1)CAMKLCAMK4ftiABmethyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylateHuman1659
CHEK1 (CHK1)CAMKLCAMK4ftjAAtrans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanolHuman1603
CHEK1 (CHK1)CAMKLCAMK4ftjABtrans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanolHuman1613
CHEK1 (CHK1)CAMKLCAMK4ftkAA3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-olHuman1608
CHEK1 (CHK1)CAMKLCAMK4ftkAB3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-olHuman1536
CHEK1 (CHK1)CAMKLCAMK4ftlAA4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-olHuman1614
CHEK1 (CHK1)CAMKLCAMK4ftlAB4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-olHuman1573
CHEK1 (CHK1)CAMKLCAMK4ftmAA4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenolHuman1546
CHEK1 (CHK1)CAMKLCAMK4ftmAB4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenolHuman1556
CHEK1 (CHK1)CAMKLCAMK4ftmAC4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenolHuman1616
CHEK1 (CHK1)CAMKLCAMK4ftnAA4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-olHuman1695
CHEK1 (CHK1)CAMKLCAMK4ftnAB4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-olHuman1678
CHEK1 (CHK1)CAMKLCAMK4ftoAA4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrileHuman1661
CHEK1 (CHK1)CAMKLCAMK4ftoAB4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrileHuman1605
CHEK1 (CHK1)CAMKLCAMK4ftqAA5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrileHuman1664
CHEK1 (CHK1)CAMKLCAMK4ftqAB5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrileHuman1550
CHEK1 (CHK1)CAMKLCAMK4ftrAA2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamideHuman1692
CHEK1 (CHK1)CAMKLCAMK4ftrAB2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamideHuman1535
CHEK1 (CHK1)CAMKLCAMK4fttAAmethyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1565
CHEK1 (CHK1)CAMKLCAMK4fttABmethyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1670
CHEK1 (CHK1)CAMKLCAMK4ftuAAmethyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1639
CHEK1 (CHK1)CAMKLCAMK4ftuABmethyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1640
CHEK1 (CHK1)CAMKLCAMK4gh2AA3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1600
CHEK1 (CHK1)CAMKLCAMK4gh2AB3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1652
CHEK1 (CHK1)CAMKLCAMK4hyhAA2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamideHuman1561
CHEK1 (CHK1)CAMKLCAMK4hyhAB2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamideHuman1626
CHEK1 (CHK1)CAMKLCAMK4hyiAA2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman1538
CHEK1 (CHK1)CAMKLCAMK4hyiAB2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman1681
CHEK1 (CHK1)CAMKLCAMK4jikA2-(4-chlorophenyl)-8-[(3s)-piperidin-3-ylamino]imidazo[1,2-c]pyrimidine-5-carboxamideHuman1698
CHEK1 (CHK1)CAMKLCAMK4qyeA4-[6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acidHuman1601
CHEK1 (CHK1)CAMKLCAMK4qyfA4-[3-amino-6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acidHuman1622
CHEK1 (CHK1)CAMKLCAMK4qygA3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acidHuman1568
CHEK1 (CHK1)CAMKLCAMK4qygB3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acidHuman1607
CHEK1 (CHK1)CAMKLCAMK4qyhA3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1689
CHEK1 (CHK1)CAMKLCAMK4qyhB3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1586
CHEK1 (CHK1)CAMKLCAMK4rvkAn-[3-(6-cyano-9h-pyrrolo[2,3-b:5,4-c']dipyridin-3-yl)phenyl]acetamideHuman1549
CHEK1 (CHK1)CAMKLCAMK4rvlA3-(2-hydroxyphenyl)-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1634
CHEK1 (CHK1)CAMKLCAMK4rvmA3-[4-(piperidin-1-ylmethyl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1624
CHEK1 (CHK1)CAMKLCAMK5dlsA1-benzyl-n-(5-{5-[3-(dimethylamino)-2,2-dimethylpropoxy]-1h-indol-2-yl}-6-oxo-1,6-dihydropyridin-3-yl)-1h-pyrazole-4-carboxamideHuman6151
CHEK1 (CHK1)CAMKLCAMK5f4nAAmethyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylateHuman6651
CHEK1 (CHK1)CAMKLCAMK5f4nABmethyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylateHuman6652
CHEK1 (CHK1)CAMKLCAMK5oopAAphosphoaminophosphonic acid-adenylate esterHuman8612
CHEK1 (CHK1)CAMKLCAMK5oopABphosphoaminophosphonic acid-adenylate esterHuman8607
CHEK1 (CHK1)CAMKLCAMK5oorAstaurosporineHuman8603
CHEK1 (CHK1)CAMKLCAMK5ootA2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman8599
CHEK1 (CHK1)CAMKLCAMK5op2AA5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8595
CHEK1 (CHK1)CAMKLCAMK5op2AB5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8611
CHEK1 (CHK1)CAMKLCAMK5op4A[4-[[4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-fluoranyl-5-methoxy-phenyl]-morpholin-4-yl-methanoneHuman8613
CHEK1 (CHK1)CAMKLCAMK5op5A3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrileHuman8600
CHEK1 (CHK1)CAMKLCAMK5op7A[4-[[5-chloranyl-4-(methylamino)-7~{h}-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-phenyl]-morpholin-4-yl-methanoneHuman8609
CHEK1 (CHK1)CAMKLCAMK5opbAA(2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholineHuman8602
CHEK1 (CHK1)CAMKLCAMK5opbAB(2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholineHuman8604
CHEK1 (CHK1)CAMKLCAMK5oprA5-[4-(morpholin-4-ylmethyl)phenyl]-3-(1-propan-2-yl-1,2,3-triazol-4-yl)pyridin-2-amineHuman8614
CHEK1 (CHK1)CAMKLCAMK5opsA4-(3-hydroxyphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrileHuman8598
CHEK1 (CHK1)CAMKLCAMK5opuA6-azanyl-4-(3-methylphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrileHuman8615
CHEK1 (CHK1)CAMKLCAMK5opvA4-(3-methylphenyl)-6-[(1-methylpyrazol-3-yl)amino]-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrileHuman8608
CHEK1 (CHK1)CAMKLCAMK5oq5A2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman8597
CHEK1 (CHK1)CAMKLCAMK5oq6A2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman8610
CHEK1 (CHK1)CAMKLCAMK5oq7AA5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8601
CHEK1 (CHK1)CAMKLCAMK5oq7AB5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8594
CHEK1 (CHK1)CAMKLCAMK5oq7BA5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8605
CHEK1 (CHK1)CAMKLCAMK5oq7BB5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8596
CHEK1 (CHK1)CAMKLCAMK5oq8A5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8606
CHEK1 (CHK1)CAMKLCAMK6fc8AA2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamideHuman9500
CHEK1 (CHK1)CAMKLCAMK6fc8AB2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamideHuman9502
CHEK1 (CHK1)CAMKLCAMK6fcfAA4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamideHuman9503
CHEK1 (CHK1)CAMKLCAMK6fcfAB4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamideHuman9498
CHEK1 (CHK1)CAMKLCAMK6fckAA2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamideHuman9501
CHEK1 (CHK1)CAMKLCAMK6fckAB2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamideHuman9499
CHEK1 (CHK1)CAMKLCAMK7akmAAphosphothiophosphoric acid-adenylate esterHuman13489
CHEK1 (CHK1)CAMKLCAMK7akmABphosphothiophosphoric acid-adenylate esterHuman13491
CHEK1 (CHK1)CAMKLCAMK7akmBA-Human13494
CHEK1 (CHK1)CAMKLCAMK7akmBB-Human13493
CHEK1 (CHK1)CAMKLCAMK7akoAAstaurosporineHuman13490
CHEK1 (CHK1)CAMKLCAMK7akoABstaurosporineHuman13495
CHEK1 (CHK1)CAMKLCAMK7akoBAstaurosporineHuman13492
CHEK1 (CHK1)CAMKLCAMK7akoBBstaurosporineHuman13496
CHEK1 (CHK1)CAMKLCAMK7bjdAA2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrileHuman13775
CHEK1 (CHK1)CAMKLCAMK7bjdAB2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrileHuman13774
CHEK1 (CHK1)CAMKLCAMK7bjeAAadenineHuman13767
CHEK1 (CHK1)CAMKLCAMK7bjeABadenineHuman13773
CHEK1 (CHK1)CAMKLCAMK7bjhAAn,n-dimethyl-7h-purin-6-amineHuman13776
CHEK1 (CHK1)CAMKLCAMK7bjhABn,n-dimethyl-7h-purin-6-amineHuman13771
CHEK1 (CHK1)CAMKLCAMK7bjjAA1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman13777
CHEK1 (CHK1)CAMKLCAMK7bjjAB1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman13779
CHEK1 (CHK1)CAMKLCAMK7bjmA4-amino-6-{[(2-fluorophenyl)methyl]amino}-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13770
CHEK1 (CHK1)CAMKLCAMK7bjoA4-amino-6-(2,3-difluorophenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13780
CHEK1 (CHK1)CAMKLCAMK7bjrA4-amino-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13778
CHEK1 (CHK1)CAMKLCAMK7bjxAA4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13772
CHEK1 (CHK1)CAMKLCAMK7bjxAB4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13768
CHEK1 (CHK1)CAMKLCAMK7bk1A4-amino-2-[(1,3-dimethyl-1h-pyrazol-4-yl)amino]-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13763
CHEK1 (CHK1)CAMKLCAMK7bk2A4-amino-7-methyl-2-({5-methyl-1-[(3r)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13766
CHEK1 (CHK1)CAMKLCAMK7bk3A4-amino-7-methyl-2-({5-methyl-1-[(3s)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13764
CHEK1 (CHK1)CAMKLCAMK7bknAadenineHuman13769
CHEK1 (CHK1)CAMKLCAMK7bkoA1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman13765
CHEK1 (CHK1)CAMKLCAMK7mckAn-{5-[(3s)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl}-6-(1-methyl-1h-pyrazol-4-yl)pyridine-2-carboxamideHuman13622
CHEK1 (CHK1)CAMKLCAMK7sufAA8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amineHuman14040
CHEK1 (CHK1)CAMKLCAMK7sufAB8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amineHuman14044
CHEK1 (CHK1)CAMKLCAMK7sugAA1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrileHuman14039
CHEK1 (CHK1)CAMKLCAMK7sugAB1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrileHuman14042
CHEK1 (CHK1)CAMKLCAMK7suhA1-[5-chloro-4-({6-chloro-7-[1-(oxetan-3-yl)piperidin-4-yl]quinazolin-2-yl}amino)-1h-pyrazol-1-yl]-2-methylpropan-2-olHuman14043
CHEK1 (CHK1)CAMKLCAMK7suiA(3r,4r)-4-{(3s,4s)-4-[6-chloro-2-({5-chloro-1-[(1r)-2,2-difluorocyclopropyl]-1h-pyrazol-4-yl}amino)quinazolin-7-yl]-3-fluoropiperidin-1-yl}oxolan-3-olHuman14045
CHEK1 (CHK1)CAMKLCAMK7sujA(3r,4r)-4-{4-[6-chloro-2-({1-[(1r)-2,2-difluorocyclopropyl]-5-methyl-1h-pyrazol-4-yl}amino)quinazolin-7-yl]piperidin-1-yl}-4-methyloxolan-3-olHuman14041
CHEK1 (CHK1)CAMKLCAMK8e80A2-[(1r,4r)-2-{(6p)-6-[(6m)-6-(1h-pyrazol-5-yl)-1h-indazol-1-yl]pyrimidin-4-yl}-2-azabicyclo[2.1.1]hexan-4-yl]propan-2-olHuman14621
CHEK1 (CHK1)CAMKLCAMK8e81A(1s)-1-[(1p)-1-{6-[(3r)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}-1h-indazol-6-yl]spiro[2.2]pentane-1-carbonitrileHuman14620
CHEK1 (CHK1)CAMKLCAMK8sivAn-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)cyclopropanecarboxamideHuman14886
CHEK1 (CHK1)CAMKLCAMK8siwA(1s,2s)-n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)-2-(1-methyl-1h-pyrazol-4-yl)cyclopropane-1-carboxamideHuman14885
CHEK1 (CHK1)CAMKLCAMK8sixA(1s)-n-(7-chloro-6-{4-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperazin-1-yl}isoquinolin-3-yl)-6-oxaspiro[2.5]octane-1-carboxamideHuman14887
CHEK2 (CHK2)RAD53CAMK2cn5Aadenosine-5'-diphosphateHuman4789
CHEK2 (CHK2)RAD53CAMK2cn8AdebromohymenialdisineHuman4808
CHEK2 (CHK2)RAD53CAMK2w0jA4,4'-diacetyldiphenylurea-bis(guanylhydrazone)Human4811
CHEK2 (CHK2)RAD53CAMK2w7xAAn-[4-[(e)-n-carbamimidamido-c-methyl-carbonimidoyl]phenyl]-7-nitro-1h-indole-2-carboxamideHuman4784
CHEK2 (CHK2)RAD53CAMK2w7xABn-[4-[(e)-n-carbamimidamido-c-methyl-carbonimidoyl]phenyl]-7-nitro-1h-indole-2-carboxamideHuman4780
CHEK2 (CHK2)RAD53CAMK2wtcA4-[2-amino-5-(4-hydroxy-3-methoxyphenyl)pyridin-3-yl]benzamideHuman4767
CHEK2 (CHK2)RAD53CAMK2wtdA4-[2-amino-5-(1,3-benzodioxol-4-yl)pyridin-3-yl]benzamideHuman4769
CHEK2 (CHK2)RAD53CAMK2wtiAA4-[2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)pyridin-3-yl]benzamideHuman4812
CHEK2 (CHK2)RAD53CAMK2wtiAB4-[2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)pyridin-3-yl]benzamideHuman4807
CHEK2 (CHK2)RAD53CAMK2wtjAA2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)-n-[2-(dimethylamino)ethyl]pyridine-3-carboxamideHuman4779
CHEK2 (CHK2)RAD53CAMK2wtjAB2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)-n-[2-(dimethylamino)ethyl]pyridine-3-carboxamideHuman4761
CHEK2 (CHK2)RAD53CAMK2xbjA4-fluoro-2-(4-{[(3s,4r)-4-(1-hydroxy-1-methylethyl)pyrrolidin-3-yl]amino}-6,7-dimethoxyquinazolin-2-yl)phenolHuman4783
CHEK2 (CHK2)RAD53CAMK2xk9An-{4-[(1e)-n-(n-hydroxycarbamimidoyl)ethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamideHuman4771
CHEK2 (CHK2)RAD53CAMK2xm8A2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenolHuman4773
CHEK2 (CHK2)RAD53CAMK2xm9AA4-(1h-pyrazol-5-yl)-2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenolHuman4785
CHEK2 (CHK2)RAD53CAMK2xm9AB4-(1h-pyrazol-5-yl)-2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenolHuman4803
CHEK2 (CHK2)RAD53CAMK2ycfAA(2e)-n-hydroxy-2-[1-(4-{[(4-{(1e)-1-[2-(n'-hydroxycarbamimidoyl)hydrazinylidene]ethyl}phenyl)carbamoyl]amino}phenyl)ethylidene]hydrazinecarboximidamideHuman4810
CHEK2 (CHK2)RAD53CAMK2ycfAB(2e)-n-hydroxy-2-[1-(4-{[(4-{(1e)-1-[2-(n'-hydroxycarbamimidoyl)hydrazinylidene]ethyl}phenyl)carbamoyl]amino}phenyl)ethylidene]hydrazinecarboximidamideHuman4774
CHEK2 (CHK2)RAD53CAMK2ycqAAn-{4-[(1e)-n-1h-imidazol-2-ylethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamideHuman4766
CHEK2 (CHK2)RAD53CAMK2ycqABn-{4-[(1e)-n-1h-imidazol-2-ylethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamideHuman4790
CHEK2 (CHK2)RAD53CAMK2ycrAA1,3-bis{4-[(1e)-n-(4,5-dihydro-1h-imidazol-2-yl)ethanehydrazonoyl]phenyl}ureaHuman4760
CHEK2 (CHK2)RAD53CAMK2ycrAB1,3-bis{4-[(1e)-n-(4,5-dihydro-1h-imidazol-2-yl)ethanehydrazonoyl]phenyl}ureaHuman4775
CHEK2 (CHK2)RAD53CAMK2ycsAAn-{4-[(1e)-n-carbamimidoylethanehydrazonoyl]phenyl}-1h-indole-3-carboxamideHuman4804
CHEK2 (CHK2)RAD53CAMK2ycsABn-{4-[(1e)-n-carbamimidoylethanehydrazonoyl]phenyl}-1h-indole-3-carboxamideHuman4764
CHEK2 (CHK2)RAD53CAMK2yiqAA(e)-5-(1-(2-carbamimidoylhydrazono)ethyl)-n-(1h-indol-6-yl)-1h-indole-2-carboxamideHuman4791
CHEK2 (CHK2)RAD53CAMK2yiqAB(e)-5-(1-(2-carbamimidoylhydrazono)ethyl)-n-(1h-indol-6-yl)-1h-indole-2-carboxamideHuman4800
CHEK2 (CHK2)RAD53CAMK2yirA(e)-n-(5-(2-carbamimidoylhydrazono)-5,6,7,8-tetrahydronaphthalen-2-yl)-7-nitro-1h-indole-2-carboxamideHuman4768
CHEK2 (CHK2)RAD53CAMK2yitAAn-{4-[(1e)-n-carbamimidoylbutanehydrazonoyl]phenyl}-5-methoxy-1h-indole-2-carboxamideHuman4777
CHEK2 (CHK2)RAD53CAMK2yitABn-{4-[(1e)-n-carbamimidoylbutanehydrazonoyl]phenyl}-5-methoxy-1h-indole-2-carboxamideHuman4770
CHEK2 (CHK2)RAD53CAMK3i6uA-Human4798
CHEK2 (CHK2)RAD53CAMK3i6uB-Human4787
CHEK2 (CHK2)RAD53CAMK3i6wA-Human4813
CHEK2 (CHK2)RAD53CAMK3i6wB-Human4792
CHEK2 (CHK2)RAD53CAMK3i6wC-Human4802
CHEK2 (CHK2)RAD53CAMK3i6wD-Human4805
CHEK2 (CHK2)RAD53CAMK3i6wE-Human4806
CHEK2 (CHK2)RAD53CAMK3i6wF-Human4776
CHEK2 (CHK2)RAD53CAMK3i6wG-Human4793
CHEK2 (CHK2)RAD53CAMK3i6wH-Human4799
CHEK2 (CHK2)RAD53CAMK4a9rA2-[4-(4-chlorophenoxy)phenyl]-1h-benzimidazole-6-carboxamideHuman4763
CHEK2 (CHK2)RAD53CAMK4a9sAA2-(4-(3-hydroxyphenoxy)phenyl)-1h-benzo[d]imidazole-5-carboxamideHuman4772
CHEK2 (CHK2)RAD53CAMK4a9sAB2-(4-(3-hydroxyphenoxy)phenyl)-1h-benzo[d]imidazole-5-carboxamideHuman4801
CHEK2 (CHK2)RAD53CAMK4a9tA2-(4-{[1-(4-chlorobenzyl)piperidin-4-yl]methoxy}phenyl)-1h-benzimidazole-5-carboxamideHuman4814
CHEK2 (CHK2)RAD53CAMK4a9uA2-{4-[(1-benzylpiperidin-4-yl)methoxy]phenyl}-1h-benzimidazole-6-carboxamideHuman4778
CHEK2 (CHK2)RAD53CAMK4bdaA3,4-dihydro[1,2,4]triazolo[1,5-a][3,1]benzimidazol-9-iumHuman4788
CHEK2 (CHK2)RAD53CAMK4bdbA4-[(e)-c-methyl-n-oxidanyl-carbonimidoyl]benzene-1,3-diolHuman4797
CHEK2 (CHK2)RAD53CAMK4bdcAn-(furan-2-ylmethyl)quinoxaline-6-carboxamideHuman4794
CHEK2 (CHK2)RAD53CAMK4bddA1-(tert-butyl)-3-(quinoxalin-6-yl)ureaHuman4786
CHEK2 (CHK2)RAD53CAMK4bdeA6-methylquinazolin-4-amineHuman4781
CHEK2 (CHK2)RAD53CAMK4bdfA5-methyl-3-phenyl-1h-pyrazoleHuman4765
CHEK2 (CHK2)RAD53CAMK4bdgA3-(pyridin-3-yl)-1h-pyrazol-5-amineHuman4796
CHEK2 (CHK2)RAD53CAMK4bdhA3-methyl-4-(thiophen-2-yl)-1h-pyrazol-5-amineHuman4782
CHEK2 (CHK2)RAD53CAMK4bdiA1-acetyl-n-(5-methylpyridin-2-yl)piperidine-4-carboxamideHuman4762
CHEK2 (CHK2)RAD53CAMK4bdjA3-cyclopropyl-4-(furan-2-yl)-1h-pyrazolo[3,4-b]pyridineHuman4795
CHEK2 (CHK2)RAD53CAMK4bdkAn-[(4-methoxyphenyl)methyl]quinoxaline-6-carboxamideHuman4809
CHUK (IKKa)IKKOther5ebzA2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7153
CHUK (IKKa)IKKOther5ebzB2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7145
CHUK (IKKa)IKKOther5ebzC2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7146
CHUK (IKKa)IKKOther5ebzD2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7144
CHUK (IKKa)IKKOther5ebzE2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7151
CHUK (IKKa)IKKOther5ebzF2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7149
CHUK (IKKa)IKKOther5ebzG2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7154
CHUK (IKKa)IKKOther5ebzH2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7155
CHUK (IKKa)IKKOther5ebzI2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7152
CHUK (IKKa)IKKOther5ebzJ2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7148
CHUK (IKKa)IKKOther5ebzK2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7150
CHUK (IKKa)IKKOther5ebzL2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7147
CHUK (IKKa)IKKOther5tqwA-Human7249
CHUK (IKKa)IKKOther5tqwB-Human7248
CHUK (IKKa)IKKOther5tqxA-Human7261
CHUK (IKKa)IKKOther5tqxB-Human7262
CHUK (IKKa)IKKOther5tqyA-Human7196
CHUK (IKKa)IKKOther5tqyB-Human7197
CLK1CLKCMGC1z57AAdebromohymenialdisineHuman106
CLK1CLKCMGC1z57ABdebromohymenialdisineHuman105
CLK1CLKCMGC2vagAAethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman104
CLK1CLKCMGC2vagABethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman103
CLK1CLKCMGC5j1vApyrido[3,4-g]quinazoline-2,10-diamineHuman6582
CLK1CLKCMGC5j1vBpyrido[3,4-g]quinazoline-2,10-diamineHuman6580
CLK1CLKCMGC5j1vCpyrido[3,4-g]quinazoline-2,10-diamineHuman6577
CLK1CLKCMGC5j1wAApyrido[3,4-g]quinazolin-2-amineHuman6579
CLK1CLKCMGC5j1wABpyrido[3,4-g]quinazolin-2-amineHuman6576
CLK1CLKCMGC5j1wBApyrido[3,4-g]quinazolin-2-amineHuman6575
CLK1CLKCMGC5j1wBBpyrido[3,4-g]quinazolin-2-amineHuman6583
CLK1CLKCMGC5j1wCApyrido[3,4-g]quinazolin-2-amineHuman6578
CLK1CLKCMGC5j1wCBpyrido[3,4-g]quinazolin-2-amineHuman6581
CLK1CLKCMGC5x8iA5-[1-[(1s)-1-(4-fluorophenyl)ethyl]-[1,2,3]triazolo[4,5-c]quinolin-8-yl]-1,3-benzoxazoleHuman8316
CLK1CLKCMGC5x8iB5-[1-[(1s)-1-(4-fluorophenyl)ethyl]-[1,2,3]triazolo[4,5-c]quinolin-8-yl]-1,3-benzoxazoleHuman8317
CLK1CLKCMGC6ft8AA3-(3-hydroxyphenyl)-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9895
CLK1CLKCMGC6ft8AB3-(3-hydroxyphenyl)-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9899
CLK1CLKCMGC6ft9AA2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9901
CLK1CLKCMGC6ft9AB2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9898
CLK1CLKCMGC6ft9BA2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9897
CLK1CLKCMGC6ft9BB2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9894
CLK1CLKCMGC6ft9CA2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9896
CLK1CLKCMGC6ft9CB2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9900
CLK1CLKCMGC6fyoAA6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHuman10324
CLK1CLKCMGC6fyoAB6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHuman10323
CLK1CLKCMGC6g33AA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9819
CLK1CLKCMGC6g33AB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9824
CLK1CLKCMGC6g33AC-Human9826
CLK1CLKCMGC6g33BA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9821
CLK1CLKCMGC6g33BB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9822
CLK1CLKCMGC6g33BC-Human9827
CLK1CLKCMGC6g33CA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9825
CLK1CLKCMGC6g33CB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9823
CLK1CLKCMGC6g33CC-Human9820
CLK1CLKCMGC6i5hAA5-(1-methylpyrazol-4-yl)-3-(3-phenoxyphenyl)furo[3,2-b]pyridineHuman10848
CLK1CLKCMGC6i5hAB5-(1-methylpyrazol-4-yl)-3-(3-phenoxyphenyl)furo[3,2-b]pyridineHuman10849
CLK1CLKCMGC6i5iAA5-(1-methylpyrazol-4-yl)-3-[1-(phenylmethyl)pyrazol-4-yl]furo[3,2-b]pyridineHuman10845
CLK1CLKCMGC6i5iAB5-(1-methylpyrazol-4-yl)-3-[1-(phenylmethyl)pyrazol-4-yl]furo[3,2-b]pyridineHuman10840
CLK1CLKCMGC6i5kAA5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10844
CLK1CLKCMGC6i5kAB5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10836
CLK1CLKCMGC6i5kBA5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10842
CLK1CLKCMGC6i5kBB5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10835
CLK1CLKCMGC6i5kCA5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10834
CLK1CLKCMGC6i5kCB5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10838
CLK1CLKCMGC6i5lAA3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10837
CLK1CLKCMGC6i5lAB3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10843
CLK1CLKCMGC6i5lBA3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10846
CLK1CLKCMGC6i5lBB3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10839
CLK1CLKCMGC6i5lCA3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10833
CLK1CLKCMGC6i5lCB3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10841
CLK1CLKCMGC6khdAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11646
CLK1CLKCMGC6khdAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11645
CLK1CLKCMGC6khdBA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11644
CLK1CLKCMGC6khdBB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11647
CLK1CLKCMGC6khdCA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11648
CLK1CLKCMGC6khdCB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11643
CLK1CLKCMGC6q8kAA~{n}2-(3-morpholin-4-ylpropyl)pyrido[3,4-g]quinazoline-2,10-diamineHuman10902
CLK1CLKCMGC6q8kAB~{n}2-(3-morpholin-4-ylpropyl)pyrido[3,4-g]quinazoline-2,10-diamineHuman10903
CLK1CLKCMGC6q8pA~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amineHuman10899
CLK1CLKCMGC6q8pB~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amineHuman10900
CLK1CLKCMGC6q8pC~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amineHuman10901
CLK1CLKCMGC6qtyAAethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman12083
CLK1CLKCMGC6qtyABethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman12084
CLK1CLKCMGC6r3dA4-[6,7-bis(chloranyl)-1~{h}-indol-3-yl]pyrimidin-2-amineHuman12128
CLK1CLKCMGC6r6eA5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amineHuman12232
CLK1CLKCMGC6r6xA5-(1-methylindol-3-yl)pyrimidin-4-amineHuman12231
CLK1CLKCMGC6r8jAA4-(1-methylindol-3-yl)pyrimidin-2-amineHuman12632
CLK1CLKCMGC6r8jAB4-(1-methylindol-3-yl)pyrimidin-2-amineHuman12631
CLK1CLKCMGC6raaAA4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11014
CLK1CLKCMGC6raaAB4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11013
CLK1CLKCMGC6tw2EAethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman11962
CLK1CLKCMGC6tw2EBethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman11963
CLK1CLKCMGC6ytaAA1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman12423
CLK1CLKCMGC6ytaAB1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman12417
CLK1CLKCMGC6ytdAA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12418
CLK1CLKCMGC6ytdAB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12420
CLK1CLKCMGC6yteCA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12419
CLK1CLKCMGC6yteCB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12422
CLK1CLKCMGC6ytgAA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12416
CLK1CLKCMGC6ytgAB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12424
CLK1CLKCMGC6ytiAAmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman12413
CLK1CLKCMGC6ytiABmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman12414
CLK1CLKCMGC6z4zAA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12315
CLK1CLKCMGC6z4zAB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12312
CLK1CLKCMGC6z4zBA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12310
CLK1CLKCMGC6z4zBB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12311
CLK1CLKCMGC6z4zCA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12309
CLK1CLKCMGC6z4zCB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12313
CLK1CLKCMGC6z50AA11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12314
CLK1CLKCMGC6z50AB11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12308
CLK1CLKCMGC6zlnAA4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman12711
CLK1CLKCMGC6zlnAB4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman12710
CLK1CLKCMGC7ak3AA~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman13142
CLK1CLKCMGC7ak3AB~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman13143
CLK1CLKCMGC7o9yA4-(1~{h}-indol-3-yl)pyrimidin-2-amineHuman14208
CLK1CLKCMGC7oa0A5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amineHuman14207
CLK1CLKCMGC7opgAA4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenolHuman13808
CLK1CLKCMGC7opgAB4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenolHuman13809
CLK1CLKCMGC8p04A(4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-oneHuman14741
CLK1CLKCMGC8p08A(4~{z})-4-(1,3-benzothiazol-6-ylmethylidene)-2-[[(2~{r})-1-methoxy-4-methyl-pentan-2-yl]amino]-1~{h}-imidazol-5-oneHuman14742
CLK2CLKCMGC3nr9A(5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman1927
CLK2CLKCMGC3nr9B(5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman1928
CLK2CLKCMGC3nr9C(5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman1929
CLK2CLKCMGC5unpAn~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamineHuman9887
CLK2CLKCMGC5unpBn~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamineHuman9888
CLK2CLKCMGC6fyiA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman10405
CLK2CLKCMGC6fykAA(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10406
CLK2CLKCMGC6fykAB(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10408
CLK2CLKCMGC6fykBA(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10407
CLK2CLKCMGC6fykBB(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10401
CLK2CLKCMGC6fykCA(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10402
CLK2CLKCMGC6fykCB(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10409
CLK2CLKCMGC6fylAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10403
CLK2CLKCMGC6fylAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10404
CLK2CLKCMGC6kheA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11651
CLK3CLKCMGC2eu9AA-Human1826
CLK3CLKCMGC2eu9AB-Human1830
CLK3CLKCMGC2exeAA-Human1822
CLK3CLKCMGC2exeAB-Human1819
CLK3CLKCMGC2wu6AA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman1823
CLK3CLKCMGC2wu6AB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman1821
CLK3CLKCMGC2wu7AAethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman1828
CLK3CLKCMGC2wu7ABethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman1827
CLK3CLKCMGC3rawAA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman1820
CLK3CLKCMGC3rawAB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman1829
CLK3CLKCMGC3rawBA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman1824
CLK3CLKCMGC3rawBB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman1825
CLK3CLKCMGC6ft7AA3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9905
CLK3CLKCMGC6ft7AB3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9903
CLK3CLKCMGC6ft7BA3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9904
CLK3CLKCMGC6ft7BB3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9902
CLK3CLKCMGC6fypAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10400
CLK3CLKCMGC6fypAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10397
CLK3CLKCMGC6fyrAA6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHuman11407
CLK3CLKCMGC6fyrAB6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHuman11406
CLK3CLKCMGC6khfAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11650
CLK3CLKCMGC6khfAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11649
CLK3CLKCMGC6rctAA4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11127
CLK3CLKCMGC6rctAB4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11126
CLK3CLKCMGC6rctBA4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11128
CLK3CLKCMGC6rctBB4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11129
CLK3CLKCMGC6ytwAA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12404
CLK3CLKCMGC6ytwAB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12407
CLK3CLKCMGC6ytwBA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12412
CLK3CLKCMGC6ytwBB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12410
CLK3CLKCMGC6ytyAA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12409
CLK3CLKCMGC6ytyAB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12406
CLK3CLKCMGC6yu1aA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12403
CLK3CLKCMGC6yu1aB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12408
CLK3CLKCMGC6yu1cA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12405
CLK3CLKCMGC6yu1cB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12411
CLK3CLKCMGC6z2vAA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12637
CLK3CLKCMGC6z2vAB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12636
CLK3CLKCMGC6z51AAn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide Human12296
CLK3CLKCMGC6z51ABn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide Human12304
CLK3CLKCMGC6z52AA11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12628
CLK3CLKCMGC6z52AB11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12627
CLK3CLKCMGC6z52BA11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12629
CLK3CLKCMGC6z52BB11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12626
CLK3CLKCMGC6z53AA6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12300
CLK3CLKCMGC6z53AB6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12305
CLK3CLKCMGC6z54AA11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12294
CLK3CLKCMGC6z54AB11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12295
CLK3CLKCMGC6z55AA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12302
CLK3CLKCMGC6z55AB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12298
CLK3CLKCMGC6z55AC7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12301
CLK3CLKCMGC6z55BA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12303
CLK3CLKCMGC6z55BB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12299
CLK3CLKCMGC6z55BC7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12297
CLK4CLKCMGC6fyvAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10511
CLK4CLKCMGC6fyvAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10510
COQ8A (ADCK3)ABC1Atypical4pedAA-Human9121
COQ8A (ADCK3)ABC1Atypical4pedAB-Human9120
COQ8A (ADCK3)ABC1Atypical5i35Aphosphoaminophosphonic acid-adenylate esterHuman9122
COQ8A (ADCK3)ABC1Atypical7udpA4-[(3,4,5-trimethoxyphenyl)amino]quinoline-7-carbonitrileHuman14589
COQ8A (ADCK3)ABC1Atypical7udqA4-[(3,4,5-trimethoxyphenyl)amino]quinoline-7-carbonitrileHuman14588
CSF1R (FMS)PDGFRTK2i0vA6-chloro-3-(3-methylisoxazol-5-yl)-4-phenylquinolin-2(1h)-oneHuman2303
CSF1R (FMS)PDGFRTK2i0yA5-cyano-furan-2-carboxylic acid [5-hydroxymethyl-2-(4-methyl-piperidin-1-yl)-phenyl]-amideHuman2315
CSF1R (FMS)PDGFRTK2i1mA5-cyano-furan-2-carboxylic acid [5-hydroxymethyl-2-(4-methyl-piperidin-1-yl)-phenyl]-amideHuman2306
CSF1R (FMS)PDGFRTK2ogvA-Human1243
CSF1R (FMS)PDGFRTK3beaA8-(2,3-dihydro-1h-inden-5-yl)-2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]phenyl}amino)-5-oxo-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman6761
CSF1R (FMS)PDGFRTK3dpkAA8-cyclohexyl-n-methoxy-5-oxo-2-{[4-(2-pyrrolidin-1-ylethyl)phenyl]amino}-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman2312
CSF1R (FMS)PDGFRTK3dpkAB8-cyclohexyl-n-methoxy-5-oxo-2-{[4-(2-pyrrolidin-1-ylethyl)phenyl]amino}-5,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman2305
CSF1R (FMS)PDGFRTK3krjAA4-cyano-n-(2-cyclohex-1-en-1-yl-4-piperidin-4-ylphenyl)-1h-imidazole-2-carboxamideHuman2302
CSF1R (FMS)PDGFRTK3krjAB4-cyano-n-(2-cyclohex-1-en-1-yl-4-piperidin-4-ylphenyl)-1h-imidazole-2-carboxamideHuman2310
CSF1R (FMS)PDGFRTK3krlAA5-cyano-n-[4-(4-methylpiperazin-1-yl)-2-piperidin-1-ylphenyl]furan-2-carboxamideHuman2309
CSF1R (FMS)PDGFRTK3krlAB5-cyano-n-[4-(4-methylpiperazin-1-yl)-2-piperidin-1-ylphenyl]furan-2-carboxamideHuman2311
CSF1R (FMS)PDGFRTK3lcdAAn~3~-(2,6-dichlorobenzyl)-5-(4-{[(2r)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]carbonyl}phenyl)pyrazine-2,3-diamineHuman1241
CSF1R (FMS)PDGFRTK3lcdABn~3~-(2,6-dichlorobenzyl)-5-(4-{[(2r)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]carbonyl}phenyl)pyrazine-2,3-diamineHuman1242
CSF1R (FMS)PDGFRTK3lcoAA3-({4-methoxy-5-[(4-methoxybenzyl)oxy]pyridin-2-yl}methoxy)-5-(1-methyl-1h-pyrazol-4-yl)pyrazin-2-amineHuman2314
CSF1R (FMS)PDGFRTK3lcoAB3-({4-methoxy-5-[(4-methoxybenzyl)oxy]pyridin-2-yl}methoxy)-5-(1-methyl-1h-pyrazol-4-yl)pyrazin-2-amineHuman2313
CSF1R (FMS)PDGFRTK4hw7A5-[(5-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-[4-(trifluoromethyl)benzyl]pyridin-2-amineHuman2304
CSF1R (FMS)PDGFRTK4r7hA5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amineHuman2308
CSF1R (FMS)PDGFRTK4r7iA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman2307
CSF1R (FMS)PDGFRTK6ig8AA(3-{4-[(4-cyclopropylphenyl)methoxy]-3-methoxyphenyl}azetidin-1-yl)(4-{[(2s)-2,3-dihydroxypropoxy]methyl}pyridin-2-yl)methanoneHuman11519
CSF1R (FMS)PDGFRTK6ig8AB(3-{4-[(4-cyclopropylphenyl)methoxy]-3-methoxyphenyl}azetidin-1-yl)(4-{[(2s)-2,3-dihydroxypropoxy]methyl}pyridin-2-yl)methanoneHuman11518
CSF1R (FMS)PDGFRTK6n33A6-fluoro-n-[(5-fluoro-2-methoxypyridin-3-yl)methyl]-5-[(5-methyl-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]pyridin-2-amineHuman11634
CSF1R (FMS)PDGFRTK6t2wA2-[(4-methoxy-2-methyl-phenyl)amino]-7-methyl-9-(4-oxidanylcyclohexyl)purin-8-oneHuman11905
CSF1R (FMS)PDGFRTK6wxjA4-(3-{[(2s)-2-(6-methoxypyridin-3-yl)-2,3-dihydro-1,4-benzodioxin-6-yl]methyl}-3h-imidazo[4,5-b]pyridin-6-yl)-2-methylbut-3-yn-2-amineHuman13337
CSF1R (FMS)PDGFRTK7mfcAAvimseltinibHuman13990
CSF1R (FMS)PDGFRTK7mfcABvimseltinibHuman13989
CSF1R (FMS)PDGFRTK7tnhA2,2-dimethyl-n-[(6-methyl-5-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}pyridin-2-yl)carbamoyl]propanamideHuman14350
CSF1R (FMS)PDGFRTK8cgcAA[4-[4-[methyl-[(3-methylphenyl)methyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]methanolHuman14766
CSF1R (FMS)PDGFRTK8cgcAB[4-[4-[methyl-[(3-methylphenyl)methyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]methanolHuman14767
CSKCskTK1bygAstaurosporineHuman2943
CSKCskTK3d7tAstaurosporineHuman2941
CSKCskTK3d7uA-Human2942
CSKCskTK3d7uC-Human2944
CSNK1A1 (CK1a)CK1CK15fqdC-Human6415
CSNK1A1 (CK1a)CK1CK15fqdF-Human6416
CSNK1A1 (CK1a)CK1CK16gzdAA[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHuman10560
CSNK1A1 (CK1a)CK1CK16gzdAB[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHuman10561
CSNK1A1 (CK1a)CK1CK18g66C-Human15006
Csnk1d (CK1d)CK1CK14jjrA-Mouse5784
Csnk1d (CK1d)CK1CK14jjrB-Mouse5785
Csnk1d (CK1d)CK1CK15x17AAadenosine-5'-diphosphateMouse8546
Csnk1d (CK1d)CK1CK15x17ABadenosine-5'-diphosphateMouse8544
Csnk1d (CK1d)CK1CK15x17BAadenosine-5'-diphosphateMouse8545
Csnk1d (CK1d)CK1CK15x17BBadenosine-5'-diphosphateMouse8547
CSNK1D (CK1d)CK1CK13uysA-Human2183
CSNK1D (CK1d)CK1CK13uysB-Human2159
CSNK1D (CK1d)CK1CK13uysC-Human2149
CSNK1D (CK1d)CK1CK13uysD-Human2180
CSNK1D (CK1d)CK1CK13uytA4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman2182
CSNK1D (CK1d)CK1CK13uytB4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman2166
CSNK1D (CK1d)CK1CK13uytC4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman2152
CSNK1D (CK1d)CK1CK13uytD4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman2163
CSNK1D (CK1d)CK1CK13uzpA4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman2158
CSNK1D (CK1d)CK1CK13uzpB4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman2177
CSNK1D (CK1d)CK1CK14hgtA2-{2-[(3,4-difluorophenoxy)methyl]-5-methoxypyridin-4-yl}-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman2181
CSNK1D (CK1d)CK1CK14hgtB2-{2-[(3,4-difluorophenoxy)methyl]-5-methoxypyridin-4-yl}-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman2179
CSNK1D (CK1d)CK1CK14hnfA3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman2194
CSNK1D (CK1d)CK1CK14hnfB3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman2193
CSNK1D (CK1d)CK1CK14kb8AA1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamineHuman2171
CSNK1D (CK1d)CK1CK14kb8AB1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamineHuman2161
CSNK1D (CK1d)CK1CK14kb8BAn-benzyl-4-(pyridin-3-yl)pyrimidin-2-amineHuman2148
CSNK1D (CK1d)CK1CK14kb8BBn-benzyl-4-(pyridin-3-yl)pyrimidin-2-amineHuman2147
CSNK1D (CK1d)CK1CK14kb8CA1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamineHuman2189
CSNK1D (CK1d)CK1CK14kb8CB1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamineHuman2164
CSNK1D (CK1d)CK1CK14kb8DAn-benzyl-4-(pyridin-3-yl)pyrimidin-2-amineHuman2146
CSNK1D (CK1d)CK1CK14kb8DBn-benzyl-4-(pyridin-3-yl)pyrimidin-2-amineHuman2188
CSNK1D (CK1d)CK1CK14kbaAA9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepineHuman2151
CSNK1D (CK1d)CK1CK14kbaAB9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepineHuman2141
CSNK1D (CK1d)CK1CK14kbaBA9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepineHuman2191
CSNK1D (CK1d)CK1CK14kbaBB9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepineHuman2175
CSNK1D (CK1d)CK1CK14kbaCA9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepineHuman2172
CSNK1D (CK1d)CK1CK14kbaCB9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepineHuman2184
CSNK1D (CK1d)CK1CK14kbaDA9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepineHuman2160
CSNK1D (CK1d)CK1CK14kbaDB9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepineHuman2142
CSNK1D (CK1d)CK1CK14kbcAA{4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanolHuman2154
CSNK1D (CK1d)CK1CK14kbcAB{4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanolHuman2156
CSNK1D (CK1d)CK1CK14kbcBA{4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanolHuman2153
CSNK1D (CK1d)CK1CK14kbcBB{4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanolHuman2150
CSNK1D (CK1d)CK1CK14kbkAA(3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholineHuman2192
CSNK1D (CK1d)CK1CK14kbkAB(3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholineHuman2176
CSNK1D (CK1d)CK1CK14kbkBA(3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholineHuman2174
CSNK1D (CK1d)CK1CK14kbkBB(3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholineHuman2187
CSNK1D (CK1d)CK1CK14kbkCA(3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholineHuman2169
CSNK1D (CK1d)CK1CK14kbkCB(3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholineHuman2165
CSNK1D (CK1d)CK1CK14kbkDA(3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholineHuman2190
CSNK1D (CK1d)CK1CK14kbkDB(3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholineHuman2145
CSNK1D (CK1d)CK1CK14tn6AA4-{4-(4-fluorophenyl)-1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1h-imidazol-5-yl}pyrimidin-2-amineHuman2168
CSNK1D (CK1d)CK1CK14tn6AB4-{4-(4-fluorophenyl)-1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1h-imidazol-5-yl}pyrimidin-2-amineHuman2186
CSNK1D (CK1d)CK1CK14tn6BA-Human2173
CSNK1D (CK1d)CK1CK14tn6BB-Human2162
CSNK1D (CK1d)CK1CK14tw9AAoctyl beta-l-talopyranosideHuman2143
CSNK1D (CK1d)CK1CK14tw9ABoctyl beta-l-talopyranosideHuman2155
CSNK1D (CK1d)CK1CK14tw9BAn-(2,2-difluoro-5h-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-2-{[2-(trifluoromethoxy)benzoyl]amino}-1,3-thiazole-4-carboxamideHuman2178
CSNK1D (CK1d)CK1CK14tw9BBn-(2,2-difluoro-5h-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-2-{[2-(trifluoromethoxy)benzoyl]amino}-1,3-thiazole-4-carboxamideHuman2167
CSNK1D (CK1d)CK1CK14twcAA2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamideHuman2185
CSNK1D (CK1d)CK1CK14twcAB2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamideHuman2157
CSNK1D (CK1d)CK1CK14twcBA2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamideHuman2170
CSNK1D (CK1d)CK1CK14twcBB2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamideHuman2144
CSNK1D (CK1d)CK1CK15ih4AA-Human6530
CSNK1D (CK1d)CK1CK15ih4AB-Human6534
CSNK1D (CK1d)CK1CK15ih4AC-Human6529
CSNK1D (CK1d)CK1CK15ih4AD-Human6531
CSNK1D (CK1d)CK1CK15ih5AA6-(3-chlorophenyl)pteridine-2,4,7-triamineHuman6527
CSNK1D (CK1d)CK1CK15ih5AB6-(3-chlorophenyl)pteridine-2,4,7-triamineHuman6533
CSNK1D (CK1d)CK1CK15ih5AC6-(3-chlorophenyl)pteridine-2,4,7-triamineHuman6526
CSNK1D (CK1d)CK1CK15ih5AD6-(3-chlorophenyl)pteridine-2,4,7-triamineHuman6528
CSNK1D (CK1d)CK1CK15ih6AA6-(3-bromophenyl)pteridine-2,4,7-triamineHuman6535
CSNK1D (CK1d)CK1CK15ih6AB6-(3-bromophenyl)pteridine-2,4,7-triamineHuman6532
CSNK1D (CK1d)CK1CK15mqvAA4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7532
CSNK1D (CK1d)CK1CK15mqvAB4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7534
CSNK1D (CK1d)CK1CK15mqvBA4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7542
CSNK1D (CK1d)CK1CK15mqvBB4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7540
CSNK1D (CK1d)CK1CK15mqvCA4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7541
CSNK1D (CK1d)CK1CK15mqvCB4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7535
CSNK1D (CK1d)CK1CK15mqvDA4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7537
CSNK1D (CK1d)CK1CK15mqvDB4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7539
CSNK1D (CK1d)CK1CK15mqvEA4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7543
CSNK1D (CK1d)CK1CK15mqvEB4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7538
CSNK1D (CK1d)CK1CK15mqvFA4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7536
CSNK1D (CK1d)CK1CK15mqvFB4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamideHuman7533
CSNK1D (CK1d)CK1CK15oktAA~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamideHuman9862
CSNK1D (CK1d)CK1CK15oktAB~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamideHuman9861
CSNK1D (CK1d)CK1CK15oktBA~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamideHuman9860
CSNK1D (CK1d)CK1CK15oktBB~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamideHuman9857
CSNK1D (CK1d)CK1CK15oktCA~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamideHuman9858
CSNK1D (CK1d)CK1CK15oktCB~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamideHuman9859
CSNK1D (CK1d)CK1CK15oktDA~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamideHuman9855
CSNK1D (CK1d)CK1CK15oktDB~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamideHuman9856
CSNK1D (CK1d)CK1CK15w4wAA4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-oneHuman8174
CSNK1D (CK1d)CK1CK15w4wAB4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-oneHuman8177
CSNK1D (CK1d)CK1CK15w4wBA4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-oneHuman8173
CSNK1D (CK1d)CK1CK15w4wBB4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-oneHuman8179
CSNK1D (CK1d)CK1CK15w4wCA4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-oneHuman8175
CSNK1D (CK1d)CK1CK15w4wCB4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-oneHuman8178
CSNK1D (CK1d)CK1CK15w4wDA4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-oneHuman8176
CSNK1D (CK1d)CK1CK15w4wDB4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-oneHuman8180
CSNK1D (CK1d)CK1CK16f1wAA(9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10959
CSNK1D (CK1d)CK1CK16f1wAB(9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10957
CSNK1D (CK1d)CK1CK16f1wBA(9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10960
CSNK1D (CK1d)CK1CK16f1wBB(9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10961
CSNK1D (CK1d)CK1CK16f26AA(9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10955
CSNK1D (CK1d)CK1CK16f26AB(9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10953
CSNK1D (CK1d)CK1CK16f26AC(9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10954
CSNK1D (CK1d)CK1CK16f26BA(9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10958
CSNK1D (CK1d)CK1CK16f26BB(9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10956
CSNK1D (CK1d)CK1CK16f26BC(9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamideHuman10952
CSNK1D (CK1d)CK1CK16gzmAA[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHuman10426
CSNK1D (CK1d)CK1CK16gzmAB[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHuman10425
CSNK1D (CK1d)CK1CK16gzmBA[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHuman10423
CSNK1D (CK1d)CK1CK16gzmBB[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHuman10424
CSNK1D (CK1d)CK1CK16hmpAA-Human11608
CSNK1D (CK1d)CK1CK16hmpAB-Human11609
CSNK1D (CK1d)CK1CK16hmpBA-Human11607
CSNK1D (CK1d)CK1CK16hmpBB-Human11610
CSNK1D (CK1d)CK1CK16hmrAA-Human11612
CSNK1D (CK1d)CK1CK16hmrAB-Human11606
CSNK1D (CK1d)CK1CK16hmrBA-Human11605
CSNK1D (CK1d)CK1CK16hmrBB-Human11611
CSNK1D (CK1d)CK1CK16pxnAA-Human11972
CSNK1D (CK1d)CK1CK16pxnAB-Human11977
CSNK1D (CK1d)CK1CK16pxnBA-Human11969
CSNK1D (CK1d)CK1CK16pxnBB-Human11978
CSNK1D (CK1d)CK1CK16pxoAA-Human11971
CSNK1D (CK1d)CK1CK16pxoAB-Human11976
CSNK1D (CK1d)CK1CK16pxoBA-Human11974
CSNK1D (CK1d)CK1CK16pxoBB-Human11975
CSNK1D (CK1d)CK1CK16pxpA-Human11970
CSNK1D (CK1d)CK1CK16pxpB-Human11973
CSNK1D (CK1d)CK1CK16rcgAA~{n}-[[6,7-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(3-fluorophenyl)-2-morpholin-4-yl-purin-6-amineHuman12112
CSNK1D (CK1d)CK1CK16rcgAB~{n}-[[6,7-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(3-fluorophenyl)-2-morpholin-4-yl-purin-6-amineHuman12109
CSNK1D (CK1d)CK1CK16rchAA~{n}-[[4,5-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-naphthalen-2-yl-purin-6-amineHuman12108
CSNK1D (CK1d)CK1CK16rchAB~{n}-[[4,5-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-naphthalen-2-yl-purin-6-amineHuman12107
CSNK1D (CK1d)CK1CK16rchAC~{n}-[[4,5-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-naphthalen-2-yl-purin-6-amineHuman12111
CSNK1D (CK1d)CK1CK16rchBA-Human12106
CSNK1D (CK1d)CK1CK16rchBB-Human12110
CSNK1D (CK1d)CK1CK16rchBC-Human12113
CSNK1D (CK1d)CK1CK16ru6AAphosphomethylphosphonic acid adenylate esterHuman12260
CSNK1D (CK1d)CK1CK16ru6ABphosphomethylphosphonic acid adenylate esterHuman12256
CSNK1D (CK1d)CK1CK16ru6BAphosphomethylphosphonic acid adenylate esterHuman12259
CSNK1D (CK1d)CK1CK16ru6BBphosphomethylphosphonic acid adenylate esterHuman12251
CSNK1D (CK1d)CK1CK16ru7AAadenosine-5'-diphosphateHuman12264
CSNK1D (CK1d)CK1CK16ru7ABadenosine-5'-diphosphateHuman12253
CSNK1D (CK1d)CK1CK16ru7BAadenosine-5'-diphosphateHuman12252
CSNK1D (CK1d)CK1CK16ru7BBadenosine-5'-diphosphateHuman12263
CSNK1D (CK1d)CK1CK16ru8AAadenosine-5'-diphosphateHuman12258
CSNK1D (CK1d)CK1CK16ru8ABadenosine-5'-diphosphateHuman12255
CSNK1D (CK1d)CK1CK16ru8BAadenosine-5'-diphosphateHuman12265
CSNK1D (CK1d)CK1CK16ru8BBadenosine-5'-diphosphateHuman12261
CSNK1D (CK1d)CK1CK16ru8CAadenosine-5'-diphosphateHuman12266
CSNK1D (CK1d)CK1CK16ru8CBadenosine-5'-diphosphateHuman12254
CSNK1D (CK1d)CK1CK16ru8DAadenosine-5'-diphosphateHuman12262
CSNK1D (CK1d)CK1CK16ru8DBadenosine-5'-diphosphateHuman12257
CSNK1D (CK1d)CK1CK17nzyAA9-chloranyl-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amineHuman14381
CSNK1D (CK1d)CK1CK17nzyAB9-chloranyl-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amineHuman14382
CSNK1D (CK1d)CK1CK17p7fAAadenosine monophosphateHuman14188
CSNK1D (CK1d)CK1CK17p7fABadenosine monophosphateHuman14185
CSNK1D (CK1d)CK1CK17p7gAAadenosine monophosphateHuman14187
CSNK1D (CK1d)CK1CK17p7gABadenosine monophosphateHuman14186
CSNK1D (CK1d)CK1CK17p7hAadenosine monophosphateHuman14184
CSNK1D (CK1d)CK1CK17qr9AA4-[5-(4-fluorophenyl)-3-(pyridin-4-ylmethyl)imidazol-4-yl]-1~{h}-pyrrolo[2,3-b]pyridineHuman14579
CSNK1D (CK1d)CK1CK17qr9AB4-[5-(4-fluorophenyl)-3-(pyridin-4-ylmethyl)imidazol-4-yl]-1~{h}-pyrrolo[2,3-b]pyridineHuman14577
CSNK1D (CK1d)CK1CK17qraA4-[3-cyclohexyl-5-(4-fluorophenyl)imidazol-4-yl]-1~{h}-pyrrolo[2,3-b]pyridineHuman14578
CSNK1D (CK1d)CK1CK17qrbAA3-(dimethylamino)-~{n}-[4-[4-(4-fluorophenyl)-5-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)imidazol-1-yl]cyclohexyl]propane-1-sulfonamideHuman14580
CSNK1D (CK1d)CK1CK17qrbAB3-(dimethylamino)-~{n}-[4-[4-(4-fluorophenyl)-5-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)imidazol-1-yl]cyclohexyl]propane-1-sulfonamideHuman14576
CSNK1D (CK1d)CK1CK18d7mA-Human14740
CSNK1D (CK1d)CK1CK18d7nA-Human14738
CSNK1D (CK1d)CK1CK18d7oA-Human14739
CSNK1D (CK1d)CK1CK18d7pA-Human14737
CSNK1E (CK1e)CK1CK14hniA3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman1722
CSNK1E (CK1e)CK1CK14hniB3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman1731
CSNK1E (CK1e)CK1CK14hokA-Human1718
CSNK1E (CK1e)CK1CK14hokC-Human1723
CSNK1E (CK1e)CK1CK14hokE-Human1720
CSNK1E (CK1e)CK1CK14hokG-Human1719
CSNK1E (CK1e)CK1CK14hokI-Human1724
CSNK1E (CK1e)CK1CK14hokK-Human1729
CSNK1E (CK1e)CK1CK14hokM-Human1727
CSNK1E (CK1e)CK1CK14hokO-Human1726
CSNK1E (CK1e)CK1CK14hokQ-Human1730
CSNK1E (CK1e)CK1CK14hokS-Human1721
CSNK1E (CK1e)CK1CK14hokU-Human1725
CSNK1E (CK1e)CK1CK14hokW-Human1728
CSNK1G1 (CK1g1)CK1CK12cmwAA2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman5567
CSNK1G1 (CK1g1)CK1CK12cmwAB2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman5566
CSNK1G2 (CK1g2)CK1CK12c47AA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman4618
CSNK1G2 (CK1g2)CK1CK12c47AB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman4621
CSNK1G2 (CK1g2)CK1CK12c47BA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman4622
CSNK1G2 (CK1g2)CK1CK12c47BB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman4620
CSNK1G2 (CK1g2)CK1CK12c47CA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman4619
CSNK1G2 (CK1g2)CK1CK12c47CB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman4624
CSNK1G2 (CK1g2)CK1CK12c47DA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman4623
CSNK1G2 (CK1g2)CK1CK12c47DB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman4617
CSNK1G3 (CK1g3)CK1CK12chlAA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman2220
CSNK1G3 (CK1g3)CK1CK12chlAB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman2217
CSNK1G3 (CK1g3)CK1CK12izrAA{(2z)-4-amino-2-[(4-methoxyphenyl)imino]-2,3-dihydro-1,3-thiazol-5-yl}(4-methoxyphenyl)methanoneHuman2222
CSNK1G3 (CK1g3)CK1CK12izrAB{(2z)-4-amino-2-[(4-methoxyphenyl)imino]-2,3-dihydro-1,3-thiazol-5-yl}(4-methoxyphenyl)methanoneHuman2221
CSNK1G3 (CK1g3)CK1CK12izsAA{[4-amino-2-(3-chloroanilino)-1,3-thiazol-5-yl](4-fluorophenyl)methanoneHuman2228
CSNK1G3 (CK1g3)CK1CK12izsAB{[4-amino-2-(3-chloroanilino)-1,3-thiazol-5-yl](4-fluorophenyl)methanoneHuman2223
CSNK1G3 (CK1g3)CK1CK12iztAAn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman2216
CSNK1G3 (CK1g3)CK1CK12iztABn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman2215
CSNK1G3 (CK1g3)CK1CK12izuAA2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHuman2218
CSNK1G3 (CK1g3)CK1CK12izuAB2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHuman2225
CSNK1G3 (CK1g3)CK1CK14g16A2-[(4-{[3-(trifluoromethyl)pyridin-2-yl]oxy}phenyl)amino]-1h-benzimidazole-6-carbonitrileHuman2219
CSNK1G3 (CK1g3)CK1CK14g17A2-[(4-tert-butylphenyl)amino]-1h-benzimidazole-6-carbonitrileHuman2226
CSNK1G3 (CK1g3)CK1CK14hglA2-[5-methoxy-2-(quinolin-3-yl)pyrimidin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman2227
CSNK1G3 (CK1g3)CK1CK14hgsA2-{2-[(3,4-difluorophenoxy)methyl]-5-methoxypyridin-4-yl}-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman2224
CSNK1G3 (CK1g3)CK1CK16groAA4-[5-(2-azanylpyrimidin-4-yl)-4-(4-fluorophenyl)imidazol-1-yl]cyclohexan-1-olHuman10002
CSNK1G3 (CK1g3)CK1CK16groAB4-[5-(2-azanylpyrimidin-4-yl)-4-(4-fluorophenyl)imidazol-1-yl]cyclohexan-1-olHuman10003
CSNK2A1 (CK2a1)CK2CMGC1jwhAphosphoaminophosphonic acid-adenylate esterHuman5485
CSNK2A1 (CK2a1)CK2CMGC1jwhB-Human5524
CSNK2A1 (CK2a1)CK2CMGC1na7A-Human5533
CSNK2A1 (CK2a1)CK2CMGC1pjkAAphosphoaminophosphonic acid-adenylate esterHuman5494
CSNK2A1 (CK2a1)CK2CMGC1pjkABphosphoaminophosphonic acid-adenylate esterHuman5410
CSNK2A1 (CK2a1)CK2CMGC2pvrAAphosphoaminophosphonic acid-adenylate esterHuman5509
CSNK2A1 (CK2a1)CK2CMGC2pvrABphosphoaminophosphonic acid-adenylate esterHuman5505
CSNK2A1 (CK2a1)CK2CMGC2zjwA2,3,7,8-tetrahydroxychromeno[5,4,3-cde]chromene-5,10-dioneHuman5423
CSNK2A1 (CK2a1)CK2CMGC3amyA5,7-dihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman5506
CSNK2A1 (CK2a1)CK2CMGC3at2AA-Human5428
CSNK2A1 (CK2a1)CK2CMGC3at2AB-Human5492
CSNK2A1 (CK2a1)CK2CMGC3at3A(1-{6-[6-(cyclopentylamino)-1h-indazol-1-yl]pyrazin-2-yl}-1h-pyrrol-3-yl)acetic acidHuman5504
CSNK2A1 (CK2a1)CK2CMGC3at4A[1-(6-{6-[(1-methylethyl)amino]-1h-indazol-1-yl}pyrazin-2-yl)-1h-pyrrol-3-yl]acetic acidHuman5413
CSNK2A1 (CK2a1)CK2CMGC3axwA4-(5-amino-1,3,4-thiadiazol-2-yl)benzoic acidHuman5440
CSNK2A1 (CK2a1)CK2CMGC3bqcAA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5486
CSNK2A1 (CK2a1)CK2CMGC3bqcAB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5490
CSNK2A1 (CK2a1)CK2CMGC3c13AA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5530
CSNK2A1 (CK2a1)CK2CMGC3c13AB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5472
CSNK2A1 (CK2a1)CK2CMGC3fwqA-Human5507
CSNK2A1 (CK2a1)CK2CMGC3fwqB-Human5479
CSNK2A1 (CK2a1)CK2CMGC3h30AA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman5496
CSNK2A1 (CK2a1)CK2CMGC3h30AB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman5460
CSNK2A1 (CK2a1)CK2CMGC3h30BA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman5484
CSNK2A1 (CK2a1)CK2CMGC3h30BB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman5480
CSNK2A1 (CK2a1)CK2CMGC3juhAAphosphoaminophosphonic acid-adenylate esterHuman5471
CSNK2A1 (CK2a1)CK2CMGC3juhABphosphoaminophosphonic acid-adenylate esterHuman5456
CSNK2A1 (CK2a1)CK2CMGC3juhBAphosphoaminophosphonic acid-adenylate esterHuman5431
CSNK2A1 (CK2a1)CK2CMGC3juhBBphosphoaminophosphonic acid-adenylate esterHuman5421
CSNK2A1 (CK2a1)CK2CMGC3mb6AAnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman5424
CSNK2A1 (CK2a1)CK2CMGC3mb6ABnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman5499
CSNK2A1 (CK2a1)CK2CMGC3mb6ACnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman5529
CSNK2A1 (CK2a1)CK2CMGC3mb7AAnaphtho[2,1-b:7,8-b']difuran-2,9-dicarboxylic acidHuman5448
CSNK2A1 (CK2a1)CK2CMGC3mb7ABnaphtho[2,1-b:7,8-b']difuran-2,9-dicarboxylic acidHuman5455
CSNK2A1 (CK2a1)CK2CMGC3ngaAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5422
CSNK2A1 (CK2a1)CK2CMGC3ngaAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5515
CSNK2A1 (CK2a1)CK2CMGC3ngaBA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5441
CSNK2A1 (CK2a1)CK2CMGC3ngaBB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5511
CSNK2A1 (CK2a1)CK2CMGC3nszAAphosphoaminophosphonic acid-adenylate esterHuman5512
CSNK2A1 (CK2a1)CK2CMGC3nszABphosphoaminophosphonic acid-adenylate esterHuman5503
CSNK2A1 (CK2a1)CK2CMGC3owjAA9-hydroxy-5,11-dimethyl-4,6-dihydro-1h-pyrido[4,3-b]carbazol-1-oneHuman5452
CSNK2A1 (CK2a1)CK2CMGC3owjAB9-hydroxy-5,11-dimethyl-4,6-dihydro-1h-pyrido[4,3-b]carbazol-1-oneHuman5470
CSNK2A1 (CK2a1)CK2CMGC3owkAA7-chloro-10-methyl-11h-benzo[g]pyrido[4,3-b]indol-3-olHuman5467
CSNK2A1 (CK2a1)CK2CMGC3owkAB7-chloro-10-methyl-11h-benzo[g]pyrido[4,3-b]indol-3-olHuman5433
CSNK2A1 (CK2a1)CK2CMGC3owlAA11-chloro-8-methyl-7h-benzo[e]pyrido[4,3-b]indol-3-olHuman5502
CSNK2A1 (CK2a1)CK2CMGC3owlAB11-chloro-8-methyl-7h-benzo[e]pyrido[4,3-b]indol-3-olHuman5416
CSNK2A1 (CK2a1)CK2CMGC3pe1AA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5487
CSNK2A1 (CK2a1)CK2CMGC3pe1AB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5500
CSNK2A1 (CK2a1)CK2CMGC3pe2AA5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acidHuman5508
CSNK2A1 (CK2a1)CK2CMGC3pe2AB5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acidHuman5519
CSNK2A1 (CK2a1)CK2CMGC3q04AA-Human5514
CSNK2A1 (CK2a1)CK2CMGC3q04AB-Human5419
CSNK2A1 (CK2a1)CK2CMGC3q9wAA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5436
CSNK2A1 (CK2a1)CK2CMGC3q9wAB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5420
CSNK2A1 (CK2a1)CK2CMGC3q9xAA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5446
CSNK2A1 (CK2a1)CK2CMGC3q9xAB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5488
CSNK2A1 (CK2a1)CK2CMGC3q9xBA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5516
CSNK2A1 (CK2a1)CK2CMGC3q9xBB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5417
CSNK2A1 (CK2a1)CK2CMGC3q9yAA1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5493
CSNK2A1 (CK2a1)CK2CMGC3q9yAB1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5526
CSNK2A1 (CK2a1)CK2CMGC3q9zAA1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5510
CSNK2A1 (CK2a1)CK2CMGC3q9zAB1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5437
CSNK2A1 (CK2a1)CK2CMGC3q9zBA1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5426
CSNK2A1 (CK2a1)CK2CMGC3q9zBB1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5430
CSNK2A1 (CK2a1)CK2CMGC3qa0AA-Human5425
CSNK2A1 (CK2a1)CK2CMGC3qa0AB-Human5451
CSNK2A1 (CK2a1)CK2CMGC3qa0BA-Human5495
CSNK2A1 (CK2a1)CK2CMGC3qa0BB-Human5528
CSNK2A1 (CK2a1)CK2CMGC3r0tAA3-(cyclopropylamino)-5-{[3-(trifluoromethyl)phenyl]amino}pyrimido[4,5-c]quinoline-8-carboxylic acidHuman5497
CSNK2A1 (CK2a1)CK2CMGC3r0tAB3-(cyclopropylamino)-5-{[3-(trifluoromethyl)phenyl]amino}pyrimido[4,5-c]quinoline-8-carboxylic acidHuman5517
CSNK2A1 (CK2a1)CK2CMGC3rpsA3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman5463
CSNK2A1 (CK2a1)CK2CMGC3rpsB-Human5450
CSNK2A1 (CK2a1)CK2CMGC3u4uA3-{5-(acetylamino)-3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1h-indol-1-yl}propanoic acidHuman5527
CSNK2A1 (CK2a1)CK2CMGC3u87Aphosphoaminophosphonic acid-adenylate esterHuman5442
CSNK2A1 (CK2a1)CK2CMGC3u87Bphosphoaminophosphonic acid-adenylate esterHuman5513
CSNK2A1 (CK2a1)CK2CMGC3u9cA7-hydroxy-3h-phenoxazin-3-oneHuman5461
CSNK2A1 (CK2a1)CK2CMGC3u9cB7-hydroxy-3h-phenoxazin-3-oneHuman5523
CSNK2A1 (CK2a1)CK2CMGC3w8lA-Human5427
CSNK2A1 (CK2a1)CK2CMGC3w8lB-Human5469
CSNK2A1 (CK2a1)CK2CMGC3warAAnicotinic acidHuman5429
CSNK2A1 (CK2a1)CK2CMGC3warABnicotinic acidHuman5464
CSNK2A1 (CK2a1)CK2CMGC3wikAn-[5-(4-nitrophenyl)-1,3,4-thiadiazol-2-yl]acetamideHuman5459
CSNK2A1 (CK2a1)CK2CMGC3wilA{[(2z)-2-(3,4-dimethoxybenzylidene)-3-oxo-2,3-dihydro-1-benzofuran-6-yl]oxy}acetic acidHuman5468
CSNK2A1 (CK2a1)CK2CMGC3wowAphosphoaminophosphonic acid-adenylate esterHuman5445
CSNK2A1 (CK2a1)CK2CMGC4dglC-Human5474
CSNK2A1 (CK2a1)CK2CMGC4dglD-Human5521
CSNK2A1 (CK2a1)CK2CMGC4fbxA-Human5415
CSNK2A1 (CK2a1)CK2CMGC4grbA5-(2-{[4-(dimethylcarbamoyl)phenyl]amino}-4-methoxypyrimidin-5-yl)thiophene-3-carboxylic acidHuman5443
CSNK2A1 (CK2a1)CK2CMGC4gubAn-[5-({3-cyano-7-[(1-methyl-1h-imidazol-4-yl)amino]pyrazolo[1,5-a]pyrimidin-5-yl}amino)-2-methylphenyl]acetamideHuman5491
CSNK2A1 (CK2a1)CK2CMGC4ib5AA-Human5501
CSNK2A1 (CK2a1)CK2CMGC4ib5AB-Human5522
CSNK2A1 (CK2a1)CK2CMGC4ib5BA-Human5532
CSNK2A1 (CK2a1)CK2CMGC4ib5BB-Human5438
CSNK2A1 (CK2a1)CK2CMGC4ib5CA-Human5498
CSNK2A1 (CK2a1)CK2CMGC4ib5CB-Human5476
CSNK2A1 (CK2a1)CK2CMGC4kwpAA4,5,6,7-tetrabromo-1-(2-deoxy-beta-d-erythro-pentofuranosyl)-1h-benzimidazoleHuman5465
CSNK2A1 (CK2a1)CK2CMGC4kwpAB4,5,6,7-tetrabromo-1-(2-deoxy-beta-d-erythro-pentofuranosyl)-1h-benzimidazoleHuman5482
CSNK2A1 (CK2a1)CK2CMGC4md7E-Human5435
CSNK2A1 (CK2a1)CK2CMGC4md7F-Human5457
CSNK2A1 (CK2a1)CK2CMGC4md7G-Human5409
CSNK2A1 (CK2a1)CK2CMGC4md7H-Human5481
CSNK2A1 (CK2a1)CK2CMGC4md8E-Human5439
CSNK2A1 (CK2a1)CK2CMGC4md8F-Human5475
CSNK2A1 (CK2a1)CK2CMGC4md8G-Human5478
CSNK2A1 (CK2a1)CK2CMGC4md8H-Human5518
CSNK2A1 (CK2a1)CK2CMGC4md9E-Human5411
CSNK2A1 (CK2a1)CK2CMGC4md9F-Human5473
CSNK2A1 (CK2a1)CK2CMGC4md9G-Human5483
CSNK2A1 (CK2a1)CK2CMGC4md9H-Human5466
CSNK2A1 (CK2a1)CK2CMGC4md9K-Human5477
CSNK2A1 (CK2a1)CK2CMGC4md9L-Human5414
CSNK2A1 (CK2a1)CK2CMGC4md9M-Human5520
CSNK2A1 (CK2a1)CK2CMGC4md9P-Human5434
CSNK2A1 (CK2a1)CK2CMGC4nh1Aphosphomethylphosphonic acid adenylate esterHuman5412
CSNK2A1 (CK2a1)CK2CMGC4nh1Bphosphomethylphosphonic acid adenylate esterHuman5531
CSNK2A1 (CK2a1)CK2CMGC4rllAA4-[(e)-(9h-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acidHuman5418
CSNK2A1 (CK2a1)CK2CMGC4rllAB4-[(e)-(9h-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acidHuman5449
CSNK2A1 (CK2a1)CK2CMGC4ub7A4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acidHuman5462
CSNK2A1 (CK2a1)CK2CMGC4ubaA4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acidHuman5432
CSNK2A1 (CK2a1)CK2CMGC4ubaB4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acidHuman5525
CSNK2A1 (CK2a1)CK2CMGC5b0xA4-[2-[(4-methoxyphenyl)carbonylamino]-1,3-thiazol-5-yl]benzoic acidHuman6475
CSNK2A1 (CK2a1)CK2CMGC5clpAA2-(3,4-dichlorophenyl)ethanamineHuman6922
CSNK2A1 (CK2a1)CK2CMGC5clpAB2-(3,4-dichlorophenyl)ethanamineHuman6920
CSNK2A1 (CK2a1)CK2CMGC5clpBA2-(3,4-dichlorophenyl)ethanamineHuman6909
CSNK2A1 (CK2a1)CK2CMGC5clpBB2-(3,4-dichlorophenyl)ethanamineHuman6911
CSNK2A1 (CK2a1)CK2CMGC5cquAA4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6035
CSNK2A1 (CK2a1)CK2CMGC5cquAB4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6038
CSNK2A1 (CK2a1)CK2CMGC5cqwAA4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6034
CSNK2A1 (CK2a1)CK2CMGC5cqwAB4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6037
CSNK2A1 (CK2a1)CK2CMGC5cqwBA4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6039
CSNK2A1 (CK2a1)CK2CMGC5cqwBB4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6036
CSNK2A1 (CK2a1)CK2CMGC5cs6AA-Human6915
CSNK2A1 (CK2a1)CK2CMGC5cs6AB-Human6901
CSNK2A1 (CK2a1)CK2CMGC5cs6BA-Human6919
CSNK2A1 (CK2a1)CK2CMGC5cs6BB-Human6926
CSNK2A1 (CK2a1)CK2CMGC5cshAAadenosine-5'-triphosphateHuman6918
CSNK2A1 (CK2a1)CK2CMGC5cshABadenosine-5'-triphosphateHuman6925
CSNK2A1 (CK2a1)CK2CMGC5cshBAadenosine-5'-triphosphateHuman6923
CSNK2A1 (CK2a1)CK2CMGC5cshBBadenosine-5'-triphosphateHuman6907
CSNK2A1 (CK2a1)CK2CMGC5cspAA2-hydroxy-5-methylbenzoic acidHuman6904
CSNK2A1 (CK2a1)CK2CMGC5cspAB2-hydroxy-5-methylbenzoic acidHuman6905
CSNK2A1 (CK2a1)CK2CMGC5cspAC2-hydroxy-5-methylbenzoic acidHuman6928
CSNK2A1 (CK2a1)CK2CMGC5csvAA3-aminobenzoic acidHuman6898
CSNK2A1 (CK2a1)CK2CMGC5csvAB3-aminobenzoic acidHuman6900
CSNK2A1 (CK2a1)CK2CMGC5ct0AA3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-olHuman7296
CSNK2A1 (CK2a1)CK2CMGC5ct0AB3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-olHuman7300
CSNK2A1 (CK2a1)CK2CMGC5ct0BA3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-olHuman7288
CSNK2A1 (CK2a1)CK2CMGC5ct0BB3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-olHuman7298
CSNK2A1 (CK2a1)CK2CMGC5ctpAAn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7304
CSNK2A1 (CK2a1)CK2CMGC5ctpABn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7289
CSNK2A1 (CK2a1)CK2CMGC5ctpBAn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7297
CSNK2A1 (CK2a1)CK2CMGC5ctpBBn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7291
CSNK2A1 (CK2a1)CK2CMGC5cu0AAn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7299
CSNK2A1 (CK2a1)CK2CMGC5cu0ABn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7293
CSNK2A1 (CK2a1)CK2CMGC5cu0BAn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7295
CSNK2A1 (CK2a1)CK2CMGC5cu0BBn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7301
CSNK2A1 (CK2a1)CK2CMGC5cu2AAmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7303
CSNK2A1 (CK2a1)CK2CMGC5cu2ABmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7302
CSNK2A1 (CK2a1)CK2CMGC5cu2BAmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7292
CSNK2A1 (CK2a1)CK2CMGC5cu2BBmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7286
CSNK2A1 (CK2a1)CK2CMGC5cu3AAn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6902
CSNK2A1 (CK2a1)CK2CMGC5cu3ABn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6903
CSNK2A1 (CK2a1)CK2CMGC5cu3BAn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6921
CSNK2A1 (CK2a1)CK2CMGC5cu3BBn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6897
CSNK2A1 (CK2a1)CK2CMGC5cu4AAn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6924
CSNK2A1 (CK2a1)CK2CMGC5cu4ABn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6895
CSNK2A1 (CK2a1)CK2CMGC5cu4ACn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6916
CSNK2A1 (CK2a1)CK2CMGC5cu6AAadenosine-5'-triphosphateHuman6899
CSNK2A1 (CK2a1)CK2CMGC5cu6ABadenosine-5'-triphosphateHuman6906
CSNK2A1 (CK2a1)CK2CMGC5cvfAAadenosine-5'-triphosphateHuman6927
CSNK2A1 (CK2a1)CK2CMGC5cvfABadenosine-5'-triphosphateHuman6910
CSNK2A1 (CK2a1)CK2CMGC5cvgAA-Human6913
CSNK2A1 (CK2a1)CK2CMGC5cvgAB-Human6908
CSNK2A1 (CK2a1)CK2CMGC5cvhAAadenosine-5'-diphosphateHuman6896
CSNK2A1 (CK2a1)CK2CMGC5cvhABadenosine-5'-diphosphateHuman6912
CSNK2A1 (CK2a1)CK2CMGC5cvhBAadenosine-5'-diphosphateHuman6914
CSNK2A1 (CK2a1)CK2CMGC5cvhBBadenosine-5'-diphosphateHuman6917
CSNK2A1 (CK2a1)CK2CMGC5cx9AAmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7287
CSNK2A1 (CK2a1)CK2CMGC5cx9ABmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7290
CSNK2A1 (CK2a1)CK2CMGC5cx9BAmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7285
CSNK2A1 (CK2a1)CK2CMGC5cx9BBmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7294
CSNK2A1 (CK2a1)CK2CMGC5h8bA~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman6408
CSNK2A1 (CK2a1)CK2CMGC5h8bB~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman6406
CSNK2A1 (CK2a1)CK2CMGC5h8eA~{n}-[2-[2-azanylethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman6409
CSNK2A1 (CK2a1)CK2CMGC5h8eB~{n}-[2-[2-azanylethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman6407
CSNK2A1 (CK2a1)CK2CMGC5h8gA~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]ethanamideHuman6405
CSNK2A1 (CK2a1)CK2CMGC5ku8A~{n}-[2-[(1~{s},2~{s})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman8664
CSNK2A1 (CK2a1)CK2CMGC5ku8B~{n}-[2-[(1~{s},2~{s})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman8663
CSNK2A1 (CK2a1)CK2CMGC5kwhAA~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman8617
CSNK2A1 (CK2a1)CK2CMGC5kwhAB~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman8619
CSNK2A1 (CK2a1)CK2CMGC5kwhBA~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman8618
CSNK2A1 (CK2a1)CK2CMGC5kwhBB~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman8620
CSNK2A1 (CK2a1)CK2CMGC5m44A3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acidHuman7404
CSNK2A1 (CK2a1)CK2CMGC5m4cAA3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acidHuman7402
CSNK2A1 (CK2a1)CK2CMGC5m4cAB3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acidHuman7403
CSNK2A1 (CK2a1)CK2CMGC5m4fAA4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7405
CSNK2A1 (CK2a1)CK2CMGC5m4fAB4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7401
CSNK2A1 (CK2a1)CK2CMGC5m4iA4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7400
CSNK2A1 (CK2a1)CK2CMGC5mmfAA(3-chloranyl-4-phenyl-phenyl)methyl-propyl-azaniumHuman7682
CSNK2A1 (CK2a1)CK2CMGC5mmfAB(3-chloranyl-4-phenyl-phenyl)methyl-propyl-azaniumHuman7666
CSNK2A1 (CK2a1)CK2CMGC5mmfBA-Human7696
CSNK2A1 (CK2a1)CK2CMGC5mmfBB-Human7657
CSNK2A1 (CK2a1)CK2CMGC5mmrAA~{n}'-[(3-chloranyl-4-phenyl-phenyl)methyl]butane-1,4-diamineHuman7668
CSNK2A1 (CK2a1)CK2CMGC5mmrAB~{n}'-[(3-chloranyl-4-phenyl-phenyl)methyl]butane-1,4-diamineHuman7659
CSNK2A1 (CK2a1)CK2CMGC5mmrBA-Human7651
CSNK2A1 (CK2a1)CK2CMGC5mmrBB-Human7680
CSNK2A1 (CK2a1)CK2CMGC5mo5AA~{n}-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propyl]methanesulfonamideHuman7676
CSNK2A1 (CK2a1)CK2CMGC5mo5AB~{n}-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propyl]methanesulfonamideHuman7661
CSNK2A1 (CK2a1)CK2CMGC5mo5BA-Human7689
CSNK2A1 (CK2a1)CK2CMGC5mo5BB-Human7656
CSNK2A1 (CK2a1)CK2CMGC5mo6AA3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoic acidHuman7672
CSNK2A1 (CK2a1)CK2CMGC5mo6AB3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoic acidHuman7665
CSNK2A1 (CK2a1)CK2CMGC5mo6BA-Human7664
CSNK2A1 (CK2a1)CK2CMGC5mo6BB-Human7652
CSNK2A1 (CK2a1)CK2CMGC5mo7AA3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanamideHuman7669
CSNK2A1 (CK2a1)CK2CMGC5mo7AB3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanamideHuman7697
CSNK2A1 (CK2a1)CK2CMGC5mo7BA-Human7698
CSNK2A1 (CK2a1)CK2CMGC5mo7BB-Human7685
CSNK2A1 (CK2a1)CK2CMGC5mo8AA3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acidHuman7653
CSNK2A1 (CK2a1)CK2CMGC5mo8AB3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acidHuman7673
CSNK2A1 (CK2a1)CK2CMGC5mo8BA3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acidHuman7654
CSNK2A1 (CK2a1)CK2CMGC5mo8BB3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acidHuman7688
CSNK2A1 (CK2a1)CK2CMGC5modAA-Human7678
CSNK2A1 (CK2a1)CK2CMGC5modAB-Human7667
CSNK2A1 (CK2a1)CK2CMGC5modBA-Human7679
CSNK2A1 (CK2a1)CK2CMGC5modBB-Human7694
CSNK2A1 (CK2a1)CK2CMGC5moeAAadenosine-5'-diphosphateHuman7650
CSNK2A1 (CK2a1)CK2CMGC5moeABadenosine-5'-diphosphateHuman7662
CSNK2A1 (CK2a1)CK2CMGC5moeBAadenosine-5'-diphosphateHuman7693
CSNK2A1 (CK2a1)CK2CMGC5moeBBadenosine-5'-diphosphateHuman7687
CSNK2A1 (CK2a1)CK2CMGC5mohAA2-(3-methoxy-4-oxidanyl-phenyl)ethanoic acidHuman7658
CSNK2A1 (CK2a1)CK2CMGC5mohAB2-(3-methoxy-4-oxidanyl-phenyl)ethanoic acidHuman7681
CSNK2A1 (CK2a1)CK2CMGC5motAA4-hydroxybenzamideHuman7660
CSNK2A1 (CK2a1)CK2CMGC5motAB4-hydroxybenzamideHuman7691
CSNK2A1 (CK2a1)CK2CMGC5movAA4'-hydroxycinnamic acidHuman7655
CSNK2A1 (CK2a1)CK2CMGC5movAB4'-hydroxycinnamic acidHuman7674
CSNK2A1 (CK2a1)CK2CMGC5mowAA5-bromopyridine-2,3-diamineHuman7670
CSNK2A1 (CK2a1)CK2CMGC5mowAB5-bromopyridine-2,3-diamineHuman7684
CSNK2A1 (CK2a1)CK2CMGC5mowBA-Human7671
CSNK2A1 (CK2a1)CK2CMGC5mowBB-Human7686
CSNK2A1 (CK2a1)CK2CMGC5mp8AAadenosine-5'-diphosphateHuman7690
CSNK2A1 (CK2a1)CK2CMGC5mp8ABadenosine-5'-diphosphateHuman7649
CSNK2A1 (CK2a1)CK2CMGC5mp8BAadenosine-5'-diphosphateHuman7695
CSNK2A1 (CK2a1)CK2CMGC5mp8BBadenosine-5'-diphosphateHuman7692
CSNK2A1 (CK2a1)CK2CMGC5mpjAAadenosine-5'-diphosphateHuman7677
CSNK2A1 (CK2a1)CK2CMGC5mpjABadenosine-5'-diphosphateHuman7663
CSNK2A1 (CK2a1)CK2CMGC5mpjBA-Human7675
CSNK2A1 (CK2a1)CK2CMGC5mpjBB-Human7683
CSNK2A1 (CK2a1)CK2CMGC5n1vAApyrazolo-pyrimidine macrocycleHuman7588
CSNK2A1 (CK2a1)CK2CMGC5n1vABpyrazolo-pyrimidine macrocycleHuman7589
CSNK2A1 (CK2a1)CK2CMGC5n1vBApyrazolo-pyrimidine macrocycleHuman7587
CSNK2A1 (CK2a1)CK2CMGC5n1vBBpyrazolo-pyrimidine macrocycleHuman7586
CSNK2A1 (CK2a1)CK2CMGC5n9kAA1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diolHuman9682
CSNK2A1 (CK2a1)CK2CMGC5n9kAB1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diolHuman9695
CSNK2A1 (CK2a1)CK2CMGC5n9lAA(4~{z})-6,7-bis(chloranyl)-4-[[(4-methylphenyl)amino]methylidene]-8-oxidanyl-1,2-dihydrodibenzofuran-3-oneHuman9652
CSNK2A1 (CK2a1)CK2CMGC5n9lAB(4~{z})-6,7-bis(chloranyl)-4-[[(4-methylphenyl)amino]methylidene]-8-oxidanyl-1,2-dihydrodibenzofuran-3-oneHuman9621
CSNK2A1 (CK2a1)CK2CMGC5n9nAA1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diolHuman9661
CSNK2A1 (CK2a1)CK2CMGC5n9nAB1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diolHuman9628
CSNK2A1 (CK2a1)CK2CMGC5nqcAA(3e)-6,7-dichloro-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-oneHuman8112
CSNK2A1 (CK2a1)CK2CMGC5nqcAB(3e)-6,7-dichloro-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-oneHuman8111
CSNK2A1 (CK2a1)CK2CMGC5omyAA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9457
CSNK2A1 (CK2a1)CK2CMGC5omyAB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9456
CSNK2A1 (CK2a1)CK2CMGC5oniAA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9455
CSNK2A1 (CK2a1)CK2CMGC5oniAB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9459
CSNK2A1 (CK2a1)CK2CMGC5oniBA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9458
CSNK2A1 (CK2a1)CK2CMGC5oniBB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9454
CSNK2A1 (CK2a1)CK2CMGC5oquAAadenosine-5'-diphosphateHuman9615
CSNK2A1 (CK2a1)CK2CMGC5oquABadenosine-5'-diphosphateHuman9627
CSNK2A1 (CK2a1)CK2CMGC5oquBAadenosine-5'-diphosphateHuman9623
CSNK2A1 (CK2a1)CK2CMGC5oquBBadenosine-5'-diphosphateHuman9678
CSNK2A1 (CK2a1)CK2CMGC5orhAA-Human9620
CSNK2A1 (CK2a1)CK2CMGC5orhAB-Human9671
CSNK2A1 (CK2a1)CK2CMGC5orhBA-Human9694
CSNK2A1 (CK2a1)CK2CMGC5orhBB-Human9639
CSNK2A1 (CK2a1)CK2CMGC5orjAAadenosine-5'-diphosphateHuman9653
CSNK2A1 (CK2a1)CK2CMGC5orjABadenosine-5'-diphosphateHuman9624
CSNK2A1 (CK2a1)CK2CMGC5orjBAadenosine-5'-diphosphateHuman9607
CSNK2A1 (CK2a1)CK2CMGC5orjBBadenosine-5'-diphosphateHuman9665
CSNK2A1 (CK2a1)CK2CMGC5orkAAadenosine-5'-diphosphateHuman9693
CSNK2A1 (CK2a1)CK2CMGC5orkABadenosine-5'-diphosphateHuman9655
CSNK2A1 (CK2a1)CK2CMGC5orkBAadenosine-5'-diphosphateHuman9674
CSNK2A1 (CK2a1)CK2CMGC5orkBBadenosine-5'-diphosphateHuman9646
CSNK2A1 (CK2a1)CK2CMGC5os7AAadenosine-5'-triphosphateHuman9644
CSNK2A1 (CK2a1)CK2CMGC5os7ABadenosine-5'-triphosphateHuman9609
CSNK2A1 (CK2a1)CK2CMGC5os7BAadenosine-5'-triphosphateHuman9626
CSNK2A1 (CK2a1)CK2CMGC5os7BBadenosine-5'-triphosphateHuman9645
CSNK2A1 (CK2a1)CK2CMGC5os8AAadenosine-5'-triphosphateHuman9608
CSNK2A1 (CK2a1)CK2CMGC5os8ABadenosine-5'-triphosphateHuman9666
CSNK2A1 (CK2a1)CK2CMGC5oslAAadenosine-5'-diphosphateHuman9673
CSNK2A1 (CK2a1)CK2CMGC5oslABadenosine-5'-diphosphateHuman9629
CSNK2A1 (CK2a1)CK2CMGC5ospAAadenosine-5'-triphosphateHuman10587
CSNK2A1 (CK2a1)CK2CMGC5ospABadenosine-5'-triphosphateHuman10600
CSNK2A1 (CK2a1)CK2CMGC5osrAAadenosine-5'-triphosphateHuman10601
CSNK2A1 (CK2a1)CK2CMGC5osrABadenosine-5'-triphosphateHuman10594
CSNK2A1 (CK2a1)CK2CMGC5osuAA-Human10595
CSNK2A1 (CK2a1)CK2CMGC5osuAB-Human10598
CSNK2A1 (CK2a1)CK2CMGC5oszAA2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azaniumHuman9669
CSNK2A1 (CK2a1)CK2CMGC5oszAB2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azaniumHuman9685
CSNK2A1 (CK2a1)CK2CMGC5oszAC2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azaniumHuman9683
CSNK2A1 (CK2a1)CK2CMGC5ot5AA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9656
CSNK2A1 (CK2a1)CK2CMGC5ot5AB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9676
CSNK2A1 (CK2a1)CK2CMGC5ot5BA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9689
CSNK2A1 (CK2a1)CK2CMGC5ot5BB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9605
CSNK2A1 (CK2a1)CK2CMGC5ot6AA(3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-pyrrol-2-yl)ethyl]azaniumHuman9619
CSNK2A1 (CK2a1)CK2CMGC5ot6AB(3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-pyrrol-2-yl)ethyl]azaniumHuman9643
CSNK2A1 (CK2a1)CK2CMGC5ot6BA-Human9613
CSNK2A1 (CK2a1)CK2CMGC5ot6BB-Human9649
CSNK2A1 (CK2a1)CK2CMGC5otdAA[2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azaniumHuman9697
CSNK2A1 (CK2a1)CK2CMGC5otdAB[2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azaniumHuman9696
CSNK2A1 (CK2a1)CK2CMGC5otdBA[2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azaniumHuman9690
CSNK2A1 (CK2a1)CK2CMGC5otdBB[2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azaniumHuman9632
CSNK2A1 (CK2a1)CK2CMGC5othAA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9612
CSNK2A1 (CK2a1)CK2CMGC5othAB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9659
CSNK2A1 (CK2a1)CK2CMGC5othBA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9625
CSNK2A1 (CK2a1)CK2CMGC5othBB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9670
CSNK2A1 (CK2a1)CK2CMGC5otiAA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9672
CSNK2A1 (CK2a1)CK2CMGC5otiAB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9667
CSNK2A1 (CK2a1)CK2CMGC5otlAA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9681
CSNK2A1 (CK2a1)CK2CMGC5otlAB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9633
CSNK2A1 (CK2a1)CK2CMGC5otlBA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9660
CSNK2A1 (CK2a1)CK2CMGC5otlBB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9616
CSNK2A1 (CK2a1)CK2CMGC5otoAA2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9648
CSNK2A1 (CK2a1)CK2CMGC5otoAB2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9637
CSNK2A1 (CK2a1)CK2CMGC5otoBA2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9688
CSNK2A1 (CK2a1)CK2CMGC5otoBB2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9611
CSNK2A1 (CK2a1)CK2CMGC5otpAA2-[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman10588
CSNK2A1 (CK2a1)CK2CMGC5otpAB2-[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman10586
CSNK2A1 (CK2a1)CK2CMGC5otpBA-Human10602
CSNK2A1 (CK2a1)CK2CMGC5otpBB-Human10591
CSNK2A1 (CK2a1)CK2CMGC5otqAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methoxy-phenyl]methyl]ethanamineHuman9638
CSNK2A1 (CK2a1)CK2CMGC5otqAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methoxy-phenyl]methyl]ethanamineHuman9651
CSNK2A1 (CK2a1)CK2CMGC5otrAAadenosine-5'-triphosphateHuman9640
CSNK2A1 (CK2a1)CK2CMGC5otrABadenosine-5'-triphosphateHuman9634
CSNK2A1 (CK2a1)CK2CMGC5otsAA2-(1~{h}-benzimidazol-2-yl)ethyl-[[3,5-bis(chloranyl)-4-phenyl-phenyl]methyl]azaniumHuman10589
CSNK2A1 (CK2a1)CK2CMGC5otsAB2-(1~{h}-benzimidazol-2-yl)ethyl-[[3,5-bis(chloranyl)-4-phenyl-phenyl]methyl]azaniumHuman10599
CSNK2A1 (CK2a1)CK2CMGC5otyAAtrifluoroacetic acidHuman9692
CSNK2A1 (CK2a1)CK2CMGC5otyABtrifluoroacetic acidHuman9680
CSNK2A1 (CK2a1)CK2CMGC5otzAAtrifluoroacetic acidHuman9650
CSNK2A1 (CK2a1)CK2CMGC5otzABtrifluoroacetic acidHuman9618
CSNK2A1 (CK2a1)CK2CMGC5oueAA3-methyl-5-oxidanyl-benzoic acidHuman9686
CSNK2A1 (CK2a1)CK2CMGC5oueAB3-methyl-5-oxidanyl-benzoic acidHuman9614
CSNK2A1 (CK2a1)CK2CMGC5oueBA(3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-imidazol-4-yl)ethyl]azaniumHuman9635
CSNK2A1 (CK2a1)CK2CMGC5oueBB(3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-imidazol-4-yl)ethyl]azaniumHuman9631
CSNK2A1 (CK2a1)CK2CMGC5oulAA[3-chloranyl-4-(3-fluorophenyl)phenyl]methanamineHuman9622
CSNK2A1 (CK2a1)CK2CMGC5oulAB[3-chloranyl-4-(3-fluorophenyl)phenyl]methanamineHuman9675
CSNK2A1 (CK2a1)CK2CMGC5oumAA~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]-2-(1~{h}-imidazol-2-yl)ethanamineHuman9668
CSNK2A1 (CK2a1)CK2CMGC5oumAB~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]-2-(1~{h}-imidazol-2-yl)ethanamineHuman9677
CSNK2A1 (CK2a1)CK2CMGC5oumBA-Human9679
CSNK2A1 (CK2a1)CK2CMGC5oumBB-Human9606
CSNK2A1 (CK2a1)CK2CMGC5ouuAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman9610
CSNK2A1 (CK2a1)CK2CMGC5ouuAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman9662
CSNK2A1 (CK2a1)CK2CMGC5ouuBA2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman9657
CSNK2A1 (CK2a1)CK2CMGC5ouuBB2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman9636
CSNK2A1 (CK2a1)CK2CMGC5owhA3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10597
CSNK2A1 (CK2a1)CK2CMGC5owlAA3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10593
CSNK2A1 (CK2a1)CK2CMGC5owlAB3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10596
CSNK2A1 (CK2a1)CK2CMGC5owlBA3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10590
CSNK2A1 (CK2a1)CK2CMGC5owlBB3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10592
CSNK2A1 (CK2a1)CK2CMGC5oyfAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methyl-phenyl]methyl]ethanamineHuman9617
CSNK2A1 (CK2a1)CK2CMGC5oyfAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methyl-phenyl]methyl]ethanamineHuman9658
CSNK2A1 (CK2a1)CK2CMGC5t1hAA7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman8685
CSNK2A1 (CK2a1)CK2CMGC5t1hAB7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman8682
CSNK2A1 (CK2a1)CK2CMGC5t1hBA7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman8683
CSNK2A1 (CK2a1)CK2CMGC5t1hBB7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman8684
CSNK2A1 (CK2a1)CK2CMGC5zn0AA-Human10697
CSNK2A1 (CK2a1)CK2CMGC5zn0AB-Human10699
CSNK2A1 (CK2a1)CK2CMGC5zn0AC-Human10704
CSNK2A1 (CK2a1)CK2CMGC5zn0AD-Human10709
CSNK2A1 (CK2a1)CK2CMGC5zn1AA-Human10696
CSNK2A1 (CK2a1)CK2CMGC5zn1AB-Human10707
CSNK2A1 (CK2a1)CK2CMGC5zn2AA-Human10698
CSNK2A1 (CK2a1)CK2CMGC5zn2AB-Human10702
CSNK2A1 (CK2a1)CK2CMGC5zn3AA-Human10703
CSNK2A1 (CK2a1)CK2CMGC5zn3AB-Human10706
CSNK2A1 (CK2a1)CK2CMGC5zn4AA-Human10700
CSNK2A1 (CK2a1)CK2CMGC5zn4AB-Human10708
CSNK2A1 (CK2a1)CK2CMGC5zn5AA-Human10705
CSNK2A1 (CK2a1)CK2CMGC5zn5AB-Human10701
CSNK2A1 (CK2a1)CK2CMGC6a1cAA5-bromanyl-2-methoxy-4-[(e)-(3-methylsulfanyl-5-phenyl-1,2,4-triazol-4-yl)iminomethyl]phenolHuman11273
CSNK2A1 (CK2a1)CK2CMGC6a1cAB5-bromanyl-2-methoxy-4-[(e)-(3-methylsulfanyl-5-phenyl-1,2,4-triazol-4-yl)iminomethyl]phenolHuman11286
CSNK2A1 (CK2a1)CK2CMGC6ehkAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[3,5-bis(chloranyl)-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9641
CSNK2A1 (CK2a1)CK2CMGC6ehkAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[3,5-bis(chloranyl)-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9663
CSNK2A1 (CK2a1)CK2CMGC6ehuAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamineHuman9684
CSNK2A1 (CK2a1)CK2CMGC6ehuAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamineHuman9691
CSNK2A1 (CK2a1)CK2CMGC6ehuBA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamineHuman9630
CSNK2A1 (CK2a1)CK2CMGC6ehuBB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamineHuman9664
CSNK2A1 (CK2a1)CK2CMGC6eiiAA(3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azaniumHuman9687
CSNK2A1 (CK2a1)CK2CMGC6eiiAB(3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azaniumHuman9647
CSNK2A1 (CK2a1)CK2CMGC6eiiBA(3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azaniumHuman9654
CSNK2A1 (CK2a1)CK2CMGC6eiiBB(3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azaniumHuman9642
CSNK2A1 (CK2a1)CK2CMGC6fvfAA-Human11342
CSNK2A1 (CK2a1)CK2CMGC6fvfAB-Human11341
CSNK2A1 (CK2a1)CK2CMGC6fvgAAadenosine-5'-triphosphateHuman11340
CSNK2A1 (CK2a1)CK2CMGC6fvgABadenosine-5'-triphosphateHuman11339
CSNK2A1 (CK2a1)CK2CMGC6gihAA-Human9941
CSNK2A1 (CK2a1)CK2CMGC6gihAB-Human9942
CSNK2A1 (CK2a1)CK2CMGC6gmdAAadenosine-5'-triphosphateHuman9993
CSNK2A1 (CK2a1)CK2CMGC6gmdABadenosine-5'-triphosphateHuman9990
CSNK2A1 (CK2a1)CK2CMGC6gmdBAadenosine-5'-triphosphateHuman9991
CSNK2A1 (CK2a1)CK2CMGC6gmdBBadenosine-5'-triphosphateHuman9992
CSNK2A1 (CK2a1)CK2CMGC6hbnAA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11287
CSNK2A1 (CK2a1)CK2CMGC6hbnAB5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11284
CSNK2A1 (CK2a1)CK2CMGC6hbnBA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11270
CSNK2A1 (CK2a1)CK2CMGC6hbnBB5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11272
CSNK2A1 (CK2a1)CK2CMGC6hmeAA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11275
CSNK2A1 (CK2a1)CK2CMGC6hmeAB5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11283
CSNK2A1 (CK2a1)CK2CMGC6hmeBA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11279
CSNK2A1 (CK2a1)CK2CMGC6hmeBB5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11282
CSNK2A1 (CK2a1)CK2CMGC6hnwAAcoumestrolHuman11523
CSNK2A1 (CK2a1)CK2CMGC6hnwABcoumestrolHuman11521
CSNK2A1 (CK2a1)CK2CMGC6hnyAAboldineHuman11520
CSNK2A1 (CK2a1)CK2CMGC6hnyABboldineHuman11522
CSNK2A1 (CK2a1)CK2CMGC6hopAA3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acidHuman11661
CSNK2A1 (CK2a1)CK2CMGC6hopAB4-hydroxy-3-methoxybenzaldehydeHuman11660
CSNK2A1 (CK2a1)CK2CMGC6hopAC(~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-oneHuman11662
CSNK2A1 (CK2a1)CK2CMGC6hopAD(2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enalHuman11666
CSNK2A1 (CK2a1)CK2CMGC6hoqAA3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acidHuman11669
CSNK2A1 (CK2a1)CK2CMGC6hoqAB3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acidHuman11665
CSNK2A1 (CK2a1)CK2CMGC6horAA(~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-oneHuman11668
CSNK2A1 (CK2a1)CK2CMGC6horAB(~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-oneHuman11663
CSNK2A1 (CK2a1)CK2CMGC6hotAA(2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enalHuman11667
CSNK2A1 (CK2a1)CK2CMGC6hotAB(2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enalHuman11670
CSNK2A1 (CK2a1)CK2CMGC6houAA4-hydroxy-3-methoxybenzaldehydeHuman11671
CSNK2A1 (CK2a1)CK2CMGC6houAB4-hydroxy-3-methoxybenzaldehydeHuman11664
CSNK2A1 (CK2a1)CK2CMGC6jwaA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman11467
CSNK2A1 (CK2a1)CK2CMGC6l1zA(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12010
CSNK2A1 (CK2a1)CK2CMGC6l21A(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12011
CSNK2A1 (CK2a1)CK2CMGC6l22AA(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12009
CSNK2A1 (CK2a1)CK2CMGC6l22AB(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12014
CSNK2A1 (CK2a1)CK2CMGC6l23AA(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman13455
CSNK2A1 (CK2a1)CK2CMGC6l23AB(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman13454
CSNK2A1 (CK2a1)CK2CMGC6l24AA(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12013
CSNK2A1 (CK2a1)CK2CMGC6l24AB(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12012
CSNK2A1 (CK2a1)CK2CMGC6q38AAbenzoic acidHuman11271
CSNK2A1 (CK2a1)CK2CMGC6q38ABbenzoic acidHuman11285
CSNK2A1 (CK2a1)CK2CMGC6q4qAAbenzoic acidHuman11281
CSNK2A1 (CK2a1)CK2CMGC6q4qABbenzoic acidHuman11276
CSNK2A1 (CK2a1)CK2CMGC6q4qACbenzoic acidHuman11277
CSNK2A1 (CK2a1)CK2CMGC6q4qBAbenzoic acidHuman11274
CSNK2A1 (CK2a1)CK2CMGC6q4qBBbenzoic acidHuman11278
CSNK2A1 (CK2a1)CK2CMGC6q4qBCbenzoic acidHuman11280
CSNK2A1 (CK2a1)CK2CMGC6qy7AA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12122
CSNK2A1 (CK2a1)CK2CMGC6qy7AB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12123
CSNK2A1 (CK2a1)CK2CMGC6qy7BA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12125
CSNK2A1 (CK2a1)CK2CMGC6qy7BB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12124
CSNK2A1 (CK2a1)CK2CMGC6rb1AA(~{e})-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)-~{n}-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]prop-2-enamideHuman12145
CSNK2A1 (CK2a1)CK2CMGC6rb1AB(~{e})-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)-~{n}-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]prop-2-enamideHuman12142
CSNK2A1 (CK2a1)CK2CMGC6rcbA(~{e})-2-cyano-~{n}-(2-hydroxyphenyl)-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12144
CSNK2A1 (CK2a1)CK2CMGC6rcmAA(~{e})-~{n}-(5-~{tert}-butyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12150
CSNK2A1 (CK2a1)CK2CMGC6rcmAB(~{e})-~{n}-(5-~{tert}-butyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12143
CSNK2A1 (CK2a1)CK2CMGC6rfeAA(~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12148
CSNK2A1 (CK2a1)CK2CMGC6rfeAB(~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12147
CSNK2A1 (CK2a1)CK2CMGC6rffAA(~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-nitro-4-oxidanyl-phenyl)prop-2-enamideHuman12146
CSNK2A1 (CK2a1)CK2CMGC6rffAB(~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-nitro-4-oxidanyl-phenyl)prop-2-enamideHuman12149
CSNK2A1 (CK2a1)CK2CMGC6spwAA-Human11961
CSNK2A1 (CK2a1)CK2CMGC6spwAB-Human11959
CSNK2A1 (CK2a1)CK2CMGC6spxA-Human11960
CSNK2A1 (CK2a1)CK2CMGC6teiAA3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12461
CSNK2A1 (CK2a1)CK2CMGC6teiAB3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12459
CSNK2A1 (CK2a1)CK2CMGC6teiBA3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12460
CSNK2A1 (CK2a1)CK2CMGC6teiBB3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12457
CSNK2A1 (CK2a1)CK2CMGC6tllAA4,5,6,7-tetrabromobenzotriazoleHuman13093
CSNK2A1 (CK2a1)CK2CMGC6tllAB4,5,6,7-tetrabromobenzotriazoleHuman13081
CSNK2A1 (CK2a1)CK2CMGC6tllAC4,5,6,7-tetrabromobenzotriazoleHuman13076
CSNK2A1 (CK2a1)CK2CMGC6tllAD4,5,6,7-tetrabromobenzotriazoleHuman13087
CSNK2A1 (CK2a1)CK2CMGC6tloAA5,6,7-tris(bromanyl)-1~{h}-benzotriazoleHuman13092
CSNK2A1 (CK2a1)CK2CMGC6tloAB5,6,7-tris(bromanyl)-1~{h}-benzotriazoleHuman13074
CSNK2A1 (CK2a1)CK2CMGC6tloAC-Human13075
CSNK2A1 (CK2a1)CK2CMGC6tlpAA5,6-dibromobenzotriazoleHuman13080
CSNK2A1 (CK2a1)CK2CMGC6tlpAB5,6-dibromobenzotriazoleHuman13078
CSNK2A1 (CK2a1)CK2CMGC6tlrAA4,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13089
CSNK2A1 (CK2a1)CK2CMGC6tlrAB4,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13083
CSNK2A1 (CK2a1)CK2CMGC6tlsAA5,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13077
CSNK2A1 (CK2a1)CK2CMGC6tlsAB5,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13082
CSNK2A1 (CK2a1)CK2CMGC6tluAA6,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13091
CSNK2A1 (CK2a1)CK2CMGC6tluAB6,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13090
CSNK2A1 (CK2a1)CK2CMGC6tlvAA6-bromanyl-1~{h}-benzotriazoleHuman13079
CSNK2A1 (CK2a1)CK2CMGC6tlvAB6-bromanyl-1~{h}-benzotriazoleHuman13084
CSNK2A1 (CK2a1)CK2CMGC6tlwAA7-bromanyl-1~{h}-benzotriazoleHuman13088
CSNK2A1 (CK2a1)CK2CMGC6tlwAB7-bromanyl-1~{h}-benzotriazoleHuman13085
CSNK2A1 (CK2a1)CK2CMGC6tlwAC7-bromanyl-1~{h}-benzotriazoleHuman13086
CSNK2A1 (CK2a1)CK2CMGC6ypgAA4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12425
CSNK2A1 (CK2a1)CK2CMGC6ypgAB4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12432
CSNK2A1 (CK2a1)CK2CMGC6yphAA4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12433
CSNK2A1 (CK2a1)CK2CMGC6yphAB4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12431
CSNK2A1 (CK2a1)CK2CMGC6yphBA4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12428
CSNK2A1 (CK2a1)CK2CMGC6yphBB4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12429
CSNK2A1 (CK2a1)CK2CMGC6ypjAA4-[(4-phenyl-1,3-thiazol-2-yl)amino]benzoic acidHuman12435
CSNK2A1 (CK2a1)CK2CMGC6ypjAB4-[(4-phenyl-1,3-thiazol-2-yl)amino]benzoic acidHuman12434
CSNK2A1 (CK2a1)CK2CMGC6ypkAA-Human12430
CSNK2A1 (CK2a1)CK2CMGC6ypkAB-Human12426
CSNK2A1 (CK2a1)CK2CMGC6ypnBAadenosine-5'-diphosphateHuman12427
CSNK2A1 (CK2a1)CK2CMGC6ypnBBadenosine-5'-diphosphateHuman12436
CSNK2A1 (CK2a1)CK2CMGC6yulA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12458
CSNK2A1 (CK2a1)CK2CMGC6yumA4-[5-[2-(2-hydroxyethyloxy)ethyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]pyrazolo[1,5-a]pyrimidin-3-yl]-2-oxidanyl-benzoic acidHuman12462
CSNK2A1 (CK2a1)CK2CMGC6yzhAAadenosine-5'-diphosphateHuman13559
CSNK2A1 (CK2a1)CK2CMGC6yzhABadenosine-5'-diphosphateHuman13560
CSNK2A1 (CK2a1)CK2CMGC6z83A~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamideHuman12652
CSNK2A1 (CK2a1)CK2CMGC6z83B~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamideHuman12651
CSNK2A1 (CK2a1)CK2CMGC6z84A~{n}-[1-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]ethanamideHuman12650
CSNK2A1 (CK2a1)CK2CMGC6z84B~{n}-[1-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]ethanamideHuman12649
CSNK2A1 (CK2a1)CK2CMGC7a49A6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13169
CSNK2A1 (CK2a1)CK2CMGC7a49B6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13168
CSNK2A1 (CK2a1)CK2CMGC7a4bAA 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13167
CSNK2A1 (CK2a1)CK2CMGC7a4bAB 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13165
CSNK2A1 (CK2a1)CK2CMGC7a4bBA 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13172
CSNK2A1 (CK2a1)CK2CMGC7a4bBB 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13166
CSNK2A1 (CK2a1)CK2CMGC7a4cAA5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13170
CSNK2A1 (CK2a1)CK2CMGC7a4cAB5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13174
CSNK2A1 (CK2a1)CK2CMGC7a4cBA5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13173
CSNK2A1 (CK2a1)CK2CMGC7a4cBB5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13171
CSNK2A1 (CK2a1)CK2CMGC7a4qAA2-methoxyimino-5-(quinolin-6-ylmethyl)-1,3-thiazol-4-oneHuman14238
CSNK2A1 (CK2a1)CK2CMGC7a4qAB2-methoxyimino-5-(quinolin-6-ylmethyl)-1,3-thiazol-4-oneHuman14239
CSNK2A1 (CK2a1)CK2CMGC7at5AA~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamideHuman13840
CSNK2A1 (CK2a1)CK2CMGC7at5AB~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamideHuman13839
CSNK2A1 (CK2a1)CK2CMGC7ay9A7-(cyclopropylamino)-5-(5-(6-oxo-1,6-dihydropyridin-3-yl)-1-(2-(piperidin-1-yl)ethyl)-1h-1,2,3-triazol-4-yl)pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman13993
CSNK2A1 (CK2a1)CK2CMGC7ayaAA~{n}-[2-[(1~{r},2~{r})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman13991
CSNK2A1 (CK2a1)CK2CMGC7ayaAB~{n}-[2-[(1~{r},2~{r})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman13992
CSNK2A1 (CK2a1)CK2CMGC7b8hAAnicotinic acidHuman13260
CSNK2A1 (CK2a1)CK2CMGC7b8hABnicotinic acidHuman13259
CSNK2A1 (CK2a1)CK2CMGC7b8iAA-Human13263
CSNK2A1 (CK2a1)CK2CMGC7b8iAB-Human13261
CSNK2A1 (CK2a1)CK2CMGC7b8iBA-Human13264
CSNK2A1 (CK2a1)CK2CMGC7b8iBB-Human13262
CSNK2A1 (CK2a1)CK2CMGC7bu4AA4-(6-aminocarbonyl-8-oxidanylidene-9-phenyl-7h-purin-2-yl)benzoic acidHuman13486
CSNK2A1 (CK2a1)CK2CMGC7bu4AB4-(6-aminocarbonyl-8-oxidanylidene-9-phenyl-7h-purin-2-yl)benzoic acidHuman13485
CSNK2A1 (CK2a1)CK2CMGC7l1xAA(2~{z})-6-[[2,6-bis(chloranyl)phenyl]methylsulfonyl]-2-[[4-oxidanyl-3-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methylidene]-4~{h}-1,4-benzothiazin-3-oneHuman13847
CSNK2A1 (CK2a1)CK2CMGC7l1xAB(2~{z})-6-[[2,6-bis(chloranyl)phenyl]methylsulfonyl]-2-[[4-oxidanyl-3-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methylidene]-4~{h}-1,4-benzothiazin-3-oneHuman13848
CSNK2A1 (CK2a1)CK2CMGC7psuAA-Human14163
CSNK2A1 (CK2a1)CK2CMGC7psuAB-Human14164
CSNK2A1 (CK2a1)CK2CMGC7qgbAA5,6-dibromobenzotriazoleHuman14468
CSNK2A1 (CK2a1)CK2CMGC7qgbAB5,6-dibromobenzotriazoleHuman14470
CSNK2A1 (CK2a1)CK2CMGC7qgcAA5,6-dibromobenzotriazoleHuman14433
CSNK2A1 (CK2a1)CK2CMGC7qgcAB5,6-dibromobenzotriazoleHuman14434
CSNK2A1 (CK2a1)CK2CMGC7qgdAA5,6-dibromobenzotriazoleHuman14472
CSNK2A1 (CK2a1)CK2CMGC7qgdAB5,6-dibromobenzotriazoleHuman14471
CSNK2A1 (CK2a1)CK2CMGC7qgeAA4,5,6,7-tetrabromobenzotriazoleHuman14469
CSNK2A1 (CK2a1)CK2CMGC7qgeAB4,5,6,7-tetrabromobenzotriazoleHuman14467
CSNK2A1 (CK2a1)CK2CMGC7quxAAadenosine-5'-diphosphateHuman14574
CSNK2A1 (CK2a1)CK2CMGC7quxABadenosine-5'-diphosphateHuman14573
CSNK2A1 (CK2a1)CK2CMGC7x4hAA5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrileHuman14595
CSNK2A1 (CK2a1)CK2CMGC7x4hAB5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrileHuman14596
CSNK2A1 (CK2a1)CK2CMGC7z39AA2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamideHuman14449
CSNK2A1 (CK2a1)CK2CMGC7z39AB2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamideHuman14445
CSNK2A1 (CK2a1)CK2CMGC7zweAA7-(1~{h}-indol-2-yl)-5-methyl-~{n}-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman14775
CSNK2A1 (CK2a1)CK2CMGC7zweAB7-(1~{h}-indol-2-yl)-5-methyl-~{n}-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman14771
CSNK2A1 (CK2a1)CK2CMGC7zwgAA(5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dioneHuman14772
CSNK2A1 (CK2a1)CK2CMGC7zwgAB(5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dioneHuman14774
CSNK2A1 (CK2a1)CK2CMGC7zwgAC(5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dioneHuman14773
CSNK2A1 (CK2a1)CK2CMGC7zy0AAadenosine-5'-diphosphateHuman14452
CSNK2A1 (CK2a1)CK2CMGC7zy0ABadenosine-5'-diphosphateHuman14439
CSNK2A1 (CK2a1)CK2CMGC7zy2AAadenosine-5'-triphosphateHuman14443
CSNK2A1 (CK2a1)CK2CMGC7zy2ABadenosine-5'-triphosphateHuman14458
CSNK2A1 (CK2a1)CK2CMGC7zy5AA-Human14457
CSNK2A1 (CK2a1)CK2CMGC7zy5AB-Human14453
CSNK2A1 (CK2a1)CK2CMGC7zy8AA-Human14441
CSNK2A1 (CK2a1)CK2CMGC7zy8AB-Human14454
CSNK2A1 (CK2a1)CK2CMGC7zydAAadenosine-5'-triphosphateHuman14438
CSNK2A1 (CK2a1)CK2CMGC7zydABadenosine-5'-triphosphateHuman14450
CSNK2A1 (CK2a1)CK2CMGC7zykAAadenosine-5'-diphosphateHuman14547
CSNK2A1 (CK2a1)CK2CMGC7zykABadenosine-5'-diphosphateHuman14546
CSNK2A1 (CK2a1)CK2CMGC7zyoAAadenosine-5'-triphosphateHuman14448
CSNK2A1 (CK2a1)CK2CMGC7zyoABadenosine-5'-triphosphateHuman14440
CSNK2A1 (CK2a1)CK2CMGC7zyrAAadenosine-5'-triphosphateHuman14444
CSNK2A1 (CK2a1)CK2CMGC7zyrABadenosine-5'-triphosphateHuman14456
CSNK2A1 (CK2a1)CK2CMGC8ae7AAadenosine-5'-diphosphateHuman14682
CSNK2A1 (CK2a1)CK2CMGC8ae7ABadenosine-5'-diphosphateHuman14684
CSNK2A1 (CK2a1)CK2CMGC8aecAAadenosine-5'-triphosphateHuman14455
CSNK2A1 (CK2a1)CK2CMGC8aecABadenosine-5'-triphosphateHuman14451
CSNK2A1 (CK2a1)CK2CMGC8aecACadenosine-5'-triphosphateHuman14446
CSNK2A1 (CK2a1)CK2CMGC8aekAAadenosine-5'-triphosphateHuman14442
CSNK2A1 (CK2a1)CK2CMGC8aekABadenosine-5'-triphosphateHuman14447
CSNK2A1 (CK2a1)CK2CMGC8aemAAadenosine-5'-triphosphateHuman14685
CSNK2A1 (CK2a1)CK2CMGC8aemABadenosine-5'-triphosphateHuman14683
CSNK2A1 (CK2a1)CK2CMGC8bgcA5-[(phenylmethyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acidHuman14545
CSNK2A1 (CK2a1)CK2CMGC8c5qAA2-methylpropyl 5-fluoranyl-3-[1-[[1-[2-[[4-(2-methylpropyl)phenyl]sulfonylamino]ethyl]piperidin-4-yl]methyl]-1,2,3-triazol-4-yl]-1~{h}-indole-2-carboxylateHuman15177
CSNK2A1 (CK2a1)CK2CMGC8c5qAB2-methylpropyl 5-fluoranyl-3-[1-[[1-[2-[[4-(2-methylpropyl)phenyl]sulfonylamino]ethyl]piperidin-4-yl]methyl]-1,2,3-triazol-4-yl]-1~{h}-indole-2-carboxylateHuman15175
CSNK2A1 (CK2a1)CK2CMGC8p05A(4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-oneHuman14744
CSNK2A1 (CK2a1)CK2CMGC8p06A7-(cyclopropylamino)-5-[[2-(1,2,4-triazol-4-yl)pyridin-4-yl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman14813
CSNK2A1 (CK2a1)CK2CMGC8p07A7-(cyclopropylamino)-5-[[3-(1,2,4-triazol-4-yl)phenyl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman14743
CSNK2A1 (CK2a1)CK2CMGC8pvoA2-[1-(1,3-benzothiazol-6-ylsulfonyl)piperidin-4-yl]-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman14976
CSNK2A1 (CK2a1)CK2CMGC8pvpA~{n}-[5-[(3-chloranyl-4-phenyl-phenyl)methylamino]pentyl]isoquinoline-5-sulfonamideHuman14977
CSNK2A1 (CK2a1)CK2CMGC8qwyA4-[6-[(2-methoxy-5-propan-2-yloxy-phenyl)amino]pyrazin-2-yl]benzoic acidHuman15174
CSNK2A1 (CK2a1)CK2CMGC8qwzA4-[6-(6-propan-2-yloxyindol-1-yl)pyrazin-2-yl]benzoic acidHuman15176
CSNK2A2 (CK2a2)CK2CMGC3e3bX[1-(6-{6-[(1-methylethyl)amino]-1h-indazol-1-yl}pyrazin-2-yl)-1h-pyrrol-3-yl]acetic acidHuman2729
CSNK2A2 (CK2a2)CK2CMGC3ofmAA3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman2728
CSNK2A2 (CK2a2)CK2CMGC3ofmAB3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman2730
CSNK2A2 (CK2a2)CK2CMGC5m4uAA4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7390
CSNK2A2 (CK2a2)CK2CMGC5m4uAB4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7391
CSNK2A2 (CK2a2)CK2CMGC5m56A4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7388
CSNK2A2 (CK2a2)CK2CMGC5m56B4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7389
CSNK2A2 (CK2a2)CK2CMGC5ooiAA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9447
CSNK2A2 (CK2a2)CK2CMGC5ooiAB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9446
CSNK2A2 (CK2a2)CK2CMGC5ooiBA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9445
CSNK2A2 (CK2a2)CK2CMGC5ooiBB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9444
CSNK2A2 (CK2a2)CK2CMGC5y9mAnicotinic acidHuman9908
CSNK2A2 (CK2a2)CK2CMGC5y9mXnicotinic acidHuman9909
CSNK2A2 (CK2a2)CK2CMGC5yf9BAnicotinic acidHuman11415
CSNK2A2 (CK2a2)CK2CMGC5yf9BBnicotinic acidHuman11416
CSNK2A2 (CK2a2)CK2CMGC5yf9XAnicotinic acidHuman11417
CSNK2A2 (CK2a2)CK2CMGC5yf9XBnicotinic acidHuman11414
CSNK2A2 (CK2a2)CK2CMGC5ywmXnicotinic acidHuman10759
CSNK2A2 (CK2a2)CK2CMGC6hmbAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10994
CSNK2A2 (CK2a2)CK2CMGC6hmbAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10995
CSNK2A2 (CK2a2)CK2CMGC6hmcAA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman10996
CSNK2A2 (CK2a2)CK2CMGC6hmcAB-Human10993
CSNK2A2 (CK2a2)CK2CMGC6hmdAA5-[2-(diethylamino)ethyl]-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman10997
CSNK2A2 (CK2a2)CK2CMGC6hmdAB-Human10992
CSNK2A2 (CK2a2)CK2CMGC6hmdAC-Human10990
CSNK2A2 (CK2a2)CK2CMGC6hmqAA3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman10991
CSNK2A2 (CK2a2)CK2CMGC6hmqAB3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman10998
CSNK2A2 (CK2a2)CK2CMGC6l20A(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman11993
CSNK2A2 (CK2a2)CK2CMGC6l20D(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman11996
CSNK2A2 (CK2a2)CK2CMGC6l20G(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman11995
CSNK2A2 (CK2a2)CK2CMGC6l20J(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman11994
CSNK2A2 (CK2a2)CK2CMGC6qy8AA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12117
CSNK2A2 (CK2a2)CK2CMGC6qy8AB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12120
CSNK2A2 (CK2a2)CK2CMGC6qy8BA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12114
CSNK2A2 (CK2a2)CK2CMGC6qy8BB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12121
CSNK2A2 (CK2a2)CK2CMGC6qy8CA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12115
CSNK2A2 (CK2a2)CK2CMGC6qy8CB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12119
CSNK2A2 (CK2a2)CK2CMGC6qy8DA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12116
CSNK2A2 (CK2a2)CK2CMGC6qy8DB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12118
CSNK2A2 (CK2a2)CK2CMGC6qy9AA3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrileHuman11012
CSNK2A2 (CK2a2)CK2CMGC6qy9AB3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrileHuman11011
CSNK2A2 (CK2a2)CK2CMGC6te2AA3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12444
CSNK2A2 (CK2a2)CK2CMGC6te2AB3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12446
CSNK2A2 (CK2a2)CK2CMGC6tewAA4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12443
CSNK2A2 (CK2a2)CK2CMGC6tewAB4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12447
CSNK2A2 (CK2a2)CK2CMGC6tguAA4-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxidanyl-benzoic acidHuman12448
CSNK2A2 (CK2a2)CK2CMGC6tguAB4-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxidanyl-benzoic acidHuman12445
CSNK2A2 (CK2a2)CK2CMGC7a1bAA 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13149
CSNK2A2 (CK2a2)CK2CMGC7a1bAB 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13144
CSNK2A2 (CK2a2)CK2CMGC7a1zAA6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13145
CSNK2A2 (CK2a2)CK2CMGC7a1zAB6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13147
CSNK2A2 (CK2a2)CK2CMGC7a22AA5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13148
CSNK2A2 (CK2a2)CK2CMGC7a22AB5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13151
CSNK2A2 (CK2a2)CK2CMGC7a2hAA5,6,7-tris(bromanyl)-1~{h}-imidazo[4,5-b]pyridineHuman13150
CSNK2A2 (CK2a2)CK2CMGC7a2hAB5,6,7-tris(bromanyl)-1~{h}-imidazo[4,5-b]pyridineHuman13146
CSNK2A2 (CK2a2)CK2CMGC7at9AA3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman13832
CSNK2A2 (CK2a2)CK2CMGC7at9AB3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman13829
CSNK2A2 (CK2a2)CK2CMGC7at9AC2-(3,4-dichlorophenyl)ethanamineHuman13830
CSNK2A2 (CK2a2)CK2CMGC7atvAA~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamideHuman13831
CSNK2A2 (CK2a2)CK2CMGC7atvAB~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamideHuman13828
CSNK2A2 (CK2a2)CK2CMGC7xyhA5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrileHuman14587
CSNK2A2 (CK2a2)CK2CMGC8q77AA(2~{s})-2-[[(2~{s})-2-[[(2~{s})-2-[12-[[4-[[5-(4-carboxyphenyl)-1,3-thiazol-2-yl]amino]-4-oxidanylidene-butanoyl]-(2-hydroxy-2-oxoethyl)amino]dodecanoylamino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]butanedioic acidHuman15024
CSNK2A2 (CK2a2)CK2CMGC8q77AB(2~{s})-2-[[(2~{s})-2-[[(2~{s})-2-[12-[[4-[[5-(4-carboxyphenyl)-1,3-thiazol-2-yl]amino]-4-oxidanylidene-butanoyl]-(2-hydroxy-2-oxoethyl)amino]dodecanoylamino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]butanedioic acidHuman15022
CSNK2A2 (CK2a2)CK2CMGC8q9sAA~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamideHuman15028
CSNK2A2 (CK2a2)CK2CMGC8q9sAB~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamideHuman15031
CSNK2A2 (CK2a2)CK2CMGC8qbuAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman15029
CSNK2A2 (CK2a2)CK2CMGC8qbuAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman15025
CSNK2A2 (CK2a2)CK2CMGC8qcdAA4,5,6,7-tetrabromobenzotriazoleHuman15023
CSNK2A2 (CK2a2)CK2CMGC8qcdAB4,5,6,7-tetrabromobenzotriazoleHuman15019
CSNK2A2 (CK2a2)CK2CMGC8qcgAAphosphoaminophosphonic acid-adenylate esterHuman15026
CSNK2A2 (CK2a2)CK2CMGC8qcgABphosphoaminophosphonic acid-adenylate esterHuman15030
CSNK2A2 (CK2a2)CK2CMGC8qcgACphosphoaminophosphonic acid-adenylate esterHuman15027
CSNK2A2 (CK2a2)CK2CMGC8qf1AA-Human15020
CSNK2A2 (CK2a2)CK2CMGC8qf1AB-Human15021
DAPK1DAPKCAMK1ig1Aphosphoaminophosphonic acid-adenylate esterHuman5615
DAPK1DAPKCAMK1jkkAphosphoaminophosphonic acid-adenylate esterHuman5644
DAPK1DAPKCAMK1jklAAphosphoaminophosphonic acid-adenylate esterHuman5685
DAPK1DAPKCAMK1jklABphosphoaminophosphonic acid-adenylate esterHuman5619
DAPK1DAPKCAMK1jksAA-Human5657
DAPK1DAPKCAMK1jksAB-Human5633
DAPK1DAPKCAMK1jktA-Human5650
DAPK1DAPKCAMK1jktB-Human5663
DAPK1DAPKCAMK1p4fAA5,6-dihydro-benzo[h]cinnolin-3-ylamineHuman5625
DAPK1DAPKCAMK1p4fAB5,6-dihydro-benzo[h]cinnolin-3-ylamineHuman5664
DAPK1DAPKCAMK1wvwA-Human5652
DAPK1DAPKCAMK1wvxA6-(3-aminopropyl)-4,9-dimethylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman5616
DAPK1DAPKCAMK1wvyAstaurosporineHuman5661
DAPK1DAPKCAMK2w4jAAadenosine-5'-diphosphateHuman5678
DAPK1DAPKCAMK2w4jABadenosine-5'-diphosphateHuman5682
DAPK1DAPKCAMK2w4kAAadenosine-5'-diphosphateHuman5653
DAPK1DAPKCAMK2w4kABadenosine-5'-diphosphateHuman5660
DAPK1DAPKCAMK2x0gAA-Human5672
DAPK1DAPKCAMK2x0gAB-Human5676
DAPK1DAPKCAMK2xuuAadenosine-5'-diphosphateHuman5627
DAPK1DAPKCAMK2xzsAA-Human5618
DAPK1DAPKCAMK2xzsAB-Human5642
DAPK1DAPKCAMK2xzsBA-Human5658
DAPK1DAPKCAMK2xzsBB-Human5671
DAPK1DAPKCAMK2y0aA-Human5651
DAPK1DAPKCAMK2y4pA-Human5659
DAPK1DAPKCAMK2y4pB-Human5626
DAPK1DAPKCAMK2y4pC-Human5688
DAPK1DAPKCAMK2y4pD-Human5640
DAPK1DAPKCAMK2yakAAruthenium octasporine 4Human7259
DAPK1DAPKCAMK2yakABruthenium octasporine 4Human7260
DAPK1DAPKCAMK3dfcBAphosphoaminophosphonic acid-adenylate esterHuman5645
DAPK1DAPKCAMK3dfcBBphosphoaminophosphonic acid-adenylate esterHuman5620
DAPK1DAPKCAMK3dgkAA-Human5656
DAPK1DAPKCAMK3dgkAB-Human5629
DAPK1DAPKCAMK3eh9AAadenosine-5'-diphosphateHuman5621
DAPK1DAPKCAMK3eh9ABadenosine-5'-diphosphateHuman5622
DAPK1DAPKCAMK3eh9ACadenosine-5'-diphosphateHuman5655
DAPK1DAPKCAMK3ehaAAphosphoaminophosphonic acid-adenylate esterHuman5636
DAPK1DAPKCAMK3ehaABphosphoaminophosphonic acid-adenylate esterHuman5687
DAPK1DAPKCAMK3ehaACphosphoaminophosphonic acid-adenylate esterHuman5647
DAPK1DAPKCAMK3f5gAAadenosine-5'-diphosphateHuman5635
DAPK1DAPKCAMK3f5gABadenosine-5'-diphosphateHuman5675
DAPK1DAPKCAMK3f5uAAphosphoaminophosphonic acid-adenylate esterHuman5677
DAPK1DAPKCAMK3f5uABphosphoaminophosphonic acid-adenylate esterHuman5632
DAPK1DAPKCAMK3f5uACphosphoaminophosphonic acid-adenylate esterHuman5630
DAPK1DAPKCAMK3gu4AAphosphoaminophosphonic acid-adenylate esterHuman5670
DAPK1DAPKCAMK3gu4ABphosphoaminophosphonic acid-adenylate esterHuman5681
DAPK1DAPKCAMK3gu5AAphosphoaminophosphonic acid-adenylate esterHuman5680
DAPK1DAPKCAMK3gu5ABphosphoaminophosphonic acid-adenylate esterHuman5669
DAPK1DAPKCAMK3gu5ACphosphoaminophosphonic acid-adenylate esterHuman5662
DAPK1DAPKCAMK3gu6AAadenosine-5'-diphosphateHuman5631
DAPK1DAPKCAMK3gu6ABadenosine-5'-diphosphateHuman5638
DAPK1DAPKCAMK3gu7AAadenosine-5'-diphosphateHuman5624
DAPK1DAPKCAMK3gu7ABadenosine-5'-diphosphateHuman5665
DAPK1DAPKCAMK3gu8AAn6-cyclopentyladenosineHuman5679
DAPK1DAPKCAMK3gu8ABn6-cyclopentyladenosineHuman5628
DAPK1DAPKCAMK3gubAA9-alpha-l-lyxofuranosyl-n-(2-phenylethyl)-9h-purin-6-amineHuman5674
DAPK1DAPKCAMK3gubAB9-alpha-l-lyxofuranosyl-n-(2-phenylethyl)-9h-purin-6-amineHuman5673
DAPK1DAPKCAMK3zxtAphosphomethylphosphonic acid adenylate esterHuman5634
DAPK1DAPKCAMK3zxtBphosphomethylphosphonic acid adenylate esterHuman5666
DAPK1DAPKCAMK3zxtCphosphomethylphosphonic acid adenylate esterHuman5646
DAPK1DAPKCAMK3zxtDphosphomethylphosphonic acid adenylate esterHuman5617
DAPK1DAPKCAMK4b4lAA-Human5683
DAPK1DAPKCAMK4b4lAB-Human5684
DAPK1DAPKCAMK4pf4AA-Human5643
DAPK1DAPKCAMK4pf4AB-Human5648
DAPK1DAPKCAMK4tl0A-Human5641
DAPK1DAPKCAMK4txcA4-(3-{3-[(r)-{[2-(dimethylamino)ethyl]amino}(hydroxy)methyl]phenyl}imidazo[1,2-b]pyridazin-6-yl)-2-methoxyphenolHuman5668
DAPK1DAPKCAMK4uv0A-Human5639
DAPK1DAPKCAMK4yo4AAphthalazineHuman5686
DAPK1DAPKCAMK4yo4ABphthalazineHuman5649
DAPK1DAPKCAMK4ypdAA4-methylpyridazineHuman5654
DAPK1DAPKCAMK4ypdAB4-methylpyridazineHuman5623
DAPK1DAPKCAMK5autA8-anilino-1-naphthalene sulfonateHuman6137
DAPK1DAPKCAMK5auuA2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4h-chromen-4-oneHuman6145
DAPK1DAPKCAMK5auvA5,7-dihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman6139
DAPK1DAPKCAMK5auwA3,5,7,3',4'-pentahydroxyflavoneHuman6144
DAPK1DAPKCAMK5auxA3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman6136
DAPK1DAPKCAMK5auyA2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-oneHuman6134
DAPK1DAPKCAMK5auzAgenisteinHuman6140
DAPK1DAPKCAMK5av0A3-(3,4-dihydroxyphenyl)-7-hydroxy-4h-chromen-4-oneHuman6142
DAPK1DAPKCAMK5av1A-Human6138
DAPK1DAPKCAMK5av2A3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman6133
DAPK1DAPKCAMK5av3A3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman6143
DAPK1DAPKCAMK5av4AAgenisteinHuman6135
DAPK1DAPKCAMK5av4ABgenisteinHuman6141
DAPK1DAPKCAMK6aarA-Human11468
DAPK1DAPKCAMK6fhaAA-Human11289
DAPK1DAPKCAMK6fhaAB-Human11288
DAPK1DAPKCAMK6fhbAA-Human11290
DAPK1DAPKCAMK6fhbAB-Human11291
DAPK1DAPKCAMK6in4A-Human11795
DAPK1DAPKCAMK6qmoAA-Human11587
DAPK1DAPKCAMK6qmoAB-Human11588
DAPK1DAPKCAMK6qn4A-Human11589
DAPK1DAPKCAMK7ccuAAresveratrolHuman13234
DAPK1DAPKCAMK7ccuABresveratrolHuman13237
DAPK1DAPKCAMK7ccvAApiceatannolHuman13232
DAPK1DAPKCAMK7ccvABpiceatannolHuman13233
DAPK1DAPKCAMK7ccwAAresveratrolHuman13235
DAPK1DAPKCAMK7ccwABresveratrolHuman13236
DAPK1DAPKCAMK8ie5Atrans-oxyresveratrolHuman14749
DAPK1DAPKCAMK8ie6A3-[(e)-2-(4-hydroxyphenyl)ethenyl]-5-methoxy-phenolHuman14751
DAPK1DAPKCAMK8ie7ApterostilbeneHuman14752
DAPK1DAPKCAMK8ie8A5-[(~{e})-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]benzene-1,3-diolHuman14750
Dapk2 (DAPK2)DAPKCAMK2ya9AA-Mouse5749
Dapk2 (DAPK2)DAPKCAMK2ya9AB-Mouse5752
Dapk2 (DAPK2)DAPKCAMK2ya9BA-Mouse5743
Dapk2 (DAPK2)DAPKCAMK2ya9BB-Mouse5744
Dapk2 (DAPK2)DAPKCAMK2yaaAAadenosine-5'-triphosphateMouse5746
Dapk2 (DAPK2)DAPKCAMK2yaaABadenosine-5'-triphosphateMouse5747
Dapk2 (DAPK2)DAPKCAMK2yaaBAadenosine-5'-triphosphateMouse5751
Dapk2 (DAPK2)DAPKCAMK2yaaBBadenosine-5'-triphosphateMouse5754
Dapk2 (DAPK2)DAPKCAMK2yabAAadenosine monophosphateMouse5750
Dapk2 (DAPK2)DAPKCAMK2yabABadenosine monophosphateMouse5753
Dapk2 (DAPK2)DAPKCAMK2yabBAadenosine monophosphateMouse5748
Dapk2 (DAPK2)DAPKCAMK2yabBBadenosine monophosphateMouse5745
DAPK2DAPKCAMK1wmkA-Human1124
DAPK2DAPKCAMK1wmkB-Human1140
DAPK2DAPKCAMK1wmkC-Human1138
DAPK2DAPKCAMK1wmkD-Human1139
DAPK2DAPKCAMK1wmkE-Human1117
DAPK2DAPKCAMK1wmkF-Human1126
DAPK2DAPKCAMK1wmkG-Human1142
DAPK2DAPKCAMK1wmkH-Human1151
DAPK2DAPKCAMK1z9xA-Human1144
DAPK2DAPKCAMK1z9xB-Human1136
DAPK2DAPKCAMK1z9xC-Human1116
DAPK2DAPKCAMK1zwsA-Human1121
DAPK2DAPKCAMK1zwsB-Human1128
DAPK2DAPKCAMK1zwsC-Human1134
DAPK2DAPKCAMK1zwsD-Human1131
DAPK2DAPKCAMK1zwsE-Human1130
DAPK2DAPKCAMK1zwsF-Human1114
DAPK2DAPKCAMK1zwsG-Human1150
DAPK2DAPKCAMK1zwsH-Human1133
DAPK2DAPKCAMK2a27A-Human1113
DAPK2DAPKCAMK2a27B-Human1129
DAPK2DAPKCAMK2a27C-Human1125
DAPK2DAPKCAMK2a27D-Human1118
DAPK2DAPKCAMK2a27E-Human1147
DAPK2DAPKCAMK2a27F-Human1127
DAPK2DAPKCAMK2a27G-Human1146
DAPK2DAPKCAMK2a27H-Human1137
DAPK2DAPKCAMK2a2aAA-Human1145
DAPK2DAPKCAMK2a2aAB-Human1123
DAPK2DAPKCAMK2a2aBA-Human1115
DAPK2DAPKCAMK2a2aBB-Human1119
DAPK2DAPKCAMK2a2aCA-Human1122
DAPK2DAPKCAMK2a2aCB-Human1148
DAPK2DAPKCAMK2a2aDA-Human1120
DAPK2DAPKCAMK2a2aDB-Human1149
DAPK2DAPKCAMK2ckeAn-(2-aminoethyl)isoquinoline-5-sulfonamideHuman1143
DAPK2DAPKCAMK2ckeBn-(2-aminoethyl)isoquinoline-5-sulfonamideHuman1132
DAPK2DAPKCAMK2ckeCn-(2-aminoethyl)isoquinoline-5-sulfonamideHuman1135
DAPK2DAPKCAMK2ckeDn-(2-aminoethyl)isoquinoline-5-sulfonamideHuman1141
DAPK2DAPKCAMK6pawA-Human12442
DAPK2DAPKCAMK6pawB-Human12440
DAPK2DAPKCAMK6pawE-Human12439
DAPK2DAPKCAMK6pawF-Human12441
DAPK3DAPKCAMK1yrpA-Human384
DAPK3DAPKCAMK1yrpB-Human383
DAPK3DAPKCAMK2j90AA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman387
DAPK3DAPKCAMK2j90AB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman382
DAPK3DAPKCAMK2j90BA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman378
DAPK3DAPKCAMK2j90BB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman379
DAPK3DAPKCAMK3bhyAA(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman385
DAPK3DAPKCAMK3bhyAB(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman381
DAPK3DAPKCAMK3bqrAA4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acidHuman380
DAPK3DAPKCAMK3bqrAB4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acidHuman386
DAPK3DAPKCAMK5a6nAA5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ideHuman6164
DAPK3DAPKCAMK5a6nAB5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ideHuman6165
DAPK3DAPKCAMK5a6nBA-Human6162
DAPK3DAPKCAMK5a6nBB-Human6161
DAPK3DAPKCAMK5a6oAA-Human6167
DAPK3DAPKCAMK5a6oAB-Human6163
DAPK3DAPKCAMK5a6oBA-Human6168
DAPK3DAPKCAMK5a6oBB-Human6166
DAPK3DAPKCAMK5vjaAA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10351
DAPK3DAPKCAMK5vjaAB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10349
DAPK3DAPKCAMK5vjaBA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10346
DAPK3DAPKCAMK5vjaBB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10350
DAPK3DAPKCAMK5vjaCA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10345
DAPK3DAPKCAMK5vjaCB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10352
DAPK3DAPKCAMK5vjaDA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10348
DAPK3DAPKCAMK5vjaDB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10347
DCLK1DCAMKLCAMK5jzjAAamp phosphoramidateHuman6984
DCLK1DCAMKLCAMK5jzjABamp phosphoramidateHuman6987
DCLK1DCAMKLCAMK5jzjBAamp phosphoramidateHuman6985
DCLK1DCAMKLCAMK5jzjBBamp phosphoramidateHuman6983
DCLK1DCAMKLCAMK5jznA5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHuman6986
DCLK1DCAMKLCAMK5jznB5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHuman6982
DCLK1DCAMKLCAMK6kyqAA-Human12799
DCLK1DCAMKLCAMK6kyqAB-Human12798
DCLK1DCAMKLCAMK6kyqBA-Human12802
DCLK1DCAMKLCAMK6kyqBB-Human12801
DCLK1DCAMKLCAMK6kyrAA-Human12803
DCLK1DCAMKLCAMK6kyrAB-Human12800
DCLK1DCAMKLCAMK6kyrBA-Human12805
DCLK1DCAMKLCAMK6kyrBB-Human12804
DCLK1DCAMKLCAMK7f3gA(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13853
DCLK1DCAMKLCAMK7kx6A2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman13907
DCLK1DCAMKLCAMK7kx8A5-ethyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman13909
DCLK1DCAMKLCAMK7kxwA2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman13910
DCLK1DCAMKLCAMK7kxwB2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman13908
DDR1DDRTK3zosAA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3253
DDR1DDRTK3zosAB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3262
DDR1DDRTK3zosBA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3258
DDR1DDRTK3zosBB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3260
DDR1DDRTK4bkjAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman3263
DDR1DDRTK4bkjAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman3256
DDR1DDRTK4bkjBA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman3255
DDR1DDRTK4bkjBB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman3259
DDR1DDRTK4ckrAA4-[(4-ethylpiperazin-1-yl)methyl]-n-{4-methyl-3-[(2-oxo-2,3-dihydro-1h-indol-5-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHuman3257
DDR1DDRTK4ckrAB4-[(4-ethylpiperazin-1-yl)methyl]-n-{4-methyl-3-[(2-oxo-2,3-dihydro-1h-indol-5-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHuman3252
DDR1DDRTK5bvkA1-(2-chlorophenyl)-3-(pyridin-3-ylmethyl)ureaHuman3251
DDR1DDRTK5bvnAn-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamideHuman3261
DDR1DDRTK5bvoAn-(5-{(1s)-1-[(5-fluoro-1,3-benzoxazol-2-yl)amino]ethyl}-2-methylphenyl)imidazo[1,2-a]pyridine-3-carboxamideHuman3250
DDR1DDRTK5bvwAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman3254
DDR1DDRTK5fdpA(4~{s})-4-methyl-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinoline-7-carboxamideHuman6676
DDR1DDRTK5fdxA3-[(4-methylpiperazin-1-yl)methyl]-~{n}-[(4~{r})-4-methyl-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinolin-7-yl]-5-(trifluoromethyl)benzamideHuman7131
DDR1DDRTK5fdxB3-[(4-methylpiperazin-1-yl)methyl]-~{n}-[(4~{r})-4-methyl-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinolin-7-yl]-5-(trifluoromethyl)benzamideHuman7130
DDR1DDRTK5sauAA3-[(6-aminopyridin-3-yl)ethynyl]-n-[3-(trifluoromethyl)phenyl]benzamideHuman14253
DDR1DDRTK5sauAB3-[(6-aminopyridin-3-yl)ethynyl]-n-[3-(trifluoromethyl)phenyl]benzamideHuman14258
DDR1DDRTK5savAAn-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamideHuman14265
DDR1DDRTK5savABn-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamideHuman14261
DDR1DDRTK5sawAA2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamideHuman14259
DDR1DDRTK5sawAB2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamideHuman14251
DDR1DDRTK5saxAA2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamideHuman14262
DDR1DDRTK5saxAB2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamideHuman14263
DDR1DDRTK5sayAn-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamideHuman14256
DDR1DDRTK5sazAA2-chloro-5-{3-chloro-4-[(2-hydroxyethyl)amino]benzamido}-n-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamideHuman14255
DDR1DDRTK5sazAB2-chloro-5-{3-chloro-4-[(2-hydroxyethyl)amino]benzamido}-n-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamideHuman14260
DDR1DDRTK5sb0An-{[(1r,2s)-2-{2-[(pyridin-3-yl)oxy]ethyl}cyclohexyl]methyl}-3-(trifluoromethoxy)benzamideHuman14264
DDR1DDRTK5sb1AA4-chloro-n-[(3s,4r)-4-phenylpyrrolidin-3-yl]-3-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamideHuman14252
DDR1DDRTK5sb1AB4-chloro-n-[(3s,4r)-4-phenylpyrrolidin-3-yl]-3-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamideHuman14257
DDR1DDRTK5sb2AA3-chloro-n-[(1r,2s)-2-phenylcyclopropyl]-5-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamideHuman14250
DDR1DDRTK5sb2AB3-chloro-n-[(1r,2s)-2-phenylcyclopropyl]-5-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamideHuman14254
DDR1DDRTK6brjAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman10760
DDR1DDRTK6bsdAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman10761
DDR1DDRTK6fewAA2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamideHuman10738
DDR1DDRTK6fewAB2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamideHuman10740
DDR1DDRTK6fexAA2-[4-bromanyl-2-oxidanylidene-1'-(1~{h}-pyrazolo[4,3-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10741
DDR1DDRTK6fexAB2-[4-bromanyl-2-oxidanylidene-1'-(1~{h}-pyrazolo[4,3-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10744
DDR1DDRTK6filAA2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamideHuman10746
DDR1DDRTK6filAB2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamideHuman10739
DDR1DDRTK6finAA3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-8-(1~{h}-indazol-5-ylcarbonyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-oneHuman10743
DDR1DDRTK6finAB3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-8-(1~{h}-indazol-5-ylcarbonyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-oneHuman10747
DDR1DDRTK6fioAA2-[1'-(1~{h}-indazol-5-ylcarbonyl)-4-methyl-2-oxidanylidene-spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10748
DDR1DDRTK6fioAB2-[1'-(1~{h}-indazol-5-ylcarbonyl)-4-methyl-2-oxidanylidene-spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10749
DDR1DDRTK6fiqA1-(1~{h}-indazol-5-ylcarbonyl)-5'-methoxy-1'-[2-oxidanylidene-2-[(2~{s})-2-(trifluoromethyl)pyrrolidin-1-yl]ethyl]spiro[piperidine-4,3'-pyrrolo[3,2-b]pyridine]-2'-oneHuman10742
DDR1DDRTK6gwrAA3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamideHuman10485
DDR1DDRTK6gwrAB3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamideHuman10484
DDR1DDRTK6gwrBA3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamideHuman10486
DDR1DDRTK6gwrBB3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamideHuman10487
DDR1DDRTK6hp9A(2~{r})-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-2-(pyrimidin-5-ylamino)-2,3-dihydro-1~{h}-indene-5-carboxamideHuman10885
DDR1DDRTK6hp9B(2~{r})-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-2-(pyrimidin-5-ylamino)-2,3-dihydro-1~{h}-indene-5-carboxamideHuman10884
DDR1DDRTK6y23A-Human12741
DDR1DDRTK6y23B-Human12742
DDR1DDRTK6y23C-Human12743
DDR1DDRTK7bcmA~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamideHuman13379
DDR1DDRTK7bcmB~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamideHuman13381
DDR1DDRTK7be6AA5-amino-n-(4-(((2s)-4-cyclohexyl-1-((1-(methylsulfonyl)piperidin-3-yl)amino)-1-oxobutan-2-yl)carbamoyl)benzyl)-1-phenyl-1h-pyrazole-4-carboxamideHuman13378
DDR1DDRTK7be6AB5-amino-n-(4-(((2s)-4-cyclohexyl-1-((1-(methylsulfonyl)piperidin-3-yl)amino)-1-oxobutan-2-yl)carbamoyl)benzyl)-1-phenyl-1h-pyrazole-4-carboxamideHuman13380
DDR1DDRTK7fehAAn-[(5-chloranyl-2-ethylsulfonyl-phenyl)methyl]-3-piperazin-1-yl-5-(trifluoromethyloxy)benzamideHuman14309
DDR1DDRTK7fehABn-[(5-chloranyl-2-ethylsulfonyl-phenyl)methyl]-3-piperazin-1-yl-5-(trifluoromethyloxy)benzamideHuman14308
DDR2DDRTK6ferA2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10729
DDR2DDRTK6ferB2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10736
DDR2DDRTK6ferC2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10731
DDR2DDRTK6ferD2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10730
DDR2DDRTK6ferE2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10726
DDR2DDRTK6ferF2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10732
DDR2DDRTK6ferG2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10734
DDR2DDRTK6ferH2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10727
DDR2DDRTK6ferI2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10735
DDR2DDRTK6ferJ2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10728
DDR2DDRTK6ferK2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10725
DDR2DDRTK6ferL2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamideHuman10733
DDR2DDRTK7aymAAn-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamideHuman13071
DDR2DDRTK7aymABn-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamideHuman13072
DMPK (DMPK1)DMPKAGC2vd5A3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman1901
DMPK (DMPK1)DMPKAGC2vd5B3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman1902
DYRK1ADYRKCMGC2vx3AAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3776
DYRK1ADYRKCMGC2vx3ABn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3762
DYRK1ADYRKCMGC2vx3BAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3766
DYRK1ADYRKCMGC2vx3BBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3769
DYRK1ADYRKCMGC2vx3CAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3740
DYRK1ADYRKCMGC2vx3CBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3735
DYRK1ADYRKCMGC2vx3DAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3786
DYRK1ADYRKCMGC2vx3DBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3790
DYRK1ADYRKCMGC2wo6AAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3758
DYRK1ADYRKCMGC2wo6ABn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3764
DYRK1ADYRKCMGC2wo6BAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3749
DYRK1ADYRKCMGC2wo6BBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3739
DYRK1ADYRKCMGC3anqA(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3767
DYRK1ADYRKCMGC3anqB(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3745
DYRK1ADYRKCMGC3anqC(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3791
DYRK1ADYRKCMGC3anqD(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3795
DYRK1ADYRKCMGC3anrA7-methoxy-1-methyl-9h-beta-carbolineHuman3778
DYRK1ADYRKCMGC3anrB7-methoxy-1-methyl-9h-beta-carbolineHuman3729
DYRK1ADYRKCMGC3anrC7-methoxy-1-methyl-9h-beta-carbolineHuman3783
DYRK1ADYRKCMGC3anrD7-methoxy-1-methyl-9h-beta-carbolineHuman3755
DYRK1ADYRKCMGC4azeA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3761
DYRK1ADYRKCMGC4azeB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3768
DYRK1ADYRKCMGC4azeC5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3788
DYRK1ADYRKCMGC4mq1AAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3796
DYRK1ADYRKCMGC4mq1ABn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3736
DYRK1ADYRKCMGC4mq1BAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3773
DYRK1ADYRKCMGC4mq1BBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3770
DYRK1ADYRKCMGC4mq1CAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3781
DYRK1ADYRKCMGC4mq1CBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3750
DYRK1ADYRKCMGC4mq1DAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3744
DYRK1ADYRKCMGC4mq1DBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3763
DYRK1ADYRKCMGC4mq2AAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3752
DYRK1ADYRKCMGC4mq2ABmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3771
DYRK1ADYRKCMGC4mq2BAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3792
DYRK1ADYRKCMGC4mq2BBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3787
DYRK1ADYRKCMGC4mq2CAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3730
DYRK1ADYRKCMGC4mq2CBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3780
DYRK1ADYRKCMGC4mq2DAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3757
DYRK1ADYRKCMGC4mq2DBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3734
DYRK1ADYRKCMGC4nctApkc412Human3794
DYRK1ADYRKCMGC4nctBpkc412Human3743
DYRK1ADYRKCMGC4nctCpkc412Human3779
DYRK1ADYRKCMGC4nctDpkc412Human3751
DYRK1ADYRKCMGC4yljAA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3782
DYRK1ADYRKCMGC4yljAB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3746
DYRK1ADYRKCMGC4yljBA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3753
DYRK1ADYRKCMGC4yljBB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3785
DYRK1ADYRKCMGC4yljCA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3777
DYRK1ADYRKCMGC4yljCB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3748
DYRK1ADYRKCMGC4yljDA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3784
DYRK1ADYRKCMGC4yljDB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3793
DYRK1ADYRKCMGC4ylkAA10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3789
DYRK1ADYRKCMGC4ylkAB10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3756
DYRK1ADYRKCMGC4yllAA10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3747
DYRK1ADYRKCMGC4yllAB10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3772
DYRK1ADYRKCMGC4yllAC10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3731
DYRK1ADYRKCMGC4yu2AA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3774
DYRK1ADYRKCMGC4yu2AB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3765
DYRK1ADYRKCMGC4yu2BA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3737
DYRK1ADYRKCMGC4yu2BB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3738
DYRK1ADYRKCMGC4yu2CA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3741
DYRK1ADYRKCMGC4yu2CB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3775
DYRK1ADYRKCMGC4yu2DA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3760
DYRK1ADYRKCMGC4yu2DB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3733
DYRK1ADYRKCMGC5a3xAn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6723
DYRK1ADYRKCMGC5a3xBn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6724
DYRK1ADYRKCMGC5a3xCn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6722
DYRK1ADYRKCMGC5a3xDn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6718
DYRK1ADYRKCMGC5a4eAAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6741
DYRK1ADYRKCMGC5a4eABn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6740
DYRK1ADYRKCMGC5a4eBAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6713
DYRK1ADYRKCMGC5a4eBBn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6726
DYRK1ADYRKCMGC5a4eCAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6725
DYRK1ADYRKCMGC5a4eCBn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6727
DYRK1ADYRKCMGC5a4eDAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6714
DYRK1ADYRKCMGC5a4eDBn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6733
DYRK1ADYRKCMGC5a4lAAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6731
DYRK1ADYRKCMGC5a4lABn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6728
DYRK1ADYRKCMGC5a4lBAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6719
DYRK1ADYRKCMGC5a4lBBn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6735
DYRK1ADYRKCMGC5a4lCAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6721
DYRK1ADYRKCMGC5a4lCBn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6711
DYRK1ADYRKCMGC5a4lDAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6739
DYRK1ADYRKCMGC5a4lDBn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6730
DYRK1ADYRKCMGC5a4qAn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6717
DYRK1ADYRKCMGC5a4qBn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6729
DYRK1ADYRKCMGC5a4qCn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6738
DYRK1ADYRKCMGC5a4qDn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6737
DYRK1ADYRKCMGC5a4tAn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6732
DYRK1ADYRKCMGC5a4tBn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6715
DYRK1ADYRKCMGC5a4tCn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6734
DYRK1ADYRKCMGC5a4tDn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6712
DYRK1ADYRKCMGC5a54An-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6736
DYRK1ADYRKCMGC5a54Bn-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6716
DYRK1ADYRKCMGC5a54Cn-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6720
DYRK1ADYRKCMGC5a54Dn-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6710
DYRK1ADYRKCMGC5aikA4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3732
DYRK1ADYRKCMGC5aikB4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3759
DYRK1ADYRKCMGC5aikC4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3754
DYRK1ADYRKCMGC5aikD4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3742
DYRK1ADYRKCMGC6a1fAA8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10522
DYRK1ADYRKCMGC6a1fAB8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10521
DYRK1ADYRKCMGC6a1gA5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10530
DYRK1ADYRKCMGC6a1gB5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10539
DYRK1ADYRKCMGC6eifA4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10534
DYRK1ADYRKCMGC6eifB4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10544
DYRK1ADYRKCMGC6eifC4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10525
DYRK1ADYRKCMGC6eifD4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10532
DYRK1ADYRKCMGC6eijA~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10518
DYRK1ADYRKCMGC6eijB~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10516
DYRK1ADYRKCMGC6eijC~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10538
DYRK1ADYRKCMGC6eijD~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10559
DYRK1ADYRKCMGC6eilA[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHuman10546
DYRK1ADYRKCMGC6eilB[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHuman10557
DYRK1ADYRKCMGC6eilC-Human10552
DYRK1ADYRKCMGC6eilD[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHuman10551
DYRK1ADYRKCMGC6eipA4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10555
DYRK1ADYRKCMGC6eipB4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10517
DYRK1ADYRKCMGC6eipC4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10533
DYRK1ADYRKCMGC6eipD4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10531
DYRK1ADYRKCMGC6eiqA[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10554
DYRK1ADYRKCMGC6eiqB[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10529
DYRK1ADYRKCMGC6eiqC[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10524
DYRK1ADYRKCMGC6eiqD[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10541
DYRK1ADYRKCMGC6eirA~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10550
DYRK1ADYRKCMGC6eirB~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10558
DYRK1ADYRKCMGC6eirC~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10528
DYRK1ADYRKCMGC6eirD~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10549
DYRK1ADYRKCMGC6eisAA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10553
DYRK1ADYRKCMGC6eisAB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10526
DYRK1ADYRKCMGC6eisBA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10556
DYRK1ADYRKCMGC6eisBB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10537
DYRK1ADYRKCMGC6eisCA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10535
DYRK1ADYRKCMGC6eisCB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10548
DYRK1ADYRKCMGC6eisDA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10547
DYRK1ADYRKCMGC6eisDB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10543
DYRK1ADYRKCMGC6eivA~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10540
DYRK1ADYRKCMGC6eivB~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10536
DYRK1ADYRKCMGC6eivC~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10542
DYRK1ADYRKCMGC6eivD~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10527
DYRK1ADYRKCMGC6ej4A3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10520
DYRK1ADYRKCMGC6ej4B3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10523
DYRK1ADYRKCMGC6ej4C3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10519
DYRK1ADYRKCMGC6ej4D3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10545
DYRK1ADYRKCMGC6ln1A1,3,5,8-tetrakis(oxidanyl)xanthen-9-oneHuman13935
DYRK1ADYRKCMGC6qu2AA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12085
DYRK1ADYRKCMGC6qu2AB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12092
DYRK1ADYRKCMGC6qu2BA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12086
DYRK1ADYRKCMGC6qu2BB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12088
DYRK1ADYRKCMGC6qu2CA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12090
DYRK1ADYRKCMGC6qu2CB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12087
DYRK1ADYRKCMGC6qu2DA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12091
DYRK1ADYRKCMGC6qu2DB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12089
DYRK1ADYRKCMGC6s11AA6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11361
DYRK1ADYRKCMGC6s11AB6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11364
DYRK1ADYRKCMGC6s11BA6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11378
DYRK1ADYRKCMGC6s11BB6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11372
DYRK1ADYRKCMGC6s14AA~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11418
DYRK1ADYRKCMGC6s14AB~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11421
DYRK1ADYRKCMGC6s17AA~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11369
DYRK1ADYRKCMGC6s17AB~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11375
DYRK1ADYRKCMGC6s1bAA~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11359
DYRK1ADYRKCMGC6s1bAB~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11377
DYRK1ADYRKCMGC6s1hAA~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman11419
DYRK1ADYRKCMGC6s1hAB~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman11420
DYRK1ADYRKCMGC6s1iAA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11370
DYRK1ADYRKCMGC6s1iAB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11376
DYRK1ADYRKCMGC6s1iBA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11371
DYRK1ADYRKCMGC6s1iBB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11367
DYRK1ADYRKCMGC6s1iCA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11366
DYRK1ADYRKCMGC6s1iCB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11373
DYRK1ADYRKCMGC6s1iDA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11362
DYRK1ADYRKCMGC6s1iDB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11379
DYRK1ADYRKCMGC6s1jAA3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazineHuman11365
DYRK1ADYRKCMGC6s1jAB3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazineHuman11360
DYRK1ADYRKCMGC6t6aAA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11857
DYRK1ADYRKCMGC6t6aAB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11858
DYRK1ADYRKCMGC6t6aBA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11860
DYRK1ADYRKCMGC6t6aBB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11861
DYRK1ADYRKCMGC6t6aCA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11863
DYRK1ADYRKCMGC6t6aCB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11859
DYRK1ADYRKCMGC6t6aDA-Human11862
DYRK1ADYRKCMGC6t6aDB-Human11856
DYRK1ADYRKCMGC6uipA4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHuman12027
DYRK1ADYRKCMGC6uipB4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHuman12025
DYRK1ADYRKCMGC6uipC4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHuman12026
DYRK1ADYRKCMGC6uwyAA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11989
DYRK1ADYRKCMGC6uwyAB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11987
DYRK1ADYRKCMGC6uwyBA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11983
DYRK1ADYRKCMGC6uwyBB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11982
DYRK1ADYRKCMGC6uwyCA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11984
DYRK1ADYRKCMGC6uwyCB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11985
DYRK1ADYRKCMGC6uwyDA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11988
DYRK1ADYRKCMGC6uwyDB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11986
DYRK1ADYRKCMGC6yf8A~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13462
DYRK1ADYRKCMGC6yf8B~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13461
DYRK1ADYRKCMGC6yf8C~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13463
DYRK1ADYRKCMGC6yf8D~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13460
DYRK1ADYRKCMGC7a4oAphosphoaminophosphonic acid-adenylate esterHuman13744
DYRK1ADYRKCMGC7a4rAA2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-oneHuman13751
DYRK1ADYRKCMGC7a4rAB2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-oneHuman13743
DYRK1ADYRKCMGC7a4sA7-chlorothieno[3,2-c]pyridin-4-amineHuman13749
DYRK1ADYRKCMGC7a4wA6-(4-methoxyphenyl)pyrimidine-2,4-diamineHuman13754
DYRK1ADYRKCMGC7a4zA3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amineHuman13752
DYRK1ADYRKCMGC7a51A4-azanyl-6-bromanyl-7-methyl-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13753
DYRK1ADYRKCMGC7a52AA3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-oneHuman13748
DYRK1ADYRKCMGC7a52AB3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-oneHuman13750
DYRK1ADYRKCMGC7a53AA(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-oneHuman13755
DYRK1ADYRKCMGC7a53AB(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-oneHuman13741
DYRK1ADYRKCMGC7a55A3-(1-methylpyrazol-4-yl)-1~{h}-pyrazole-5-carboxylic acidHuman13746
DYRK1ADYRKCMGC7a5bA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman13756
DYRK1ADYRKCMGC7a5dAA4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13742
DYRK1ADYRKCMGC7a5dAB4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13745
DYRK1ADYRKCMGC7a5lAA4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amineHuman13747
DYRK1ADYRKCMGC7a5lAB4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amineHuman13758
DYRK1ADYRKCMGC7a5nA5-(2-azanylpyridin-4-yl)-~{n}-[[2,6-bis(fluoranyl)phenyl]methyl]-2-methyl-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman13757
DYRK1ADYRKCMGC7aj2AA4-(4-methoxyphenyl)pyridin-2-amineHuman13609
DYRK1ADYRKCMGC7aj2AB4-(4-methoxyphenyl)pyridin-2-amineHuman13592
DYRK1ADYRKCMGC7aj4AA4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amineHuman13605
DYRK1ADYRKCMGC7aj4AB4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amineHuman13588
DYRK1ADYRKCMGC7aj5AA4-(1-benzofuran-5-yl)pyridine-2,6-diamineHuman13602
DYRK1ADYRKCMGC7aj5AB4-(1-benzofuran-5-yl)pyridine-2,6-diamineHuman13591
DYRK1ADYRKCMGC7aj7A4-(3-methylbenzimidazol-5-yl)pyridine-2,6-diamineHuman13600
DYRK1ADYRKCMGC7aj8AA4-(1-benzofuran-5-yl)pyridin-2-amineHuman13587
DYRK1ADYRKCMGC7aj8AB4-(1-benzofuran-5-yl)pyridin-2-amineHuman13603
DYRK1ADYRKCMGC7ajaAA1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazineHuman13610
DYRK1ADYRKCMGC7ajaAB1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazineHuman13597
DYRK1ADYRKCMGC7ajmAA~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamideHuman13590
DYRK1ADYRKCMGC7ajmAB~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamideHuman13598
DYRK1ADYRKCMGC7ajsAA4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13599
DYRK1ADYRKCMGC7ajsAB4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13607
DYRK1ADYRKCMGC7ajvA4-(2,3-dibutylimidazo[4,5-b]pyridin-5-yl)pyridine-2,6-diamineHuman13594
DYRK1ADYRKCMGC7ajwAA4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13612
DYRK1ADYRKCMGC7ajwAB4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13611
DYRK1ADYRKCMGC7ajyA4-[2-methyl-3-[(2~{r})-2-phenoxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13606
DYRK1ADYRKCMGC7ak2A4-[2-methyl-3-(2-pyridin-2-yloxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13593
DYRK1ADYRKCMGC7akaAA4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13596
DYRK1ADYRKCMGC7akaAB4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13595
DYRK1ADYRKCMGC7akbAA4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13608
DYRK1ADYRKCMGC7akbAB4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13604
DYRK1ADYRKCMGC7akeA4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13601
DYRK1ADYRKCMGC7aklA4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13589
DYRK1ADYRKCMGC7fhsAA(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14160
DYRK1ADYRKCMGC7fhsAB(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14159
DYRK1ADYRKCMGC7fhtAA(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14161
DYRK1ADYRKCMGC7fhtAB(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14162
DYRK1ADYRKCMGC7o7kAAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman13988
DYRK1ADYRKCMGC7o7kABn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman13987
DYRK1ADYRKCMGC7z5nA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman14667
DYRK1ADYRKCMGC7zh8AA6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridineHuman14489
DYRK1ADYRKCMGC7zh8AB6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridineHuman14488
DYRK1ADYRKCMGC8c3gAAn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15155
DYRK1ADYRKCMGC8c3gABn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15153
DYRK1ADYRKCMGC8c3qAArutinHuman15158
DYRK1ADYRKCMGC8c3qABrutinHuman15154
DYRK1ADYRKCMGC8c3rAAgossypinHuman15156
DYRK1ADYRKCMGC8c3rABgossypinHuman15157
DYRK1BDYRKCMGC8c2zAAn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15180
DYRK1BDYRKCMGC8c2zABn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15181
DYRK2DYRKCMGC3k2lAA-Human3147
DYRK2DYRKCMGC3k2lAB-Human3145
DYRK2DYRKCMGC3kvwAA(2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acidHuman3148
DYRK2DYRKCMGC3kvwAB(2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acidHuman3149
DYRK2DYRKCMGC4azfAA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3144
DYRK2DYRKCMGC4azfAB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3146
DYRK2DYRKCMGC5lxcAAmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7122
DYRK2DYRKCMGC5lxcABmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7129
DYRK2DYRKCMGC5lxcBAmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7125
DYRK2DYRKCMGC5lxcBBmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7126
DYRK2DYRKCMGC5lxdAAmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7124
DYRK2DYRKCMGC5lxdABmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7128
DYRK2DYRKCMGC5lxdBAmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7123
DYRK2DYRKCMGC5lxdBBmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7127
DYRK2DYRKCMGC5ztnA(1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneHuman10482
DYRK2DYRKCMGC5ztnB(1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneHuman10483
DYRK2DYRKCMGC6hdpAAscorzodihydrostilbene aHuman11572
DYRK2DYRKCMGC6hdpABscorzodihydrostilbene aHuman11573
DYRK2DYRKCMGC6hdrAAcurcuminHuman11570
DYRK2DYRKCMGC6hdrABcurcuminHuman11571
DYRK2DYRKCMGC6k0jA3-(2,7-dimethoxyacridin-9-yl)sulfanylpropan-1-amineHuman11817
DYRK2DYRKCMGC7akfAA4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13613
DYRK2DYRKCMGC7akfAB4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13614
DYRK2DYRKCMGC7akhA4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13615
DYRK2DYRKCMGC7dg4A2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridineHuman13967
DYRK2DYRKCMGC7dh3A2,7-dimethoxy-9-piperidin-4-ylsulfanyl-acridineHuman13978
DYRK2DYRKCMGC7dh9A[2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridin-4-yl]methanolHuman13976
DYRK2DYRKCMGC7dhcA4-[bis(fluoranyl)methyl]-2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridineHuman13973
DYRK2DYRKCMGC7dhhA[9-(azetidin-3-ylmethylsulfanyl)-2,7-dimethoxy-acridin-4-yl]methanolHuman13975
DYRK2DYRKCMGC7dhkA2-methoxy-7-phenylmethoxy-9-(piperidin-4-ylmethylsulfanyl)acridineHuman13977
DYRK2DYRKCMGC7dhnA7-methoxy-2-methylsulfanyl-9-(piperidin-4-ylmethylsulfanyl)-[1,3]thiazolo[5,4-b]quinolineHuman13971
DYRK2DYRKCMGC7dhoA2-methoxy-9-(piperidin-4-ylmethylsulfanyl)-7-propan-2-yloxy-acridineHuman13972
DYRK2DYRKCMGC7dhvA2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine-4-carboxylic acidHuman13974
DYRK2DYRKCMGC7djoA[2,7-dimethoxy-9-[[(3s)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanolHuman13994
DYRK2DYRKCMGC7dl6A[2,7-dimethoxy-9-[[(3r)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanolHuman14013
DYRK2DYRKCMGC7ejvAA[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14180
DYRK2DYRKCMGC7ejvAB[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14181
DYRK2DYRKCMGC7ejvBA[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14183
DYRK2DYRKCMGC7ejvBB[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14182
DYRK2DYRKCMGC8hltA(6-{[(4p)-4-(1,3-benzothiazol-5-yl)-5-fluoropyrimidin-2-yl]amino}pyridin-3-yl)(piperazin-1-yl)methanoneHuman15091
DYRK3DYRKCMGC5y86A7-methoxy-1-methyl-9h-beta-carbolineHuman9876
EGFREGFRTK1m14A-Human826
EGFREGFRTK1m17AA[6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amineHuman873
EGFREGFRTK1m17AB[6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amineHuman905
EGFREGFRTK1xkkAn-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamineHuman844
EGFREGFRTK2eb2A-Human787
EGFREGFRTK2eb3Aphosphoaminophosphonic acid-adenylate esterHuman816
EGFREGFRTK2gs2A-Human849
EGFREGFRTK2gs6A-Human815
EGFREGFRTK2gs7Aphosphoaminophosphonic acid-adenylate esterHuman842
EGFREGFRTK2gs7Bphosphoaminophosphonic acid-adenylate esterHuman795
EGFREGFRTK2itnAAphosphoaminophosphonic acid-adenylate esterHuman879
EGFREGFRTK2itnABphosphoaminophosphonic acid-adenylate esterHuman833
EGFREGFRTK2itoAgefitinibHuman783
EGFREGFRTK2itpAA6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman880
EGFREGFRTK2itpAB6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman871
EGFREGFRTK2itqAA1,2,3,4-tetrahydrogen staurosporineHuman813
EGFREGFRTK2itqAB1,2,3,4-tetrahydrogen staurosporineHuman846
EGFREGFRTK2ittAA6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman892
EGFREGFRTK2ittAB6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman891
EGFREGFRTK2ituAA1,2,3,4-tetrahydrogen staurosporineHuman779
EGFREGFRTK2ituAB1,2,3,4-tetrahydrogen staurosporineHuman859
EGFREGFRTK2itvAAphosphoaminophosphonic acid-adenylate esterHuman911
EGFREGFRTK2itvABphosphoaminophosphonic acid-adenylate esterHuman834
EGFREGFRTK2itwAA1,2,3,4-tetrahydrogen staurosporineHuman817
EGFREGFRTK2itwAB1,2,3,4-tetrahydrogen staurosporineHuman914
EGFREGFRTK2itxAphosphoaminophosphonic acid-adenylate esterHuman865
EGFREGFRTK2ityAgefitinibHuman790
EGFREGFRTK2itzAgefitinibHuman789
EGFREGFRTK2j5eA-Human7215
EGFREGFRTK2j5fAn-[4-(3-bromo-phenylamino)-quinazolin-6-yl]-acrylamideHuman862
EGFREGFRTK2j6mA6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman900
EGFREGFRTK2jitA-Human888
EGFREGFRTK2jitB-Human805
EGFREGFRTK2jiuA6-{4-[(4-ethylpiperazin-1-yl)methyl]phenyl}-n-[(1r)-1-phenylethyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman858
EGFREGFRTK2jiuB-Human895
EGFREGFRTK2jivAAn-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamideHuman893
EGFREGFRTK2jivABn-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamideHuman851
EGFREGFRTK2jivBAn-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamideHuman830
EGFREGFRTK2jivBBn-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamideHuman812
EGFREGFRTK2rf9A-Human876
EGFREGFRTK2rf9B-Human883
EGFREGFRTK2rfdA-Human875
EGFREGFRTK2rfdB-Human840
EGFREGFRTK2rfeA-Human836
EGFREGFRTK2rfeB-Human896
EGFREGFRTK2rfeC-Human907
EGFREGFRTK2rfeD-Human807
EGFREGFRTK2rgpAn-[1-(3-fluorobenzyl)-1h-indazol-5-yl]-5-[(piperidin-1-ylamino)methyl]pyrimidine-4,6-diamineHuman6757
EGFREGFRTK3belA4-amino-6-{[1-(3-fluorobenzyl)-1h-indazol-5-yl]amino}pyrimidine-5-carbaldehyde o-(2-methoxyethyl)oximeHuman6758
EGFREGFRTK3gopAA-Human853
EGFREGFRTK3gopAB-Human886
EGFREGFRTK3gt8Aphosphoaminophosphonic acid-adenylate esterHuman908
EGFREGFRTK3gt8Bphosphoaminophosphonic acid-adenylate esterHuman847
EGFREGFRTK3gt8Cphosphoaminophosphonic acid-adenylate esterHuman882
EGFREGFRTK3gt8Dphosphoaminophosphonic acid-adenylate esterHuman860
EGFREGFRTK3ikaAAn-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamideHuman802
EGFREGFRTK3ikaABn-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamideHuman855
EGFREGFRTK3ikaBA-Human863
EGFREGFRTK3ikaBB-Human868
EGFREGFRTK3lzbAn-[3-(5-{2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}imidazo[2,1-b][1,3]thiazol-6-yl)phenyl]-2-phenylacetamideHuman800
EGFREGFRTK3lzbBn-[3-(5-{2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}imidazo[2,1-b][1,3]thiazol-6-yl)phenyl]-2-phenylacetamideHuman810
EGFREGFRTK3lzbCn-[3-(5-{2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}imidazo[2,1-b][1,3]thiazol-6-yl)phenyl]-2-phenylacetamideHuman808
EGFREGFRTK3lzbDn-[3-(5-{2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl}imidazo[2,1-b][1,3]thiazol-6-yl)phenyl]-2-phenylacetamideHuman820
EGFREGFRTK3pozAn-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamideHuman7308
EGFREGFRTK3ug1AA-Human864
EGFREGFRTK3ug1AB-Human799
EGFREGFRTK3ug2AAgefitinibHuman898
EGFREGFRTK3ug2ABgefitinibHuman819
EGFREGFRTK3vjnAphosphoaminophosphonic acid-adenylate esterHuman872
EGFREGFRTK3vjoAphosphoaminophosphonic acid-adenylate esterHuman777
EGFREGFRTK3w2oAAn-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamideHuman9119
EGFREGFRTK3w2oABn-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamideHuman9118
EGFREGFRTK3w2pAAn-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-4-(dimethylamino)butanamideHuman829
EGFREGFRTK3w2pABn-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-4-(dimethylamino)butanamideHuman838
EGFREGFRTK3w2qAAn-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamideHuman845
EGFREGFRTK3w2qABn-(4-{[3-chloro-4-(pyridin-2-ylmethoxy)phenyl]amino}-3-cyano-7-ethoxyquinolin-6-yl)-4-(dimethylamino)butanamideHuman874
EGFREGFRTK3w2rAA1-{3-[2-chloro-4-({5-[2-(2-hydroxyethoxy)ethyl]-5h-pyrrolo[3,2-d]pyrimidin-4-yl}amino)phenoxy]phenyl}-3-cyclohexylureaHuman822
EGFREGFRTK3w2rAB1-{3-[2-chloro-4-({5-[2-(2-hydroxyethoxy)ethyl]-5h-pyrrolo[3,2-d]pyrimidin-4-yl}amino)phenoxy]phenyl}-3-cyclohexylureaHuman885
EGFREGFRTK3w2sAA1-{3-[2-chloro-4-({5-[2-(2-hydroxyethoxy)ethyl]-5h-pyrrolo[3,2-d]pyrimidin-4-yl}amino)phenoxy]phenyl}-3-cyclohexylureaHuman778
EGFREGFRTK3w2sAB1-{3-[2-chloro-4-({5-[2-(2-hydroxyethoxy)ethyl]-5h-pyrrolo[3,2-d]pyrimidin-4-yl}amino)phenoxy]phenyl}-3-cyclohexylureaHuman792
EGFREGFRTK3w32A4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-n-[2-(methylsulfonyl)ethyl]-8,9-dihydro-7h-pyrimido[4,5-b]azepine-6-carboxamideHuman784
EGFREGFRTK3w33AA4-{[4-(1-benzothiophen-4-yloxy)-3-chlorophenyl]amino}-n-(2-hydroxyethyl)-8,9-dihydro-7h-pyrimido[4,5-b]azepine-6-carboxamideHuman782
EGFREGFRTK3w33AB4-{[4-(1-benzothiophen-4-yloxy)-3-chlorophenyl]amino}-n-(2-hydroxyethyl)-8,9-dihydro-7h-pyrimido[4,5-b]azepine-6-carboxamideHuman869
EGFREGFRTK4g5jAAn-{4-[(3-chloro-4-fluorophenyl)amino]-7-[(3s)-tetrahydrofuran-3-yloxy]quinazolin-6-yl}-4-(dimethylamino)butanamideHuman794
EGFREGFRTK4g5jABn-{4-[(3-chloro-4-fluorophenyl)amino]-7-[(3s)-tetrahydrofuran-3-yloxy]quinazolin-6-yl}-4-(dimethylamino)butanamideHuman852
EGFREGFRTK4g5pAn-{4-[(3-chloro-4-fluorophenyl)amino]-7-[(3s)-tetrahydrofuran-3-yloxy]quinazolin-6-yl}-4-(dimethylamino)butanamideHuman809
EGFREGFRTK4g5pB-Human788
EGFREGFRTK4hjoA[6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amineHuman835
EGFREGFRTK4i1zAA-Human903
EGFREGFRTK4i1zAB-Human906
EGFREGFRTK4i20A-Human850
EGFREGFRTK4i21A-Human824
EGFREGFRTK4i21B-Human776
EGFREGFRTK4i22AgefitinibHuman823
EGFREGFRTK4i23A(2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamideHuman870
EGFREGFRTK4i24A(2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamideHuman831
EGFREGFRTK4i24B(2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamideHuman910
EGFREGFRTK4jq7A(2s)-2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]-2-phenylethanolHuman801
EGFREGFRTK4jq8An-[3-(4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-6-phenylfuro[2,3-d]pyrimidin-5-yl)phenyl]-n~3~,n~3~-dimethyl-beta-alaninamideHuman821
EGFREGFRTK4jr3An-[3-(4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-6-phenylfuro[2,3-d]pyrimidin-5-yl)phenyl]acetamideHuman915
EGFREGFRTK4jrvA4-(dimethylamino)-n-[3-(4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-6-phenylfuro[2,3-d]pyrimidin-5-yl)phenyl]butanamideHuman857
EGFREGFRTK4li5AAn-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-4-methoxyphenyl)propanamideHuman841
EGFREGFRTK4li5ABn-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-4-methoxyphenyl)propanamideHuman797
EGFREGFRTK4ll0An-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHuman804
EGFREGFRTK4ll0Bn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHuman796
EGFREGFRTK4lqmAn-[4-(3-bromo-phenylamino)-quinazolin-6-yl]-acrylamideHuman785
EGFREGFRTK4lrmAn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHuman901
EGFREGFRTK4lrmBn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHuman867
EGFREGFRTK4lrmCn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHuman781
EGFREGFRTK4lrmDn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHuman786
EGFREGFRTK4lrmEn-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamideHuman825
EGFREGFRTK4r3pA-Human827
EGFREGFRTK4r3rA-Human887
EGFREGFRTK4r5sAn-[4-({[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino}methyl)phenyl]propanamideHuman775
EGFREGFRTK4riwBadenosine-5'-diphosphateHuman877
EGFREGFRTK4riwDadenosine-5'-diphosphateHuman848
EGFREGFRTK4rixBadenosine-5'-diphosphateHuman811
EGFREGFRTK4rixDadenosine-5'-diphosphateHuman909
EGFREGFRTK4riyBadenosine-5'-diphosphateHuman806
EGFREGFRTK4riyDadenosine-5'-diphosphateHuman856
EGFREGFRTK4rj4An-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1-(propan-2-yl)-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amineHuman866
EGFREGFRTK4rj5An-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amineHuman912
EGFREGFRTK4rj6An-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-2-(1h-pyrazol-4-yl)-3h-imidazo[4,5-c]pyridin-6-amineHuman832
EGFREGFRTK4rj7AA2,6-dichloro-n-{2-[(2-{[(2s)-1-hydroxypropan-2-yl]amino}-6-methylpyrimidin-4-yl)amino]pyridin-4-yl}benzamideHuman793
EGFREGFRTK4rj7AB2,6-dichloro-n-{2-[(2-{[(2s)-1-hydroxypropan-2-yl]amino}-6-methylpyrimidin-4-yl)amino]pyridin-4-yl}benzamideHuman828
EGFREGFRTK4rj8A1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHuman899
EGFREGFRTK4tksA-Human897
EGFREGFRTK4wd5An-{2-methyl-5-[2-oxo-9-(1h-pyrazol-4-yl)benzo[h][1,6]naphthyridin-1(2h)-yl]phenyl}propanamideHuman6594
EGFREGFRTK4wd5B-Human6593
EGFREGFRTK4wkqAAgefitinibHuman889
EGFREGFRTK4wkqABgefitinibHuman837
EGFREGFRTK4wrgAA-Human854
EGFREGFRTK4wrgAB-Human814
EGFREGFRTK4zauAn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHuman6221
EGFREGFRTK4zjvAA-Human798
EGFREGFRTK4zjvAB-Human843
EGFREGFRTK4zjvBA-Human904
EGFREGFRTK4zjvBB-Human780
EGFREGFRTK4zseAAphosphoaminophosphonic acid-adenylate esterHuman6696
EGFREGFRTK4zseABphosphoaminophosphonic acid-adenylate esterHuman6697
EGFREGFRTK4zseBAphosphoaminophosphonic acid-adenylate esterHuman6695
EGFREGFRTK4zseBBphosphoaminophosphonic acid-adenylate esterHuman6699
EGFREGFRTK4zseCAphosphoaminophosphonic acid-adenylate esterHuman6693
EGFREGFRTK4zseCBphosphoaminophosphonic acid-adenylate esterHuman6698
EGFREGFRTK4zseDAphosphoaminophosphonic acid-adenylate esterHuman6694
EGFREGFRTK4zseDBphosphoaminophosphonic acid-adenylate esterHuman6700
EGFREGFRTK5c8kA1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-imidazo[4,5-c]pyridin-6-amineHuman6201
EGFREGFRTK5c8mA2-methyl-n-{2-[4-(methylsulfonyl)piperidin-1-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amineHuman6202
EGFREGFRTK5c8nAn-{2-[4-(2-aminoethyl)-4-methoxypiperidin-1-yl]pyrimidin-4-yl}-2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amineHuman6199
EGFREGFRTK5calA2,2-dimethyl-3-[(4-{[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]amino}pyrimidin-2-yl)amino]propanamideHuman6195
EGFREGFRTK5canA(3r)-3-methyl-1-(4-{[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]amino}pyrimidin-2-yl)pyrrolidine-3-carboxamideHuman6203
EGFREGFRTK5caoAn~2~-[2-methyl-2-(methylsulfonyl)propyl]-n~4~-[2-methyl-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-yl]pyrimidine-2,4-diamineHuman6206
EGFREGFRTK5capAA2-methyl-n-[2-(2-methyl-2-methylsulfonyl-propoxy)pyrimidin-4-yl]-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amineHuman6200
EGFREGFRTK5capAB2-methyl-n-[2-(2-methyl-2-methylsulfonyl-propoxy)pyrimidin-4-yl]-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amineHuman6198
EGFREGFRTK5caqAn-[2-[(3r,4s)-3-fluoranyl-4-methoxy-piperidin-1-yl]pyrimidin-4-yl]-2-methyl-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amineHuman6204
EGFREGFRTK5casA(1r)-1-{6-({2-[(3r,4s)-3-fluoro-4-methoxypiperidin-1-yl]pyrimidin-4-yl}amino)-1-[(2s)-1,1,1-trifluoropropan-2-yl]-1h-imidazo[4,5-c]pyridin-2-yl}ethanolHuman6205
EGFREGFRTK5cauA(1r)-1-{6-({2-[(3s,4r)-3-fluoro-4-methoxypiperidin-1-yl]pyrimidin-4-yl}amino)-1-[(2s)-1,1,1-trifluoropropan-2-yl]-1h-imidazo[4,5-c]pyridin-2-yl}ethanolHuman6196
EGFREGFRTK5cavA(1r)-1-{6-({2-[(3r,4s)-3-fluoro-4-methoxypiperidin-1-yl]pyrimidin-4-yl}amino)-1-[(2s)-1,1,1-trifluoropropan-2-yl]-1h-imidazo[4,5-c]pyridin-2-yl}ethanolHuman6197
EGFREGFRTK5cnnAAphosphoaminophosphonic acid-adenylate esterHuman791
EGFREGFRTK5cnnABphosphoaminophosphonic acid-adenylate esterHuman902
EGFREGFRTK5cnnBAphosphoaminophosphonic acid-adenylate esterHuman839
EGFREGFRTK5cnnBBphosphoaminophosphonic acid-adenylate esterHuman803
EGFREGFRTK5cnoAAphosphoaminophosphonic acid-adenylate esterHuman884
EGFREGFRTK5cnoABphosphoaminophosphonic acid-adenylate esterHuman894
EGFREGFRTK5cnoBAphosphoaminophosphonic acid-adenylate esterHuman878
EGFREGFRTK5cnoBBphosphoaminophosphonic acid-adenylate esterHuman861
EGFREGFRTK5czhA-Human6111
EGFREGFRTK5cziA-Human6110
EGFREGFRTK5d41AAphosphoaminophosphonic acid-adenylate esterHuman6665
EGFREGFRTK5d41ABphosphoaminophosphonic acid-adenylate esterHuman6667
EGFREGFRTK5d41BAphosphoaminophosphonic acid-adenylate esterHuman6666
EGFREGFRTK5d41BBphosphoaminophosphonic acid-adenylate esterHuman6664
EGFREGFRTK5edpA-Human6252
EGFREGFRTK5edqA~{n}-(7-chloranyl-1~{h}-indazol-3-yl)-7,7-dimethyl-2-(1~{h}-pyrazol-4-yl)-5~{h}-furo[3,4-d]pyrimidin-4-amineHuman6253
EGFREGFRTK5edrAA~{n}-(1~{h}-indazol-3-yl)-7,7-dimethyl-2-(2-methylpyrazol-3-yl)-5~{h}-furo[3,4-d]pyrimidin-4-amineHuman6254
EGFREGFRTK5edrAB~{n}-(1~{h}-indazol-3-yl)-7,7-dimethyl-2-(2-methylpyrazol-3-yl)-5~{h}-furo[3,4-d]pyrimidin-4-amineHuman6255
EGFREGFRTK5em5A4-[2-(4-chlorophenyl)ethylamino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamideHuman6307
EGFREGFRTK5em6A4-[(2-azanylpyrimidin-4-yl)amino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamideHuman6305
EGFREGFRTK5em7AA4-[(2-methoxyphenyl)amino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamideHuman6304
EGFREGFRTK5em7AB4-[(2-methoxyphenyl)amino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamideHuman6303
EGFREGFRTK5em8A4-[(2-methoxyphenyl)amino]-~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-2-oxidanylidene-1~{h}-pyridine-3-carboxamideHuman6306
EGFREGFRTK5fedA~{n}-[7-methyl-1-[(3~{r})-1-propanoylazepan-3-yl]benzimidazol-2-yl]-3-(trifluoromethyl)benzamideHuman6882
EGFREGFRTK5feeA~{n}-[7-methyl-1-[(3~{r})-1-propanoylazepan-3-yl]benzimidazol-2-yl]-3-(trifluoromethyl)benzamideHuman6881
EGFREGFRTK5feqA~{n}-[1-[(3~{r})-1-[4-(dimethylamino)but-2-enoyl]azepan-3-yl]-7-methyl-benzimidazol-2-yl]-2-methyl-pyridine-4-carboxamideHuman6883
EGFREGFRTK5gmpAAn-[3-[2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-5-methyl-7-oxidanylidene-pyrido[2,3-d]pyrimidin-8-yl]phenyl]prop-2-enamideHuman8167
EGFREGFRTK5gmpABn-[3-[2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-5-methyl-7-oxidanylidene-pyrido[2,3-d]pyrimidin-8-yl]phenyl]prop-2-enamideHuman8168
EGFREGFRTK5gnkAA1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(1-methylimidazol-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman7525
EGFREGFRTK5gnkAB1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(1-methylimidazol-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman7524
EGFREGFRTK5gtyAA1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8363
EGFREGFRTK5gtyAB1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8352
EGFREGFRTK5gtyBA1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8360
EGFREGFRTK5gtyBB1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8367
EGFREGFRTK5gtyCA1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8366
EGFREGFRTK5gtyCB1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8358
EGFREGFRTK5gtyDA1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8356
EGFREGFRTK5gtyDB1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8368
EGFREGFRTK5gtyEA1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8359
EGFREGFRTK5gtyEB1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8353
EGFREGFRTK5gtyFA1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8354
EGFREGFRTK5gtyFB1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8364
EGFREGFRTK5gtyGA1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8355
EGFREGFRTK5gtyGB1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8369
EGFREGFRTK5gtyHA1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8362
EGFREGFRTK5gtyHB1-[(3r)-3-[4-azanyl-3-[3-chloranyl-4-[(6-methylpyridin-2-yl)methoxy]phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]prop-2-en-1-oneHuman8357
EGFREGFRTK5gtzAAn-[5-[[5-chloranyl-4-[(2-propan-2-ylsulfonylphenyl)amino]pyrimidin-2-yl]amino]-2-(4-ethylpiperazin-1-yl)-4-methoxy-phenyl]prop-2-enamideHuman8365
EGFREGFRTK5gtzABn-[5-[[5-chloranyl-4-[(2-propan-2-ylsulfonylphenyl)amino]pyrimidin-2-yl]amino]-2-(4-ethylpiperazin-1-yl)-4-methoxy-phenyl]prop-2-enamideHuman8361
EGFREGFRTK5hcxA~{n}-[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]-2-methyl-1-propan-2-yl-imidazo[4,5-c]pyridin-6-amineHuman7040
EGFREGFRTK5hcyA6-[[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]amino]-~{n}-(oxan-4-yl)-1-propan-2-yl-pyrrolo[3,2-c]pyridine-3-carboxamideHuman7039
EGFREGFRTK5hczA2-[1-[1-[(2~{s})-butan-2-yl]-6-[[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]amino]pyrazolo[4,3-c]pyridin-3-yl]azetidin-3-yl]propan-2-olHuman7041
EGFREGFRTK5hg5AAn-{3-[(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy]phenyl}propanamideHuman6375
EGFREGFRTK5hg5ABn-{3-[(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy]phenyl}propanamideHuman6376
EGFREGFRTK5hg7A1-{(3r,4r)-3-[({5-chloro-2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-methoxypyrrolidin-1-yl}propan-1-oneHuman6367
EGFREGFRTK5hg8AAn-[3-({2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)phenyl]propanamideHuman6380
EGFREGFRTK5hg8ABn-[3-({2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)phenyl]propanamideHuman6378
EGFREGFRTK5hg9AA1-[(3r,4r)-3-[({2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-(trifluoromethyl)pyrrolidin-1-yl]propan-1-oneHuman6379
EGFREGFRTK5hg9AB1-[(3r,4r)-3-[({2-[(1-methyl-1h-pyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}oxy)methyl]-4-(trifluoromethyl)pyrrolidin-1-yl]propan-1-oneHuman6377
EGFREGFRTK5hibAn-tert-butyl-5-{[(1-methyl-1h-pyrazol-5-yl)sulfonyl]amino}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman6490
EGFREGFRTK5hicAn-{2-[1-(cyclopropylsulfonyl)-1h-pyrazol-4-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-imidazo[4,5-c]pyridin-6-amineHuman6491
EGFREGFRTK5j9yAA(r)-1-(3-(4-amino-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-oneHuman6946
EGFREGFRTK5j9yAB(r)-1-(3-(4-amino-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-oneHuman6945
EGFREGFRTK5j9zA(r)-1-(3-(4-amino-3-(1-methyl-1h-indol-3-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-oneHuman6947
EGFREGFRTK5jebA3-(furan-2-yl)-n-[5-(furan-2-yl)-2-methoxyphenyl]-1h-pyrazolo[3,4-d]pyrimidin-4-amine Human7038
EGFREGFRTK5u8lAA4-[(4-{4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-6-[(prop-2-yn-1-yl)carbamoyl]pyrimidin-2-yl}piperazin-1-yl)methyl]benzene-1-sulfonyl fluorideHuman7387
EGFREGFRTK5u8lAB4-[(4-{4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-6-[(prop-2-yn-1-yl)carbamoyl]pyrimidin-2-yl}piperazin-1-yl)methyl]benzene-1-sulfonyl fluorideHuman7386
EGFREGFRTK5ug8AAn-[(3r,4r)-4-fluoro-1-{6-[(1-methyl-1h-pyrazol-4-yl)amino]-9-(propan-2-yl)-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman7519
EGFREGFRTK5ug8ABn-[(3r,4r)-4-fluoro-1-{6-[(1-methyl-1h-pyrazol-4-yl)amino]-9-(propan-2-yl)-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman7514
EGFREGFRTK5ug9AAn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-(propan-2-yl)-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman7512
EGFREGFRTK5ug9ABn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-(propan-2-yl)-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman7513
EGFREGFRTK5ugaAA4-(4-{[2-{[(3s)-1-acetylpyrrolidin-3-yl]amino}-9-(propan-2-yl)-9h-purin-6-yl]amino}phenyl)-1-methylpiperazin-1-iumHuman7517
EGFREGFRTK5ugaAB4-(4-{[2-{[(3s)-1-acetylpyrrolidin-3-yl]amino}-9-(propan-2-yl)-9h-purin-6-yl]amino}phenyl)-1-methylpiperazin-1-iumHuman7511
EGFREGFRTK5ugbA4-(4-{[2-{[(3s)-1-acetylpyrrolidin-3-yl]amino}-9-(propan-2-yl)-9h-purin-6-yl]amino}phenyl)-1-methylpiperazin-1-iumHuman7515
EGFREGFRTK5ugcAAn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman7516
EGFREGFRTK5ugcABn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman7518
EGFREGFRTK5uwdAn-(3-{[2-{[4-(4-acetylpiperazin-1-yl)-2-methoxyphenyl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]amino}phenyl)propanamideHuman8568
EGFREGFRTK5x26An2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9536
EGFREGFRTK5x27A9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9534
EGFREGFRTK5x28A9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9538
EGFREGFRTK5x2aAAn2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9545
EGFREGFRTK5x2aABn2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9530
EGFREGFRTK5x2aACn2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9539
EGFREGFRTK5x2aBAn2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9526
EGFREGFRTK5x2aBBn2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9548
EGFREGFRTK5x2aBCn2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9543
EGFREGFRTK5x2aCAn2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9537
EGFREGFRTK5x2aCBn2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9531
EGFREGFRTK5x2aCCn2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-9-propan-2-yl-purine-2,8-diamineHuman9547
EGFREGFRTK5x2aDAphosphoaminophosphonic acid-adenylate esterHuman9529
EGFREGFRTK5x2aDBphosphoaminophosphonic acid-adenylate esterHuman9532
EGFREGFRTK5x2aDCphosphoaminophosphonic acid-adenylate esterHuman9533
EGFREGFRTK5x2cAA9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9572
EGFREGFRTK5x2cAB9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9567
EGFREGFRTK5x2cAC9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9566
EGFREGFRTK5x2cBA9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9569
EGFREGFRTK5x2cBB9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9571
EGFREGFRTK5x2cBC9-cyclopentyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9570
EGFREGFRTK5x2fAA9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9540
EGFREGFRTK5x2fAB9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9535
EGFREGFRTK5x2fBA9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9546
EGFREGFRTK5x2fBB9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9541
EGFREGFRTK5x2fCA9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9527
EGFREGFRTK5x2fCB9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9542
EGFREGFRTK5x2fDA9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9544
EGFREGFRTK5x2fDB9-cyclohexyl-n2-[4-(4-methylpiperazin-1-yl)phenyl]-n8-phenyl-purine-2,8-diamineHuman9528
EGFREGFRTK5x2kAn-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamideHuman9568
EGFREGFRTK5xdkAn-[3-[[2-[[4-(4-ethanoylpiperazin-1-yl)-2-methoxy-phenyl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]prop-2-enamideHuman9065
EGFREGFRTK5xdlAn-[3-[[2-[[4-(4-ethanoylpiperazin-1-yl)-2-methoxy-phenyl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]prop-2-enamideHuman9066
EGFREGFRTK5xgmA12-(2-cyanoethyl)-6,7,12,13-tetrahydro-13-methyl-5-oxo-5h-indolo[2,3-a]pyrrolo[3,4-c]carbazoleHuman8552
EGFREGFRTK5xgnA12-(2-cyanoethyl)-6,7,12,13-tetrahydro-13-methyl-5-oxo-5h-indolo[2,3-a]pyrrolo[3,4-c]carbazoleHuman8553
EGFREGFRTK5xgnB-Human8554
EGFREGFRTK5y25A(2r)-n-[4-[(3-chloranyl-4-fluoranyl-phenyl)amino]-7-(3-morpholin-4-ylpropoxy)quinazolin-6-yl]-1-(2-fluoranylethanoyl)pyrrolidine-2-carboxamideHuman10373
EGFREGFRTK5y9tA6-ethyl-3-[[4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-5-[(3r)-1-prop-2-enoylpyrrolidin-3-yl]oxy-pyrazine-2-carboxamideHuman10053
EGFREGFRTK5yu9AA1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman9430
EGFREGFRTK5yu9AB1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman9428
EGFREGFRTK5yu9BA1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman9433
EGFREGFRTK5yu9BB1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman9434
EGFREGFRTK5yu9CA1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman9432
EGFREGFRTK5yu9CB1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman9427
EGFREGFRTK5yu9DA1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman9431
EGFREGFRTK5yu9DB1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}prop-2-en-1-oneHuman9429
EGFREGFRTK5ztoAn-{trans-4-[3-(2-chlorophenyl)-7-{[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]cyclohexyl}propanamideHuman11070
EGFREGFRTK5zwjA(2r)-2-(5-fluoro-2-hydroxyphenyl)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-(1,3-thiazol-2-yl)acetamideHuman10372
EGFREGFRTK6d8eA(4-fluorophenyl)methyl {2-[(1-methyl-1h-pyrazol-3-yl)amino]pyrimidin-4-yl}[3-(propanoylamino)phenyl]carbamateHuman10374
EGFREGFRTK6dukAAphosphoaminophosphonic acid-adenylate esterHuman11067
EGFREGFRTK6dukABphosphoaminophosphonic acid-adenylate esterHuman11066
EGFREGFRTK6dukBAphosphoaminophosphonic acid-adenylate esterHuman11060
EGFREGFRTK6dukBBphosphoaminophosphonic acid-adenylate esterHuman11069
EGFREGFRTK6dukCAphosphoaminophosphonic acid-adenylate esterHuman11061
EGFREGFRTK6dukCBphosphoaminophosphonic acid-adenylate esterHuman11068
EGFREGFRTK6dukDAphosphoaminophosphonic acid-adenylate esterHuman11064
EGFREGFRTK6dukDBphosphoaminophosphonic acid-adenylate esterHuman11062
EGFREGFRTK6dukEAphosphoaminophosphonic acid-adenylate esterHuman11058
EGFREGFRTK6dukEBphosphoaminophosphonic acid-adenylate esterHuman11059
EGFREGFRTK6dukFAphosphoaminophosphonic acid-adenylate esterHuman11065
EGFREGFRTK6dukFBphosphoaminophosphonic acid-adenylate esterHuman11063
EGFREGFRTK6jrjA6-(2-chloranyl-3-fluoranyl-phenyl)-5-methyl-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[(3s)-1-propanoylpiperidin-3-yl]pyrido[2,3-d]pyrimidin-7-oneHuman12158
EGFREGFRTK6jrkA6-(2-chloranyl-3-fluoranyl-phenyl)-5-methyl-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[(3s)-1-propanoylpiperidin-3-yl]pyrido[2,3-d]pyrimidin-7-oneHuman12159
EGFREGFRTK6jrxAn-{trans-4-[3-(2-chlorophenyl)-7-{[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]cyclohexyl}propanamideHuman12157
EGFREGFRTK6jwlAn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHuman12173
EGFREGFRTK6jx0An-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHuman12175
EGFREGFRTK6jx4An-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHuman12176
EGFREGFRTK6jxtAAn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHuman12240
EGFREGFRTK6jxtABn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHuman12239
EGFREGFRTK6jz0Ae-4-(dimethylamino)-n-[3-[4-[[(1s)-2-oxidanyl-1-phenyl-ethyl]amino]-6-phenyl-furo[2,3-d]pyrimidin-5-yl]phenyl]but-2-enamideHuman11845
EGFREGFRTK6lubAAn-[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]-7-(4-methylpiperazin-1-yl)-5-propan-2-yl-9-[2,2,2-tris(fluoranyl)ethoxy]pyrido[4,3-b]indol-3-amineHuman12918
EGFREGFRTK6lubABn-[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]-7-(4-methylpiperazin-1-yl)-5-propan-2-yl-9-[2,2,2-tris(fluoranyl)ethoxy]pyrido[4,3-b]indol-3-amineHuman12917
EGFREGFRTK6ludAn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHuman12919
EGFREGFRTK6p1dAAphosphoaminophosphonic acid-adenylate esterHuman11872
EGFREGFRTK6p1dABphosphoaminophosphonic acid-adenylate esterHuman11868
EGFREGFRTK6p1dBAphosphoaminophosphonic acid-adenylate esterHuman11873
EGFREGFRTK6p1dBBphosphoaminophosphonic acid-adenylate esterHuman11883
EGFREGFRTK6p1dCA10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman11880
EGFREGFRTK6p1dCB10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman11869
EGFREGFRTK6p1dDA10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman11884
EGFREGFRTK6p1dDB10-benzyl-8-fluoro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman11885
EGFREGFRTK6p1lAphosphoaminophosphonic acid-adenylate esterHuman11878
EGFREGFRTK6p1lBphosphoaminophosphonic acid-adenylate esterHuman11886
EGFREGFRTK6p1lCphosphoaminophosphonic acid-adenylate esterHuman11876
EGFREGFRTK6p1lDphosphoaminophosphonic acid-adenylate esterHuman11870
EGFREGFRTK6p8qAAphosphoaminophosphonic acid-adenylate esterHuman11875
EGFREGFRTK6p8qABphosphoaminophosphonic acid-adenylate esterHuman11882
EGFREGFRTK6p8qBAadenosine monophosphateHuman11867
EGFREGFRTK6p8qBBadenosine monophosphateHuman11874
EGFREGFRTK6p8qCAadenosine monophosphateHuman11881
EGFREGFRTK6p8qCBadenosine monophosphateHuman11879
EGFREGFRTK6p8qDAadenosine monophosphateHuman11871
EGFREGFRTK6p8qDBadenosine monophosphateHuman11877
EGFREGFRTK6s89A~{n}-[3-[6-[4-(4-methylpiperazin-1-yl)phenyl]-4-propan-2-yloxy-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamideHuman11729
EGFREGFRTK6s8aA~{n}-[3-[6-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-methylpropoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamideHuman11728
EGFREGFRTK6s9bA3-fluoranyl-~{n}-[1-(2-methyl-2-oxidanyl-propyl)benzimidazol-2-yl]-5-pyridin-3-yl-benzamideHuman11805
EGFREGFRTK6s9cAA~{n}-[1-(2-methyl-2-oxidanyl-propyl)benzimidazol-2-yl]-2-phenyl-pyridine-4-carboxamideHuman11806
EGFREGFRTK6s9cAB~{n}-[1-(2-methyl-2-oxidanyl-propyl)benzimidazol-2-yl]-2-phenyl-pyridine-4-carboxamideHuman11804
EGFREGFRTK6s9dA8-oxa-14,21,23,28-tetraazapentacyclo[23.3.1.02,7.014,22.015,20]nonacosa-1(28),2(7),3,5,15,17,19,21,25(29),26-decaen-24-oneHuman11803
EGFREGFRTK6tfuA~{n}-[3-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamideHuman12844
EGFREGFRTK6tfuB~{n}-[3-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamideHuman12842
EGFREGFRTK6tfvAA~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamideHuman12828
EGFREGFRTK6tfvAB~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamideHuman12832
EGFREGFRTK6tfvBA~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamideHuman12845
EGFREGFRTK6tfvBB~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamideHuman12827
EGFREGFRTK6tfwA~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamideHuman12838
EGFREGFRTK6tfwB~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamideHuman12837
EGFREGFRTK6tfyAA~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamideHuman12825
EGFREGFRTK6tfyAB~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamideHuman12841
EGFREGFRTK6tfyBA~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamideHuman12847
EGFREGFRTK6tfyBB~{n}-[5-[4-[[3-chloranyl-4-(pyridin-2-ylmethoxy)phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(3-oxidanylpropoxy)phenyl]propanamideHuman12831
EGFREGFRTK6tfzAA~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamideHuman12840
EGFREGFRTK6tfzAB~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamideHuman12846
EGFREGFRTK6tfzBA~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamideHuman12830
EGFREGFRTK6tfzBB~{n}-[2-(2-hydroxyethyloxy)-5-[4-[[1-(phenylmethyl)indazol-5-yl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]phenyl]propanamideHuman12839
EGFREGFRTK6tg0AA~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamideHuman12833
EGFREGFRTK6tg0AB~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamideHuman12829
EGFREGFRTK6tg0BA~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamideHuman12834
EGFREGFRTK6tg0BB~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-(2-hydroxyethyloxy)phenyl]propanamideHuman12835
EGFREGFRTK6tg1AA~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamideHuman12826
EGFREGFRTK6tg1AB~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamideHuman12843
EGFREGFRTK6tg1BA~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamideHuman12836
EGFREGFRTK6tg1BB~{n}-[5-[4-[[4-[[1,3-bis(oxidanylidene)isoindol-2-yl]methyl]phenyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-2-[2-(dimethylamino)ethoxy]phenyl]propanamideHuman12824
EGFREGFRTK6v5nAA3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-olHuman12170
EGFREGFRTK6v5nAB3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-olHuman12180
EGFREGFRTK6v5nBA3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-olHuman12227
EGFREGFRTK6v5nBB3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-olHuman12185
EGFREGFRTK6v5nCA3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-olHuman12197
EGFREGFRTK6v5nCB3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-olHuman12196
EGFREGFRTK6v5nDA3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-olHuman12199
EGFREGFRTK6v5nDB3-[4-(4-fluorophenyl)-5-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)-1h-imidazol-2-yl]propan-1-olHuman12201
EGFREGFRTK6v5pAA4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridineHuman12174
EGFREGFRTK6v5pAB4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridineHuman12172
EGFREGFRTK6v5pBA4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridineHuman12203
EGFREGFRTK6v5pBB4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridineHuman12200
EGFREGFRTK6v5pCA4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridineHuman12210
EGFREGFRTK6v5pCB4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridineHuman12192
EGFREGFRTK6v5pDA4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridineHuman12218
EGFREGFRTK6v5pDB4-[4-(4-fluorophenyl)-2-(3-methoxypropyl)-1h-imidazol-5-yl]-2-phenyl-3h-pyrrolo[2,3-b]pyridineHuman12186
EGFREGFRTK6v66AAn-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamideHuman12178
EGFREGFRTK6v66ABn-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamideHuman12177
EGFREGFRTK6v66BAn-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamideHuman12205
EGFREGFRTK6v66BBn-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamideHuman12217
EGFREGFRTK6v66CAn-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamideHuman12184
EGFREGFRTK6v66CBn-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamideHuman12208
EGFREGFRTK6v66DAn-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamideHuman12221
EGFREGFRTK6v66DBn-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamideHuman12224
EGFREGFRTK6v6kAAn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12179
EGFREGFRTK6v6kABn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12168
EGFREGFRTK6v6kBAn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12202
EGFREGFRTK6v6kBBn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12229
EGFREGFRTK6v6kCAn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12207
EGFREGFRTK6v6kCBn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12209
EGFREGFRTK6v6kDAn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12223
EGFREGFRTK6v6kDBn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12212
EGFREGFRTK6v6kEAn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12187
EGFREGFRTK6v6kEBn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12193
EGFREGFRTK6v6kFAn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12204
EGFREGFRTK6v6kFBn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12214
EGFREGFRTK6v6kGAn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12195
EGFREGFRTK6v6kGBn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12222
EGFREGFRTK6v6kHAn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12216
EGFREGFRTK6v6kHBn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12190
EGFREGFRTK6v6oAAn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12169
EGFREGFRTK6v6oABn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12181
EGFREGFRTK6v6oBAn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12198
EGFREGFRTK6v6oBBn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12228
EGFREGFRTK6v6oCAn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12188
EGFREGFRTK6v6oCBn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12226
EGFREGFRTK6v6oDAn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12213
EGFREGFRTK6v6oDBn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12219
EGFREGFRTK6v6oEAn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12225
EGFREGFRTK6v6oEBn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12191
EGFREGFRTK6v6oFAn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12206
EGFREGFRTK6v6oFBn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12220
EGFREGFRTK6v6oGAn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12215
EGFREGFRTK6v6oGBn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12189
EGFREGFRTK6v6oHAn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12194
EGFREGFRTK6v6oHBn-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12211
EGFREGFRTK6vh4An-[3-({4-[4-(4-fluorophenyl)-2-(3-hydroxypropyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12183
EGFREGFRTK6vhnAn-[3-({4-[4-(4-fluorophenyl)-2-(methylsulfanyl)-1h-imidazol-5-yl]pyridin-2-yl}amino)-4-methoxyphenyl]propanamideHuman12171
EGFREGFRTK6vhpAn-{3-[(4-{4-(4-fluorophenyl)-2-[(2-methoxyethyl)sulfanyl]-1h-imidazol-5-yl}pyridin-2-yl)amino]-4-methoxyphenyl}propanamideHuman12182
EGFREGFRTK6wa2AAn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamideHuman13434
EGFREGFRTK6wa2ABn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamideHuman13442
EGFREGFRTK6wa2BAn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamideHuman13443
EGFREGFRTK6wa2BBn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamideHuman13444
EGFREGFRTK6wa2CAn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamideHuman13447
EGFREGFRTK6wa2CBn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamideHuman13436
EGFREGFRTK6wa2DAn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamideHuman13439
EGFREGFRTK6wa2DBn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-fluoro-5-hydroxybenzamideHuman13437
EGFREGFRTK6wakAAphosphoaminophosphonic acid-adenylate esterHuman13438
EGFREGFRTK6wakABphosphoaminophosphonic acid-adenylate esterHuman13440
EGFREGFRTK6wakBAphosphoaminophosphonic acid-adenylate esterHuman13435
EGFREGFRTK6wakBBphosphoaminophosphonic acid-adenylate esterHuman13448
EGFREGFRTK6wakCAn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-[(1-oxo-1,3-dihydro-2h-isoindol-2-yl)methyl]benzamideHuman13449
EGFREGFRTK6wakCBn-(3-{5-[2-(acetylamino)pyridin-4-yl]-2-(methylsulfanyl)-1h-imidazol-4-yl}phenyl)-2-[(1-oxo-1,3-dihydro-2h-isoindol-2-yl)methyl]benzamideHuman13441
EGFREGFRTK6wakDAphosphoaminophosphonic acid-adenylate esterHuman13446
EGFREGFRTK6wakDBphosphoaminophosphonic acid-adenylate esterHuman13445
EGFREGFRTK6wxnAA-Human13558
EGFREGFRTK6wxnAB-Human13557
EGFREGFRTK6xl4A~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamideHuman13759
EGFREGFRTK6z4bAA~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamideHuman12975
EGFREGFRTK6z4bAB~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamideHuman12974
EGFREGFRTK6z4dAAn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman12971
EGFREGFRTK6z4dABn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman12972
EGFREGFRTK6z4dBAn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman12979
EGFREGFRTK6z4dBBn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman12978
EGFREGFRTK7a2aAA(2r)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-2-phenyl-n-(1,3-thiazol-2-yl)acetamideHuman12977
EGFREGFRTK7a2aAB(2r)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-2-phenyl-n-(1,3-thiazol-2-yl)acetamideHuman12976
EGFREGFRTK7a2aBA(2r)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-2-phenyl-n-(1,3-thiazol-2-yl)acetamideHuman12970
EGFREGFRTK7a2aBB(2r)-2-(1-oxo-1,3-dihydro-2h-isoindol-2-yl)-2-phenyl-n-(1,3-thiazol-2-yl)acetamideHuman12973
EGFREGFRTK7a6iA~{n}-[5-[4-chloranyl-2-[4-(4-methylpiperazin-1-yl)phenyl]-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]-2-methyl-phenyl]propanamideHuman14123
EGFREGFRTK7a6jAA1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-oneHuman14125
EGFREGFRTK7a6jAB1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-oneHuman14124
EGFREGFRTK7a6kAApropan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylateHuman14111
EGFREGFRTK7a6kABpropan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylateHuman14113
EGFREGFRTK7a6kACpropan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylateHuman14112
EGFREGFRTK7aeiA5-chloranyl-~{n}2-[4-[4-(dimethylamino)piperidin-1-yl]-2-methoxy-5-(1-methylpyrazol-4-yl)phenyl]-~{n}4-(2-dimethylphosphorylphenyl)pyrimidine-2,4-diamineHuman13619
EGFREGFRTK7aemA5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamineHuman13482
EGFREGFRTK7b85Apropan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylateHuman14121
EGFREGFRTK7er2A5-chloranyl-n2-[3-chloranyl-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n4-(2-dimethylphosphorylphenyl)pyrimidine-2,4-diamineHuman14194
EGFREGFRTK7jxiAAn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman13885
EGFREGFRTK7jxiABn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman13882
EGFREGFRTK7jxkAAn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman13884
EGFREGFRTK7jxkABn-[(3r,4r)-4-fluoro-1-{6-[(3-methoxy-1-methyl-1h-pyrazol-4-yl)amino]-9-methyl-9h-purin-2-yl}pyrrolidin-3-yl]propanamideHuman13876
EGFREGFRTK7jxlAAn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-5-{[4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-4-methoxyphenyl)propanamideHuman13878
EGFREGFRTK7jxlABn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-5-{[4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-4-methoxyphenyl)propanamideHuman13879
EGFREGFRTK7jxmAphosphoaminophosphonic acid-adenylate esterHuman13883
EGFREGFRTK7jxpAAphosphoaminophosphonic acid-adenylate esterHuman13881
EGFREGFRTK7jxpABphosphoaminophosphonic acid-adenylate esterHuman13874
EGFREGFRTK7jxqAA(2r)-2-(5-fluoro-2-hydroxyphenyl)-2-{6-[4-(1-methylpiperidin-4-yl)phenyl]-1-oxo-1,3-dihydro-2h-isoindol-2-yl}-n-(1,3-thiazol-2-yl)acetamideHuman13886
EGFREGFRTK7jxqAB(2r)-2-(5-fluoro-2-hydroxyphenyl)-2-{6-[4-(1-methylpiperidin-4-yl)phenyl]-1-oxo-1,3-dihydro-2h-isoindol-2-yl}-n-(1,3-thiazol-2-yl)acetamideHuman13880
EGFREGFRTK7jxwAAn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHuman13875
EGFREGFRTK7jxwABn-(2-{[2-(dimethylamino)ethyl](methyl)amino}-4-methoxy-5-{[4-(1-methyl-1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)prop-2-enamideHuman13877
EGFREGFRTK7k1hA(2r)-2-(5-fluoro-2-hydroxyphenyl)-2-{6-[4-(1-methylpiperidin-4-yl)phenyl]-1-oxo-1,3-dihydro-2h-isoindol-2-yl}-n-(1,3-thiazol-2-yl)acetamideHuman13902
EGFREGFRTK7k1iAAphosphoaminophosphonic acid-adenylate esterHuman13904
EGFREGFRTK7k1iABphosphoaminophosphonic acid-adenylate esterHuman13903
EGFREGFRTK7kxzA(20r)-10,15,20-trimethyl-2-[(4-methylpiperazin-1-yl)methyl]-18,19,20,21-tetrahydro-15h,17h-12,8-(metheno)pyrazolo[3',4':2,3][1,5,10,12]oxatriazacycloheptadecino[12,11-a]benzimidazol-7(6h)-oneHuman14074
EGFREGFRTK7ky0A(20r)-10,15,20-trimethyl-2-[(4-methylpiperazin-1-yl)methyl]-18,19,20,21-tetrahydro-15h,17h-12,8-(metheno)pyrazolo[3',4':2,3][1,5,10,12]oxatriazacycloheptadecino[12,11-a]benzimidazol-7(6h)-oneHuman14073
EGFREGFRTK7lg8A6-ethyl-3-[[4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-5-[(3r)-1-prop-2-enoylpyrrolidin-3-yl]oxy-pyrazine-2-carboxamideHuman14120
EGFREGFRTK7lgsAA~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamideHuman13906
EGFREGFRTK7lgsAB~{n}-[2-[2-(dimethylamino)ethyl-methyl-amino]-4-methoxy-5-[[4-(1-methylindol-3-yl)pyrimidin-2-yl]amino]phenyl]propanamideHuman13905
EGFREGFRTK7ltxAphosphoaminophosphonic acid-adenylate esterHuman14122
EGFREGFRTK7oxbA2-[2-(3-methoxyphenyl)pyrimidin-4-yl]-1'-prop-2-enoyl-spiro[5,6-dihydro-1~{h}-pyrrolo[3,2-c]pyridine-7,4'-piperidine]-4-oneHuman13948
EGFREGFRTK7si1AA-Human14478
EGFREGFRTK7si1AB-Human14480
EGFREGFRTK7si1AC-Human14479
EGFREGFRTK7sydAB-Human14027
EGFREGFRTK7syeA-Human14028
EGFREGFRTK7sz0AB-Human14031
EGFREGFRTK7sz1A-Human14029
EGFREGFRTK7sz5A-Human14030
EGFREGFRTK7sz7A-Human14016
EGFREGFRTK7t4iApropan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylateHuman14530
EGFREGFRTK7t4jApropan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylateHuman14529
EGFREGFRTK7tvdA-Human14107
EGFREGFRTK7u98A19-chloro-18-fluoro-22-methoxy-8,9,11,12,14,15-hexahydro-21h-4,6-ethenopyrimido[5,4-m][1,4,7,10,15]benzotetraoxazacycloheptadecineHuman14526
EGFREGFRTK7u99A19-chloro-22-methoxy-8,9,11,12,14,15-hexahydro-21h-4,6-ethenopyrimido[5,4-m][1,4,7,10,15]benzotetraoxazacycloheptadecineHuman14533
EGFREGFRTK7u9aA4-(5-chloro-4-fluoro-2-hydroxyanilino)-7-methoxyquinazolin-6-olHuman14527
EGFREGFRTK7ukvAn-[5-{[(4p)-4-{4-[(dimethylamino)methyl]-3-phenyl-1h-pyrazol-1-yl}pyrimidin-2-yl]amino}-4-methoxy-2-(morpholin-4-yl)phenyl]propanamideHuman14528
EGFREGFRTK7ukwAA-Human14531
EGFREGFRTK7ukwAB-Human14532
EGFREGFRTK7vraAA25-chloro-11-(ethylsulfonyl)-44-morpholino-11h-5,12-dioxa-3-aza-1(3,6)-indola-2(4,2)-pyrimidina-4(1,3)-benzenacyclododecaphaneHuman14235
EGFREGFRTK7vraAB25-chloro-11-(ethylsulfonyl)-44-morpholino-11h-5,12-dioxa-3-aza-1(3,6)-indola-2(4,2)-pyrimidina-4(1,3)-benzenacyclododecaphaneHuman14237
EGFREGFRTK7vreA5-chloranyl-n-[5-chloranyl-2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-4-(1-ethylsulfonylindol-3-yl)pyrimidin-2-amineHuman14236
EGFREGFRTK7zymA5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamineHuman14726
EGFREGFRTK7zynAAn-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamideHuman14727
EGFREGFRTK7zynABn-{3-[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamideHuman14728
EGFREGFRTK7zypApropan-2-yl 2-[[4-(4-azanylpiperidin-1-yl)-2-methoxy-phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylateHuman14731
EGFREGFRTK7zyqAAphenyl 2-[[4-[4-(dimethylamino)piperidin-1-yl]-2-methoxy-phenyl]amino]-4-(1h-indol-3-yl)pyrimidine-5-carboxylateHuman14730
EGFREGFRTK7zyqABphenyl 2-[[4-[4-(dimethylamino)piperidin-1-yl]-2-methoxy-phenyl]amino]-4-(1h-indol-3-yl)pyrimidine-5-carboxylateHuman14729
EGFREGFRTK8a27AA(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHuman14462
EGFREGFRTK8a27AB(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHuman14465
EGFREGFRTK8a2aAA(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHuman14466
EGFREGFRTK8a2aAB(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHuman14460
EGFREGFRTK8a2bAA(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHuman14464
EGFREGFRTK8a2bAB(2r)-2-(6,7-dihydro-5h-pyrrolo[1,2-c]imidazol-1-yl)-2-[5-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-3-oxidanylidene-7-(trifluoromethyl)-1h-isoindol-2-yl]-n-(1,3-thiazol-2-yl)ethanamideHuman14459
EGFREGFRTK8a2dAA(2r)-2-[4-[bis(fluoranyl)methyl]-6-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-7-methyl-indazol-2-yl]-2-spiro[6,7-dihydropyrrolo[1,2-c]imidazole-5,1'-cyclopropane]-1-yl-n-(1,3-thiazol-2-yl)ethanamideHuman14463
EGFREGFRTK8a2dAB(2r)-2-[4-[bis(fluoranyl)methyl]-6-[2-[4-[[4-(hydroxymethyl)piperidin-1-yl]methyl]phenyl]ethynyl]-7-methyl-indazol-2-yl]-2-spiro[6,7-dihydropyrrolo[1,2-c]imidazole-5,1'-cyclopropane]-1-yl-n-(1,3-thiazol-2-yl)ethanamideHuman14461
EGFREGFRTK8d73AA(3s,4r)-3-fluoro-1-(4-{[4-(methylamino)-1-(propan-2-yl)pyrido[3,4-d]pyridazin-7-yl]amino}pyrimidin-2-yl)piperidin-4-olHuman14312
EGFREGFRTK8d73AB(3s,4r)-3-fluoro-1-(4-{[4-(methylamino)-1-(propan-2-yl)pyrido[3,4-d]pyridazin-7-yl]amino}pyrimidin-2-yl)piperidin-4-olHuman14310
EGFREGFRTK8d76AA(3s,4r)-3-fluoro-1-(4-{[8-{3-[(methanesulfonyl)methyl]azetidin-1-yl}-5-(propan-2-yl)-2,7-naphthyridin-3-yl]amino}pyrimidin-2-yl)-3-methylpiperidin-4-olHuman14311
EGFREGFRTK8d76AB(3s,4r)-3-fluoro-1-(4-{[8-{3-[(methanesulfonyl)methyl]azetidin-1-yl}-5-(propan-2-yl)-2,7-naphthyridin-3-yl]amino}pyrimidin-2-yl)-3-methylpiperidin-4-olHuman14313
EGFREGFRTK8dswAphosphoaminophosphonic acid-adenylate esterHuman14946
EGFREGFRTK8emeA-Human14938
EGFREGFRTK8f1hAn-[(5p,8s,10r)-4-amino-6-methyl-5-(quinolin-3-yl)-8,9-dihydropyrimido[5,4-b]indolizin-8-yl]prop-2-enamideHuman14947
EGFREGFRTK8f1wA1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-oneHuman14944
EGFREGFRTK8f1xAApropan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylateHuman14942
EGFREGFRTK8f1xABpropan-2-yl 2-[[4-[2-(dimethylamino)ethyl-methyl-amino]-2-methoxy-5-(propanoylamino)phenyl]amino]-4-(1-methylindol-3-yl)pyrimidine-5-carboxylateHuman14943
EGFREGFRTK8f1yA1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-oneHuman14940
EGFREGFRTK8f1zA(2p)-3-(3-chloro-2-methoxyanilino)-2-[3-(2-methoxy-2-methylpropoxy)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman14939
EGFREGFRTK8fv3AAphosphoaminophosphonic acid-adenylate esterHuman15168
EGFREGFRTK8fv3ABphosphoaminophosphonic acid-adenylate esterHuman15167
EGFREGFRTK8fv4AAphosphoaminophosphonic acid-adenylate esterHuman15166
EGFREGFRTK8fv4ABphosphoaminophosphonic acid-adenylate esterHuman15165
EGFREGFRTK8g63AralimetinibHuman14937
EGFREGFRTK8h7xA5-chloro-n~4~-[2-(dimethylphosphoryl)phenyl]-n~2~-{2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl}pyrimidine-2,4-diamineHuman14945
EGFREGFRTK8hv1A3-(3-bromophenyl)-1,4-dihydro-1,2,4-triazole-5-thioneHuman15072
EGFREGFRTK8hv2AA~{n}-pyridin-2-ylprop-2-enamideHuman15077
EGFREGFRTK8hv2AB~{n}-pyridin-2-ylprop-2-enamideHuman15068
EGFREGFRTK8hv3A~{n}-pyridin-2-ylprop-2-enamideHuman15067
EGFREGFRTK8hv4A~{n}-pyridin-2-ylprop-2-enamideHuman15075
EGFREGFRTK8hv5AA~{n}-(1-methylbenzimidazol-4-yl)prop-2-enamideHuman15069
EGFREGFRTK8hv5AB~{n}-(1-methylbenzimidazol-4-yl)prop-2-enamideHuman15065
EGFREGFRTK8hv6AA~{n}-quinolin-7-ylprop-2-enamideHuman15071
EGFREGFRTK8hv6AB~{n}-quinolin-7-ylprop-2-enamideHuman15064
EGFREGFRTK8hv7A~{n}-[7-(dimethylamino)-2-methyl-pyrazolo[1,5-a]pyrimidin-5-yl]prop-2-enamideHuman15066
EGFREGFRTK8hv8A~{n}-pyrazolo[1,5-a]pyridin-2-ylprop-2-enamideHuman15073
EGFREGFRTK8hv9AA~{n}-(4-phenylpyridin-2-yl)prop-2-enamideHuman15063
EGFREGFRTK8hv9AB~{n}-(4-phenylpyridin-2-yl)prop-2-enamideHuman15070
EGFREGFRTK8hvaA~{n}-[6-(1-methylindol-3-yl)pyrimidin-4-yl]prop-2-enamideHuman15076
EGFREGFRTK8hy7A~{n}-[3-[[6-fluoranyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]quinazolin-4-yl]amino]phenyl]prop-2-enamideHuman14941
EGFREGFRTK8wd4A~{n}-[3,3-bis(fluoranyl)propyl]-4-[[(2~{s})-butan-2-yl]amino]-6-[[2-(1-cyclopropylsulfonylpyrazol-4-yl)pyrimidin-4-yl]amino]pyridine-3-carboxamideHuman15074
EIF2AK2 (PKR)PEKOther2a19Bphosphoaminophosphonic acid-adenylate esterHuman920
EIF2AK2 (PKR)PEKOther2a19Cphosphoaminophosphonic acid-adenylate esterHuman918
EIF2AK2 (PKR)PEKOther2a1aB-Human919
EIF2AK2 (PKR)PEKOther3uiuA-Human917
EIF2AK2 (PKR)PEKOther3uiuB-Human916
EIF2AK2 (PKR)PEKOther6d3kAadenosine-5'-diphosphateHuman11386
EIF2AK2 (PKR)PEKOther6d3kBadenosine-5'-diphosphateHuman11385
EIF2AK2 (PKR)PEKOther6d3kCadenosine-5'-diphosphateHuman11387
EIF2AK2 (PKR)PEKOther6d3lA-Human11384
EIF2AK2 (PKR)PEKOther8qelB(3~{z})-3-[(4-methyl-1~{h}-imidazol-5-yl)methylidene]-2-oxidanylidene-1~{h}-indole-5-carboxamideHuman14954
Eif2ak3 (PEK)PEKOther3qd2B-Mouse5802
EIF2AK3 (PEK)PEKOther4g31AA1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanoneHuman2672
EIF2AK3 (PEK)PEKOther4g31AB1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanoneHuman2671
EIF2AK3 (PEK)PEKOther4g34AA1-[5-(4-aminothieno[3,2-c]pyridin-3-yl)-2,3-dihydro-1h-indol-1-yl]-2-phenylethanoneHuman2674
EIF2AK3 (PEK)PEKOther4g34AB1-[5-(4-aminothieno[3,2-c]pyridin-3-yl)-2,3-dihydro-1h-indol-1-yl]-2-phenylethanoneHuman2670
EIF2AK3 (PEK)PEKOther4m7iA1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-1h-indol-1-yl]-2-(6-methylpyridin-2-yl)ethanoneHuman2673
EIF2AK3 (PEK)PEKOther4x7hAAn-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1h-pyrazole-4-carboxamideHuman7247
EIF2AK3 (PEK)PEKOther4x7hABn-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1h-pyrazole-4-carboxamideHuman7240
EIF2AK3 (PEK)PEKOther4x7jAA2-amino-n-[4-methoxy-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamideHuman6848
EIF2AK3 (PEK)PEKOther4x7jAB2-amino-n-[4-methoxy-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamideHuman6841
EIF2AK3 (PEK)PEKOther4x7kAA4-{2-amino-3-[5-fluoro-2-(methylamino)quinazolin-6-yl]-4-methylbenzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman7246
EIF2AK3 (PEK)PEKOther4x7kAB4-{2-amino-3-[5-fluoro-2-(methylamino)quinazolin-6-yl]-4-methylbenzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman7242
EIF2AK3 (PEK)PEKOther4x7lAA4-{2-amino-4-methyl-3-[2-(methylamino)-1,3-benzothiazol-6-yl]benzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman6844
EIF2AK3 (PEK)PEKOther4x7lAB4-{2-amino-4-methyl-3-[2-(methylamino)-1,3-benzothiazol-6-yl]benzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman6843
EIF2AK3 (PEK)PEKOther4x7nAA4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman7245
EIF2AK3 (PEK)PEKOther4x7nAB4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman7241
EIF2AK3 (PEK)PEKOther4x7oAA1-[5-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanoneHuman7243
EIF2AK3 (PEK)PEKOther4x7oAB1-[5-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanoneHuman7244
EIF2AK3 (PEK)PEKOther7mf0A2-amino-n-cyclopropyl-5-(4-{[(2r)-2-(3,5-difluorophenyl)-2-hydroxyacetyl]amino}-2-methylphenyl)pyridine-3-carboxamideHuman13577
EIF2AK3 (PEK)PEKOther8eq9AA(2r)-n-[(4m)-4-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamideHuman14524
EIF2AK3 (PEK)PEKOther8eq9AB(2r)-n-[(4m)-4-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamideHuman14521
EIF2AK3 (PEK)PEKOther8eqdA(2r)-n-[(4m)-4-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamideHuman14523
EIF2AK3 (PEK)PEKOther8eqeA(2r)-n-[(4m)-4-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-hydroxy-2-[3-(trifluoromethyl)phenyl]acetamideHuman14522
EIF2AK4 (GCN2)PEKOther6n3lAAn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHuman11691
EIF2AK4 (GCN2)PEKOther6n3lABn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHuman11694
EIF2AK4 (GCN2)PEKOther6n3lBAn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHuman11693
EIF2AK4 (GCN2)PEKOther6n3lBBn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHuman11692
EIF2AK4 (GCN2)PEKOther6n3nAn-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-2,5-dichloro-3-(hydroxymethyl)benzene-1-sulfonamideHuman11690
EIF2AK4 (GCN2)PEKOther6n3oAn-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-5-chloro-2-methoxypyridine-3-sulfonamideHuman11695
EIF2AK4 (GCN2)PEKOther7qq6A4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman14116
EIF2AK4 (GCN2)PEKOther7qwkA(2~{s})-~{n}-[(1~{s})-1-[4-[(6-pyridin-4-ylquinazolin-2-yl)amino]phenyl]ethyl]piperidine-2-carboxamideHuman14209
EPHA2 (EphA2)EphTK1mqbAphosphoaminophosphonic acid-adenylate esterHuman2088
EPHA2 (EphA2)EphTK1mqbBphosphoaminophosphonic acid-adenylate esterHuman2089
EPHA2 (EphA2)EphTK4p2kA-Human2091
EPHA2 (EphA2)EphTK4pdoA-Human2086
EPHA2 (EphA2)EphTK4pdoB-Human2087
EPHA2 (EphA2)EphTK4trlA-Human2090
EPHA2 (EphA2)EphTK5ek7A-Human6322
EPHA2 (EphA2)EphTK5ek7B-Human6321
EPHA2 (EphA2)EphTK5i9uAA-Human7190
EPHA2 (EphA2)EphTK5i9uAB-Human7185
EPHA2 (EphA2)EphTK5i9vAAphosphothiophosphoric acid-adenylate esterHuman7188
EPHA2 (EphA2)EphTK5i9vABphosphothiophosphoric acid-adenylate esterHuman7173
EPHA2 (EphA2)EphTK5i9wAAphosphoaminophosphonic acid-adenylate esterHuman7187
EPHA2 (EphA2)EphTK5i9wABphosphoaminophosphonic acid-adenylate esterHuman7178
EPHA2 (EphA2)EphTK5i9xAA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman7182
EPHA2 (EphA2)EphTK5i9xAB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman7177
EPHA2 (EphA2)EphTK5i9yAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7194
EPHA2 (EphA2)EphTK5i9yABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7176
EPHA2 (EphA2)EphTK5i9zAAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman7180
EPHA2 (EphA2)EphTK5i9zABn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman7181
EPHA2 (EphA2)EphTK5ia0AAalisertibHuman7169
EPHA2 (EphA2)EphTK5ia0ABalisertibHuman7171
EPHA2 (EphA2)EphTK5ia0BAalisertibHuman7174
EPHA2 (EphA2)EphTK5ia0BBalisertibHuman7179
EPHA2 (EphA2)EphTK5ia0CAalisertibHuman7186
EPHA2 (EphA2)EphTK5ia0CBalisertibHuman7175
EPHA2 (EphA2)EphTK5ia1A4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman7191
EPHA2 (EphA2)EphTK5ia2AA7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman7170
EPHA2 (EphA2)EphTK5ia2AB7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman7172
EPHA2 (EphA2)EphTK5ia3AA6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-oneHuman7193
EPHA2 (EphA2)EphTK5ia3AB6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-oneHuman7184
EPHA2 (EphA2)EphTK5ia4AAn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman7189
EPHA2 (EphA2)EphTK5ia4ABn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman7168
EPHA2 (EphA2)EphTK5ia5AAgolvatinibHuman7192
EPHA2 (EphA2)EphTK5ia5ABgolvatinibHuman7183
EPHA2 (EphA2)EphTK5njzAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8093
EPHA2 (EphA2)EphTK5njzAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8085
EPHA2 (EphA2)EphTK5nk0AA2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8095
EPHA2 (EphA2)EphTK5nk0AB2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8096
EPHA2 (EphA2)EphTK5nk1AA2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8064
EPHA2 (EphA2)EphTK5nk1AB2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8059
EPHA2 (EphA2)EphTK5nk2AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8100
EPHA2 (EphA2)EphTK5nk2AB-Human8060
EPHA2 (EphA2)EphTK5nk2AC~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8065
EPHA2 (EphA2)EphTK5nk3AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8092
EPHA2 (EphA2)EphTK5nk3AB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8080
EPHA2 (EphA2)EphTK5nk4AA2-[[3-[[(4~{r})-3,3-bis(fluoranyl)piperidin-4-yl]carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8070
EPHA2 (EphA2)EphTK5nk4AB2-[[3-[[(4~{r})-3,3-bis(fluoranyl)piperidin-4-yl]carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8076
EPHA2 (EphA2)EphTK5nk5AA2-[[3-[(3-aminophenyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8068
EPHA2 (EphA2)EphTK5nk5AB2-[[3-[(3-aminophenyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8066
EPHA2 (EphA2)EphTK5nk5AC-Human8091
EPHA2 (EphA2)EphTK5nk6AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(4-oxidanylcyclohexyl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8094
EPHA2 (EphA2)EphTK5nk6AB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(4-oxidanylcyclohexyl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8061
EPHA2 (EphA2)EphTK5nk7AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8089
EPHA2 (EphA2)EphTK5nk7AB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8081
EPHA2 (EphA2)EphTK5nk8AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(2,2,6,6-tetramethyl-1-oxidanyl-piperidin-4-yl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8062
EPHA2 (EphA2)EphTK5nk8AB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(2,2,6,6-tetramethyl-1-oxidanyl-piperidin-4-yl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8088
EPHA2 (EphA2)EphTK5nk9AA(2~{z})-~{n}-(2-chloranyl-6-methyl-phenyl)-2-[3-[(4-methyl-4-oxidanyl-cyclohexyl)carbamoyl]phenyl]imino-1,3-thiazolidine-5-carboxamideHuman8073
EPHA2 (EphA2)EphTK5nk9AB(2~{z})-~{n}-(2-chloranyl-6-methyl-phenyl)-2-[3-[(4-methyl-4-oxidanyl-cyclohexyl)carbamoyl]phenyl]imino-1,3-thiazolidine-5-carboxamideHuman8067
EPHA2 (EphA2)EphTK5nkaAA4-[[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylamino]cyclohexane-1-carboxylic acidHuman8075
EPHA2 (EphA2)EphTK5nkaAB4-[[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylamino]cyclohexane-1-carboxylic acidHuman8086
EPHA2 (EphA2)EphTK5nkaAC-Human8083
EPHA2 (EphA2)EphTK5nkbAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3,5-dimorpholin-4-ylphenyl)amino]-1,3-thiazole-5-carboxamideHuman8098
EPHA2 (EphA2)EphTK5nkbAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3,5-dimorpholin-4-ylphenyl)amino]-1,3-thiazole-5-carboxamideHuman8097
EPHA2 (EphA2)EphTK5nkcAA(3~{s})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidine-3-carboxylic acidHuman8099
EPHA2 (EphA2)EphTK5nkcAB(3~{s})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidine-3-carboxylic acidHuman8072
EPHA2 (EphA2)EphTK5nkdAA2-[(3~{r})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidin-3-yl]ethanoic acidHuman8058
EPHA2 (EphA2)EphTK5nkdAB2-[(3~{r})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidin-3-yl]ethanoic acidHuman8082
EPHA2 (EphA2)EphTK5nkeAA2-[[3-bromanyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8078
EPHA2 (EphA2)EphTK5nkeAB2-[[3-bromanyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8063
EPHA2 (EphA2)EphTK5nkfAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)-5-(trifluoromethyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8087
EPHA2 (EphA2)EphTK5nkfAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)-5-(trifluoromethyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8071
EPHA2 (EphA2)EphTK5nkgAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-ethyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8079
EPHA2 (EphA2)EphTK5nkgAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-ethyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8090
EPHA2 (EphA2)EphTK5nkhAA2-[[3-(2-aminophenyl)-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8074
EPHA2 (EphA2)EphTK5nkhAB2-[[3-(2-aminophenyl)-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8077
EPHA2 (EphA2)EphTK5nkiAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]-1,3-thiazole-5-carboxamideHuman8084
EPHA2 (EphA2)EphTK5nkiAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]-1,3-thiazole-5-carboxamideHuman8069
EPHA2 (EphA2)EphTK6fnfAA4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10417
EPHA2 (EphA2)EphTK6fnfAB4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10420
EPHA2 (EphA2)EphTK6fngAA4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10414
EPHA2 (EphA2)EphTK6fngAB4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10416
EPHA2 (EphA2)EphTK6fnhAA1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10422
EPHA2 (EphA2)EphTK6fnhAB1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10418
EPHA2 (EphA2)EphTK6fnhBA1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10421
EPHA2 (EphA2)EphTK6fnhBB1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10413
EPHA2 (EphA2)EphTK6fnhCA1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10415
EPHA2 (EphA2)EphTK6fnhCB1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10419
EPHA2 (EphA2)EphTK6hesAA4-methyl-3-[(2-pyridin-3-ylquinazolin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11550
EPHA2 (EphA2)EphTK6hesAB4-methyl-3-[(2-pyridin-3-ylquinazolin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11566
EPHA2 (EphA2)EphTK6hesAC-Human11554
EPHA2 (EphA2)EphTK6hetAA~{n}-(3-chlorophenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman11564
EPHA2 (EphA2)EphTK6hetAB~{n}-(3-chlorophenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman11560
EPHA2 (EphA2)EphTK6hetAC-Human11562
EPHA2 (EphA2)EphTK6heuAA3-[(4,6-dipyridin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11563
EPHA2 (EphA2)EphTK6heuAB3-[(4,6-dipyridin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11552
EPHA2 (EphA2)EphTK6hevAA4-methyl-3-[(2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11561
EPHA2 (EphA2)EphTK6hevAB4-methyl-3-[(2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11565
EPHA2 (EphA2)EphTK6hewAA4-methyl-3-[(1-methyl-6-pyrimidin-5-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11549
EPHA2 (EphA2)EphTK6hewAB4-methyl-3-[(1-methyl-6-pyrimidin-5-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11556
EPHA2 (EphA2)EphTK6hewAC-Human11553
EPHA2 (EphA2)EphTK6hexAA4-methyl-3-[(1-methyl-6-pyrazin-2-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11559
EPHA2 (EphA2)EphTK6hexAB4-methyl-3-[(1-methyl-6-pyrazin-2-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11555
EPHA2 (EphA2)EphTK6hexAC-Human11551
EPHA2 (EphA2)EphTK6heyAA3-[(4,6-dipyridin-3-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11557
EPHA2 (EphA2)EphTK6heyAB3-[(4,6-dipyridin-3-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11558
EPHA2 (EphA2)EphTK6q7bAA3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11927
EPHA2 (EphA2)EphTK6q7bAB3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11935
EPHA2 (EphA2)EphTK6q7cAA3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpiperidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11931
EPHA2 (EphA2)EphTK6q7cAB3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpiperidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11930
EPHA2 (EphA2)EphTK6q7dAA3-[[4-imidazol-1-yl-6-(4-oxidanylpiperidin-1-yl)-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11937
EPHA2 (EphA2)EphTK6q7dAB3-[[4-imidazol-1-yl-6-(4-oxidanylpiperidin-1-yl)-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11928
EPHA2 (EphA2)EphTK6q7eAA3-[[4-imidazol-1-yl-6-[(3~{r})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11926
EPHA2 (EphA2)EphTK6q7eAB3-[[4-imidazol-1-yl-6-[(3~{r})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11932
EPHA2 (EphA2)EphTK6q7fAA3-[(4-imidazol-1-yl-6-piperazin-1-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11929
EPHA2 (EphA2)EphTK6q7fAB3-[(4-imidazol-1-yl-6-piperazin-1-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11936
EPHA2 (EphA2)EphTK6q7gAA3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11933
EPHA2 (EphA2)EphTK6q7gAB3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11938
EPHA2 (EphA2)EphTK6q7gAC3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11934
EPHA2 (EphA2)EphTK7kjaAAphosphomethylphosphonic acid adenylate esterHuman13250
EPHA2 (EphA2)EphTK7kjaABphosphomethylphosphonic acid adenylate esterHuman13255
EPHA2 (EphA2)EphTK7kjaBAphosphomethylphosphonic acid adenylate esterHuman13249
EPHA2 (EphA2)EphTK7kjaBBphosphomethylphosphonic acid adenylate esterHuman13251
EPHA2 (EphA2)EphTK7kjbA-Human13253
EPHA2 (EphA2)EphTK7kjcAAphosphomethylphosphonic acid adenylate esterHuman13257
EPHA2 (EphA2)EphTK7kjcABphosphomethylphosphonic acid adenylate esterHuman13256
EPHA2 (EphA2)EphTK7kjcBAphosphomethylphosphonic acid adenylate esterHuman13252
EPHA2 (EphA2)EphTK7kjcBBphosphomethylphosphonic acid adenylate esterHuman13254
EPHA2 (EphA2)EphTK8binAA8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14514
EPHA2 (EphA2)EphTK8binAB8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14515
EPHA2 (EphA2)EphTK8binAC8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14512
EPHA2 (EphA2)EphTK8bioAB8-(4-azanylbutyl)-6-[2-chloranyl-5-(trifluoromethyl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14513
EPHA2 (EphA2)EphTK8bk0AA~{n}-(2-chlorophenyl)-6-piperidin-4-yl-imidazo[1,2-a]pyridine-3-carboxamideHuman14504
EPHA2 (EphA2)EphTK8bk0AB~{n}-(2-chlorophenyl)-6-piperidin-4-yl-imidazo[1,2-a]pyridine-3-carboxamideHuman14503
EPHA2 (EphA2)EphTK8bocAA~{n}-[3,5-bis(trifluoromethyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman15003
EPHA2 (EphA2)EphTK8bocAB~{n}-[3,5-bis(trifluoromethyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman15002
EPHA2 (EphA2)EphTK8bodAA~{n}-[3,5-bis(chloranyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14657
EPHA2 (EphA2)EphTK8bodAB~{n}-[3,5-bis(chloranyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14646
EPHA2 (EphA2)EphTK8bofAA4-methyl-~{n}-(3-methylphenyl)-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14656
EPHA2 (EphA2)EphTK8bofAB4-methyl-~{n}-(3-methylphenyl)-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14652
EPHA2 (EphA2)EphTK8bogAA~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamideHuman14650
EPHA2 (EphA2)EphTK8bogAB~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamideHuman14649
EPHA2 (EphA2)EphTK8bogAC~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamideHuman14654
EPHA2 (EphA2)EphTK8bohAA4-methyl-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14647
EPHA2 (EphA2)EphTK8bohAB4-methyl-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14651
EPHA2 (EphA2)EphTK8boiAA4-methyl-~{n}-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14645
EPHA2 (EphA2)EphTK8boiAB4-methyl-~{n}-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14655
EPHA2 (EphA2)EphTK8bokAA~{n}-(3,5-dimethoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14648
EPHA2 (EphA2)EphTK8bokAB~{n}-(3,5-dimethoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14659
EPHA2 (EphA2)EphTK8bomAA~{n}-(3-methoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14658
EPHA2 (EphA2)EphTK8bomAB~{n}-(3-methoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14653
EPHA2 (EphA2)EphTK8qqyAA6-(4-fluoranyl-3-methoxy-phenyl)-13$l^{6}-thia-2,4,8,12,19-pentazatricyclo[12.3.1.1^{3,7}]nonadeca-1(18),3,5,7(19),14,16-hexaene 13,13-dioxideHuman15001
EPHA2 (EphA2)EphTK8qqyAB6-(4-fluoranyl-3-methoxy-phenyl)-13$l^{6}-thia-2,4,8,12,19-pentazatricyclo[12.3.1.1^{3,7}]nonadeca-1(18),3,5,7(19),14,16-hexaene 13,13-dioxideHuman15000
EPHA2 (EphA2)EphTK8xpvAA1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman15134
EPHA2 (EphA2)EphTK8xpvAB1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman15135
EPHA3 (EphA3)EphTK2gsfA-Human2861
EPHA3 (EphA3)EphTK2qo2AA-Human2880
EPHA3 (EphA3)EphTK2qo2AB-Human2886
EPHA3 (EphA3)EphTK2qo7AAphosphoaminophosphonic acid-adenylate esterHuman2874
EPHA3 (EphA3)EphTK2qo7ABphosphoaminophosphonic acid-adenylate esterHuman2857
EPHA3 (EphA3)EphTK2qo7ACphosphoaminophosphonic acid-adenylate esterHuman2839
EPHA3 (EphA3)EphTK2qo9AAphosphoaminophosphonic acid-adenylate esterHuman2862
EPHA3 (EphA3)EphTK2qo9ABphosphoaminophosphonic acid-adenylate esterHuman2864
EPHA3 (EphA3)EphTK2qobAA-Human2889
EPHA3 (EphA3)EphTK2qobAB-Human2872
EPHA3 (EphA3)EphTK2qobAC-Human2850
EPHA3 (EphA3)EphTK2qocAAphosphoaminophosphonic acid-adenylate esterHuman2882
EPHA3 (EphA3)EphTK2qocAB-Human2856
EPHA3 (EphA3)EphTK2qocAC-Human2871
EPHA3 (EphA3)EphTK2qodAA-Human2869
EPHA3 (EphA3)EphTK2qodAB-Human2842
EPHA3 (EphA3)EphTK2qodAC-Human2866
EPHA3 (EphA3)EphTK2qofAA-Human2888
EPHA3 (EphA3)EphTK2qofAB-Human2859
EPHA3 (EphA3)EphTK2qofAC-Human2870
EPHA3 (EphA3)EphTK2qoiAA-Human2855
EPHA3 (EphA3)EphTK2qoiAB-Human2891
EPHA3 (EphA3)EphTK2qokAA-Human2873
EPHA3 (EphA3)EphTK2qokAB-Human2876
EPHA3 (EphA3)EphTK2qokAC-Human2884
EPHA3 (EphA3)EphTK2qolAA-Human2863
EPHA3 (EphA3)EphTK2qolAB-Human2836
EPHA3 (EphA3)EphTK2qolAC-Human2845
EPHA3 (EphA3)EphTK2qolAD-Human2877
EPHA3 (EphA3)EphTK2qonAA-Human2867
EPHA3 (EphA3)EphTK2qonAB-Human2853
EPHA3 (EphA3)EphTK2qooAA-Human2847
EPHA3 (EphA3)EphTK2qooAB-Human2881
EPHA3 (EphA3)EphTK2qoqAAphosphoaminophosphonic acid-adenylate esterHuman2890
EPHA3 (EphA3)EphTK2qoqABphosphoaminophosphonic acid-adenylate esterHuman2849
EPHA3 (EphA3)EphTK2qoqACphosphoaminophosphonic acid-adenylate esterHuman2879
EPHA3 (EphA3)EphTK3dzqAAn-[2-methyl-5-({[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamideHuman2852
EPHA3 (EphA3)EphTK3dzqABn-[2-methyl-5-({[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamideHuman2868
EPHA3 (EphA3)EphTK3fxxAAphosphoaminophosphonic acid-adenylate esterHuman2883
EPHA3 (EphA3)EphTK3fxxABphosphoaminophosphonic acid-adenylate esterHuman2860
EPHA3 (EphA3)EphTK3fy2AA-Human2851
EPHA3 (EphA3)EphTK3fy2AB-Human2837
EPHA3 (EphA3)EphTK4g2fAA1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-oneHuman2843
EPHA3 (EphA3)EphTK4g2fAB1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-oneHuman2838
EPHA3 (EphA3)EphTK4gk2AA7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2841
EPHA3 (EphA3)EphTK4gk2AB7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2858
EPHA3 (EphA3)EphTK4gk3AA8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2844
EPHA3 (EphA3)EphTK4gk3AB8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2885
EPHA3 (EphA3)EphTK4gk4AA8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2854
EPHA3 (EphA3)EphTK4gk4AB8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2840
EPHA3 (EphA3)EphTK4p4cA2-amino-1-(3-methoxyphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman2875
EPHA3 (EphA3)EphTK4p5qAA2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman2892
EPHA3 (EphA3)EphTK4p5qAB2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman2878
EPHA3 (EphA3)EphTK4p5zA2-amino-1-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenyl]-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman2887
EPHA3 (EphA3)EphTK4twnAA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman2846
EPHA3 (EphA3)EphTK4twnAB1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman2865
EPHA3 (EphA3)EphTK4twoAA5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acidHuman2893
EPHA3 (EphA3)EphTK4twoAB5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acidHuman2848
EPHA3 (EphA3)EphTK6in0AA1,4,7,10,13,16-hexaoxacyclooctadecaneHuman11792
EPHA3 (EphA3)EphTK6in0AB1,4,7,10,13,16-hexaoxacyclooctadecaneHuman11793
Epha4 (EphA4)EphTK2helA-Mouse5812
Epha4 (EphA4)EphTK2xyuA5-(5-fluoro-2-methylphenyl)-6,7,8,9-tetrahydro-3h-pyrazolo[3,4-c]isoquinolin-1-amineMouse5810
Epha4 (EphA4)EphTK2y6mAA-Mouse5809
Epha4 (EphA4)EphTK2y6mAB-Mouse5813
Epha4 (EphA4)EphTK2y6oAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideMouse5814
Epha4 (EphA4)EphTK2y6oABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideMouse5811
EPHA5 (EphA5)EphTK2r2pAA-Human3412
EPHA5 (EphA5)EphTK2r2pAB-Human3413
EPHA7 (EphA7)EphTK2reiAA-Human4
EPHA7 (EphA7)EphTK2reiAB-Human2
EPHA7 (EphA7)EphTK3dkoAA5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamideHuman1
EPHA7 (EphA7)EphTK3dkoAB5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamideHuman3
EPHA7 (EphA7)EphTK7eecAA-Human13792
EPHA7 (EphA7)EphTK7eecAB-Human13790
EPHA7 (EphA7)EphTK7eedA-Human13791
EPHA7 (EphA7)EphTK7eefA-Human13793
EPHA8 (EphA8)EphTK3kulAA-Human1251
EPHA8 (EphA8)EphTK3kulAB-Human1252
EPHA8 (EphA8)EphTK3kulBA-Human1249
EPHA8 (EphA8)EphTK3kulBB-Human1250
EPHB1 (EphB1)EphTK3zfxA-Human560
EPHB1 (EphB1)EphTK3zfxB-Human558
EPHB1 (EphB1)EphTK3zfxC-Human557
EPHB1 (EphB1)EphTK3zfxD-Human552
EPHB1 (EphB1)EphTK3zfxE-Human555
EPHB1 (EphB1)EphTK3zfxF-Human553
EPHB1 (EphB1)EphTK3zfxG-Human554
EPHB1 (EphB1)EphTK3zfxH-Human556
EPHB1 (EphB1)EphTK3zfxI-Human559
EPHB1 (EphB1)EphTK5mjaA2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamideHuman7582
EPHB1 (EphB1)EphTK5mjaB2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamideHuman7583
EPHB1 (EphB1)EphTK5mjbA2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamideHuman7584
EPHB1 (EphB1)EphTK5mjbB2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamideHuman7585
EPHB1 (EphB1)EphTK6umwAA-Human12924
EPHB1 (EphB1)EphTK6umwAB-Human12923
EPHB1 (EphB1)EphTK7kplAA-Human13384
EPHB1 (EphB1)EphTK7kplAB-Human13383
EPHB1 (EphB1)EphTK7kpmAAadenosine-5'-diphosphateHuman13385
EPHB1 (EphB1)EphTK7kpmABadenosine-5'-diphosphateHuman13382
Ephb2 (EphB2)EphTK1jpaAphosphoaminophosphonic acid-adenylate esterMouse5806
Ephb2 (EphB2)EphTK1jpaBphosphoaminophosphonic acid-adenylate esterMouse5805
Ephb2 (EphB2)EphTK2henAadenosine-5'-diphosphateMouse5807
Ephb2 (EphB2)EphTK2henBadenosine-5'-diphosphateMouse5804
Ephb2 (EphB2)EphTK2henCadenosine-5'-diphosphateMouse5808
Ephb2 (EphB2)EphTK2henDadenosine-5'-diphosphateMouse5803
EPHB2 (EphB2)EphTK3zfmA-Human2731
EPHB3 (EphB3)EphTK3zfyAA-Human537
EPHB3 (EphB3)EphTK3zfyAB-Human538
EPHB3 (EphB3)EphTK3zfyBA-Human539
EPHB3 (EphB3)EphTK3zfyBB-Human536
EPHB3 (EphB3)EphTK5l6oA1-(4-phenylazanylquinazolin-7-yl)ethanoneHuman6938
EPHB3 (EphB3)EphTK5l6pA~{n}-(4-phenylazanylquinazolin-7-yl)ethanamideHuman6937
EPHB4 (EphB4)EphTK2vwuAn-(5-chloro-1,3-benzodioxol-4-yl)-6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin-4-amineHuman370
EPHB4 (EphB4)EphTK2vwvAAn'-(3-chloro-4-methoxy-phenyl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazine-2,4-diamineHuman365
EPHB4 (EphB4)EphTK2vwvABn'-(3-chloro-4-methoxy-phenyl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazine-2,4-diamineHuman369
EPHB4 (EphB4)EphTK2vwwAAn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3,4,5- trimethoxyphenyl)pyrimidine-2,4-diamineHuman356
EPHB4 (EphB4)EphTK2vwwABn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3,4,5- trimethoxyphenyl)pyrimidine-2,4-diamineHuman358
EPHB4 (EphB4)EphTK2vwxAA3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamideHuman361
EPHB4 (EphB4)EphTK2vwxAB3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamideHuman350
EPHB4 (EphB4)EphTK2vwyAAn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-methylsulfonylphenyl)pyrimidine-2,4-diamineHuman353
EPHB4 (EphB4)EphTK2vwyABn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-methylsulfonylphenyl)pyrimidine-2,4-diamineHuman355
EPHB4 (EphB4)EphTK2vwzAAn-[3-[[4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl]amino]phenyl]methanesulfonamideHuman360
EPHB4 (EphB4)EphTK2vwzABn-[3-[[4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl]amino]phenyl]methanesulfonamideHuman362
EPHB4 (EphB4)EphTK2vx0AAn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-morpholin-4-ylphenyl)pyrimidine-2,4-diamineHuman375
EPHB4 (EphB4)EphTK2vx0ABn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-morpholin-4-ylphenyl)pyrimidine-2,4-diamineHuman368
EPHB4 (EphB4)EphTK2vx1AA3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzamideHuman371
EPHB4 (EphB4)EphTK2vx1AB3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzamideHuman374
EPHB4 (EphB4)EphTK2x9fAAn^4^-1h-indazol-4-yl-n^2^-[3-(methylsulfonyl)phenyl]pyrimidine-2,4-diamineHuman354
EPHB4 (EphB4)EphTK2x9fABn^4^-1h-indazol-4-yl-n^2^-[3-(methylsulfonyl)phenyl]pyrimidine-2,4-diamineHuman359
EPHB4 (EphB4)EphTK2xvdAA{4-methyl-3-[(1-methylethyl)(2-{[3-(methylsulfonyl)-5-morpholin-4-ylphenyl]amino}pyrimidin-4-yl)amino]phenyl}methanolHuman363
EPHB4 (EphB4)EphTK2xvdAB{4-methyl-3-[(1-methylethyl)(2-{[3-(methylsulfonyl)-5-morpholin-4-ylphenyl]amino}pyrimidin-4-yl)amino]phenyl}methanolHuman372
EPHB4 (EphB4)EphTK2yn8AstaurosporineHuman352
EPHB4 (EphB4)EphTK2yn8BstaurosporineHuman349
EPHB4 (EphB4)EphTK3zewAAstaurosporineHuman373
EPHB4 (EphB4)EphTK3zewABstaurosporineHuman377
EPHB4 (EphB4)EphTK3zewBAstaurosporineHuman351
EPHB4 (EphB4)EphTK3zewBBstaurosporineHuman357
EPHB4 (EphB4)EphTK4aw5AA(3z)-5-[(1-ethylpiperidin-4-yl)amino]-3-[(5-methoxy-1h-benzimidazol-2-yl)(phenyl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman367
EPHB4 (EphB4)EphTK4aw5AB(3z)-5-[(1-ethylpiperidin-4-yl)amino]-3-[(5-methoxy-1h-benzimidazol-2-yl)(phenyl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman376
EPHB4 (EphB4)EphTK4bb4AAn-(2-methoxyethyl)-4-[(6-pyridin-4-ylquinazolin-2-yl)amino]benzamideHuman364
EPHB4 (EphB4)EphTK4bb4ABn-(2-methoxyethyl)-4-[(6-pyridin-4-ylquinazolin-2-yl)amino]benzamideHuman366
EPHB4 (EphB4)EphTK6fniAA4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10338
EPHB4 (EphB4)EphTK6fniAB4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10333
EPHB4 (EphB4)EphTK6fnjAA4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10336
EPHB4 (EphB4)EphTK6fnjAB4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10334
EPHB4 (EphB4)EphTK6fnjBA4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10340
EPHB4 (EphB4)EphTK6fnjBB4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10341
EPHB4 (EphB4)EphTK6fnkAA1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10344
EPHB4 (EphB4)EphTK6fnkAB1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10337
EPHB4 (EphB4)EphTK6fnlAA-Human10343
EPHB4 (EphB4)EphTK6fnlAB-Human10335
EPHB4 (EphB4)EphTK6fnmAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman10342
EPHB4 (EphB4)EphTK6fnmABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman10339
ERBB2 (ErbB2)EGFRTK3pp0AA2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanolHuman4815
ERBB2 (ErbB2)EGFRTK3pp0AB2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanolHuman4820
ERBB2 (ErbB2)EGFRTK3pp0BA2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanolHuman4816
ERBB2 (ErbB2)EGFRTK3pp0BB2-{2-[4-({5-chloro-6-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethoxy}ethanolHuman4819
ERBB2 (ErbB2)EGFRTK3rcdAn-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamideHuman9325
ERBB2 (ErbB2)EGFRTK3rcdB-Human9322
ERBB2 (ErbB2)EGFRTK3rcdCn-{2-[4-({3-chloro-4-[3-(trifluoromethyl)phenoxy]phenyl}amino)-5h-pyrrolo[3,2-d]pyrimidin-5-yl]ethyl}-3-hydroxy-3-methylbutanamideHuman9323
ERBB2 (ErbB2)EGFRTK3rcdD-Human9324
ERBB2 (ErbB2)EGFRTK7jxhAA(2e)-n-[3-cyano-7-ethoxy-4-({3-methyl-4-[([1,2,4]triazolo[1,5-a]pyridin-7-yl)oxy]phenyl}amino)quinolin-6-yl]-4-(dimethylamino)but-2-enamideHuman13888
ERBB2 (ErbB2)EGFRTK7jxhAB(2e)-n-[3-cyano-7-ethoxy-4-({3-methyl-4-[([1,2,4]triazolo[1,5-a]pyridin-7-yl)oxy]phenyl}amino)quinolin-6-yl]-4-(dimethylamino)but-2-enamideHuman13887
ERBB2 (ErbB2)EGFRTK7pcdAA1-[4-[4-[[3,5-bis(chloranyl)-4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)phenyl]amino]pyrimido[5,4-d]pyrimidin-6-yl]piperazin-1-yl]-4-(3-fluoranylazetidin-1-yl)butan-1-oneHuman14320
ERBB2 (ErbB2)EGFRTK7pcdAB1-[4-[4-[[3,5-bis(chloranyl)-4-([1,2,4]triazolo[1,5-a]pyridin-7-yloxy)phenyl]amino]pyrimido[5,4-d]pyrimidin-6-yl]piperazin-1-yl]-4-(3-fluoranylazetidin-1-yl)butan-1-oneHuman14319
ERBB3 (ErbB3)EGFRTK3kexAphosphoaminophosphonic acid-adenylate esterHuman1939
ERBB3 (ErbB3)EGFRTK3kexBphosphoaminophosphonic acid-adenylate esterHuman1933
ERBB3 (ErbB3)EGFRTK3lmgAphosphoaminophosphonic acid-adenylate esterHuman1935
ERBB3 (ErbB3)EGFRTK3lmgBphosphoaminophosphonic acid-adenylate esterHuman1936
ERBB3 (ErbB3)EGFRTK4riwAphosphoaminophosphonic acid-adenylate esterHuman1930
ERBB3 (ErbB3)EGFRTK4riwCphosphoaminophosphonic acid-adenylate esterHuman1932
ERBB3 (ErbB3)EGFRTK4rixAphosphoaminophosphonic acid-adenylate esterHuman1931
ERBB3 (ErbB3)EGFRTK4rixCphosphoaminophosphonic acid-adenylate esterHuman1934
ERBB3 (ErbB3)EGFRTK4riyAphosphoaminophosphonic acid-adenylate esterHuman1937
ERBB3 (ErbB3)EGFRTK4riyCphosphoaminophosphonic acid-adenylate esterHuman1938
ERBB3 (ErbB3)EGFRTK6op9AA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman11545
ERBB3 (ErbB3)EGFRTK6op9AB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman11544
ERBB3 (ErbB3)EGFRTK7mn5A-Human13953
ERBB3 (ErbB3)EGFRTK7mn6A-Human13952
ERBB3 (ErbB3)EGFRTK7mn8A-Human13966
ERBB4 (ErbB4)EGFRTK2r4bAAn-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amineHuman2822
ERBB4 (ErbB4)EGFRTK2r4bABn-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amineHuman2827
ERBB4 (ErbB4)EGFRTK2r4bBAn-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amineHuman2818
ERBB4 (ErbB4)EGFRTK2r4bBBn-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amineHuman2823
ERBB4 (ErbB4)EGFRTK3bbtBn-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamineHuman2825
ERBB4 (ErbB4)EGFRTK3bbtDn-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamineHuman2819
ERBB4 (ErbB4)EGFRTK3bbwA-Human2820
ERBB4 (ErbB4)EGFRTK3bbwB-Human2817
ERBB4 (ErbB4)EGFRTK3bceA-Human2821
ERBB4 (ErbB4)EGFRTK3bceB-Human2826
ERBB4 (ErbB4)EGFRTK3bceC-Human2824
Ern1 (IRE1)IREOther4pl3Aadenosine-5'-diphosphateMouse5769
Ern1 (IRE1)IREOther4pl3Badenosine-5'-diphosphateMouse5768
Ern1 (IRE1)IREOther4pl4Aadenosine-5'-diphosphateMouse5770
Ern1 (IRE1)IREOther4pl4Badenosine-5'-diphosphateMouse5767
Ern1 (IRE1)IREOther4pl4Cadenosine-5'-diphosphateMouse5761
Ern1 (IRE1)IREOther4pl4Dadenosine-5'-diphosphateMouse5765
Ern1 (IRE1)IREOther4pl5Aadenosine-5'-diphosphateMouse5762
Ern1 (IRE1)IREOther4pl5Badenosine-5'-diphosphateMouse5764
Ern1 (IRE1)IREOther4pl5Cadenosine-5'-diphosphateMouse5766
Ern1 (IRE1)IREOther4pl5Dadenosine-5'-diphosphateMouse5763
ERN1 (IRE1)IREOther3p23Aadenosine-5'-diphosphateHuman1795
ERN1 (IRE1)IREOther3p23Badenosine-5'-diphosphateHuman1797
ERN1 (IRE1)IREOther3p23Cadenosine-5'-diphosphateHuman1798
ERN1 (IRE1)IREOther3p23Dadenosine-5'-diphosphateHuman1800
ERN1 (IRE1)IREOther4u6rAn-{4-[(3-{2-[(trans-4-aminocyclohexyl)amino]pyrimidin-4-yl}pyridin-2-yl)oxy]-3-methylnaphthalen-1-yl}-2-chlorobenzenesulfonamideHuman1802
ERN1 (IRE1)IREOther4yz9AA(5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamideHuman6233
ERN1 (IRE1)IREOther4yz9AB(5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamideHuman6224
ERN1 (IRE1)IREOther4yz9BA(5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamideHuman6225
ERN1 (IRE1)IREOther4yz9BB(5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamideHuman6229
ERN1 (IRE1)IREOther4yz9CA(5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamideHuman6223
ERN1 (IRE1)IREOther4yz9CB(5r)-2-(3,4-dichlorobenzyl)-n-(4-methylbenzyl)-2,7-diazaspiro[4.5]decane-7-carboxamideHuman6222
ERN1 (IRE1)IREOther4yzcAAstaurosporineHuman6235
ERN1 (IRE1)IREOther4yzcABstaurosporineHuman6232
ERN1 (IRE1)IREOther4yzcBAstaurosporineHuman6227
ERN1 (IRE1)IREOther4yzcBBstaurosporineHuman6231
ERN1 (IRE1)IREOther4yzdAAadenosine-5'-diphosphateHuman6234
ERN1 (IRE1)IREOther4yzdABadenosine-5'-diphosphateHuman6228
ERN1 (IRE1)IREOther4yzdBAadenosine-5'-diphosphateHuman6236
ERN1 (IRE1)IREOther4yzdBBadenosine-5'-diphosphateHuman6230
ERN1 (IRE1)IREOther4yzdCAadenosine-5'-diphosphateHuman6237
ERN1 (IRE1)IREOther4yzdCBadenosine-5'-diphosphateHuman6226
ERN1 (IRE1)IREOther4z7gA-Human1799
ERN1 (IRE1)IREOther4z7gB-Human1796
ERN1 (IRE1)IREOther4z7hA2-methoxy-4-[6-(propan-2-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman1794
ERN1 (IRE1)IREOther4z7hB2-methoxy-4-[6-(propan-2-ylamino)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman1801
ERN1 (IRE1)IREOther5hgiA-Human6669
ERN1 (IRE1)IREOther6hv0A6-chloranyl-3-(2~{h}-indazol-5-yl)-~{n}-propan-2-yl-imidazo[1,2-b]pyridazin-8-amineHuman10928
ERN1 (IRE1)IREOther6hx1AA6-chloranyl-~{n}-(cyclopropylmethyl)-3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-8-amineHuman10927
ERN1 (IRE1)IREOther6hx1AB6-chloranyl-~{n}-(cyclopropylmethyl)-3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-8-amineHuman10929
ERN1 (IRE1)IREOther6urcA2-chloro-n-(6-methyl-5-{[3-(2-{[(3s)-piperidin-3-yl]amino}pyrimidin-4-yl)pyridin-2-yl]oxy}naphthalen-1-yl)benzene-1-sulfonamideHuman11799
ERN1 (IRE1)IREOther6urcB2-chloro-n-(6-methyl-5-{[3-(2-{[(3s)-piperidin-3-yl]amino}pyrimidin-4-yl)pyridin-2-yl]oxy}naphthalen-1-yl)benzene-1-sulfonamideHuman11798
ERN1 (IRE1)IREOther6w39AAethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamateHuman13120
ERN1 (IRE1)IREOther6w39ABethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamateHuman13122
ERN1 (IRE1)IREOther6w39BAethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamateHuman13117
ERN1 (IRE1)IREOther6w39BBethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamateHuman13124
ERN1 (IRE1)IREOther6w3aAA~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]but-2-ynamideHuman13125
ERN1 (IRE1)IREOther6w3aAB~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]but-2-ynamideHuman13116
ERN1 (IRE1)IREOther6w3aBA~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]but-2-ynamideHuman13118
ERN1 (IRE1)IREOther6w3aBB~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]but-2-ynamideHuman13119
ERN1 (IRE1)IREOther6w3bA-Human13039
ERN1 (IRE1)IREOther6w3cA-Human13040
ERN1 (IRE1)IREOther6w3cB-Human13038
ERN1 (IRE1)IREOther6w3cC-Human13036
ERN1 (IRE1)IREOther6w3cD-Human13037
ERN1 (IRE1)IREOther6w3eAmethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamateHuman13121
ERN1 (IRE1)IREOther6w3eBmethyl ~{n}-[6-methyl-5-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxy-naphthalen-1-yl]carbamateHuman13126
ERN1 (IRE1)IREOther6w3kA4-[5-[2,6-bis(fluoranyl)phenyl]-2~{h}-pyrazolo[3,4-b]pyridin-3-yl]-2-(4-oxidanylpiperidin-1-yl)-1~{h}-pyrimidin-6-oneHuman13123
ERN1 (IRE1)IREOther6xdbA4-amino-n-(6-chloro-2-fluoro-3-{[(2-fluorophenyl)sulfonyl]amino}phenyl)-6-(1,3-dimethyl-1h-pyrazol-4-yl)quinazoline-8-carboxamideHuman13531
ERN1 (IRE1)IREOther6xddA4-[(trans-4-aminocyclohexyl)amino]-n-(6-chloro-3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)thieno[3,2-d]pyrimidine-7-carboxamideHuman13529
ERN1 (IRE1)IREOther6xddB4-[(trans-4-aminocyclohexyl)amino]-n-(6-chloro-3-{[(2,5-difluorophenyl)sulfonyl]amino}-2-fluorophenyl)thieno[3,2-d]pyrimidine-7-carboxamideHuman13530
ERN1 (IRE1)IREOther6xdfBA-Human13508
ERN1 (IRE1)IREOther6xdfBB-Human13507
ERN1 (IRE1)IREOther7bmkAA2,2,2-tris(fluoranyl)-~{n}-[4-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxynaphthalen-1-yl]ethanesulfonamideHuman13911
ERN1 (IRE1)IREOther7bmkAB2,2,2-tris(fluoranyl)-~{n}-[4-[3-[2-[[(3~{s})-piperidin-3-yl]amino]pyrimidin-4-yl]pyridin-2-yl]oxynaphthalen-1-yl]ethanesulfonamideHuman13912
FESFerTK3bkbAAstaurosporineHuman2810
FESFerTK3bkbABstaurosporineHuman2813
FESFerTK3bkbACstaurosporineHuman2812
FESFerTK3cblAAstaurosporineHuman2808
FESFerTK3cblABstaurosporineHuman2811
FESFerTK3cd3AAstaurosporineHuman2814
FESFerTK3cd3ABstaurosporineHuman2815
FESFerTK4e93AA5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHuman2816
FESFerTK4e93AB5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHuman2809
FESFerTK6jmfA6-{[(1r,2s)-2-aminocyclohexyl]amino}-5-cyano-2-[(3-methylphenyl)amino]pyridine-3-carboxamideHuman11140
FGFR1FGFRTK1agwAA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3520
FGFR1FGFRTK1agwAB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3528
FGFR1FGFRTK1agwBA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3568
FGFR1FGFRTK1agwBB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3510
FGFR1FGFRTK1fgiAA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3555
FGFR1FGFRTK1fgiAB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3552
FGFR1FGFRTK1fgiBA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3586
FGFR1FGFRTK1fgiBB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3580
FGFR1FGFRTK1fgkAA-Human3592
FGFR1FGFRTK1fgkAB-Human3546
FGFR1FGFRTK1fgkBA-Human3513
FGFR1FGFRTK1fgkBB-Human3557
FGFR1FGFRTK2fgiA1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHuman3490
FGFR1FGFRTK2fgiB1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHuman3541
FGFR1FGFRTK3c4fAA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3515
FGFR1FGFRTK3c4fAB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3564
FGFR1FGFRTK3c4fBA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3573
FGFR1FGFRTK3c4fBB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3562
FGFR1FGFRTK3gqiAphosphomethylphosphonic acid adenylate esterHuman3566
FGFR1FGFRTK3gqlA(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHuman3509
FGFR1FGFRTK3gqlB(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHuman3506
FGFR1FGFRTK3gqlC(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHuman3536
FGFR1FGFRTK3js2A5-(2-thienyl)nicotinic acidHuman3523
FGFR1FGFRTK3js2B5-(2-thienyl)nicotinic acidHuman3504
FGFR1FGFRTK3kxxA-Human3495
FGFR1FGFRTK3kxxB-Human3575
FGFR1FGFRTK3kxxC-Human3549
FGFR1FGFRTK3kxxD-Human3503
FGFR1FGFRTK3ky2A-Human3534
FGFR1FGFRTK3ky2B-Human3525
FGFR1FGFRTK3rhxA(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman3554
FGFR1FGFRTK3rhxB(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman3522
FGFR1FGFRTK3tt0AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3567
FGFR1FGFRTK3tt0AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3538
FGFR1FGFRTK3tt0BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3547
FGFR1FGFRTK3tt0BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3581
FGFR1FGFRTK4f63A5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHuman3563
FGFR1FGFRTK4f63B5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHuman3574
FGFR1FGFRTK4f64AA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3548
FGFR1FGFRTK4f64AB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3589
FGFR1FGFRTK4f64BA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3576
FGFR1FGFRTK4f64BB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3553
FGFR1FGFRTK4f65AA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3558
FGFR1FGFRTK4f65AB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3508
FGFR1FGFRTK4f65BA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3545
FGFR1FGFRTK4f65BB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3502
FGFR1FGFRTK4nk9An~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3550
FGFR1FGFRTK4nk9Bn~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3535
FGFR1FGFRTK4nkaAn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3501
FGFR1FGFRTK4nkaBn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3539
FGFR1FGFRTK4nksAAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3570
FGFR1FGFRTK4nksABn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3561
FGFR1FGFRTK4nksBAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3492
FGFR1FGFRTK4nksBBn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3577
FGFR1FGFRTK4rwiAA-Human3499
FGFR1FGFRTK4rwiAB-Human3551
FGFR1FGFRTK4rwiBA-Human3569
FGFR1FGFRTK4rwiBB-Human3527
FGFR1FGFRTK4rwjAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3584
FGFR1FGFRTK4rwjABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3519
FGFR1FGFRTK4rwjBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3579
FGFR1FGFRTK4rwjBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3559
FGFR1FGFRTK4rwkAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3500
FGFR1FGFRTK4rwkABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3517
FGFR1FGFRTK4rwkBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3591
FGFR1FGFRTK4rwkBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3530
FGFR1FGFRTK4rwlA-Human3516
FGFR1FGFRTK4rwlB6-({7-[(1-aminocyclopropyl)methoxy]-6-methoxyquinolin-4-yl}oxy)-n-methylnaphthalene-1-carboxamideHuman3596
FGFR1FGFRTK4uwbAAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6020
FGFR1FGFRTK4uwbABn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6023
FGFR1FGFRTK4uwbBAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6018
FGFR1FGFRTK4uwbBBn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6022
FGFR1FGFRTK4uwcAA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6019
FGFR1FGFRTK4uwcAB3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6017
FGFR1FGFRTK4uwcBA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6021
FGFR1FGFRTK4uwcBB3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6016
FGFR1FGFRTK4uwyAA-Human3489
FGFR1FGFRTK4uwyAB-Human3582
FGFR1FGFRTK4uwyBA-Human3537
FGFR1FGFRTK4uwyBB-Human3583
FGFR1FGFRTK4v01AA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3556
FGFR1FGFRTK4v01AB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3590
FGFR1FGFRTK4v01BA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3497
FGFR1FGFRTK4v01BB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3594
FGFR1FGFRTK4v04AA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3542
FGFR1FGFRTK4v04AB-Human3571
FGFR1FGFRTK4v04BA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3524
FGFR1FGFRTK4v04BB-Human3496
FGFR1FGFRTK4v05AAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3560
FGFR1FGFRTK4v05ABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3593
FGFR1FGFRTK4v05BAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3518
FGFR1FGFRTK4v05BBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3493
FGFR1FGFRTK4wunAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3511
FGFR1FGFRTK4wunABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3595
FGFR1FGFRTK4wunBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3529
FGFR1FGFRTK4wunBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3565
FGFR1FGFRTK4zsaAA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3491
FGFR1FGFRTK4zsaAB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3487
FGFR1FGFRTK4zsaBA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3572
FGFR1FGFRTK4zsaBB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3512
FGFR1FGFRTK5a46AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3532
FGFR1FGFRTK5a46AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3505
FGFR1FGFRTK5a46BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3526
FGFR1FGFRTK5a46BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3578
FGFR1FGFRTK5a4cAA1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3543
FGFR1FGFRTK5a4cAB1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3498
FGFR1FGFRTK5a4cBA1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3585
FGFR1FGFRTK5a4cBB1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3540
FGFR1FGFRTK5am6AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3494
FGFR1FGFRTK5am6AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3514
FGFR1FGFRTK5am6BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3587
FGFR1FGFRTK5am6BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3521
FGFR1FGFRTK5am7AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3533
FGFR1FGFRTK5am7AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3488
FGFR1FGFRTK5am7BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3588
FGFR1FGFRTK5am7BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3531
FGFR1FGFRTK5b7vA[5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanoneHuman6705
FGFR1FGFRTK5b7vB[5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanoneHuman6704
FGFR1FGFRTK5ew8AA~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6470
FGFR1FGFRTK5ew8AB~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6461
FGFR1FGFRTK5ew8BA~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6474
FGFR1FGFRTK5ew8BB~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6471
FGFR1FGFRTK5flfAA-Human6462
FGFR1FGFRTK5flfAB-Human6464
FGFR1FGFRTK5flfBA-Human6465
FGFR1FGFRTK5flfBB-Human6467
FGFR1FGFRTK5flfCA-Human6469
FGFR1FGFRTK5flfCB-Human6466
FGFR1FGFRTK5flfDA-Human6468
FGFR1FGFRTK5flfDB-Human6463
FGFR1FGFRTK5flfEA-Human6473
FGFR1FGFRTK5flfEB-Human6472
FGFR1FGFRTK5o49AA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9560
FGFR1FGFRTK5o49AB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9556
FGFR1FGFRTK5o49BA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9561
FGFR1FGFRTK5o49BB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9557
FGFR1FGFRTK5o4aAA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9554
FGFR1FGFRTK5o4aAB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9558
FGFR1FGFRTK5o4aBA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9559
FGFR1FGFRTK5o4aBB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9555
FGFR1FGFRTK5uq0AA2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7456
FGFR1FGFRTK5uq0AB2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7458
FGFR1FGFRTK5uq0BA2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7459
FGFR1FGFRTK5uq0BB2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7457
FGFR1FGFRTK5ur1AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7970
FGFR1FGFRTK5ur1AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7972
FGFR1FGFRTK5ur1BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7969
FGFR1FGFRTK5ur1BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7971
FGFR1FGFRTK5vndAAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7646
FGFR1FGFRTK5vndABn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7648
FGFR1FGFRTK5vndBAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7647
FGFR1FGFRTK5vndBBn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7645
FGFR1FGFRTK5z0sAA1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10813
FGFR1FGFRTK5z0sAB1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10815
FGFR1FGFRTK5z0sBA1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10812
FGFR1FGFRTK5z0sBB1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10814
FGFR1FGFRTK5zv2A4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHuman10055
FGFR1FGFRTK5zv2B4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHuman10054
FGFR1FGFRTK6c18AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11155
FGFR1FGFRTK6c18AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11168
FGFR1FGFRTK6c18BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10854
FGFR1FGFRTK6c18BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11170
FGFR1FGFRTK6c19AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11163
FGFR1FGFRTK6c19AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10859
FGFR1FGFRTK6c19BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10855
FGFR1FGFRTK6c19BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10862
FGFR1FGFRTK6c1bAA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11169
FGFR1FGFRTK6c1bAB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10861
FGFR1FGFRTK6c1bBA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10856
FGFR1FGFRTK6c1bBB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11167
FGFR1FGFRTK6c1cAA7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11164
FGFR1FGFRTK6c1cAB7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10853
FGFR1FGFRTK6c1cBA7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10858
FGFR1FGFRTK6c1cBB7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11158
FGFR1FGFRTK6c1oAAn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11159
FGFR1FGFRTK6c1oABn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11166
FGFR1FGFRTK6c1oBAn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11160
FGFR1FGFRTK6c1oBBn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11154
FGFR1FGFRTK6itjAA4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11773
FGFR1FGFRTK6itjAB4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11774
FGFR1FGFRTK6itjBA4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11775
FGFR1FGFRTK6itjBB4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11772
FGFR1FGFRTK6mzqAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman10860
FGFR1FGFRTK6mzqAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11156
FGFR1FGFRTK6mzqBA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11161
FGFR1FGFRTK6mzqBB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11171
FGFR1FGFRTK6mzwAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11162
FGFR1FGFRTK6mzwAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11157
FGFR1FGFRTK6mzwBA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11165
FGFR1FGFRTK6mzwBB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman10857
FGFR1FGFRTK6nvlAAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11400
FGFR1FGFRTK6nvlABn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11401
FGFR1FGFRTK6nvlBAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11403
FGFR1FGFRTK6nvlBBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11399
FGFR1FGFRTK6nvlCAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11404
FGFR1FGFRTK6nvlCBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11405
FGFR1FGFRTK6nvlDAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11402
FGFR1FGFRTK6nvlDBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11398
FGFR1FGFRTK6p68An-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHuman11336
FGFR1FGFRTK6p68Bn-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHuman11334
FGFR1FGFRTK6p68Cn-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHuman11332
FGFR1FGFRTK6p69AAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11333
FGFR1FGFRTK6p69ABn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11330
FGFR1FGFRTK6p69BAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11331
FGFR1FGFRTK6p69BBn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11335
FGFR1FGFRTK7ozbAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman14010
FGFR1FGFRTK7ozbAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman14008
FGFR1FGFRTK7ozdAAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHuman14007
FGFR1FGFRTK7ozdABn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHuman14009
FGFR1FGFRTK7ozfAAn-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamideHuman14011
FGFR1FGFRTK7ozfABn-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamideHuman14006
FGFR1FGFRTK7wclAA11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-oneHuman14364
FGFR1FGFRTK7wclAB11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-oneHuman14363
FGFR2FGFRTK1gjoA-Human478
FGFR2FGFRTK1oecA4-aryl-2-phenylamino pyrimidineHuman479
FGFR2FGFRTK2psqA-Human515
FGFR2FGFRTK2psqB-Human530
FGFR2FGFRTK2pvfAphosphomethylphosphonic acid adenylate esterHuman525
FGFR2FGFRTK2pvyAphosphomethylphosphonic acid adenylate esterHuman489
FGFR2FGFRTK2pvyBphosphomethylphosphonic acid adenylate esterHuman504
FGFR2FGFRTK2pvyCphosphomethylphosphonic acid adenylate esterHuman501
FGFR2FGFRTK2pvyDphosphomethylphosphonic acid adenylate esterHuman482
FGFR2FGFRTK2pwlAphosphomethylphosphonic acid adenylate esterHuman523
FGFR2FGFRTK2pwlBphosphomethylphosphonic acid adenylate esterHuman534
FGFR2FGFRTK2py3Aphosphomethylphosphonic acid adenylate esterHuman509
FGFR2FGFRTK2py3Bphosphomethylphosphonic acid adenylate esterHuman484
FGFR2FGFRTK2pz5Aphosphomethylphosphonic acid adenylate esterHuman511
FGFR2FGFRTK2pz5Bphosphomethylphosphonic acid adenylate esterHuman513
FGFR2FGFRTK2pzpAphosphomethylphosphonic acid adenylate esterHuman497
FGFR2FGFRTK2pzpBphosphomethylphosphonic acid adenylate esterHuman524
FGFR2FGFRTK2pzrAphosphomethylphosphonic acid adenylate esterHuman526
FGFR2FGFRTK2pzrBphosphomethylphosphonic acid adenylate esterHuman508
FGFR2FGFRTK2q0bAphosphomethylphosphonic acid adenylate esterHuman512
FGFR2FGFRTK2q0bBphosphomethylphosphonic acid adenylate esterHuman499
FGFR2FGFRTK3b2tA5'-o-[(s)-hydroxy{[(s)-hydroxy(methyl)phosphoryl]oxy}phosphoryl]adenosineHuman520
FGFR2FGFRTK3b2tB5'-o-[(s)-hydroxy{[(s)-hydroxy(methyl)phosphoryl]oxy}phosphoryl]adenosineHuman517
FGFR2FGFRTK3clyAphosphomethylphosphonic acid adenylate esterHuman522
FGFR2FGFRTK3ri1A(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman503
FGFR2FGFRTK3ri1B(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman528
FGFR2FGFRTK4j95AAphosphomethylphosphonic acid adenylate esterHuman529
FGFR2FGFRTK4j95ABphosphomethylphosphonic acid adenylate esterHuman477
FGFR2FGFRTK4j95BAphosphomethylphosphonic acid adenylate esterHuman498
FGFR2FGFRTK4j95BBphosphomethylphosphonic acid adenylate esterHuman519
FGFR2FGFRTK4j95CAphosphomethylphosphonic acid adenylate esterHuman531
FGFR2FGFRTK4j95CBphosphomethylphosphonic acid adenylate esterHuman502
FGFR2FGFRTK4j95DAphosphomethylphosphonic acid adenylate esterHuman490
FGFR2FGFRTK4j95DBphosphomethylphosphonic acid adenylate esterHuman492
FGFR2FGFRTK4j96AA-Human473
FGFR2FGFRTK4j96AB-Human470
FGFR2FGFRTK4j96BAphosphomethylphosphonic acid adenylate esterHuman485
FGFR2FGFRTK4j96BBphosphomethylphosphonic acid adenylate esterHuman486
FGFR2FGFRTK4j97AAphosphomethylphosphonic acid adenylate esterHuman496
FGFR2FGFRTK4j97ABphosphomethylphosphonic acid adenylate esterHuman527
FGFR2FGFRTK4j97ACphosphomethylphosphonic acid adenylate esterHuman521
FGFR2FGFRTK4j97BAphosphomethylphosphonic acid adenylate esterHuman476
FGFR2FGFRTK4j97BBphosphomethylphosphonic acid adenylate esterHuman493
FGFR2FGFRTK4j97BCphosphomethylphosphonic acid adenylate esterHuman510
FGFR2FGFRTK4j97CAphosphomethylphosphonic acid adenylate esterHuman488
FGFR2FGFRTK4j97CBphosphomethylphosphonic acid adenylate esterHuman487
FGFR2FGFRTK4j97CCphosphomethylphosphonic acid adenylate esterHuman483
FGFR2FGFRTK4j97DAphosphomethylphosphonic acid adenylate esterHuman507
FGFR2FGFRTK4j97DBphosphomethylphosphonic acid adenylate esterHuman532
FGFR2FGFRTK4j97DCphosphomethylphosphonic acid adenylate esterHuman514
FGFR2FGFRTK4j98AA-Human500
FGFR2FGFRTK4j98AB-Human475
FGFR2FGFRTK4j98BAphosphomethylphosphonic acid adenylate esterHuman516
FGFR2FGFRTK4j98BBphosphomethylphosphonic acid adenylate esterHuman472
FGFR2FGFRTK4j99AAphosphomethylphosphonic acid adenylate esterHuman474
FGFR2FGFRTK4j99ABphosphomethylphosphonic acid adenylate esterHuman494
FGFR2FGFRTK4j99ACphosphomethylphosphonic acid adenylate esterHuman469
FGFR2FGFRTK4j99BAphosphomethylphosphonic acid adenylate esterHuman518
FGFR2FGFRTK4j99BBphosphomethylphosphonic acid adenylate esterHuman495
FGFR2FGFRTK4j99BCphosphomethylphosphonic acid adenylate esterHuman491
FGFR2FGFRTK4j99CAphosphomethylphosphonic acid adenylate esterHuman505
FGFR2FGFRTK4j99CBphosphomethylphosphonic acid adenylate esterHuman506
FGFR2FGFRTK4j99CCphosphomethylphosphonic acid adenylate esterHuman471
FGFR2FGFRTK4j99DAphosphomethylphosphonic acid adenylate esterHuman533
FGFR2FGFRTK4j99DBphosphomethylphosphonic acid adenylate esterHuman481
FGFR2FGFRTK4j99DCphosphomethylphosphonic acid adenylate esterHuman480
FGFR2FGFRTK5eg3Aphosphomethylphosphonic acid adenylate esterHuman6368
FGFR2FGFRTK5uglAAphosphoaminophosphonic acid-adenylate esterHuman7442
FGFR2FGFRTK5uglABphosphoaminophosphonic acid-adenylate esterHuman7452
FGFR2FGFRTK5uglBAphosphoaminophosphonic acid-adenylate esterHuman7450
FGFR2FGFRTK5uglBBphosphoaminophosphonic acid-adenylate esterHuman7449
FGFR2FGFRTK5ugxAAphosphomethylphosphonic acid adenylate esterHuman7443
FGFR2FGFRTK5ugxABphosphomethylphosphonic acid adenylate esterHuman7448
FGFR2FGFRTK5ugxBAphosphomethylphosphonic acid adenylate esterHuman7454
FGFR2FGFRTK5ugxBBphosphomethylphosphonic acid adenylate esterHuman7445
FGFR2FGFRTK5uhnAAphosphomethylphosphonic acid adenylate esterHuman7455
FGFR2FGFRTK5uhnABphosphomethylphosphonic acid adenylate esterHuman7441
FGFR2FGFRTK5uhnBAphosphomethylphosphonic acid adenylate esterHuman7451
FGFR2FGFRTK5uhnBBphosphomethylphosphonic acid adenylate esterHuman7444
FGFR2FGFRTK5ui0AA-Human7446
FGFR2FGFRTK5ui0AB-Human7447
FGFR2FGFRTK5ui0BAphosphomethylphosphonic acid adenylate esterHuman7453
FGFR2FGFRTK5ui0BBphosphomethylphosphonic acid adenylate esterHuman7440
FGFR2FGFRTK6agxAAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11541
FGFR2FGFRTK6agxABethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11542
FGFR2FGFRTK6agxBAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11540
FGFR2FGFRTK6agxBBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11536
FGFR2FGFRTK6agxCAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11538
FGFR2FGFRTK6agxCBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11537
FGFR2FGFRTK6agxDAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11543
FGFR2FGFRTK6agxDBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11539
FGFR2FGFRTK6lvkAn-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12131
FGFR2FGFRTK6lvkBn-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12129
FGFR2FGFRTK6lvlAn-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12132
FGFR2FGFRTK6lvlBn-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12130
FGFR2FGFRTK6v6qAphosphomethylphosphonic acid adenylate esterHuman12968
FGFR2FGFRTK6v6qBphosphomethylphosphonic acid adenylate esterHuman12966
FGFR2FGFRTK6v6qCphosphomethylphosphonic acid adenylate esterHuman12969
FGFR2FGFRTK6v6qDphosphomethylphosphonic acid adenylate esterHuman12967
FGFR2FGFRTK7kiaAA1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13283
FGFR2FGFRTK7kiaAB1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13285
FGFR2FGFRTK7kiaBA1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13281
FGFR2FGFRTK7kiaBB1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13288
FGFR2FGFRTK7kieAAn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13287
FGFR2FGFRTK7kieABn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13286
FGFR2FGFRTK7kieBAn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13282
FGFR2FGFRTK7kieBBn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13284
FGFR2FGFRTK7ozyAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman13999
FGFR2FGFRTK7ozyAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman13998
FGFR2FGFRTK8e1xA(5m)-n-methyl-5-{(6m,8s)-5-{[(3s)-oxolan-3-yl]amino}-6-[1-(propan-2-yl)-1h-pyrazol-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl}pyridine-3-carboxamideHuman14511
FGFR2FGFRTK8h75A4-[9-(2-chlorophenyl)-6-methyl-2,4,5,8,12-pentazatricyclo[8.4.0.0^{3,7}]tetradeca-1(10),3,6,8,11,13-hexaen-13-yl]morpholineHuman14860
FGFR2FGFRTK8stgAn-{4-[(5p)-4-amino-5-{3-fluoro-4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}-2-methylprop-2-enamideHuman14762
FGFR3FGFRTK4k33AAphosphomethylphosphonic acid adenylate esterHuman1871
FGFR3FGFRTK4k33ABphosphomethylphosphonic acid adenylate esterHuman1870
FGFR3FGFRTK6lvmA2-[[5-[2-(3,5-dimethoxyphenyl)ethyl]-2-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]pyrimidin-4-yl]amino]-n-ethyl-benzenesulfonamideHuman12134
FGFR3FGFRTK6pnxAAphosphomethylphosphonic acid adenylate esterHuman11948
FGFR3FGFRTK6pnxABphosphomethylphosphonic acid adenylate esterHuman11946
FGFR3FGFRTK6pnxBAphosphomethylphosphonic acid adenylate esterHuman11947
FGFR3FGFRTK6pnxBBphosphomethylphosphonic acid adenylate esterHuman11949
FGFR3FGFRTK7dhlA5-[2-(3,5-dimethoxyphenyl)ethyl]-n-[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]pyrimidin-2-amineHuman13258
FGFR4FGFRTK4qq5An-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamideHuman921
FGFR4FGFRTK4qqcAAn-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamideHuman934
FGFR4FGFRTK4qqcABn-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamideHuman932
FGFR4FGFRTK4qqjA-Human935
FGFR4FGFRTK4qqtA-Human922
FGFR4FGFRTK4qrcA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman923
FGFR4FGFRTK4r6vAn-[4-({[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino}methyl)phenyl]propanamideHuman931
FGFR4FGFRTK4tyeA-Human927
FGFR4FGFRTK4tygAA-Human929
FGFR4FGFRTK4tygAB-Human933
FGFR4FGFRTK4tyiA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman926
FGFR4FGFRTK4tyjA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman925
FGFR4FGFRTK4uxqA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman930
FGFR4FGFRTK4xcuAAn-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamideHuman928
FGFR4FGFRTK4xcuABn-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamideHuman924
FGFR4FGFRTK5jkgA2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanolHuman7089
FGFR4FGFRTK5nudA3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amineHuman9787
FGFR4FGFRTK5nudB3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amineHuman9790
FGFR4FGFRTK5nwzA~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamideHuman9789
FGFR4FGFRTK5nwzB~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamideHuman9788
FGFR4FGFRTK5xffA2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanolHuman10375
FGFR4FGFRTK5xfjA2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanolHuman10376
FGFR4FGFRTK6iuoAn-({4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}methyl)prop-2-enamideHuman11757
FGFR4FGFRTK6iupAAn-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamideHuman11797
FGFR4FGFRTK6iupABn-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamideHuman11796
FGFR4FGFRTK6jpeAn-[2-[[6-[2-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]amino]pyridin-3-yl]pyrimidin-4-yl]amino]-3-methyl-phenyl]prop-2-enamideHuman12230
FGFR4FGFRTK6jpjAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman11051
FGFR4FGFRTK6nvgAn-[3,5-dichloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)phenyl]propanamideHuman11394
FGFR4FGFRTK6nvhAAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11388
FGFR4FGFRTK6nvhABn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11393
FGFR4FGFRTK6nviAAn-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamideHuman11392
FGFR4FGFRTK6nviABn-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamideHuman11389
FGFR4FGFRTK6nvjAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-fluorophenyl]propanamideHuman11391
FGFR4FGFRTK6nvkAAn-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamideHuman11395
FGFR4FGFRTK6nvkABn-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamideHuman11390
FGFR4FGFRTK6v9cAAn-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamideHuman12096
FGFR4FGFRTK6v9cABn-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamideHuman12095
FGFR4FGFRTK6yi8AAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12812
FGFR4FGFRTK6yi8ABn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12811
FGFR4FGFRTK6yi8BAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12813
FGFR4FGFRTK6yi8BBn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12814
FGFR4FGFRTK7dtzAn-[2-[[5-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]methoxy]pyrimidin-2-yl]amino]-3-methyl-phenyl]-2-fluoranyl-prop-2-enamideHuman13506
FGFR4FGFRTK7f3mA6-[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]-2-(methylamino)-8-[3-(4-prop-2-enoylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidin-7-oneHuman14034
FGFR4FGFRTK7v29An-[2-[[3-(3,5-dimethoxyphenyl)-2-oxidanylidene-1-[3-(4-propanoylpiperazin-1-yl)propyl]-4h-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]propanamideHuman14165
FGFR4FGFRTK7vjlAn-[5-(aminomethyl)-4-(2-methoxyethylamino)pyridin-2-yl]-7-[2,2,2-tris(fluoranyl)ethanoyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman14109
FGFR4FGFRTK7wctA~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamideHuman14167
FGFR4FGFRTK7wcwA~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamideHuman14168
FGFR4FGFRTK7wcxA~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamideHuman14166
FGFR4FGFRTK7yboA~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14499
FGFR4FGFRTK7ybpA~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14500
FGFR4FGFRTK7ybxA~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14502
FGFR4FGFRTK7yc1A~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-propyl-pyrrolo[3,2-b]pyridine-3-carboxamideHuman14498
FGFR4FGFRTK7yc3A6-bromanyl-~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14501
FGRSrcTK7uy0AA7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman14568
FGRSrcTK7uy0AB7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman14563
FGRSrcTK7uy0AC7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman14564
FGRSrcTK7uy0BA7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman14566
FGRSrcTK7uy0BB7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman14565
FGRSrcTK7uy0BC7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman14562
FGRSrcTK7uy3A3-[(6,7-dimethoxyquinazolin-4-yl)oxy]-n-{4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-4-methylbenzamideHuman14567
FLT1VEGFRTK3hngAAn-(4-chlorophenyl)-2-[(pyridin-4-ylmethyl)amino]benzamideHuman3837
FLT1VEGFRTK3hngABn-(4-chlorophenyl)-2-[(pyridin-4-ylmethyl)amino]benzamideHuman3838
FLT3PDGFRTK1rjbA-Human625
FLT3PDGFRTK4rt7AA1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)ureaHuman626
FLT3PDGFRTK4rt7AB1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)ureaHuman627
FLT3PDGFRTK4xufA1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)ureaHuman624
FLT3PDGFRTK4xufB1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-{7-[2-(morpholin-4-yl)ethoxy]imidazo[2,1-b][1,3]benzothiazol-2-yl}phenyl)ureaHuman623
FLT3PDGFRTK5x02An-[(2s)-1-[5-[2-[(4-cyanophenyl)amino]-4-(propylamino)pyrimidin-5-yl]pent-4-ynylamino]-1-oxidanylidene-propan-2-yl]-4-(dimethylamino)-n-methyl-but-2-enamideHuman9522
FLT3PDGFRTK6il3AA7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)-3-(pyridin-2-yl)imidazo[1,2-a]pyridineHuman10785
FLT3PDGFRTK6il3AB7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)-3-(pyridin-2-yl)imidazo[1,2-a]pyridineHuman10786
FLT3PDGFRTK6jqrA6-ethyl-3-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-5-(oxan-4-ylamino)pyrazine-2-carboxamideHuman11802
FYNSrcTK2dq7XstaurosporineHuman1941
GAKNAKOther4c57AA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human341
GAKNAKOther4c57AB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human340
GAKNAKOther4c57BA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human334
GAKNAKOther4c57BB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human348
GAKNAKOther4c58AA9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman336
GAKNAKOther4c58AB9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman333
GAKNAKOther4c59AA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human337
GAKNAKOther4c59AB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human346
GAKNAKOther4o38AA-Human345
GAKNAKOther4o38AB-Human335
GAKNAKOther4o38BA-Human338
GAKNAKOther4o38BB-Human343
GAKNAKOther4y8dAA2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]anilineHuman344
GAKNAKOther4y8dAB2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]anilineHuman339
GAKNAKOther4y8dBA2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]anilineHuman347
GAKNAKOther4y8dBB2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]anilineHuman342
GAKNAKOther5y7zAgefitinibHuman10332
GAKNAKOther5y7zBgefitinibHuman10331
GAKNAKOther5y80AAgefitinibHuman10329
GAKNAKOther5y80ABgefitinibHuman10330
GRK2 (BARK1)GRKAGC3cikA-Human1706
GRK2 (BARK1)GRKAGC3krwAbalanolHuman1707
GRK2 (BARK1)GRKAGC3krxAbalanolHuman1709
GRK2 (BARK1)GRKAGC3v5wAAparoxetineHuman1705
GRK2 (BARK1)GRKAGC3v5wABparoxetineHuman1711
GRK2 (BARK1)GRKAGC4mk0AA5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-oneHuman1710
GRK2 (BARK1)GRKAGC4mk0AB5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-oneHuman1704
GRK2 (BARK1)GRKAGC4pnkAA(4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamideHuman1703
GRK2 (BARK1)GRKAGC4pnkAB(4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamideHuman1708
GRK2 (BARK1)GRKAGC5he1AA(4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamideHuman6605
GRK2 (BARK1)GRKAGC5he1AB(4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamideHuman6606
GRK2 (BARK1)GRKAGC5ukkAA5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamideHuman7529
GRK2 (BARK1)GRKAGC5ukkAB5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamideHuman7530
GRK2 (BARK1)GRKAGC5uklAA2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamideHuman7528
GRK2 (BARK1)GRKAGC5uklAB2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamideHuman7531
GRK2 (BARK1)GRKAGC5uuuAA3-({[4-methyl-5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)-n-[2-(trifluoromethyl)benzyl]benzamideHuman8255
GRK2 (BARK1)GRKAGC5uuuAB3-({[4-methyl-5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)-n-[2-(trifluoromethyl)benzyl]benzamideHuman8254
GRK2 (BARK1)GRKAGC5uvcAn-benzyl-3-({[5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)benzamideHuman8256
GRK2 (BARK1)GRKAGC5wg3A2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(1h-pyrazol-3-yl)methyl]benzamideHuman9439
GRK2 (BARK1)GRKAGC5wg4AA2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamideHuman9441
GRK2 (BARK1)GRKAGC5wg4AB2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamideHuman9438
GRK2 (BARK1)GRKAGC5wg5AA5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazoleHuman9437
GRK2 (BARK1)GRKAGC5wg5AB5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazoleHuman9440
GRK2 (BARK1)GRKAGC6c2yA(4r,5r,6s)-4-[4-fluoro-3-({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}carbamoyl)phenyl]-n-(2h-indazol-5-yl)-6-methyl-2-oxohexahydropyrimidine-5-carboxamideHuman9854
GRK2 (BARK1)GRKAGC6u7cA5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(2h-indazol-3-yl)methyl]benzamideHuman12162
GRK2 (BARK1)GRKAGC7k7lAA3-benzyl-6-(1h-pyrazol-4-yl)quinazolin-4(3h)-oneHuman12960
GRK2 (BARK1)GRKAGC7k7lAB3-benzyl-6-(1h-pyrazol-4-yl)quinazolin-4(3h)-oneHuman12958
GRK2 (BARK1)GRKAGC7k7zAA3-benzyl-7-(1h-pyrazol-4-yl)quinazolin-4(3h)-oneHuman12959
GRK2 (BARK1)GRKAGC7k7zAB3-benzyl-7-(1h-pyrazol-4-yl)quinazolin-4(3h)-oneHuman12961
GRK2 (BARK1)GRKAGC7pwdAA4-chloranyl-n-[2-(4-chlorophenyl)ethyl]thieno[2,3-c]pyridine-2-carboxamideHuman13949
GRK2 (BARK1)GRKAGC7pwdAB4-chloranyl-n-[2-(4-chlorophenyl)ethyl]thieno[2,3-c]pyridine-2-carboxamideHuman13950
GRK4 (GPRK4)GRKAGC4yhjAamp phosphoramidateHuman422
GRK4 (GPRK4)GRKAGC4yhjBamp phosphoramidateHuman423
GRK5 (GPRK5)GRKAGC4tnbAsangivamycinHuman3276
GRK5 (GPRK5)GRKAGC4tndAphosphoaminophosphonic acid-adenylate esterHuman3275
GRK5 (GPRK5)GRKAGC6pjxAAsangivamycinHuman13042
GRK5 (GPRK5)GRKAGC6pjxABsangivamycinHuman13041
GRK5 (GPRK5)GRKAGC8uapA(3z)-3-{[4-(2-chloroacetamido)-3,5-dimethyl-1h-pyrrol-2-yl]methylidene}-n-[(1r)-1-(4-fluorophenyl)ethyl]-2-oxo-2,3-dihydro-1h-indole-5-carboxamideHuman15093
GRK5 (GPRK5)GRKAGC8uaqA(3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-[(4-{[(2s)-2-(furan-2-yl)-2-hydroxyacetyl]amino}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamideHuman15092
GRK6 (GPRK6)GRKAGC2acxAphosphoaminophosphonic acid-adenylate esterHuman420
GRK6 (GPRK6)GRKAGC2acxBphosphoaminophosphonic acid-adenylate esterHuman417
GRK6 (GPRK6)GRKAGC3nynAsangivamycinHuman419
GRK6 (GPRK6)GRKAGC3nynBsangivamycinHuman416
GRK6 (GPRK6)GRKAGC3nyoAadenosine monophosphateHuman418
GRK6 (GPRK6)GRKAGC3nyoBadenosine monophosphateHuman421
GSK3AGSKCMGC7sxfAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14781
GSK3AGSKCMGC7sxfAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14780
GSK3AGSKCMGC7sxgAA(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14783
GSK3AGSKCMGC7sxgAB(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14782
Gsk3b (GSK3B)GSKCMGC4nu1AAadenosine-5'-diphosphateMouse5699
Gsk3b (GSK3B)GSKCMGC4nu1ABadenosine-5'-diphosphateMouse5700
Gsk3b (GSK3B)GSKCMGC5airA-Mouse6863
Gsk3b (GSK3B)GSKCMGC5airB-Mouse6864
Gsk3b (GSK3B)GSKCMGC6ae3A2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-oneMouse10607
Gsk3b (GSK3B)GSKCMGC6ae3B2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-oneMouse10606
Gsk3b (GSK3B)GSKCMGC6ae3C-Mouse10605
Gsk3b (GSK3B)GSKCMGC6ae3D-Mouse10604
GSK3BGSKCMGC1gngA-Human665
GSK3BGSKCMGC1gngB-Human700
GSK3BGSKCMGC1h8fA-Human745
GSK3BGSKCMGC1h8fB-Human666
GSK3BGSKCMGC1i09A-Human630
GSK3BGSKCMGC1i09B-Human638
GSK3BGSKCMGC1j1bAphosphoaminophosphonic acid-adenylate esterHuman707
GSK3BGSKCMGC1j1bBphosphoaminophosphonic acid-adenylate esterHuman657
GSK3BGSKCMGC1j1cAadenosine-5'-diphosphateHuman696
GSK3BGSKCMGC1j1cBadenosine-5'-diphosphateHuman677
GSK3BGSKCMGC1o9uA9-methyl-9h-purin-6-amineHuman708
GSK3BGSKCMGC1pyxAphosphoaminophosphonic acid-adenylate esterHuman645
GSK3BGSKCMGC1pyxBphosphoaminophosphonic acid-adenylate esterHuman663
GSK3BGSKCMGC1q3dAstaurosporineHuman705
GSK3BGSKCMGC1q3dBstaurosporineHuman752
GSK3BGSKCMGC1q3wA9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-oneHuman635
GSK3BGSKCMGC1q3wB9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-oneHuman693
GSK3BGSKCMGC1q41A(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman628
GSK3BGSKCMGC1q41B(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman658
GSK3BGSKCMGC1q4lA2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acidHuman714
GSK3BGSKCMGC1q4lB2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acidHuman655
GSK3BGSKCMGC1q5kAn-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)ureaHuman680
GSK3BGSKCMGC1q5kBn-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)ureaHuman651
GSK3BGSKCMGC1r0eAA3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman733
GSK3BGSKCMGC1r0eAB3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman672
GSK3BGSKCMGC1r0eBA3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman687
GSK3BGSKCMGC1r0eBB3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman639
GSK3BGSKCMGC1uv5A6-bromoindirubin-3'-oximeHuman759
GSK3BGSKCMGC2jldAAruthenium pyridocarbazoleHuman7213
GSK3BGSKCMGC2jldABruthenium pyridocarbazoleHuman7214
GSK3BGSKCMGC2jldBAruthenium pyridocarbazoleHuman7205
GSK3BGSKCMGC2jldBBruthenium pyridocarbazoleHuman7209
GSK3BGSKCMGC2o5kA2-(2,4-dichloro-phenyl)-7-hydroxy-1h-benzoimidazole-4-carboxylic acid [2-(4-methanesulfonylamino-phenyl)-ethyl]-amideHuman633
GSK3BGSKCMGC2ow3Abis-(indole)maleimide pyridinophaneHuman698
GSK3BGSKCMGC2ow3Bbis-(indole)maleimide pyridinophaneHuman649
GSK3BGSKCMGC3du8A(7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman701
GSK3BGSKCMGC3du8B(7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman737
GSK3BGSKCMGC3f7zAA2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman743
GSK3BGSKCMGC3f7zAB2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman647
GSK3BGSKCMGC3f7zAC2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman685
GSK3BGSKCMGC3f7zBA2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman749
GSK3BGSKCMGC3f7zBB2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman670
GSK3BGSKCMGC3f7zBC2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman686
GSK3BGSKCMGC3f88AA5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman741
GSK3BGSKCMGC3f88AB5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman679
GSK3BGSKCMGC3f88BA5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman744
GSK3BGSKCMGC3f88BB5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman756
GSK3BGSKCMGC3gb2AA2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazoleHuman727
GSK3BGSKCMGC3gb2AB2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazoleHuman734
GSK3BGSKCMGC3i4bAn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHuman646
GSK3BGSKCMGC3i4bBn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHuman629
GSK3BGSKCMGC3l1sA(4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-oneHuman757
GSK3BGSKCMGC3l1sB(4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-oneHuman713
GSK3BGSKCMGC3m1sAAruthenium pyridocarbazoleHuman7212
GSK3BGSKCMGC3m1sABruthenium pyridocarbazoleHuman7206
GSK3BGSKCMGC3m1sBAruthenium pyridocarbazoleHuman7210
GSK3BGSKCMGC3m1sBBruthenium pyridocarbazoleHuman7208
GSK3BGSKCMGC3pupAruthenium octasporineHuman7207
GSK3BGSKCMGC3pupBruthenium octasporineHuman7211
GSK3BGSKCMGC3q3bA4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHuman660
GSK3BGSKCMGC3q3bB4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHuman674
GSK3BGSKCMGC3sayAA(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman738
GSK3BGSKCMGC3sayAB(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman661
GSK3BGSKCMGC3sayBA(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman682
GSK3BGSKCMGC3sayBB(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman710
GSK3BGSKCMGC3sd0A3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dioneHuman720
GSK3BGSKCMGC3sd0B3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dioneHuman673
GSK3BGSKCMGC3zdiA3,6-diamino-4-(2-chlorophenyl)thieno[2,3-b]pyridine-2,5-dicarbonitrileHuman748
GSK3BGSKCMGC3zrkAA2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman675
GSK3BGSKCMGC3zrkAB2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman644
GSK3BGSKCMGC3zrkAC2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman697
GSK3BGSKCMGC3zrkBA2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman637
GSK3BGSKCMGC3zrkBB2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman662
GSK3BGSKCMGC3zrkBC2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman731
GSK3BGSKCMGC3zrlAA7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman712
GSK3BGSKCMGC3zrlAB7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman725
GSK3BGSKCMGC3zrlAC7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman654
GSK3BGSKCMGC3zrlBA7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman718
GSK3BGSKCMGC3zrlBB7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman691
GSK3BGSKCMGC3zrlBC7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman676
GSK3BGSKCMGC3zrmAA7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman751
GSK3BGSKCMGC3zrmAB7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman648
GSK3BGSKCMGC3zrmAC7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman724
GSK3BGSKCMGC3zrmBA7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman753
GSK3BGSKCMGC3zrmBB7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman652
GSK3BGSKCMGC3zrmBC7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman706
GSK3BGSKCMGC4accA3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman704
GSK3BGSKCMGC4accB3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman669
GSK3BGSKCMGC4acdA3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamideHuman723
GSK3BGSKCMGC4acdB3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamideHuman692
GSK3BGSKCMGC4acgA2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamideHuman681
GSK3BGSKCMGC4acgB2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamideHuman721
GSK3BGSKCMGC4achA3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamideHuman653
GSK3BGSKCMGC4achB3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamideHuman702
GSK3BGSKCMGC4afjAA5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman632
GSK3BGSKCMGC4afjAB5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman683
GSK3BGSKCMGC4afjAC5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman742
GSK3BGSKCMGC4afjBA5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman678
GSK3BGSKCMGC4afjBB5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman726
GSK3BGSKCMGC4afjBC5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman711
GSK3BGSKCMGC4b7tA(5z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-methyl-2-(propan-2-ylamino)imidazol-4-oneHuman732
GSK3BGSKCMGC4ditAn-(pyridin-3-yl)-2-(thiophen-3-yl)-3h-imidazo[4,5-b]pyridine-7-carboxamideHuman689
GSK3BGSKCMGC4iq6A6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amineHuman728
GSK3BGSKCMGC4iq6B6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amineHuman750
GSK3BGSKCMGC4j1rA(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman709
GSK3BGSKCMGC4j1rB(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman656
GSK3BGSKCMGC4j1rC(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman688
GSK3BGSKCMGC4j1rD(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman736
GSK3BGSKCMGC4j71AA(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman642
GSK3BGSKCMGC4j71AB(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman690
GSK3BGSKCMGC4j71BA(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman641
GSK3BGSKCMGC4j71BB(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman739
GSK3BGSKCMGC4nm0AAadenosine-5'-diphosphateHuman715
GSK3BGSKCMGC4nm0ABadenosine-5'-diphosphateHuman671
GSK3BGSKCMGC4nm3AAadenosine-5'-diphosphateHuman730
GSK3BGSKCMGC4nm3ABadenosine-5'-diphosphateHuman640
GSK3BGSKCMGC4nm5AAadenosine-5'-diphosphateHuman755
GSK3BGSKCMGC4nm5ABadenosine-5'-diphosphateHuman694
GSK3BGSKCMGC4nm7AAadenosine-5'-diphosphateHuman695
GSK3BGSKCMGC4nm7ABadenosine-5'-diphosphateHuman684
GSK3BGSKCMGC4ptcAA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman664
GSK3BGSKCMGC4ptcAB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman659
GSK3BGSKCMGC4ptcBA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman747
GSK3BGSKCMGC4ptcBB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman758
GSK3BGSKCMGC4pteAAn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman716
GSK3BGSKCMGC4pteABn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman717
GSK3BGSKCMGC4pteBAn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman722
GSK3BGSKCMGC4pteBBn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman667
GSK3BGSKCMGC4ptgAA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman735
GSK3BGSKCMGC4ptgAB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman634
GSK3BGSKCMGC4ptgBA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman740
GSK3BGSKCMGC4ptgBB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman754
GSK3BGSKCMGC5f94AA2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6374
GSK3BGSKCMGC5f94AB2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6369
GSK3BGSKCMGC5f94BA2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6372
GSK3BGSKCMGC5f94BB2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6371
GSK3BGSKCMGC5f95A2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamideHuman6373
GSK3BGSKCMGC5f95B2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamideHuman6370
GSK3BGSKCMGC5hlnAchir99021Human6649
GSK3BGSKCMGC5hlnBchir99021Human6650
GSK3BGSKCMGC5hlpAA4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6647
GSK3BGSKCMGC5hlpAB4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6648
GSK3BGSKCMGC5hlpBA4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6646
GSK3BGSKCMGC5hlpBB4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6645
GSK3BGSKCMGC5k5nA5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamideHuman7411
GSK3BGSKCMGC5k5nB5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamideHuman7410
GSK3BGSKCMGC5kpkA(4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9735
GSK3BGSKCMGC5kpkB(4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9731
GSK3BGSKCMGC5kplAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9729
GSK3BGSKCMGC5kplAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9730
GSK3BGSKCMGC5kplBA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9728
GSK3BGSKCMGC5kplBB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9733
GSK3BGSKCMGC5kpmA(4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9732
GSK3BGSKCMGC5kpmB(4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9734
GSK3BGSKCMGC5oy4A~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamideHuman8621
GSK3BGSKCMGC5oy4B~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamideHuman8622
GSK3BGSKCMGC5t31A(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9565
GSK3BGSKCMGC5t31B(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9564
GSK3BGSKCMGC6b8jAAchir99021Human8658
GSK3BGSKCMGC6b8jABchir99021Human8659
GSK3BGSKCMGC6gjoA(3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-oneHuman10974
GSK3BGSKCMGC6gjoB(3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-oneHuman10973
GSK3BGSKCMGC6gn1A~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamideHuman9997
GSK3BGSKCMGC6gn1B~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamideHuman9996
GSK3BGSKCMGC6h0uA(2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamideHuman11049
GSK3BGSKCMGC6h0uB(2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamideHuman11050
GSK3BGSKCMGC6hk3AA3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11425
GSK3BGSKCMGC6hk3AB3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11426
GSK3BGSKCMGC6hk3BA3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11422
GSK3BGSKCMGC6hk3BB3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11424
GSK3BGSKCMGC6hk4AA3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11429
GSK3BGSKCMGC6hk4AB3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11423
GSK3BGSKCMGC6hk4BA3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11430
GSK3BGSKCMGC6hk4BB3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11427
GSK3BGSKCMGC6hk7A3-azanyl-~{n}-(2-methoxyethyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11428
GSK3BGSKCMGC6tcuAA5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamideHuman12780
GSK3BGSKCMGC6tcuAB5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamideHuman12781
GSK3BGSKCMGC6v6lAA-Human11913
GSK3BGSKCMGC6v6lAB-Human11912
GSK3BGSKCMGC6y9rAA~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamideHuman12287
GSK3BGSKCMGC6y9rAB~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamideHuman12289
GSK3BGSKCMGC6y9sAA~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12286
GSK3BGSKCMGC6y9sAB~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12290
GSK3BGSKCMGC6y9sBA~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12285
GSK3BGSKCMGC6y9sBB~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12288
GSK3BGSKCMGC7b6fAA3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrileHuman13069
GSK3BGSKCMGC7b6fAB3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrileHuman13070
GSK3BGSKCMGC7oy5AA~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHuman14118
GSK3BGSKCMGC7oy5AB~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHuman14119
GSK3BGSKCMGC7sxhAA(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14787
GSK3BGSKCMGC7sxhAB(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14784
GSK3BGSKCMGC7sxjAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14785
GSK3BGSKCMGC7sxjAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14786
GSK3BGSKCMGC7u2zAA(3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHuman14203
GSK3BGSKCMGC7u2zAB(3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHuman14202
GSK3BGSKCMGC7u31AA5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amineHuman14199
GSK3BGSKCMGC7u31AB5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amineHuman14201
GSK3BGSKCMGC7u33AA3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamideHuman14198
GSK3BGSKCMGC7u33AB3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamideHuman14200
GSK3BGSKCMGC7u36A(3s)-1-[(2-fluorophenoxy)acetyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHuman14204
GSK3BGSKCMGC7z1fA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman14663
GSK3BGSKCMGC7z1gA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman14662
GSK3BGSKCMGC8auzAA8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14707
GSK3BGSKCMGC8auzAB8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14708
GSK3BGSKCMGC8av1AA2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14706
GSK3BGSKCMGC8av1AB2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14709
GSK3BGSKCMGC8djcAA(4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamideHuman14672
GSK3BGSKCMGC8djcAB(4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamideHuman14669
GSK3BGSKCMGC8djdAA2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamideHuman14673
GSK3BGSKCMGC8djdAB2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamideHuman14668
GSK3BGSKCMGC8djeAA(4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamideHuman14670
GSK3BGSKCMGC8djeAB(4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamideHuman14671
GSK3BGSKCMGC8ff8A2-(4-cyanoanilino)-n-(4-phenylpyridin-3-yl)pyrimidine-4-carboxamideHuman14763
GUCY2C (HSER)RGCRGC8fx4D-Human14837
HASPIN (Haspin)HaspinOther2vuwAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman3809
HASPIN (Haspin)HaspinOther2vuwAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman3801
HASPIN (Haspin)HaspinOther2wb8AA-Human3802
HASPIN (Haspin)HaspinOther2wb8AB-Human3815
HASPIN (Haspin)HaspinOther3dlzAAadenosine monophosphateHuman3804
HASPIN (Haspin)HaspinOther3dlzABadenosine monophosphateHuman3808
HASPIN (Haspin)HaspinOther3e7vAA3-(3-aminophenyl)-n-(3-chlorophenyl)pyrazolo[1,5-a]pyrimidin-5-amineHuman3814
HASPIN (Haspin)HaspinOther3e7vAB3-(3-aminophenyl)-n-(3-chlorophenyl)pyrazolo[1,5-a]pyrimidin-5-amineHuman3799
HASPIN (Haspin)HaspinOther3f2nAA(2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-olHuman3803
HASPIN (Haspin)HaspinOther3f2nAB(2s)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-olHuman3813
HASPIN (Haspin)HaspinOther3fmdAAn-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamideHuman3798
HASPIN (Haspin)HaspinOther3fmdABn-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamideHuman3810
HASPIN (Haspin)HaspinOther3iq7AA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman3807
HASPIN (Haspin)HaspinOther3iq7AB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman3811
HASPIN (Haspin)HaspinOther4oucAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman3806
HASPIN (Haspin)HaspinOther4oucAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman3812
HASPIN (Haspin)HaspinOther4qtcAA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman3805
HASPIN (Haspin)HaspinOther4qtcAB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman3800
HASPIN (Haspin)HaspinOther5htbAA-Human6620
HASPIN (Haspin)HaspinOther5htbAB-Human6621
HASPIN (Haspin)HaspinOther5htcAA-Human6445
HASPIN (Haspin)HaspinOther5htcAB-Human6446
HASPIN (Haspin)HaspinOther5htcAC-Human6444
HASPIN (Haspin)HaspinOther6g34AA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9832
HASPIN (Haspin)HaspinOther6g34AB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9846
HASPIN (Haspin)HaspinOther6g35AA5-bromotubercidinHuman9843
HASPIN (Haspin)HaspinOther6g35AB5-bromotubercidinHuman9841
HASPIN (Haspin)HaspinOther6g35AC-Human9837
HASPIN (Haspin)HaspinOther6g35AD-Human9829
HASPIN (Haspin)HaspinOther6g36AA5-chlorotubercidinHuman9834
HASPIN (Haspin)HaspinOther6g36AB5-chlorotubercidinHuman9844
HASPIN (Haspin)HaspinOther6g37AA5-fluorotubercidinHuman9840
HASPIN (Haspin)HaspinOther6g37AB5-fluorotubercidinHuman9845
HASPIN (Haspin)HaspinOther6g38AA'2-(4-amino-pyrrolo[2,3-d]pyrimidin-7-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diolHuman9830
HASPIN (Haspin)HaspinOther6g38AB'2-(4-amino-pyrrolo[2,3-d]pyrimidin-7-yl)-5-hydroxymethyl-tetrahydro-furan-3,4-diolHuman9842
HASPIN (Haspin)HaspinOther6g39AA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9839
HASPIN (Haspin)HaspinOther6g39AB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9831
HASPIN (Haspin)HaspinOther6g39AC-Human9838
HASPIN (Haspin)HaspinOther6g39AD-Human9833
HASPIN (Haspin)HaspinOther6g3aAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9836
HASPIN (Haspin)HaspinOther6g3aAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9835
HASPIN (Haspin)HaspinOther6z56AA6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12322
HASPIN (Haspin)HaspinOther6z56AB6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12333
HASPIN (Haspin)HaspinOther6z56AC6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12320
HASPIN (Haspin)HaspinOther6z57AA10-(2-morpholin-4-ylethyl)-7-oxa-10,13,17,18,21-pentazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaeneHuman12321
HASPIN (Haspin)HaspinOther6z57AB10-(2-morpholin-4-ylethyl)-7-oxa-10,13,17,18,21-pentazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaeneHuman12323
HASPIN (Haspin)HaspinOther6z58AA8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-oneHuman12327
HASPIN (Haspin)HaspinOther6z58AB8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-oneHuman12332
HASPIN (Haspin)HaspinOther6z59AA11-oxa-8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-oneHuman12326
HASPIN (Haspin)HaspinOther6z59AB11-oxa-8,14,18,19,22-pentazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2,4,6(23),15(22),16,19-heptaen-7-oneHuman12316
HASPIN (Haspin)HaspinOther6z5aAAn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide Human12328
HASPIN (Haspin)HaspinOther6z5aABn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide Human12324
HASPIN (Haspin)HaspinOther6z5bAA6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12331
HASPIN (Haspin)HaspinOther6z5bAB6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12334
HASPIN (Haspin)HaspinOther6z5cAA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12319
HASPIN (Haspin)HaspinOther6z5cAB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12318
HASPIN (Haspin)HaspinOther6z5dAA11-methyl-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one Human12325
HASPIN (Haspin)HaspinOther6z5dAB11-methyl-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one Human12330
HASPIN (Haspin)HaspinOther6z5eAA11-cyclopropyl-14-(2-hydroxyethyl)-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one Human12317
HASPIN (Haspin)HaspinOther6z5eAB11-cyclopropyl-14-(2-hydroxyethyl)-8,11,14,18,19,22-hexazatetracyclo[13.5.2.12,6.018,21]tricosa-1(21),2(23),3,5,15(22),16,19-heptaen-7-one Human12329
HASPIN (Haspin)HaspinOther7avqAA(2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olHuman13176
HASPIN (Haspin)HaspinOther7avqAB(2~{r})-2-[[3-(2~{h}-indazol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olHuman13175
HASPIN (Haspin)HaspinOther7opsA2-methylsulfanyl-10-nitro-pyrido[3,4-g]quinazolineHuman13815
HASPIN (Haspin)HaspinOther7sqmAA1-[(4s)-5-(2,4-difluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-4-methylpiperidin-4-amineHuman14033
HASPIN (Haspin)HaspinOther7sqmAB1-[(4s)-5-(2,4-difluorophenyl)imidazo[2,1-b][1,3,4]thiadiazol-2-yl]-4-methylpiperidin-4-amineHuman14032
HCKSrcTK1ad5Aphosphoaminophosphonic acid-adenylate esterHuman9480
HCKSrcTK1ad5Bphosphoaminophosphonic acid-adenylate esterHuman9483
HCKSrcTK1qcfA1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamineHuman2641
HCKSrcTK2c0iAAn-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2662
HCKSrcTK2c0iABn-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2649
HCKSrcTK2c0iBAn-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2650
HCKSrcTK2c0iBBn-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2640
HCKSrcTK2c0oAAn-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2666
HCKSrcTK2c0oABn-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2652
HCKSrcTK2c0oBAn-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2663
HCKSrcTK2c0oBBn-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2657
HCKSrcTK2c0tAAn-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2653
HCKSrcTK2c0tABn-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2667
HCKSrcTK2c0tBAn-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2642
HCKSrcTK2c0tBBn-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamideHuman2634
HCKSrcTK2hckA3,5,7,3',4'-pentahydroxyflavoneHuman9481
HCKSrcTK2hckB3,5,7,3',4'-pentahydroxyflavoneHuman9482
HCKSrcTK2hk5A3-{[2-(1h-benzimidazol-1-yl)-6-{[2-(diethylamino)ethyl]amino}pyrimidin-4-yl]amino}-4-methylphenolHuman2639
HCKSrcTK3vryA4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentaneHuman2647
HCKSrcTK3vryB4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentaneHuman2646
HCKSrcTK3vrzA1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-benzylureaHuman2658
HCKSrcTK3vrzB1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-benzylureaHuman2661
HCKSrcTK3vs0An-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]benzamideHuman2633
HCKSrcTK3vs0Bn-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]benzamideHuman2644
HCKSrcTK3vs1A1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-phenylureaHuman2635
HCKSrcTK3vs1B1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-phenylureaHuman2636
HCKSrcTK3vs2A7-[cis-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2651
HCKSrcTK3vs2B7-[cis-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2632
HCKSrcTK3vs3A7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2643
HCKSrcTK3vs3B7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2665
HCKSrcTK3vs4A5-(4-phenoxyphenyl)-7-(tetrahydro-2h-pyran-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2654
HCKSrcTK3vs4B5-(4-phenoxyphenyl)-7-(tetrahydro-2h-pyran-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2638
HCKSrcTK3vs5A7-(1-methylpiperidin-4-yl)-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2645
HCKSrcTK3vs5B7-(1-methylpiperidin-4-yl)-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2669
HCKSrcTK3vs6Atert-butyl {4-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl}carbamateHuman2664
HCKSrcTK3vs6Btert-butyl {4-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl}carbamateHuman2656
HCKSrcTK3vs7A1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman2659
HCKSrcTK3vs7B1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman2648
HCKSrcTK4ludA6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazoleHuman2660
HCKSrcTK4ludB6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazoleHuman2637
HCKSrcTK4lueA7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2655
HCKSrcTK4lueB7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman2668
HCKSrcTK5h09Aethyl (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-4-methyl-pentanoateHuman8537
HCKSrcTK5h0bA(2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]azaniumyl]-4-methyl-pentanoateHuman8567
HCKSrcTK5h0eA(2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-4-methyl-pentanamideHuman8538
HCKSrcTK5h0gA(2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-~{n},4-dimethyl-pentanamideHuman8536
HCKSrcTK5h0hA(2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-~{n},~{n},4-trimethyl-pentanamideHuman8539
HCKSrcTK5zj6A7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman9987
HCKSrcTK5zj6B7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman9988
HIPK2DYRKCMGC6p5sAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11512
HIPK2DYRKCMGC6p5sAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11513
HIPK2DYRKCMGC7ncfA3-(4-tert-butylphenyl)-5-(1h-pyrazol-4-yl)furo[3,2-b]pyridineHuman13393
HIPK3DYRKCMGC7o7iA-Human13996
HIPK3DYRKCMGC7o7jAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman13997
Igf1r (IGF1R)InsRTK6pyhA-Mouse11777
Igf1r (IGF1R)InsRTK6pyhD-Mouse11776
IGF1RInsRTK1jqhAphosphoaminophosphonic acid-adenylate esterHuman999
IGF1RInsRTK1jqhBphosphoaminophosphonic acid-adenylate esterHuman994
IGF1RInsRTK1jqhCphosphoaminophosphonic acid-adenylate esterHuman1038
IGF1RInsRTK1k3aAphosphomethylphosphonic acid adenylate esterHuman1028
IGF1RInsRTK1m7nA-Human1007
IGF1RInsRTK1m7nB-Human1012
IGF1RInsRTK1p4oA-Human1002
IGF1RInsRTK1p4oB-Human1026
IGF1RInsRTK2oj9A3-[5-(1h-imidazol-1-yl)-7-methyl-1h-benzimidazol-2-yl]-4-[(pyridin-2-ylmethyl)amino]pyridin-2(1h)-oneHuman1017
IGF1RInsRTK2zm3A(4z)-6-bromo-4-({[4-(pyrrolidin-1-ylmethyl)phenyl]amino}methylidene)isoquinoline-1,3(2h,4h)-dioneHuman1004
IGF1RInsRTK2zm3B(4z)-6-bromo-4-({[4-(pyrrolidin-1-ylmethyl)phenyl]amino}methylidene)isoquinoline-1,3(2h,4h)-dioneHuman1000
IGF1RInsRTK2zm3C(4z)-6-bromo-4-({[4-(pyrrolidin-1-ylmethyl)phenyl]amino}methylidene)isoquinoline-1,3(2h,4h)-dioneHuman1010
IGF1RInsRTK2zm3D(4z)-6-bromo-4-({[4-(pyrrolidin-1-ylmethyl)phenyl]amino}methylidene)isoquinoline-1,3(2h,4h)-dioneHuman1023
IGF1RInsRTK3d94AA3-[cis-3-(4-methylpiperazin-1-yl)cyclobutyl]-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-8-amineHuman6759
IGF1RInsRTK3d94AB3-[cis-3-(4-methylpiperazin-1-yl)cyclobutyl]-1-(2-phenylquinolin-7-yl)imidazo[1,5-a]pyrazin-8-amineHuman6760
IGF1RInsRTK3f5pA4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman995
IGF1RInsRTK3f5pB4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1044
IGF1RInsRTK3f5pC4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1022
IGF1RInsRTK3f5pD4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1015
IGF1RInsRTK3f5pE4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1042
IGF1RInsRTK3f5pF4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1029
IGF1RInsRTK3f5pG4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1005
IGF1RInsRTK3f5pH4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1006
IGF1RInsRTK3f5pI4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1016
IGF1RInsRTK3f5pJ4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1040
IGF1RInsRTK3f5pK4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1013
IGF1RInsRTK3f5pL4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1039
IGF1RInsRTK3f5pM4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1001
IGF1RInsRTK3f5pR4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1019
IGF1RInsRTK3f5pS4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman996
IGF1RInsRTK3f5pT4-[[3-chloro-4-(1-methylimidazol-2-yl)sulfanyl-phenyl]amino]-7-[3-(2-hydroxyethyl-methyl-amino)propoxy]-6-methoxy-quinoline-3-carbonitrileHuman1037
IGF1RInsRTK3i81A1-{4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}-n-(6-fluoropyridin-3-yl)-2-methyl-l-prolinamideHuman1041
IGF1RInsRTK3lvpA3-(4-chloro-1h-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dimethoxy-1-methyl-1h-pyrrolo[3,2-b]pyridineHuman1032
IGF1RInsRTK3lvpB3-(4-chloro-1h-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dimethoxy-1-methyl-1h-pyrrolo[3,2-b]pyridineHuman1035
IGF1RInsRTK3lvpC3-(4-chloro-1h-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dimethoxy-1-methyl-1h-pyrrolo[3,2-b]pyridineHuman1003
IGF1RInsRTK3lvpD3-(4-chloro-1h-pyrrolo[2,3-b]pyridin-2-yl)-5,6-dimethoxy-1-methyl-1h-pyrrolo[3,2-b]pyridineHuman1009
IGF1RInsRTK3lw0AA-Human1021
IGF1RInsRTK3lw0AB-Human1031
IGF1RInsRTK3lw0BA-Human993
IGF1RInsRTK3lw0BB-Human1008
IGF1RInsRTK3lw0CA-Human1011
IGF1RInsRTK3lw0CB-Human1025
IGF1RInsRTK3lw0DA-Human1033
IGF1RInsRTK3lw0DB-Human1027
IGF1RInsRTK3nw5An-(5-cyclopropyl-1h-pyrazol-3-yl)-2-{(2r)-1-[(6-fluoropyridin-3-yl)carbonyl]pyrrolidin-2-yl}pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman998
IGF1RInsRTK3nw6An-(5-cyclopropyl-1h-pyrazol-3-yl)-2-{(2s)-1-[(6-fluoropyridin-3-yl)carbonyl]pyrrolidin-2-yl}pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman1043
IGF1RInsRTK3nw7An-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}methyl)-6-fluoropyridine-3-carboxamideHuman1030
IGF1RInsRTK3o23A(5s)-5-methyl-1-(quinolin-4-ylmethyl)-3-{4-[(trifluoromethyl)sulfonyl]phenyl}imidazolidine-2,4-dioneHuman1036
IGF1RInsRTK3qquAn~2~-[3-methoxy-4-(morpholin-4-yl)phenyl]-n~4~-(quinolin-3-yl)pyrimidine-2,4-diamineHuman1024
IGF1RInsRTK3qquBn~2~-[3-methoxy-4-(morpholin-4-yl)phenyl]-n~4~-(quinolin-3-yl)pyrimidine-2,4-diamineHuman1020
IGF1RInsRTK3qquCn~2~-[3-methoxy-4-(morpholin-4-yl)phenyl]-n~4~-(quinolin-3-yl)pyrimidine-2,4-diamineHuman1014
IGF1RInsRTK3qquDn~2~-[3-methoxy-4-(morpholin-4-yl)phenyl]-n~4~-(quinolin-3-yl)pyrimidine-2,4-diamineHuman997
IGF1RInsRTK4d2rAAn-{2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]phenyl}-4-(1h-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman1018
IGF1RInsRTK4d2rABn-{2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]phenyl}-4-(1h-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman1034
IGF1RInsRTK5fxqA5-chloranyl-4-imidazo[1,2-a]pyridin-3-yl-n-(5-methyl-1-piperidin-4-yl-pyrazol-4-yl)pyrimidin-2-amineHuman7093
IGF1RInsRTK5fxrAA5-chloranyl-4-imidazo[1,2-a]pyridin-3-yl-n-(3-methyl-1-piperidin-4-yl-pyrazol-4-yl)pyrimidin-2-amineHuman7095
IGF1RInsRTK5fxrAB5-chloranyl-4-imidazo[1,2-a]pyridin-3-yl-n-(3-methyl-1-piperidin-4-yl-pyrazol-4-yl)pyrimidin-2-amineHuman7094
IGF1RInsRTK5fxsAA2-[4-[4-[[(6z)-5-chloranyl-6-pyrazolo[1,5-a]pyridin-3-ylidene-1h-pyrimidin-2-yl]amino]-3,5-dimethyl-pyrazol-1-yl]piperidin-1-yl]-n,n-dimethyl-ethanamideHuman7096
IGF1RInsRTK5fxsAB2-[4-[4-[[(6z)-5-chloranyl-6-pyrazolo[1,5-a]pyridin-3-ylidene-1h-pyrimidin-2-yl]amino]-3,5-dimethyl-pyrazol-1-yl]piperidin-1-yl]-n,n-dimethyl-ethanamideHuman7097
IGF1RInsRTK5hznA7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6493
IGF1RInsRTK5hznB7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6495
IGF1RInsRTK5hznC7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6498
IGF1RInsRTK5hznD7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6496
IGF1RInsRTK5hznE7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6494
IGF1RInsRTK5hznF7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6497
IGF1RInsRTK5hznG7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6499
IGF1RInsRTK5hznH7-[cis-3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-(benzyloxy)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman6492
IGF1RInsRTK6jk8AA-Human12015
IGF1RInsRTK6jk8AB-Human12016
IGF1RInsRTK6jk8BA-Human12018
IGF1RInsRTK6jk8BB-Human12017
IGF1RInsRTK8pyiA3-[8-azanyl-1-(4-ethoxy-8-fluoranyl-2-phenyl-quinolin-7-yl)imidazo[1,5-a]pyrazin-3-yl]-1-methyl-cyclobutan-1-olHuman14903
IGF1RInsRTK8pyjA5,5-dimethyl-1-(quinolin-4-ylmethyl)-3-[4-(trifluoromethylsulfonyl)phenyl]imidazolidine-2,4-dioneHuman14905
IGF1RInsRTK8pykAA5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-3-[4-(trifluoromethylsulfanyl)phenyl]imidazolidine-2,4-dioneHuman14900
IGF1RInsRTK8pykAB5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-3-[4-(trifluoromethylsulfanyl)phenyl]imidazolidine-2,4-dioneHuman14904
IGF1RInsRTK8pylA(5s)-5-methyl-1-(1h-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfanyl)phenyl]imidazolidine-2,4-dioneHuman14906
IGF1RInsRTK8pymA5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfanyl)phenyl]imidazolidine-2,4-dioneHuman14901
IGF1RInsRTK8pynAA5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfonyl)phenyl]imidazolidine-2,4-dioneHuman14902
IGF1RInsRTK8pynAB5,5-dimethyl-1-(1h-pyrrolo[2,3-b]pyridin-4-ylmethyl)-3-[4-(trifluoromethylsulfonyl)phenyl]imidazolidine-2,4-dioneHuman14907
IKBKB (IKKb)IKKOther4e3cA-Human297
IKBKB (IKKb)IKKOther4e3cB-Human294
IKBKB (IKKb)IKKOther4e3cC-Human296
IKBKB (IKKb)IKKOther4e3cD-Human291
IKBKB (IKKb)IKKOther4e3cE-Human289
IKBKB (IKKb)IKKOther4e3cF-Human292
IKBKB (IKKb)IKKOther4kikAAk-252aHuman290
IKBKB (IKKb)IKKOther4kikABk-252aHuman288
IKBKB (IKKb)IKKOther4kikBAk-252aHuman295
IKBKB (IKKb)IKKOther4kikBBk-252aHuman293
ILKMLKTKL3kmuA-Human4606
ILKMLKTKL3kmwAadenosine-5'-triphosphateHuman4605
ILKMLKTKL3repAadenosine-5'-triphosphateHuman4604
ILKMLKTKL6mibA-Human10687
Insr (INSR)InsRTK7sl4A-Mouse14172
Insr (INSR)InsRTK7sl6A-Mouse14171
Insr (INSR)InsRTK7sl7A-Mouse14169
Insr (INSR)InsRTK7stjA-Mouse14170
Insr (INSR)InsRTK8dtlB-Mouse14362
Insr (INSR)InsRTK8eyxA-Mouse14496
Insr (INSR)InsRTK8eyyA-Mouse14497
INSRInsRTK1gagA-Human586
INSRInsRTK1i44Aphosphomethylphosphonic acid adenylate esterHuman582
INSRInsRTK1ir3Aphosphoaminophosphonic acid-adenylate esterHuman602
INSRInsRTK1irkAA-Human596
INSRInsRTK1irkAB-Human603
INSRInsRTK1p14A-Human593
INSRInsRTK1rqqAthiophosphoric acid o-((adenosyl-phospho)phospho)-s-acetamidyl-diesterHuman7407
INSRInsRTK1rqqBthiophosphoric acid o-((adenosyl-phospho)phospho)-s-acetamidyl-diesterHuman7406
INSRInsRTK2auhA-Human584
INSRInsRTK2b4sB-Human585
INSRInsRTK2b4sD-Human583
INSRInsRTK2z8cA[4-({5-(aminocarbonyl)-4-[(3-methylphenyl)amino]pyrimidin-2-yl}amino)phenyl]acetic acidHuman587
INSRInsRTK3bu3A-Human591
INSRInsRTK3bu5Aadenosine-5'-triphosphateHuman595
INSRInsRTK3bu6A-Human601
INSRInsRTK3ekkAA2-[(2-{[1-(n,n-dimethylglycyl)-5-methoxy-1h-indol-6-yl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-6-fluoro-n-methylbenzamideHuman578
INSRInsRTK3ekkAB2-[(2-{[1-(n,n-dimethylglycyl)-5-methoxy-1h-indol-6-yl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-6-fluoro-n-methylbenzamideHuman581
INSRInsRTK3eknAA2-fluoro-6-{[2-({2-methoxy-4-[4-(1-methylethyl)piperazin-1-yl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamideHuman597
INSRInsRTK3eknAB2-fluoro-6-{[2-({2-methoxy-4-[4-(1-methylethyl)piperazin-1-yl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamideHuman594
INSRInsRTK3etaAA1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)ureaHuman590
INSRInsRTK3etaAB1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)ureaHuman579
INSRInsRTK3etaBA1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)ureaHuman588
INSRInsRTK3etaBB1-(3-{5-[4-(aminomethyl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)-3-(2-phenoxyphenyl)ureaHuman600
INSRInsRTK4ibmAA5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-oneHuman589
INSRInsRTK4ibmAB5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-oneHuman598
INSRInsRTK4ibmBA5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-oneHuman604
INSRInsRTK4ibmBB5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-3h-pyrazolo[3,4-c]pyridazin-3-oneHuman599
INSRInsRTK4xlvAphosphomethylphosphonic acid adenylate esterHuman577
INSRInsRTK5e1sAA(5r)-n-(1-{2-[4-(2-methoxyethyl)piperazin-1-yl]ethyl}-1h-pyrazol-3-yl)-5,8-dimethyl-9-phenyl-6,8-dihydro-5h-pyrazolo[3,4-h]quinazolin-2-amineHuman6146
INSRInsRTK5e1sAB(5r)-n-(1-{2-[4-(2-methoxyethyl)piperazin-1-yl]ethyl}-1h-pyrazol-3-yl)-5,8-dimethyl-9-phenyl-6,8-dihydro-5h-pyrazolo[3,4-h]quinazolin-2-amineHuman6147
INSRInsRTK5hhwAA7-[3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-[[(2~{r})-oxan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-4-amineHuman6523
INSRInsRTK5hhwAB7-[3-(azetidin-1-ylmethyl)cyclobutyl]-5-[3-[[(2~{r})-oxan-2-yl]methoxy]phenyl]pyrrolo[2,3-d]pyrimidin-4-amineHuman6522
INSRInsRTK6pxvA-Human11592
INSRInsRTK6pxvC-Human11590
INSRInsRTK6pxwA-Human11593
INSRInsRTK6pxwB-Human11591
INSRInsRTK7bw7A-Human13504
INSRInsRTK7bw7C-Human13505
INSRInsRTK7bw8A-Human13502
INSRInsRTK7bw8C-Human13503
INSRInsRTK7pg0A-Human14097
INSRInsRTK7pg2A-Human14098
INSRInsRTK7pg3A-Human14099
INSRInsRTK7pg4A-Human14100
INSRInsRTK8dwnA-Human14975
INSRR (IRR)InsRTK7tykA-Human14612
INSRR (IRR)InsRTK7tymA-Human14611
IRAK1IRAKTKL6bfnAAn-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamideHuman8698
IRAK1IRAKTKL6bfnABn-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamideHuman8700
IRAK1IRAKTKL6bfnBAn-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamideHuman8701
IRAK1IRAKTKL6bfnBBn-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamideHuman8699
IRAK3IRAKTKL6ruuA-Human12770
IRAK3IRAKTKL6ruuB-Human12769
IRAK3IRAKTKL6ruuC-Human12771
IRAK3IRAKTKL6ziwIphosphothiophosphoric acid-adenylate esterHuman12483
IRAK4IRAKTKL2nruAA1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalateHuman1748
IRAK4IRAKTKL2nruAB1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalateHuman1760
IRAK4IRAKTKL2nruBA1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalateHuman1773
IRAK4IRAKTKL2nruBB1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalateHuman1749
IRAK4IRAKTKL2nruCA1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalateHuman1776
IRAK4IRAKTKL2nruCB1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalateHuman1771
IRAK4IRAKTKL2nruDA1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalateHuman1762
IRAK4IRAKTKL2nruDB1-(3-hydroxypropyl)-2-[(3-nitrobenzoyl)amino]-1h-benzimidazol-5-yl pivalateHuman1787
IRAK4IRAKTKL2nryAAstaurosporineHuman1753
IRAK4IRAKTKL2nryABstaurosporineHuman1777
IRAK4IRAKTKL2nryBAstaurosporineHuman1758
IRAK4IRAKTKL2nryBBstaurosporineHuman1772
IRAK4IRAKTKL2nryCAstaurosporineHuman1779
IRAK4IRAKTKL2nryCBstaurosporineHuman1750
IRAK4IRAKTKL2nryDAstaurosporineHuman1789
IRAK4IRAKTKL2nryDBstaurosporineHuman1746
IRAK4IRAKTKL2o8yA-Human1744
IRAK4IRAKTKL2o8yB-Human1732
IRAK4IRAKTKL2oibAA-Human1756
IRAK4IRAKTKL2oibAB-Human1766
IRAK4IRAKTKL2oibBA-Human1785
IRAK4IRAKTKL2oibBB-Human1743
IRAK4IRAKTKL2oibCA-Human1781
IRAK4IRAKTKL2oibCB-Human1741
IRAK4IRAKTKL2oibDA-Human1736
IRAK4IRAKTKL2oibDB-Human1783
IRAK4IRAKTKL2oicAstaurosporineHuman1739
IRAK4IRAKTKL2oicBstaurosporineHuman1752
IRAK4IRAKTKL2oicCstaurosporineHuman1734
IRAK4IRAKTKL2oicDstaurosporineHuman1755
IRAK4IRAKTKL2oidAphosphoaminophosphonic acid-adenylate esterHuman1764
IRAK4IRAKTKL2oidBphosphoaminophosphonic acid-adenylate esterHuman1759
IRAK4IRAKTKL2oidCphosphoaminophosphonic acid-adenylate esterHuman1775
IRAK4IRAKTKL2oidDphosphoaminophosphonic acid-adenylate esterHuman1733
IRAK4IRAKTKL4rmzAA3-nitro-n-[1-phenyl-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl]benzamideHuman6349
IRAK4IRAKTKL4rmzAB3-nitro-n-[1-phenyl-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl]benzamideHuman6352
IRAK4IRAKTKL4rmzBA3-nitro-n-[1-phenyl-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl]benzamideHuman6351
IRAK4IRAKTKL4rmzBB3-nitro-n-[1-phenyl-5-(piperidin-1-ylmethyl)-1h-benzimidazol-2-yl]benzamideHuman6350
IRAK4IRAKTKL4u97AstaurosporineHuman1754
IRAK4IRAKTKL4u97BstaurosporineHuman1742
IRAK4IRAKTKL4u9aAstaurosporineHuman1751
IRAK4IRAKTKL4u9aBstaurosporineHuman1792
IRAK4IRAKTKL4xs2A(1r,2s,3r,5r)-3-({5-(1,3-benzothiazol-2-yl)-6-chloro-2-[(3-methoxypropyl)amino]pyrimidin-4-yl}amino)-5-(hydroxymethyl)cyclopentane-1,2-diolHuman1765
IRAK4IRAKTKL4xs2B(1r,2s,3r,5r)-3-({5-(1,3-benzothiazol-2-yl)-6-chloro-2-[(3-methoxypropyl)amino]pyrimidin-4-yl}amino)-5-(hydroxymethyl)cyclopentane-1,2-diolHuman1778
IRAK4IRAKTKL4xs2C(1r,2s,3r,5r)-3-({5-(1,3-benzothiazol-2-yl)-6-chloro-2-[(3-methoxypropyl)amino]pyrimidin-4-yl}amino)-5-(hydroxymethyl)cyclopentane-1,2-diolHuman1791
IRAK4IRAKTKL4xs2D(1r,2s,3r,5r)-3-({5-(1,3-benzothiazol-2-yl)-6-chloro-2-[(3-methoxypropyl)amino]pyrimidin-4-yl}amino)-5-(hydroxymethyl)cyclopentane-1,2-diolHuman1738
IRAK4IRAKTKL4y73AA5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman9123
IRAK4IRAKTKL4y73AB5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman9129
IRAK4IRAKTKL4y73BA5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman9128
IRAK4IRAKTKL4y73BB5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman9125
IRAK4IRAKTKL4y73CA5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman9130
IRAK4IRAKTKL4y73CB5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman9124
IRAK4IRAKTKL4y73DA5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman9127
IRAK4IRAKTKL4y73DB5-{[(1r,2s)-2-aminocyclohexyl]amino}-n-[1-methyl-3-(trifluoromethyl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman9126
IRAK4IRAKTKL4yo6AAn-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1793
IRAK4IRAKTKL4yo6ABn-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1763
IRAK4IRAKTKL4yo6BAn-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1747
IRAK4IRAKTKL4yo6BBn-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1769
IRAK4IRAKTKL4yo6CAn-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1780
IRAK4IRAKTKL4yo6CBn-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1737
IRAK4IRAKTKL4yo6DAn-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1768
IRAK4IRAKTKL4yo6DBn-(3-methyl-1-phenyl-1h-pyrazol-5-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1788
IRAK4IRAKTKL4yp8An-{1-(4-cyclopropyl-2-fluorophenyl)-3-[1-(propan-2-yl)piperidin-4-yl]-1h-pyrazol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1740
IRAK4IRAKTKL4yp8Bn-{1-(4-cyclopropyl-2-fluorophenyl)-3-[1-(propan-2-yl)piperidin-4-yl]-1h-pyrazol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1786
IRAK4IRAKTKL4yp8Cn-{1-(4-cyclopropyl-2-fluorophenyl)-3-[1-(propan-2-yl)piperidin-4-yl]-1h-pyrazol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1735
IRAK4IRAKTKL4yp8Dn-{1-(4-cyclopropyl-2-fluorophenyl)-3-[1-(propan-2-yl)piperidin-4-yl]-1h-pyrazol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman1745
IRAK4IRAKTKL4ztlAA(1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diolHuman6003
IRAK4IRAKTKL4ztlAB(1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diolHuman5994
IRAK4IRAKTKL4ztlBA(1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diolHuman6009
IRAK4IRAKTKL4ztlBB(1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diolHuman6004
IRAK4IRAKTKL4ztlCA(1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diolHuman5998
IRAK4IRAKTKL4ztlCB(1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diolHuman5990
IRAK4IRAKTKL4ztlDA(1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diolHuman5996
IRAK4IRAKTKL4ztlDB(1r,2s,3r,5r)-3-{[5-(1,3-benzothiazol-2-yl)-2-(propylamino)pyrimidin-4-yl]amino}-5-(hydroxymethyl)cyclopentane-1,2-diolHuman6000
IRAK4IRAKTKL4ztmA5-(1,3-benzothiazol-2-yl)-2-(cyclopropylamino)-6-{[(1r,2s,3r,4r)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino}pyrimidin-4(3h)-oneHuman5997
IRAK4IRAKTKL4ztmB5-(1,3-benzothiazol-2-yl)-2-(cyclopropylamino)-6-{[(1r,2s,3r,4r)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino}pyrimidin-4(3h)-oneHuman5992
IRAK4IRAKTKL4ztmC5-(1,3-benzothiazol-2-yl)-2-(cyclopropylamino)-6-{[(1r,2s,3r,4r)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino}pyrimidin-4(3h)-oneHuman6006
IRAK4IRAKTKL4ztmD5-(1,3-benzothiazol-2-yl)-2-(cyclopropylamino)-6-{[(1r,2s,3r,4r)-2,3-dihydroxy-4-(hydroxymethyl)cyclopentyl]amino}pyrimidin-4(3h)-oneHuman5999
IRAK4IRAKTKL4ztnAA5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-oneHuman5993
IRAK4IRAKTKL4ztnAB5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-oneHuman6007
IRAK4IRAKTKL4ztnBA5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-oneHuman6005
IRAK4IRAKTKL4ztnBB5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-oneHuman6001
IRAK4IRAKTKL4ztnCA5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-oneHuman6008
IRAK4IRAKTKL4ztnCB5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-oneHuman5991
IRAK4IRAKTKL4ztnDA5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-oneHuman5995
IRAK4IRAKTKL4ztnDB5-(1,3-benzothiazol-2-yl)-2-(morpholin-4-yl)-6-[(3r)-piperidin-3-ylamino]pyrimidin-4(3h)-oneHuman6002
IRAK4IRAKTKL5k72A~{n}4,~{n}4-dimethyl-~{n}1-[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]cyclohexane-1,4-diamineHuman8720
IRAK4IRAKTKL5k72B~{n}4,~{n}4-dimethyl-~{n}1-[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]cyclohexane-1,4-diamineHuman8711
IRAK4IRAKTKL5k72C~{n}4,~{n}4-dimethyl-~{n}1-[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]cyclohexane-1,4-diamineHuman8723
IRAK4IRAKTKL5k72D~{n}4,~{n}4-dimethyl-~{n}1-[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]cyclohexane-1,4-diamineHuman8721
IRAK4IRAKTKL5k75AA~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamineHuman8725
IRAK4IRAKTKL5k75AB~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamineHuman8727
IRAK4IRAKTKL5k75BA~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamineHuman8713
IRAK4IRAKTKL5k75BB~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamineHuman8717
IRAK4IRAKTKL5k75CA~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamineHuman8724
IRAK4IRAKTKL5k75CB~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamineHuman8710
IRAK4IRAKTKL5k75DA~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamineHuman8718
IRAK4IRAKTKL5k75DB~{n}1-(7,8-dihydro-6~{h}-cyclopenta[2,3]thieno[2,4-~{c}]pyrimidin-1-yl)-~{n}4,~{n}4-dimethyl-cyclohexane-1,4-diamineHuman8714
IRAK4IRAKTKL5k76AA~{n}-(4-morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman8712
IRAK4IRAKTKL5k76AB~{n}-(4-morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman8715
IRAK4IRAKTKL5k76BA~{n}-(4-morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman8709
IRAK4IRAKTKL5k76BB~{n}-(4-morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman8708
IRAK4IRAKTKL5k7gA(3~{a}~{s},7~{a}~{r})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-oneHuman8722
IRAK4IRAKTKL5k7gB(3~{a}~{s},7~{a}~{r})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-oneHuman8706
IRAK4IRAKTKL5k7gC(3~{a}~{s},7~{a}~{r})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-oneHuman8707
IRAK4IRAKTKL5k7gD(3~{a}~{s},7~{a}~{r})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-oneHuman8716
IRAK4IRAKTKL5k7iA(3~{a}~{r},7~{a}~{s})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-oneHuman9521
IRAK4IRAKTKL5k7iB(3~{a}~{r},7~{a}~{s})-1-methyl-5-[4-[[5-(oxan-4-yl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]amino]cyclohexyl]-3,3~{a},4,6,7,7~{a}-hexahydropyrrolo[3,2-c]pyridin-2-oneHuman9520
IRAK4IRAKTKL5kx7A-Human6956
IRAK4IRAKTKL5kx7B~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-6-(1-methylpyrazol-4-yl)pyridine-2-carboxamideHuman6957
IRAK4IRAKTKL5kx8A~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-5-piperazin-1-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman6958
IRAK4IRAKTKL5kx8B~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-5-piperazin-1-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman6959
IRAK4IRAKTKL5kx8C~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-5-piperazin-1-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman6960
IRAK4IRAKTKL5kx8D~{n}-(3-aminocarbonyl-1-methyl-pyrazol-4-yl)-5-piperazin-1-yl-pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman6961
IRAK4IRAKTKL5t1sA5-[3-(3,5-dimethylphenyl)-4-[4-(methylamino)butyl]quinolin-6-yl]pyridin-3-olHuman7568
IRAK4IRAKTKL5t1sB5-[3-(3,5-dimethylphenyl)-4-[4-(methylamino)butyl]quinolin-6-yl]pyridin-3-olHuman7566
IRAK4IRAKTKL5t1sC5-[3-(3,5-dimethylphenyl)-4-[4-(methylamino)butyl]quinolin-6-yl]pyridin-3-olHuman7561
IRAK4IRAKTKL5t1sD5-[3-(3,5-dimethylphenyl)-4-[4-(methylamino)butyl]quinolin-6-yl]pyridin-3-olHuman7563
IRAK4IRAKTKL5t1tA~{n},~{n}-dimethyl-4-(6-nitroquinazolin-4-yl)oxy-cyclohexan-1-amineHuman7567
IRAK4IRAKTKL5t1tB~{n},~{n}-dimethyl-4-(6-nitroquinazolin-4-yl)oxy-cyclohexan-1-amineHuman7562
IRAK4IRAKTKL5t1tC~{n},~{n}-dimethyl-4-(6-nitroquinazolin-4-yl)oxy-cyclohexan-1-amineHuman7564
IRAK4IRAKTKL5t1tD~{n},~{n}-dimethyl-4-(6-nitroquinazolin-4-yl)oxy-cyclohexan-1-amineHuman7565
IRAK4IRAKTKL5uiqAA2-[(propan-2-yl)oxy]benzamideHuman7596
IRAK4IRAKTKL5uiqAB2-[(propan-2-yl)oxy]benzamideHuman7612
IRAK4IRAKTKL5uiqBA2-[(propan-2-yl)oxy]benzamideHuman7617
IRAK4IRAKTKL5uiqBB2-[(propan-2-yl)oxy]benzamideHuman7619
IRAK4IRAKTKL5uiqCA2-[(propan-2-yl)oxy]benzamideHuman7616
IRAK4IRAKTKL5uiqCB2-[(propan-2-yl)oxy]benzamideHuman7608
IRAK4IRAKTKL5uiqDA2-[(propan-2-yl)oxy]benzamideHuman7620
IRAK4IRAKTKL5uiqDB2-[(propan-2-yl)oxy]benzamideHuman7610
IRAK4IRAKTKL5uirAA5-(4-cyanophenyl)-3-[(propan-2-yl)oxy]naphthalene-2-carboxamideHuman7599
IRAK4IRAKTKL5uirAB5-(4-cyanophenyl)-3-[(propan-2-yl)oxy]naphthalene-2-carboxamideHuman7600
IRAK4IRAKTKL5uirBA5-(4-cyanophenyl)-3-[(propan-2-yl)oxy]naphthalene-2-carboxamideHuman7595
IRAK4IRAKTKL5uirBB5-(4-cyanophenyl)-3-[(propan-2-yl)oxy]naphthalene-2-carboxamideHuman7605
IRAK4IRAKTKL5uisAA4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamideHuman7604
IRAK4IRAKTKL5uisAB4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamideHuman7598
IRAK4IRAKTKL5uisBA4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamideHuman7601
IRAK4IRAKTKL5uisBB4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamideHuman7618
IRAK4IRAKTKL5uisCA4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamideHuman7611
IRAK4IRAKTKL5uisCB4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamideHuman7613
IRAK4IRAKTKL5uisDA4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamideHuman7602
IRAK4IRAKTKL5uisDB4-{[(3r)-piperidin-3-yl]oxy}-6-[(propan-2-yl)oxy]quinoline-7-carboxamideHuman7614
IRAK4IRAKTKL5uitA1-{[(2s)-5-oxopyrrolidin-2-yl]methoxy}-7-[(propan-2-yl)oxy]isoquinoline-6-carboxamideHuman7606
IRAK4IRAKTKL5uitB1-{[(2s)-5-oxopyrrolidin-2-yl]methoxy}-7-[(propan-2-yl)oxy]isoquinoline-6-carboxamideHuman7597
IRAK4IRAKTKL5uiuAA1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamideHuman7603
IRAK4IRAKTKL5uiuAB1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamideHuman7615
IRAK4IRAKTKL5uiuBA1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamideHuman7607
IRAK4IRAKTKL5uiuBB1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamideHuman7609
IRAK4IRAKTKL5w84A4-(benzylamino)-6-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]pyridine-3-carboxamideHuman8559
IRAK4IRAKTKL5w84B4-(benzylamino)-6-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]pyridine-3-carboxamideHuman8561
IRAK4IRAKTKL5w85A6-[(1,3-benzothiazol-6-yl)amino]-4-{[(2s)-1-hydroxy-3-phenylpropan-2-yl]amino}-n-methylpyridine-3-carboxamideHuman8560
IRAK4IRAKTKL5w85B6-[(1,3-benzothiazol-6-yl)amino]-4-{[(2s)-1-hydroxy-3-phenylpropan-2-yl]amino}-n-methylpyridine-3-carboxamideHuman8558
IRAK4IRAKTKL6eg9AA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman10906
IRAK4IRAKTKL6eg9AB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman10905
IRAK4IRAKTKL6eg9BA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman10909
IRAK4IRAKTKL6eg9BB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman10911
IRAK4IRAKTKL6egaAA3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}-n-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman10908
IRAK4IRAKTKL6egaAB3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}-n-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman10907
IRAK4IRAKTKL6egaBA3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}-n-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman10912
IRAK4IRAKTKL6egaBB3-{2-[(cyclopropanecarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}-n-{4-[(piperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman10910
IRAK4IRAKTKL6egdAAn-[2-methoxy-4-(morpholin-4-yl)phenyl]-2-(pyridin-3-yl)-1,3-thiazole-5-carboxamideHuman10895
IRAK4IRAKTKL6egdABn-[2-methoxy-4-(morpholin-4-yl)phenyl]-2-(pyridin-3-yl)-1,3-thiazole-5-carboxamideHuman10892
IRAK4IRAKTKL6egdDAn-[2-methoxy-4-(morpholin-4-yl)phenyl]-2-(pyridin-3-yl)-1,3-thiazole-5-carboxamideHuman10894
IRAK4IRAKTKL6egdDBn-[2-methoxy-4-(morpholin-4-yl)phenyl]-2-(pyridin-3-yl)-1,3-thiazole-5-carboxamideHuman10890
IRAK4IRAKTKL6egeAAn-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamideHuman10897
IRAK4IRAKTKL6egeABn-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamideHuman10891
IRAK4IRAKTKL6egeDAn-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamideHuman10896
IRAK4IRAKTKL6egeDBn-[2-methoxy-4-(morpholin-4-yl)phenyl]-6-(1h-pyrazol-5-yl)pyridine-2-carboxamideHuman10889
IRAK4IRAKTKL6egfBphosphoaminophosphonic acid-adenylate esterHuman10893
IRAK4IRAKTKL6f3dA4-[4-[[4-(dimethylamino)cyclohexyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]cyclohexane-1-carboxamideHuman9925
IRAK4IRAKTKL6f3dB4-[4-[[4-(dimethylamino)cyclohexyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]cyclohexane-1-carboxamideHuman9924
IRAK4IRAKTKL6f3eA2-[(3~{r})-12-(4-morpholin-4-ylcyclohexyl)oxy-7-thia-9,11-diazatricyclo[6.4.0.0^{2,6}]dodeca-1(8),2(6),9,11-tetraen-3-yl]ethanamideHuman9923
IRAK4IRAKTKL6f3eB2-[(3~{r})-12-(4-morpholin-4-ylcyclohexyl)oxy-7-thia-9,11-diazatricyclo[6.4.0.0^{2,6}]dodeca-1(8),2(6),9,11-tetraen-3-yl]ethanamideHuman9926
IRAK4IRAKTKL6f3gA~{n}4,~{n}4-dimethyl-~{n}1-(5-propan-2-ylpyrrolo[3,2-d]pyrimidin-4-yl)cyclohexane-1,4-diamineHuman9921
IRAK4IRAKTKL6f3gB~{n}4,~{n}4-dimethyl-~{n}1-(5-propan-2-ylpyrrolo[3,2-d]pyrimidin-4-yl)cyclohexane-1,4-diamineHuman9927
IRAK4IRAKTKL6f3iA(3~{r})-3-[4-[[4-(4-ethanoylpiperazin-1-yl)cyclohexyl]amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]butanamideHuman9928
IRAK4IRAKTKL6f3iB(3~{r})-3-[4-[[4-(4-ethanoylpiperazin-1-yl)cyclohexyl]amino]pyrrolo[2,1-f][1,2,4]triazin-5-yl]butanamideHuman9922
IRAK4IRAKTKL6lxyBn-[(2r)-2-fluoranyl-3-methyl-3-oxidanyl-butyl]-6-[(6-fluoranylpyrazolo[1,5-a]pyrimidin-5-yl)amino]-4-(propan-2-ylamino)pyridine-3-carboxamideHuman13163
IRAK4IRAKTKL6lxyDn-[(2r)-2-fluoranyl-3-methyl-3-oxidanyl-butyl]-6-[(6-fluoranylpyrazolo[1,5-a]pyrimidin-5-yl)amino]-4-(propan-2-ylamino)pyridine-3-carboxamideHuman13161
IRAK4IRAKTKL6lxyEn-[(2r)-2-fluoranyl-3-methyl-3-oxidanyl-butyl]-6-[(6-fluoranylpyrazolo[1,5-a]pyrimidin-5-yl)amino]-4-(propan-2-ylamino)pyridine-3-carboxamideHuman13162
IRAK4IRAKTKL6momAA6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amineHuman11742
IRAK4IRAKTKL6momAB6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amineHuman11740
IRAK4IRAKTKL6momBA6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amineHuman11743
IRAK4IRAKTKL6momBB6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amineHuman11745
IRAK4IRAKTKL6momCA6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amineHuman11738
IRAK4IRAKTKL6momCB6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amineHuman11739
IRAK4IRAKTKL6momDA6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amineHuman11744
IRAK4IRAKTKL6momDB6-[7-methoxy-6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-3-yl]-n-[(3r)-pyrrolidin-3-yl]pyridin-2-amineHuman11741
IRAK4IRAKTKL6n8gAAn-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamideHuman10796
IRAK4IRAKTKL6n8gABn-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamideHuman10795
IRAK4IRAKTKL6n8gBAn-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamideHuman10791
IRAK4IRAKTKL6n8gBBn-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamideHuman10790
IRAK4IRAKTKL6n8gCAn-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamideHuman10794
IRAK4IRAKTKL6n8gCBn-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamideHuman10793
IRAK4IRAKTKL6n8gDAn-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamideHuman10792
IRAK4IRAKTKL6n8gDBn-[2-(morpholin-4-yl)-6-(piperidin-1-yl)-1,3-benzoxazol-5-yl]-6-(1h-pyrrolo[2,3-b]pyridin-5-yl)pyridine-2-carboxamideHuman10789
IRAK4IRAKTKL6o8uAAn-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11113
IRAK4IRAKTKL6o8uABn-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11121
IRAK4IRAKTKL6o8uBAn-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11120
IRAK4IRAKTKL6o8uBBn-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11096
IRAK4IRAKTKL6o8uCAn-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11116
IRAK4IRAKTKL6o8uCBn-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11093
IRAK4IRAKTKL6o8uDAn-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11119
IRAK4IRAKTKL6o8uDBn-[2,2-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11103
IRAK4IRAKTKL6o94AAn-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11092
IRAK4IRAKTKL6o94ABn-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11091
IRAK4IRAKTKL6o94BAn-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11098
IRAK4IRAKTKL6o94BBn-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11117
IRAK4IRAKTKL6o94CAn-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11118
IRAK4IRAKTKL6o94CBn-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11095
IRAK4IRAKTKL6o94DAn-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11111
IRAK4IRAKTKL6o94DBn-{5-[4-(hydroxymethyl)piperidin-1-yl]-1-methyl-2-(morpholin-4-yl)-1h-benzimidazol-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11108
IRAK4IRAKTKL6o95AAn-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11104
IRAK4IRAKTKL6o95ABn-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11102
IRAK4IRAKTKL6o95BAn-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11090
IRAK4IRAKTKL6o95BBn-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11106
IRAK4IRAKTKL6o95CAn-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11110
IRAK4IRAKTKL6o95CBn-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11097
IRAK4IRAKTKL6o95DAn-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11105
IRAK4IRAKTKL6o95DBn-[(2r)-2-(hydroxymethyl)-2-methyl-6-(morpholin-4-yl)-2,3-dihydro-1-benzofuran-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11101
IRAK4IRAKTKL6o9dAAn-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11099
IRAK4IRAKTKL6o9dABn-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11109
IRAK4IRAKTKL6o9dBAn-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11107
IRAK4IRAKTKL6o9dBBn-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11094
IRAK4IRAKTKL6o9dCAn-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11115
IRAK4IRAKTKL6o9dCBn-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11112
IRAK4IRAKTKL6o9dDAn-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11100
IRAK4IRAKTKL6o9dDBn-{7-[4-(aminomethyl)piperidin-1-yl]quinolin-6-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11114
IRAK4IRAKTKL6rfiAAmethyl 4-[4-[(6-cyanoquinazolin-4-yl)amino]cyclohexyl]piperazine-1-carboxylateHuman11788
IRAK4IRAKTKL6rfiABmethyl 4-[4-[(6-cyanoquinazolin-4-yl)amino]cyclohexyl]piperazine-1-carboxylateHuman11787
IRAK4IRAKTKL6rfiBAmethyl 4-[4-[(6-cyanoquinazolin-4-yl)amino]cyclohexyl]piperazine-1-carboxylateHuman11790
IRAK4IRAKTKL6rfiBBmethyl 4-[4-[(6-cyanoquinazolin-4-yl)amino]cyclohexyl]piperazine-1-carboxylateHuman11791
IRAK4IRAKTKL6rfjAmethyl 4-[4-[[6-(cyanomethyl)-2-[(1-methylpyrazol-4-yl)amino]pyrido[3,2-d]pyrimidin-4-yl]amino]cyclohexyl]piperazine-1-carboxylateHuman11786
IRAK4IRAKTKL6rfjBmethyl 4-[4-[[6-(cyanomethyl)-2-[(1-methylpyrazol-4-yl)amino]pyrido[3,2-d]pyrimidin-4-yl]amino]cyclohexyl]piperazine-1-carboxylateHuman11789
IRAK4IRAKTKL6thwA7-fluoranyl-4-(1-methylcyclopropyl)oxy-~{n}-[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]-6-(2-methylpyrimidin-5-yl)pyrido[3,2-d]pyrimidin-2-amineHuman12950
IRAK4IRAKTKL6thwB7-fluoranyl-4-(1-methylcyclopropyl)oxy-~{n}-[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]-6-(2-methylpyrimidin-5-yl)pyrido[3,2-d]pyrimidin-2-amineHuman12956
IRAK4IRAKTKL6thxA2-[4-[(1-methylcyclopropyl)amino]-2-[(1-methylpyrazol-4-yl)amino]pyrido[3,2-d]pyrimidin-6-yl]ethanenitrileHuman12944
IRAK4IRAKTKL6thxB2-[4-[(1-methylcyclopropyl)amino]-2-[(1-methylpyrazol-4-yl)amino]pyrido[3,2-d]pyrimidin-6-yl]ethanenitrileHuman12953
IRAK4IRAKTKL6thzA7-fluoranyl-~{n}-[1-(2-methyl-2-azaspiro[3.3]heptan-6-yl)pyrazol-4-yl]-4-(1-methylcyclopropyl)oxy-6-(2-methylpyrimidin-5-yl)pyrido[3,2-d]pyrimidin-2-amineHuman12948
IRAK4IRAKTKL6thzB7-fluoranyl-~{n}-[1-(2-methyl-2-azaspiro[3.3]heptan-6-yl)pyrazol-4-yl]-4-(1-methylcyclopropyl)oxy-6-(2-methylpyrimidin-5-yl)pyrido[3,2-d]pyrimidin-2-amineHuman12951
IRAK4IRAKTKL6ti8AA~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamideHuman12947
IRAK4IRAKTKL6ti8AB~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamideHuman12954
IRAK4IRAKTKL6ti8BA~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamideHuman12949
IRAK4IRAKTKL6ti8BB~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamideHuman12952
IRAK4IRAKTKL6ti8CA~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamideHuman12945
IRAK4IRAKTKL6ti8CB~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamideHuman12946
IRAK4IRAKTKL6ti8DA~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamideHuman12957
IRAK4IRAKTKL6ti8DB~{n},~{n}-dimethyl-4-(1-methylcyclopropyl)oxy-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[3,2-d]pyrimidine-6-carboxamideHuman12942
IRAK4IRAKTKL6tiaA4-(1-methylcyclopropyl)oxy-~{n}-[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]-6-(1-methylpyrazol-4-yl)pyrido[3,2-d]pyrimidin-2-amineHuman12955
IRAK4IRAKTKL6tiaB4-(1-methylcyclopropyl)oxy-~{n}-[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]-6-(1-methylpyrazol-4-yl)pyrido[3,2-d]pyrimidin-2-amineHuman12943
IRAK4IRAKTKL6uyaAAn-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11810
IRAK4IRAKTKL6uyaABn-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11811
IRAK4IRAKTKL6uyaBAn-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11807
IRAK4IRAKTKL6uyaBBn-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11812
IRAK4IRAKTKL6uyaCAn-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11814
IRAK4IRAKTKL6uyaCBn-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11808
IRAK4IRAKTKL6uyaDAn-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11813
IRAK4IRAKTKL6uyaDBn-{2-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]-6-(morpholin-4-yl)-1-oxo-2,3-dihydro-1h-isoindol-5-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11809
IRAK4IRAKTKL6vqlA6-[(1,3-benzothiazol-6-yl)amino]-4-(cyclopropylamino)-n-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamideHuman12395
IRAK4IRAKTKL6vqlB6-[(1,3-benzothiazol-6-yl)amino]-4-(cyclopropylamino)-n-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamideHuman12394
IRAK4IRAKTKL6vqlC6-[(1,3-benzothiazol-6-yl)amino]-4-(cyclopropylamino)-n-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamideHuman12393
IRAK4IRAKTKL6vqlD6-[(1,3-benzothiazol-6-yl)amino]-4-(cyclopropylamino)-n-[(2r)-2-fluoro-3-hydroxy-3-methylbutyl]pyridine-3-carboxamideHuman12392
IRAK4IRAKTKL7c2vAA2-(2-methylpyridin-4-yl)-n-[2-morpholin-4-yl-5-[(3r)-3-oxidanylpyrrolidin-1-yl]-[1,3]oxazolo[4,5-b]pyridin-6-yl]-1,3-oxazole-4-carboxamideHuman12997
IRAK4IRAKTKL7c2vAB2-(2-methylpyridin-4-yl)-n-[2-morpholin-4-yl-5-[(3r)-3-oxidanylpyrrolidin-1-yl]-[1,3]oxazolo[4,5-b]pyridin-6-yl]-1,3-oxazole-4-carboxamideHuman13001
IRAK4IRAKTKL7c2vCA2-(2-methylpyridin-4-yl)-n-[2-morpholin-4-yl-5-[(3r)-3-oxidanylpyrrolidin-1-yl]-[1,3]oxazolo[4,5-b]pyridin-6-yl]-1,3-oxazole-4-carboxamideHuman12999
IRAK4IRAKTKL7c2vCB2-(2-methylpyridin-4-yl)-n-[2-morpholin-4-yl-5-[(3r)-3-oxidanylpyrrolidin-1-yl]-[1,3]oxazolo[4,5-b]pyridin-6-yl]-1,3-oxazole-4-carboxamideHuman13003
IRAK4IRAKTKL7c2wAA-Human12996
IRAK4IRAKTKL7c2wBA-Human12998
IRAK4IRAKTKL7c2wCA-Human13002
IRAK4IRAKTKL7c2wDA-Human13000
IRAK4IRAKTKL7qg1Amethyl 4-[4-[[6-(cyanomethyl)-2-[(1-methylpyrazol-4-yl)amino]-5-oxidanylidene-pyrido[4,3-d]pyrimidin-4-yl]amino]cyclohexyl]piperazine-1-carboxylateHuman14212
IRAK4IRAKTKL7qg2AA6-methyl-4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[4,3-d]pyrimidin-5-oneHuman14210
IRAK4IRAKTKL7qg2AB6-methyl-4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[4,3-d]pyrimidin-5-oneHuman14215
IRAK4IRAKTKL7qg3A6-[(2~{s})-2-fluoranylpropyl]-4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]pyrido[4,3-d]pyrimidin-5-oneHuman14213
IRAK4IRAKTKL7qg5AA4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-6-pyrimidin-5-yl-pyrido[4,3-d]pyrimidin-5-oneHuman14211
IRAK4IRAKTKL7qg5AB4-[(1-methylcyclopropyl)amino]-2-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-6-pyrimidin-5-yl-pyrido[4,3-d]pyrimidin-5-oneHuman14214
IRAK4IRAKTKL8atbAA~{n}-[6-ethoxy-2-[2-(4-methylpiperazin-1-yl)-2-oxidanylidene-ethyl]indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamideHuman15080
IRAK4IRAKTKL8atbAB~{n}-[6-ethoxy-2-[2-(4-methylpiperazin-1-yl)-2-oxidanylidene-ethyl]indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamideHuman15079
IRAK4IRAKTKL8atlAA~{n}-[6-methoxy-2-(2-morpholin-4-yl-2-oxidanylidene-ethyl)indazol-5-yl]-6-[(1~{r})-2,2,2-tris(fluoranyl)-1-oxidanyl-ethyl]pyridine-2-carboxamideHuman14964
IRAK4IRAKTKL8atlAB~{n}-[6-methoxy-2-(2-morpholin-4-yl-2-oxidanylidene-ethyl)indazol-5-yl]-6-[(1~{r})-2,2,2-tris(fluoranyl)-1-oxidanyl-ethyl]pyridine-2-carboxamideHuman14959
IRAK4IRAKTKL8atlBA~{n}-[6-methoxy-2-(2-morpholin-4-yl-2-oxidanylidene-ethyl)indazol-5-yl]-6-[(1~{r})-2,2,2-tris(fluoranyl)-1-oxidanyl-ethyl]pyridine-2-carboxamideHuman14961
IRAK4IRAKTKL8atlBB~{n}-[6-methoxy-2-(2-morpholin-4-yl-2-oxidanylidene-ethyl)indazol-5-yl]-6-[(1~{r})-2,2,2-tris(fluoranyl)-1-oxidanyl-ethyl]pyridine-2-carboxamideHuman14966
IRAK4IRAKTKL8atnAA~{n}-[3-methyl-2-(3-methyl-3-oxidanyl-butyl)-6-(2-oxidanylpropan-2-yl)benzimidazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamideHuman14965
IRAK4IRAKTKL8atnAB~{n}-[3-methyl-2-(3-methyl-3-oxidanyl-butyl)-6-(2-oxidanylpropan-2-yl)benzimidazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamideHuman14962
IRAK4IRAKTKL8br5AA~{n}-[2,3-dimethyl-6-(1~{h}-pyrazol-5-yl)benzimidazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamideHuman15187
IRAK4IRAKTKL8br5AB~{n}-[2,3-dimethyl-6-(1~{h}-pyrazol-5-yl)benzimidazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamideHuman15189
IRAK4IRAKTKL8br6AA~{n}-[6-methoxy-2-(2-methylsulfonylethyl)-1,3-dihydroindazol-5-yl]-6-(2-oxidanylpropan-2-yl)pyridine-2-carboxamideHuman15191
IRAK4IRAKTKL8br6AB~{n}-[6-methoxy-2-(2-methylsulfonylethyl)-1,3-dihydroindazol-5-yl]-6-(2-oxidanylpropan-2-yl)pyridine-2-carboxamideHuman15190
IRAK4IRAKTKL8br7A3-nitro-~{n}-[2-[2-oxidanylidene-2-[4-(phenylcarbonyl)piperazin-1-yl]ethyl]indazol-5-yl]benzamideHuman15188
IRAK4IRAKTKL8dksAA(1s,2s,3r,4r)-3-({2-[3-(pyrrolidine-1-carbonyl)anilino]thieno[3,2-d]pyrimidin-4-yl}amino)bicyclo[2.2.1]hept-5-ene-2-carboxamideHuman14316
IRAK4IRAKTKL8dksAB(1s,2s,3r,4r)-3-({2-[3-(pyrrolidine-1-carbonyl)anilino]thieno[3,2-d]pyrimidin-4-yl}amino)bicyclo[2.2.1]hept-5-ene-2-carboxamideHuman14315
IRAK4IRAKTKL8wtfAA1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamideHuman14960
IRAK4IRAKTKL8wtfAB1-{[(2s,3s,4s)-3-ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamideHuman14963
ITKTecTK1sm2AstaurosporineHuman74
ITKTecTK1sm2BstaurosporineHuman73
ITKTecTK1snuAstaurosporineHuman82
ITKTecTK1snuBstaurosporineHuman33
ITKTecTK1snxA-Human61
ITKTecTK1snxB-Human62
ITKTecTK3miyAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman46
ITKTecTK3miyBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman8
ITKTecTK3mj1A7-[(4-methylpiperazin-1-yl)methyl]-4-[(3-methyl-1h-pyrazol-5-yl)amino]-2-(tetrahydro-2h-pyran-4-yl)phthalazin-1(2h)-oneHuman27
ITKTecTK3mj2An-[5-({5-[(4-acetylpiperazin-1-yl)carbonyl]-4-methoxy-2-methylphenyl}sulfanyl)-1,3-thiazol-2-yl]-4-({[(1s)-1,2,2-trimethylpropyl]amino}methyl)benzamideHuman67
ITKTecTK3qgwAA3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamideHuman11
ITKTecTK3qgwAB3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamideHuman57
ITKTecTK3qgwBAn-(6-oxo-1,6-dihydro-3,4'-bipyridin-5-yl)benzamideHuman65
ITKTecTK3qgwBBn-(6-oxo-1,6-dihydro-3,4'-bipyridin-5-yl)benzamideHuman14
ITKTecTK3qgyAA3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamideHuman35
ITKTecTK3qgyAB3-[(8-phenylthieno[2,3-h]quinazolin-2-yl)amino]benzenesulfonamideHuman72
ITKTecTK3qgyBAn-{5-[2-(methylamino)pyrimidin-4-yl]-2-oxo-1,2-dihydropyridin-3-yl}-4-(piperidin-1-yl)benzamideHuman52
ITKTecTK3qgyBBn-{5-[2-(methylamino)pyrimidin-4-yl]-2-oxo-1,2-dihydropyridin-3-yl}-4-(piperidin-1-yl)benzamideHuman66
ITKTecTK3t9tAA(2z)-4-(dimethylamino)-n-{7-fluoro-4-[(2-methylphenyl)amino]imidazo[1,5-a]quinoxalin-8-yl}-n-methylbut-2-enamideHuman16
ITKTecTK3t9tAB(2z)-4-(dimethylamino)-n-{7-fluoro-4-[(2-methylphenyl)amino]imidazo[1,5-a]quinoxalin-8-yl}-n-methylbut-2-enamideHuman83
ITKTecTK3v5jA3-{4-[2-(morpholin-4-yl)ethoxy]-2-(4lambda~4~-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl}pentan-3-olHuman80
ITKTecTK3v5jB3-{4-[2-(morpholin-4-yl)ethoxy]-2-(4lambda~4~-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl}pentan-3-olHuman60
ITKTecTK3v5lA3-[3-(4-methoxyphenyl)-2-(1h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-olHuman30
ITKTecTK3v5lB3-[3-(4-methoxyphenyl)-2-(1h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-olHuman54
ITKTecTK3v5lC3-[3-(4-methoxyphenyl)-2-(1h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-olHuman26
ITKTecTK3v5lD3-[3-(4-methoxyphenyl)-2-(1h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-olHuman56
ITKTecTK3v8tAA3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-olHuman55
ITKTecTK3v8tAB3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-olHuman5
ITKTecTK3v8tBA3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-olHuman39
ITKTecTK3v8tBB3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-olHuman49
ITKTecTK3v8wA3-[2-(5-phenyl-2h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-olHuman43
ITKTecTK3v8wB3-[2-(5-phenyl-2h-thieno[3,2-c]pyrazol-3-yl)-1h-indol-6-yl]pentan-3-olHuman10
ITKTecTK4hctA3-{1-[(3r)-1-acryloylpiperidin-3-yl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-n-(3-tert-butylphenyl)benzamideHuman44
ITKTecTK4hcuA3-{4-amino-1-[(3r)-1-propanoylpiperidin-3-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-n-[4-(propan-2-yl)phenyl]benzamideHuman81
ITKTecTK4hcvA3-{4-amino-1-[(3s)-1-propanoylpiperidin-3-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-n-[4-(propan-2-yl)phenyl]benzamideHuman32
ITKTecTK4kioAA1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-oneHuman76
ITKTecTK4kioAB1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-oneHuman79
ITKTecTK4kioBA1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-oneHuman36
ITKTecTK4kioBB1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-oneHuman48
ITKTecTK4kioCA1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]propan-1-oneHuman75
ITKTecTK4kioCB1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]prop-2-en-1-oneHuman7
ITKTecTK4kioDA1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]propan-1-oneHuman6
ITKTecTK4kioDB1-[(3s)-3-{[4-(morpholin-4-ylmethyl)-6-([1,3]thiazolo[5,4-b]pyridin-2-ylamino)pyrimidin-2-yl]amino}pyrrolidin-1-yl]propan-1-oneHuman85
ITKTecTK4l7sAAtrans-4-({4-[difluoro(4-fluorophenyl)methyl]-6-[(5-methoxy[1,3]thiazolo[5,4-b]pyridin-2-yl)amino]pyrimidin-2-yl}amino)cyclohexanolHuman50
ITKTecTK4l7sABtrans-4-({4-[difluoro(4-fluorophenyl)methyl]-6-[(5-methoxy[1,3]thiazolo[5,4-b]pyridin-2-yl)amino]pyrimidin-2-yl}amino)cyclohexanolHuman64
ITKTecTK4l7sBAtrans-4-({4-[difluoro(4-fluorophenyl)methyl]-6-[(5-methoxy[1,3]thiazolo[5,4-b]pyridin-2-yl)amino]pyrimidin-2-yl}amino)cyclohexanolHuman37
ITKTecTK4l7sBBtrans-4-({4-[difluoro(4-fluorophenyl)methyl]-6-[(5-methoxy[1,3]thiazolo[5,4-b]pyridin-2-yl)amino]pyrimidin-2-yl}amino)cyclohexanolHuman25
ITKTecTK4m0yAA4-(carbamoylamino)-1-(naphthalen-1-yl)-1h-pyrazole-3-carboxamideHuman9
ITKTecTK4m0yAB4-(carbamoylamino)-1-(naphthalen-1-yl)-1h-pyrazole-3-carboxamideHuman70
ITKTecTK4m0zAA4-(carbamoylamino)-1-(7-methoxynaphthalen-1-yl)-1h-pyrazole-3-carboxamideHuman45
ITKTecTK4m0zAB4-(carbamoylamino)-1-(7-methoxynaphthalen-1-yl)-1h-pyrazole-3-carboxamideHuman47
ITKTecTK4m12AA-Human22
ITKTecTK4m12AB-Human51
ITKTecTK4m13AA-Human17
ITKTecTK4m13AB-Human15
ITKTecTK4m14A4-(carbamoylamino)-1-[7-(propan-2-yloxy)naphthalen-1-yl]-1h-pyrazole-3-carboxamideHuman58
ITKTecTK4m15Aadenosine-5'-diphosphateHuman31
ITKTecTK4mf0A(1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(pyridin-3-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamideHuman77
ITKTecTK4mf0B(1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(pyridin-3-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamideHuman28
ITKTecTK4mf1AA(1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(1h-pyrazol-4-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamideHuman41
ITKTecTK4mf1AB(1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(1h-pyrazol-4-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamideHuman34
ITKTecTK4mf1BA(1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(1h-pyrazol-4-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamideHuman12
ITKTecTK4mf1BB(1s,2s)-2-{4-[(dimethylamino)methyl]phenyl}-n-[6-(1h-pyrazol-4-yl)-1,3-benzothiazol-2-yl]cyclopropanecarboxamideHuman18
ITKTecTK4pp9An-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-2h-indazole-3-carboxamideHuman20
ITKTecTK4pp9Bn-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-2h-indazole-3-carboxamideHuman40
ITKTecTK4ppaAn-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman38
ITKTecTK4ppaBn-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman21
ITKTecTK4ppbAn-{1-[(1s)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman29
ITKTecTK4ppbBn-{1-[(1s)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman84
ITKTecTK4ppcAAn-{1-[(1r)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman53
ITKTecTK4ppcABn-{1-[(1r)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman13
ITKTecTK4ppcBAn-{1-[(1r)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman78
ITKTecTK4ppcBBn-{1-[(1r)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman63
ITKTecTK4pqnAAn-{1-[(1s)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6,6-dimethyl-4,5,6,7-tetrahydro-1h-indazole-3-carboxamideHuman42
ITKTecTK4pqnABn-{1-[(1s)-3-(dimethylamino)-1-phenylpropyl]-1h-pyrazol-4-yl}-6,6-dimethyl-4,5,6,7-tetrahydro-1h-indazole-3-carboxamideHuman19
ITKTecTK4qd6AAtrans-4-({6-[(5-phenyl-1h-pyrazol-3-yl)amino]-4-(phenylsulfonyl)pyridin-2-yl}amino)cyclohexanolHuman23
ITKTecTK4qd6ABtrans-4-({6-[(5-phenyl-1h-pyrazol-3-yl)amino]-4-(phenylsulfonyl)pyridin-2-yl}amino)cyclohexanolHuman59
ITKTecTK4qd6BAtrans-4-({6-[(5-phenyl-1h-pyrazol-3-yl)amino]-4-(phenylsulfonyl)pyridin-2-yl}amino)cyclohexanolHuman24
ITKTecTK4qd6BBtrans-4-({6-[(5-phenyl-1h-pyrazol-3-yl)amino]-4-(phenylsulfonyl)pyridin-2-yl}amino)cyclohexanolHuman71
ITKTecTK4rfmAA(4as,5ar)-n-{1-[(r)-[(2r)-1,1-dioxidotetrahydro-2h-thiopyran-2-yl](phenyl)methyl]-1h-pyrazol-4-yl}-5,5-difluoro-5a-methyl-1,4,4a,5,5a,6-hexahydrocyclopropa[f]indazole-3-carboxamideHuman68
ITKTecTK4rfmAB(4as,5ar)-n-{1-[(r)-[(2r)-1,1-dioxidotetrahydro-2h-thiopyran-2-yl](phenyl)methyl]-1h-pyrazol-4-yl}-5,5-difluoro-5a-methyl-1,4,4a,5,5a,6-hexahydrocyclopropa[f]indazole-3-carboxamideHuman69
Jak1 (JAK1)JakATK8ewyA-Mouse14664
JAK1JakATK3eygAA3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHuman1445
JAK1JakATK3eygAB3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHuman1453
JAK1JakATK3eyhA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman1462
JAK1JakATK4e4lAA1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1450
JAK1JakATK4e4lAB1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1488
JAK1JakATK4e4lBA1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1464
JAK1JakATK4e4lBB1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1466
JAK1JakATK4e4lDA1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1455
JAK1JakATK4e4lDB1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1468
JAK1JakATK4e4lEA-Human1469
JAK1JakATK4e4lEB-Human1484
JAK1JakATK4e4nAtert-butyl [(1r,3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)cyclopentyl]carbamateHuman1443
JAK1JakATK4e4nBtert-butyl [(1r,3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)cyclopentyl]carbamateHuman1454
JAK1JakATK4e5wAA[4-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl][(2s)-1-(propan-2-yl)pyrrolidin-2-yl]methanoneHuman1452
JAK1JakATK4e5wAB[4-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl][(2s)-1-(propan-2-yl)pyrrolidin-2-yl]methanoneHuman1473
JAK1JakATK4e5wBA[4-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl][(2s)-1-(propan-2-yl)pyrrolidin-2-yl]methanoneHuman1447
JAK1JakATK4e5wBB[4-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl][(2s)-1-(propan-2-yl)pyrrolidin-2-yl]methanoneHuman1477
JAK1JakATK4ehzAA2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1482
JAK1JakATK4ehzAB2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1463
JAK1JakATK4ehzBA2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1448
JAK1JakATK4ehzBB2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1481
JAK1JakATK4ehzCA2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1470
JAK1JakATK4ehzCB2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1476
JAK1JakATK4ehzDA2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1485
JAK1JakATK4ehzDB2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman1451
JAK1JakATK4ei4A(1r,3r)-3-(2-methylimidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(8h)-yl)cyclohexanolHuman1480
JAK1JakATK4ei4B(1r,3r)-3-(2-methylimidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(8h)-yl)cyclohexanolHuman1483
JAK1JakATK4fk6AAn-({1-[(1r,2r,4s)-bicyclo[2.2.1]hept-2-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2-yl}methyl)methanesulfonamideHuman1465
JAK1JakATK4fk6ABn-({1-[(1r,2r,4s)-bicyclo[2.2.1]hept-2-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2-yl}methyl)methanesulfonamideHuman1460
JAK1JakATK4fk6BAn-({1-[(1r,2r,4s)-bicyclo[2.2.1]hept-2-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2-yl}methyl)methanesulfonamideHuman1487
JAK1JakATK4fk6BBn-({1-[(1r,2r,4s)-bicyclo[2.2.1]hept-2-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-2-yl}methyl)methanesulfonamideHuman1459
JAK1JakATK4i5cAA3-oxo-3-[(3r)-3-(pyrrolo[2,3-b][1,2,3]triazolo[4,5-d]pyridin-1(6h)-yl)piperidin-1-yl]propanenitrileHuman1446
JAK1JakATK4i5cAB3-oxo-3-[(3r)-3-(pyrrolo[2,3-b][1,2,3]triazolo[4,5-d]pyridin-1(6h)-yl)piperidin-1-yl]propanenitrileHuman1471
JAK1JakATK4i5cBA3-oxo-3-[(3r)-3-(pyrrolo[2,3-b][1,2,3]triazolo[4,5-d]pyridin-1(6h)-yl)piperidin-1-yl]propanenitrileHuman1467
JAK1JakATK4i5cBB3-oxo-3-[(3r)-3-(pyrrolo[2,3-b][1,2,3]triazolo[4,5-d]pyridin-1(6h)-yl)piperidin-1-yl]propanenitrileHuman1458
JAK1JakATK4ivbAAtrans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrileHuman1486
JAK1JakATK4ivbABtrans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrileHuman1479
JAK1JakATK4ivbBAtrans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrileHuman1472
JAK1JakATK4ivbBBtrans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrileHuman1444
JAK1JakATK4ivcA(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)acetonitrileHuman1461
JAK1JakATK4ivcB(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)acetonitrileHuman1456
JAK1JakATK4ivdAA3-(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)propanenitrileHuman1489
JAK1JakATK4ivdAB3-(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)propanenitrileHuman1474
JAK1JakATK4ivdBA3-(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)propanenitrileHuman1490
JAK1JakATK4ivdBB3-(trans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexyl)propanenitrileHuman1457
JAK1JakATK4k6zA(1r,2s)-2-{[8-oxo-2-(1h-pyrazol-4-yl)-5,8-dihydropyrido[3,4-d]pyrimidin-4-yl]amino}cyclopentanecarbonitrileHuman1478
JAK1JakATK4k77A4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-8(7h)-oneHuman1449
JAK1JakATK4k77B4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-8(7h)-oneHuman1475
JAK1JakATK5e1eAA6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amineHuman6250
JAK1JakATK5e1eAB6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amineHuman6248
JAK1JakATK5e1eBA6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amineHuman6249
JAK1JakATK5e1eBB6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amineHuman6251
JAK1JakATK5hx8AA4-[(4-aminocyclohexyl)amino]-3-(1h-benzimidazol-2-yl)-1h-pyridin-2-oneHuman6441
JAK1JakATK5hx8AB4-[(4-aminocyclohexyl)amino]-3-(1h-benzimidazol-2-yl)-1h-pyridin-2-oneHuman6438
JAK1JakATK5hx8BA4-[(4-aminocyclohexyl)amino]-3-(1h-benzimidazol-2-yl)-1h-pyridin-2-oneHuman6440
JAK1JakATK5hx8BB4-[(4-aminocyclohexyl)amino]-3-(1h-benzimidazol-2-yl)-1h-pyridin-2-oneHuman6439
JAK1JakATK5khwAadenosine-5'-diphosphateHuman7164
JAK1JakATK5khwBadenosine-5'-diphosphateHuman7165
JAK1JakATK5khxAA~{n}-[3-[methyl(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl]methanesulfonamideHuman7167
JAK1JakATK5khxAB~{n}-[3-[methyl(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl]methanesulfonamideHuman7166
JAK1JakATK5wo4AA3-[(4-chloro-3-methoxyphenyl)amino]-1-[(3r,4s)-4-cyanooxan-3-yl]-1h-pyrazole-4-carboxamideHuman8702
JAK1JakATK5wo4AB3-[(4-chloro-3-methoxyphenyl)amino]-1-[(3r,4s)-4-cyanooxan-3-yl]-1h-pyrazole-4-carboxamideHuman8705
JAK1JakATK5wo4BA3-[(4-chloro-3-methoxyphenyl)amino]-1-[(3r,4s)-4-cyanooxan-3-yl]-1h-pyrazole-4-carboxamideHuman8704
JAK1JakATK5wo4BB3-[(4-chloro-3-methoxyphenyl)amino]-1-[(3r,4s)-4-cyanooxan-3-yl]-1h-pyrazole-4-carboxamideHuman8703
JAK1JakATK6aahAA4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10392
JAK1JakATK6aahAB4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10396
JAK1JakATK6aahBA4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10394
JAK1JakATK6aahBB4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10395
JAK1JakATK6bbuAAn-{cis-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamideHuman9497
JAK1JakATK6bbuABn-{cis-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamideHuman9496
JAK1JakATK6c7yAAadenosine-5'-diphosphateHuman9866
JAK1JakATK6c7yABadenosine-5'-diphosphateHuman9867
JAK1JakATK6dbnAA[(1s)-2,2-difluorocyclopropyl][(1r,5s)-3-{2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octan-8-yl]methanoneHuman10393
JAK1JakATK6dbnAB[(1s)-2,2-difluorocyclopropyl][(1r,5s)-3-{2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octan-8-yl]methanoneHuman10391
JAK1JakATK6elrAA[3-[[5-methyl-2-[[3-(4-methylpiperazin-1-yl)-5-methylsulfonyl-phenyl]amino]pyrimidin-4-yl]amino]phenyl]methanolHuman10618
JAK1JakATK6elrAB[3-[[5-methyl-2-[[3-(4-methylpiperazin-1-yl)-5-methylsulfonyl-phenyl]amino]pyrimidin-4-yl]amino]phenyl]methanolHuman10616
JAK1JakATK6elrBA[3-[[5-methyl-2-[[3-(4-methylpiperazin-1-yl)-5-methylsulfonyl-phenyl]amino]pyrimidin-4-yl]amino]phenyl]methanolHuman10619
JAK1JakATK6elrBB[3-[[5-methyl-2-[[3-(4-methylpiperazin-1-yl)-5-methylsulfonyl-phenyl]amino]pyrimidin-4-yl]amino]phenyl]methanolHuman10617
JAK1JakATK6gghAA~{n}-[5-methyl-4-[7-[[(2~{r})-2-(4-methylpiperazin-1-yl)propanoyl]amino]-1~{h}-indol-3-yl]pyrimidin-2-yl]cyclopropanecarboxamideHuman11087
JAK1JakATK6gghAB~{n}-[5-methyl-4-[7-[[(2~{r})-2-(4-methylpiperazin-1-yl)propanoyl]amino]-1~{h}-indol-3-yl]pyrimidin-2-yl]cyclopropanecarboxamideHuman11088
JAK1JakATK6gghBA~{n}-[5-methyl-4-[7-[[(2~{r})-2-(4-methylpiperazin-1-yl)propanoyl]amino]-1~{h}-indol-3-yl]pyrimidin-2-yl]cyclopropanecarboxamideHuman11089
JAK1JakATK6gghBB~{n}-[5-methyl-4-[7-[[(2~{r})-2-(4-methylpiperazin-1-yl)propanoyl]amino]-1~{h}-indol-3-yl]pyrimidin-2-yl]cyclopropanecarboxamideHuman11086
JAK1JakATK6hzuAA2-[4-[8-oxidanylidene-2-[(~{e})-(2-oxidanylidenepyridin-3-ylidene)amino]-7~{h}-purin-9-yl]cyclohexyl]ethanenitrileHuman11764
JAK1JakATK6hzuAB2-[4-[8-oxidanylidene-2-[(~{e})-(2-oxidanylidenepyridin-3-ylidene)amino]-7~{h}-purin-9-yl]cyclohexyl]ethanenitrileHuman11762
JAK1JakATK6hzuBA2-[4-[8-oxidanylidene-2-[(~{e})-(2-oxidanylidenepyridin-3-ylidene)amino]-7~{h}-purin-9-yl]cyclohexyl]ethanenitrileHuman11765
JAK1JakATK6hzuBB2-[4-[8-oxidanylidene-2-[(~{e})-(2-oxidanylidenepyridin-3-ylidene)amino]-7~{h}-purin-9-yl]cyclohexyl]ethanenitrileHuman11763
JAK1JakATK6n77AAn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11024
JAK1JakATK6n77ABn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11021
JAK1JakATK6n77ACn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11029
JAK1JakATK6n77BAn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11030
JAK1JakATK6n77BBn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11018
JAK1JakATK6n77BCn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11034
JAK1JakATK6n78AAn-{3-[5-chloro-2-(difluoromethoxy)phenyl]-1-methyl-1h-pyrazol-4-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11019
JAK1JakATK6n78ABn-{3-[5-chloro-2-(difluoromethoxy)phenyl]-1-methyl-1h-pyrazol-4-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11022
JAK1JakATK6n79An-{5-[5-chloro-2-(difluoromethoxy)phenyl]-1h-pyrazol-4-yl}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11031
JAK1JakATK6n7aAAn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-2-methyl-2h-pyrazolo[4,3-c]pyridine-7-carboxamideHuman11017
JAK1JakATK6n7aABn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-2-methyl-2h-pyrazolo[4,3-c]pyridine-7-carboxamideHuman11028
JAK1JakATK6n7aBAn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-2-methyl-2h-pyrazolo[4,3-c]pyridine-7-carboxamideHuman11015
JAK1JakATK6n7aBBn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-2-methyl-2h-pyrazolo[4,3-c]pyridine-7-carboxamideHuman11026
JAK1JakATK6n7bAn-[3-(5-chloro-2-methoxyphenyl)-1-methyl-1h-pyrazol-4-yl]-1h-pyrazolo[4,3-c]pyridine-7-carboxamideHuman11020
JAK1JakATK6n7cAAn-[5-(3-methoxynaphthalen-2-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11016
JAK1JakATK6n7cABn-[5-(3-methoxynaphthalen-2-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11027
JAK1JakATK6n7cBAn-[5-(3-methoxynaphthalen-2-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11033
JAK1JakATK6n7cBBn-[5-(3-methoxynaphthalen-2-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11023
JAK1JakATK6n7dAAn-[5-(6-methoxy-1h-indazol-5-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11032
JAK1JakATK6n7dABn-[5-(6-methoxy-1h-indazol-5-yl)-1h-pyrazol-4-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman11025
JAK1JakATK6rsbA1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[[4-(cyclohexen-1-yl)phenyl]methyl]-3-fluoranyl-piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12482
JAK1JakATK6rsbB1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[[4-(cyclohexen-1-yl)phenyl]methyl]-3-fluoranyl-piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12479
JAK1JakATK6rscAA1-[4-(cyanomethyl)-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12477
JAK1JakATK6rscAB1-[4-(cyanomethyl)-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12468
JAK1JakATK6rscBA1-[4-(cyanomethyl)-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12474
JAK1JakATK6rscBB1-[4-(cyanomethyl)-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12469
JAK1JakATK6rsdAA1-[4-(cyanomethyl)-1-[(3-oxidanyl-4-phenyl-phenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12472
JAK1JakATK6rsdAB1-[4-(cyanomethyl)-1-[(3-oxidanyl-4-phenyl-phenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12478
JAK1JakATK6rsdBA1-[4-(cyanomethyl)-1-[(3-oxidanyl-4-phenyl-phenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12466
JAK1JakATK6rsdBB1-[4-(cyanomethyl)-1-[(3-oxidanyl-4-phenyl-phenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12475
JAK1JakATK6rseAAmethyl ~{n}-[4-aminocarbonyl-1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[(4-ethenyl-2-fluoranyl-5-oxidanyl-phenyl)methyl]-3-fluoranyl-piperidin-4-yl]pyrazol-3-yl]carbamateHuman12481
JAK1JakATK6rseABmethyl ~{n}-[4-aminocarbonyl-1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[(4-ethenyl-2-fluoranyl-5-oxidanyl-phenyl)methyl]-3-fluoranyl-piperidin-4-yl]pyrazol-3-yl]carbamateHuman12476
JAK1JakATK6rseBAmethyl ~{n}-[4-aminocarbonyl-1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[(4-ethenyl-2-fluoranyl-5-oxidanyl-phenyl)methyl]-3-fluoranyl-piperidin-4-yl]pyrazol-3-yl]carbamateHuman12465
JAK1JakATK6rseBBmethyl ~{n}-[4-aminocarbonyl-1-[(3~{r},4~{r})-4-(cyanomethyl)-1-[(4-ethenyl-2-fluoranyl-5-oxidanyl-phenyl)methyl]-3-fluoranyl-piperidin-4-yl]pyrazol-3-yl]carbamateHuman12471
JAK1JakATK6rshAA1-[(3~{r},4~{r})-4-(cyanomethyl)-3-fluoranyl-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12470
JAK1JakATK6rshAB1-[(3~{r},4~{r})-4-(cyanomethyl)-3-fluoranyl-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12473
JAK1JakATK6rshBA1-[(3~{r},4~{r})-4-(cyanomethyl)-3-fluoranyl-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12467
JAK1JakATK6rshBB1-[(3~{r},4~{r})-4-(cyanomethyl)-3-fluoranyl-1-[(4-phenylphenyl)methyl]piperidin-4-yl]-3-(cyclopropylcarbonylamino)pyrazole-4-carboxamideHuman12480
JAK1JakATK6sm8AA2-chloranyl-6-[(3~{s})-3-[(1~{s})-2-cyano-1-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethyl]pyrrolidin-1-yl]benzenecarbonitrileHuman12248
JAK1JakATK6sm8AB2-chloranyl-6-[(3~{s})-3-[(1~{s})-2-cyano-1-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethyl]pyrrolidin-1-yl]benzenecarbonitrileHuman12250
JAK1JakATK6sm8BA2-chloranyl-6-[(3~{s})-3-[(1~{s})-2-cyano-1-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethyl]pyrrolidin-1-yl]benzenecarbonitrileHuman12245
JAK1JakATK6sm8BB2-chloranyl-6-[(3~{s})-3-[(1~{s})-2-cyano-1-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]ethyl]pyrrolidin-1-yl]benzenecarbonitrileHuman12249
JAK1JakATK6smbAA~{n}-[3-[2-[(3-methoxy-1-methyl-pyrazol-4-yl)amino]-5-methyl-pyrimidin-4-yl]-1~{h}-indol-7-yl]-2-methyl-pyridine-3-carboxamideHuman12246
JAK1JakATK6smbAB~{n}-[3-[2-[(3-methoxy-1-methyl-pyrazol-4-yl)amino]-5-methyl-pyrimidin-4-yl]-1~{h}-indol-7-yl]-2-methyl-pyridine-3-carboxamideHuman12247
JAK1JakATK6smbBA~{n}-[3-[2-[(3-methoxy-1-methyl-pyrazol-4-yl)amino]-5-methyl-pyrimidin-4-yl]-1~{h}-indol-7-yl]-2-methyl-pyridine-3-carboxamideHuman12244
JAK1JakATK6smbBB~{n}-[3-[2-[(3-methoxy-1-methyl-pyrazol-4-yl)amino]-5-methyl-pyrimidin-4-yl]-1~{h}-indol-7-yl]-2-methyl-pyridine-3-carboxamideHuman12243
JAK1JakATK6tpeA2-[4-(3-methyl-6-oxidanylidene-1,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]ethanenitrileHuman12364
JAK1JakATK6tpeB2-[4-(3-methyl-6-oxidanylidene-1,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]ethanenitrileHuman12368
JAK1JakATK6tpfAA(1~{s})-2,2-bis(fluoranyl)-~{n}-[4-(3-methyl-6-oxidanylidene-2,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]cyclopropane-1-carboxamideHuman12366
JAK1JakATK6tpfAB(1~{s})-2,2-bis(fluoranyl)-~{n}-[4-(3-methyl-6-oxidanylidene-2,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]cyclopropane-1-carboxamideHuman12365
JAK1JakATK6tpfBA(1~{s})-2,2-bis(fluoranyl)-~{n}-[4-(3-methyl-6-oxidanylidene-2,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]cyclopropane-1-carboxamideHuman12363
JAK1JakATK6tpfBB(1~{s})-2,2-bis(fluoranyl)-~{n}-[4-(3-methyl-6-oxidanylidene-2,7-dihydropyrazolo[3,4-b]pyridin-4-yl)cyclohexyl]cyclopropane-1-carboxamideHuman12367
JAK1JakATK6w8lAn-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropanecarboxamideHuman12133
JAK1-bJakBTK4l00AA-Human1421
JAK1-bJakBTK4l00AB-Human1420
JAK1-bJakBTK4l00BA-Human1422
JAK1-bJakBTK4l00BB-Human1423
JAK1-bJakBTK4l01AA-Human1424
JAK1-bJakBTK4l01AB-Human1418
JAK1-bJakBTK4l01BA-Human1417
JAK1-bJakBTK4l01BB-Human1419
Jak2 (JAK2)JakATK4gl9A2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouse6933
Jak2 (JAK2)JakATK4gl9B2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouse6936
Jak2 (JAK2)JakATK4gl9C2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouse6934
Jak2 (JAK2)JakATK4gl9D2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouse6935
JAK2JakATK2b7aA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman3708
JAK2JakATK2b7aB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman3728
JAK2JakATK2w1iA4-[(2-{4-[(cyclopropylcarbamoyl)amino]-1h-pyrazol-3-yl}-1h-benzimidazol-6-yl)methyl]morpholin-4-iumHuman3652
JAK2JakATK2w1iB-Human3648
JAK2JakATK2xa4AA5-chloro-n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(5-methyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman3664
JAK2JakATK2xa4AB5-chloro-n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(5-methyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman3623
JAK2JakATK2xa4BA5-chloro-n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(5-methyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman3628
JAK2JakATK2xa4BB5-chloro-n2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(5-methyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman3707
JAK2JakATK3e62AA5-bromo-1h-indazol-3-amineHuman3665
JAK2JakATK3e62AB5-bromo-1h-indazol-3-amineHuman3630
JAK2JakATK3e63AA5-phenyl-1h-indazol-3-amineHuman3675
JAK2JakATK3e63AB5-phenyl-1h-indazol-3-amineHuman3711
JAK2JakATK3e64AA4-(3-amino-1h-indazol-5-yl)-n-tert-butylbenzenesulfonamideHuman3646
JAK2JakATK3e64AB4-(3-amino-1h-indazol-5-yl)-n-tert-butylbenzenesulfonamideHuman3653
JAK2JakATK3fupA3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHuman3721
JAK2JakATK3fupB3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHuman3654
JAK2JakATK3io7A(3s)-1-[6-(2-aminopyrazolo[1,5-a]pyrimidin-3-yl)pyrimidin-4-yl]-n,n-diethylpiperidine-3-carboxamideHuman3636
JAK2JakATK3iokAA3-(6-{[(1s)-1-(4-fluorophenyl)ethyl]amino}pyrimidin-4-yl)pyrazolo[1,5-a]pyrimidin-2-amineHuman3694
JAK2JakATK3iokAB3-(6-{[(1s)-1-(4-fluorophenyl)ethyl]amino}pyrimidin-4-yl)pyrazolo[1,5-a]pyrimidin-2-amineHuman3718
JAK2JakATK3jy9AA(3s)-3-(4-hydroxyphenyl)-1,5-dihydro-1,5,12-triazabenzo[4,5]cycloocta[1,2,3-cd]inden-4(3h)-oneHuman3668
JAK2JakATK3jy9AB(3s)-3-(4-hydroxyphenyl)-1,5-dihydro-1,5,12-triazabenzo[4,5]cycloocta[1,2,3-cd]inden-4(3h)-oneHuman3716
JAK2JakATK3kckAA3-chloro-4-(4h-3,4,7-triazadibenzo[cd,f]azulen-6-yl)phenolHuman3683
JAK2JakATK3kckAB3-chloro-4-(4h-3,4,7-triazadibenzo[cd,f]azulen-6-yl)phenolHuman3722
JAK2JakATK3krrAA8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-(1-piperidin-4-yl-1h-pyrazol-4-yl)quinoxalineHuman3643
JAK2JakATK3krrAB8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-(1-piperidin-4-yl-1h-pyrazol-4-yl)quinoxalineHuman3695
JAK2JakATK3lpbAAn-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]benzenesulfonamideHuman3672
JAK2JakATK3lpbABn-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]benzenesulfonamideHuman3698
JAK2JakATK3lpbBAn-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]benzenesulfonamideHuman3635
JAK2JakATK3lpbBBn-methyl-4-[3-(3,4,5-trimethoxyphenyl)quinoxalin-5-yl]benzenesulfonamideHuman3681
JAK2JakATK3q32A2-(2,6-difluoro-4-methoxyphenyl)-1-(4-{4-[(3-methyl-1h-pyrazol-5-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}piperazin-1-yl)ethanoneHuman3700
JAK2JakATK3q32B2-(2,6-difluoro-4-methoxyphenyl)-1-(4-{4-[(3-methyl-1h-pyrazol-5-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl}piperazin-1-yl)ethanoneHuman3639
JAK2JakATK3rvgA1-(cyclohexylamino)-7-(1-methyl-1h-pyrazol-4-yl)-5h-pyrido[4,3-b]indole-4-carboxamideHuman3638
JAK2JakATK3tjcA4-amino-n-methyl-2-[4-(morpholin-4-yl)phenyl]thieno[3,2-c]pyridine-7-carboxamideHuman3685
JAK2JakATK3tjcB4-amino-n-methyl-2-[4-(morpholin-4-yl)phenyl]thieno[3,2-c]pyridine-7-carboxamideHuman3688
JAK2JakATK3tjdA4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-n-methylthieno[3,2-c]pyridine-7-carboxamideHuman3677
JAK2JakATK3tjdB4-amino-2-[4-(tert-butylsulfamoyl)phenyl]-n-methylthieno[3,2-c]pyridine-7-carboxamideHuman3626
JAK2JakATK3ugcAA5-{[6-(acetylamino)pyrimidin-4-yl]oxy}-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-2,3-dihydro-1h-indole-1-carboxamideHuman3632
JAK2JakATK3ugcAB5-{[6-(acetylamino)pyrimidin-4-yl]oxy}-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-2,3-dihydro-1h-indole-1-carboxamideHuman3651
JAK2JakATK3zmmAA5-fluoro-4-[(1s)-1-(5-fluoropyrimidin-2-yl)ethoxy]-n-(5-methyl-1h-pyrazol-3-yl)-6-morpholino-pyrimidin-2-amineHuman3674
JAK2JakATK3zmmAB5-fluoro-4-[(1s)-1-(5-fluoropyrimidin-2-yl)ethoxy]-n-(5-methyl-1h-pyrazol-3-yl)-6-morpholino-pyrimidin-2-amineHuman3667
JAK2JakATK3zmmBA5-fluoro-4-[(1s)-1-(5-fluoropyrimidin-2-yl)ethoxy]-n-(5-methyl-1h-pyrazol-3-yl)-6-morpholino-pyrimidin-2-amineHuman3709
JAK2JakATK3zmmBB5-fluoro-4-[(1s)-1-(5-fluoropyrimidin-2-yl)ethoxy]-n-(5-methyl-1h-pyrazol-3-yl)-6-morpholino-pyrimidin-2-amineHuman3678
JAK2JakATK4aqcAA8-(4-methylsulfonylphenyl)-n-(4-morpholin-4-ylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amineHuman3720
JAK2JakATK4aqcAB8-(4-methylsulfonylphenyl)-n-(4-morpholin-4-ylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amineHuman3696
JAK2JakATK4aqcBA8-(4-methylsulfonylphenyl)-n-(4-morpholin-4-ylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amineHuman3679
JAK2JakATK4aqcBB8-(4-methylsulfonylphenyl)-n-(4-morpholin-4-ylphenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-amineHuman3676
JAK2JakATK4bbeAn-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]ethanamideHuman3670
JAK2JakATK4bbeBn-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]ethanamideHuman3727
JAK2JakATK4bbeCn-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]ethanamideHuman3649
JAK2JakATK4bbeDn-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]ethanamideHuman3726
JAK2JakATK4bbfA(2r)-n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]pyrrolidine-2-carboxamideHuman3723
JAK2JakATK4bbfB(2r)-n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]pyrrolidine-2-carboxamideHuman3717
JAK2JakATK4bbfC(2r)-n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]pyrrolidine-2-carboxamideHuman3644
JAK2JakATK4bbfD(2r)-n-[4-[2-[(4-morpholin-4-ylphenyl)amino]pyrimidin-4-yl]phenyl]pyrrolidine-2-carboxamideHuman3663
JAK2JakATK4c61An2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-7-methyl-n4-(1-methylimidazol-4-yl)thieno[3,2-d]pyrimidine-2,4-diamineHuman3661
JAK2JakATK4c61Bn2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-7-methyl-n4-(1-methylimidazol-4-yl)thieno[3,2-d]pyrimidine-2,4-diamineHuman3645
JAK2JakATK4c62An2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(1-methylimidazol-4-yl)-6-morpholino-1,3,5-triazine-2,4-diamineHuman3655
JAK2JakATK4c62Bn2-[(1s)-1-(5-fluoropyrimidin-2-yl)ethyl]-n4-(1-methylimidazol-4-yl)-6-morpholino-1,3,5-triazine-2,4-diamineHuman3625
JAK2JakATK4d0wAA5-(2-aminopyrimidin-4-yl)-2-(5-chloro-2-methylphenyl)-1h-pyrrole-3-carboxamideHuman3666
JAK2JakATK4d0wAB5-(2-aminopyrimidin-4-yl)-2-(5-chloro-2-methylphenyl)-1h-pyrrole-3-carboxamideHuman3650
JAK2JakATK4d0xAA5-(2-aminopyrimidin-4-yl)-2-[2-chloro-5-(trifluoromethyl)phenyl]-1h-pyrrole-3-carboxamideHuman3699
JAK2JakATK4d0xAB5-(2-aminopyrimidin-4-yl)-2-[2-chloro-5-(trifluoromethyl)phenyl]-1h-pyrrole-3-carboxamideHuman3642
JAK2JakATK4d1sAA2-(5-chloro-2-methylphenyl)-1-methyl-5-(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1h-pyrrole-3-carboxamideHuman3634
JAK2JakATK4d1sAB2-(5-chloro-2-methylphenyl)-1-methyl-5-(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1h-pyrrole-3-carboxamideHuman3627
JAK2JakATK4e4mA1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman3713
JAK2JakATK4e4mB1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman3712
JAK2JakATK4e4mD1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman3669
JAK2JakATK4e4mE1-[4-methyl-1-(methylsulfonyl)piperidin-4-yl]-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman3637
JAK2JakATK4e6dAA3-[(3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl]-3-oxopropanenitrileHuman3689
JAK2JakATK4e6dAB3-[(3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl]-3-oxopropanenitrileHuman3656
JAK2JakATK4e6dBA3-[(3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl]-3-oxopropanenitrileHuman3631
JAK2JakATK4e6dBB3-[(3r)-3-(imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl)piperidin-1-yl]-3-oxopropanenitrileHuman3647
JAK2JakATK4e6qA1-(1-benzylpiperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman3624
JAK2JakATK4e6qB1-(1-benzylpiperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman3671
JAK2JakATK4f08A1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman3662
JAK2JakATK4f08B1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman3719
JAK2JakATK4f09A2-methyl-1-(piperidin-4-yl)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridineHuman3622
JAK2JakATK4gfmAA2,6-dichloro-n-(2-oxo-2,5-dihydropyridin-4-yl)benzamideHuman3680
JAK2JakATK4gfmAB2,6-dichloro-n-(2-oxo-2,5-dihydropyridin-4-yl)benzamideHuman3705
JAK2JakATK4gmyA2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman3684
JAK2JakATK4hgeAAn-[1-(3-chlorophenyl)-3-methyl-1h-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman3703
JAK2JakATK4hgeABn-[1-(3-chlorophenyl)-3-methyl-1h-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman3658
JAK2JakATK4hgeBAn-[1-(3-chlorophenyl)-3-methyl-1h-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman3706
JAK2JakATK4hgeBBn-[1-(3-chlorophenyl)-3-methyl-1h-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman3715
JAK2JakATK4ivaAAtrans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrileHuman3673
JAK2JakATK4ivaABtrans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrileHuman3725
JAK2JakATK4ivaACtrans-4-{2-[(1r)-1-hydroxyethyl]imidazo[4,5-d]pyrrolo[2,3-b]pyridin-1(6h)-yl}cyclohexanecarbonitrileHuman3714
JAK2JakATK4ji9An-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamideHuman3692
JAK2JakATK4ji9Bn-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamideHuman3724
JAK2JakATK4jiaAA5-(4-methoxyphenyl)-n-[4-(4-methylpiperazin-1-yl)phenyl][1,2,4]triazolo[1,5-a]pyridin-2-amineHuman3691
JAK2JakATK4jiaAB5-(4-methoxyphenyl)-n-[4-(4-methylpiperazin-1-yl)phenyl][1,2,4]triazolo[1,5-a]pyridin-2-amineHuman3640
JAK2JakATK4p7eAn-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamideHuman3682
JAK2JakATK4p7eBn-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamideHuman3701
JAK2JakATK4ytcAAn~3~-phenyl-1-[6-(phenylamino)pyrimidin-4-yl]-1h-1,2,4-triazole-3,5-diamineHuman3633
JAK2JakATK4ytcABn~3~-phenyl-1-[6-(phenylamino)pyrimidin-4-yl]-1h-1,2,4-triazole-3,5-diamineHuman3687
JAK2JakATK4ytfAAn~2~-[2-(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl]-n-(2,2,2-trifluoroethyl)-l-alaninamideHuman3690
JAK2JakATK4ytfABn~2~-[2-(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl]-n-(2,2,2-trifluoroethyl)-l-alaninamideHuman3693
JAK2JakATK4ythAAn~2~-[2-(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl]-2-methyl-n-(2,2,2-trifluoroethyl)-d-alaninamideHuman3710
JAK2JakATK4ythABn~2~-[2-(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)-5-fluoropyrimidin-4-yl]-2-methyl-n-(2,2,2-trifluoroethyl)-d-alaninamideHuman3702
JAK2JakATK4ytiAA(2r)-2-methyl-2-[[2-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl]amino]-n-[2,2,2-tris(fluoranyl)ethyl]butanamideHuman3641
JAK2JakATK4ytiAB(2r)-2-methyl-2-[[2-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-4-yl]amino]-n-[2,2,2-tris(fluoranyl)ethyl]butanamideHuman3657
JAK2JakATK4zimAA3-(3,4-dichlorophenyl)-6-(morpholin-4-ylcarbonyl)-9h-carbazole-1-carboxamideHuman3704
JAK2JakATK4zimAB3-(3,4-dichlorophenyl)-6-(morpholin-4-ylcarbonyl)-9h-carbazole-1-carboxamideHuman3659
JAK2JakATK4zimBA3-(3,4-dichlorophenyl)-6-(morpholin-4-ylcarbonyl)-9h-carbazole-1-carboxamideHuman3660
JAK2JakATK4zimBB3-(3,4-dichlorophenyl)-6-(morpholin-4-ylcarbonyl)-9h-carbazole-1-carboxamideHuman3697
JAK2JakATK5aepAA1-(5-chloro-2-methylphenyl)-4-(pyrrolo[2,1-f][1,2,4]triazin-4-yl)-1h-pyrrole-2-carboxamideHuman3629
JAK2JakATK5aepAB1-(5-chloro-2-methylphenyl)-4-(pyrrolo[2,1-f][1,2,4]triazin-4-yl)-1h-pyrrole-2-carboxamideHuman3686
JAK2JakATK5cf4An,n-dicyclopropyl-6-ethyl-4-[(3-methoxypropyl)amino]-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5980
JAK2JakATK5cf4Bn,n-dicyclopropyl-6-ethyl-4-[(3-methoxypropyl)amino]-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5982
JAK2JakATK5cf5An,n-dicyclopropyl-4-[(4,5-dimethyl-1,3-thiazol-2-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5984
JAK2JakATK5cf5Bn,n-dicyclopropyl-4-[(4,5-dimethyl-1,3-thiazol-2-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5976
JAK2JakATK5cf6An,n-dicyclopropyl-6-[(2s)-2,3-dihydroxypropyl]-1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5979
JAK2JakATK5cf6Bn,n-dicyclopropyl-6-[(2s)-2,3-dihydroxypropyl]-1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5977
JAK2JakATK5cf8AAn,n-dicyclopropyl-4-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5978
JAK2JakATK5cf8ABn,n-dicyclopropyl-4-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5981
JAK2JakATK5cf8BAn,n-dicyclopropyl-4-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5985
JAK2JakATK5cf8BBn,n-dicyclopropyl-4-[(1,5-dimethyl-1h-pyrazol-3-yl)amino]-6-ethyl-1-methyl-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridine-7-carboxamideHuman5983
JAK2JakATK5hezAn-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamideHuman7254
JAK2JakATK5hezBn-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamideHuman7255
JAK2JakATK5hezCn-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamideHuman7253
JAK2JakATK5hezDn-tert-butyl-3-[(5-methyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]benzenesulfonamideHuman7252
JAK2JakATK5l3aAA~{n}-(1~{h}-indazol-4-yl)methanesulfonamideHuman6561
JAK2JakATK5l3aAB~{n}-(1~{h}-indazol-4-yl)methanesulfonamideHuman6560
JAK2JakATK5tq3AA4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-3-ethylphenolHuman7359
JAK2JakATK5tq3AB4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-3-ethylphenolHuman7356
JAK2JakATK5tq3BA4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-3-ethylphenolHuman7360
JAK2JakATK5tq3BB4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-3-ethylphenolHuman7352
JAK2JakATK5tq4A6-(2-ethyl-4-hydroxyphenyl)-1h-indazole-3-carboxamideHuman7351
JAK2JakATK5tq5A6-(2-ethyl-4-hydroxyphenyl)-n-(6-methylpyridin-3-yl)-1h-indazole-3-carboxamideHuman7358
JAK2JakATK5tq6A{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}(pyrrolidin-1-yl)methanoneHuman7354
JAK2JakATK5tq6B{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}(pyrrolidin-1-yl)methanoneHuman7361
JAK2JakATK5tq7A{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}[(3r)-3-(phenylsulfonyl)pyrrolidin-1-yl]methanoneHuman7355
JAK2JakATK5tq7B{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}[(3r)-3-(phenylsulfonyl)pyrrolidin-1-yl]methanoneHuman7353
JAK2JakATK5tq8A{2-[6-(2-ethyl-5-fluoro-4-hydroxyphenyl)-2h-indazol-3-yl]-3,4,6,7-tetrahydro-5h-imidazo[4,5-c]pyridin-5-yl}[5-(piperidin-1-yl)pyrazin-2-yl]methanoneHuman7357
JAK2JakATK5usyAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8101
JAK2JakATK5usyAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8102
JAK2JakATK5usyBA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8103
JAK2JakATK5usyBB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8104
JAK2JakATK5wevAAn-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamideHuman8377
JAK2JakATK5wevABn-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamideHuman8376
JAK2JakATK6aajA4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10515
JAK2JakATK6aajB4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10514
JAK2JakATK6bbvAn-{cis-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]cyclobutyl}propane-1-sulfonamideHuman9504
JAK2JakATK6drwAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman10512
JAK2JakATK6drwAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman10513
JAK2JakATK6tpdA3-methyl-4-phenyl-2,7-dihydropyrazolo[3,4-b]pyridin-6-oneHuman12350
JAK2JakATK6vglA(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13223
JAK2JakATK6vglB(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13222
JAK2JakATK6vglC(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13221
JAK2JakATK6vglD(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13220
JAK2JakATK6vn8AbaricitinibHuman13291
JAK2JakATK6vn8BbaricitinibHuman13301
JAK2JakATK6vnbA(3s)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13298
JAK2JakATK6vncA(3r)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13359
JAK2JakATK6vncB(3r)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13348
JAK2JakATK6vneAn-tert-butyl-3-{[5-methyl-2-({4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}amino)pyrimidin-4-yl]amino}benzenesulfonamideHuman13296
JAK2JakATK6vneBn-tert-butyl-3-{[5-methyl-2-({4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}amino)pyrimidin-4-yl]amino}benzenesulfonamideHuman13302
JAK2JakATK6vnfAAn~4~-[1-(tert-butylsulfonyl)-2,3-dihydro-1h-indol-6-yl]-n~2~-[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]-5-methylpyrimidine-2,4-diamineHuman13347
JAK2JakATK6vnfABn~4~-[1-(tert-butylsulfonyl)-2,3-dihydro-1h-indol-6-yl]-n~2~-[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]-5-methylpyrimidine-2,4-diamineHuman13357
JAK2JakATK6vnfBAn~4~-[1-(tert-butylsulfonyl)-2,3-dihydro-1h-indol-6-yl]-n~2~-[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]-5-methylpyrimidine-2,4-diamineHuman13346
JAK2JakATK6vnfBBn~4~-[1-(tert-butylsulfonyl)-2,3-dihydro-1h-indol-6-yl]-n~2~-[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]-5-methylpyrimidine-2,4-diamineHuman13352
JAK2JakATK6vngAn-{2-fluoro-5-[(2-{[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]phenyl}-2-methylpropane-2-sulfonamideHuman13358
JAK2JakATK6vngBn-{2-fluoro-5-[(2-{[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]phenyl}-2-methylpropane-2-sulfonamideHuman13341
JAK2JakATK6vnhAn-{5-[(2-{[3,5-difluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]-2-fluorophenyl}-2-methylpropane-2-sulfonamideHuman13344
JAK2JakATK6vnhBn-{5-[(2-{[3,5-difluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]-2-fluorophenyl}-2-methylpropane-2-sulfonamideHuman13342
JAK2JakATK6vniA2-{5-[(2-{[3,5-difluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-5-methylpyrimidin-4-yl)amino]-2-fluorophenyl}-1lambda~6~,2-thiazolidine-1,1-dioneHuman13294
JAK2JakATK6vnjAA3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13340
JAK2JakATK6vnjBA3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13355
JAK2JakATK6vnkA(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13293
JAK2JakATK6vnkB(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13295
JAK2JakATK6vnkC(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13304
JAK2JakATK6vnkD(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13292
JAK2JakATK6vnlA4-[[4-[[3-(~{tert}-butylsulfonylamino)-4-chloranyl-phenyl]amino]-5-methyl-pyrimidin-2-yl]amino]-2-fluoranyl-~{n}-(1-methylpiperidin-4-yl)benzamideHuman13303
JAK2JakATK6vnlB4-[[4-[[3-(~{tert}-butylsulfonylamino)-4-chloranyl-phenyl]amino]-5-methyl-pyrimidin-2-yl]amino]-2-fluoranyl-~{n}-(1-methylpiperidin-4-yl)benzamideHuman13299
JAK2JakATK6vnlC4-[[4-[[3-(~{tert}-butylsulfonylamino)-4-chloranyl-phenyl]amino]-5-methyl-pyrimidin-2-yl]amino]-2-fluoranyl-~{n}-(1-methylpiperidin-4-yl)benzamideHuman13300
JAK2JakATK6vnlD4-[[4-[[3-(~{tert}-butylsulfonylamino)-4-chloranyl-phenyl]amino]-5-methyl-pyrimidin-2-yl]amino]-2-fluoranyl-~{n}-(1-methylpiperidin-4-yl)benzamideHuman13297
JAK2JakATK6vnmA4-[1-(but-3-en-1-yl)-1h-pyrazol-4-yl]-n-[4-(piperidin-4-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-2-amineHuman13354
JAK2JakATK6vnmB4-[1-(but-3-en-1-yl)-1h-pyrazol-4-yl]-n-[4-(piperidin-4-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-2-amineHuman13351
JAK2JakATK6vs3A(3r)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13349
JAK2JakATK6vs3B(3r)-3-cyclopentyl-3-[4-(2-{[4-(piperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13345
JAK2JakATK6vsnA(3s)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13353
JAK2JakATK6vsnB(3s)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13356
JAK2JakATK6vsnC(3s)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13350
JAK2JakATK6vsnD(3s)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13343
JAK2JakATK6wtnAA(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13538
JAK2JakATK6wtnAB(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13540
JAK2JakATK6wtoAAbaricitinibHuman13536
JAK2JakATK6wtoABbaricitinibHuman13539
JAK2JakATK6wtpAAtert-butyl 4-[(4-{1-[3-(cyanomethyl)-1-(ethylsulfonyl)azetidin-3-yl]-1h-pyrazol-4-yl}-7h-pyrrolo[2,3-d]pyrimidin-2-yl)amino]benzoateHuman13541
JAK2JakATK6wtpABtert-butyl 4-[(4-{1-[3-(cyanomethyl)-1-(ethylsulfonyl)azetidin-3-yl]-1h-pyrazol-4-yl}-7h-pyrrolo[2,3-d]pyrimidin-2-yl)amino]benzoateHuman13542
JAK2JakATK6wtqAAn-methyl-4-{[4-(1-propyl-1h-pyrazol-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-2-yl]amino}benzamideHuman13535
JAK2JakATK6wtqABn-methyl-4-{[4-(1-propyl-1h-pyrazol-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-2-yl]amino}benzamideHuman13537
JAK2JakATK6x8eAA[3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrileHuman13154
JAK2JakATK6x8eAB[3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrileHuman13152
JAK2JakATK6x8eBA[3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrileHuman13155
JAK2JakATK6x8eBB[3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrileHuman13153
JAK2JakATK7ll4AA{1-(ethylsulfonyl)-3-[4-(2-{[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]azetidin-3-yl}acetonitrileHuman14035
JAK2JakATK7ll4AB{1-(ethylsulfonyl)-3-[4-(2-{[3-fluoro-4-(1-methylpiperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]azetidin-3-yl}acetonitrileHuman14037
JAK2JakATK7ll5AA{1-(ethylsulfonyl)-3-[4-(2-{[4-(1-methylpiperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]azetidin-3-yl}acetonitrileHuman14036
JAK2JakATK7ll5AB{1-(ethylsulfonyl)-3-[4-(2-{[4-(1-methylpiperidin-4-yl)phenyl]amino}-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]azetidin-3-yl}acetonitrileHuman14038
JAK2JakATK7q7iAA4-[8-methoxy-2-[(1-methylpyrazol-4-yl)amino]quinazolin-6-yl]phenolHuman14085
JAK2JakATK7q7iAB4-[8-methoxy-2-[(1-methylpyrazol-4-yl)amino]quinazolin-6-yl]phenolHuman14088
JAK2JakATK7q7kAA4-(2-azanyl-8-methoxy-quinazolin-6-yl)phenolHuman14091
JAK2JakATK7q7kAB4-(2-azanyl-8-methoxy-quinazolin-6-yl)phenolHuman14086
JAK2JakATK7q7lAA4-[2-azanyl-8-[[(2~{s})-1-oxidanylpropan-2-yl]amino]quinazolin-6-yl]-5-ethyl-2-fluoranyl-phenolHuman14092
JAK2JakATK7q7lAB4-[2-azanyl-8-[[(2~{s})-1-oxidanylpropan-2-yl]amino]quinazolin-6-yl]-5-ethyl-2-fluoranyl-phenolHuman14090
JAK2JakATK7q7wAA4-[2-[5-(dimethylamino)pentylamino]-8-[[(2~{s})-1-oxidanylpropan-2-yl]amino]quinazolin-6-yl]-5-ethyl-2-fluoranyl-phenolHuman14087
JAK2JakATK7q7wAB4-[2-[5-(dimethylamino)pentylamino]-8-[[(2~{s})-1-oxidanylpropan-2-yl]amino]quinazolin-6-yl]-5-ethyl-2-fluoranyl-phenolHuman14089
JAK2JakATK7reeAA[3-(4-{2-[3,5-difluoro-4-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)anilino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}-1h-pyrazol-1-yl)-1-(ethanesulfonyl)azetidin-3-yl]acetonitrileHuman13855
JAK2JakATK7reeAB[3-(4-{2-[3,5-difluoro-4-(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)anilino]-7h-pyrrolo[2,3-d]pyrimidin-4-yl}-1h-pyrazol-1-yl)-1-(ethanesulfonyl)azetidin-3-yl]acetonitrileHuman13856
JAK2JakATK7rn6AA5-{[6-(acetylamino)pyrimidin-4-yl]oxy}-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-2,3-dihydro-1h-indole-1-carboxamideHuman13956
JAK2JakATK7rn6AB5-{[6-(acetylamino)pyrimidin-4-yl]oxy}-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-2,3-dihydro-1h-indole-1-carboxamideHuman13955
JAK2JakATK7teuAA3-{(4s)-2-[(cyclopropanecarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}-4-methylbenzamideHuman14806
JAK2JakATK7teuAB3-{(4s)-2-[(cyclopropanecarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}-4-methylbenzamideHuman14811
JAK2JakATK7uywAA2-(2,6-difluorophenyl)-4-[4-(pyrrolidine-1-carbonyl)anilino]-5h-pyrrolo[3,4-b]pyridin-5-oneHuman14333
JAK2JakATK7uywAB2-(2,6-difluorophenyl)-4-[4-(pyrrolidine-1-carbonyl)anilino]-5h-pyrrolo[3,4-b]pyridin-5-oneHuman14334
JAK2JakATK8bm2AA3-[(4-chloranyl-2-fluoranyl-phenyl)methyl]-2-methyl-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)-8-(morpholin-4-ylmethyl)imidazo[1,2-b]pyridazin-6-amineHuman15043
JAK2JakATK8bm2AB3-[(4-chloranyl-2-fluoranyl-phenyl)methyl]-2-methyl-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)-8-(morpholin-4-ylmethyl)imidazo[1,2-b]pyridazin-6-amineHuman15035
JAK2JakATK8bpvAA11-(2-pyrrolidin-1-yl-ethoxy)-14,19-dioxa-5,7,26-triaza-tetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaeneHuman15040
JAK2JakATK8bpvAB11-(2-pyrrolidin-1-yl-ethoxy)-14,19-dioxa-5,7,26-triaza-tetracyclo[19.3.1.1(2,6).1(8,12)]heptacosa-1(25),2(26),3,5,8,10,12(27),16,21,23-decaeneHuman15036
JAK2JakATK8bpwAAlestaurtinibHuman15044
JAK2JakATK8bpwABlestaurtinibHuman15039
JAK2JakATK8bx6AAcerdulatinibHuman15033
JAK2JakATK8bx6ABcerdulatinibHuman15042
JAK2JakATK8bx9AAilginatinibHuman15038
JAK2JakATK8bx9ABilginatinibHuman15034
JAK2JakATK8bxcAAitacitinibHuman15037
JAK2JakATK8bxcABitacitinibHuman15041
JAK2JakATK8bxhAAmomelotinibHuman15032
JAK2JakATK8bxhABmomelotinibHuman15045
JAK2JakATK8g6zAA(3r)-3-cyclopentyl-3-[(4m)-4-{5-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-1h-pyrazol-1-yl]propanenitrileHuman14808
JAK2JakATK8g6zAB(3r)-3-cyclopentyl-3-[(4m)-4-{5-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-1h-pyrazol-1-yl]propanenitrileHuman14810
JAK2JakATK8g8oAA[1-{5-methyl-2-[(3-methyl-1,2-thiazol-5-yl)amino]pyrimidin-4-yl}-3-(4-methylpiperazin-1-yl)azetidin-3-yl]acetonitrileHuman14807
JAK2JakATK8g8oAB[1-{5-methyl-2-[(3-methyl-1,2-thiazol-5-yl)amino]pyrimidin-4-yl}-3-(4-methylpiperazin-1-yl)azetidin-3-yl]acetonitrileHuman14809
JAK2JakATK8g8xAA3-cyclopropyl-1-{5-methyl-2-[(3-methyl-1,2-thiazol-5-yl)amino]pyrimidin-4-yl}azetidin-3-olHuman14804
JAK2JakATK8g8xAB3-cyclopropyl-1-{5-methyl-2-[(3-methyl-1,2-thiazol-5-yl)amino]pyrimidin-4-yl}azetidin-3-olHuman14805
JAK2-bJakBTK4fvpA-Human1222
JAK2-bJakBTK4fvqAadenosine-5'-triphosphateHuman1224
JAK2-bJakBTK4fvrAadenosine-5'-triphosphateHuman1223
JAK2-bJakBTK5i4nAAadenosine-5'-triphosphateHuman6525
JAK2-bJakBTK5i4nABadenosine-5'-triphosphateHuman6524
JAK2-bJakBTK5uszAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8048
JAK2-bJakBTK5uszAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8043
JAK2-bJakBTK5ut0AA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman8041
JAK2-bJakBTK5ut0AB1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman8047
JAK2-bJakBTK5ut1AA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman8046
JAK2-bJakBTK5ut1AB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman8049
JAK2-bJakBTK5ut2AA2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamideHuman8040
JAK2-bJakBTK5ut2AB2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamideHuman8039
JAK2-bJakBTK5ut3A5-phenyl-2-ureidothiophene-3-carboxamideHuman8044
JAK2-bJakBTK5ut4A8-[3,5-difluoro-4-(morpholin-4-ylmethyl)phenyl]-2-(1-piperidin-4-yl-1h-pyrazol-4-yl)quinoxalineHuman8038
JAK2-bJakBTK5ut5AAn-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamideHuman8042
JAK2-bJakBTK5ut5ABn-(5-{4-[(1,1-dioxidothiomorpholin-4-yl)methyl]phenyl}[1,2,4]triazolo[1,5-a]pyridin-2-yl)cyclopropanecarboxamideHuman8037
JAK2-bJakBTK5ut6AA4-({4-amino-6-[3-(hydroxymethyl)-1h-pyrazol-1-yl]pyrimidin-2-yl}amino)benzonitrileHuman8036
JAK2-bJakBTK5ut6AB4-({4-amino-6-[3-(hydroxymethyl)-1h-pyrazol-1-yl]pyrimidin-2-yl}amino)benzonitrileHuman8045
JAK2-bJakBTK5wijA4-{[6-(cyclohexylmethoxy)-7h-purin-2-yl]amino}-n,n-diethylbenzamideHuman10388
JAK2-bJakBTK5wikB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman10387
JAK2-bJakBTK5wilA5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman10379
JAK2-bJakBTK5wimA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10385
JAK2-bJakBTK5winA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman10378
JAK2-bJakBTK6brwAA4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman10382
JAK2-bJakBTK6brwAB4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman10377
JAK2-bJakBTK6bs0AA4-(5-aminopyrazin-2-yl)-1h-pyrrolo[2,3-b]pyridin-6-amineHuman10380
JAK2-bJakBTK6bs0AB4-(5-aminopyrazin-2-yl)-1h-pyrrolo[2,3-b]pyridin-6-amineHuman10381
JAK2-bJakBTK6bssAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman10386
JAK2-bJakBTK6d2iA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10967
JAK2-bJakBTK6d2iB1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10966
JAK2-bJakBTK6g3cAA2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-oneHuman10978
JAK2-bJakBTK6g3cAB2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-oneHuman10976
JAK2-bJakBTK6g3cBA2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-oneHuman10977
JAK2-bJakBTK6g3cBB2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7,7-trimethyl-8-(3-methylbutyl)pteridin-6-oneHuman10975
JAK2-bJakBTK6m9hAA4-({4-amino-6-[4-(2-hydroxyethyl)-1h-imidazol-1-yl]pyrimidin-2-yl}amino)benzonitrileHuman10384
JAK2-bJakBTK6m9hAB4-({4-amino-6-[4-(2-hydroxyethyl)-1h-imidazol-1-yl]pyrimidin-2-yl}amino)benzonitrileHuman10383
JAK2-bJakBTK6oavA5-amino-3-[(4-cyanophenyl)amino]-n-phenyl-1h-1,2,4-triazole-1-carboxamideHuman12099
JAK2-bJakBTK6obbA5-amino-n-phenyl-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carboxamideHuman12097
JAK2-bJakBTK6obfA[4-({5-amino-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenoxy]acetic acidHuman12098
JAK2-bJakBTK6oblA[4-({5-amino-3-[(4-cyanophenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenoxy]acetic acidHuman12101
JAK2-bJakBTK6occA2-[4-({5-amino-3-[(4-sulfamoylphenyl)amino]-1h-1,2,4-triazole-1-carbonyl}amino)phenyl]-1,3-oxazole-4-carboxylic acidHuman12100
JAK3JakATK1yvjAA1,2,3,4-tetrahydrogen-staurosporineHuman460
JAK3JakATK1yvjAB1,2,3,4-tetrahydrogen-staurosporineHuman451
JAK3JakATK3lxkA3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHuman436
JAK3JakATK3lxlAA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman434
JAK3JakATK3lxlAB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman443
JAK3JakATK3pjcA3-(1h-indol-3-yl)-4-[2-(4-oxopiperidin-1-yl)-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrrole-2,5-dioneHuman444
JAK3JakATK3zc6AAn-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman442
JAK3JakATK3zc6ABn-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman461
JAK3JakATK3zc6BAn-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman449
JAK3JakATK3zc6BBn-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman447
JAK3JakATK3zc6CAn-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman433
JAK3JakATK3zc6CBn-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman445
JAK3JakATK3zc6DAn-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman446
JAK3JakATK3zc6DBn-[(2r)-1-(3-cyanoazetidin-1-yl)-1-oxidanylidene-propan-2-yl]-2-(6-fluoranyl-1-methyl-indazol-3-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman459
JAK3JakATK3zepAA2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman448
JAK3JakATK3zepAB2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman456
JAK3JakATK3zepBA2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman430
JAK3JakATK3zepBB2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman437
JAK3JakATK3zepCA2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman439
JAK3JakATK3zepCB2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman462
JAK3JakATK3zepDA2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman454
JAK3JakATK3zepDB2-[[(3r)-3-acetamido-2,3-dihydro-1h-inden-5-yl]oxy]-n-[(1s)-1-cyclopropylethyl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman457
JAK3JakATK4hvdA2-cyclopropyl-n-[(2s)-3,3-dimethylbutan-2-yl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman431
JAK3JakATK4hvgA2-cyclopropyl-n-[(2s)-3-hydroxy-3-methylbutan-2-yl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman450
JAK3JakATK4hvhA2-cyclopropyl-n-[(2r)-3-hydroxy-3-methylbutan-2-yl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman441
JAK3JakATK4hviA2-cyclopropyl-n-[(2r)-1-oxo-1-(piperidin-1-yl)propan-2-yl]-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman438
JAK3JakATK4i6qAn-[(1s)-1-cyclopropylethyl]-2-phenoxy-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman432
JAK3JakATK4qpsAAn-{1-[6-(phenylamino)pyrazin-2-yl]-1h-benzimidazol-6-yl}prop-2-enamideHuman453
JAK3JakATK4qpsABn-{1-[6-(phenylamino)pyrazin-2-yl]-1h-benzimidazol-6-yl}prop-2-enamideHuman458
JAK3JakATK4qpsCAn-{1-[6-(phenylamino)pyrazin-2-yl]-1h-benzimidazol-6-yl}prop-2-enamideHuman435
JAK3JakATK4qpsCBn-{1-[6-(phenylamino)pyrazin-2-yl]-1h-benzimidazol-6-yl}prop-2-enamideHuman455
JAK3JakATK4qt1A1-{(3s)-1-[(2-methylpropyl)sulfonyl]piperidin-3-yl}-3-(5h-pyrrolo[2,3-b]pyrazin-2-yl)ureaHuman452
JAK3JakATK4rioA4-{[(1r,2s)-2-fluoro-2-methylcyclopentyl]amino}pyrrolo[1,2-b]pyridazine-3-carboxamideHuman440
JAK3JakATK4v0gAAn-[3-(2-{3-amino-6-[1-(1-methylpiperidin-4-yl)-1h-pyrazol-4-yl]pyrazin-2-yl}-1h-benzimidazol-1-yl)phenyl]propanamideHuman6347
JAK3JakATK4v0gABn-[3-(2-{3-amino-6-[1-(1-methylpiperidin-4-yl)-1h-pyrazol-4-yl]pyrazin-2-yl}-1h-benzimidazol-1-yl)phenyl]propanamideHuman6346
JAK3JakATK4v0gBAn-[3-(2-{3-amino-6-[1-(1-methylpiperidin-4-yl)-1h-pyrazol-4-yl]pyrazin-2-yl}-1h-benzimidazol-1-yl)phenyl]propanamideHuman6348
JAK3JakATK4v0gBBn-[3-(2-{3-amino-6-[1-(1-methylpiperidin-4-yl)-1h-pyrazol-4-yl]pyrazin-2-yl}-1h-benzimidazol-1-yl)phenyl]propanamideHuman6345
JAK3JakATK4z16An-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamideHuman6395
JAK3JakATK4z16Bn-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamideHuman6396
JAK3JakATK4z16Cn-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamideHuman6397
JAK3JakATK4z16Dn-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamideHuman6394
JAK3JakATK5lwmAA2-cyano-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1,4,6,8,11-pentaen-4-yl)furan-2-yl]-~{n},~{n}-dimethyl-prop-2-enamideHuman7115
JAK3JakATK5lwmAB2-cyano-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1,4,6,8,11-pentaen-4-yl)furan-2-yl]-~{n},~{n}-dimethyl-prop-2-enamideHuman7118
JAK3JakATK5lwnAA(~{z})-2-cyano-~{n},~{n}-dimethyl-3-[5-[3-[(1~{s},2~{r})-2-methylcyclohexyl]-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1,4,6,8,11-pentaen-4-yl]furan-2-yl]prop-2-enamideHuman7117
JAK3JakATK5lwnAB(2~{s})-2-cyano-~{n},~{n}-dimethyl-3-[5-[3-[(1~{s},2~{r})-2-methylcyclohexyl]-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1,4,6,8,11-pentaen-4-yl]furan-2-yl]propanamideHuman7116
JAK3JakATK5tozA1-{(2s,5r)-2-methyl-5-[(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}propan-1-oneHuman7163
JAK3JakATK5ttsA1-{(3r)-3-[(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}propan-1-oneHuman7439
JAK3JakATK5ttuAA1-[(3ar,7ar)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)octahydro-6h-pyrrolo[2,3-c]pyridin-6-yl]propan-1-oneHuman7435
JAK3JakATK5ttuAB1-[(3ar,7ar)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)octahydro-6h-pyrrolo[2,3-c]pyridin-6-yl]propan-1-oneHuman7438
JAK3JakATK5ttvAAn-[3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]propanamideHuman7437
JAK3JakATK5ttvABn-[3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl]propanamideHuman7436
JAK3JakATK5vo6A4-{[(1r,3s)-3-amino-2,2,3-trimethylcyclopentyl]amino}-6-phenylpyrrolo[1,2-b]pyridazine-3-carboxamideHuman7960
JAK3JakATK5w86AA4-(benzylamino)-6-({4-[(1-methylpiperidin-4-yl)carbamoyl]phenyl}amino)pyridine-3-carboxamideHuman8549
JAK3JakATK5w86BA4-(benzylamino)-6-({4-[(1-methylpiperidin-4-yl)carbamoyl]phenyl}amino)pyridine-3-carboxamideHuman8551
JAK3JakATK5w86CA4-(benzylamino)-6-({4-[(1-methylpiperidin-4-yl)carbamoyl]phenyl}amino)pyridine-3-carboxamideHuman8550
JAK3JakATK5w86DA4-(benzylamino)-6-({4-[(1-methylpiperidin-4-yl)carbamoyl]phenyl}amino)pyridine-3-carboxamideHuman8548
JAK3JakATK5wfjA4-({[3-(propanoylamino)phenyl]methyl}amino)pyrrolo[1,2-b]pyridazine-3-carboxamideHuman8535
JAK3JakATK6aakA4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10366
JAK3JakATK6aakB4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10367
JAK3JakATK6aakC4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10368
JAK3JakATK6aakD4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10365
JAK3JakATK6da4A(z)-1-{2,2-difluoro-6-[5-(2-methoxyethyl)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]-2,3-dihydro-4h-1,4-benzoxazin-4-yl}methanimineHuman10723
JAK3JakATK6db3AA[(1s)-1-methyl-6-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]cyanamideHuman10718
JAK3JakATK6db3AB[(1s)-1-methyl-6-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]cyanamideHuman10719
JAK3JakATK6db4AAn-[(1s)-6-(5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]imidoformamideHuman10724
JAK3JakATK6db4ABn-[(1s)-6-(5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]imidoformamideHuman10721
JAK3JakATK6dudAAn-[(1s)-6-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]imidoformamideHuman10722
JAK3JakATK6dudABn-[(1s)-6-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1h-inden-1-yl]imidoformamideHuman10720
JAK3JakATK6gl9AA(~{e})-3-[3-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)phenyl]prop-2-enenitrileHuman10014
JAK3JakATK6gl9AB(~{e})-3-[3-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)phenyl]prop-2-enenitrileHuman10016
JAK3JakATK6gl9BA(~{e})-3-[3-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)phenyl]prop-2-enenitrileHuman10019
JAK3JakATK6gl9BB(~{e})-3-[3-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)phenyl]prop-2-enenitrileHuman10013
JAK3JakATK6glaAA(~{e})-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]prop-2-enenitrileHuman10018
JAK3JakATK6glaAB(~{e})-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]prop-2-enenitrileHuman10012
JAK3JakATK6glaBA(~{e})-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]prop-2-enenitrileHuman10017
JAK3JakATK6glaBB(~{e})-3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]prop-2-enenitrileHuman10022
JAK3JakATK6glbAA3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]propanenitrileHuman10020
JAK3JakATK6glbAB3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]propanenitrileHuman10023
JAK3JakATK6glbBA3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]propanenitrileHuman10021
JAK3JakATK6glbBB3-[5-(3-cyclohexyl-3,5,8,10-tetrazatricyclo[7.3.0.0^{2,6}]dodeca-1(9),2(6),4,7,11-pentaen-4-yl)furan-2-yl]propanenitrileHuman10015
JAK3JakATK6hzvAA3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrileHuman11756
JAK3JakATK6hzvAB3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrileHuman11751
JAK3JakATK6hzvBA3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrileHuman11753
JAK3JakATK6hzvBB3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrileHuman11754
JAK3JakATK6hzvCA3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrileHuman11752
JAK3JakATK6hzvCB3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrileHuman11755
JAK3JakATK6hzvDA3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrileHuman11749
JAK3JakATK6hzvDB3-[7-(2-hydroxyethyl)-9-(oxan-4-yl)-8-oxidanylidene-purin-2-yl]imidazo[1,2-a]pyridine-6-carbonitrileHuman11750
JAK3JakATK6ny4A4-{[(2r,3r)-1,3-dihydroxybutan-2-yl]amino}-6-phenylpyrrolo[1,2-b]pyridazine-3-carboxamideHuman11052
JAK3JakATK7apfAA3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamideHuman13141
JAK3JakATK7apfAB3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamideHuman13130
JAK3JakATK7apfBA3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamideHuman13137
JAK3JakATK7apfBB3-[3-(propanoylamino)phenyl]-1~{h}-pyrrolo[2,3-b]pyridine-5-carboxamideHuman13132
JAK3JakATK7apgAA~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamideHuman13134
JAK3JakATK7apgAB~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamideHuman13135
JAK3JakATK7apgBA~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamideHuman13131
JAK3JakATK7apgBB~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamideHuman13136
JAK3JakATK7apgCA~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamideHuman13140
JAK3JakATK7apgCB~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamideHuman13139
JAK3JakATK7apgDA~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamideHuman13138
JAK3JakATK7apgDB~{n}-[3-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)phenyl]propanamideHuman13133
JAK3JakATK7c3nAA3-[(3s,4r)-3-methyl-7-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1,7-diazaspiro[3.4]octan-1-yl]-3-oxidanylidene-propanenitrileHuman12389
JAK3JakATK7c3nAB3-[(3s,4r)-3-methyl-7-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1,7-diazaspiro[3.4]octan-1-yl]-3-oxidanylidene-propanenitrileHuman12391
JAK3JakATK7c3nAC3-[(3s,4r)-3-methyl-7-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1,7-diazaspiro[3.4]octan-1-yl]-3-oxidanylidene-propanenitrileHuman12390
JAK3JakATK7q6hAA1-[4-[[2-[(1-methylpyrazol-4-yl)amino]quinazolin-8-yl]amino]piperidin-1-yl]ethanoneHuman14080
JAK3JakATK7q6hAB1-[4-[[2-[(1-methylpyrazol-4-yl)amino]quinazolin-8-yl]amino]piperidin-1-yl]ethanoneHuman14082
JAK3JakATK7q6hAC1-[4-[[2-[(1-methylpyrazol-4-yl)amino]quinazolin-8-yl]amino]piperidin-1-yl]ethanoneHuman14081
JAK3JakATK7uyvAA6-{[(2m)-2-(2-chloro-6-fluorophenyl)-5-oxo-5h-pyrrolo[3,4-b]pyridin-4-yl]amino}-n-ethylpyridine-3-carboxamideHuman14331
JAK3JakATK7uyvAB6-{[(2m)-2-(2-chloro-6-fluorophenyl)-5-oxo-5h-pyrrolo[3,4-b]pyridin-4-yl]amino}-n-ethylpyridine-3-carboxamideHuman14332
KDRVEGFRTK1vr2A-Human5338
KDRVEGFRTK1y6aAAn-[5-(ethylsulfonyl)-2-methoxyphenyl]-5-[3-(2-pyridinyl)phenyl]-1,3-oxazol-2-amineHuman5339
KDRVEGFRTK1y6aABn-[5-(ethylsulfonyl)-2-methoxyphenyl]-5-[3-(2-pyridinyl)phenyl]-1,3-oxazol-2-amineHuman5323
KDRVEGFRTK1y6bAn-(cyclopropylmethyl)-4-(methyloxy)-3-({5-[3-(3-pyridinyl)phenyl]-1,3-oxazol-2-yl}amino)benzenesulfonamideHuman5345
KDRVEGFRTK1ywnAn-{4-[4-amino-6-(4-methoxyphenyl)furo[2,3-d]pyrimidin-5-yl]phenyl}-n'-[2-fluoro-5-(trifluoromethyl)phenyl]ureaHuman5314
KDRVEGFRTK2oh4AAmethyl (5-{4-[({[2-fluoro-5-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-1h-benzimidazol-2-yl)carbamateHuman5347
KDRVEGFRTK2oh4ABmethyl (5-{4-[({[2-fluoro-5-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-1h-benzimidazol-2-yl)carbamateHuman5324
KDRVEGFRTK2p2hA4-(2-anilinopyridin-3-yl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazin-2-amineHuman5310
KDRVEGFRTK2p2iAn-(4-phenoxyphenyl)-2-[(pyridin-4-ylmethyl)amino]nicotinamideHuman5326
KDRVEGFRTK2p2iBn-(4-phenoxyphenyl)-2-[(pyridin-4-ylmethyl)amino]nicotinamideHuman5315
KDRVEGFRTK2qu5A4-[[2-[[4-chloro-3-(trifluoromethyl)phenyl]amino]-3h-benzimidazol-5-yl]oxy]-n-methyl-pyridine-2-carboxamideHuman5317
KDRVEGFRTK2qu6A4-({2-[(4-chloro-3-{[(2s)-1-methylpyrrolidin-2-yl]methoxy}phenyl)amino]-1,3-benzoxazol-5-yl}oxy)-n-methylpyridine-2-carboxamideHuman5316
KDRVEGFRTK2qu6B4-({2-[(4-chloro-3-{[(2s)-1-methylpyrrolidin-2-yl]methoxy}phenyl)amino]-1,3-benzoxazol-5-yl}oxy)-n-methylpyridine-2-carboxamideHuman5340
KDRVEGFRTK2rl5An-(4-chlorophenyl)-7-[(6,7-dimethoxyquinolin-4-yl)oxy]-2,3-dihydro-1,4-benzoxazine-4-carboxamideHuman5348
KDRVEGFRTK2xirAn,2-dimethyl-6-{[7-(2-morpholin-4-ylethoxy)quinolin-4-yl]oxy}-1-benzofuran-3-carboxamideHuman6789
KDRVEGFRTK3b8qAn-(4-chlorophenyl)-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamideHuman5332
KDRVEGFRTK3b8qBn-(4-chlorophenyl)-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamideHuman5319
KDRVEGFRTK3b8rAn-cyclopropyl-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamideHuman5327
KDRVEGFRTK3b8rBn-cyclopropyl-6-[(6,7-dimethoxyquinolin-4-yl)oxy]naphthalene-1-carboxamideHuman5341
KDRVEGFRTK3be2An-{3-[3-(dimethylamino)propyl]-5-(trifluoromethyl)phenyl}-4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]benzamideHuman5337
KDRVEGFRTK3c7qAmethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman5334
KDRVEGFRTK3cjfAAn~4~-(3-methyl-1h-indazol-6-yl)-n~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamineHuman6792
KDRVEGFRTK3cjfABn~4~-(3-methyl-1h-indazol-6-yl)-n~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamineHuman6794
KDRVEGFRTK3cjgAAn~4~-methyl-n~4~-(3-methyl-1h-indazol-6-yl)-n~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamineHuman6791
KDRVEGFRTK3cjgABn~4~-methyl-n~4~-(3-methyl-1h-indazol-6-yl)-n~2~-(3,4,5-trimethoxyphenyl)pyrimidine-2,4-diamineHuman6788
KDRVEGFRTK3cp9A3-(2-aminoquinazolin-6-yl)-1-(3,3-dimethylindolin-6-yl)-4-methylpyridin-2(1h)-oneHuman6786
KDRVEGFRTK3cp9B3-(2-aminoquinazolin-6-yl)-1-(3,3-dimethylindolin-6-yl)-4-methylpyridin-2(1h)-oneHuman6790
KDRVEGFRTK3cpbAn'-(6-aminopyridin-3-yl)-n-(2-cyclopentylethyl)-4-methyl-benzene-1,3-dicarboxamideHuman6787
KDRVEGFRTK3cpbBn'-(6-aminopyridin-3-yl)-n-(2-cyclopentylethyl)-4-methyl-benzene-1,3-dicarboxamideHuman6793
KDRVEGFRTK3cpcA3-(2-aminoquinazolin-6-yl)-4-methyl-1-[3-(trifluoromethyl)phenyl]pyridin-2(1h)-oneHuman5346
KDRVEGFRTK3cpcB3-(2-aminoquinazolin-6-yl)-4-methyl-1-[3-(trifluoromethyl)phenyl]pyridin-2(1h)-oneHuman5309
KDRVEGFRTK3dtwA6-chloro-n-pyrimidin-5-yl-3-{[3-(trifluoromethyl)phenyl]amino}-1,2-benzisoxazole-7-carboxamideHuman5313
KDRVEGFRTK3dtwB6-chloro-n-pyrimidin-5-yl-3-{[3-(trifluoromethyl)phenyl]amino}-1,2-benzisoxazole-7-carboxamideHuman5308
KDRVEGFRTK3eflAn-(3,3-dimethyl-2,3-dihydro-1h-indol-6-yl)-2-[(pyridin-4-ylmethyl)amino]pyridine-3-carboxamideHuman5344
KDRVEGFRTK3eflBn-(3,3-dimethyl-2,3-dihydro-1h-indol-6-yl)-2-[(pyridin-4-ylmethyl)amino]pyridine-3-carboxamideHuman5330
KDRVEGFRTK3ewhAn-[4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)naphthalen-1-yl]-6-(trifluoromethyl)-1h-benzimidazol-2-amineHuman5351
KDRVEGFRTK3u6jAn-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamideHuman5318
KDRVEGFRTK3vheA1-{2-fluoro-4-[(5-methyl-5h-pyrrolo[3,2-d]pyrimidin-4-yl)oxy]phenyl}-3-[3-(trifluoromethyl)phenyl]ureaHuman5331
KDRVEGFRTK3vhkA{3-[(5-methyl-2-phenyl-1,3-oxazol-4-yl)methoxy]phenyl}methanolHuman5342
KDRVEGFRTK3vidA4,5,6,11-tetrahydro-1h-pyrazolo[4',3':6,7]cyclohepta[1,2-b]indoleHuman5335
KDRVEGFRTK3vntAA2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamideHuman5312
KDRVEGFRTK3vntAB2-chloro-3-(1-cyanocyclopropyl)-n-[5-({2-[(cyclopropylcarbonyl)amino][1,3]thiazolo[5,4-b]pyridin-5-yl}oxy)-2-fluorophenyl]benzamideHuman5328
KDRVEGFRTK3vo3AAn-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}oxy)phenyl]-1,3-dimethyl-1h-pyrazole-5-carboxamideHuman5329
KDRVEGFRTK3vo3ABn-[3-({2-[(cyclopropylcarbonyl)amino]imidazo[1,2-b]pyridazin-6-yl}oxy)phenyl]-1,3-dimethyl-1h-pyrazole-5-carboxamideHuman5321
KDRVEGFRTK3wzdAA4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHuman5325
KDRVEGFRTK3wzdAB4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHuman5350
KDRVEGFRTK3wzeAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5336
KDRVEGFRTK3wzeAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5320
KDRVEGFRTK4ag8AaxitinibHuman5311
KDRVEGFRTK4agcAaxitinibHuman5343
KDRVEGFRTK4agdAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman5322
KDRVEGFRTK4asdA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5333
KDRVEGFRTK4aseAtivozanibHuman5349
KDRVEGFRTK5ew3A2-(pyridin-4-ylmethylamino)-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman6289
KDRVEGFRTK5ew3B2-(pyridin-4-ylmethylamino)-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman6290
KDRVEGFRTK6gqoAA2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamideHuman10580
KDRVEGFRTK6gqoAB2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamideHuman10583
KDRVEGFRTK6gqpAA~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamideHuman10582
KDRVEGFRTK6gqpAB~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamideHuman10584
KDRVEGFRTK6gqqAA~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamideHuman10581
KDRVEGFRTK6gqqAB~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamideHuman10585
KDRVEGFRTK6xvjA~{n}-[3-[(dimethylamino)methyl]-5-methyl-phenyl]-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamideHuman12274
KDRVEGFRTK6xvkA~{n}-(4,4-dimethyl-2-prop-1-ynyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamideHuman12273
KITPDGFRTK1pkgAadenosine-5'-diphosphateHuman397
KITPDGFRTK1pkgBadenosine-5'-diphosphateHuman402
KITPDGFRTK1t45AA-Human399
KITPDGFRTK1t45AB-Human394
KITPDGFRTK1t46AA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman393
KITPDGFRTK1t46AB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman404
KITPDGFRTK3g0eAAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman401
KITPDGFRTK3g0eABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman398
KITPDGFRTK3g0fAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman395
KITPDGFRTK3g0fBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman400
KITPDGFRTK4hvsA5-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-n-[4-(trifluoromethyl)benzyl]pyridin-2-amineHuman403
KITPDGFRTK4u0iAA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman405
KITPDGFRTK4u0iAB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman396
KITPDGFRTK6gqjAA2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamideHuman10364
KITPDGFRTK6gqjAB2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamideHuman10354
KITPDGFRTK6gqjBA2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamideHuman10358
KITPDGFRTK6gqjBB2-[4-(6,7-dimethoxyquinazolin-4-yl)oxy-2-methoxy-phenyl]-~{n}-(1-propan-2-ylpyrazol-4-yl)ethanamideHuman10356
KITPDGFRTK6gqkAA~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamideHuman10355
KITPDGFRTK6gqkAB~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamideHuman10353
KITPDGFRTK6gqkBA~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamideHuman10363
KITPDGFRTK6gqkBB~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(1-ethylpyrazol-4-yl)ethanamideHuman10360
KITPDGFRTK6gqlA~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamideHuman10362
KITPDGFRTK6gqlB~{n}-[4-(6,7-dimethoxyquinazolin-4-yl)oxyphenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamideHuman10357
KITPDGFRTK6gqmA~{n}-[4-[[5-fluoranyl-7-(2-methoxyethoxy)quinazolin-4-yl]amino]phenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamideHuman10359
KITPDGFRTK6gqmB~{n}-[4-[[5-fluoranyl-7-(2-methoxyethoxy)quinazolin-4-yl]amino]phenyl]-2-(4-propan-2-yl-1,2,3-triazol-1-yl)ethanamideHuman10361
KITPDGFRTK6hh1AA~{n}-(2,3-dimethylphenyl)-5-(4-pyridin-4-yloxyphenyl)-4~{h}-1,2,4-triazol-3-amineHuman11629
KITPDGFRTK6hh1AB~{n}-(2,3-dimethylphenyl)-5-(4-pyridin-4-yloxyphenyl)-4~{h}-1,2,4-triazol-3-amineHuman11628
KITPDGFRTK6ittAAn-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]ureaHuman11826
KITPDGFRTK6ittABn-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]ureaHuman11824
KITPDGFRTK6ittBAn-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]ureaHuman11821
KITPDGFRTK6ittBBn-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]ureaHuman11820
KITPDGFRTK6itvAAn-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]ureaHuman11822
KITPDGFRTK6itvABn-(5-ethyl-1,2-oxazol-3-yl)-n'-[4-(2-{[6-(4-ethylpyrazin-1(4h)-yl)pyrimidin-4-yl]amino}-1,3-thiazol-5-yl)phenyl]ureaHuman11827
KITPDGFRTK6klaAAn-[6-(4-ethylpiperazin-1-yl)-2-methyl-pyrimidin-4-yl]-5-pyridin-4-yl-1,3-thiazol-2-amineHuman11825
KITPDGFRTK6klaABn-[6-(4-ethylpiperazin-1-yl)-2-methyl-pyrimidin-4-yl]-5-pyridin-4-yl-1,3-thiazol-2-amineHuman11823
KITPDGFRTK6mobAAn-{4-chloro-5-[1-ethyl-7-(methylamino)-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl]-2-fluorophenyl}-n'-phenylureaHuman11469
KITPDGFRTK6mobABn-{4-chloro-5-[1-ethyl-7-(methylamino)-2-oxo-1,2-dihydro-1,6-naphthyridin-3-yl]-2-fluorophenyl}-n'-phenylureaHuman11470
KITPDGFRTK6xv9A~{n}-[3-[(dimethylamino)methyl]-5-methyl-phenyl]-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamideHuman12282
KITPDGFRTK6xv9B~{n}-[3-[(dimethylamino)methyl]-5-methyl-phenyl]-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamideHuman12283
KITPDGFRTK6xvaA~{n}-[[3-[2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanoylamino]-5-methyl-phenyl]methyl]propanamideHuman12284
KITPDGFRTK6xvaB~{n}-[[3-[2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanoylamino]-5-methyl-phenyl]methyl]propanamideHuman12281
KITPDGFRTK6xvbA~{n}-(4,4-dimethyl-2-propyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamideHuman12279
KITPDGFRTK6xvbB~{n}-(4,4-dimethyl-2-propyl-3,1-benzoxazin-6-yl)-2-[3-methoxy-5-(7-methoxyquinolin-4-yl)oxy-pyridin-2-yl]ethanamideHuman12280
KITPDGFRTK7khgAA5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amineHuman13786
KITPDGFRTK7khgAB5-[(5-chloro-1h-pyrrolo[2,3-b]pyridin-3-yl)methyl]-n-{[6-(trifluoromethyl)pyridin-3-yl]methyl}pyridin-2-amineHuman13788
KITPDGFRTK7khjA2-phenyl-5-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman13789
KITPDGFRTK7khkA4,5-dimethyl-n-(2-phenyl-1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazole-3-carboxamideHuman13787
KITPDGFRTK7zw8AA~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amineHuman14622
KITPDGFRTK7zw8AB~{n}-[[4-(1-methylpyrazol-4-yl)phenyl]methyl]-6-[7-(3-pyrrolidin-1-ylpropoxy)imidazo[1,2-a]pyridin-3-yl]pyrimidin-4-amineHuman14624
KITPDGFRTK7zy6A5-imidazo[1,2-a]pyridin-3-yl-~{n}-[(1~{r})-1-(6-pyrrolidin-1-ylpyridin-3-yl)ethyl]pyridin-3-amineHuman14623
KITPDGFRTK8dfmA-Human14677
KITPDGFRTK8dfpA-Human14678
KITPDGFRTK8dfqA-Human14679
KITPDGFRTK8pq9AA(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15118
KITPDGFRTK8pq9AB(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15125
KITPDGFRTK8pqaAA6-(1-methylpyrazol-4-yl)-4-(4-pyrimidin-2-ylpiperazin-1-yl)pyrrolo[2,1-f][1,2,4]triazineHuman15124
KITPDGFRTK8pqaAB6-(1-methylpyrazol-4-yl)-4-(4-pyrimidin-2-ylpiperazin-1-yl)pyrrolo[2,1-f][1,2,4]triazineHuman15115
KITPDGFRTK8pqbAA(1~{s})-1-(4-fluorophenyl)-~{n},~{n}-dimethyl-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15121
KITPDGFRTK8pqbAB(1~{s})-1-(4-fluorophenyl)-~{n},~{n}-dimethyl-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15120
KITPDGFRTK8pqcAA(1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15122
KITPDGFRTK8pqcAB(1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15123
KITPDGFRTK8pqdAA~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]ethanamideHuman15113
KITPDGFRTK8pqdAB~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]ethanamideHuman15126
KITPDGFRTK8pqeAA~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]prop-2-enamideHuman15119
KITPDGFRTK8pqeAB~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]prop-2-enamideHuman15117
KITPDGFRTK8pqfAAmethyl ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]carbamateHuman15116
KITPDGFRTK8pqfABmethyl ~{n}-[(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethyl]carbamateHuman15127
KITPDGFRTK8pqgAA(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15114
KITPDGFRTK8pqgAB(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15112
KSR1RAFTKL7juwBphosphoaminophosphonic acid-adenylate esterHuman12855
KSR1RAFTKL7juxAphosphoaminophosphonic acid-adenylate esterHuman14018
KSR1RAFTKL7juyBphosphoaminophosphonic acid-adenylate esterHuman12920
KSR1RAFTKL7juzA-Human12856
KSR1RAFTKL7juzBphosphoaminophosphonic acid-adenylate esterHuman12851
KSR1RAFTKL7jv0A-Human12848
KSR1RAFTKL7jv0Bphosphoaminophosphonic acid-adenylate esterHuman12853
KSR1RAFTKL7jv1Bphosphoaminophosphonic acid-adenylate esterHuman12854
KSR1RAFTKL7jv1D-Human12849
KSR2RAFTKL2y4iBadenosine-5'-triphosphateHuman1244
KSR2RAFTKL5kkrB6,7-dimethoxy-~{n}-(2-methyl-4-phenoxy-phenyl)quinazolin-4-amineHuman7027
KSR2RAFTKL7juqBadenosine-5'-diphosphateHuman12821
KSR2RAFTKL7jurBphosphoaminophosphonic acid-adenylate esterHuman12822
KSR2RAFTKL7jusBphosphoaminophosphonic acid-adenylate esterHuman12823
KSR2RAFTKL7jutBphosphoaminophosphonic acid-adenylate esterHuman12818
KSR2RAFTKL7juuBphosphoaminophosphonic acid-adenylate esterHuman12820
KSR2RAFTKL7juvBphosphoaminophosphonic acid-adenylate esterHuman12819
LCKSrcTK1qpcAphosphoaminophosphonic acid-adenylate esterHuman2291
LCKSrcTK1qpdAstaurosporineHuman2267
LCKSrcTK1qpeA1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamineHuman2271
LCKSrcTK1qpjAstaurosporineHuman2283
LCKSrcTK2of2A2,3-diphenyl-n-(2-piperazin-1-ylethyl)furo[2,3-b]pyridin-4-amineHuman2261
LCKSrcTK2of4A5,6-diphenyl-n-(2-piperazin-1-ylethyl)furo[2,3-d]pyrimidin-4-amineHuman2296
LCKSrcTK2ofuA2,6-dimethylphenyl 2-(3,5-dimethoxy-4-(3-(4-methylpiperazin-1-yl)propoxy)phenylamino)pyrimidin- 4-yl(2,4-dimethoxyphenyl)carbamateHuman2259
LCKSrcTK2ofvA3-(2-aminoquinazolin-6-yl)-4-methyl-n-[3-(trifluoromethyl)phenyl]benzamideHuman2280
LCKSrcTK2ofvB3-(2-aminoquinazolin-6-yl)-4-methyl-n-[3-(trifluoromethyl)phenyl]benzamideHuman2294
LCKSrcTK2og8An-{2-[(n,n-diethylglycyl)amino]-5-(trifluoromethyl)phenyl}-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamideHuman2286
LCKSrcTK2og8Bn-{2-[(n,n-diethylglycyl)amino]-5-(trifluoromethyl)phenyl}-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamideHuman2282
LCKSrcTK2pl0A4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman2290
LCKSrcTK2zm1An-(2-chlorophenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amineHuman2273
LCKSrcTK2zm4An-(2-chloro-6-methylphenyl)-8-[(3s)-3-methylpiperazin-1-yl]imidazo[1,5-a]quinoxalin-4-amineHuman2262
LCKSrcTK2zybAn-(2,6-dimethylphenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amineHuman2275
LCKSrcTK3ac1A5-{[(1r,2s)-2-aminocyclohexyl]amino}-3-[(3,5-dimethoxyphenyl)amino]pyrazine-2-carboxamideHuman2287
LCKSrcTK3ac2A7-[(2-amino-2-methylpropyl)amino]-2-[(3,5-dimethoxyphenyl)amino]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2266
LCKSrcTK3ac3A2-[(3,5-dimethoxyphenyl)amino]-5-ethyl-7-[(2r)-2-(hydroxymethyl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2292
LCKSrcTK3ac4A5-[(2-amino-1,1-dimethylethyl)amino]-7-[(3,5-dimethoxyphenyl)amino][1,2,4]triazolo[4,3-c]pyrimidine-8-carboxamideHuman2278
LCKSrcTK3ac5A5-{[(1r,2s)-2-aminocyclohexyl]amino}-7-[(3,5-dimethoxyphenyl)amino]-2-(3-hydroxyphenyl)[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxamideHuman2277
LCKSrcTK3ac8A7-[(2-amino-2-methylpropyl)amino]-5-cyclopropyl-2-[(3,5-dimethoxyphenyl)amino]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2300
LCKSrcTK3acjA7-(3,4-dimethoxyphenyl)-5-(ethylsulfanyl)imidazo[1,2-c]pyrimidineHuman2260
LCKSrcTK3ackA6-(5-methoxy-1-methyl-1h-indol-3-yl)-5h-pyrrolo[2,3-b]pyrazineHuman2284
LCKSrcTK3ad4A(4-chlorophenyl)(5-methoxy-1-benzofuran-2-yl)methanoneHuman2268
LCKSrcTK3ad5A4-[4-(benzyloxy)phenyl]-5-{[2-(4-chlorophenyl)-2-oxoethyl]sulfanyl}-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman2270
LCKSrcTK3ad6A7-[(cyclopropylmethyl)amino]-2-[(4-methoxyphenyl)amino]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2274
LCKSrcTK3b2wAn-[5-({[2-fluoro-3-(trifluoromethyl)phenyl]amino}carbonyl)-2-methylphenyl]-4-methoxy-2-[(4-piperazin-1-ylphenyl)amino]pyrimidine-5-carboxamideHuman2299
LCKSrcTK3bymAn-phenyl-1-{4-[(3,4,5-trimethoxyphenyl)amino]-1,3,5-triazin-2-yl}-1h-benzimidazol-2-amineHuman2264
LCKSrcTK3byoA6-(2,6-dimethylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimido[5',4':5,6]pyrimido[1,2-a]benzimidazol-5(6h)-oneHuman2272
LCKSrcTK3bysA4-methyl-n~3~-(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-5-yl)-n~1~-[3-(trifluoromethyl)phenyl]benzene-1,3-dicarboxamideHuman2293
LCKSrcTK3byuA2-methyl-n-{4-methyl-3-[(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-5-yl)carbamoyl]phenyl}-3-(trifluoromethyl)benzamideHuman2288
LCKSrcTK3kmmA3-(2,6-dichlorophenyl)-7-({4-[2-(diethylamino)ethoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman2265
LCKSrcTK3kxzA3-[7-[(3-hydroxyphenyl)amino]pyrazolo[1,5-a]pyrimidin-2-yl]-n-(1-hydroxy-2,2,6,6-tetramethyl-piperidin-4-yl)benzamideHuman2281
LCKSrcTK3lckAA-Human2263
LCKSrcTK3lckAB-Human2301
LCKSrcTK3mpmAA4-{(6r,7r)-7-amino-3-[3-(4-methylpiperazin-1-yl)phenyl]-6,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl}phenolHuman2279
LCKSrcTK3mpmAB4-{(6r,7r)-7-amino-3-[3-(4-methylpiperazin-1-yl)phenyl]-6,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl}phenolHuman2295
LCKSrcTK4c3fAAn-phenyl-4-(5-phenyl-1h-pyrazol-4-yl)pyrimidin-2-amineHuman2276
LCKSrcTK4c3fABn-phenyl-4-(5-phenyl-1h-pyrazol-4-yl)pyrimidin-2-amineHuman2297
LCKSrcTK6pdjAAn-{4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]-3-methylphenyl}-1-methyl-1h-indazole-3-carboxamideHuman11698
LCKSrcTK6pdjABn-{4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]-3-methylphenyl}-1-methyl-1h-indazole-3-carboxamideHuman11699
LIMK1LISKTKL3s95AAstaurosporineHuman1246
LIMK1LISKTKL3s95ABstaurosporineHuman1248
LIMK1LISKTKL3s95BAstaurosporineHuman1245
LIMK1LISKTKL3s95BBstaurosporineHuman1247
LIMK1LISKTKL5hvjAAphosphoaminophosphonic acid-adenylate esterHuman6599
LIMK1LISKTKL5hvjABphosphoaminophosphonic acid-adenylate esterHuman6598
LIMK1LISKTKL5hvjBA-Human6597
LIMK1LISKTKL5hvjBB-Human6595
LIMK1LISKTKL5hvkAphosphoaminophosphonic acid-adenylate esterHuman6600
LIMK1LISKTKL5hvkCphosphoaminophosphonic acid-adenylate esterHuman6596
LIMK1LISKTKL5l6wLphosphothiophosphoric acid-adenylate esterHuman6668
LIMK1LISKTKL5nxcL(2~{r})-2-azanyl-2-cyclohexyl-~{n}-[2-(1-methylpyrazol-4-yl)-9-oxidanylidene-3,10,11-triazatricyclo[6.4.1.0^{4,13}]trideca-1,4,6,8(13),11-pentaen-6-yl]ethanamideHuman7592
LIMK1LISKTKL7atsAn-[3-[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]benzenesulfonamideHuman13164
LIMK1LISKTKL7atuA(s)-2-benzyl-6-(8-chloro-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-7-oxo-4,5,6,7-tetrahydro-2h-pyrazolo[3,4-c]pyridine-3-carboxamideHuman14019
LIMK1LISKTKL7b8wA2-(2-methylpropanoylamino)-~{n}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamideHuman14126
LIMK1LISKTKL8aauLA~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamideHuman14555
LIMK1LISKTKL8aauLB~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamideHuman14554
LIMK2LISKTKL4tptAn-{4-[(1s)-1,2-dihydroxyethyl]benzyl}-n-methyl-4-(phenylsulfamoyl)benzamideHuman2476
LIMK2LISKTKL4tptBn-{4-[(1s)-1,2-dihydroxyethyl]benzyl}-n-methyl-4-(phenylsulfamoyl)benzamideHuman2475
LIMK2LISKTKL5nxdAA4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamideHuman7623
LIMK2LISKTKL5nxdAB4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamideHuman7621
LIMK2LISKTKL5nxdBA4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamideHuman7624
LIMK2LISKTKL5nxdBB4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamideHuman7622
LIMK2LISKTKL7qhgAA2-(2-methylpropanoylamino)-~{n}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamideHuman14021
LIMK2LISKTKL7qhgAB2-(2-methylpropanoylamino)-~{n}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamideHuman14020
LIMK2LISKTKL8wswAA~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamideHuman14862
LIMK2LISKTKL8wswAB~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamideHuman14861
LMTK3 (LMR3)LmrTK6seqAA-Human12994
LMTK3 (LMR3)LmrTK6seqAB-Human12995
LRRK1LRRKTKL8e04A-Human14879
LRRK1LRRKTKL8e05A-Human14882
LRRK1LRRKTKL8e06A-Human14881
LRRK1LRRKTKL8facA-Human14880
LRRK2LRRKTKL6vnoA1-Human12735
LRRK2LRRKTKL6vnoA10-Human12717
LRRK2LRRKTKL6vnoA2-Human12725
LRRK2LRRKTKL6vnoA3-Human12731
LRRK2LRRKTKL6vnoA4-Human12719
LRRK2LRRKTKL6vnoA5-Human12715
LRRK2LRRKTKL6vnoA6-Human12732
LRRK2LRRKTKL6vnoA7-Human12712
LRRK2LRRKTKL6vnoA8-Human12718
LRRK2LRRKTKL6vnoA9-Human12728
LRRK2LRRKTKL6vp6A-Human12714
LRRK2LRRKTKL6vp6B-Human12726
LRRK2LRRKTKL6vp7A1-Human12713
LRRK2LRRKTKL6vp7A10-Human12730
LRRK2LRRKTKL6vp7A2-Human12724
LRRK2LRRKTKL6vp7A3-Human12733
LRRK2LRRKTKL6vp7A4-Human12720
LRRK2LRRKTKL6vp7A5-Human12716
LRRK2LRRKTKL6vp7A6-Human12721
LRRK2LRRKTKL6vp7A7-Human12727
LRRK2LRRKTKL6vp7A8-Human12722
LRRK2LRRKTKL6vp7A9-Human12729
LRRK2LRRKTKL6vp8A-Human12723
LRRK2LRRKTKL6vp8B-Human12734
LRRK2LRRKTKL7lhtA-Human13623
LRRK2LRRKTKL7lhwA-Human13625
LRRK2LRRKTKL7li3A-Human13626
LRRK2LRRKTKL7li4A-Human13624
LRRK2LRRKTKL8fo8C-Human15133
LRRK2LRRKTKL8fo9A-Human15132
LRRK2LRRKTKL8txzAA-Human15056
LRRK2LRRKTKL8txzAB-Human15057
LRRK2LRRKTKL8tyqAA4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-3-[(1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]benzamideHuman15058
LRRK2LRRKTKL8tyqAB4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-3-[(1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]benzamideHuman15055
LRRK2LRRKTKL8tzbA-Human15052
LRRK2LRRKTKL8tzcA-Human15050
LRRK2LRRKTKL8tzeA4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-3-[(1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]benzamideHuman15054
LRRK2LRRKTKL8tzfA-Human15059
LRRK2LRRKTKL8tzgAA-Human15051
LRRK2LRRKTKL8tzgAB-Human15053
LRRK2LRRKTKL8u7lA-Human15184
LRRK2LRRKTKL8u8bA-Human15185
Lyn (LYN)SrcTK2zv7A-Mouse5771
Lyn (LYN)SrcTK2zv8Aphosphoaminophosphonic acid-adenylate esterMouse5772
Lyn (LYN)SrcTK2zv9A1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamineMouse5773
Lyn (LYN)SrcTK2zvaAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideMouse5774
LYNSrcTK3a4oXstaurosporineHuman1812
LYNSrcTK5xy1An-(1h-indazol-6-yl)-8-piperidin-4-yloxy-6-propyl-quinazolin-2-amineHuman8271
MAP2K1STE7STE1s9jAadenosine-5'-triphosphateHuman3316
MAP2K1STE7STE2p55A2-[(4-ethynyl-2-fluorophenyl)amino]-3,4-difluoro-n-(2-hydroxyethoxy)benzamideHuman3327
MAP2K1STE7STE3dv3AAadenosine-5'-triphosphateHuman3322
MAP2K1STE7STE3dv3ABadenosine-5'-triphosphateHuman3311
MAP2K1STE7STE3dy7Aadenosine-5'-triphosphateHuman3282
MAP2K1STE7STE3e8nAadenosine-5'-triphosphateHuman3323
MAP2K1STE7STE3eqbAAadenosine-5'-triphosphateHuman3324
MAP2K1STE7STE3eqbABadenosine-5'-triphosphateHuman3310
MAP2K1STE7STE3eqcAA2-[(2-chloro-4-iodophenyl)amino]-n-{[(2r)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamideHuman3280
MAP2K1STE7STE3eqcAB2-[(2-chloro-4-iodophenyl)amino]-n-{[(2r)-2,3-dihydroxypropyl]oxy}-3,4-difluorobenzamideHuman3300
MAP2K1STE7STE3eqdAphosphothiophosphoric acid-adenylate esterHuman3284
MAP2K1STE7STE3eqfAk-252aHuman3317
MAP2K1STE7STE3eqgAadenosine-5'-diphosphateHuman3304
MAP2K1STE7STE3eqhA(2z)-bis{amino[(2-aminophenyl)sulfanyl]methylidene}butanedinitrileHuman3290
MAP2K1STE7STE3eqiAadenosine-5'-diphosphateHuman3308
MAP2K1STE7STE3mblAAadenosine-5'-diphosphateHuman3292
MAP2K1STE7STE3mblABadenosine-5'-diphosphateHuman3318
MAP2K1STE7STE3ornAphosphoaminophosphonic acid-adenylate esterHuman3277
MAP2K1STE7STE3os3Aadenosine-5'-triphosphateHuman3281
MAP2K1STE7STE3pp1AAadenosine-5'-triphosphateHuman3294
MAP2K1STE7STE3pp1ABadenosine-5'-triphosphateHuman3285
MAP2K1STE7STE3slsAAphosphoaminophosphonic acid-adenylate esterHuman9486
MAP2K1STE7STE3slsABphosphoaminophosphonic acid-adenylate esterHuman9485
MAP2K1STE7STE3slsBAphosphoaminophosphonic acid-adenylate esterHuman9487
MAP2K1STE7STE3slsBBphosphoaminophosphonic acid-adenylate esterHuman9484
MAP2K1STE7STE3v01An-{[(2r)-2,3-dihydroxypropyl]oxy}-3-[(2-fluoro-4-iodophenyl)amino]furo[3,2-c]pyridine-2-carboxamideHuman3291
MAP2K1STE7STE3v04A4-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)-1h-indazole-5-carboxamideHuman3325
MAP2K1STE7STE3vvhAAadenosine-5'-triphosphateHuman3288
MAP2K1STE7STE3vvhABadenosine-5'-triphosphateHuman3296
MAP2K1STE7STE3vvhBAadenosine-5'-triphosphateHuman3321
MAP2K1STE7STE3vvhBBadenosine-5'-triphosphateHuman3289
MAP2K1STE7STE3vvhCAadenosine-5'-triphosphateHuman3306
MAP2K1STE7STE3vvhCBadenosine-5'-triphosphateHuman3287
MAP2K1STE7STE3w8qAphosphothiophosphoric acid-adenylate esterHuman3298
MAP2K1STE7STE3wigAphosphoaminophosphonic acid-adenylate esterHuman3329
MAP2K1STE7STE3zlsA1h-pyrrolo[2,3-b]pyridine-3-carboxylic acidHuman3279
MAP2K1STE7STE3zlwA(1r)-1-hydroxy-1-methyl-2,3,6,7-tetrahydro-1h,5h-pyrido[3,2,1-ij]quinolin-5-oneHuman3278
MAP2K1STE7STE3zlxA7-choro-6-[(3r)-pyrrolidin-3-ylmethoxy]isoquinolin-1(2h)-oneHuman3312
MAP2K1STE7STE3zlyA3-amino-1h-indazole-4-carbonitrileHuman3320
MAP2K1STE7STE3zm4A7-chloranyl-6-[(3s)-pyrrolidin-3-yl]oxy-2h-isoquinolin-1-oneHuman3303
MAP2K1STE7STE4an2AA[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]-[3-oxidanyl-3-[(2s)-piperidin-2-yl]azetidin-1-yl]methanoneHuman3309
MAP2K1STE7STE4an2AB[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]-[3-oxidanyl-3-[(2s)-piperidin-2-yl]azetidin-1-yl]methanoneHuman3326
MAP2K1STE7STE4an3Aadenosine-5'-triphosphateHuman3295
MAP2K1STE7STE4an9Aphosphomethylphosphonic acid adenylate esterHuman3330
MAP2K1STE7STE4anbA[3-(aminomethyl)-3-oxidanyl-azetidin-1-yl]-[3,4-bis(fluoranyl)-2-[(2-fluoranyl-4-iodanyl-phenyl)amino]phenyl]methanoneHuman3302
MAP2K1STE7STE4arkAadenosine-5'-diphosphateHuman3299
MAP2K1STE7STE4lmnAphosphoaminophosphonic acid-adenylate esterHuman3283
MAP2K1STE7STE4mneAAphosphomethylphosphonic acid adenylate esterHuman3293
MAP2K1STE7STE4mneABphosphomethylphosphonic acid adenylate esterHuman3307
MAP2K1STE7STE4mneDAphosphomethylphosphonic acid adenylate esterHuman3313
MAP2K1STE7STE4mneDBphosphomethylphosphonic acid adenylate esterHuman3315
MAP2K1STE7STE4mneEAphosphomethylphosphonic acid adenylate esterHuman3314
MAP2K1STE7STE4mneEBphosphomethylphosphonic acid adenylate esterHuman3286
MAP2K1STE7STE4mneHAphosphomethylphosphonic acid adenylate esterHuman3319
MAP2K1STE7STE4mneHBphosphomethylphosphonic acid adenylate esterHuman3328
MAP2K1STE7STE4u7zA5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamideHuman3297
MAP2K1STE7STE4u80Aphosphoaminophosphonic acid-adenylate esterHuman3305
MAP2K1STE7STE4u81A8-[(4-cyclopropyl-2-fluorophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-7-carboxamideHuman3301
MAP2K1STE7STE5bx0Aethyl 2h-indazole-5-carboxylateHuman6300
MAP2K1STE7STE5eymAA3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman6966
MAP2K1STE7STE5eymAB3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman6969
MAP2K1STE7STE5eymBA3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman6968
MAP2K1STE7STE5eymBB3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman6967
MAP2K1STE7STE5hzeAA(3s,4r,8s,9s,11e)-8,9,16-trihydroxy-3,4-dimethyl-14-(methylamino)-3,4,5,6,9,10-hexahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman7569
MAP2K1STE7STE5hzeAB(3s,4r,8s,9s,11e)-8,9,16-trihydroxy-3,4-dimethyl-14-(methylamino)-3,4,5,6,9,10-hexahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman7570
MAP2K1STE7STE5yt3Aphosphoaminophosphonic acid-adenylate esterHuman10692
MAP2K1STE7STE5yt3Bphosphoaminophosphonic acid-adenylate esterHuman10694
MAP2K1STE7STE5yt3Cphosphoaminophosphonic acid-adenylate esterHuman10693
MAP2K1STE7STE5yt3Dphosphoaminophosphonic acid-adenylate esterHuman10695
MAP2K1STE7STE6nybBadenosine-5'-diphosphateHuman11719
MAP2K1STE7STE6pp9BAphosphoaminophosphonic acid-adenylate esterHuman11716
MAP2K1STE7STE6pp9BBphosphoaminophosphonic acid-adenylate esterHuman11720
MAP2K1STE7STE6q0jCA5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11721
MAP2K1STE7STE6q0jCB5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11713
MAP2K1STE7STE6q0jDA5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11714
MAP2K1STE7STE6q0jDB5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11718
MAP2K1STE7STE6q0tCA5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11715
MAP2K1STE7STE6q0tCB5-[(2-fluoro-4-iodophenyl)amino]-n-(2-hydroxyethoxy)imidazo[1,5-a]pyridine-6-carboxamideHuman11717
MAP2K1STE7STE6u2gAphosphomethylphosphonic acid adenylate esterHuman11574
MAP2K1STE7STE6v2wBAphosphoaminophosphonic acid-adenylate esterHuman13015
MAP2K1STE7STE6v2wBBphosphoaminophosphonic acid-adenylate esterHuman13017
MAP2K1STE7STE7b3mAphosphoaminophosphonic acid-adenylate esterHuman13365
MAP2K1STE7STE7b3mBphosphoaminophosphonic acid-adenylate esterHuman13363
MAP2K1STE7STE7b7rAphosphoaminophosphonic acid-adenylate esterHuman13397
MAP2K1STE7STE7b7rBphosphoaminophosphonic acid-adenylate esterHuman13400
MAP2K1STE7STE7b94Bphosphoaminophosphonic acid-adenylate esterHuman13364
MAP2K1STE7STE7b9lAAphosphoaminophosphonic acid-adenylate esterHuman13402
MAP2K1STE7STE7b9lABphosphoaminophosphonic acid-adenylate esterHuman13401
MAP2K1STE7STE7b9lBAphosphoaminophosphonic acid-adenylate esterHuman13398
MAP2K1STE7STE7b9lBBphosphoaminophosphonic acid-adenylate esterHuman13399
MAP2K1STE7STE7f2xAphosphoaminophosphonic acid-adenylate esterHuman14243
MAP2K1STE7STE7m0tB5-[(4-bromo-2-chlorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamideHuman13512
MAP2K1STE7STE7m0uB5-[(4-bromo-2-fluorophenyl)amino]-4-fluoro-n-(2-hydroxyethoxy)-1-methyl-1h-benzimidazole-6-carboxamideHuman13517
MAP2K1STE7STE7m0vBAphosphoaminophosphonic acid-adenylate esterHuman13518
MAP2K1STE7STE7m0vBBphosphoaminophosphonic acid-adenylate esterHuman13511
MAP2K1STE7STE7m0wBphosphoaminophosphonic acid-adenylate esterHuman13515
MAP2K1STE7STE7m0xBAphosphoaminophosphonic acid-adenylate esterHuman13514
MAP2K1STE7STE7m0xBBphosphoaminophosphonic acid-adenylate esterHuman13519
MAP2K1STE7STE7m0yBphosphoaminophosphonic acid-adenylate esterHuman13513
MAP2K1STE7STE7m0zBphosphoaminophosphonic acid-adenylate esterHuman13516
MAP2K1STE7STE7mfdBn-(3-fluoro-4-{[4-methyl-2-oxo-7-(pyrimidin-2-yloxy)-2h-chromen-3-yl]methyl}pyridin-2-yl)-n'-methylsulfuric diamideHuman14076
MAP2K1STE7STE7pqvAA8-(2-chloranyl-4-methoxy-phenyl)-7-fluoranyl-1-piperidin-4-yl-imidazo[4,5-c]quinolineHuman14157
MAP2K1STE7STE7pqvAB8-(2-chloranyl-4-methoxy-phenyl)-7-fluoranyl-1-piperidin-4-yl-imidazo[4,5-c]quinolineHuman14158
MAP2K1STE7STE7umbBphosphoaminophosphonic acid-adenylate esterHuman14989
MAP2K1STE7STE7xlpA(1~{r},3~{s})-3-[[6-[2-chloranyl-4-(4-methylpyrimidin-2-yl)oxy-phenyl]-3-methyl-1~{h}-indazol-4-yl]oxy]cyclohexan-1-amineHuman14644
MAP2K1STE7STE7xncA~{n}-[4-[[6-(3-chloranylpyridin-4-yl)-3-methyl-1~{h}-indazol-4-yl]oxy]cyclohexyl]ethanamideHuman14643
MAP2K1STE7STE8dgsBAphosphothiophosphoric acid-adenylate esterHuman14825
MAP2K1STE7STE8dgsBBphosphothiophosphoric acid-adenylate esterHuman14826
MAP2K1STE7STE8dgtBAphosphothiophosphoric acid-adenylate esterHuman14828
MAP2K1STE7STE8dgtBBphosphothiophosphoric acid-adenylate esterHuman14827
MAP2K2STE7STE1s9iAadenosine-5'-triphosphateHuman2772
MAP2K2STE7STE1s9iBadenosine-5'-triphosphateHuman2770
MAP2K4STE7STE3alnAphosphoaminophosphonic acid-adenylate esterHuman2832
MAP2K4STE7STE3alnBphosphoaminophosphonic acid-adenylate esterHuman2830
MAP2K4STE7STE3alnCphosphoaminophosphonic acid-adenylate esterHuman2831
MAP2K4STE7STE3aloAphosphoaminophosphonic acid-adenylate esterHuman2835
MAP2K4STE7STE3vutA-Human2834
MAP2K4STE7STE3vutB-Human2833
MAP2K6STE7STE3enmAA-Human1225
MAP2K6STE7STE3enmAB-Human1229
MAP2K6STE7STE3enmBA-Human1227
MAP2K6STE7STE3enmBB-Human1232
MAP2K6STE7STE3enmCA-Human1234
MAP2K6STE7STE3enmCB-Human1226
MAP2K6STE7STE3enmDA-Human1230
MAP2K6STE7STE3enmDB-Human1233
MAP2K6STE7STE3fmeAstaurosporineHuman1231
MAP2K6STE7STE3vn9A9-{5-o-[(r)-hydroxy{[(s)-hydroxy(phosphonoamino)phosphoryl]oxy}phosphoryl]-beta-l-ribofuranosyl}-9h-purin-6-amineHuman1228
MAP2K6STE7STE8a8mBphosphomethylphosphonic acid adenosyl esterHuman14292
MAP2K6STE7STE8p7jAn-[3-(1h-pyrrolo[2,3-b]pyridin-4-yl)phenyl]prop-2-enamideHuman14833
MAP2K6STE7STE8pm3A~{n}-[3-(2-azanylpyridin-4-yl)phenyl]propanamideHuman14994
MAP2K7STE7STE2dylA-Human1240
MAP2K7STE7STE3wzuA(3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman1239
MAP2K7STE7STE5b2kA-Human6503
MAP2K7STE7STE5b2lAA-Human6501
MAP2K7STE7STE5b2lAB-Human6502
MAP2K7STE7STE5b2mA-Human6500
MAP2K7STE7STE5y8uA-Human8556
MAP2K7STE7STE5y90AA-Human8555
MAP2K7STE7STE5y90AB-Human8557
MAP2K7STE7STE5z1dAn-[3-(6-methyl-1h-indazol-3-yl)phenyl]prop-2-enamideHuman10827
MAP2K7STE7STE5z1eAn-[3-(6-methyl-1h-indazol-3-yl)phenyl]prop-2-enamideHuman10828
MAP2K7STE7STE6ib0A1-[(3~{r})-3-(4-azanyl-3-ethynyl-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]prop-2-en-1-oneHuman10922
MAP2K7STE7STE6ib2A1-[(3~{r})-3-[4-azanyl-3-[1-(4-ethanoylphenyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman10921
MAP2K7STE7STE6qflA-Human11080
MAP2K7STE7STE6qfrA-Human11081
MAP2K7STE7STE6qftA1-[(3~{r})-3-(4-azanyl-3-iodanyl-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]propan-1-oneHuman11085
MAP2K7STE7STE6qg4A1-[(3~{r})-3-[4-azanyl-3-(4-hydroxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman11084
MAP2K7STE7STE6qg7A(r)-1-(3-(4-amino-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-oneHuman11083
MAP2K7STE7STE6qhoA1-[(3~{r})-3-(4-azanylpyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl]propan-1-oneHuman11079
MAP2K7STE7STE6qhrA1-[(3~{r})-3-[4-azanyl-3-(1~{h}-pyrrolo[2,3-b]pyridin-5-yl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman11082
MAP2K7STE7STE6yfzAA-Human12679
MAP2K7STE7STE6yfzAB-Human12682
MAP2K7STE7STE6yg0A-Human12695
MAP2K7STE7STE6yg1AA-Human12690
MAP2K7STE7STE6yg1AB-Human12684
MAP2K7STE7STE6yg1BA-Human12691
MAP2K7STE7STE6yg1BB-Human12680
MAP2K7STE7STE6yg1CA-Human12692
MAP2K7STE7STE6yg1CB-Human12688
MAP2K7STE7STE6yg2AA1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman12678
MAP2K7STE7STE6yg2AB1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman12686
MAP2K7STE7STE6yg3AAn-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamideHuman12689
MAP2K7STE7STE6yg3ABn-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamideHuman12681
MAP2K7STE7STE6yg4A(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman12693
MAP2K7STE7STE6yg5A[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}amino)phenyl]acetonitrileHuman12677
MAP2K7STE7STE6yg6AA~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHuman12676
MAP2K7STE7STE6yg6AB~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHuman12687
MAP2K7STE7STE6yg6BA~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHuman12673
MAP2K7STE7STE6yg6BB~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{s})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHuman12694
MAP2K7STE7STE6yg7AA~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHuman12683
MAP2K7STE7STE6yg7AB~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHuman12674
MAP2K7STE7STE6yg7BA~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHuman12696
MAP2K7STE7STE6yg7BB~{n}-[4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-[[(3~{r})-1-propanoylpyrrolidin-3-yl]amino]pyrimidin-4-yl]oxy-benzamideHuman12685
MAP2K7STE7STE6yz4AA-Human12697
MAP2K7STE7STE6yz4AB-Human12675
MAP2K7STE7STE7cbxAA3-(1h-indazol-3-yl)-5-(prop-2-enoylamino)-n-prop-2-ynyl-benzamideHuman12815
MAP2K7STE7STE7cbxAB3-(1h-indazol-3-yl)-5-(prop-2-enoylamino)-n-prop-2-ynyl-benzamideHuman12816
MAP2K7STE7STE7oviA1-[(3~{r})-3-[4-azanyl-3-[1-(2-phenylethyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman14301
MAP2K7STE7STE7ovjAA1-[(3~{r})-3-[4-azanyl-3-[1-[2,2-bis(fluoranyl)-2-phenyl-ethyl]-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman14306
MAP2K7STE7STE7ovjAB1-[(3~{r})-3-[4-azanyl-3-[1-[2,2-bis(fluoranyl)-2-phenyl-ethyl]-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman14299
MAP2K7STE7STE7ovkA1-[(3~{r})-3-[4-azanyl-3-[1-(5-bromanyl-2-oxidanyl-phenyl)-1,2,3-triazol-4-yl]pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-oneHuman14298
MAP2K7STE7STE7ovlAA3-(2~{h}-indazol-3-yl)-~{n}-[[1-[(1~{r},2~{r})-2-methoxycyclohexyl]-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamideHuman14307
MAP2K7STE7STE7ovlAB3-(2~{h}-indazol-3-yl)-~{n}-[[1-[(1~{r},2~{r})-2-methoxycyclohexyl]-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamideHuman14304
MAP2K7STE7STE7ovmAA~{n}-[(1-cyclobutyl-1,2,3-triazol-4-yl)methyl]-3-(1~{h}-indazol-3-yl)-5-(propanoylamino)benzamideHuman14305
MAP2K7STE7STE7ovmAB~{n}-[(1-cyclobutyl-1,2,3-triazol-4-yl)methyl]-3-(1~{h}-indazol-3-yl)-5-(propanoylamino)benzamideHuman14302
MAP2K7STE7STE7ovnAA3-(1~{h}-indazol-3-yl)-~{n}-[[1-(2-methylphenyl)-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamideHuman14303
MAP2K7STE7STE7ovnAB3-(1~{h}-indazol-3-yl)-~{n}-[[1-(2-methylphenyl)-1,2,3-triazol-4-yl]methyl]-5-(propanoylamino)benzamideHuman14300
MAP3K12 (DLK)MLKTKL5cenAA-Human6157
MAP3K12 (DLK)MLKTKL5cenAB-Human6160
MAP3K12 (DLK)MLKTKL5ceoAA2-[[6-[3,3-bis(fluoranyl)pyrrolidin-1-yl]-4-[1-(oxetan-3-yl)piperidin-4-yl]pyridin-2-yl]amino]pyridine-4-carbonitrileHuman6156
MAP3K12 (DLK)MLKTKL5ceoAB2-[[6-[3,3-bis(fluoranyl)pyrrolidin-1-yl]-4-[1-(oxetan-3-yl)piperidin-4-yl]pyridin-2-yl]amino]pyridine-4-carbonitrileHuman6155
MAP3K12 (DLK)MLKTKL5cepAAn-(5-piperidin-4-yl-1-propan-2-yl-pyrazol-3-yl)-4-(trifluoromethyl)pyridin-2-amineHuman6158
MAP3K12 (DLK)MLKTKL5cepABn-(5-piperidin-4-yl-1-propan-2-yl-pyrazol-3-yl)-4-(trifluoromethyl)pyridin-2-amineHuman6154
MAP3K12 (DLK)MLKTKL5ceqAA2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrileHuman6159
MAP3K12 (DLK)MLKTKL5ceqAB2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrileHuman6153
MAP3K12 (DLK)MLKTKL5vo1AA5-{5-[(1r,5s,6r)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amineHuman8540
MAP3K12 (DLK)MLKTKL5vo1AB5-{5-[(1r,5s,6r)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amineHuman8541
MAP3K12 (DLK)MLKTKL5vo2AA5-{5-[1-(oxetan-3-yl)piperidin-4-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amineHuman8543
MAP3K12 (DLK)MLKTKL5vo2AB5-{5-[1-(oxetan-3-yl)piperidin-4-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amineHuman8542
MAP3K12 (DLK)MLKTKL8degAmethyl (1s,4s)-5-{(4p)-4-[5-amino-6-(difluoromethoxy)pyrazin-2-yl]-6-[(1r,4r)-2-azabicyclo[2.1.1]hexan-2-yl]pyridin-2-yl}-2,5-diazabicyclo[2.2.1]heptane-2-carboxylateHuman14557
MAP3K12 (DLK)MLKTKL8ourAA5-[1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)-2-propan-2-yl-imidazol-4-yl]-3-(trifluoromethyloxy)pyridin-2-amineHuman14856
MAP3K12 (DLK)MLKTKL8ourAB5-[1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)-2-propan-2-yl-imidazol-4-yl]-3-(trifluoromethyloxy)pyridin-2-amineHuman14852
MAP3K12 (DLK)MLKTKL8ousAA(1s)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2-methyl-propan-1-olHuman14857
MAP3K12 (DLK)MLKTKL8ousAB(1s)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2-methyl-propan-1-olHuman14854
MAP3K12 (DLK)MLKTKL8outAA(1r)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-fluoranyl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2,2,2-tris(fluoranyl)ethanolHuman14853
MAP3K12 (DLK)MLKTKL8outAB(1r)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-fluoranyl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2,2,2-tris(fluoranyl)ethanolHuman14855
Map3k14 (NIK)STE-UniqueSTE4g3cAA-Mouse5797
Map3k14 (NIK)STE-UniqueSTE4g3cAB-Mouse5786
Map3k14 (NIK)STE-UniqueSTE4g3cBA-Mouse5792
Map3k14 (NIK)STE-UniqueSTE4g3cBB-Mouse5787
Map3k14 (NIK)STE-UniqueSTE4g3eAA(2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-olMouse5790
Map3k14 (NIK)STE-UniqueSTE4g3eAB(2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-olMouse5795
Map3k14 (NIK)STE-UniqueSTE4g3eBA(2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-olMouse5796
Map3k14 (NIK)STE-UniqueSTE4g3eBB(2r)-4-[1-(2-amino-5-chloropyrimidin-4-yl)-2,3-dihydro-1h-indol-6-yl]-2-(1,3-thiazol-2-yl)but-3-yn-2-olMouse5794
Map3k14 (NIK)STE-UniqueSTE4g3fAA3-{2-[(5-fluoro-2-hydroxyphenyl)amino]-1,3-thiazol-4-yl}benzonitrileMouse5789
Map3k14 (NIK)STE-UniqueSTE4g3fAB3-{2-[(5-fluoro-2-hydroxyphenyl)amino]-1,3-thiazol-4-yl}benzonitrileMouse5788
Map3k14 (NIK)STE-UniqueSTE4g3gAA4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenolMouse5793
Map3k14 (NIK)STE-UniqueSTE4g3gAB4-fluoro-2-{[4-(pyridin-4-yl)-1,3-thiazol-2-yl]amino}phenolMouse5791
Map3k14 (NIK)STE-UniqueSTE5t8oAA10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamideMouse7373
Map3k14 (NIK)STE-UniqueSTE5t8oAB10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamideMouse7371
Map3k14 (NIK)STE-UniqueSTE5t8oBA10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamideMouse7372
Map3k14 (NIK)STE-UniqueSTE5t8oBB10-(3-methyl-3-oxidanyl-but-1-ynyl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2-carboxamideMouse7378
Map3k14 (NIK)STE-UniqueSTE5t8pAA6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamideMouse7368
Map3k14 (NIK)STE-UniqueSTE5t8pAB6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamideMouse7377
Map3k14 (NIK)STE-UniqueSTE5t8pBA6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamideMouse7376
Map3k14 (NIK)STE-UniqueSTE5t8pBB6,7-dihydrothieno[4,5]oxepino[1,2-~{c}]pyridine-2-carboxamideMouse7379
Map3k14 (NIK)STE-UniqueSTE5t8qAA1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamideMouse7370
Map3k14 (NIK)STE-UniqueSTE5t8qAB1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamideMouse7369
Map3k14 (NIK)STE-UniqueSTE5t8qBA1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamideMouse7374
Map3k14 (NIK)STE-UniqueSTE5t8qBB1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamideMouse7375
Map3k14 (NIK)STE-UniqueSTE6g4yAA10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamideMouse10041
Map3k14 (NIK)STE-UniqueSTE6g4yAB10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamideMouse10043
Map3k14 (NIK)STE-UniqueSTE6g4yBA10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamideMouse10047
Map3k14 (NIK)STE-UniqueSTE6g4yBB10-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrolidin-3-yl]ethynyl]-~{n}3-(oxan-4-yl)-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepine-2,3-dicarboxamideMouse10045
Map3k14 (NIK)STE-UniqueSTE6g4zAA5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamideMouse10044
Map3k14 (NIK)STE-UniqueSTE6g4zAB5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamideMouse10046
Map3k14 (NIK)STE-UniqueSTE6g4zBA5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamideMouse10048
Map3k14 (NIK)STE-UniqueSTE6g4zBB5-fluoranyl-1-[4-[2-[(3~{r})-1-methyl-3-oxidanyl-2-oxidanylidene-pyrrol-3-yl]ethynyl]pyridin-2-yl]indazole-3-carboxamideMouse10042
Map3k14 (NIK)STE-UniqueSTE6mynAA(5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamideMouse11525
Map3k14 (NIK)STE-UniqueSTE6mynAB(5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamideMouse11526
Map3k14 (NIK)STE-UniqueSTE6mynBA(5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamideMouse11524
Map3k14 (NIK)STE-UniqueSTE6mynBB(5s,7s)-9-fluoro-10-[(3r)-3-hydroxy-3-(5-methyl-1,2-oxazol-3-yl)but-1-yn-1-yl]-n~3~-methyl-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamideMouse11527
Map3k14 (NIK)STE-UniqueSTE7szrAA1-(3-{[(1r,4r,5s)-4-hydroxy-2-methyl-3-oxo-2-azabicyclo[3.1.0]hexan-4-yl]ethynyl}phenyl)-1h-pyrazolo[3,4-b]pyridine-3-carboxamideMouse14777
Map3k14 (NIK)STE-UniqueSTE7szrAB1-(3-{[(1r,4r,5s)-4-hydroxy-2-methyl-3-oxo-2-azabicyclo[3.1.0]hexan-4-yl]ethynyl}phenyl)-1h-pyrazolo[3,4-b]pyridine-3-carboxamideMouse14776
MAP3K14 (NIK)STE-UniqueSTE4dn5Aphosphothiophosphoric acid-adenylate esterHuman2205
MAP3K14 (NIK)STE-UniqueSTE4dn5Bphosphothiophosphoric acid-adenylate esterHuman2202
MAP3K14 (NIK)STE-UniqueSTE4g3dA-Human2208
MAP3K14 (NIK)STE-UniqueSTE4g3dB-Human2209
MAP3K14 (NIK)STE-UniqueSTE4g3dD-Human2212
MAP3K14 (NIK)STE-UniqueSTE4g3dE-Human2214
MAP3K14 (NIK)STE-UniqueSTE4idtAA11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amineHuman2203
MAP3K14 (NIK)STE-UniqueSTE4idtAB11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amineHuman2204
MAP3K14 (NIK)STE-UniqueSTE4idtBA11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amineHuman2210
MAP3K14 (NIK)STE-UniqueSTE4idtBB11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amineHuman2207
MAP3K14 (NIK)STE-UniqueSTE4idvAA4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-olHuman2211
MAP3K14 (NIK)STE-UniqueSTE4idvBA4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-olHuman2206
MAP3K14 (NIK)STE-UniqueSTE4idvCA4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-olHuman2201
MAP3K14 (NIK)STE-UniqueSTE4idvDA4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-olHuman2213
MAP3K14 (NIK)STE-UniqueSTE6wppAA5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amineHuman12737
MAP3K14 (NIK)STE-UniqueSTE6wppAB5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amineHuman12736
MAP3K14 (NIK)STE-UniqueSTE6wppBA5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amineHuman12738
MAP3K14 (NIK)STE-UniqueSTE6wppBB5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amineHuman12739
MAP3K14 (NIK)STE-UniqueSTE6z1qAAdesf-3r/4076Human12451
MAP3K14 (NIK)STE-UniqueSTE6z1qABdesf-3r/4076Human12454
MAP3K14 (NIK)STE-UniqueSTE6z1qBAdesf-3r/4076Human12455
MAP3K14 (NIK)STE-UniqueSTE6z1qBBdesf-3r/4076Human12449
MAP3K14 (NIK)STE-UniqueSTE6z1tAA4s/3694Human12450
MAP3K14 (NIK)STE-UniqueSTE6z1tAB4s/3694Human12456
MAP3K14 (NIK)STE-UniqueSTE6z1tBA4s/3694Human12453
MAP3K14 (NIK)STE-UniqueSTE6z1tBB4s/3694Human12452
MAP3K20 (ZAK)MLKTKL5hesAAn-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6460
MAP3K20 (ZAK)MLKTKL5hesABn-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6458
MAP3K20 (ZAK)MLKTKL5hesBAn-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6459
MAP3K20 (ZAK)MLKTKL5hesBBn-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamideHuman6457
MAP3K20 (ZAK)MLKTKL5x5oAAn-[2,4-bis(fluoranyl)-3-[2-(3-methoxy-1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-bromanyl-benzenesulfonamideHuman9449
MAP3K20 (ZAK)MLKTKL5x5oABn-[2,4-bis(fluoranyl)-3-[2-(3-methoxy-1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-bromanyl-benzenesulfonamideHuman9448
MAP3K20 (ZAK)MLKTKL6jutA~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]-3-bromanyl-benzenesulfonamideHuman11462
MAP3K20 (ZAK)MLKTKL6juuAA~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamideHuman12167
MAP3K20 (ZAK)MLKTKL6juuAB~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamideHuman12166
MAP3K20 (ZAK)MLKTKL7yawAA~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamideHuman14891
MAP3K20 (ZAK)MLKTKL7yawAB~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamideHuman14893
MAP3K20 (ZAK)MLKTKL7yazAA~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamideHuman14894
MAP3K20 (ZAK)MLKTKL7yazAB~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamideHuman14892
MAP3K21 (MLK4)MLKTKL4uyaAphosphothiophosphoric acid-adenylate esterHuman6126
MAP3K5STE11STE2clqAAstaurosporineHuman4740
MAP3K5STE11STE2clqABstaurosporineHuman4736
MAP3K5STE11STE2clqBAstaurosporineHuman4755
MAP3K5STE11STE2clqBBstaurosporineHuman4732
MAP3K5STE11STE3vw6AA4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHuman4747
MAP3K5STE11STE3vw6AB4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHuman4752
MAP3K5STE11STE3vw6BA4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHuman4738
MAP3K5STE11STE3vw6BB4-tert-butyl-n-[6-(1h-imidazol-1-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHuman4737
MAP3K5STE11STE4bf2AstaurosporineHuman4743
MAP3K5STE11STE4bf2BstaurosporineHuman4745
MAP3K5STE11STE4bhnAA4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHuman4754
MAP3K5STE11STE4bhnAB4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHuman4758
MAP3K5STE11STE4bhnBA4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHuman4734
MAP3K5STE11STE4bhnBB4-tert-butyl-n-[6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyridin-2-yl]benzamideHuman4748
MAP3K5STE11STE4bibAA3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamideHuman4750
MAP3K5STE11STE4bibAB3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamideHuman4759
MAP3K5STE11STE4bibBA3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamideHuman4733
MAP3K5STE11STE4bibBB3-cyano-4-(piperidin-4-yloxy)-1h-indole-7-carboxamideHuman4749
MAP3K5STE11STE4bicAn-(2-aminoethyl)-5-{1h-pyrrolo[2,3-b]pyridin-3-yl}thiophene-2-sulfonamideHuman4739
MAP3K5STE11STE4bicB-Human4741
MAP3K5STE11STE4bidAA5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridineHuman4756
MAP3K5STE11STE4bidAB5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridineHuman4753
MAP3K5STE11STE4bidBA5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridineHuman4742
MAP3K5STE11STE4bidBB5-[(1r)-2-amino-1-phenylethoxy]-2-(furan-3-yl)-3-{1h-pyrrolo[2,3-b]pyridin-3-yl}pyridineHuman4744
MAP3K5STE11STE4bieAAn-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamideHuman4746
MAP3K5STE11STE4bieABn-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamideHuman4757
MAP3K5STE11STE4bieBAn-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamideHuman4735
MAP3K5STE11STE4bieBBn-(2-aminoethyl)-5-{2-methyl-1h-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-sulfonamideHuman4751
MAP3K5STE11STE5uorA6-{[(2s)-4-methylmorpholin-2-yl]methoxy}-2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-oneHuman8107
MAP3K5STE11STE5uorB6-{[(2s)-4-methylmorpholin-2-yl]methoxy}-2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-oneHuman8108
MAP3K5STE11STE5uoxA2-(6-{4-[(2r)-1-hydroxypropan-2-yl]-4h-1,2,4-triazol-3-yl}pyridin-2-yl)-6-[(propan-2-yl)oxy]-2,3-dihydro-1h-isoindol-1-oneHuman8109
MAP3K5STE11STE5uoxB2-(6-{4-[(2r)-1-hydroxypropan-2-yl]-4h-1,2,4-triazol-3-yl}pyridin-2-yl)-6-[(propan-2-yl)oxy]-2,3-dihydro-1h-isoindol-1-oneHuman8106
MAP3K5STE11STE5up3A2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-oneHuman8105
MAP3K5STE11STE5up3B2-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-2,3-dihydro-1h-isoindol-1-oneHuman8110
MAP3K5STE11STE5v19An-(1-ethyl-1h-pyrazol-4-yl)furan-3-carboxamideHuman8025
MAP3K5STE11STE5v19Bn-(1-ethyl-1h-pyrazol-4-yl)furan-3-carboxamideHuman8024
MAP3K5STE11STE5v24AA2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamideHuman8022
MAP3K5STE11STE5v24AB2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamideHuman8021
MAP3K5STE11STE5v24BA2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamideHuman8026
MAP3K5STE11STE5v24BB2-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]-n-(pyridin-2-yl)-1,3-thiazole-4-carboxamideHuman8023
MAP3K5STE11STE5vilA2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamideHuman9512
MAP3K5STE11STE5vilB2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamideHuman9509
MAP3K5STE11STE5vilC2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamideHuman9506
MAP3K5STE11STE5vilD2-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-5-sulfamoylbenzamideHuman9508
MAP3K5STE11STE5vioA4-methoxy-n~1~-methyl-n~3~-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzene-1,3-dicarboxamideHuman9510
MAP3K5STE11STE5vioB4-methoxy-n~1~-methyl-n~3~-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzene-1,3-dicarboxamideHuman9507
MAP3K5STE11STE5vioC-Human9511
MAP3K5STE11STE5vioD4-methoxy-n~1~-methyl-n~3~-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzene-1,3-dicarboxamideHuman9505
MAP3K5STE11STE6e2mAn-[3-(4-methyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamideHuman10575
MAP3K5STE11STE6e2mBn-[3-(4-methyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamideHuman10576
MAP3K5STE11STE6e2nAn-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl][3,4'-bipyridine]-2'-carboxamideHuman10577
MAP3K5STE11STE6e2nBn-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl][3,4'-bipyridine]-2'-carboxamideHuman10572
MAP3K5STE11STE6e2oA4-(4-cyclopropyl-1h-imidazol-1-yl)-n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamideHuman10574
MAP3K5STE11STE6e2oB4-(4-cyclopropyl-1h-imidazol-1-yl)-n-[3-(4-cyclopropyl-4h-1,2,4-triazol-3-yl)phenyl]pyridine-2-carboxamideHuman10573
MAP3K5STE11STE6oytA5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamideHuman11837
MAP3K5STE11STE6oytB5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamideHuman11835
MAP3K5STE11STE6oytC5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamideHuman11840
MAP3K5STE11STE6oytD5-(4-cyclopropyl-1h-imidazol-1-yl)-2-fluoro-4-methyl-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}benzamideHuman11844
MAP3K5STE11STE6oywAA(19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-oneHuman11836
MAP3K5STE11STE6oywAB(19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-oneHuman11842
MAP3K5STE11STE6oywBA(19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-oneHuman11839
MAP3K5STE11STE6oywBB(19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-oneHuman11841
MAP3K5STE11STE6oywCA(19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-oneHuman11838
MAP3K5STE11STE6oywCB(19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-oneHuman11843
MAP3K5STE11STE6oywDA(19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-oneHuman11834
MAP3K5STE11STE6oywDB(19s)-19-methyl-16,17,18,19-tetrahydro-8,4-(azeno)[1,2,4]triazolo[4,3-f][1,6,13]benzoxadiazacyclohexadecin-10(9h)-oneHuman11833
MAP3K5STE11STE6vreAA3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamideHuman12236
MAP3K5STE11STE6vreAB3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamideHuman12233
MAP3K5STE11STE6vreBA3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamideHuman12235
MAP3K5STE11STE6vreBB3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamideHuman12234
MAP3K5STE11STE6xihAA(2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamideHuman12703
MAP3K5STE11STE6xihAB(2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamideHuman12700
MAP3K5STE11STE6xihBA(2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamideHuman12702
MAP3K5STE11STE6xihBB(2r)-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}oxane-2-carboxamideHuman12701
MAP3K5STE11STE7mu7AA3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamideHuman14221
MAP3K5STE11STE7mu7AB3-methoxy-n-{6-[4-(propan-2-yl)-4h-1,2,4-triazol-3-yl]pyridin-2-yl}-1-(pyrazin-2-yl)-1h-pyrazole-4-carboxamideHuman14220
MAP3K7 (TAK1)MLKTKL2evaAAadenosineHuman1884
MAP3K7 (TAK1)MLKTKL2evaABadenosineHuman1882
MAP3K7 (TAK1)MLKTKL2yiyA(1e)-1-[5-tert-butyl-2-(3-fluorophenyl)-1h-pyrazol-3-ylidene]-3-(4-pyridin-3-yloxyphenyl)ureaHuman1890
MAP3K7 (TAK1)MLKTKL4gs6AA(3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman1885
MAP3K7 (TAK1)MLKTKL4gs6AB(3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman1886
MAP3K7 (TAK1)MLKTKL4l3pA2-(1-benzothiophen-7-yl)-4-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[2,3-c]pyridin-7-amineHuman1891
MAP3K7 (TAK1)MLKTKL4l52AA1-(4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}piperidin-1-yl)ethanoneHuman1883
MAP3K7 (TAK1)MLKTKL4l52AB1-(4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}piperidin-1-yl)ethanoneHuman1889
MAP3K7 (TAK1)MLKTKL4l53AAtrans-4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}cyclohexanolHuman1887
MAP3K7 (TAK1)MLKTKL4l53ABtrans-4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}cyclohexanolHuman1892
MAP3K7 (TAK1)MLKTKL4o91An-{4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-4-methyl-3-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)benzamideHuman1888
MAP3K7 (TAK1)MLKTKL5e7rA2-chloro-n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}acetamideHuman7412
MAP3K7 (TAK1)MLKTKL5gjdA1-(4-((1h-pyrrolo[2,3-b]pyridin-4-yl)oxy)phenyl)-3-(5-(4-methylpiperazin-1-yl)naphthalen-2-yl)ureaHuman7263
MAP3K7 (TAK1)MLKTKL5gjfAn-(2-isopropoxy-4-(4-methylpiperazine-1-carbonyl)phenyl)-2-(3-(3-phenylureido)phenyl)thiazole-4-carboxamideHuman7264
MAP3K7 (TAK1)MLKTKL5gjgAn-(2-isopropoxy-4-(4-methylpiperazine-1-carbonyl)phenyl)-2-(3-(phenylcarbamoyl)phenyl)thiazole-4-carboxamideHuman7265
MAP3K7 (TAK1)MLKTKL5j7sAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman7429
MAP3K7 (TAK1)MLKTKL5j8iAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamideHuman7428
MAP3K7 (TAK1)MLKTKL5j9lAn-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamideHuman7426
MAP3K7 (TAK1)MLKTKL5jgaAn-[5-(4-methylpiperazine-1-carbonyl)[1,1'-biphenyl]-2-yl]-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamideHuman6886
MAP3K7 (TAK1)MLKTKL5jgbAn-(2-methoxy-4-{[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamideHuman6885
MAP3K7 (TAK1)MLKTKL5jgdAn-(2-isopropoxy-3-(4-methylpiperazine-1-carbonyl)phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamideHuman6884
MAP3K7 (TAK1)MLKTKL5jh6A2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl prop-2-enoateHuman7427
MAP3K7 (TAK1)MLKTKL5jk3A~{n}-[2-[5-chloranyl-2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]oxyphenyl]prop-2-enamideHuman7430
MAP3K7 (TAK1)MLKTKL5v5nAAn~1~-(1-propyl-1,3-dihydro-2h-benzimidazol-2-ylidene)benzene-1,3-dicarboxamideHuman8350
MAP3K7 (TAK1)MLKTKL5v5nABn~1~-(1-propyl-1,3-dihydro-2h-benzimidazol-2-ylidene)benzene-1,3-dicarboxamideHuman8351
MAP3K7 (TAK1)MLKTKL7nthAA2-[[5-[[2-[bis(fluoranyl)methoxy]phenyl]methyl-[(2~{r})-1-(methylamino)-1-oxidanylidene-propan-2-yl]carbamoyl]-1~{h}-imidazol-2-yl]carbonyl]isoindole-5-carboxamideHuman13456
MAP3K7 (TAK1)MLKTKL7nthAB2-[[5-[[2-[bis(fluoranyl)methoxy]phenyl]methyl-[(2~{r})-1-(methylamino)-1-oxidanylidene-propan-2-yl]carbamoyl]-1~{h}-imidazol-2-yl]carbonyl]isoindole-5-carboxamideHuman13458
MAP3K7 (TAK1)MLKTKL7ntiAA~{n}-[[2-[bis(fluoranyl)methoxy]phenyl]methyl]-~{n}-[2-(methylamino)-2-oxidanylidene-ethyl]-2-pyrrolidin-1-ylcarbonyl-1~{h}-imidazole-4-carboxamideHuman13459
MAP3K7 (TAK1)MLKTKL7ntiAB~{n}-[[2-[bis(fluoranyl)methoxy]phenyl]methyl]-~{n}-[2-(methylamino)-2-oxidanylidene-ethyl]-2-pyrrolidin-1-ylcarbonyl-1~{h}-imidazole-4-carboxamideHuman13457
MAP3K7 (TAK1)MLKTKL8gw3A-Human14877
MAP3K8 (COT)STE-UniqueSTE4y83A5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman428
MAP3K8 (COT)STE-UniqueSTE4y83B5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman426
MAP3K8 (COT)STE-UniqueSTE4y83C5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman425
MAP3K8 (COT)STE-UniqueSTE4y85A5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amineHuman427
MAP3K8 (COT)STE-UniqueSTE4y85B5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amineHuman429
MAP3K8 (COT)STE-UniqueSTE4y85C5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amineHuman424
MAP3K8 (COT)STE-UniqueSTE5iu2AAn-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amineHuman6980
MAP3K8 (COT)STE-UniqueSTE5iu2ABn-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amineHuman6981
MAP3K8 (COT)STE-UniqueSTE5iu2BAn-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amineHuman6979
MAP3K8 (COT)STE-UniqueSTE5iu2BBn-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amineHuman6978
MAP3K9 (MLK1)MLKTKL3dtcA12-(2-hydroxyethyl)-2-(1-methylethoxy)-13,14-dihydronaphtho[2,1-a]pyrrolo[3,4-c]carbazol-5(12h)-oneHuman3839
MAP3K9 (MLK1)MLKTKL4uy9AA-Human6127
MAP3K9 (MLK1)MLKTKL4uy9AB-Human6128
MAP3K9 (MLK1)MLKTKL4uy9BA-Human6129
MAP3K9 (MLK1)MLKTKL4uy9BB-Human6130
MAP4K1 (HPK1)STE20STE6cqdAphosphoaminophosphonic acid-adenylate esterHuman10803
MAP4K1 (HPK1)STE20STE6cqdBphosphoaminophosphonic acid-adenylate esterHuman10801
MAP4K1 (HPK1)STE20STE6cqeAA-Human10802
MAP4K1 (HPK1)STE20STE6cqeAB-Human10804
MAP4K1 (HPK1)STE20STE6cqeBA-Human10805
MAP4K1 (HPK1)STE20STE6cqeBB-Human10800
MAP4K1 (HPK1)STE20STE6cqfAn-{2-(3,3-difluoropyrrolidin-1-yl)-6-[(3r)-pyrrolidin-3-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-pyrazolo[4,3-c]pyridin-6-amineHuman10806
MAP4K1 (HPK1)STE20STE6nfyAAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman11075
MAP4K1 (HPK1)STE20STE6nfyABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman11072
MAP4K1 (HPK1)STE20STE6nfyBAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman11076
MAP4K1 (HPK1)STE20STE6nfyBBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman11077
MAP4K1 (HPK1)STE20STE6nfzAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman11078
MAP4K1 (HPK1)STE20STE6nfzBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman11074
MAP4K1 (HPK1)STE20STE6ng0An-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman11071
MAP4K1 (HPK1)STE20STE6ng0Bn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman11073
MAP4K1 (HPK1)STE20STE7kacA5-{[4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-5-(1,3,4-oxadiazol-2-yl)pyrimidin-2-yl]amino}-3,3-dimethyl-2-benzofuran-1(3h)-oneHuman13231
MAP4K1 (HPK1)STE20STE7kacB5-{[4-{[(1s)-2-hydroxy-1-phenylethyl]amino}-5-(1,3,4-oxadiazol-2-yl)pyrimidin-2-yl]amino}-3,3-dimethyl-2-benzofuran-1(3h)-oneHuman13230
MAP4K1 (HPK1)STE20STE7l24AA6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridineHuman13416
MAP4K1 (HPK1)STE20STE7l24AB6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridineHuman13418
MAP4K1 (HPK1)STE20STE7l24BA6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridineHuman13422
MAP4K1 (HPK1)STE20STE7l24BB6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridineHuman13426
MAP4K1 (HPK1)STE20STE7l24CA6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridineHuman13423
MAP4K1 (HPK1)STE20STE7l24CB6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridineHuman13417
MAP4K1 (HPK1)STE20STE7l24DA6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridineHuman13415
MAP4K1 (HPK1)STE20STE7l24DB6-(2-fluoro-6-methoxyphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrazolo[4,3-c]pyridineHuman13421
MAP4K1 (HPK1)STE20STE7l25AA6-(2-fluoro-6-methoxyphenyl)-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[4,3-c]pyridineHuman13428
MAP4K1 (HPK1)STE20STE7l25AB6-(2-fluoro-6-methoxyphenyl)-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[4,3-c]pyridineHuman13424
MAP4K1 (HPK1)STE20STE7l25BA6-(2-fluoro-6-methoxyphenyl)-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[4,3-c]pyridineHuman13413
MAP4K1 (HPK1)STE20STE7l25BB6-(2-fluoro-6-methoxyphenyl)-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[4,3-c]pyridineHuman13425
MAP4K1 (HPK1)STE20STE7l26AA6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrileHuman13427
MAP4K1 (HPK1)STE20STE7l26AB6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrileHuman13429
MAP4K1 (HPK1)STE20STE7l26BA6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrileHuman13430
MAP4K1 (HPK1)STE20STE7l26BB6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrileHuman13414
MAP4K1 (HPK1)STE20STE7l26CA6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrileHuman13419
MAP4K1 (HPK1)STE20STE7l26CB6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrileHuman13420
MAP4K1 (HPK1)STE20STE7l26DA6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrileHuman13431
MAP4K1 (HPK1)STE20STE7l26DB6-(2-fluoro-6-methylphenyl)-1-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-5-carbonitrileHuman13432
MAP4K1 (HPK1)STE20STE7m0kAA4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13480
MAP4K1 (HPK1)STE20STE7m0kAB4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13481
MAP4K1 (HPK1)STE20STE7m0kBA4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13476
MAP4K1 (HPK1)STE20STE7m0kBB4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13470
MAP4K1 (HPK1)STE20STE7m0kCA4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13473
MAP4K1 (HPK1)STE20STE7m0kCB4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13474
MAP4K1 (HPK1)STE20STE7m0kDA4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13479
MAP4K1 (HPK1)STE20STE7m0kDB4-anilino-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13471
MAP4K1 (HPK1)STE20STE7m0lA4-(2-bromoanilino)-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13475
MAP4K1 (HPK1)STE20STE7m0lB4-(2-bromoanilino)-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13466
MAP4K1 (HPK1)STE20STE7m0lC4-(2-bromoanilino)-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13478
MAP4K1 (HPK1)STE20STE7m0lD4-(2-bromoanilino)-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13468
MAP4K1 (HPK1)STE20STE7m0mAA4-[2-fluoro-6-(trifluoromethyl)anilino]-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13469
MAP4K1 (HPK1)STE20STE7m0mAB4-[2-fluoro-6-(trifluoromethyl)anilino]-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13477
MAP4K1 (HPK1)STE20STE7m0mBA4-[2-fluoro-6-(trifluoromethyl)anilino]-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13467
MAP4K1 (HPK1)STE20STE7m0mBB4-[2-fluoro-6-(trifluoromethyl)anilino]-2-[(6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino]pyrimidine-5-carboxamideHuman13472
MAP4K1 (HPK1)STE20STE7r9lA2-amino-n,n-dimethyl-5-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamideHuman14026
MAP4K1 (HPK1)STE20STE7r9nAAn-{2-(3,3-difluoropyrrolidin-1-yl)-6-[(3r)-pyrrolidin-3-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-pyrazolo[4,3-c]pyridin-6-amineHuman14025
MAP4K1 (HPK1)STE20STE7r9nABn-{2-(3,3-difluoropyrrolidin-1-yl)-6-[(3r)-pyrrolidin-3-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1h-pyrazolo[4,3-c]pyridin-6-amineHuman14023
MAP4K1 (HPK1)STE20STE7r9pA6-amino-2-fluoro-n,n-dimethyl-3-(4'-methylspiro[cyclopropane-1,3'-pyrrolo[2,3-b]pyridin]-5'-yl)benzamideHuman14022
MAP4K1 (HPK1)STE20STE7r9tA6-amino-3-[(1s,3r)-4'-chloro-3-hydroxy-1',2'-dihydrospiro[cyclopentane-1,3'-pyrrolo[2,3-b]pyridin]-5'-yl]-2-fluoro-n,n-dimethylbenzamideHuman14024
MAP4K1 (HPK1)STE20STE7siuA6-[(5r)-5-benzamidocyclohex-1-en-1-yl]-3-[(1-methyl-1h-pyrazol-4-yl)amino]pyrazine-2-carboxamideHuman14117
MAP4K1 (HPK1)STE20STE8cdwAA~{n}-[4-(1-methylpiperidin-4-yl)phenyl]-7-(1-methylpyrazol-4-yl)quinazolin-2-amineHuman14896
MAP4K1 (HPK1)STE20STE8cdwAB~{n}-[4-(1-methylpiperidin-4-yl)phenyl]-7-(1-methylpyrazol-4-yl)quinazolin-2-amineHuman14895
MAP4K1 (HPK1)STE20STE8cijA2-[[8-azanyl-7-fluoranyl-6-(8-methyl-2,3-dihydro-1~{h}-pyrido[2,3-b][1,4]oxazin-7-yl)isoquinolin-3-yl]amino]-6-propan-2-yl-5,8-dihydro-4~{h}-pyrazolo[1,5-d][1,4]diazepin-7-oneHuman14897
MAP4K1 (HPK1)STE20STE8fh4AA(3p)-3-[6-chloro-4-(9-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrileHuman14688
MAP4K1 (HPK1)STE20STE8fh4AB(3p)-3-[6-chloro-4-(9-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrileHuman14690
MAP4K1 (HPK1)STE20STE8fjzA(3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrileHuman14691
MAP4K1 (HPK1)STE20STE8fkoA(3p)-3-{4-[(2s,5r)-5-amino-2-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrileHuman14689
MAP4K3 (KHS2)STE20STE5j5tA5-[2-(piperidin-4-yl)-1,3-thiazol-5-yl]-3-[(pyridin-4-yl)methoxy]pyridin-2-amineHuman7133
MAP4K4 (HGK)STE20STE4oboAA6-(3-chlorophenyl)quinazolin-4-amineHuman2746
MAP4K4 (HGK)STE20STE4oboAB6-(3-chlorophenyl)quinazolin-4-amineHuman2744
MAP4K4 (HGK)STE20STE4oboBA-Human2762
MAP4K4 (HGK)STE20STE4oboBB-Human2748
MAP4K4 (HGK)STE20STE4obpAA6-(2-fluoropyridin-4-yl)pyrido[3,2-d]pyrimidin-4-amineHuman2750
MAP4K4 (HGK)STE20STE4obpAB6-(2-fluoropyridin-4-yl)pyrido[3,2-d]pyrimidin-4-amineHuman2761
MAP4K4 (HGK)STE20STE4obpBA-Human2754
MAP4K4 (HGK)STE20STE4obpBB-Human2757
MAP4K4 (HGK)STE20STE4obqAAn-[3-(4-aminoquinazolin-6-yl)-5-fluorophenyl]-2-(pyrrolidin-1-yl)acetamideHuman2758
MAP4K4 (HGK)STE20STE4obqABn-[3-(4-aminoquinazolin-6-yl)-5-fluorophenyl]-2-(pyrrolidin-1-yl)acetamideHuman2755
MAP4K4 (HGK)STE20STE4obqBA-Human2736
MAP4K4 (HGK)STE20STE4obqBB-Human2742
MAP4K4 (HGK)STE20STE4rvtAA3-hexanoyl-4-hydroxy-5-(4-hydroxyphenyl)pyridin-2(1h)-oneHuman2751
MAP4K4 (HGK)STE20STE4rvtAB3-hexanoyl-4-hydroxy-5-(4-hydroxyphenyl)pyridin-2(1h)-oneHuman2760
MAP4K4 (HGK)STE20STE4rvtBA-Human2749
MAP4K4 (HGK)STE20STE4rvtBB-Human2739
MAP4K4 (HGK)STE20STE4u3yAA-Human6339
MAP4K4 (HGK)STE20STE4u3yAB-Human6340
MAP4K4 (HGK)STE20STE4u3yBA-Human6344
MAP4K4 (HGK)STE20STE4u3yBB-Human6343
MAP4K4 (HGK)STE20STE4u3zAA-Human6333
MAP4K4 (HGK)STE20STE4u3zAB-Human6326
MAP4K4 (HGK)STE20STE4u3zBA-Human6336
MAP4K4 (HGK)STE20STE4u3zBB-Human6327
MAP4K4 (HGK)STE20STE4u40AAphosphoaminophosphonic acid-adenylate esterHuman6332
MAP4K4 (HGK)STE20STE4u40ABphosphoaminophosphonic acid-adenylate esterHuman6329
MAP4K4 (HGK)STE20STE4u40BA-Human6342
MAP4K4 (HGK)STE20STE4u40BB-Human6331
MAP4K4 (HGK)STE20STE4u41AA6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amineHuman6338
MAP4K4 (HGK)STE20STE4u41AB6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amineHuman6334
MAP4K4 (HGK)STE20STE4u41BA-Human6341
MAP4K4 (HGK)STE20STE4u41BB-Human6328
MAP4K4 (HGK)STE20STE4u42AA6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amineHuman6335
MAP4K4 (HGK)STE20STE4u42AB6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amineHuman6337
MAP4K4 (HGK)STE20STE4u42BA6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amineHuman6330
MAP4K4 (HGK)STE20STE4u42BB6-[(3s)-3-(4-methyl-1h-pyrazol-3-yl)piperidin-1-yl]pyrido[3,2-d]pyrimidin-4-amineHuman6325
MAP4K4 (HGK)STE20STE4u43AAn-(pyridin-3-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman2763
MAP4K4 (HGK)STE20STE4u43ABn-(pyridin-3-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman2738
MAP4K4 (HGK)STE20STE4u43BA-Human2753
MAP4K4 (HGK)STE20STE4u43BB-Human2743
MAP4K4 (HGK)STE20STE4u44AA6-phenyl-n-(pyridin-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman2752
MAP4K4 (HGK)STE20STE4u44AB6-phenyl-n-(pyridin-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman2745
MAP4K4 (HGK)STE20STE4u44BA-Human2737
MAP4K4 (HGK)STE20STE4u44BB-Human2740
MAP4K4 (HGK)STE20STE4u45AA6-(1h-pyrazol-4-yl)-n-(pyridin-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman2747
MAP4K4 (HGK)STE20STE4u45AB6-(1h-pyrazol-4-yl)-n-(pyridin-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman2759
MAP4K4 (HGK)STE20STE4u45BA-Human2741
MAP4K4 (HGK)STE20STE4u45BB-Human2756
MAP4K4 (HGK)STE20STE4zk5A8-amino-n-[1-(cyclopropylcarbonyl)azetidin-3-yl]-2-(3-fluorophenyl)-1,7-naphthyridine-5-carboxamideHuman6015
MAP4K4 (HGK)STE20STE4zk5B-Human6014
MAP4K4 (HGK)STE20STE4zp5A4-[5-(4-chlorophenyl)-1,3-oxazol-2-yl]benzamideHuman7091
MAP4K4 (HGK)STE20STE4zp5B-Human7090
MAP4K4 (HGK)STE20STE5di1A4-{6-amino-5-[4-(methylsulfonyl)phenyl]pyridin-3-yl}phenolHuman6354
MAP4K4 (HGK)STE20STE5di1B-Human6353
MAP4K4 (HGK)STE20STE5j95A1-{4-[6-amino-5-(4-chlorophenyl)pyridin-3-yl]phenyl}cyclopentane-1-carboxylic acidHuman7999
MAP4K4 (HGK)STE20STE5j95B-Human8000
MAP4K4 (HGK)STE20STE5w5qAA(5s,7s)-n~3~-methyl-10-[3-methyl-3-(5-methyl-1,3-oxazol-2-yl)but-1-yn-1-yl]-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamideHuman10008
MAP4K4 (HGK)STE20STE5w5qAB(5s,7s)-n~3~-methyl-10-[3-methyl-3-(5-methyl-1,3-oxazol-2-yl)but-1-yn-1-yl]-6,7-dihydro-5h-5,7-methanoimidazo[2,1-a][2]benzazepine-2,3-dicarboxamideHuman10005
MAP4K4 (HGK)STE20STE5w5qBA-Human10007
MAP4K4 (HGK)STE20STE5w5qBB-Human10006
MAPK1 (Erk2)MAPKCMGC1pmeA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman2583
MAPK1 (Erk2)MAPKCMGC1tvoA5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman2581
MAPK1 (Erk2)MAPKCMGC1wzyA1-allyl-5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman2618
MAPK1 (Erk2)MAPKCMGC2ojgAn,n-dimethyl-4-(4-phenyl-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamideHuman2603
MAPK1 (Erk2)MAPKCMGC2ojiAn-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamideHuman2570
MAPK1 (Erk2)MAPKCMGC2ojjA(s)-n-(1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamideHuman2612
MAPK1 (Erk2)MAPKCMGC2y9qAAphosphoaminophosphonic acid-adenylate esterHuman2626
MAPK1 (Erk2)MAPKCMGC2y9qABphosphoaminophosphonic acid-adenylate esterHuman2556
MAPK1 (Erk2)MAPKCMGC2y9qACphosphoaminophosphonic acid-adenylate esterHuman2567
MAPK1 (Erk2)MAPKCMGC3i5zAn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHuman2579
MAPK1 (Erk2)MAPKCMGC3i60A4-{2-[(2-chlorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-phenylethyl]-1h-pyrrole-2-carboxamideHuman2584
MAPK1 (Erk2)MAPKCMGC3sa0AAnorathyriolHuman2596
MAPK1 (Erk2)MAPKCMGC3sa0ABnorathyriolHuman2557
MAPK1 (Erk2)MAPKCMGC3teiAphosphoaminophosphonic acid-adenylate esterHuman2608
MAPK1 (Erk2)MAPKCMGC3w55A(3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman2573
MAPK1 (Erk2)MAPKCMGC4fmqAAphosphoaminophosphonic acid-adenylate esterHuman2604
MAPK1 (Erk2)MAPKCMGC4fmqABphosphoaminophosphonic acid-adenylate esterHuman2619
MAPK1 (Erk2)MAPKCMGC4fuxAtrans-4-{[4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)pyrimidin-2-yl]amino}cyclohexanolHuman2568
MAPK1 (Erk2)MAPKCMGC4fuyAA{4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanoneHuman2622
MAPK1 (Erk2)MAPKCMGC4fuyAB{4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanoneHuman2587
MAPK1 (Erk2)MAPKCMGC4fv0AAn-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amineHuman2562
MAPK1 (Erk2)MAPKCMGC4fv0ABn-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amineHuman2599
MAPK1 (Erk2)MAPKCMGC4fv1AAn-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamideHuman2594
MAPK1 (Erk2)MAPKCMGC4fv1ABn-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamideHuman2613
MAPK1 (Erk2)MAPKCMGC4fv2AA4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHuman2592
MAPK1 (Erk2)MAPKCMGC4fv2AB4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHuman2571
MAPK1 (Erk2)MAPKCMGC4fv3AAethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman2617
MAPK1 (Erk2)MAPKCMGC4fv3ABethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman2580
MAPK1 (Erk2)MAPKCMGC4fv4AA9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrileHuman2623
MAPK1 (Erk2)MAPKCMGC4fv4AB9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrileHuman2558
MAPK1 (Erk2)MAPKCMGC4fv5An-[(1s)-2-hydroxy-1-phenylethyl]-4-(5-methyl-2-phenylpyrimidin-4-yl)-1h-pyrrole-2-carboxamideHuman2598
MAPK1 (Erk2)MAPKCMGC4fv6An-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-4-(2-{[(2s)-1-hydroxybutan-2-yl]amino}-5-methylpyrimidin-4-yl)-1h-pyrrole-2-carboxamideHuman2551
MAPK1 (Erk2)MAPKCMGC4fv7AA4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrileHuman2572
MAPK1 (Erk2)MAPKCMGC4fv7AB4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrileHuman2614
MAPK1 (Erk2)MAPKCMGC4fv8AA6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-oneHuman2625
MAPK1 (Erk2)MAPKCMGC4fv8AB6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-oneHuman2601
MAPK1 (Erk2)MAPKCMGC4fv9AA3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman2582
MAPK1 (Erk2)MAPKCMGC4fv9AB3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman2552
MAPK1 (Erk2)MAPKCMGC4g6nAA3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazoleHuman2609
MAPK1 (Erk2)MAPKCMGC4g6nAB3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazoleHuman2593
MAPK1 (Erk2)MAPKCMGC4g6oA4-{4-[4-(aminomethyl)-3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHuman2565
MAPK1 (Erk2)MAPKCMGC4h3pAphosphoaminophosphonic acid-adenylate esterHuman2624
MAPK1 (Erk2)MAPKCMGC4h3pDphosphoaminophosphonic acid-adenylate esterHuman2575
MAPK1 (Erk2)MAPKCMGC4h3qAphosphoaminophosphonic acid-adenylate esterHuman2611
MAPK1 (Erk2)MAPKCMGC4iz5Aadenosine-5'-diphosphateHuman2554
MAPK1 (Erk2)MAPKCMGC4iz5Badenosine-5'-diphosphateHuman2600
MAPK1 (Erk2)MAPKCMGC4iz5Cadenosine-5'-diphosphateHuman2595
MAPK1 (Erk2)MAPKCMGC4iz5Dadenosine-5'-diphosphateHuman2578
MAPK1 (Erk2)MAPKCMGC4iz7AA-Human2615
MAPK1 (Erk2)MAPKCMGC4iz7AB-Human2577
MAPK1 (Erk2)MAPKCMGC4iz7CA-Human2569
MAPK1 (Erk2)MAPKCMGC4iz7CB-Human2597
MAPK1 (Erk2)MAPKCMGC4izaAA-Human2586
MAPK1 (Erk2)MAPKCMGC4izaAB-Human2607
MAPK1 (Erk2)MAPKCMGC4izaCA-Human2588
MAPK1 (Erk2)MAPKCMGC4izaCB-Human2627
MAPK1 (Erk2)MAPKCMGC4n0sAAcaffeic acidHuman2589
MAPK1 (Erk2)MAPKCMGC4n0sABcaffeic acidHuman2555
MAPK1 (Erk2)MAPKCMGC4nifBAphosphoaminophosphonic acid-adenylate esterHuman2585
MAPK1 (Erk2)MAPKCMGC4nifBBphosphoaminophosphonic acid-adenylate esterHuman2566
MAPK1 (Erk2)MAPKCMGC4nifEAphosphoaminophosphonic acid-adenylate esterHuman2621
MAPK1 (Erk2)MAPKCMGC4nifEBphosphoaminophosphonic acid-adenylate esterHuman2591
MAPK1 (Erk2)MAPKCMGC4o6eAAn-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamideHuman2559
MAPK1 (Erk2)MAPKCMGC4o6eABn-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamideHuman2553
MAPK1 (Erk2)MAPKCMGC4qp1An-benzyl-9h-purin-6-amineHuman6092
MAPK1 (Erk2)MAPKCMGC4qp1Bn-benzyl-9h-purin-6-amineHuman6080
MAPK1 (Erk2)MAPKCMGC4qp2A5-chloro-1,3-benzoxazol-2-amineHuman6078
MAPK1 (Erk2)MAPKCMGC4qp2B-Human6081
MAPK1 (Erk2)MAPKCMGC4qp3A(2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-olHuman6084
MAPK1 (Erk2)MAPKCMGC4qp3B(2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-olHuman6079
MAPK1 (Erk2)MAPKCMGC4qp4AAn-cyclohexyl-9h-purin-6-amineHuman6088
MAPK1 (Erk2)MAPKCMGC4qp4ABn-cyclohexyl-9h-purin-6-amineHuman6075
MAPK1 (Erk2)MAPKCMGC4qp4BAn-cyclohexyl-9h-purin-6-amineHuman6086
MAPK1 (Erk2)MAPKCMGC4qp4BBn-cyclohexyl-9h-purin-6-amineHuman6083
MAPK1 (Erk2)MAPKCMGC4qp6A5h-pyrrolo[2,3-b]pyrazineHuman6089
MAPK1 (Erk2)MAPKCMGC4qp6B5h-pyrrolo[2,3-b]pyrazineHuman6091
MAPK1 (Erk2)MAPKCMGC4qp7A2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6082
MAPK1 (Erk2)MAPKCMGC4qp7B2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6093
MAPK1 (Erk2)MAPKCMGC4qp8A2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6087
MAPK1 (Erk2)MAPKCMGC4qp8B2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6076
MAPK1 (Erk2)MAPKCMGC4qp9A7-(1-propyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6085
MAPK1 (Erk2)MAPKCMGC4qpaA7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6077
MAPK1 (Erk2)MAPKCMGC4qpaB7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6090
MAPK1 (Erk2)MAPKCMGC4qtaAA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman2602
MAPK1 (Erk2)MAPKCMGC4qtaAB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman2576
MAPK1 (Erk2)MAPKCMGC4qteAA4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamideHuman2590
MAPK1 (Erk2)MAPKCMGC4qteAB4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamideHuman2564
MAPK1 (Erk2)MAPKCMGC4xj0A1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-oneHuman6048
MAPK1 (Erk2)MAPKCMGC4xj0B1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-oneHuman6049
MAPK1 (Erk2)MAPKCMGC4zxtAAcatecholHuman6654
MAPK1 (Erk2)MAPKCMGC4zxtABcatecholHuman6653
MAPK1 (Erk2)MAPKCMGC4zzmA7-ethylsulfonyl-n-(oxan-4-yl)-6,8-dihydro-5h-pyrido[3,4-d]pyrimidin-2-amineHuman2616
MAPK1 (Erk2)MAPKCMGC4zznAA2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamideHuman2605
MAPK1 (Erk2)MAPKCMGC4zznAB2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamideHuman2610
MAPK1 (Erk2)MAPKCMGC4zzoAAn-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamideHuman2620
MAPK1 (Erk2)MAPKCMGC4zzoABn-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamideHuman2606
MAPK1 (Erk2)MAPKCMGC5ax3A(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman6398
MAPK1 (Erk2)MAPKCMGC5bueA1-benzyl-4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-oneHuman2574
MAPK1 (Erk2)MAPKCMGC5buiA3-(4-fluorophenyl)-5-(pyridin-2-yl)-4,5,6,7-tetrahydro-2h-pyrazolo[4,3-c]pyridineHuman2563
MAPK1 (Erk2)MAPKCMGC5bujAA4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-oneHuman2560
MAPK1 (Erk2)MAPKCMGC5bujAB4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-oneHuman2561
MAPK1 (Erk2)MAPKCMGC5bvdAA2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-oneHuman6030
MAPK1 (Erk2)MAPKCMGC5bvdAB2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-oneHuman6028
MAPK1 (Erk2)MAPKCMGC5bveAA2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6029
MAPK1 (Erk2)MAPKCMGC5bveAB2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6026
MAPK1 (Erk2)MAPKCMGC5bvfAA2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6031
MAPK1 (Erk2)MAPKCMGC5bvfAB2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6027
MAPK1 (Erk2)MAPKCMGC5k4iA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6744
MAPK1 (Erk2)MAPKCMGC5lcjAA[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman6833
MAPK1 (Erk2)MAPKCMGC5lcjAB[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman6834
MAPK1 (Erk2)MAPKCMGC5lckAA~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamideHuman6835
MAPK1 (Erk2)MAPKCMGC5lckAB~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamideHuman6836
MAPK1 (Erk2)MAPKCMGC5nguA2-[2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneHuman7991
MAPK1 (Erk2)MAPKCMGC5nhfA2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-5-(phenylmethyl)-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7997
MAPK1 (Erk2)MAPKCMGC5nhhA5-(2-methoxyethyl)-2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7996
MAPK1 (Erk2)MAPKCMGC5nhjA5-(2-methoxyethyl)-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7994
MAPK1 (Erk2)MAPKCMGC5nhlA(6~{r})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7992
MAPK1 (Erk2)MAPKCMGC5nhoA(6~{s})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7993
MAPK1 (Erk2)MAPKCMGC5nhpA5-(2-methoxyethyl)-1-methyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydropyrrolo[3,2-c]pyridin-4-oneHuman7998
MAPK1 (Erk2)MAPKCMGC5nhvA7-[2-(oxan-4-ylamino)pyrimidin-4-yl]-3,4-dihydro-2~{h}-pyrrolo[1,2-a]pyrazin-1-oneHuman7995
MAPK1 (Erk2)MAPKCMGC5v60AAphosphomethylphosphonic acid adenylate esterHuman8261
MAPK1 (Erk2)MAPKCMGC5v60ABphosphomethylphosphonic acid adenylate esterHuman8263
MAPK1 (Erk2)MAPKCMGC5v61AA-Human8265
MAPK1 (Erk2)MAPKCMGC5v61AB-Human8266
MAPK1 (Erk2)MAPKCMGC5v62AA5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman8264
MAPK1 (Erk2)MAPKCMGC5v62AB5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman8262
MAPK1 (Erk2)MAPKCMGC5wp1AA5,7-dihydroxy-4h-1-benzopyran-4-oneHuman10441
MAPK1 (Erk2)MAPKCMGC5wp1AB5,7-dihydroxy-4h-1-benzopyran-4-oneHuman10440
MAPK1 (Erk2)MAPKCMGC6d5yA-Human10939
MAPK1 (Erk2)MAPKCMGC6dmgAA-Human10811
MAPK1 (Erk2)MAPKCMGC6dmgABethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman10810
MAPK1 (Erk2)MAPKCMGC6dmgACethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman10809
MAPK1 (Erk2)MAPKCMGC6g54AAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10938
MAPK1 (Erk2)MAPKCMGC6g54ABn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10937
MAPK1 (Erk2)MAPKCMGC6g8xAA4-chloranyl-1~{h}-indazol-3-amineHuman9957
MAPK1 (Erk2)MAPKCMGC6g8xAB4-chloranyl-1~{h}-indazol-3-amineHuman9954
MAPK1 (Erk2)MAPKCMGC6g91AA5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amineHuman9965
MAPK1 (Erk2)MAPKCMGC6g91AB5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amineHuman9956
MAPK1 (Erk2)MAPKCMGC6g92AA~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amineHuman11409
MAPK1 (Erk2)MAPKCMGC6g92AB~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amineHuman11411
MAPK1 (Erk2)MAPKCMGC6g93AA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-oneHuman9955
MAPK1 (Erk2)MAPKCMGC6g93AB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-oneHuman9959
MAPK1 (Erk2)MAPKCMGC6g97AA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-oneHuman9960
MAPK1 (Erk2)MAPKCMGC6g97AB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-oneHuman9970
MAPK1 (Erk2)MAPKCMGC6g9aAA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-oneHuman11408
MAPK1 (Erk2)MAPKCMGC6g9aAB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-oneHuman11412
MAPK1 (Erk2)MAPKCMGC6g9dAA~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamideHuman9972
MAPK1 (Erk2)MAPKCMGC6g9dAB~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamideHuman9953
MAPK1 (Erk2)MAPKCMGC6g9hAA~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamideHuman9971
MAPK1 (Erk2)MAPKCMGC6g9hAB~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamideHuman9958
MAPK1 (Erk2)MAPKCMGC6g9jAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamideHuman9952
MAPK1 (Erk2)MAPKCMGC6g9jAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamideHuman9949
MAPK1 (Erk2)MAPKCMGC6g9kAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamideHuman9966
MAPK1 (Erk2)MAPKCMGC6g9kAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamideHuman9947
MAPK1 (Erk2)MAPKCMGC6g9mAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamideHuman9964
MAPK1 (Erk2)MAPKCMGC6g9mAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamideHuman9944
MAPK1 (Erk2)MAPKCMGC6g9nAA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamideHuman11410
MAPK1 (Erk2)MAPKCMGC6g9nAB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamideHuman11413
MAPK1 (Erk2)MAPKCMGC6gdmAA(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamideHuman9968
MAPK1 (Erk2)MAPKCMGC6gdmAB(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamideHuman9946
MAPK1 (Erk2)MAPKCMGC6gdqAA4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamideHuman9948
MAPK1 (Erk2)MAPKCMGC6gdqAB4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamideHuman9973
MAPK1 (Erk2)MAPKCMGC6ge0AA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamideHuman9950
MAPK1 (Erk2)MAPKCMGC6ge0AB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamideHuman9961
MAPK1 (Erk2)MAPKCMGC6gjbAA[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman10832
MAPK1 (Erk2)MAPKCMGC6gjbAB[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman10831
MAPK1 (Erk2)MAPKCMGC6gjdAAcyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamateHuman10829
MAPK1 (Erk2)MAPKCMGC6gjdABcyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamateHuman10830
MAPK1 (Erk2)MAPKCMGC6nbsAA-Human11510
MAPK1 (Erk2)MAPKCMGC6nbsAB-Human11508
MAPK1 (Erk2)MAPKCMGC6opgAphosphoaminophosphonic acid-adenylate esterHuman11507
MAPK1 (Erk2)MAPKCMGC6ophA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman11509
MAPK1 (Erk2)MAPKCMGC6opiA(3r)-n-[3-(2-cyclopropylpyridin-4-yl)-1h-indazol-5-yl]-3-(methoxymethyl)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]-3,6-dihydropyridin-1(2h)-yl}ethyl)pyrrolidine-3-carboxamideHuman11511
MAPK1 (Erk2)MAPKCMGC6q7kA1h-imidazol-2-amineHuman10985
MAPK1 (Erk2)MAPKCMGC6q7sAA-Human11349
MAPK1 (Erk2)MAPKCMGC6q7sAB-Human11343
MAPK1 (Erk2)MAPKCMGC6q7tAA1,2-oxazol-3-amineHuman11350
MAPK1 (Erk2)MAPKCMGC6q7tAB1,2-oxazol-3-amineHuman11347
MAPK1 (Erk2)MAPKCMGC6qa1AApyridin-2-amineHuman11352
MAPK1 (Erk2)MAPKCMGC6qa1ABpyridin-2-amineHuman11346
MAPK1 (Erk2)MAPKCMGC6qa3AApyrazoleHuman11353
MAPK1 (Erk2)MAPKCMGC6qa3ABpyrazoleHuman11345
MAPK1 (Erk2)MAPKCMGC6qa4AA1~{h}-pyridin-2-oneHuman11344
MAPK1 (Erk2)MAPKCMGC6qa4AB1~{h}-pyridin-2-oneHuman11351
MAPK1 (Erk2)MAPKCMGC6qagAA1~{h}-1,2,3-triazoleHuman10988
MAPK1 (Erk2)MAPKCMGC6qagAB1~{h}-1,2,3-triazoleHuman10982
MAPK1 (Erk2)MAPKCMGC6qahAA1-azanylpropylideneazaniumHuman11354
MAPK1 (Erk2)MAPKCMGC6qahAB1-azanylpropylideneazaniumHuman11348
MAPK1 (Erk2)MAPKCMGC6qalAA1,1-bis(oxidanylidene)thietan-3-olHuman10987
MAPK1 (Erk2)MAPKCMGC6qalAB1,1-bis(oxidanylidene)thietan-3-olHuman10981
MAPK1 (Erk2)MAPKCMGC6qaqAAthiophen-3-ylmethylazaniumHuman10983
MAPK1 (Erk2)MAPKCMGC6qaqABthiophen-3-ylmethylazaniumHuman10989
MAPK1 (Erk2)MAPKCMGC6qawAA[1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazaniumHuman10984
MAPK1 (Erk2)MAPKCMGC6qawAB[1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazaniumHuman10986
MAPK1 (Erk2)MAPKCMGC6rfoA-Human12341
MAPK1 (Erk2)MAPKCMGC6rq4AA6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-oneHuman11854
MAPK1 (Erk2)MAPKCMGC6rq4AB6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-oneHuman11855
MAPK1 (Erk2)MAPKCMGC6slgAA(6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-oneHuman11815
MAPK1 (Erk2)MAPKCMGC6slgAB(6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-oneHuman11816
MAPK1 (Erk2)MAPKCMGC7auvAA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13925
MAPK1 (Erk2)MAPKCMGC7auvAB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13930
MAPK1 (Erk2)MAPKCMGC7e73A-Human14114
MAPK1 (Erk2)MAPKCMGC7e75A-Human14115
MAPK1 (Erk2)MAPKCMGC7nqqAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamideHuman13926
MAPK1 (Erk2)MAPKCMGC7nqqAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamideHuman13928
MAPK1 (Erk2)MAPKCMGC7nqwAA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-oneHuman13927
MAPK1 (Erk2)MAPKCMGC7nqwAB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-oneHuman13924
MAPK1 (Erk2)MAPKCMGC7nr3AA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-oneHuman13923
MAPK1 (Erk2)MAPKCMGC7nr3AB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-oneHuman13922
MAPK1 (Erk2)MAPKCMGC7nr5AA(2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13921
MAPK1 (Erk2)MAPKCMGC7nr5AB(2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13934
MAPK1 (Erk2)MAPKCMGC7nr8AA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamideHuman13933
MAPK1 (Erk2)MAPKCMGC7nr8AB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamideHuman13929
MAPK1 (Erk2)MAPKCMGC7nr9AA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamideHuman13932
MAPK1 (Erk2)MAPKCMGC7nr9AB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamideHuman13931
MAPK1 (Erk2)MAPKCMGC7opmAA1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]ureaHuman14084
MAPK1 (Erk2)MAPKCMGC7opmAB1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]ureaHuman14083
MAPK1 (Erk2)MAPKCMGC7w5oA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14110
MAPK1 (Erk2)MAPKCMGC7x4uAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14660
MAPK1 (Erk2)MAPKCMGC7x4uAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14661
MAPK1 (Erk2)MAPKCMGC7xc1A(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14665
MAPK1 (Erk2)MAPKCMGC8ao2AA~{n}-(1~{h}-indazol-5-ylmethyl)propanamideHuman14415
MAPK1 (Erk2)MAPKCMGC8ao2AB~{n}-(1~{h}-indazol-5-ylmethyl)propanamideHuman14394
MAPK1 (Erk2)MAPKCMGC8ao3AA2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14386
MAPK1 (Erk2)MAPKCMGC8ao3AB2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14414
MAPK1 (Erk2)MAPKCMGC8ao4AA~{n}-(1~{h}-indazol-5-yl)ethanesulfonamideHuman14416
MAPK1 (Erk2)MAPKCMGC8ao4AB~{n}-(1~{h}-indazol-5-yl)ethanesulfonamideHuman14399
MAPK1 (Erk2)MAPKCMGC8ao5AA~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamideHuman14392
MAPK1 (Erk2)MAPKCMGC8ao5AB~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamideHuman14400
MAPK1 (Erk2)MAPKCMGC8ao6AA~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14397
MAPK1 (Erk2)MAPKCMGC8ao6AB~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14396
MAPK1 (Erk2)MAPKCMGC8ao7AA~{n}-[(1-methylindazol-6-yl)methyl]propanamideHuman14389
MAPK1 (Erk2)MAPKCMGC8ao7AB~{n}-[(1-methylindazol-6-yl)methyl]propanamideHuman14398
MAPK1 (Erk2)MAPKCMGC8ao8AA1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-oneHuman14410
MAPK1 (Erk2)MAPKCMGC8ao8AB1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-oneHuman14405
MAPK1 (Erk2)MAPKCMGC8ao9AA1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-oneHuman14420
MAPK1 (Erk2)MAPKCMGC8ao9AB1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-oneHuman14390
MAPK1 (Erk2)MAPKCMGC8ao9AC1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-oneHuman14401
MAPK1 (Erk2)MAPKCMGC8aoaAA~{n}-pyridin-3-ylprop-2-enamideHuman14391
MAPK1 (Erk2)MAPKCMGC8aoaAB~{n}-pyridin-3-ylpropanamideHuman14407
MAPK1 (Erk2)MAPKCMGC8aobAA~{n}-[(1-methylindazol-3-yl)methyl]propanamideHuman14402
MAPK1 (Erk2)MAPKCMGC8aobAB~{n}-[(1-methylindazol-3-yl)methyl]propanamideHuman14413
MAPK1 (Erk2)MAPKCMGC8aocAA~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamideHuman14409
MAPK1 (Erk2)MAPKCMGC8aocAB~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamideHuman14406
MAPK1 (Erk2)MAPKCMGC8aodAA1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-oneHuman14417
MAPK1 (Erk2)MAPKCMGC8aodAB1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-oneHuman14388
MAPK1 (Erk2)MAPKCMGC8aoeAA~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamideHuman14395
MAPK1 (Erk2)MAPKCMGC8aoeAB~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamideHuman14411
MAPK1 (Erk2)MAPKCMGC8aofAA~{n}-(2-methylpyrimidin-5-yl)propanamideHuman14419
MAPK1 (Erk2)MAPKCMGC8aofAB~{n}-(2-methylpyrimidin-5-yl)propanamideHuman14408
MAPK1 (Erk2)MAPKCMGC8aogAA~{n}-(5-methyl-1,2-oxazol-3-yl)propanamideHuman14403
MAPK1 (Erk2)MAPKCMGC8aogAB~{n}-(5-methyl-1,2-oxazol-3-yl)propanamideHuman14421
MAPK1 (Erk2)MAPKCMGC8aohAA~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamideHuman14385
MAPK1 (Erk2)MAPKCMGC8aohAB~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamideHuman14404
MAPK1 (Erk2)MAPKCMGC8aoiAA1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-oneHuman14387
MAPK1 (Erk2)MAPKCMGC8aoiAB1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-oneHuman14393
MAPK1 (Erk2)MAPKCMGC8aojAA1-[(2~{s})-2-(5-methyl-3-pyridin-4-yl-1~{h}-pyrazol-4-yl)pyrrolidin-1-yl]propan-1-oneHuman14412
MAPK1 (Erk2)MAPKCMGC8aojAB-Human14418
MAPK10 (JNK3)MAPKCMGC1jnkAphosphoaminophosphonic acid-adenylate esterHuman3451
MAPK10 (JNK3)MAPKCMGC1pmnAcyclopropyl-{4-[5-(3,4-dichlorophenyl)-2-[(1-methyl)-piperidin]-4-yl-3-propyl-3h-imidazol-4-yl]-pyrimidin-2-yl}amineHuman3439
MAPK10 (JNK3)MAPKCMGC1pmuA9-(4-hydroxyphenyl)-2,7-phenanthrolineHuman3474
MAPK10 (JNK3)MAPKCMGC1pmvA2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHuman3434
MAPK10 (JNK3)MAPKCMGC2b1pA3-{6-[(2-chlorophenyl)amino]-1h-indazol-3-yl}-5-{[4-(dimethylamino)butanoyl]amino}benzoic acidHuman3464
MAPK10 (JNK3)MAPKCMGC2excXn-{2'-[(4-fluorophenyl)amino]-4,4'-bipyridin-2-yl}-4-methoxycyclohexanecarboxamideHuman3478
MAPK10 (JNK3)MAPKCMGC2o0uAn-{3-cyano-6-[3-(1-piperidinyl)propanoyl]-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-yl}1-naphthalenecarboxamideHuman3415
MAPK10 (JNK3)MAPKCMGC2o2uAn-(3-cyano-4,5,6,7-tetrahydro-1-benzothien-2-yl)-2-fluorobenzamideHuman3457
MAPK10 (JNK3)MAPKCMGC2ok1AAn-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamideHuman3444
MAPK10 (JNK3)MAPKCMGC2ok1ABn-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamideHuman3473
MAPK10 (JNK3)MAPKCMGC2p33A4-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-n-ethylpiperidine-1-carboxamideHuman3455
MAPK10 (JNK3)MAPKCMGC2r9sAn-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamideHuman3450
MAPK10 (JNK3)MAPKCMGC2r9sBn-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamideHuman3420
MAPK10 (JNK3)MAPKCMGC2wajAA1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinolineHuman3472
MAPK10 (JNK3)MAPKCMGC2wajAB1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinolineHuman3471
MAPK10 (JNK3)MAPKCMGC2zdtAA4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acidHuman3421
MAPK10 (JNK3)MAPKCMGC2zdtAB4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acidHuman3424
MAPK10 (JNK3)MAPKCMGC2zduA4-[(4-{[6-bromo-3-(methoxycarbonyl)-1-oxo-4-phenylisoquinolin-2(1h)-yl]methyl}phenyl)amino]-4-oxobutanoic acidHuman3479
MAPK10 (JNK3)MAPKCMGC3cgfAn-cyclohexyl-4-imidazo[1,2-a]pyridin-3-yl-n-methylpyrimidin-2-amineHuman6770
MAPK10 (JNK3)MAPKCMGC3cgoA2-{4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidin-1-yl}-n-methylacetamideHuman6771
MAPK10 (JNK3)MAPKCMGC3da6An-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)naphthalen-1-yl]-1h-benzimidazol-2-amineHuman3476
MAPK10 (JNK3)MAPKCMGC3fi2AA3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHuman3463
MAPK10 (JNK3)MAPKCMGC3fi2AB3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHuman3452
MAPK10 (JNK3)MAPKCMGC3fi3AA3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHuman3442
MAPK10 (JNK3)MAPKCMGC3fi3AB3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHuman3445
MAPK10 (JNK3)MAPKCMGC3fv8AA5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamideHuman3468
MAPK10 (JNK3)MAPKCMGC3fv8AB5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamideHuman3426
MAPK10 (JNK3)MAPKCMGC3g90X(3e)-5-fluoro-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-1h-indole-2,3-dione 3-oximeHuman3477
MAPK10 (JNK3)MAPKCMGC3g9lX(3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-[(e)-2-phenylethenyl]-1h-indole-2,3-dione 3-oximeHuman3435
MAPK10 (JNK3)MAPKCMGC3g9nA(3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-phenyl-1h-indole-2,3-dione 3-oximeHuman3416
MAPK10 (JNK3)MAPKCMGC3kvxAAn-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)anilineHuman3433
MAPK10 (JNK3)MAPKCMGC3kvxABn-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)anilineHuman3430
MAPK10 (JNK3)MAPKCMGC3oxiAmethyl 3-[(thiophen-2-ylacetyl)amino]thiophene-2-carboxylateHuman3423
MAPK10 (JNK3)MAPKCMGC3oy1A5-[2-(cyclohexylamino)pyridin-4-yl]-4-naphthalen-2-yl-2-(tetrahydro-2h-pyran-4-yl)-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman3469
MAPK10 (JNK3)MAPKCMGC3ptgAn-[4-methyl-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamideHuman3470
MAPK10 (JNK3)MAPKCMGC3rtpAn-[4-cyano-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamideHuman3467
MAPK10 (JNK3)MAPKCMGC3ttiAtrans-4-({9-[(3s)-tetrahydrofuran-3-yl]-8-[(2,4,6-trifluorophenyl)amino]-9h-purin-2-yl}amino)cyclohexanolHuman3456
MAPK10 (JNK3)MAPKCMGC3ttjAA9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamineHuman3458
MAPK10 (JNK3)MAPKCMGC3ttjAB9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamineHuman3428
MAPK10 (JNK3)MAPKCMGC3v6rAA4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3441
MAPK10 (JNK3)MAPKCMGC3v6rAB4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3436
MAPK10 (JNK3)MAPKCMGC3v6rBA4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3427
MAPK10 (JNK3)MAPKCMGC3v6rBB4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3417
MAPK10 (JNK3)MAPKCMGC3v6sAB3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3449
MAPK10 (JNK3)MAPKCMGC3v6sBB3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3425
MAPK10 (JNK3)MAPKCMGC4h36AA-Human3459
MAPK10 (JNK3)MAPKCMGC4h36AB-Human3461
MAPK10 (JNK3)MAPKCMGC4h39AA-Human3460
MAPK10 (JNK3)MAPKCMGC4h39AB-Human3462
MAPK10 (JNK3)MAPKCMGC4h3bAA-Human3480
MAPK10 (JNK3)MAPKCMGC4h3bAB-Human3454
MAPK10 (JNK3)MAPKCMGC4h3bAC-Human3453
MAPK10 (JNK3)MAPKCMGC4h3bCA-Human3475
MAPK10 (JNK3)MAPKCMGC4h3bCB-Human3465
MAPK10 (JNK3)MAPKCMGC4h3bCC-Human3446
MAPK10 (JNK3)MAPKCMGC4kkeAadenosine monophosphateHuman3448
MAPK10 (JNK3)MAPKCMGC4kkgA-Human3443
MAPK10 (JNK3)MAPKCMGC4kkhAcyclopropyl[(3r)-3-({4-[6-hydroxy-2-(naphthalen-2-yl)-1h-benzimidazol-1-yl]pyrimidin-2-yl}amino)piperidin-1-yl]methanoneHuman3419
MAPK10 (JNK3)MAPKCMGC4u79An-{4-[(3-{2-[(trans-4-aminocyclohexyl)amino]pyrimidin-4-yl}pyridin-2-yl)oxy]naphthalen-1-yl}benzenesulfonamideHuman3466
MAPK10 (JNK3)MAPKCMGC4w4vA3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamideHuman3437
MAPK10 (JNK3)MAPKCMGC4w4wAn-(2-methylpyridin-4-yl)-3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}benzamideHuman3418
MAPK10 (JNK3)MAPKCMGC4w4xA3-(4-{[(4-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamideHuman3440
MAPK10 (JNK3)MAPKCMGC4w4yA3-(4-{[(4-methylphenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamideHuman3447
MAPK10 (JNK3)MAPKCMGC4whzAA3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamideHuman3429
MAPK10 (JNK3)MAPKCMGC4whzAB3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamideHuman3422
MAPK10 (JNK3)MAPKCMGC4x21An-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamideHuman6240
MAPK10 (JNK3)MAPKCMGC4x21Bn-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamideHuman6239
MAPK10 (JNK3)MAPKCMGC4y46A1-{trans-4-[(8-cyclopentyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]cyclohexyl}-3-propan-2-ylureaHuman3414
MAPK10 (JNK3)MAPKCMGC4y5hA1-(trans-4-{[7-oxo-8-(propan-2-yl)-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}cyclohexyl)-3-propan-2-ylureaHuman3431
MAPK10 (JNK3)MAPKCMGC4z9lAAphosphoaminophosphonic acid-adenylate esterHuman3432
MAPK10 (JNK3)MAPKCMGC4z9lABphosphoaminophosphonic acid-adenylate esterHuman3438
MAPK10 (JNK3)MAPKCMGC6ekdAA4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10498
MAPK10 (JNK3)MAPKCMGC6ekdAB4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10502
MAPK10 (JNK3)MAPKCMGC6emhAA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10508
MAPK10 (JNK3)MAPKCMGC6emhAB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10503
MAPK10 (JNK3)MAPKCMGC6emhBA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10506
MAPK10 (JNK3)MAPKCMGC6emhBB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10501
MAPK10 (JNK3)MAPKCMGC6emhCA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10507
MAPK10 (JNK3)MAPKCMGC6emhCB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10505
MAPK10 (JNK3)MAPKCMGC6emhDA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10497
MAPK10 (JNK3)MAPKCMGC6emhDB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10496
MAPK10 (JNK3)MAPKCMGC6eq9AAphosphomethylphosphonic acid adenylate esterHuman10500
MAPK10 (JNK3)MAPKCMGC6eq9ABphosphomethylphosphonic acid adenylate esterHuman10509
MAPK10 (JNK3)MAPKCMGC6eq9BAphosphomethylphosphonic acid adenylate esterHuman10504
MAPK10 (JNK3)MAPKCMGC6eq9BBphosphomethylphosphonic acid adenylate esterHuman10499
MAPK10 (JNK3)MAPKCMGC7ksiA4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13387
MAPK10 (JNK3)MAPKCMGC7ksjA4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13388
MAPK10 (JNK3)MAPKCMGC7kskA4-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13386
MAPK10 (JNK3)MAPKCMGC7oreAA4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamideHuman13811
MAPK10 (JNK3)MAPKCMGC7oreAB4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamideHuman13810
MAPK10 (JNK3)MAPKCMGC7oreAC4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamideHuman13813
MAPK10 (JNK3)MAPKCMGC7orfAAn-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamideHuman13812
MAPK10 (JNK3)MAPKCMGC7orfABn-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamideHuman13814
MAPK10 (JNK3)MAPKCMGC7s1nAA4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13958
MAPK10 (JNK3)MAPKCMGC7s1nAB4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13957
MAPK10 (JNK3)MAPKCMGC7yl1A7-hexyl-3-methyl-8-sulfanylidene-9h-purine-2,6-dioneHuman14845
MAPK10 (JNK3)MAPKCMGC8bzpAA2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamideHuman14859
MAPK10 (JNK3)MAPKCMGC8bzpAB2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamideHuman14858
MAPK10 (JNK3)MAPKCMGC8enjAn-[3-({(4p)-4-[(3m)-1-tert-butyl-3-(3-hydroxyphenyl)-1h-pyrazol-4-yl]pyridin-2-yl}amino)propyl]-4-hydroxybenzene-1-sulfonamideHuman14884
MAPK10 (JNK3)MAPKCMGC8wgfAAphosphoaminophosphonic acid-adenylate esterHuman15046
MAPK10 (JNK3)MAPKCMGC8wgfABphosphoaminophosphonic acid-adenylate esterHuman15047
MAPK11 (p38b)MAPKCMGC3gc8A5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman2766
MAPK11 (p38b)MAPKCMGC3gc8B5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman2769
MAPK11 (p38b)MAPKCMGC3gc9A5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman2765
MAPK11 (p38b)MAPKCMGC3gc9B5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman2767
MAPK11 (p38b)MAPKCMGC3gp0AAnilotinibHuman2768
MAPK11 (p38b)MAPKCMGC3gp0ABnilotinibHuman2764
MAPK12 (p38g)MAPKCMGC1cm8Aphosphoaminophosphonic acid-adenylate esterHuman4625
MAPK12 (p38g)MAPKCMGC1cm8Bphosphoaminophosphonic acid-adenylate esterHuman4626
MAPK12 (p38g)MAPKCMGC6unaAA-Human11898
MAPK12 (p38g)MAPKCMGC6unaAB-Human11900
MAPK12 (p38g)MAPKCMGC6unaBA-Human11901
MAPK12 (p38g)MAPKCMGC6unaBB-Human11899
MAPK12 (p38g)MAPKCMGC7cgaA-Human13762
MAPK13 (p38d)MAPKCMGC3coiAA-Human2948
MAPK13 (p38d)MAPKCMGC3coiAB-Human2946
MAPK13 (p38d)MAPKCMGC4eyjA1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-yloxy)phenyl]ureaHuman2949
MAPK13 (p38d)MAPKCMGC4eymA2-(morpholin-4-yl)-n-[4-(pyridin-4-yloxy)phenyl]pyridine-4-carboxamideHuman2945
MAPK13 (p38d)MAPKCMGC4mygA-Human2951
MAPK13 (p38d)MAPKCMGC4mygB-Human2950
MAPK13 (p38d)MAPKCMGC4ynoA-Human2947
MAPK13 (p38d)MAPKCMGC5eknA1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-ylsulfanyl)phenyl]ureaHuman6745
MAPK13 (p38d)MAPKCMGC5ekoA3-(4-methyl-1h-imidazol-1-yl)-n-[4-(pyridin-4-yloxy)phenyl]benzamideHuman6746
MAPK13 (p38d)MAPKCMGC8x23AA-Human15129
MAPK13 (p38d)MAPKCMGC8x23AB-Human15128
Mapk14 (p38a)MAPKCMGC1lewA-Mouse5864
Mapk14 (p38a)MAPKCMGC1lezA-Mouse5863
Mapk14 (p38a)MAPKCMGC1yw2A2-(ethoxymethyl)-4-(4-fluorophenyl)-3-[2-(2-hydroxyphenoxy)pyrimidin-4-yl]isoxazol-5(2h)-oneMouse5869
Mapk14 (p38a)MAPKCMGC1ywrA4-(4-fluorophenyl)-1-methyl-5-(2-{[(1s)-1-phenylethyl]amino}pyrimidin-4-yl)-2-piperidin-4-yl-1,2-dihydro-3h-pyrazol-3-oneMouse5840
Mapk14 (p38a)MAPKCMGC2ewaAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse5859
Mapk14 (p38a)MAPKCMGC2ewaAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse5870
Mapk14 (p38a)MAPKCMGC2ghlA3-(2-chlorophenyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)ureaMouse5871
Mapk14 (p38a)MAPKCMGC2ghmA3-(2-chlorobenzyl)-1-(2-{[(1s)-2-hydroxy-1,2-dimethylpropyl]amino}pyrimidin-4-yl)-1-(4-methoxyphenyl)ureaMouse5845
Mapk14 (p38a)MAPKCMGC2gtmA8-(2-chlorophenylamino)-2-(2,6-difluorophenylamino)-9-ethyl-9h-purine-1,7-diiumMouse5867
Mapk14 (p38a)MAPKCMGC2gtnA2-(2,6-difluorophenoxy)-n-(2-fluorophenyl)-9-isopropyl-9h-purin-8-amineMouse5860
Mapk14 (p38a)MAPKCMGC2ozaB-Mouse5862
Mapk14 (p38a)MAPKCMGC2puuA5-tert-butyl-2-(4-methylphenyl)-3-{[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]-1-naphthyl}amino)carbonyl]amino}-1h-pyrazol-2-iumMouse6866
Mapk14 (p38a)MAPKCMGC3p4kA-Mouse5842
Mapk14 (p38a)MAPKCMGC3p5kA1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylureaMouse5854
Mapk14 (p38a)MAPKCMGC3p78A1-{5-tert-butyl-3-[(1,1-dioxidothiomorpholin-4-yl)carbonyl]thiophen-2-yl}-3-naphthalen-2-ylureaMouse5866
Mapk14 (p38a)MAPKCMGC3p79A1-{3-tert-butyl-1-[2-(1,1-dioxidothiomorpholin-4-yl)-2-oxoethyl]-1h-pyrazol-5-yl}-3-naphthalen-2-ylureaMouse5849
Mapk14 (p38a)MAPKCMGC3p7aA1-[5-tert-butyl-2-(1,1-dioxidothiomorpholin-4-yl)thiophen-3-yl]-3-naphthalen-1-ylureaMouse5853
Mapk14 (p38a)MAPKCMGC3p7bA1-{5-tert-butyl-3-[(5-oxo-1,4-diazepan-1-yl)carbonyl]thiophen-2-yl}-3-naphthalen-1-ylureaMouse5856
Mapk14 (p38a)MAPKCMGC3p7cA1-[5-tert-butyl-3-({4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepan-1-yl}carbonyl)thiophen-2-yl]-3-(2,3-dichlorophenyl)ureaMouse5838
Mapk14 (p38a)MAPKCMGC3py3A-Mouse5857
Mapk14 (p38a)MAPKCMGC3tg1A-Mouse5850
Mapk14 (p38a)MAPKCMGC4ka3A-Mouse5852
Mapk14 (p38a)MAPKCMGC4looAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5851
Mapk14 (p38a)MAPKCMGC4looAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5832
Mapk14 (p38a)MAPKCMGC4lopAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5848
Mapk14 (p38a)MAPKCMGC4lopAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5861
Mapk14 (p38a)MAPKCMGC4lopBA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5839
Mapk14 (p38a)MAPKCMGC4lopBB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5831
Mapk14 (p38a)MAPKCMGC4lopCA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5847
Mapk14 (p38a)MAPKCMGC4lopCB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5855
Mapk14 (p38a)MAPKCMGC4lopDA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5865
Mapk14 (p38a)MAPKCMGC4lopDB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5837
Mapk14 (p38a)MAPKCMGC4loqAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5872
Mapk14 (p38a)MAPKCMGC4loqAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5836
Mapk14 (p38a)MAPKCMGC4loqBA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5834
Mapk14 (p38a)MAPKCMGC4loqBB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5833
Mapk14 (p38a)MAPKCMGC4loqCA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5858
Mapk14 (p38a)MAPKCMGC4loqCB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5846
Mapk14 (p38a)MAPKCMGC4loqDA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5835
Mapk14 (p38a)MAPKCMGC4loqDB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse5843
Mapk14 (p38a)MAPKCMGC4tyhBAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideMouse5841
Mapk14 (p38a)MAPKCMGC4tyhBBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideMouse5844
Mapk14 (p38a)MAPKCMGC5larAA5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse6753
Mapk14 (p38a)MAPKCMGC5larAB5-azanyl-~{n}-[[4-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse6752
Mapk14 (p38a)MAPKCMGC5nzzEAphosphothiophosphoric acid-adenylate esterMouse9981
Mapk14 (p38a)MAPKCMGC5nzzEBphosphothiophosphoric acid-adenylate esterMouse9980
Mapk14 (p38a)MAPKCMGC5nzzFAphosphothiophosphoric acid-adenylate esterMouse9983
Mapk14 (p38a)MAPKCMGC5nzzFBphosphothiophosphoric acid-adenylate esterMouse9979
Mapk14 (p38a)MAPKCMGC5nzzGAphosphothiophosphoric acid-adenylate esterMouse9977
Mapk14 (p38a)MAPKCMGC5nzzGBphosphothiophosphoric acid-adenylate esterMouse9982
Mapk14 (p38a)MAPKCMGC5nzzHAphosphothiophosphoric acid-adenylate esterMouse9978
Mapk14 (p38a)MAPKCMGC5nzzHBphosphothiophosphoric acid-adenylate esterMouse9984
Mapk14 (p38a)MAPKCMGC5o90A4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse9525
Mapk14 (p38a)MAPKCMGC5r8uAA3,4-dihydro-2~{h}-chromene-6-carboxamideMouse12555
Mapk14 (p38a)MAPKCMGC5r8uAB3,4-dihydro-2~{h}-chromene-6-carboxamideMouse12583
Mapk14 (p38a)MAPKCMGC5r8vAA-Mouse12553
Mapk14 (p38a)MAPKCMGC5r8vAB-Mouse12556
Mapk14 (p38a)MAPKCMGC5r8wAA-Mouse12535
Mapk14 (p38a)MAPKCMGC5r8wAB-Mouse12534
Mapk14 (p38a)MAPKCMGC5r8xAA-Mouse12573
Mapk14 (p38a)MAPKCMGC5r8xAB-Mouse12521
Mapk14 (p38a)MAPKCMGC5r8yAAthiophene-2-carbothioamideMouse12584
Mapk14 (p38a)MAPKCMGC5r8yABthiophene-2-carbothioamideMouse12524
Mapk14 (p38a)MAPKCMGC5r8zAA6-methoxypyridine-3-carbothioamideMouse12575
Mapk14 (p38a)MAPKCMGC5r8zAB6-methoxypyridine-3-carbothioamideMouse12544
Mapk14 (p38a)MAPKCMGC5r90AA2,5-diphenyl-4~{h}-pyrazol-3-oneMouse12603
Mapk14 (p38a)MAPKCMGC5r90AB2,5-diphenyl-4~{h}-pyrazol-3-oneMouse12582
Mapk14 (p38a)MAPKCMGC5r91AA-Mouse12560
Mapk14 (p38a)MAPKCMGC5r91AB-Mouse12539
Mapk14 (p38a)MAPKCMGC5r92AA(3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamideMouse12590
Mapk14 (p38a)MAPKCMGC5r92AB(3~{s})-~{n}-methoxy-1-(4-methoxyphenyl)-~{n}-methyl-5-oxidanylidene-pyrrolidine-3-carboxamideMouse12620
Mapk14 (p38a)MAPKCMGC5r93AA-Mouse12571
Mapk14 (p38a)MAPKCMGC5r93AB-Mouse12545
Mapk14 (p38a)MAPKCMGC5r94AA-Mouse12532
Mapk14 (p38a)MAPKCMGC5r94AB-Mouse12589
Mapk14 (p38a)MAPKCMGC5r95AA-Mouse12586
Mapk14 (p38a)MAPKCMGC5r95AB-Mouse12597
Mapk14 (p38a)MAPKCMGC5r96AA-Mouse12610
Mapk14 (p38a)MAPKCMGC5r96AB-Mouse12559
Mapk14 (p38a)MAPKCMGC5r97AA4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amineMouse12529
Mapk14 (p38a)MAPKCMGC5r97AB4-(piperidin-1-yl)-1,2,5-oxadiazol-3-amineMouse12525
Mapk14 (p38a)MAPKCMGC5r98AA-Mouse12563
Mapk14 (p38a)MAPKCMGC5r98AB-Mouse12606
Mapk14 (p38a)MAPKCMGC5r99AA3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrileMouse12572
Mapk14 (p38a)MAPKCMGC5r99AB3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrileMouse12533
Mapk14 (p38a)MAPKCMGC5r9aAA-Mouse12565
Mapk14 (p38a)MAPKCMGC5r9aAB-Mouse12604
Mapk14 (p38a)MAPKCMGC5r9bAA-Mouse12577
Mapk14 (p38a)MAPKCMGC5r9bAB-Mouse12540
Mapk14 (p38a)MAPKCMGC5r9cAA-Mouse12591
Mapk14 (p38a)MAPKCMGC5r9cAB-Mouse12522
Mapk14 (p38a)MAPKCMGC5r9dAAbenzyl hydroxycarbamateMouse12550
Mapk14 (p38a)MAPKCMGC5r9dABbenzyl hydroxycarbamateMouse12554
Mapk14 (p38a)MAPKCMGC5r9eAA-Mouse12602
Mapk14 (p38a)MAPKCMGC5r9eAB-Mouse12564
Mapk14 (p38a)MAPKCMGC5r9fAA-Mouse12526
Mapk14 (p38a)MAPKCMGC5r9fAB-Mouse12569
Mapk14 (p38a)MAPKCMGC5r9gAA-Mouse12547
Mapk14 (p38a)MAPKCMGC5r9gAB-Mouse12595
Mapk14 (p38a)MAPKCMGC5r9hAA-Mouse12615
Mapk14 (p38a)MAPKCMGC5r9hAB-Mouse12587
Mapk14 (p38a)MAPKCMGC5r9iAAmethyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoateMouse12548
Mapk14 (p38a)MAPKCMGC5r9iABmethyl (2~{r})-3-(4-bromophenyl)-2-pyridin-4-yl-propanoateMouse12551
Mapk14 (p38a)MAPKCMGC5r9jAA3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dioneMouse12609
Mapk14 (p38a)MAPKCMGC5r9jAB3-ethyl-1-[(1~{r},8~{s},9~{s},10~{s})-10-oxidanyl-11-oxatricyclo[6.2.1.0^{2,7}]undeca-2(7),3,5-trien-9-yl]imidazolidine-2,4-dioneMouse12527
Mapk14 (p38a)MAPKCMGC5r9kAA2,3-dihydro-1-benzoxepine-5-carboxylic acidMouse12611
Mapk14 (p38a)MAPKCMGC5r9kAB2,3-dihydro-1-benzoxepine-5-carboxylic acidMouse12549
Mapk14 (p38a)MAPKCMGC5r9lAA(3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-olMouse12562
Mapk14 (p38a)MAPKCMGC5r9lAB(3~{s})-2-(cyclopropylmethyl)-3-[(~{s})-oxidanyl(phenyl)methyl]-2-azabicyclo[2.2.2]octan-4-olMouse12523
Mapk14 (p38a)MAPKCMGC5r9mAA-Mouse12574
Mapk14 (p38a)MAPKCMGC5r9mAB-Mouse12570
Mapk14 (p38a)MAPKCMGC5r9nAA[4-(1h-benzimidazol-1-yl)phenyl]methanolMouse12593
Mapk14 (p38a)MAPKCMGC5r9nAB[4-(1h-benzimidazol-1-yl)phenyl]methanolMouse12596
Mapk14 (p38a)MAPKCMGC5r9oAA-Mouse12588
Mapk14 (p38a)MAPKCMGC5r9oAB-Mouse12616
Mapk14 (p38a)MAPKCMGC5r9pAA4-amino-n-(pyridin-2-yl)benzenesulfonamideMouse12518
Mapk14 (p38a)MAPKCMGC5r9pAB4-amino-n-(pyridin-2-yl)benzenesulfonamideMouse12576
Mapk14 (p38a)MAPKCMGC5r9qAA1-phenylmethoxyureaMouse12557
Mapk14 (p38a)MAPKCMGC5r9qAB1-phenylmethoxyureaMouse12612
Mapk14 (p38a)MAPKCMGC5r9rAA4-acetyl-n-ethylpiperazine-1-carboxamideMouse12519
Mapk14 (p38a)MAPKCMGC5r9rAB4-acetyl-n-ethylpiperazine-1-carboxamideMouse12536
Mapk14 (p38a)MAPKCMGC5r9sAA-Mouse12531
Mapk14 (p38a)MAPKCMGC5r9sAB-Mouse12561
Mapk14 (p38a)MAPKCMGC5r9tAA-Mouse12618
Mapk14 (p38a)MAPKCMGC5r9tAB-Mouse12538
Mapk14 (p38a)MAPKCMGC5r9uAA[4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanoneMouse12541
Mapk14 (p38a)MAPKCMGC5r9uAB[4-(cyclopropanecarbonyl)piperazin-1-yl](furan-2-yl)methanoneMouse12546
Mapk14 (p38a)MAPKCMGC5r9vAA-Mouse12530
Mapk14 (p38a)MAPKCMGC5r9vAB-Mouse12528
Mapk14 (p38a)MAPKCMGC5r9wAA~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamideMouse12605
Mapk14 (p38a)MAPKCMGC5r9wAB~{n}-(1,3-benzodioxol-5-ylmethyl)ethanesulfonamideMouse12542
Mapk14 (p38a)MAPKCMGC5r9xAA-Mouse12566
Mapk14 (p38a)MAPKCMGC5r9xAB-Mouse12543
Mapk14 (p38a)MAPKCMGC5r9yAA3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrileMouse12537
Mapk14 (p38a)MAPKCMGC5r9yAB3-oxidanylidene-3-[4-(phenylmethyl)piperidin-1-yl]propanenitrileMouse12621
Mapk14 (p38a)MAPKCMGC5r9zAA-Mouse12580
Mapk14 (p38a)MAPKCMGC5r9zAB-Mouse12613
Mapk14 (p38a)MAPKCMGC5ra0AA[4-(1h-benzimidazol-1-yl)phenyl]methanolMouse12592
Mapk14 (p38a)MAPKCMGC5ra0AB[4-(1h-benzimidazol-1-yl)phenyl]methanolMouse12617
Mapk14 (p38a)MAPKCMGC5ra1AA2-phenoxyacetamideMouse12600
Mapk14 (p38a)MAPKCMGC5ra1AB2-phenoxyacetamideMouse12579
Mapk14 (p38a)MAPKCMGC5ra2AA1-(3-methylpyridin-2-yl)-1,4-diazepaneMouse12568
Mapk14 (p38a)MAPKCMGC5ra2AB1-(3-methylpyridin-2-yl)-1,4-diazepaneMouse12520
Mapk14 (p38a)MAPKCMGC5ra3AA-Mouse12599
Mapk14 (p38a)MAPKCMGC5ra3AB-Mouse12581
Mapk14 (p38a)MAPKCMGC5ra4AA-Mouse12552
Mapk14 (p38a)MAPKCMGC5ra4AB-Mouse12594
Mapk14 (p38a)MAPKCMGC5ra5AA-Mouse12558
Mapk14 (p38a)MAPKCMGC5ra5AB-Mouse12619
Mapk14 (p38a)MAPKCMGC5ra6AA1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thioureaMouse12614
Mapk14 (p38a)MAPKCMGC5ra6AB1-[(1~{r},2~{r},4~{s})-2-bicyclo[2.2.1]heptanyl]-3-(2-pyridin-2-ylethyl)thioureaMouse12598
Mapk14 (p38a)MAPKCMGC5ra7AA4-methylbenzamideMouse12567
Mapk14 (p38a)MAPKCMGC5ra7AB4-methylbenzamideMouse12578
Mapk14 (p38a)MAPKCMGC5ra8AA5-(trifluoromethyl)-1,2-benzoxazol-3-amineMouse12585
Mapk14 (p38a)MAPKCMGC5ra8AB5-(trifluoromethyl)-1,2-benzoxazol-3-amineMouse12608
Mapk14 (p38a)MAPKCMGC5ra9AA4-chloranylthieno[3,2-d]pyrimidineMouse12601
Mapk14 (p38a)MAPKCMGC5ra9AB4-chloranylthieno[3,2-d]pyrimidineMouse12607
Mapk14 (p38a)MAPKCMGC5uojA-Mouse7466
Mapk14 (p38a)MAPKCMGC6so1AA-Mouse11681
Mapk14 (p38a)MAPKCMGC6so1AB-Mouse11675
Mapk14 (p38a)MAPKCMGC6so2AA-Mouse11678
Mapk14 (p38a)MAPKCMGC6so2AB-Mouse11679
Mapk14 (p38a)MAPKCMGC6so4AA-Mouse11627
Mapk14 (p38a)MAPKCMGC6so4AB-Mouse11626
Mapk14 (p38a)MAPKCMGC6sodAA-Mouse11673
Mapk14 (p38a)MAPKCMGC6sodAB-Mouse11674
Mapk14 (p38a)MAPKCMGC6soiAA-Mouse11676
Mapk14 (p38a)MAPKCMGC6soiAB-Mouse11682
Mapk14 (p38a)MAPKCMGC6sotAA-Mouse11689
Mapk14 (p38a)MAPKCMGC6sotAB-Mouse11688
Mapk14 (p38a)MAPKCMGC6souAA2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanoneMouse11680
Mapk14 (p38a)MAPKCMGC6souAB2-(4-methylphenoxy)-1-(4-methylpiperazin-4-ium-1-yl)ethanoneMouse11672
Mapk14 (p38a)MAPKCMGC6sovAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11685
Mapk14 (p38a)MAPKCMGC6sovAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11677
Mapk14 (p38a)MAPKCMGC6sp9AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11684
Mapk14 (p38a)MAPKCMGC6sp9AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11686
Mapk14 (p38a)MAPKCMGC6splAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11687
Mapk14 (p38a)MAPKCMGC6splAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse11683
Mapk14 (p38a)MAPKCMGC6y4tAA5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12030
Mapk14 (p38a)MAPKCMGC6y4tAB5-azanyl-~{n}-[[4-[[(2~{s})-1-[[(2~{s})-butan-2-yl]amino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12036
Mapk14 (p38a)MAPKCMGC6y4uAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12035
Mapk14 (p38a)MAPKCMGC6y4uAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pentan-3-ylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12038
Mapk14 (p38a)MAPKCMGC6y4vAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12037
Mapk14 (p38a)MAPKCMGC6y4vAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(3-methylbutylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12031
Mapk14 (p38a)MAPKCMGC6y4wAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12034
Mapk14 (p38a)MAPKCMGC6y4wAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(cyclohexylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12033
Mapk14 (p38a)MAPKCMGC6y4xAA5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12039
Mapk14 (p38a)MAPKCMGC6y4xAB5-azanyl-~{n}-[[4-[[(2~{s})-1-[2-(4-chlorophenyl)ethylamino]-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12032
Mapk14 (p38a)MAPKCMGC6y6vAA5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12066
Mapk14 (p38a)MAPKCMGC6y6vAB5-azanyl-~{n}-[[4-[[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12067
Mapk14 (p38a)MAPKCMGC6y7wAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12065
Mapk14 (p38a)MAPKCMGC6y7wAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12071
Mapk14 (p38a)MAPKCMGC6y7xAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12072
Mapk14 (p38a)MAPKCMGC6y7xAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12060
Mapk14 (p38a)MAPKCMGC6y7yAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12063
Mapk14 (p38a)MAPKCMGC6y7yAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12076
Mapk14 (p38a)MAPKCMGC6y7zAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12070
Mapk14 (p38a)MAPKCMGC6y7zAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12082
Mapk14 (p38a)MAPKCMGC6y80AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12081
Mapk14 (p38a)MAPKCMGC6y80AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12080
Mapk14 (p38a)MAPKCMGC6y81AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12079
Mapk14 (p38a)MAPKCMGC6y81AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12073
Mapk14 (p38a)MAPKCMGC6y82AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12077
Mapk14 (p38a)MAPKCMGC6y82AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12061
Mapk14 (p38a)MAPKCMGC6y85AA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12069
Mapk14 (p38a)MAPKCMGC6y85AB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12068
Mapk14 (p38a)MAPKCMGC6y8hAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12075
Mapk14 (p38a)MAPKCMGC6y8hAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12078
Mapk14 (p38a)MAPKCMGC6ycuAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12152
Mapk14 (p38a)MAPKCMGC6ycuAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12154
Mapk14 (p38a)MAPKCMGC6ycwAA4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12153
Mapk14 (p38a)MAPKCMGC6ycwAB4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleMouse12151
Mapk14 (p38a)MAPKCMGC6yjcAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12437
Mapk14 (p38a)MAPKCMGC6yjcAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-piperazin-1-yl-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12438
Mapk14 (p38a)MAPKCMGC6yk7AA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12163
Mapk14 (p38a)MAPKCMGC6yk7AB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-(ethylamino)-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12164
Mapk14 (p38a)MAPKCMGC6zwrAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12708
Mapk14 (p38a)MAPKCMGC6zwrAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-oxidanylidene-1-(pyridin-4-ylmethylamino)butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse12709
Mapk14 (p38a)MAPKCMGC7bdoAA~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamideMouse13409
Mapk14 (p38a)MAPKCMGC7bdoAB~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamideMouse13405
Mapk14 (p38a)MAPKCMGC7bdqA~{n}-[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]-4-[[(1-phenylpyrazolo[3,4-d]pyrimidin-4-yl)amino]methyl]benzamideMouse13408
Mapk14 (p38a)MAPKCMGC7be4A5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideMouse13406
Mapk14 (p38a)MAPKCMGC7be5A5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{r})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-methyl-pyrazole-4-carboxamideMouse13407
Mapk14 (p38a)MAPKCMGC7pvuAA-Mouse14747
Mapk14 (p38a)MAPKCMGC7pvuAB-Mouse14748
Mapk14 (p38a)MAPKCMGC7z6iAA4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridineMouse14801
Mapk14 (p38a)MAPKCMGC7z6iAB4-[4-(4-fluorophenyl)-2-[4-[methyl(oxidanyl)-$l^{3}-sulfanyl]phenyl]-1~{h}-imidazol-5-yl]pyridineMouse14800
Mapk14 (p38a)MAPKCMGC7z9tAn-(2-cyclobutyl-1h-1,3-benzodiazol-5-yl)benzenesulfonamideMouse14799
Mapk14 (p38a)MAPKCMGC8acmA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse15096
Mapk14 (p38a)MAPKCMGC8acoAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse15095
Mapk14 (p38a)MAPKCMGC8acoAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineMouse15094
Mapk14 (p38a)MAPKCMGC8efjA(4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamideMouse14995
MAPK14 (p38a)MAPKCMGC1a9uA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5229
MAPK14 (p38a)MAPKCMGC1bl6A4-(4-fluorophenyl)-1-cycloropropylmethyl-5-(4-pyridyl)-imidazoleHuman5243
MAPK14 (p38a)MAPKCMGC1bl7A4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleHuman5193
MAPK14 (p38a)MAPKCMGC1bmkA4-(fluorophenyl)-1-cyclopropylmethyl-5-(2-amino-4-pyrimidinyl)imidazoleHuman5235
MAPK14 (p38a)MAPKCMGC1di9A4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazolineHuman5251
MAPK14 (p38a)MAPKCMGC1kv1A1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5252
MAPK14 (p38a)MAPKCMGC1kv2A1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman5255
MAPK14 (p38a)MAPKCMGC1m7qA1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2(1h)-oneHuman5128
MAPK14 (p38a)MAPKCMGC1oukA4-[5-[2-(1-phenyl-ethylamino)-pyrimidin-4-yl]-1-methyl-4-(3-trifluoromethylphenyl)-1h-imidazol-2-yl]-piperidineHuman5146
MAPK14 (p38a)MAPKCMGC1ouyA1-(2,6-dichlorophenyl)-6-[(2,4-difluorophenyl)sulfanyl]-7-(1,2,3,6-tetrahydro-4-pyridinyl)-3,4-dihydropyrido[3,2-d]pyrimidin-2(1h)-oneHuman7258
MAPK14 (p38a)MAPKCMGC1oveAA1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-oneHuman5178
MAPK14 (p38a)MAPKCMGC1oveAB1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-oneHuman5087
MAPK14 (p38a)MAPKCMGC1oveAC1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-oneHuman5199
MAPK14 (p38a)MAPKCMGC1oz1AA3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-olHuman5230
MAPK14 (p38a)MAPKCMGC1oz1AB3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-olHuman5261
MAPK14 (p38a)MAPKCMGC1r39A-Human5116
MAPK14 (p38a)MAPKCMGC1r3cAA-Human5170
MAPK14 (p38a)MAPKCMGC1r3cAB-Human4996
MAPK14 (p38a)MAPKCMGC1w7hA3-(benzyloxy)pyridin-2-amineHuman5023
MAPK14 (p38a)MAPKCMGC1w82An-[(3z)-5-tert-butyl-2-phenyl-1,2-dihydro-3h-pyrazol-3-ylidene]-n'-(4-chlorophenyl)ureaHuman5165
MAPK14 (p38a)MAPKCMGC1w83An-[4-chloro-3-(pyridin-3-yloxymethyl)-phenyl]-3-fluoro-Human4986
MAPK14 (p38a)MAPKCMGC1w84A3-(2-pyridin-4-ylethyl)-1h-indoleHuman5065
MAPK14 (p38a)MAPKCMGC1wbnAn-(3-tert-butyl-1h-pyrazol-5-yl)-n'-{4-chloro-3-[(pyridin-3-yloxy)methyl]phenyl}ureaHuman5257
MAPK14 (p38a)MAPKCMGC1wboA2-chlorophenolHuman5039
MAPK14 (p38a)MAPKCMGC1wbsA3-fluoro-5-morpholin-4-yl-n-[3-(2-pyridin-4-ylethyl)-1h-indol-5-yl]benzamideHuman5258
MAPK14 (p38a)MAPKCMGC1wbtA3-fluoro-5-morpholin-4-yl-n-[1-(2-pyridin-4-ylethyl)-1h-indol-6-yl]benzamideHuman5082
MAPK14 (p38a)MAPKCMGC1wbvA3-fluoro-n-1h-indol-5-yl-5-morpholin-4-ylbenzamideHuman5148
MAPK14 (p38a)MAPKCMGC1wbwA3-(1-naphthylmethoxy)pyridin-2-amineHuman5179
MAPK14 (p38a)MAPKCMGC1wfcA-Human4989
MAPK14 (p38a)MAPKCMGC1yqjA6((s)-3-benzylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyrazineHuman5152
MAPK14 (p38a)MAPKCMGC1zyjA4-phenoxy-n-(pyridin-2-ylmethyl)benzamideHuman5058
MAPK14 (p38a)MAPKCMGC1zz2An-[3-(4-fluorophenoxy)phenyl]-4-[(2-hydroxybenzyl)amino]piperidine-1-sulfonamideHuman5164
MAPK14 (p38a)MAPKCMGC1zzlA6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-3-isopropyl[1,2,4]triazolo[4,3-a]pyridineHuman5249
MAPK14 (p38a)MAPKCMGC2bajA1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2,3-dichlorophenyl)ureaHuman5176
MAPK14 (p38a)MAPKCMGC2bakAn-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamideHuman5114
MAPK14 (p38a)MAPKCMGC2balA[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl][3-(piperidin-4-yloxy)phenyl]methanoneHuman5260
MAPK14 (p38a)MAPKCMGC2baqA[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanoneHuman5184
MAPK14 (p38a)MAPKCMGC2fslX-Human5264
MAPK14 (p38a)MAPKCMGC2fsmX-Human5044
MAPK14 (p38a)MAPKCMGC2fsoX-Human5117
MAPK14 (p38a)MAPKCMGC2fstXA-Human5080
MAPK14 (p38a)MAPKCMGC2fstXB-Human5195
MAPK14 (p38a)MAPKCMGC2gfsAA[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanoneHuman5227
MAPK14 (p38a)MAPKCMGC2gfsAB[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanoneHuman5050
MAPK14 (p38a)MAPKCMGC2i0hAA2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dioneHuman5062
MAPK14 (p38a)MAPKCMGC2i0hAB2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dioneHuman5009
MAPK14 (p38a)MAPKCMGC2lgcA1-Human5021
MAPK14 (p38a)MAPKCMGC2lgcA10-Human5063
MAPK14 (p38a)MAPKCMGC2lgcA2-Human5093
MAPK14 (p38a)MAPKCMGC2lgcA3-Human5040
MAPK14 (p38a)MAPKCMGC2lgcA4-Human5067
MAPK14 (p38a)MAPKCMGC2lgcA5-Human5107
MAPK14 (p38a)MAPKCMGC2lgcA6-Human5219
MAPK14 (p38a)MAPKCMGC2lgcA7-Human5161
MAPK14 (p38a)MAPKCMGC2lgcA8-Human5078
MAPK14 (p38a)MAPKCMGC2lgcA9-Human5127
MAPK14 (p38a)MAPKCMGC2npqA-Human5205
MAPK14 (p38a)MAPKCMGC2okrA-Human5136
MAPK14 (p38a)MAPKCMGC2okrD-Human5100
MAPK14 (p38a)MAPKCMGC2onlA-Human5177
MAPK14 (p38a)MAPKCMGC2onlB-Human5007
MAPK14 (p38a)MAPKCMGC2qd9A1-[(3ar)-5-{[3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8h)-yl]carbonyl}-6-methoxy-3ah-pyrrolo[2,3-b]pyridin-3-yl]-2-[(3r)-3-hydroxypyrrolidin-1-yl]-2-oxoethanoneHuman5197
MAPK14 (p38a)MAPKCMGC2rg5An-ethyl-4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5254
MAPK14 (p38a)MAPKCMGC2rg6A4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methyl-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5228
MAPK14 (p38a)MAPKCMGC2y8oAA-Human5079
MAPK14 (p38a)MAPKCMGC2y8oAB-Human5030
MAPK14 (p38a)MAPKCMGC2yisA1-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1h-pyrazol-5-yl]-3-{2-[(3-{2-[(2-hydroxyethyl)sulfanyl]phenyl}[1,2,4]triazolo[4,3-a]pyridin-6-yl)sulfanyl]benzyl}ureaHuman5240
MAPK14 (p38a)MAPKCMGC2yiwA1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)ureaHuman4988
MAPK14 (p38a)MAPKCMGC2yixA1-ethyl-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)ureaHuman5143
MAPK14 (p38a)MAPKCMGC2zazAA4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehydeHuman4980
MAPK14 (p38a)MAPKCMGC2zazAB4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehydeHuman5034
MAPK14 (p38a)MAPKCMGC2zb0AAn-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamideHuman5099
MAPK14 (p38a)MAPKCMGC2zb0ABn-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamideHuman5147
MAPK14 (p38a)MAPKCMGC2zb1AAn-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamideHuman5038
MAPK14 (p38a)MAPKCMGC2zb1ABn-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamideHuman5103
MAPK14 (p38a)MAPKCMGC3bv2A5-methyl-4-[(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)amino]-n-(1-phenylethenyl)pyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5191
MAPK14 (p38a)MAPKCMGC3bv3A5-methyl-4-[(2-methyl-5-{[(3-morpholin-4-ylphenyl)carbonyl]amino}phenyl)amino]-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5207
MAPK14 (p38a)MAPKCMGC3bx5An-[2-methyl-5-(methylcarbamoyl)phenyl]-2-{[(1r)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamideHuman5000
MAPK14 (p38a)MAPKCMGC3c5uA6-[4-(2-fluorophenyl)-1,3-oxazol-5-yl]-n-(1-methylethyl)-1,3-benzothiazol-2-amineHuman5125
MAPK14 (p38a)MAPKCMGC3ctqAn-benzyl-1-[5-({5-tert-butyl-2-methoxy-3-[(methylsulfonyl)amino]phenyl}carbamoyl)-2-methylphenyl]-1h-1,2,3-triazole-4-carboxamideHuman5220
MAPK14 (p38a)MAPKCMGC3d7zAAn~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamideHuman5247
MAPK14 (p38a)MAPKCMGC3d7zABn~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamideHuman5108
MAPK14 (p38a)MAPKCMGC3d83An-{4'-[(cyclopropylmethyl)carbamoyl]-6-methylbiphenyl-3-yl}-2-morpholin-4-ylpyridine-4-carboxamideHuman5028
MAPK14 (p38a)MAPKCMGC3ds6An-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5074
MAPK14 (p38a)MAPKCMGC3ds6Bn-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5188
MAPK14 (p38a)MAPKCMGC3ds6Cn-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5182
MAPK14 (p38a)MAPKCMGC3ds6Dn-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5123
MAPK14 (p38a)MAPKCMGC3dt1An-cyclopropyl-4-methyl-3-{2-[(2-morpholin-4-ylethyl)amino]quinazolin-6-yl}benzamideHuman5086
MAPK14 (p38a)MAPKCMGC3e92An-cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamideHuman5149
MAPK14 (p38a)MAPKCMGC3e93AA4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamideHuman5241
MAPK14 (p38a)MAPKCMGC3e93AB4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamideHuman5004
MAPK14 (p38a)MAPKCMGC3fc1X5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman5110
MAPK14 (p38a)MAPKCMGC3fi4A(2s)-1-{[3-(2-chlorophenyl)-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-olHuman5051
MAPK14 (p38a)MAPKCMGC3fklAn-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-2h-pyran-4-ylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]benzamideHuman5172
MAPK14 (p38a)MAPKCMGC3fknA3-[2-chloro-5-(methylsulfonyl)phenyl]-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidineHuman5049
MAPK14 (p38a)MAPKCMGC3fkoA3-(2-chlorophenyl)-6-(2-fluorophenoxy)-2h-indazoleHuman5075
MAPK14 (p38a)MAPKCMGC3fl4A6-(2,4-difluorophenoxy)-3-(2-methylphenyl)-1h-pyrazolo[3,4-d]pyrimidineHuman5151
MAPK14 (p38a)MAPKCMGC3flnC6-(2,4-difluorophenoxy)-8-methyl-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5090
MAPK14 (p38a)MAPKCMGC3flqA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5168
MAPK14 (p38a)MAPKCMGC3flsA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5119
MAPK14 (p38a)MAPKCMGC3flwA6-(2,4-difluorophenoxy)-2-{[3-hydroxy-1-(2-hydroxyethyl)propyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman5153
MAPK14 (p38a)MAPKCMGC3flyA6-(2,4-difluorophenoxy)-8-methyl-2-[(1-methylethyl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5113
MAPK14 (p38a)MAPKCMGC3flzA8-methyl-6-phenoxy-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5204
MAPK14 (p38a)MAPKCMGC3fmhA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5024
MAPK14 (p38a)MAPKCMGC3fmjA4-(5-methyl-3-phenylisoxazol-4-yl)pyrimidin-2-amineHuman5129
MAPK14 (p38a)MAPKCMGC3fmkA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5209
MAPK14 (p38a)MAPKCMGC3fmlA6-(2,4-difluorophenoxy)-n-[(1s)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman5010
MAPK14 (p38a)MAPKCMGC3fmmA6-(2,4-difluorophenoxy)-n-[(1r)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman5186
MAPK14 (p38a)MAPKCMGC3fmnAA6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman5196
MAPK14 (p38a)MAPKCMGC3fmnAB6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman4995
MAPK14 (p38a)MAPKCMGC3fsfA3-(2,6-dichlorophenyl)-7-({4-[(diethylamino)methoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman5097
MAPK14 (p38a)MAPKCMGC3fskA3-(2-chlorophenyl)-7-[(trans-4-hydroxycyclohexyl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman5008
MAPK14 (p38a)MAPKCMGC3gc7AA5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman5061
MAPK14 (p38a)MAPKCMGC3gc7AB5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman5256
MAPK14 (p38a)MAPKCMGC3gcpAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5194
MAPK14 (p38a)MAPKCMGC3gcpAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5157
MAPK14 (p38a)MAPKCMGC3gcqAA1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5066
MAPK14 (p38a)MAPKCMGC3gcqAB1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5053
MAPK14 (p38a)MAPKCMGC3gcsAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5077
MAPK14 (p38a)MAPKCMGC3gcsAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5052
MAPK14 (p38a)MAPKCMGC3gcuAA1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5032
MAPK14 (p38a)MAPKCMGC3gcuAB1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5162
MAPK14 (p38a)MAPKCMGC3gcuBA1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5175
MAPK14 (p38a)MAPKCMGC3gcuBB1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5126
MAPK14 (p38a)MAPKCMGC3gcvAA1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5088
MAPK14 (p38a)MAPKCMGC3gcvAB1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5174
MAPK14 (p38a)MAPKCMGC3gfeAn-cyclopropyl-3-{[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-4-yl]amino}-4-methylbenzamideHuman4991
MAPK14 (p38a)MAPKCMGC3gi3An-{5-tert-butyl-2-methoxy-3-[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]naphthalen-1-yl}carbamoyl)amino]phenyl}methanesulfonamideHuman5226
MAPK14 (p38a)MAPKCMGC3ha8AAn~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamideHuman5253
MAPK14 (p38a)MAPKCMGC3ha8ABn~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamideHuman5187
MAPK14 (p38a)MAPKCMGC3hecAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman5166
MAPK14 (p38a)MAPKCMGC3hecAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman5035
MAPK14 (p38a)MAPKCMGC3hegAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5112
MAPK14 (p38a)MAPKCMGC3hegAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5218
MAPK14 (p38a)MAPKCMGC3hl7A2-{4-[5-(4-chlorophenyl)-4-pyrimidin-4-yl-1h-pyrazol-3-yl]piperidin-1-yl}-2-oxoethanolHuman5236
MAPK14 (p38a)MAPKCMGC3hllAA3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamideHuman5115
MAPK14 (p38a)MAPKCMGC3hllAB3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamideHuman5104
MAPK14 (p38a)MAPKCMGC3hp2AA1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-oneHuman5217
MAPK14 (p38a)MAPKCMGC3hp2AB1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-oneHuman5031
MAPK14 (p38a)MAPKCMGC3hp5A5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman5158
MAPK14 (p38a)MAPKCMGC3hrbA[3-amino-2-(2-methylphenyl)-1-oxidopyridin-4-yl](2,4-difluorophenyl)methanoneHuman5202
MAPK14 (p38a)MAPKCMGC3hubA2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamideHuman5029
MAPK14 (p38a)MAPKCMGC3hucAAn-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamideHuman5027
MAPK14 (p38a)MAPKCMGC3hucABn-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamideHuman5111
MAPK14 (p38a)MAPKCMGC3hv3AA1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5012
MAPK14 (p38a)MAPKCMGC3hv3AB1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5232
MAPK14 (p38a)MAPKCMGC3hv4A1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5121
MAPK14 (p38a)MAPKCMGC3hv4B1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5064
MAPK14 (p38a)MAPKCMGC3hv5AA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5203
MAPK14 (p38a)MAPKCMGC3hv5AB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5263
MAPK14 (p38a)MAPKCMGC3hv5BA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5085
MAPK14 (p38a)MAPKCMGC3hv5BB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5137
MAPK14 (p38a)MAPKCMGC3hv6A1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(2-morpholin-4-ylethoxy)phenyl]ureaHuman5101
MAPK14 (p38a)MAPKCMGC3hv7A1-[1-(3-aminophenyl)-3-tert-butyl-1h-pyrazol-5-yl]-3-naphthalen-1-ylureaHuman5223
MAPK14 (p38a)MAPKCMGC3hvcA4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridineHuman5054
MAPK14 (p38a)MAPKCMGC3iphAA6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamideHuman4999
MAPK14 (p38a)MAPKCMGC3iphAB6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamideHuman5156
MAPK14 (p38a)MAPKCMGC3itzA4-chloro-n-cyclopropyl-3-{[1-(2,6-difluorophenyl)-1h-pyrazolo[3,4-d]pyridazin-4-yl]amino}benzamideHuman5135
MAPK14 (p38a)MAPKCMGC3iw5An-[2-(3-{[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl}-1h-indol-1-yl)ethyl]-3-(trifluoromethyl)benzamideHuman5076
MAPK14 (p38a)MAPKCMGC3iw6AAethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylateHuman4990
MAPK14 (p38a)MAPKCMGC3iw6ABethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylateHuman5154
MAPK14 (p38a)MAPKCMGC3iw7A2-({4-[(4-benzylpiperidin-1-yl)carbonyl]benzyl}sulfanyl)-3h-imidazo[4,5-c]pyridineHuman5084
MAPK14 (p38a)MAPKCMGC3iw8A1-{4-[(1s)-1-amino-2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-(3-chloro-4-fluorophenyl)ureaHuman5181
MAPK14 (p38a)MAPKCMGC3k3iAA(3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinolineHuman5212
MAPK14 (p38a)MAPKCMGC3k3iAB(3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinolineHuman5022
MAPK14 (p38a)MAPKCMGC3k3jA2-(4-fluorophenyl)-3-oxo-6-pyridin-4-yl-n-[2-(trifluoromethyl)benzyl]-2,3-dihydropyridazine-4-carboxamideHuman5047
MAPK14 (p38a)MAPKCMGC3kf7A3-{6-[2-(2,4-difluorophenyl)ethyl][1,2,4]triazolo[4,3-a]pyridin-3-yl}-4-methylbenzamideHuman5201
MAPK14 (p38a)MAPKCMGC3kq7AAn-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamideHuman5081
MAPK14 (p38a)MAPKCMGC3kq7ABn-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamideHuman5057
MAPK14 (p38a)MAPKCMGC3l8sA3-[(4-bromo-2,6-difluorobenzyl)oxy]-5-{[(4-pyrrolidin-1-ylbutyl)carbamoyl]amino}isothiazole-4-carboxamideHuman5055
MAPK14 (p38a)MAPKCMGC3l8xAn,4-dimethyl-3-[(1-phenyl-1h-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman5041
MAPK14 (p38a)MAPKCMGC3lfaAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman5018
MAPK14 (p38a)MAPKCMGC3lfbAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)ureaHuman4998
MAPK14 (p38a)MAPKCMGC3lfbAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)ureaHuman5001
MAPK14 (p38a)MAPKCMGC3lfcA(4-{5-[({4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}carbamoyl)amino]-3-tert-butyl-1h-pyrazol-1-yl}phenyl)acetic acidHuman5160
MAPK14 (p38a)MAPKCMGC3lfdA1-{4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5102
MAPK14 (p38a)MAPKCMGC3lfeA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-4-ylmethoxy)ethyl]-1,3-thiazol-2-yl}ureaHuman5173
MAPK14 (p38a)MAPKCMGC3lffAA(4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acidHuman5140
MAPK14 (p38a)MAPKCMGC3lffAB(4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acidHuman5120
MAPK14 (p38a)MAPKCMGC3lhjAn-cyclopropyl-3-[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamideHuman5234
MAPK14 (p38a)MAPKCMGC3mgyA-Human5171
MAPK14 (p38a)MAPKCMGC3mh0A-Human5124
MAPK14 (p38a)MAPKCMGC3mh1A-Human5003
MAPK14 (p38a)MAPKCMGC3mh2A-Human4985
MAPK14 (p38a)MAPKCMGC3mh3A-Human5109
MAPK14 (p38a)MAPKCMGC3mpaA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5026
MAPK14 (p38a)MAPKCMGC3mptAAn-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamideHuman5224
MAPK14 (p38a)MAPKCMGC3mptABn-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamideHuman5246
MAPK14 (p38a)MAPKCMGC3mvlA4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5060
MAPK14 (p38a)MAPKCMGC3mvlB4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5091
MAPK14 (p38a)MAPKCMGC3mvmA4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman4993
MAPK14 (p38a)MAPKCMGC3mvmB4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5210
MAPK14 (p38a)MAPKCMGC3mw1A8-(2,6-dichlorophenyl)-4-(2,4-difluorophenyl)-2-piperidin-4-yl-1,7-naphthyridine 7-oxideHuman5072
MAPK14 (p38a)MAPKCMGC3newAA-Human5025
MAPK14 (p38a)MAPKCMGC3newAB-Human5248
MAPK14 (p38a)MAPKCMGC3nnuAA2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamideHuman5094
MAPK14 (p38a)MAPKCMGC3nnuAB2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamideHuman5059
MAPK14 (p38a)MAPKCMGC3nnvAA1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylureaHuman5037
MAPK14 (p38a)MAPKCMGC3nnvAB1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylureaHuman5046
MAPK14 (p38a)MAPKCMGC3nnwAA2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamideHuman5139
MAPK14 (p38a)MAPKCMGC3nnwAB2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamideHuman5138
MAPK14 (p38a)MAPKCMGC3nnxA2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamideHuman5002
MAPK14 (p38a)MAPKCMGC3nwwA1-[2-(2-{[2-(dimethylamino)ethyl]amino}-6-{2-[(1-methylethyl)amino]-1,3-thiazol-5-yl}pyrimidin-4-yl)benzyl]-3-ethylureaHuman5068
MAPK14 (p38a)MAPKCMGC3o8pA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5071
MAPK14 (p38a)MAPKCMGC3o8tA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5167
MAPK14 (p38a)MAPKCMGC3o8uA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5250
MAPK14 (p38a)MAPKCMGC3obgA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5211
MAPK14 (p38a)MAPKCMGC3objA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman4994
MAPK14 (p38a)MAPKCMGC3oc1A1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5019
MAPK14 (p38a)MAPKCMGC3ocgA5-amino-n-[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]-1-phenyl-1h-pyrazole-4-carboxamideHuman4984
MAPK14 (p38a)MAPKCMGC3od6X-Human5134
MAPK14 (p38a)MAPKCMGC3odyX-Human5233
MAPK14 (p38a)MAPKCMGC3odzX-Human5069
MAPK14 (p38a)MAPKCMGC3oefXA-Human5163
MAPK14 (p38a)MAPKCMGC3oefXB-Human5231
MAPK14 (p38a)MAPKCMGC3pg3AA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}ureaHuman5122
MAPK14 (p38a)MAPKCMGC3pg3AB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}ureaHuman5096
MAPK14 (p38a)MAPKCMGC3qudAA{4-[(2-aminophenyl)amino]phenyl}(phenyl)methanoneHuman5006
MAPK14 (p38a)MAPKCMGC3qudAB{4-[(2-aminophenyl)amino]phenyl}(phenyl)methanoneHuman5262
MAPK14 (p38a)MAPKCMGC3queA2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-oneHuman5095
MAPK14 (p38a)MAPKCMGC3rinAn-cyclopropyl-4-methyl-3-(2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indol]-6'-yl)benzamideHuman5239
MAPK14 (p38a)MAPKCMGC3rocA3-{5-chloro-4-[(2,4-difluorobenzyl)oxy]-6-oxopyrimidin-1(6h)-yl}-n-(2-hydroxyethyl)-4-methylbenzamideHuman5011
MAPK14 (p38a)MAPKCMGC3s3iA3-(3-tert-butyl[1,2,4]triazolo[4,3-a]pyridin-7-yl)-n-cyclopropyl-4-methylbenzamideHuman5169
MAPK14 (p38a)MAPKCMGC3s4qA3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-n-cyclopropyl-4-methylbenzamideHuman5133
MAPK14 (p38a)MAPKCMGC3u8wA3-[3-(2-chloro-6-fluorophenyl)-5-ethyl-6-oxo-5,6-dihydro[1,2,4]triazolo[4,3-b]pyridazin-7-yl]-n-cyclopropyl-4-methylbenzamideHuman5192
MAPK14 (p38a)MAPKCMGC3uvpAAn-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamideHuman5070
MAPK14 (p38a)MAPKCMGC3uvpABn-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamideHuman5155
MAPK14 (p38a)MAPKCMGC3uvqAAn-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamideHuman5183
MAPK14 (p38a)MAPKCMGC3uvqABn-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamideHuman5214
MAPK14 (p38a)MAPKCMGC3uvrAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}ureaHuman6880
MAPK14 (p38a)MAPKCMGC3uvrAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}ureaHuman6879
MAPK14 (p38a)MAPKCMGC3zs5AA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman4987
MAPK14 (p38a)MAPKCMGC3zs5AB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman4977
MAPK14 (p38a)MAPKCMGC3zsgAAtak-715Human5033
MAPK14 (p38a)MAPKCMGC3zsgABtak-715Human5098
MAPK14 (p38a)MAPKCMGC3zshAA2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamideHuman5216
MAPK14 (p38a)MAPKCMGC3zshAB2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamideHuman5118
MAPK14 (p38a)MAPKCMGC3zsiAA5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman5056
MAPK14 (p38a)MAPKCMGC3zsiAB5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman4983
MAPK14 (p38a)MAPKCMGC3zyaAA2-amino-phenylamino-dibenzosuberoneHuman5105
MAPK14 (p38a)MAPKCMGC3zyaAB2-amino-phenylamino-dibenzosuberoneHuman5089
MAPK14 (p38a)MAPKCMGC4a9yAn-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamideHuman5073
MAPK14 (p38a)MAPKCMGC4aa0AAn-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamideHuman5213
MAPK14 (p38a)MAPKCMGC4aa0ABn-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamideHuman5132
MAPK14 (p38a)MAPKCMGC4aa4An-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]furan-3-carboxamideHuman5045
MAPK14 (p38a)MAPKCMGC4aa5An-cyclopropyl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]benzamideHuman5206
MAPK14 (p38a)MAPKCMGC4aacAn-isoxazol-3-yl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxo-quinazolin-3-yl]benzamideHuman5048
MAPK14 (p38a)MAPKCMGC4dliA-Human5092
MAPK14 (p38a)MAPKCMGC4dljA2-phenyl-n~4~-(2-phenylethyl)quinazoline-4,7-diamineHuman5242
MAPK14 (p38a)MAPKCMGC4e5aXA-Human5189
MAPK14 (p38a)MAPKCMGC4e5aXB-Human5222
MAPK14 (p38a)MAPKCMGC4e5bA-Human5221
MAPK14 (p38a)MAPKCMGC4e6aA-Human5238
MAPK14 (p38a)MAPKCMGC4e6cA-Human5015
MAPK14 (p38a)MAPKCMGC4e8aA-Human4979
MAPK14 (p38a)MAPKCMGC4eh2A3-phenylquinazolin-4(3h)-oneHuman5244
MAPK14 (p38a)MAPKCMGC4eh3AnaringeninHuman5042
MAPK14 (p38a)MAPKCMGC4eh4Aphenyl(piperidin-1-yl)methanoneHuman5043
MAPK14 (p38a)MAPKCMGC4eh5Abenzyl pyridine-3-carboxylateHuman5185
MAPK14 (p38a)MAPKCMGC4eh6An-phenylpyridine-3-carboxamideHuman5083
MAPK14 (p38a)MAPKCMGC4eh7AA(3-phenoxyphenyl)methanolHuman5208
MAPK14 (p38a)MAPKCMGC4eh7AB(3-phenoxyphenyl)methanolHuman5020
MAPK14 (p38a)MAPKCMGC4eh8AA[3-(benzyloxy)phenyl]methanolHuman4978
MAPK14 (p38a)MAPKCMGC4eh8AB[3-(benzyloxy)phenyl]methanolHuman5014
MAPK14 (p38a)MAPKCMGC4eh9A-Human4982
MAPK14 (p38a)MAPKCMGC4ehvAA-Human4997
MAPK14 (p38a)MAPKCMGC4ehvAB-Human4981
MAPK14 (p38a)MAPKCMGC4ewqAA3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazineHuman5200
MAPK14 (p38a)MAPKCMGC4ewqAB3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazineHuman5245
MAPK14 (p38a)MAPKCMGC4f9wAAn,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5130
MAPK14 (p38a)MAPKCMGC4f9wABn,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5106
MAPK14 (p38a)MAPKCMGC4f9yAAn,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5225
MAPK14 (p38a)MAPKCMGC4f9yABn,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5017
MAPK14 (p38a)MAPKCMGC4fa2AAtrans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanolHuman5150
MAPK14 (p38a)MAPKCMGC4fa2ABtrans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanolHuman5145
MAPK14 (p38a)MAPKCMGC4geoA-Human5190
MAPK14 (p38a)MAPKCMGC4kinA5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5237
MAPK14 (p38a)MAPKCMGC4kinB5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5131
MAPK14 (p38a)MAPKCMGC4kinC5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5142
MAPK14 (p38a)MAPKCMGC4kinD5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5144
MAPK14 (p38a)MAPKCMGC4kipA2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamideHuman5159
MAPK14 (p38a)MAPKCMGC4kipB2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamideHuman5180
MAPK14 (p38a)MAPKCMGC4kiqAethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5141
MAPK14 (p38a)MAPKCMGC4kiqBethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5013
MAPK14 (p38a)MAPKCMGC4kiqCethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5215
MAPK14 (p38a)MAPKCMGC4kiqDethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5016
MAPK14 (p38a)MAPKCMGC4l8mAAn-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamideHuman5005
MAPK14 (p38a)MAPKCMGC4l8mABn-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamideHuman4992
MAPK14 (p38a)MAPKCMGC4r3cAA6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazineHuman5198
MAPK14 (p38a)MAPKCMGC4r3cAB6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazineHuman5036
MAPK14 (p38a)MAPKCMGC4zthAA6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazineHuman6706
MAPK14 (p38a)MAPKCMGC4zthAB6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazineHuman6707
MAPK14 (p38a)MAPKCMGC5etaA-Human7136
MAPK14 (p38a)MAPKCMGC5etaB-Human7137
MAPK14 (p38a)MAPKCMGC5etcA-Human6361
MAPK14 (p38a)MAPKCMGC5etfAA-Human7134
MAPK14 (p38a)MAPKCMGC5etfAB-Human7135
MAPK14 (p38a)MAPKCMGC5etiA-Human6362
MAPK14 (p38a)MAPKCMGC5ml5A3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-methylsulfanyl-1~{h}-imidazol-5-yl]pyridin-2-yl]propanamideHuman7544
MAPK14 (p38a)MAPKCMGC5mtxAA3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamideHuman8382
MAPK14 (p38a)MAPKCMGC5mtxAB3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamideHuman8379
MAPK14 (p38a)MAPKCMGC5mtyA~{n}-[2,4-bis(fluoranyl)-5-[[14-(2-hydroxyethylcarbamoyl)-2-oxidanylidene-6-tricyclo[9.4.0.0^{3,8}]pentadeca-1(15),3(8),4,6,11,13-hexaenyl]amino]phenyl]thiophene-2-carboxamideHuman8383
MAPK14 (p38a)MAPKCMGC5mz3AA~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8680
MAPK14 (p38a)MAPKCMGC5mz3AB~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8681
MAPK14 (p38a)MAPKCMGC5n63A-Human8526
MAPK14 (p38a)MAPKCMGC5n64A-Human8527
MAPK14 (p38a)MAPKCMGC5n65A2-phenyl-~{n}4-(2-thiophen-2-ylethyl)quinazoline-4,7-diamineHuman8525
MAPK14 (p38a)MAPKCMGC5n66A1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman8524
MAPK14 (p38a)MAPKCMGC5n67AA-Human8523
MAPK14 (p38a)MAPKCMGC5n67AB-Human8521
MAPK14 (p38a)MAPKCMGC5n68A-Human8522
MAPK14 (p38a)MAPKCMGC5o8uA-Human8381
MAPK14 (p38a)MAPKCMGC5o8vA-Human8380
MAPK14 (p38a)MAPKCMGC5omgAA3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxideHuman11246
MAPK14 (p38a)MAPKCMGC5omgAB3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxideHuman11245
MAPK14 (p38a)MAPKCMGC5omhA1-(3-chlorophenyl)-3-methyl-4~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxideHuman11251
MAPK14 (p38a)MAPKCMGC5tbeA~{n}-[2,4-bis(fluoranyl)-5-[[9-(2-morpholin-4-ylethylcarbamoyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulen-3-yl]amino]phenyl]thiophene-2-carboxamideHuman8032
MAPK14 (p38a)MAPKCMGC5tcoA3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulene-9-carboxamideHuman8031
MAPK14 (p38a)MAPKCMGC5wjjAAn-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamideHuman9514
MAPK14 (p38a)MAPKCMGC5wjjABn-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamideHuman9516
MAPK14 (p38a)MAPKCMGC5xyxAAn-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amineHuman9519
MAPK14 (p38a)MAPKCMGC5xyxABn-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amineHuman9517
MAPK14 (p38a)MAPKCMGC5xyyA3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-4h-1,2,4-triazol-3-yl)phenolHuman9513
MAPK14 (p38a)MAPKCMGC6anlAAtak-715Human9515
MAPK14 (p38a)MAPKCMGC6anlABtak-715Human9518
MAPK14 (p38a)MAPKCMGC6hwtAA3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamideHuman11248
MAPK14 (p38a)MAPKCMGC6hwtAB3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamideHuman11254
MAPK14 (p38a)MAPKCMGC6hwuAA-Human11247
MAPK14 (p38a)MAPKCMGC6hwuAB-Human11249
MAPK14 (p38a)MAPKCMGC6hwvAA-Human11253
MAPK14 (p38a)MAPKCMGC6hwvAB-Human11250
MAPK14 (p38a)MAPKCMGC6m95A(4-benzylpiperidin-1-yl)[2-methoxy-4-(methylsulfanyl)phenyl]methanoneHuman11252
MAPK14 (p38a)MAPKCMGC6m9lA3-benzyl-6-[(2,4-difluorophenyl)amino]-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-oneHuman11255
MAPK14 (p38a)MAPKCMGC6ohdAA3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamideHuman11818
MAPK14 (p38a)MAPKCMGC6ohdAB3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamideHuman11819
MAPK14 (p38a)MAPKCMGC6qdzAA1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ureaHuman11956
MAPK14 (p38a)MAPKCMGC6qdzAB1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ureaHuman11958
MAPK14 (p38a)MAPKCMGC6qe1A1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{r})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ureaHuman11957
MAPK14 (p38a)MAPKCMGC6qyxA-Human12127
MAPK14 (p38a)MAPKCMGC6sfiAA~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamideHuman11613
MAPK14 (p38a)MAPKCMGC6sfiAB~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamideHuman11619
MAPK14 (p38a)MAPKCMGC6sfjAA~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamideHuman11614
MAPK14 (p38a)MAPKCMGC6sfjAB~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamideHuman11616
MAPK14 (p38a)MAPKCMGC6sfjAC~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamideHuman11618
MAPK14 (p38a)MAPKCMGC6sfkAA~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamideHuman11617
MAPK14 (p38a)MAPKCMGC6sfkAB~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamideHuman11620
MAPK14 (p38a)MAPKCMGC6sfoAA5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman11615
MAPK14 (p38a)MAPKCMGC6sfoAB5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman11621
MAPK14 (p38a)MAPKCMGC6tcaBAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12491
MAPK14 (p38a)MAPKCMGC6tcaBBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12488
MAPK14 (p38a)MAPKCMGC6tcaDAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12486
MAPK14 (p38a)MAPKCMGC6tcaDBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12492
MAPK14 (p38a)MAPKCMGC6tcaFAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12489
MAPK14 (p38a)MAPKCMGC6tcaFBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12490
MAPK14 (p38a)MAPKCMGC6tcaHAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12493
MAPK14 (p38a)MAPKCMGC6tcaHBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12487
MAPK14 (p38a)MAPKCMGC6zqsA2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-oneHuman12986
MAPK14 (p38a)MAPKCMGC6zwpAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman12699
MAPK14 (p38a)MAPKCMGC6zwpAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman12698
MAPK14 (p38a)MAPKCMGC8a8mAphosphomethylphosphonic acid adenosyl esterHuman14289
MAPK3 (Erk1)MAPKCMGC2zoqA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman1716
MAPK3 (Erk1)MAPKCMGC2zoqB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman1712
MAPK3 (Erk1)MAPKCMGC4qtbAA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman1714
MAPK3 (Erk1)MAPKCMGC4qtbAB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman1713
MAPK3 (Erk1)MAPKCMGC4qtbBA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman1717
MAPK3 (Erk1)MAPKCMGC4qtbBB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman1715
MAPK3 (Erk1)MAPKCMGC6gesAAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10923
MAPK3 (Erk1)MAPKCMGC6gesABn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10926
MAPK3 (Erk1)MAPKCMGC6gesBAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10925
MAPK3 (Erk1)MAPKCMGC6gesBBn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10924
MAPK6 (Erk3)MAPKCMGC6ykyAA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12788
MAPK6 (Erk3)MAPKCMGC6ykyAB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12790
MAPK6 (Erk3)MAPKCMGC6ykyBA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12792
MAPK6 (Erk3)MAPKCMGC6ykyBB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12786
MAPK6 (Erk3)MAPKCMGC6ykyCA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12787
MAPK6 (Erk3)MAPKCMGC6ykyCB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12784
MAPK6 (Erk3)MAPKCMGC6ykyDA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12796
MAPK6 (Erk3)MAPKCMGC6ykyDB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12789
MAPK6 (Erk3)MAPKCMGC6ylcA5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12791
MAPK6 (Erk3)MAPKCMGC6ylcB5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12797
MAPK6 (Erk3)MAPKCMGC6ylcC5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12794
MAPK6 (Erk3)MAPKCMGC6ylcD5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12795
MAPK6 (Erk3)MAPKCMGC6yllA~{n}4-[3-(4-methoxyphenyl)-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]cyclohexane-1,4-diamineHuman12793
MAPK6 (Erk3)MAPKCMGC6yllB-Human12785
MAPK6 (Erk3)MAPKCMGC7aqbAA-Human12982
MAPK6 (Erk3)MAPKCMGC7aqbAB-Human12981
MAPK6 (Erk3)MAPKCMGC7aqbBA-Human12980
MAPK6 (Erk3)MAPKCMGC7aqbBB-Human12983
MAPK7 (Erk5)MAPKCMGC4b99A11-cyclopentyl-2-[[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl-phenyl]amino]-5-methyl-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman388
MAPK7 (Erk5)MAPKCMGC4ic7Aphosphoaminophosphonic acid-adenylate esterHuman392
MAPK7 (Erk5)MAPKCMGC4ic7Dphosphoaminophosphonic acid-adenylate esterHuman391
MAPK7 (Erk5)MAPKCMGC4ic8A-Human390
MAPK7 (Erk5)MAPKCMGC4ic8B-Human389
MAPK7 (Erk5)MAPKCMGC4zsgAA3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6589
MAPK7 (Erk5)MAPKCMGC4zsgAB3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6584
MAPK7 (Erk5)MAPKCMGC4zsjAA3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6588
MAPK7 (Erk5)MAPKCMGC4zsjAB3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6585
MAPK7 (Erk5)MAPKCMGC4zslA3-amino-5-[(4-chlorophenyl)amino]-n-[(1s)-1-phenylethyl]-1h-1,2,4-triazole-1-carboxamideHuman6586
MAPK7 (Erk5)MAPKCMGC5byyAA2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman6591
MAPK7 (Erk5)MAPKCMGC5byyAB2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman6587
MAPK7 (Erk5)MAPKCMGC5byzAA4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamideHuman6590
MAPK7 (Erk5)MAPKCMGC5byzAB4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamideHuman6592
MAPK7 (Erk5)MAPKCMGC5o7iAA4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamideHuman9995
MAPK7 (Erk5)MAPKCMGC5o7iAB4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamideHuman9994
MAPK7 (Erk5)MAPKCMGC6hkmA[4-(6,7-dimethoxyquinazolin-4-yl)piperidin-1-yl]-[4-(trifluoromethyloxy)phenyl]methanoneHuman10917
MAPK7 (Erk5)MAPKCMGC6hknAA[2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanoneHuman10918
MAPK7 (Erk5)MAPKCMGC6hknAB[2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanoneHuman10919
MAPK7 (Erk5)MAPKCMGC7pusAA4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamideHuman14218
MAPK7 (Erk5)MAPKCMGC7pusAB4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamideHuman14219
MAPK8 (JNK1)MAPKCMGC1ukhA-Human4628
MAPK8 (JNK1)MAPKCMGC1ukiA2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHuman4630
MAPK8 (JNK1)MAPKCMGC2g01A6-chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4h-pyrazolo[3,4-b]quinolin-4-oneHuman4662
MAPK8 (JNK1)MAPKCMGC2g01B6-chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4h-pyrazolo[3,4-b]quinolin-4-oneHuman4641
MAPK8 (JNK1)MAPKCMGC2gmxAn-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-bromo-2,5-dimethoxyphenyl)acetamideHuman4674
MAPK8 (JNK1)MAPKCMGC2gmxBn-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-bromo-2,5-dimethoxyphenyl)acetamideHuman4638
MAPK8 (JNK1)MAPKCMGC2h96A5-cyano-n-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamideHuman4655
MAPK8 (JNK1)MAPKCMGC2h96B5-cyano-n-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamideHuman4668
MAPK8 (JNK1)MAPKCMGC2no3A2-({2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}amino)benzamideHuman4640
MAPK8 (JNK1)MAPKCMGC2no3B2-({2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}amino)benzamideHuman4657
MAPK8 (JNK1)MAPKCMGC2xrwAAphosphoaminophosphonic acid-adenylate esterHuman4675
MAPK8 (JNK1)MAPKCMGC2xrwABphosphoaminophosphonic acid-adenylate esterHuman4650
MAPK8 (JNK1)MAPKCMGC2xrwACphosphoaminophosphonic acid-adenylate esterHuman4660
MAPK8 (JNK1)MAPKCMGC2xs0Aphosphoaminophosphonic acid-adenylate esterHuman4629
MAPK8 (JNK1)MAPKCMGC3eljAA2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamideHuman4658
MAPK8 (JNK1)MAPKCMGC3eljAB2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamideHuman4636
MAPK8 (JNK1)MAPKCMGC3o17A-Human4670
MAPK8 (JNK1)MAPKCMGC3o17B-Human4667
MAPK8 (JNK1)MAPKCMGC3o2mA-Human4676
MAPK8 (JNK1)MAPKCMGC3o2mB-Human4649
MAPK8 (JNK1)MAPKCMGC3pzeA3-(carbamoylamino)-5-phenylthiophene-2-carboxamideHuman4642
MAPK8 (JNK1)MAPKCMGC3v3vA3,5,6,7-tetrahydroxy-2-(3,4-dihydroxyphenyl)-4h-chromen-4-oneHuman4653
MAPK8 (JNK1)MAPKCMGC3vudA-Human4664
MAPK8 (JNK1)MAPKCMGC3vugA-Human4665
MAPK8 (JNK1)MAPKCMGC3vuhA-Human4663
MAPK8 (JNK1)MAPKCMGC3vuiA-Human4652
MAPK8 (JNK1)MAPKCMGC3vukA-Human4659
MAPK8 (JNK1)MAPKCMGC3vulA-Human4633
MAPK8 (JNK1)MAPKCMGC3vumA-Human4671
MAPK8 (JNK1)MAPKCMGC4awiAAn-(1,1-dioxidotetrahydro-2h-thiopyran-4-yl)-4-[2-(1-methylethyl)-1h-pyrrolo[2,3-b]pyridin-4-yl]benzenesulfonamideHuman4661
MAPK8 (JNK1)MAPKCMGC4awiABn-(1,1-dioxidotetrahydro-2h-thiopyran-4-yl)-4-[2-(1-methylethyl)-1h-pyrrolo[2,3-b]pyridin-4-yl]benzenesulfonamideHuman4634
MAPK8 (JNK1)MAPKCMGC4e73AAmethyl 3-(4-{[(1r,2s,3s,5s,7s)-5-aminotricyclo[3.3.1.1~3,7~]dec-2-yl]carbamoyl}benzyl)-4-oxo-1-phenyl-1,4-dihydro-1,8-naphthyridine-2-carboxylateHuman4645
MAPK8 (JNK1)MAPKCMGC4e73ABmethyl 3-(4-{[(1r,2s,3s,5s,7s)-5-aminotricyclo[3.3.1.1~3,7~]dec-2-yl]carbamoyl}benzyl)-4-oxo-1-phenyl-1,4-dihydro-1,8-naphthyridine-2-carboxylateHuman4669
MAPK8 (JNK1)MAPKCMGC4g1wAmethyl 7-fluoro-3-{4-[(2-hydroxyethyl)sulfonyl]benzyl}-4-oxo-1-phenyl-1,4-dihydroquinoline-2-carboxylateHuman4631
MAPK8 (JNK1)MAPKCMGC4hysAtrans-4-{[4-(1h-indazol-1-yl)pyrimidin-2-yl]amino}cyclohexanolHuman4672
MAPK8 (JNK1)MAPKCMGC4hyuAtrans-4-[(4-{4-[3-(methylsulfonyl)propoxy]-1h-indazol-1-yl}pyrimidin-2-yl)amino]cyclohexanolHuman4632
MAPK8 (JNK1)MAPKCMGC4izyAtrans-4-[(4-{4-[4-(methylsulfonyl)piperidin-1-yl]-1h-indol-1-yl}pyrimidin-2-yl)amino]cyclohexanolHuman4654
MAPK8 (JNK1)MAPKCMGC4l7fAAn-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamideHuman4639
MAPK8 (JNK1)MAPKCMGC4l7fABn-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamideHuman4637
MAPK8 (JNK1)MAPKCMGC4l7fACn-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamideHuman4648
MAPK8 (JNK1)MAPKCMGC4qtdAA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman4651
MAPK8 (JNK1)MAPKCMGC4qtdAB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman4673
MAPK8 (JNK1)MAPKCMGC4ux9AAphosphoaminophosphonic acid-adenylate esterHuman4643
MAPK8 (JNK1)MAPKCMGC4ux9ABphosphoaminophosphonic acid-adenylate esterHuman4646
MAPK8 (JNK1)MAPKCMGC4ux9BAphosphoaminophosphonic acid-adenylate esterHuman4635
MAPK8 (JNK1)MAPKCMGC4ux9BBphosphoaminophosphonic acid-adenylate esterHuman4656
MAPK8 (JNK1)MAPKCMGC4ux9CAphosphoaminophosphonic acid-adenylate esterHuman4644
MAPK8 (JNK1)MAPKCMGC4ux9CBphosphoaminophosphonic acid-adenylate esterHuman4647
MAPK8 (JNK1)MAPKCMGC4ux9DAphosphoaminophosphonic acid-adenylate esterHuman4627
MAPK8 (JNK1)MAPKCMGC4ux9DBphosphoaminophosphonic acid-adenylate esterHuman4666
MAPK8 (JNK1)MAPKCMGC4yr8AA-Human6452
MAPK8 (JNK1)MAPKCMGC4yr8AB-Human6448
MAPK8 (JNK1)MAPKCMGC4yr8CA-Human6449
MAPK8 (JNK1)MAPKCMGC4yr8CB-Human6447
MAPK8 (JNK1)MAPKCMGC4yr8EA-Human6451
MAPK8 (JNK1)MAPKCMGC4yr8EB-Human6454
MAPK8 (JNK1)MAPKCMGC4yr8FA-Human6450
MAPK8 (JNK1)MAPKCMGC4yr8FB-Human6453
MAPK8 (JNK1)MAPKCMGC5lw1BadenosineHuman9081
MAPK8 (JNK1)MAPKCMGC5lw1EadenosineHuman9079
MAPK8 (JNK1)MAPKCMGC5lw1HadenosineHuman9080
MAPK8 (JNK1)MAPKCMGC6f5eB-Human9078
MAPK8 (JNK1)MAPKCMGC6zr5Aphosphoaminophosphonic acid-adenylate esterHuman12984
MAPK8 (JNK1)MAPKCMGC6zr5Bphosphoaminophosphonic acid-adenylate esterHuman12985
MAPK8 (JNK1)MAPKCMGC8x5mAA3-[4-(dimethylamino)butanoylamino]-~{n}-[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamideHuman15099
MAPK8 (JNK1)MAPKCMGC8x5mAB3-[4-(dimethylamino)butanoylamino]-~{n}-[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamideHuman15100
MAPK9 (JNK2)MAPKCMGC3e7oAn-{3-[5-(1h-1,2,4-triazol-3-yl)-1h-indazol-3-yl]phenyl}furan-2-carboxamideHuman1238
MAPK9 (JNK2)MAPKCMGC3e7oBn-{3-[5-(1h-1,2,4-triazol-3-yl)-1h-indazol-3-yl]phenyl}furan-2-carboxamideHuman1236
MAPK9 (JNK2)MAPKCMGC3npcA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman1235
MAPK9 (JNK2)MAPKCMGC3npcB1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman1237
MAPK9 (JNK2)MAPKCMGC7cmlAA-Human12707
MAPK9 (JNK2)MAPKCMGC7cmlAB-Human12705
MAPK9 (JNK2)MAPKCMGC7cmlBA-Human12706
MAPK9 (JNK2)MAPKCMGC7cmlBB-Human12704
MAPK9 (JNK2)MAPKCMGC7n8tAAadenosine monophosphateHuman14241
MAPK9 (JNK2)MAPKCMGC7n8tABadenosine monophosphateHuman14242
MAPK9 (JNK2)MAPKCMGC8elcA4-(dimethylamino)-n-{4-[(3s)-3-({4-[(8r)-2-phenylpyrazolo[1,5-a]pyridin-3-yl]pyrimidin-2-yl}amino)pyrrolidine-1-carbonyl]phenyl}butanamideHuman14816
MAPKAPK2MAPKAPKCAMK1kwpA-Human1280
MAPKAPK2MAPKAPKCAMK1kwpB-Human1296
MAPKAPK2MAPKAPKCAMK1nxkAstaurosporineHuman1342
MAPKAPK2MAPKAPKCAMK1nxkBstaurosporineHuman1292
MAPKAPK2MAPKAPKCAMK1nxkCstaurosporineHuman1312
MAPKAPK2MAPKAPKCAMK1nxkDstaurosporineHuman1334
MAPKAPK2MAPKAPKCAMK1ny3Aadenosine-5'-diphosphateHuman1318
MAPKAPK2MAPKAPKCAMK2jboA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1333
MAPKAPK2MAPKAPKCAMK2jbpA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1366
MAPKAPK2MAPKAPKCAMK2jbpB2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1320
MAPKAPK2MAPKAPKCAMK2jbpC2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1344
MAPKAPK2MAPKAPKCAMK2jbpD2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1327
MAPKAPK2MAPKAPKCAMK2jbpE2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1358
MAPKAPK2MAPKAPKCAMK2jbpF2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1335
MAPKAPK2MAPKAPKCAMK2jbpG2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1339
MAPKAPK2MAPKAPKCAMK2jbpH2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1326
MAPKAPK2MAPKAPKCAMK2jbpI2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1364
MAPKAPK2MAPKAPKCAMK2jbpJ-Human1359
MAPKAPK2MAPKAPKCAMK2jbpK2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1363
MAPKAPK2MAPKAPKCAMK2jbpL2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1283
MAPKAPK2MAPKAPKCAMK2onlC-Human1306
MAPKAPK2MAPKAPKCAMK2onlD-Human1345
MAPKAPK2MAPKAPKCAMK2ozaA-Human1310
MAPKAPK2MAPKAPKCAMK2p3gX2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1349
MAPKAPK2MAPKAPKCAMK2pzyA(4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamideHuman1314
MAPKAPK2MAPKAPKCAMK2pzyB(4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamideHuman1307
MAPKAPK2MAPKAPKCAMK2pzyCstaurosporineHuman1279
MAPKAPK2MAPKAPKCAMK2pzyD-Human1357
MAPKAPK2MAPKAPKCAMK3a2cAn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1330
MAPKAPK2MAPKAPKCAMK3a2cBn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1332
MAPKAPK2MAPKAPKCAMK3a2cCn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1328
MAPKAPK2MAPKAPKCAMK3a2cDn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1316
MAPKAPK2MAPKAPKCAMK3a2cEn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1315
MAPKAPK2MAPKAPKCAMK3a2cFn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1355
MAPKAPK2MAPKAPKCAMK3a2cGn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1343
MAPKAPK2MAPKAPKCAMK3a2cHn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1325
MAPKAPK2MAPKAPKCAMK3a2cIn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1311
MAPKAPK2MAPKAPKCAMK3a2cJn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1353
MAPKAPK2MAPKAPKCAMK3a2cKn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1360
MAPKAPK2MAPKAPKCAMK3a2cLn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1301
MAPKAPK2MAPKAPKCAMK3fpmA3-{[(1r)-1-phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dioneHuman1367
MAPKAPK2MAPKAPKCAMK3fyjX(10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-oneHuman1336
MAPKAPK2MAPKAPKCAMK3fykX(3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-oneHuman1297
MAPKAPK2MAPKAPKCAMK3gokA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1281
MAPKAPK2MAPKAPKCAMK3gokB2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1304
MAPKAPK2MAPKAPKCAMK3gokC2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1350
MAPKAPK2MAPKAPKCAMK3gokD2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1284
MAPKAPK2MAPKAPKCAMK3gokE2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1300
MAPKAPK2MAPKAPKCAMK3gokF2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1362
MAPKAPK2MAPKAPKCAMK3gokG2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1351
MAPKAPK2MAPKAPKCAMK3gokH2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1338
MAPKAPK2MAPKAPKCAMK3gokI2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1305
MAPKAPK2MAPKAPKCAMK3gokJ2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1319
MAPKAPK2MAPKAPKCAMK3gokK2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1299
MAPKAPK2MAPKAPKCAMK3gokL2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1365
MAPKAPK2MAPKAPKCAMK3ka0A6-{5-[(2-aminopyrimidin-4-yl)amino]-2-hydroxyphenyl}-n-methylidene-1-benzothiophene-2-carboxamideHuman1290
MAPKAPK2MAPKAPKCAMK3kc3An~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1289
MAPKAPK2MAPKAPKCAMK3kc3Bn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1298
MAPKAPK2MAPKAPKCAMK3kc3Cn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1303
MAPKAPK2MAPKAPKCAMK3kc3Dn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1288
MAPKAPK2MAPKAPKCAMK3kc3En~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1285
MAPKAPK2MAPKAPKCAMK3kc3Fn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1341
MAPKAPK2MAPKAPKCAMK3kc3G-Human1356
MAPKAPK2MAPKAPKCAMK3kc3Hn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1291
MAPKAPK2MAPKAPKCAMK3kc3In~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1354
MAPKAPK2MAPKAPKCAMK3kc3Jn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1347
MAPKAPK2MAPKAPKCAMK3kc3Kn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1317
MAPKAPK2MAPKAPKCAMK3kc3Ln~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1324
MAPKAPK2MAPKAPKCAMK3kgaAA6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-oneHuman9476
MAPKAPK2MAPKAPKCAMK3kgaAB6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-oneHuman9477
MAPKAPK2MAPKAPKCAMK3m2wAA2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-oneHuman9474
MAPKAPK2MAPKAPKCAMK3m2wAB2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-oneHuman9473
MAPKAPK2MAPKAPKCAMK3m42A2-[5-(2-methoxyethoxy)pyridin-3-yl]-8,9,10,11-tetrahydro-7h-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin-7-oneHuman9475
MAPKAPK2MAPKAPKCAMK3r2bA2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-oneHuman1287
MAPKAPK2MAPKAPKCAMK3r2bB2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-oneHuman1329
MAPKAPK2MAPKAPKCAMK3r2bC-Human1368
MAPKAPK2MAPKAPKCAMK3r2bD-Human1337
MAPKAPK2MAPKAPKCAMK3r2bE-Human1286
MAPKAPK2MAPKAPKCAMK3r2bF-Human1321
MAPKAPK2MAPKAPKCAMK3r2bG-Human1369
MAPKAPK2MAPKAPKCAMK3r2bH-Human1348
MAPKAPK2MAPKAPKCAMK3r2bI-Human1294
MAPKAPK2MAPKAPKCAMK3r2bJ-Human1331
MAPKAPK2MAPKAPKCAMK3r2bK-Human1293
MAPKAPK2MAPKAPKCAMK3r2bL-Human1295
MAPKAPK2MAPKAPKCAMK3r2yA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1361
MAPKAPK2MAPKAPKCAMK3r30AA1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acidHuman1352
MAPKAPK2MAPKAPKCAMK3r30AB1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acidHuman1309
MAPKAPK2MAPKAPKCAMK3wi6An-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1308
MAPKAPK2MAPKAPKCAMK3wi6Bn-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1282
MAPKAPK2MAPKAPKCAMK3wi6Cn-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1346
MAPKAPK2MAPKAPKCAMK3wi6Dn-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1340
MAPKAPK2MAPKAPKCAMK3wi6En-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1323
MAPKAPK2MAPKAPKCAMK3wi6Fn-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1313
MAPKAPK2MAPKAPKCAMK4tyhAA-Human1302
MAPKAPK2MAPKAPKCAMK4tyhAB-Human1322
MAPKAPK2MAPKAPKCAMK6t8xA(10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-oneHuman13548
MAPKAPK2MAPKAPKCAMK6tcaAA-Human12502
MAPKAPK2MAPKAPKCAMK6tcaAB-Human12507
MAPKAPK2MAPKAPKCAMK6tcaCA-Human12504
MAPKAPK2MAPKAPKCAMK6tcaCB-Human12506
MAPKAPK2MAPKAPKCAMK6tcaEA-Human12500
MAPKAPK2MAPKAPKCAMK6tcaEB-Human12503
MAPKAPK2MAPKAPKCAMK6tcaGA-Human12505
MAPKAPK2MAPKAPKCAMK6tcaGB-Human12501
MAPKAPK2MAPKAPKCAMK8xu4A-Human15173
MAPKAPK3MAPKAPKCAMK3fhrAA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4590
MAPKAPK3MAPKAPKCAMK3fhrAB2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4598
MAPKAPK3MAPKAPKCAMK3fxwAA2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4596
MAPKAPK3MAPKAPKCAMK3fxwAB2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4593
MAPKAPK3MAPKAPKCAMK3r1nAA2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-oneHuman4589
MAPKAPK3MAPKAPKCAMK3r1nAB2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-oneHuman4588
MAPKAPK3MAPKAPKCAMK3sheAAn-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamideHuman4594
MAPKAPK3MAPKAPKCAMK3sheABn-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamideHuman4599
MAPKAPK3MAPKAPKCAMK7nrbAA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman14052
MAPKAPK3MAPKAPKCAMK7nrbAB2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman14051
MARK1CAMKLCAMK2hakA-Human258
MARK1CAMKLCAMK2hakB-Human259
MARK1CAMKLCAMK2hakC-Human260
MARK1CAMKLCAMK2hakD-Human257
MARK1CAMKLCAMK2hakE-Human255
MARK1CAMKLCAMK2hakF-Human254
MARK1CAMKLCAMK2hakG-Human256
MARK1CAMKLCAMK2hakH-Human261
MARK1CAMKLCAMK6c9dAA-Human10052
MARK1CAMKLCAMK6c9dAB-Human10051
MARK1CAMKLCAMK6c9dBA-Human10049
MARK1CAMKLCAMK6c9dBB-Human10050
MARK2CAMKLCAMK3iecA-Human3045
MARK2CAMKLCAMK3iecB-Human3044
MARK2CAMKLCAMK3iecC-Human3046
MARK2CAMKLCAMK3iecD-Human3043
MARK2CAMKLCAMK5eakAn-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHuman6410
MARK2CAMKLCAMK5eakBn-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHuman6411
MARK2CAMKLCAMK5kz7A7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-oneHuman7967
MARK2CAMKLCAMK5kz7B7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-oneHuman7966
MARK2CAMKLCAMK5kz8A5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-oneHuman7965
MARK2CAMKLCAMK5kz8B5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-oneHuman7968
MARK2CAMKLCAMK8txyAn-[(5p,8r)-5-(2-cyano-5-{[(3r)-1-methylpyrrolidin-3-yl]methoxy}pyridin-4-yl)pyrazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamideHuman15136
MARK3CAMKLCAMK2qnjA-Human3269
MARK3CAMKLCAMK2qnjB-Human3264
MARK3CAMKLCAMK3fe3AA-Human3267
MARK3CAMKLCAMK3fe3AB-Human3266
MARK3CAMKLCAMK3fe3BA-Human3268
MARK3CAMKLCAMK3fe3BB-Human3265
MARK3CAMKLCAMK7p1lA5-bromo-4-n-[2-(1h-imidazol-5-yl)ethyl]-2-n-[3-(morpholin-4-ylmethyl)phenyl]pyrimidine-2,4-diamineHuman13799
MARK4CAMKLCAMK5es1A~{n}-[(1~{r},6~{r})-6-azanyl-2,2-bis(fluoranyl)cyclohexyl]-5-ethyl-4-[6-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHuman6260
MARK4CAMKLCAMK8xflA-Human15101
MASTLMASTAGC5lohAAstaurosporineHuman7086
MASTLMASTAGC5lohABstaurosporineHuman7085
MASTLMASTAGC5lohBAstaurosporineHuman7088
MASTLMASTAGC5lohBBstaurosporineHuman7087
Melk (MELK)CAMKLCAMK4bfmAphosphoaminophosphonic acid-adenylate esterMouse5798
Melk (MELK)CAMKLCAMK4cqgA1-[6-(3,5-dichloro-4-hydroxyphenyl)-4-({trans-4-[(dimethylamino)methyl]cyclohexyl}amino)-1,5-naphthyridin-3-yl]ethanoneMouse6865
MELKCAMKLCAMK4bkyAA3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamideHuman2480
MELKCAMKLCAMK4bkyAB3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamideHuman2490
MELKCAMKLCAMK4bkzAAn-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamideHuman2505
MELKCAMKLCAMK4bkzABn-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamideHuman2484
MELKCAMKLCAMK4bl1AAphosphoaminophosphonic acid-adenylate esterHuman2514
MELKCAMKLCAMK4bl1ABphosphoaminophosphonic acid-adenylate esterHuman2519
MELKCAMKLCAMK4d2pAA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2513
MELKCAMKLCAMK4d2pAB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2499
MELKCAMKLCAMK4d2pBA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2494
MELKCAMKLCAMK4d2pBB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2498
MELKCAMKLCAMK4d2pCA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2496
MELKCAMKLCAMK4d2pCB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2501
MELKCAMKLCAMK4d2pDA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2486
MELKCAMKLCAMK4d2pDB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2518
MELKCAMKLCAMK4d2tAA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2487
MELKCAMKLCAMK4d2tAB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2489
MELKCAMKLCAMK4d2tBA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2520
MELKCAMKLCAMK4d2tBB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2512
MELKCAMKLCAMK4d2tCA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2491
MELKCAMKLCAMK4d2tCB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2526
MELKCAMKLCAMK4d2tDA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2530
MELKCAMKLCAMK4d2tDB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2511
MELKCAMKLCAMK4d2vAA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2493
MELKCAMKLCAMK4d2vAB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2522
MELKCAMKLCAMK4d2vBA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2483
MELKCAMKLCAMK4d2vBB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2507
MELKCAMKLCAMK4d2vCA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2529
MELKCAMKLCAMK4d2vCB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2492
MELKCAMKLCAMK4d2vDA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2502
MELKCAMKLCAMK4d2vDB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2506
MELKCAMKLCAMK4d2wAA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2515
MELKCAMKLCAMK4d2wAB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2509
MELKCAMKLCAMK4d2wBA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2500
MELKCAMKLCAMK4d2wBB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2482
MELKCAMKLCAMK4d2wCA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2527
MELKCAMKLCAMK4d2wCB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2503
MELKCAMKLCAMK4d2wDA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2481
MELKCAMKLCAMK4d2wDB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2495
MELKCAMKLCAMK4ixpA-Human2528
MELKCAMKLCAMK4umpAA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2497
MELKCAMKLCAMK4umpAB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2485
MELKCAMKLCAMK4umpBA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2524
MELKCAMKLCAMK4umpBB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2504
MELKCAMKLCAMK4umpCA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2479
MELKCAMKLCAMK4umpCB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2508
MELKCAMKLCAMK4umpDA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2516
MELKCAMKLCAMK4umpDB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2525
MELKCAMKLCAMK4umqAA3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminiumHuman2488
MELKCAMKLCAMK4umqAB3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminiumHuman2523
MELKCAMKLCAMK4umrA4-fluoro-n-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamideHuman2521
MELKCAMKLCAMK4umtA1-(4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}-2-methoxybenzyl)piperazinediiumHuman2510
MELKCAMKLCAMK4umuA(2-ethoxy-4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}phenyl)methanaminiumHuman2517
MELKCAMKLCAMK5ih8An-[(pyridin-2-yl)methyl]-4-[4-(pyridin-4-yl)-1h-pyrazol-1-yl]benzamideHuman6661
MELKCAMKLCAMK5ih9AA1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazineHuman6659
MELKCAMKLCAMK5ih9AB1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazineHuman6657
MELKCAMKLCAMK5ihaAA1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazineHuman6663
MELKCAMKLCAMK5ihaAB1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazineHuman6658
MELKCAMKLCAMK5ihcAA4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridineHuman6660
MELKCAMKLCAMK5ihcAB4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridineHuman6662
MELKCAMKLCAMK5k00AA4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamideHuman7497
MELKCAMKLCAMK5k00AB4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamideHuman7498
MELKCAMKLCAMK5m5aAAk-252aHuman8735
MELKCAMKLCAMK5m5aABk-252aHuman8733
MELKCAMKLCAMK5mafAmethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman8732
MELKCAMKLCAMK5magAApf-3758309Human8736
MELKCAMKLCAMK5magABpf-3758309Human8731
MELKCAMKLCAMK5mahAA~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamideHuman8729
MELKCAMKLCAMK5mahAB~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamideHuman8734
MELKCAMKLCAMK5maiAA3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman8728
MELKCAMKLCAMK5maiAB3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman8730
MELKCAMKLCAMK5tvtA9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3-methyl-3,4-dihydropyrimido[5,4-c][1,5]naphthyridin-2(1h)-oneHuman8667
MELKCAMKLCAMK5twlA9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3,4-dihydropyrimido[5,4-c]quinolin-2(1h)-oneHuman8668
MELKCAMKLCAMK5twuA-Human8670
MELKCAMKLCAMK5twuB-Human8672
MELKCAMKLCAMK5twyA2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman8671
MELKCAMKLCAMK5twyB2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman8669
MELKCAMKLCAMK5twzA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman8675
MELKCAMKLCAMK5tx3A7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-oneHuman8673
MELKCAMKLCAMK5tx3B7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-oneHuman8674
MELKCAMKLCAMK6gvxAA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11137
MELKCAMKLCAMK6gvxAB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11139
MELKCAMKLCAMK6gvxBA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11136
MELKCAMKLCAMK6gvxBB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11138
MELKCAMKLCAMK6vxrAA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman12645
MELKCAMKLCAMK6vxrAB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman12644
MERTK (MER)AxlTK2p0cAAphosphoaminophosphonic acid-adenylate esterHuman286
MERTK (MER)AxlTK2p0cABphosphoaminophosphonic acid-adenylate esterHuman287
MERTK (MER)AxlTK2p0cBAphosphoaminophosphonic acid-adenylate esterHuman271
MERTK (MER)AxlTK2p0cBBphosphoaminophosphonic acid-adenylate esterHuman280
MERTK (MER)AxlTK3bprAA2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman278
MERTK (MER)AxlTK3bprAB2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman263
MERTK (MER)AxlTK3bprBA2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman281
MERTK (MER)AxlTK3bprBB2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman275
MERTK (MER)AxlTK3bprCA2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman284
MERTK (MER)AxlTK3bprCB2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman276
MERTK (MER)AxlTK3bprDA2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman279
MERTK (MER)AxlTK3bprDB2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurineHuman282
MERTK (MER)AxlTK3brbAAadenosine-5'-diphosphateHuman266
MERTK (MER)AxlTK3brbABadenosine-5'-diphosphateHuman273
MERTK (MER)AxlTK3brbBAadenosine-5'-diphosphateHuman267
MERTK (MER)AxlTK3brbBBadenosine-5'-diphosphateHuman274
MERTK (MER)AxlTK3tcpA1-[(trans-4-aminocyclohexyl)methyl]-n-butyl-3-(4-fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-6-amineHuman272
MERTK (MER)AxlTK3tcpB1-[(trans-4-aminocyclohexyl)methyl]-n-butyl-3-(4-fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-6-amineHuman285
MERTK (MER)AxlTK4m3qAtrans-4-{[2-(butylamino)-5-(pyridin-2-yl)pyrimidin-4-yl]amino}cyclohexanolHuman283
MERTK (MER)AxlTK4m3qBtrans-4-{[2-(butylamino)-5-(pyridin-2-yl)pyrimidin-4-yl]amino}cyclohexanolHuman269
MERTK (MER)AxlTK4mh7An-butyl-2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-methylpyrimidine-5-carboxamideHuman262
MERTK (MER)AxlTK4mh7B-Human265
MERTK (MER)AxlTK4mhaAA2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-(4-sulfamoylbenzyl)pyrimidine-5-carboxamideHuman264
MERTK (MER)AxlTK4mhaAB2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-(4-sulfamoylbenzyl)pyrimidine-5-carboxamideHuman277
MERTK (MER)AxlTK4mhaBA2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-(4-sulfamoylbenzyl)pyrimidine-5-carboxamideHuman268
MERTK (MER)AxlTK4mhaBB2-(butylamino)-4-[(trans-4-hydroxycyclohexyl)amino]-n-(4-sulfamoylbenzyl)pyrimidine-5-carboxamideHuman270
MERTK (MER)AxlTK5k0kAA15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-oneHuman7345
MERTK (MER)AxlTK5k0kAB15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-oneHuman7347
MERTK (MER)AxlTK5k0kBA15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-oneHuman7348
MERTK (MER)AxlTK5k0kBB15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-oneHuman7346
MERTK (MER)AxlTK5k0xAA(7s)-7-amino-n-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamideHuman7433
MERTK (MER)AxlTK5k0xAB(7s)-7-amino-n-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamideHuman7432
MERTK (MER)AxlTK5k0xBA(7s)-7-amino-n-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamideHuman7434
MERTK (MER)AxlTK5k0xBB(7s)-7-amino-n-[(4-fluorophenyl)methyl]-8-oxo-2,9,16,18,21-pentaazabicyclo[15.3.1]henicosa-1(21),17,19-triene-20-carboxamideHuman7431
MERTK (MER)AxlTK5tc0An-(2-{4-[(2s)-4-(methylsulfonyl)morpholin-2-yl]-1,3-thiazol-2-yl}phenyl)-1h-imidazole-2-carboxamideHuman7383
MERTK (MER)AxlTK5tc0B-Human7381
MERTK (MER)AxlTK5td2AAn-[2-{4-[(2s)-4-(methylsulfonyl)morpholin-2-yl]-1,3-thiazol-2-yl}-4-(morpholin-4-yl)phenyl]-1h-imidazole-2-carboxamideHuman7384
MERTK (MER)AxlTK5td2ABn-[2-{4-[(2s)-4-(methylsulfonyl)morpholin-2-yl]-1,3-thiazol-2-yl}-4-(morpholin-4-yl)phenyl]-1h-imidazole-2-carboxamideHuman7380
MERTK (MER)AxlTK5td2BA-Human7385
MERTK (MER)AxlTK5td2BB-Human7382
MERTK (MER)AxlTK5u6cAA(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8251
MERTK (MER)AxlTK5u6cAB(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8253
MERTK (MER)AxlTK5u6cBA(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8250
MERTK (MER)AxlTK5u6cBB(10r)-7-amino-11-chloro-12-fluoro-1-(2-hydroxyethyl)-3,10,16-trimethyl-16,17-dihydro-1h-8,4-(azeno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecin-15(10h)-oneHuman8252
MERTK (MER)AxlTK6mepAcis-4-[(2-[(4-{[4-(1,3-dioxolan-2-yl)pyridin-2-yl]ethynyl}phenyl)amino]-5-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}pyrimidin-4-yl)amino]cyclohexan-1-olHuman11602
MERTK (MER)AxlTK6mepBcis-4-[(2-[(4-{[4-(1,3-dioxolan-2-yl)pyridin-2-yl]ethynyl}phenyl)amino]-5-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}pyrimidin-4-yl)amino]cyclohexan-1-olHuman11601
MERTK (MER)AxlTK7aaxAA~{n}-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluoranyl-phenyl]-4-ethoxy-1-(4-fluoranyl-2-methyl-phenyl)pyrazole-3-carboxamideHuman12938
MERTK (MER)AxlTK7aaxAB~{n}-[4-(6,7-dimethoxyquinolin-4-yl)oxy-3-fluoranyl-phenyl]-4-ethoxy-1-(4-fluoranyl-2-methyl-phenyl)pyrazole-3-carboxamideHuman12941
MERTK (MER)AxlTK7aayAAn-(3-fluoro-4-{[1-methyl-6-(1h-pyrazol-4-yl)-1h-indazol-5-yl]oxy}phenyl)-1-(4-fluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamideHuman12940
MERTK (MER)AxlTK7aayABn-(3-fluoro-4-{[1-methyl-6-(1h-pyrazol-4-yl)-1h-indazol-5-yl]oxy}phenyl)-1-(4-fluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamideHuman12935
MERTK (MER)AxlTK7aazAA2-azanyl-~{n}-[(1~{s},2~{s})-2-[[4-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]phenyl]methoxy]cyclopentyl]-5-(1-methylpyrazol-4-yl)pyridine-3-carboxamideHuman12962
MERTK (MER)AxlTK7aazAB2-azanyl-~{n}-[(1~{s},2~{s})-2-[[4-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]phenyl]methoxy]cyclopentyl]-5-(1-methylpyrazol-4-yl)pyridine-3-carboxamideHuman12964
MERTK (MER)AxlTK7ab0AA-Human12937
MERTK (MER)AxlTK7ab0AB-Human12939
MERTK (MER)AxlTK7ab1A6-ethyl-3-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-5-(oxan-4-ylamino)pyrazine-2-carboxamideHuman12933
MERTK (MER)AxlTK7ab2AA4-[2-(butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-olHuman12934
MERTK (MER)AxlTK7ab2AB4-[2-(butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-olHuman12936
MERTK (MER)AxlTK7avxA1-(4-fluorophenyl)-n-[3-fluoro-4-[(3-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)oxy]phenyl]-2,3-dimethyl-5-oxopyrazole-4-carboxamideHuman13372
MERTK (MER)AxlTK7avxB1-(4-fluorophenyl)-n-[3-fluoro-4-[(3-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)oxy]phenyl]-2,3-dimethyl-5-oxopyrazole-4-carboxamideHuman13375
MERTK (MER)AxlTK7avyAn-(2-(2-cyclopropylethoxy)pyrimidin-5-yl)-7-methoxy-6-(piperidin-4-ylmethoxy)quinazolin-4-amineHuman13369
MERTK (MER)AxlTK7avzA(r)-n2-(4-(cyclopropylmethoxy)-3,5-difluorophenyl)-5-(3-methylpiperazin-1-yl)-n4-(tetrahydro-2h-pyran-4-yl)pyrimidine-2,4-diamineHuman13370
MERTK (MER)AxlTK7aw0A2-(cyclopentyloxy)-9-(2,6-difluorobenzyl)-n-methyl-9h-purin-6-amineHuman13373
MERTK (MER)AxlTK7aw1An-(6-(4-(3-(4-((5,6-dihydroimidazo[1,2-a]pyrazin-7(8h)-yl)methyl)-3-(trifluoromethyl)phenyl)ureido)phenoxy)pyrimidin-4-yl)cyclopropanecarboxamideHuman13366
MERTK (MER)AxlTK7aw2A5-(2'-chloro-[1,1'-biphenyl]-4-yl)-n-(imidazo[1,2-a]pyridin-6-ylmethyl)-n-methyl-1,3,4-oxadiazol-2-amineHuman13377
MERTK (MER)AxlTK7aw3A2-(1-((5-chloro-1h-pyrrolo[2,3-b]pyridine-3-carboxamido)methyl)-2-azabicyclo[2.1.1]hexan-2-yl)-n-methyl-4-(trifluoromethyl)thiazole-5-carboxamideHuman13367
MERTK (MER)AxlTK7aw4AA3-methyl-5-(4-methyl-1,2,3-thiadiazol-5-yl)-n-((r)-1-(((r)-3-(methylamino)-3-oxo-1-(4-(trifluoromethyl)phenyl)propyl)amino)-1-oxo-4-phenylbutan-2-yl)isoxazole-4-carboxamideHuman13374
MERTK (MER)AxlTK7aw4AB3-methyl-5-(4-methyl-1,2,3-thiadiazol-5-yl)-n-((r)-1-(((r)-3-(methylamino)-3-oxo-1-(4-(trifluoromethyl)phenyl)propyl)amino)-1-oxo-4-phenylbutan-2-yl)isoxazole-4-carboxamideHuman13371
MERTK (MER)AxlTK7aw4BA3-methyl-5-(4-methyl-1,2,3-thiadiazol-5-yl)-n-((r)-1-(((r)-3-(methylamino)-3-oxo-1-(4-(trifluoromethyl)phenyl)propyl)amino)-1-oxo-4-phenylbutan-2-yl)isoxazole-4-carboxamideHuman13376
MERTK (MER)AxlTK7aw4BB3-methyl-5-(4-methyl-1,2,3-thiadiazol-5-yl)-n-((r)-1-(((r)-3-(methylamino)-3-oxo-1-(4-(trifluoromethyl)phenyl)propyl)amino)-1-oxo-4-phenylbutan-2-yl)isoxazole-4-carboxamideHuman13368
MERTK (MER)AxlTK7cqeA5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman12963
MERTK (MER)AxlTK7cqeC5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman12965
MERTK (MER)AxlTK7dxlA3-[4-[6-chloranyl-5-[[(3r)-pyrrolidin-3-yl]amino]-1h-indazol-3-yl]pyrazol-1-yl]benzenecarbonitrileHuman13941
MERTK (MER)AxlTK7m5zAA2-(butylamino)-n-[1-(3-fluoropropyl)piperidin-4-yl]-4-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyrimidine-5-carboxamideHuman13919
MERTK (MER)AxlTK7m5zAB2-(butylamino)-n-[1-(3-fluoropropyl)piperidin-4-yl]-4-{[(1r,4r)-4-hydroxycyclohexyl]amino}pyrimidine-5-carboxamideHuman13920
MERTK (MER)AxlTK7oamA-Human13556
MERTK (MER)AxlTK7olsA5-[4-(1,5-dimethylpyrazol-4-yl)-2-methyl-phenyl]-~{n}-(imidazo[1,2-a]pyridin-6-ylmethyl)-~{n}-methyl-1,3,4-oxadiazol-2-amineHuman13899
MERTK (MER)AxlTK7olvA4-[4-[5-[imidazo[1,2-a]pyridin-6-ylmethyl(methyl)amino]-1,3,4-oxadiazol-2-yl]-3-methyl-phenyl]-2,5-dimethyl-pyrazole-3-carbonitrileHuman13898
MERTK (MER)AxlTK7olxA~{n}-[[3-[4-[(dimethylamino)methyl]phenyl]imidazo[1,2-a]pyridin-6-yl]methyl]-~{n}-methyl-5-[3-methyl-5-(1,3,5-trimethylpyrazol-4-yl)pyridin-2-yl]-1,3,4-oxadiazol-2-amineHuman13897
MERTK (MER)AxlTK7xhyA~{n}-[4-(2-azanyl-3-chloranyl-pyridin-4-yl)oxy-3-fluoranyl-phenyl]-5-(4-fluorophenyl)-4-oxidanylidene-1~{h}-pyridine-3-carboxamideHuman14517
METMetTK1r0pAk-252aHuman2991
METMetTK1r1wA-Human3014
METMetTK2g15A-Human2983
METMetTK2rfnA2-benzyl-5-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-3-methylpyrimidin-4(3h)-oneHuman3022
METMetTK2rfnB2-benzyl-5-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-3-methylpyrimidin-4(3h)-oneHuman2961
METMetTK2rfsAn-(3-chlorophenyl)-n-methyl-2-oxo-3-[(3,4,5-trimethyl-1h-pyrrol-2-yl)methyl]-2h-indole-5-sulfonamideHuman2974
METMetTK2wd1AA1-[(2-nitrophenyl)sulfonyl]-1h-pyrrolo[3,2-b]pyridine-6-carboxamideHuman3032
METMetTK2wd1AB1-[(2-nitrophenyl)sulfonyl]-1h-pyrrolo[3,2-b]pyridine-6-carboxamideHuman2976
METMetTK2wgjA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman3009
METMetTK2wkmA(3z)-5-[(2,6-dichlorobenzyl)sulfonyl]-3-[(3,5-dimethyl-4-{[(2s)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]carbonyl}-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman3021
METMetTK3a4pA(2e)-3-{6-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]quinolin-3-yl}-n-methylprop-2-enamideHuman3005
METMetTK3c1xAn-{[4-({5-[(4-aminopiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}oxy)-3-fluorophenyl]carbamoyl}-2-(4-fluorophenyl)acetamideHuman3020
METMetTK3ccnA4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methyl]phenolHuman2971
METMetTK3cd8AA7-methoxy-4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy]quinolineHuman3008
METMetTK3cd8AB7-methoxy-4-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methoxy]quinolineHuman2995
METMetTK3ce3A1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamideHuman6769
METMetTK3cthAn-({4-[(2-aminopyridin-4-yl)oxy]-3-fluorophenyl}carbamoyl)-2-(4-fluorophenyl)acetamideHuman6768
METMetTK3ctjAA2-(4-fluorophenyl)-n-{[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]carbamoyl}acetamideHuman6767
METMetTK3ctjAB2-(4-fluorophenyl)-n-{[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]carbamoyl}acetamideHuman6766
METMetTK3dkcAAadenosine-5'-triphosphateHuman2997
METMetTK3dkcABadenosine-5'-triphosphateHuman2952
METMetTK3dkfAA6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinolineHuman3030
METMetTK3dkfAB6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinolineHuman3029
METMetTK3dkfAC6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinolineHuman2984
METMetTK3dkgAA6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinolineHuman2993
METMetTK3dkgAB6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinolineHuman3019
METMetTK3dkgAC6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinolineHuman3006
METMetTK3efjA2-benzyl-5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-3-methylpyrimidin-4(3h)-oneHuman3015
METMetTK3efjB2-benzyl-5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-3-methylpyrimidin-4(3h)-oneHuman2957
METMetTK3efkA5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-2-[(4-fluorophenyl)amino]-3-methylpyrimidin-4(3h)-oneHuman3018
METMetTK3efkB5-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-2-[(4-fluorophenyl)amino]-3-methylpyrimidin-4(3h)-oneHuman2988
METMetTK3f66AA3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenolHuman2989
METMetTK3f66AB3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenolHuman3027
METMetTK3f66AC3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenolHuman3011
METMetTK3f66AD3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenolHuman3026
METMetTK3f66BA3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenolHuman3034
METMetTK3f66BB3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenolHuman2992
METMetTK3f66BC3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenolHuman2966
METMetTK3f66BD3-[3-(4-methylpiperazin-1-yl)-7-(trifluoromethyl)quinoxalin-5-yl]phenolHuman3000
METMetTK3f82An-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorophenyl}-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamideHuman2977
METMetTK3i5nA7-methoxy-n-[(6-phenyl[1,2,4]triazolo[4,3-b]pyridazin-3-yl)methyl]-1,5-naphthyridin-4-amineHuman3013
METMetTK3l8vA2-({4-[(2-aminopyridin-4-yl)oxy]-3-fluorophenyl}amino)-n-(2,4-difluorophenyl)pyridine-3-carboxamideHuman2978
METMetTK3lq8AAn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman2998
METMetTK3lq8ABn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman2964
METMetTK3q6uAA-Human2954
METMetTK3q6uAB-Human2962
METMetTK3q6wA3-{5-oxo-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-5h-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl}-n-(pyridin-2-ylmethyl)propanamideHuman2969
METMetTK3qtiAA6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinolineHuman2994
METMetTK3qtiAB6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinolineHuman3028
METMetTK3qtiBA6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinolineHuman3017
METMetTK3qtiBB6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinolineHuman3024
METMetTK3r7oAn-[(2r)-1,4-dioxan-2-ylmethyl]-n-methyl-n'-{5-oxo-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-5h-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl}sulfuric diamideHuman3038
METMetTK3rhkA1-[(3r,4r)-4-(1h-indol-3-yl)-2,5-dioxopyrrolidin-3-yl]pyrrolo[3,2,1-ij]quinoliniumHuman2979
METMetTK3rhkB1-[(3r,4r)-4-(1h-indol-3-yl)-2,5-dioxopyrrolidin-3-yl]pyrrolo[3,2,1-ij]quinoliniumHuman2959
METMetTK3u6hAAn-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamideHuman2996
METMetTK3u6hABn-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]-3-fluorophenyl}-1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamideHuman2965
METMetTK3u6iAn-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-1-[(2r)-2-hydroxypropyl]-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamideHuman2967
METMetTK3vw8An-({4-[(6,7-dimethoxyquinolin-4-yl)oxy]phenyl}carbamothioyl)-2-phenylacetamideHuman2985
METMetTK3zbxA6-[[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinolineHuman3036
METMetTK3zc5A6-{(1s)-1-[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]ethyl}quinolineHuman3003
METMetTK3zclA(s)-3-(1-(1h-pyrrolo(2,3-b)pyridin-3-yl)ethyl)-n-isopropyl-(1,2,4)triazolo(4,3-b)pyridazin-6-amineHuman2990
METMetTK3zxzA2-{4-[1-(quinolin-6-ylmethyl)-1h-[1,2,3]triazolo[4,5-b]pyrazin-6-yl]-1h-pyrazol-1-yl}ethanolHuman2999
METMetTK3zzeA(2s)-n'-[(3r)-4-chloro-7-methyl-2-oxo-2,3-dihydro-1h-indol-3-yl]-2-(4-hydroxyphenyl)propanehydrazideHuman2980
METMetTK4aoiA4-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylmethyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-6-yl]benzenecarbonitrileHuman2958
METMetTK4ap7A4-[[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]phenolHuman3035
METMetTK4degA7-methoxy-n-{[6-(3-methyl-1,2-thiazol-5-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]methyl}-1,5-naphthyridin-4-amineHuman2981
METMetTK4dehA5-phenyl-3-(quinolin-6-ylmethyl)-3,5,6,7-tetrahydro-4h-[1,2,3]triazolo[4,5-c]pyridin-4-oneHuman2963
METMetTK4deiA3-{(1s)-1-[3-(2-methoxyethoxy)quinolin-6-yl]ethyl}-5-(3-methyl-1,2-thiazol-5-yl)-3,5-dihydro-4h-[1,2,3]triazolo[4,5-c]pyridin-4-oneHuman3016
METMetTK4eevAAn-(3-fluoro-4-{[1-methyl-6-(1h-pyrazol-4-yl)-1h-indazol-5-yl]oxy}phenyl)-1-(4-fluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamideHuman3012
METMetTK4eevABn-(3-fluoro-4-{[1-methyl-6-(1h-pyrazol-4-yl)-1h-indazol-5-yl]oxy}phenyl)-1-(4-fluorophenyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamideHuman3023
METMetTK4gg5AA3-(4-methylpiperazin-1-yl)-n-(3-nitrobenzyl)-7-(trifluoromethyl)quinolin-5-amineHuman2956
METMetTK4gg5AB3-(4-methylpiperazin-1-yl)-n-(3-nitrobenzyl)-7-(trifluoromethyl)quinolin-5-amineHuman2953
METMetTK4gg7AAn-(3-nitrobenzyl)-6-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amineHuman3002
METMetTK4gg7ABn-(3-nitrobenzyl)-6-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-2-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amineHuman2987
METMetTK4iwdA1-{5-oxo-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-5h-benzo[4,5]cyclohepta[1,2-b]pyridin-7-yl}-n-(pyridin-2-ylmethyl)methanesulfonamideHuman2975
METMetTK4knbAA7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amineHuman2960
METMetTK4knbAB7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amineHuman3037
METMetTK4knbBA7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amineHuman3007
METMetTK4knbBB7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amineHuman2970
METMetTK4knbCA7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amineHuman2955
METMetTK4knbCB7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amineHuman3001
METMetTK4knbDA7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amineHuman3010
METMetTK4knbDB7-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-3-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[3,2-c]pyridin-6-amineHuman2968
METMetTK4mxcAAn-(3-fluoro-4-{[2-({3-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman3033
METMetTK4mxcABn-(3-fluoro-4-{[2-({3-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman3025
METMetTK4r1vAA3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrileHuman3004
METMetTK4r1vAB3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrileHuman2972
METMetTK4r1yA3-(diethylamino)propyl (3-{[5-(3,4-dimethoxyphenyl)-2-oxo-2h-1,3,4-thiadiazin-3(6h)-yl]methyl}phenyl)carbamateHuman2973
METMetTK4xmoA6-{(1r)-1-fluoro-1-[8-fluoro-6-(3-methyl-1,2-oxazol-5-yl)[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl}-3-methoxyquinolineHuman3031
METMetTK4xyfAA6-{(1s)-1-[8-fluoro-6-(3-methyl-1,2-oxazol-5-yl)[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl}-3-(2-methoxyethoxy)quinolineHuman2986
METMetTK4xyfAB6-{(1s)-1-[8-fluoro-6-(3-methyl-1,2-oxazol-5-yl)[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl}-3-(2-methoxyethoxy)quinolineHuman2982
METMetTK5dg5AAn-(2,5-difluoro-4-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman7037
METMetTK5dg5ABn-(2,5-difluoro-4-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman7034
METMetTK5dg5BAn-(2,5-difluoro-4-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman7035
METMetTK5dg5BBn-(2,5-difluoro-4-{[2-(1-methyl-1h-pyrazol-4-yl)pyridin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman7036
METMetTK5eobAA6-[bis(fluoranyl)-[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinolineHuman7100
METMetTK5eobAB6-[bis(fluoranyl)-[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinolineHuman7101
METMetTK5eycAA6-[(1~{r})-1-[8-fluoranyl-6-(3-methyl-1,2-oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl]-1,6-naphthyridin-5-oneHuman6401
METMetTK5eycAB6-[(1~{r})-1-[8-fluoranyl-6-(3-methyl-1,2-oxazol-5-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl]-1,6-naphthyridin-5-oneHuman6400
METMetTK5eydAA6-[(1~{r})-1-[8-fluoranyl-6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl]-3-(2-methoxyethoxy)-1,6-naphthyridin-5-oneHuman6402
METMetTK5eydAB6-[(1~{r})-1-[8-fluoranyl-6-(1-methylpyrazol-4-yl)-[1,2,4]triazolo[4,3-a]pyridin-3-yl]ethyl]-3-(2-methoxyethoxy)-1,6-naphthyridin-5-oneHuman6399
METMetTK5hlwA1-[2-(1-ethylpiperidin-4-yl)ethyl]-3-(6-{[6-(thiophen-2-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1,3-benzothiazol-2-yl)ureaHuman7275
METMetTK5hniXmethyl (6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1h-benzimidazol-2-yl)carbamateHuman7280
METMetTK5hniYmethyl (6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1h-benzimidazol-2-yl)carbamateHuman7278
METMetTK5ho6A1-(6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1,3-benzothiazol-2-yl)-3-[2-(morpholin-4-yl)ethyl]ureaHuman7277
METMetTK5hoaA1-(6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1,3-benzothiazol-2-yl)-3-[2-(morpholin-4-yl)ethyl]ureaHuman7279
METMetTK5horA1-(6-{[6-(4-fluorophenyl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}-1,3-benzothiazol-2-yl)-3-[2-(morpholin-4-yl)ethyl]ureaHuman7276
METMetTK5htiAAn-[3-fluoro-4-({7-[2-(morpholin-4-yl)ethoxy]-1,6-naphthyridin-4-yl}oxy)phenyl]-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman8010
METMetTK5htiABn-[3-fluoro-4-({7-[2-(morpholin-4-yl)ethoxy]-1,6-naphthyridin-4-yl}oxy)phenyl]-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman8009
METMetTK5t3qAn-{3-fluoro-4-[(7-methoxyquinolin-4-yl)oxy]phenyl}-1-(2-hydroxy-2-methylpropyl)-5-methyl-3-oxo-2-phenyl-2,3-dihydro-1h-pyrazole-4-carboxamideHuman7413
METMetTK5uabAAn-{6-[([1,2,4]triazolo[4,3-a]pyridin-3-yl)sulfanyl]imidazo[1,2-b]pyridazin-2-yl}cyclopropanecarboxamideHuman7961
METMetTK5uabABn-{6-[([1,2,4]triazolo[4,3-a]pyridin-3-yl)sulfanyl]imidazo[1,2-b]pyridazin-2-yl}cyclopropanecarboxamideHuman7964
METMetTK5uadAn-(6-{[6-(1-methyl-1h-pyrazol-4-yl)-1h-benzotriazol-1-yl]methyl}imidazo[1,2-b]pyridazin-2-yl)cyclopropanecarboxamideHuman7963
METMetTK5ya5AA2-[3-(4-methoxybenzyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1h-indoleHuman10040
METMetTK5ya5AB2-[3-(4-methoxybenzyl)[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1h-indoleHuman10039
METMetTK6sd9An-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman11531
METMetTK6sdcAAn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman11532
METMetTK6sdcABn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman11534
METMetTK6sddAn-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorophenyl}-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamideHuman11533
METMetTK6sdeAvolitinibHuman11535
METMetTK6ubwAn-(6-{difluoro[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-a]pyridin-3-yl]methyl}imidazo[1,2-b]pyridazin-2-yl)cyclopropanecarboxamideHuman11979
METMetTK7b3qAA1-(phenylmethyl)-5~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman13177
METMetTK7b3qAB1-(phenylmethyl)-5~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman13182
METMetTK7b3tAA3-(phenylmethyl)-1~{h}-pyrrolo[2,3-b]pyridineHuman13183
METMetTK7b3tAB3-(phenylmethyl)-1~{h}-pyrrolo[2,3-b]pyridineHuman13191
METMetTK7b3vAA3-(3-methyl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)-1~{h}-pyrrolo[3,4-b]pyrrol-6-oneHuman13188
METMetTK7b3vAB3-(3-methyl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)-1~{h}-pyrrolo[3,4-b]pyrrol-6-oneHuman13194
METMetTK7b3wAA3-(6-fluoranyl-1~{h}-indazol-4-yl)-4,5-dihydro-1~{h}-pyrrolo[3,4-b]pyrrol-6-oneHuman13180
METMetTK7b3wAB3-(6-fluoranyl-1~{h}-indazol-4-yl)-4,5-dihydro-1~{h}-pyrrolo[3,4-b]pyrrol-6-oneHuman13178
METMetTK7b3zAA3-[3-(phenylmethyl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-4,5-dihydro-1~{h}-pyrrolo[3,4-b]pyrrol-6-oneHuman13181
METMetTK7b3zAB3-[3-(phenylmethyl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-4,5-dihydro-1~{h}-pyrrolo[3,4-b]pyrrol-6-oneHuman13186
METMetTK7b40A3-(phenylmethyl)-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridineHuman13192
METMetTK7b41AA3-[(2-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridineHuman13184
METMetTK7b41AB3-[(2-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridineHuman13193
METMetTK7b42A3-[(3-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridineHuman13190
METMetTK7b43A3-[(4-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridineHuman13189
METMetTK7b43B3-[(4-fluorophenyl)methyl]-5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridineHuman13187
METMetTK7b44AA5-methoxy-1~{h}-indazoleHuman13185
METMetTK7b44AB5-methoxy-1~{h}-indazoleHuman13179
METMetTK7v3rAA~{n}1'-[3-fluoranyl-4-(2-phenylazanylpyrimidin-4-yl)oxy-phenyl]-~{n}1-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman14328
METMetTK7v3rAB~{n}1'-[3-fluoranyl-4-(2-phenylazanylpyrimidin-4-yl)oxy-phenyl]-~{n}1-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman14330
METMetTK7v3sAA~{n}1'-[3-fluoranyl-4-(10~{h}-pyrido[3,2-b][1,4]benzoxazin-4-yloxy)phenyl]-~{n}1-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman14329
METMetTK7v3sAB~{n}1'-[3-fluoranyl-4-(10~{h}-pyrido[3,2-b][1,4]benzoxazin-4-yloxy)phenyl]-~{n}1-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman14327
METMetTK7y4tA2-[2-[3-(1-methylpyrazol-4-yl)quinolin-6-yl]ethyl]-6-(3-nitrophenyl)pyridazin-3-oneHuman14548
METMetTK7y4uA~{n}-methyl-4-[1-[2-[3-(1-methylpyrazol-4-yl)quinolin-6-yl]ethyl]-6-oxidanylidene-pyridazin-3-yl]-2-(trifluoromethyl)benzamideHuman14550
METMetTK8an8A3-[bis(fluoranyl)methyl]-~{n}-methyl-~{n}-[(1~{r})-8-methyl-5-(3-methyl-1~{h}-indazol-6-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]pyridine-2-carboxamideHuman14355
METMetTK8ansA3-[bis(fluoranyl)methyl]-~{n}-methyl-~{n}-[(1~{r})-8-methyl-5-(3-methyl-1~{h}-indazol-6-yl)-1,2,3,4-tetrahydronaphthalen-1-yl]pyridine-2-carboxamideHuman14356
METMetTK8au3A3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrileHuman14982
METMetTK8au5A3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrileHuman14983
METMetTK8aw1AA3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrileHuman14981
METMetTK8aw1AB3-[1-(3-{5-[(1-methylpiperidin-4-yl)methoxy]pyrimidin-2-yl}benzyl)-6-oxo-1,6-dihydropyridazin-3-yl]benzonitrileHuman14980
METMetTK8gvjA(1^4z,5^2e)-6^3-(trifluoromethyl)-5^1,5^6-dihydro-1^1h-8-aza-2(3,6)-quinolina-5(1,3)-pyridazina-1(4,1)-pyrazola-6(1,4)-benzenacyclododecaphane-5^6,7-dioneHuman14549
METMetTK8ouuAA5-(3-ethynyl-5-fluoranyl-1h-indazol-7-yl)-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dioneHuman14821
METMetTK8ouuAB5-(3-ethynyl-5-fluoranyl-1h-indazol-7-yl)-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dioneHuman14824
METMetTK8ouvAA5-(1h-indazol-7-yl)-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dioneHuman14820
METMetTK8ouvAB5-(1h-indazol-7-yl)-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dioneHuman14823
METMetTK8ov7A5-[3,5-bis(fluoranyl)phenyl]-1-[(1s)-1-[3-(1h-imidazol-5-yl)phenyl]ethyl]pyrimidine-2,4-dioneHuman14817
METMetTK8ovzA1-[(1s)-1-[3-(1h-imidazol-4-yl)phenyl]ethyl]-5-(1h-indazol-7-yl)pyrimidine-2,4-dioneHuman14822
METMetTK8ow3A5-[3,5-bis(fluoranyl)phenyl]-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dioneHuman14818
METMetTK8owgA5-[3,5-bis(fluoranyl)phenyl]-1-[(1s)-1-phenylethyl]pyrimidine-2,4-dioneHuman14819
MKNK1 (MNK1)MAPKAPKCAMK2hw6A-Human2084
MKNK1 (MNK1)MAPKAPKCAMK2hw6B-Human2085
MKNK1 (MNK1)MAPKAPKCAMK5wvdA1-methyl-n-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamideHuman9464
MKNK1 (MNK1)MAPKAPKCAMK5wvdB1-methyl-n-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamideHuman9465
MKNK2 (MNK2)MAPKAPKCAMK2ac3A-Human765
MKNK2 (MNK2)MAPKAPKCAMK2ac5AA-Human763
MKNK2 (MNK2)MAPKAPKCAMK2ac5AB-Human766
MKNK2 (MNK2)MAPKAPKCAMK2hw7AstaurosporineHuman764
MKNK2 (MNK2)MAPKAPKCAMK6cj5A3-(pyridin-3-yl)imidazo[1,2-a]pyridine-8-carboxamideHuman9886
MKNK2 (MNK2)MAPKAPKCAMK6cjeA4-[(9h-purin-6-yl)amino]benzamideHuman9884
MKNK2 (MNK2)MAPKAPKCAMK6cjhA3-phenyl-5-(pyridin-4-yl)-1h-indazoleHuman9885
MKNK2 (MNK2)MAPKAPKCAMK6cjwA3-(pyridin-4-yl)imidazo[1,2-b]pyridazineHuman9879
MKNK2 (MNK2)MAPKAPKCAMK6cjyA5-[(7h-purin-6-yl)amino]-1h-isoindol-1-oneHuman9881
MKNK2 (MNK2)MAPKAPKCAMK6ck3A(3r)-3-methyl-5-[(pyrimidin-4-yl)amino]-2,3-dihydro-1h-isoindol-1-oneHuman9883
MKNK2 (MNK2)MAPKAPKCAMK6ck6A6'-[(6-aminopyrimidin-4-yl)amino]-8'-methyl-2'h-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dioneHuman9880
MKNK2 (MNK2)MAPKAPKCAMK6ckiA3,3-dimethyl-6-[(pyrimidin-4-yl)amino]-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dioneHuman9882
MKNK2 (MNK2)MAPKAPKCAMK6jlrA4-[5-(1-methylpyrazol-4-yl)pyridin-3-yl]benzamideHuman11968
Mlkl (MLKL)TKL-UniqueTKL4btfA-Mouse5816
Mlkl (MLKL)TKL-UniqueTKL4m68AA-Mouse5820
Mlkl (MLKL)TKL-UniqueTKL4m68AB-Mouse5819
Mlkl (MLKL)TKL-UniqueTKL4m69BA-Mouse5818
Mlkl (MLKL)TKL-UniqueTKL4m69BB-Mouse5817
MLKLTKL-UniqueTKL4m67A-Human3048
MLKLTKL-UniqueTKL4mwiAA-Human3047
MLKLTKL-UniqueTKL4mwiAB-Human3049
MLKLTKL-UniqueTKL5knjA1-[4-[methyl-[2-[(3-sulfamoylphenyl)amino]pyrimidin-4-yl]amino]phenyl]-3-[4-(trifluoromethyloxy)phenyl]ureaHuman7270
MLKLTKL-UniqueTKL5knjB1-[4-[methyl-[2-[(3-sulfamoylphenyl)amino]pyrimidin-4-yl]amino]phenyl]-3-[4-(trifluoromethyloxy)phenyl]ureaHuman7268
MLKLTKL-UniqueTKL5ko1AA[(1~{r})-2-[(4-fluorophenyl)amino]-2-oxidanylidene-1-phenyl-ethyl] 3-azanylpyrazine-2-carboxylateHuman7269
MLKLTKL-UniqueTKL5ko1AB[(1~{r})-2-[(4-fluorophenyl)amino]-2-oxidanylidene-1-phenyl-ethyl] 3-azanylpyrazine-2-carboxylateHuman7271
MLKLTKL-UniqueTKL6bwkA-Human10038
MLKLTKL-UniqueTKL6lk5A-Human13094
MLKLTKL-UniqueTKL6lk6A-Human13095
MLKLTKL-UniqueTKL6o5zA-Human12782
MLKLTKL-UniqueTKL6o5zB1-[2-fluoranyl-5-(trifluoromethyl)phenyl]-3-[4-[methyl-[2-[(3-sulfamoylphenyl)amino]pyrimidin-4-yl]amino]phenyl]ureaHuman12783
MLKLTKL-UniqueTKL7jw7A-Human13395
MLKLTKL-UniqueTKL7jxuA-Human13394
MLKLTKL-UniqueTKL7jxuB-Human13396
MLKLTKL-UniqueTKL7monAn-[4-({2-[(cyclopropanecarbonyl)amino]pyridin-4-yl}oxy)-3-fluorophenyl]-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamideHuman13980
MLKLTKL-UniqueTKL8slzA-Human14988
MST1R (RON)MetTK3plsAAphosphoaminophosphonic acid-adenylate esterHuman1492
MST1R (RON)MetTK3plsABphosphoaminophosphonic acid-adenylate esterHuman1491
MTOR (FRAP)PIKKAtypical3jbzAadenosine-5'-diphosphateHuman9113
MTOR (FRAP)PIKKAtypical4jsnA-Human9114
MTOR (FRAP)PIKKAtypical4jsnB-Human9115
MTOR (FRAP)PIKKAtypical4jspAphosphothiophosphoric acid-adenylate esterHuman9106
MTOR (FRAP)PIKKAtypical4jspBphosphothiophosphoric acid-adenylate esterHuman9107
MTOR (FRAP)PIKKAtypical4jsvAadenosine-5'-diphosphateHuman9109
MTOR (FRAP)PIKKAtypical4jsvBadenosine-5'-diphosphateHuman9100
MTOR (FRAP)PIKKAtypical4jsxA9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-oneHuman9112
MTOR (FRAP)PIKKAtypical4jsxB9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-oneHuman9111
MTOR (FRAP)PIKKAtypical4jt5A2-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-1h-indol-5-olHuman9116
MTOR (FRAP)PIKKAtypical4jt5B2-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-1h-indol-5-olHuman9104
MTOR (FRAP)PIKKAtypical4jt6A3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenolHuman9103
MTOR (FRAP)PIKKAtypical4jt6B3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenolHuman9102
MTOR (FRAP)PIKKAtypical5flcBA-Human9105
MTOR (FRAP)PIKKAtypical5flcBB-Human9108
MTOR (FRAP)PIKKAtypical5flcFA-Human9101
MTOR (FRAP)PIKKAtypical5flcFB-Human9117
MTOR (FRAP)PIKKAtypical5h64a-Human9110
MTOR (FRAP)PIKKAtypical5h64A-Human9099
MTOR (FRAP)PIKKAtypical5wbuA-Human9407
MTOR (FRAP)PIKKAtypical5wbuB-Human9405
MTOR (FRAP)PIKKAtypical5wbyA-Human9404
MTOR (FRAP)PIKKAtypical5wbyB-Human9406
MTOR (FRAP)PIKKAtypical5zcsA-Human9748
MTOR (FRAP)PIKKAtypical5zcsB-Human9749
MTOR (FRAP)PIKKAtypical6sb0A-Human11727
MTOR (FRAP)PIKKAtypical6sb0B-Human11725
MTOR (FRAP)PIKKAtypical6sb2A-Human11724
MTOR (FRAP)PIKKAtypical6sb2B-Human11726
MTOR (FRAP)PIKKAtypical6zwmAphosphothiophosphoric acid-adenylate esterHuman12989
MTOR (FRAP)PIKKAtypical6zwmBphosphothiophosphoric acid-adenylate esterHuman12988
MTOR (FRAP)PIKKAtypical6zwoBphosphothiophosphoric acid-adenylate esterHuman12987
MTOR (FRAP)PIKKAtypical7pe7A-Human13901
MTOR (FRAP)PIKKAtypical7pe8A-Human13870
MTOR (FRAP)PIKKAtypical7pe9A-Human13871
MTOR (FRAP)PIKKAtypical7peaA-Human13873
MTOR (FRAP)PIKKAtypical7pebA-Human13869
MTOR (FRAP)PIKKAtypical7pecA-Human13872
MTOR (FRAP)PIKKAtypical7tzoA-Human14575
MTOR (FRAP)PIKKAtypical7uxcA-Human14525
MTOR (FRAP)PIKKAtypical8eraA1-[6-{[(3m)-4-amino-3-(2-amino-1,3-benzoxazol-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-3,4-dihydroisoquinolin-2(1h)-yl]-3-hydroxypropan-1-oneHuman14569
MYLK4 (SgK085)MLCKCAMK2x4fAA4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amineHuman4865
MYLK4 (SgK085)MLCKCAMK2x4fAB4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amineHuman4867
MYLK4 (SgK085)MLCKCAMK2x4fBA4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amineHuman4866
MYLK4 (SgK085)MLCKCAMK2x4fBB4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amineHuman4868
NEK1NEKOther4apcAA-Human1215
NEK1NEKOther4apcAB-Human1208
NEK1NEKOther4apcBA-Human1212
NEK1NEKOther4apcBB-Human1210
NEK1NEKOther4b9dAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman1211
NEK1NEKOther4b9dAB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman1213
NEK1NEKOther4b9dBA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman1214
NEK1NEKOther4b9dBB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman1209
NEK2NEKOther2javAA5-[(z)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman332
NEK2NEKOther2javAB5-[(z)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman323
NEK2NEKOther2w5aAAadenosine-5'-diphosphateHuman302
NEK2NEKOther2w5aABadenosine-5'-diphosphateHuman317
NEK2NEKOther2w5bAAphosphothiophosphoric acid-adenylate esterHuman320
NEK2NEKOther2w5bABphosphothiophosphoric acid-adenylate esterHuman305
NEK2NEKOther2w5hAA-Human327
NEK2NEKOther2w5hAB-Human310
NEK2NEKOther2wqoA4-[2-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]benzoic acidHuman331
NEK2NEKOther2xk3AA4-[3-amino-6-(3-ethylthiophen-2-yl)pyrazin-2-yl]cyclohexane-1-carboxylic acidHuman309
NEK2NEKOther2xk3AB4-[3-amino-6-(3-ethylthiophen-2-yl)pyrazin-2-yl]cyclohexane-1-carboxylic acidHuman329
NEK2NEKOther2xk4AA4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acidHuman314
NEK2NEKOther2xk4AB4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acidHuman316
NEK2NEKOther2xk4AC4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acidHuman304
NEK2NEKOther2xk6Acis-4-[3-amino-6-(3-cyclopropylthiophen-2-yl)pyrazin-2-yl]cyclohexanecarboxylic acidHuman301
NEK2NEKOther2xk7AA(3r,4r)-1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-3-ethylpiperidine-4-carboxylic acidHuman326
NEK2NEKOther2xk7AB(3r,4r)-1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-3-ethylpiperidine-4-carboxylic acidHuman318
NEK2NEKOther2xk8A4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methoxybenzoic acidHuman300
NEK2NEKOther2xkcAA4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methylbenzoic acidHuman321
NEK2NEKOther2xkcAB4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methylbenzoic acidHuman307
NEK2NEKOther2xkdAA4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]benzoic acidHuman330
NEK2NEKOther2xkdAB4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]benzoic acidHuman298
NEK2NEKOther2xkeA1-[3-amino-6-(3-methoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acidHuman299
NEK2NEKOther2xkfAA1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acidHuman315
NEK2NEKOther2xkfAB1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acidHuman311
NEK2NEKOther2xnmAA5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamideHuman306
NEK2NEKOther2xnmAB5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamideHuman324
NEK2NEKOther2xnnAA5-(1h-benzimidazol-1-yl)-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamideHuman303
NEK2NEKOther2xnnAB5-(1h-benzimidazol-1-yl)-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamideHuman308
NEK2NEKOther2xnoAA5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{[2-(trifluoromethyl)benzyl]oxy}thiophene-2-carboxamideHuman319
NEK2NEKOther2xnoAB5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{[2-(trifluoromethyl)benzyl]oxy}thiophene-2-carboxamideHuman313
NEK2NEKOther2xnpAA4-{5-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamideHuman328
NEK2NEKOther2xnpAB4-{5-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamideHuman322
NEK2NEKOther4a4xA4-(2-amino-5-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridin-3-yl)-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamideHuman325
NEK2NEKOther4afeA4-(2-amino-5-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridin-3-yl)-2-{[(1r,2z)-4,4,4-trifluoro-1-methylbut-2-en-1-yl]oxy}benzamideHuman312
NEK2NEKOther5m51A3-[[6-(cyclohexylmethoxy)-9~{h}-purin-2-yl]amino]benzamideHuman7157
NEK2NEKOther5m53AA3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n},~{n}-dimethyl-benzamideHuman7159
NEK2NEKOther5m53AB3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n},~{n}-dimethyl-benzamideHuman7161
NEK2NEKOther5m55AA6-[(~{z})-2-(diethylamino)ethenyl]-~{n}-phenyl-7~{h}-purin-2-amineHuman7140
NEK2NEKOther5m55AB6-[(~{z})-2-(diethylamino)ethenyl]-~{n}-phenyl-7~{h}-purin-2-amineHuman7139
NEK2NEKOther5m57Ao6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7272
NEK2NEKOther6sgdAA4-[(6-ethenyl-7~{h}-purin-2-yl)amino]benzenesulfonamideHuman12373
NEK2NEKOther6sgdAB4-[(6-ethenyl-7~{h}-purin-2-yl)amino]benzenesulfonamideHuman12375
NEK2NEKOther6sghAA2-[4-[(6-ethenyl-9~{h}-purin-2-yl)amino]phenyl]ethanamideHuman12374
NEK2NEKOther6sghAB2-[4-[(6-ethenyl-9~{h}-purin-2-yl)amino]phenyl]ethanamideHuman12372
NEK2NEKOther6sgiAA4-[(6-ethyl-7~{h}-purin-2-yl)amino]benzenesulfonamideHuman12378
NEK2NEKOther6sgiAB4-[(6-ethyl-7~{h}-purin-2-yl)amino]benzenesulfonamideHuman12380
NEK2NEKOther6sgkA2-phenylazanyl-9~{h}-purine-6-carbonitrileHuman12377
NEK2NEKOther6sk9AA3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12376
NEK2NEKOther6sk9AB3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12379
NEK7NEKOther2wqmAA-Human3854
NEK7NEKOther2wqmAB-Human3857
NEK7NEKOther2wqnAAadenosine-5'-diphosphateHuman3855
NEK7NEKOther2wqnABadenosine-5'-diphosphateHuman3856
NEK7NEKOther5de2AA-Human6246
NEK7NEKOther5de2AB-Human6244
NEK7NEKOther5de2BA-Human6245
NEK7NEKOther5de2BB-Human6247
NEK7NEKOther6npyBA-Human11338
NEK7NEKOther6npyBB-Human11337
NEK7NEKOther6s73A3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12357
NEK7NEKOther6s73B3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12353
NEK7NEKOther6s73C3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12362
NEK7NEKOther6s73D-Human12355
NEK7NEKOther6s75A3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12356
NEK7NEKOther6s75B3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12358
NEK7NEKOther6s75C3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12360
NEK7NEKOther6s75D-Human12359
NEK7NEKOther6s76A-Human12351
NEK7NEKOther6s76B-Human12354
NEK7NEKOther6s76C-Human12352
NEK7NEKOther6s76D-Human12361
NTRK1 (TRKA)TrkTK4aojAA5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamineHuman3602
NTRK1 (TRKA)TrkTK4aojAB5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamineHuman3610
NTRK1 (TRKA)TrkTK4aojBA5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamineHuman3607
NTRK1 (TRKA)TrkTK4aojBB5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamineHuman3604
NTRK1 (TRKA)TrkTK4aojCA5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamineHuman3617
NTRK1 (TRKA)TrkTK4aojCB5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamineHuman3621
NTRK1 (TRKA)TrkTK4f0iA-Human3603
NTRK1 (TRKA)TrkTK4f0iB-Human3605
NTRK1 (TRKA)TrkTK4gt5AA-Human3616
NTRK1 (TRKA)TrkTK4gt5AB-Human3609
NTRK1 (TRKA)TrkTK4pmmAAn-(3-cyclopropyl-1-phenyl-1h-pyrazol-5-yl)-2-{4-[3-methoxy-4-(4-methyl-1h-imidazol-1-yl)phenyl]-1h-1,2,3-triazol-1-yl}acetamideHuman3618
NTRK1 (TRKA)TrkTK4pmmABn-(3-cyclopropyl-1-phenyl-1h-pyrazol-5-yl)-2-{4-[3-methoxy-4-(4-methyl-1h-imidazol-1-yl)phenyl]-1h-1,2,3-triazol-1-yl}acetamideHuman3619
NTRK1 (TRKA)TrkTK4pmpAA1-cyclopropyl-1-[3-(1,3-thiazol-2-yl)benzyl]-3-[4-(trifluoromethoxy)phenyl]ureaHuman3613
NTRK1 (TRKA)TrkTK4pmpAB1-cyclopropyl-1-[3-(1,3-thiazol-2-yl)benzyl]-3-[4-(trifluoromethoxy)phenyl]ureaHuman3608
NTRK1 (TRKA)TrkTK4pmsAA4-(naphthalen-1-yl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1h-pyrrolo[3,2-c]pyridine-2-carboxylic acidHuman3606
NTRK1 (TRKA)TrkTK4pmsAB4-(naphthalen-1-yl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1h-pyrrolo[3,2-c]pyridine-2-carboxylic acidHuman3601
NTRK1 (TRKA)TrkTK4pmtAAn~4~-[4-(morpholin-4-yl)phenyl]-n~6~-(pyridin-3-ylmethyl)pyrido[3,2-d]pyrimidine-4,6-diamineHuman3614
NTRK1 (TRKA)TrkTK4pmtABn~4~-[4-(morpholin-4-yl)phenyl]-n~6~-(pyridin-3-ylmethyl)pyrido[3,2-d]pyrimidine-4,6-diamineHuman3612
NTRK1 (TRKA)TrkTK4yneAA6-[(2r)-2-(3-fluorophenyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)imidazo[1,2-b]pyridazineHuman3620
NTRK1 (TRKA)TrkTK4yneAB6-[(2r)-2-(3-fluorophenyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)imidazo[1,2-b]pyridazineHuman3611
NTRK1 (TRKA)TrkTK4ypsA4-{6-[(3r)-3-(3-fluorophenyl)morpholin-4-yl]imidazo[1,2-b]pyridazin-3-yl}benzonitrileHuman3615
NTRK1 (TRKA)TrkTK5h3qAA1-[(3s,4r)-4-[3,4-bis(fluoranyl)phenyl]-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(5-ethoxy-4-methyl-2-phenyl-pyrazol-3-yl)ureaHuman7461
NTRK1 (TRKA)TrkTK5h3qAB1-[(3s,4r)-4-[3,4-bis(fluoranyl)phenyl]-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(5-ethoxy-4-methyl-2-phenyl-pyrazol-3-yl)ureaHuman7460
NTRK1 (TRKA)TrkTK5i8aAA(6r)-3-(methylsulfanyl)-6-phenyl-1-(1h-pyrazol-3-yl)-6,7-dihydrothieno[3,4-c]pyridin-4(5h)-oneHuman8311
NTRK1 (TRKA)TrkTK5i8aAB(6r)-3-(methylsulfanyl)-6-phenyl-1-(1h-pyrazol-3-yl)-6,7-dihydrothieno[3,4-c]pyridin-4(5h)-oneHuman8312
NTRK1 (TRKA)TrkTK5jfsAAn-{4-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-2-yl}-n'-(2,4-difluorophenyl)ureaHuman7506
NTRK1 (TRKA)TrkTK5jfsABn-{4-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-2-yl}-n'-(2,4-difluorophenyl)ureaHuman7502
NTRK1 (TRKA)TrkTK5jfvAAn-{5-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}-2-(4-chlorophenyl)acetamideHuman7504
NTRK1 (TRKA)TrkTK5jfvABn-{5-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}-2-(4-chlorophenyl)acetamideHuman7503
NTRK1 (TRKA)TrkTK5jfwAA2-(4-cyanophenyl)-n-{5-[7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}acetamideHuman7500
NTRK1 (TRKA)TrkTK5jfwAB2-(4-cyanophenyl)-n-{5-[7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}acetamideHuman7505
NTRK1 (TRKA)TrkTK5jfxAn-{5-[2-amino-7-(1-hydroxy-2-methylpropan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}-2-(5-chloropyridin-2-yl)acetamideHuman7501
NTRK1 (TRKA)TrkTK5kmiA1-(9~{h}-fluoren-9-yl)-3-(2-methyl-4-phenyl-pyrimidin-5-yl)ureaHuman7330
NTRK1 (TRKA)TrkTK5kmjAA~{n}-(pyridin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)ethanamideHuman7334
NTRK1 (TRKA)TrkTK5kmjAB~{n}-(pyridin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)ethanamideHuman7335
NTRK1 (TRKA)TrkTK5kmkA2-fluoranyl-~{n}-[2-(4-fluorophenyl)-6-methyl-pyridin-3-yl]-4-(trifluoromethyl)benzamideHuman7336
NTRK1 (TRKA)TrkTK5kmlA1-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-3-[[2-(trifluoromethyl)phenyl]methyl]ureaHuman7333
NTRK1 (TRKA)TrkTK5kmmA1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-naphthalen-1-yl-ureaHuman7331
NTRK1 (TRKA)TrkTK5kmnA1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-[[2-(trifluoromethyl)phenyl]methyl]ureaHuman7332
NTRK1 (TRKA)TrkTK5kmoA1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-pyridin-2-yl-ureaHuman7329
NTRK1 (TRKA)TrkTK5kvtAAentrectinibHuman9450
NTRK1 (TRKA)TrkTK5kvtABentrectinibHuman9451
NTRK1 (TRKA)TrkTK5wr7An-tert-butyl-2-[2-[6,6-dimethyl-8-(methylsulfonylamino)-11-oxidanylidene-naphtho[2,3-b][1]benzofuran-3-yl]ethynyl]-6-methyl-pyridine-4-carboxamideHuman8737
NTRK1 (TRKA)TrkTK6d1yAA2,4-dichloro-n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)benzamideHuman9873
NTRK1 (TRKA)TrkTK6d1yAB2,4-dichloro-n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)benzamideHuman9871
NTRK1 (TRKA)TrkTK6d1zAA5-{[5-(6-aminopyridin-2-yl)-2-chlorobenzene-1-carbonyl]amino}-1-phenyl-1h-pyrazole-3-carboxamideHuman9874
NTRK1 (TRKA)TrkTK6d1zAB5-{[5-(6-aminopyridin-2-yl)-2-chlorobenzene-1-carbonyl]amino}-1-phenyl-1h-pyrazole-3-carboxamideHuman9870
NTRK1 (TRKA)TrkTK6d20A5-{[2,4-dichloro-5-(pyridin-2-yl)benzene-1-carbonyl]amino}-n-(2-hydroxy-2-methylpropyl)-1-phenyl-1h-pyrazole-3-carboxamideHuman9875
NTRK1 (TRKA)TrkTK6d22A-Human9872
NTRK1 (TRKA)TrkTK6dkbA2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamideHuman10057
NTRK1 (TRKA)TrkTK6dkgAA2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-4-(2-hydroxy-2-methylpropoxy)benzamideHuman10059
NTRK1 (TRKA)TrkTK6dkgAB2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-4-(2-hydroxy-2-methylpropoxy)benzamideHuman10063
NTRK1 (TRKA)TrkTK6dkiAA6-amino-5-{[(3s)-4,4-difluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}pyrrolidin-3-yl]oxy}-n-methylpyridine-3-carboxamideHuman10060
NTRK1 (TRKA)TrkTK6dkiAB6-amino-5-{[(3s)-4,4-difluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}pyrrolidin-3-yl]oxy}-n-methylpyridine-3-carboxamideHuman10061
NTRK1 (TRKA)TrkTK6dkwAA5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamideHuman10056
NTRK1 (TRKA)TrkTK6dkwAB5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamideHuman10058
NTRK1 (TRKA)TrkTK6dkwBA5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamideHuman10062
NTRK1 (TRKA)TrkTK6dkwBB5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamideHuman10064
NTRK1 (TRKA)TrkTK6iqnA4-[[4-azanyl-3-(4-cyclohexylpiperazin-1-yl)-9,10-bis(oxidanylidene)anthracen-1-yl]amino]benzoic acidHuman11951
NTRK1 (TRKA)TrkTK6iqnB4-[[4-azanyl-3-(4-cyclohexylpiperazin-1-yl)-9,10-bis(oxidanylidene)anthracen-1-yl]amino]benzoic acidHuman11950
NTRK1 (TRKA)TrkTK6j5lAAn-{2-[({3-[6-(piperazin-1-yl)pyridin-3-yl]-1h-indazol-5-yl}amino)methyl]phenyl}methanesulfonamideHuman11436
NTRK1 (TRKA)TrkTK6j5lABn-{2-[({3-[6-(piperazin-1-yl)pyridin-3-yl]-1h-indazol-5-yl}amino)methyl]phenyl}methanesulfonamideHuman11435
NTRK1 (TRKA)TrkTK6j5lACn-{2-[({3-[6-(piperazin-1-yl)pyridin-3-yl]-1h-indazol-5-yl}amino)methyl]phenyl}methanesulfonamideHuman11437
NTRK1 (TRKA)TrkTK6nptA4-tert-butyl-n-(1,3-diphenyl-1h-pyrazol-5-yl)benzamideHuman11172
NTRK1 (TRKA)TrkTK6nspAAn-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)-2-(3-oxo-2,3-dihydro-4h-1,4-benzothiazin-4-yl)acetamideHuman11173
NTRK1 (TRKA)TrkTK6nspABn-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)-2-(3-oxo-2,3-dihydro-4h-1,4-benzothiazin-4-yl)acetamideHuman11175
NTRK1 (TRKA)TrkTK6nssAAn-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)-2-(10h-phenoxazin-10-yl)acetamideHuman11174
NTRK1 (TRKA)TrkTK6nssABn-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)-2-(10h-phenoxazin-10-yl)acetamideHuman11176
NTRK1 (TRKA)TrkTK6pl1AAn-(5-{[(7-methyl-4-oxo-4h-pyrido[1,2-a]pyrimidin-2-yl)methyl]sulfanyl}-1,3,4-thiadiazol-2-yl)-n'-[3-(trifluoromethyl)phenyl]ureaHuman11722
NTRK1 (TRKA)TrkTK6pl1ABn-(5-{[(7-methyl-4-oxo-4h-pyrido[1,2-a]pyrimidin-2-yl)methyl]sulfanyl}-1,3,4-thiadiazol-2-yl)-n'-[3-(trifluoromethyl)phenyl]ureaHuman11723
NTRK1 (TRKA)TrkTK6pl2An-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-2-{[1-(4-hydroxyphenyl)-1h-tetrazol-5-yl]sulfanyl}acetamideHuman11598
NTRK1 (TRKA)TrkTK6pl3AA2-[(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)amino]-2-oxoethyl 4-(1h-tetrazol-1-yl)benzoateHuman11599
NTRK1 (TRKA)TrkTK6pl3AB2-[(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)amino]-2-oxoethyl 4-(1h-tetrazol-1-yl)benzoateHuman11600
NTRK1 (TRKA)TrkTK6pl4AAn-{[5-(methoxymethyl)-2-(trifluoromethoxy)phenyl]methyl}-n'-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)ureaHuman12463
NTRK1 (TRKA)TrkTK6pl4ABn-{[5-(methoxymethyl)-2-(trifluoromethoxy)phenyl]methyl}-n'-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)ureaHuman12464
NTRK1 (TRKA)TrkTK6pmaAn-[2-chloro-5-(trifluoromethyl)phenyl]-2-[1-(4-methoxyphenyl)-4-oxo-1,4-dihydro-5h-pyrazolo[3,4-d]pyrimidin-5-yl]acetamideHuman12006
NTRK1 (TRKA)TrkTK6pmbA2-[5,7-dimethyl-2-(pyridin-3-yl)[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-n-[3-(trifluoromethyl)phenyl]acetamideHuman12001
NTRK1 (TRKA)TrkTK6pmcAn-(6-{[(5-chloro-2-methoxyphenyl)carbamoyl]amino}-1,3-benzothiazol-2-yl)benzamideHuman12002
NTRK1 (TRKA)TrkTK6pmeAAn-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamideHuman12004
NTRK1 (TRKA)TrkTK6pmeABn-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamideHuman12005
NTRK1 (TRKA)TrkTK6pmeBAn-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamideHuman12007
NTRK1 (TRKA)TrkTK6pmeBBn-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamideHuman12000
NTRK1 (TRKA)TrkTK6pmeCAn-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamideHuman11999
NTRK1 (TRKA)TrkTK6pmeCBn-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamideHuman12003
NTRK1 (TRKA)TrkTK7vkmAA-Human13946
NTRK1 (TRKA)TrkTK7vkmAB-Human13942
NTRK1 (TRKA)TrkTK7vknAArepotrectinibHuman13945
NTRK1 (TRKA)TrkTK7vknABrepotrectinibHuman13944
NTRK1 (TRKA)TrkTK7vkoArepotrectinibHuman13943
NTRK1 (TRKA)TrkTK7xafA4^6,14-dimethyl-n-(3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-10-oxo-5-oxa-11,14-diaza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclo-tetradecaphan-2-yne-45-carboxamideHuman14232
NTRK1 (TRKA)TrkTK7xbiAA4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]-~{n}-[3-(1-methylpyrazol-4-yl)-1~{h}-indazol-5-yl]-2-(trifluoromethyl)benzamideHuman14687
NTRK1 (TRKA)TrkTK7xbiAB4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]-~{n}-[3-(1-methylpyrazol-4-yl)-1~{h}-indazol-5-yl]-2-(trifluoromethyl)benzamideHuman14686
NTRK1 (TRKA)TrkTK8j5wAn-(3-cyclopropyl-5-((4-methylpiperazin-1-yl)methyl)phenyl)-4^6-methyl-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamideHuman14985
NTRK1 (TRKA)TrkTK8j5xAn-(3-cyclopropyl-5-((4-methylpiperazin-1-yl)methyl)phenyl)-4^6-methyl-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamideHuman14987
NTRK1 (TRKA)TrkTK8j61A4^6-methyl-n-(3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamideHuman14986
NTRK1 (TRKA)TrkTK8j63A4^6-methyl-n-(3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-11-oxo-5-oxa-10,14-diaza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamideHuman14984
NTRK2 (TRKB)TrkTK4aszA-Human3599
NTRK2 (TRKB)TrkTK4at3A(5z)-5-(carbamoylimino)-3-[(5r)-6,7,8,9-tetrahydro-5h-benzo[7]annulen-5-ylsulfanyl]-2,5-dihydroisothiazole-4-carboxamideHuman3600
NTRK2 (TRKB)TrkTK4at4A1-[4-(4-aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]ureaHuman3598
NTRK2 (TRKB)TrkTK4at5A5-{3-methoxy-4-[(4-methoxybenzyl)oxy]benzyl}pyrimidine-2,4-diamineHuman3597
NTRK3 (TRKC)TrkTK3v5qA1-(3-{[(3z)-2-oxo-3-(1h-pyrrol-2-ylmethylidene)-2,3-dihydro-1h-indol-6-yl]amino}phenyl)-3-[3-(trifluoromethyl)phenyl]ureaHuman102
NTRK3 (TRKC)TrkTK3v5qB1-(3-{[(3z)-2-oxo-3-(1h-pyrrol-2-ylmethylidene)-2,3-dihydro-1h-indol-6-yl]amino}phenyl)-3-[3-(trifluoromethyl)phenyl]ureaHuman97
NTRK3 (TRKC)TrkTK4ymjAA4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrileHuman101
NTRK3 (TRKC)TrkTK4ymjAB4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrileHuman98
NTRK3 (TRKC)TrkTK4ymjBA4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrileHuman100
NTRK3 (TRKC)TrkTK4ymjBB4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrileHuman99
NTRK3 (TRKC)TrkTK6kzcA3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-2-methyl-~{n}-[3-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]benzamideHuman11696
NTRK3 (TRKC)TrkTK6kzdA3-[2-[6-(4-aminophenyl)imidazo[1,2-a]pyrazin-3-yl]ethynyl]-2-methyl-~{n}-[3-(4-methylpiperazin-1-yl)-5-propan-2-yl-phenyl]benzamideHuman11697
OXSR1 (OSR1)STE20STE2vwiAAphosphoaminophosphonic acid-adenylate esterHuman4842
OXSR1 (OSR1)STE20STE2vwiABphosphoaminophosphonic acid-adenylate esterHuman4839
OXSR1 (OSR1)STE20STE2vwiBAphosphoaminophosphonic acid-adenylate esterHuman4843
OXSR1 (OSR1)STE20STE2vwiBBphosphoaminophosphonic acid-adenylate esterHuman4836
OXSR1 (OSR1)STE20STE2vwiCAphosphoaminophosphonic acid-adenylate esterHuman4838
OXSR1 (OSR1)STE20STE2vwiCBphosphoaminophosphonic acid-adenylate esterHuman4844
OXSR1 (OSR1)STE20STE2vwiDAphosphoaminophosphonic acid-adenylate esterHuman4835
OXSR1 (OSR1)STE20STE2vwiDBphosphoaminophosphonic acid-adenylate esterHuman4833
OXSR1 (OSR1)STE20STE3dakAphosphoaminophosphonic acid-adenylate esterHuman4834
OXSR1 (OSR1)STE20STE3dakBphosphoaminophosphonic acid-adenylate esterHuman4841
OXSR1 (OSR1)STE20STE3dakCphosphoaminophosphonic acid-adenylate esterHuman4837
OXSR1 (OSR1)STE20STE3dakDphosphoaminophosphonic acid-adenylate esterHuman4840
PAK1STE20STE1f3mC-Human161
PAK1STE20STE1f3mD-Human158
PAK1STE20STE1yhvA-Human177
PAK1STE20STE1yhwA-Human160
PAK1STE20STE2hy81(5s,6r,7r,9r)-12-hydroxy-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9-tetrahydro-5h,14h-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-oneHuman172
PAK1STE20STE3fxzAAoctahedral ru-pyridocarbazoleHuman7198
PAK1STE20STE3fxzABoctahedral ru-pyridocarbazoleHuman7200
PAK1STE20STE3fy0Aruthenium pyridocarbazoleHuman7202
PAK1STE20STE3q4zAAphosphoaminophosphonic acid-adenylate esterHuman166
PAK1STE20STE3q4zABphosphoaminophosphonic acid-adenylate esterHuman174
PAK1STE20STE3q4zBA-Human144
PAK1STE20STE3q4zBB-Human183
PAK1STE20STE3q52A-Human146
PAK1STE20STE3q53Aadenosine-5'-triphosphateHuman165
PAK1STE20STE4dawAA[1,3-dioxo-6-(pyridin-2-yl-kappan)-2,3-dihydro-1h-isoindol-5-yl-kappac~5~][(thioxomethylidene)azanido-kappan](1,4,7-trithionane-kappa~3~s~1~,s~4~,s~7~)rutheniumHuman7201
PAK1STE20STE4dawAB[1,3-dioxo-6-(pyridin-2-yl-kappan)-2,3-dihydro-1h-isoindol-5-yl-kappac~5~][(thioxomethylidene)azanido-kappan](1,4,7-trithionane-kappa~3~s~1~,s~4~,s~7~)rutheniumHuman7199
PAK1STE20STE4eqcAA6-[2-chloro-4-(1,3-thiazol-5-yl)phenyl]-8-ethyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman180
PAK1STE20STE4eqcAB6-[2-chloro-4-(1,3-thiazol-5-yl)phenyl]-8-ethyl-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman147
PAK1STE20STE4o0rApf-3758309Human171
PAK1STE20STE4o0rB-Human145
PAK1STE20STE4o0tA1-({1-(2-aminopyrimidin-4-yl)-2-[(2-methoxyethyl)amino]-1h-benzimidazol-6-yl}ethynyl)cyclohexanolHuman143
PAK1STE20STE4o0tB-Human141
PAK1STE20STE4p90A[2-chloro-5-(hydroxymethyl)phenyl]{5-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl}methanoneHuman164
PAK1STE20STE4p90B[2-chloro-5-(hydroxymethyl)phenyl]{5-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl}methanoneHuman151
PAK1STE20STE4zjiAA2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepineHuman159
PAK1STE20STE4zjiAB2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepineHuman175
PAK1STE20STE4zjiBA2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepineHuman168
PAK1STE20STE4zjiBB2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepineHuman185
PAK1STE20STE4zjiCA2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepineHuman167
PAK1STE20STE4zjiCB2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepineHuman152
PAK1STE20STE4zjiDA2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepineHuman139
PAK1STE20STE4zjiDB2-chloro-5-ethyl-8-fluoro-11-(4-methylpiperazin-1-yl)-dibenzodiazepineHuman150
PAK1STE20STE4zjjAA(s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamideHuman157
PAK1STE20STE4zjjAB(s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamideHuman153
PAK1STE20STE4zjjBA(s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamideHuman176
PAK1STE20STE4zjjBB(s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamideHuman137
PAK1STE20STE4zjjCA(s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamideHuman182
PAK1STE20STE4zjjCB(s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamideHuman178
PAK1STE20STE4zjjDA(s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamideHuman169
PAK1STE20STE4zjjDB(s)-n-(tert-butyl)-3-((2-chloro-5-ethyl-8-fluoro-dibenzodiazepin-11-yl)amino)pyrrolidine-1-carboxamideHuman162
PAK1STE20STE4zloAA2,8-difluoro-11-(4-methylpiperazin-1-yl)-5h-dibenzo[b,e][1,4]diazepineHuman142
PAK1STE20STE4zloAB2,8-difluoro-11-(4-methylpiperazin-1-yl)-5h-dibenzo[b,e][1,4]diazepineHuman181
PAK1STE20STE4zloBA-Human188
PAK1STE20STE4zloBB-Human170
PAK1STE20STE4zy4A2-(4-aminopiperidin-1-yl)-n-(5-cyclopropyl-1h-pyrazol-3-yl)thieno[3,2-d]pyrimidin-4-amineHuman187
PAK1STE20STE4zy4B2-(4-aminopiperidin-1-yl)-n-(5-cyclopropyl-1h-pyrazol-3-yl)thieno[3,2-d]pyrimidin-4-amineHuman154
PAK1STE20STE4zy5An~2~-[(trans-4-aminocyclohexyl)methyl]-n~4~-(3-cyclopropyl-1h-pyrazol-5-yl)pyrimidine-2,4-diamineHuman155
PAK1STE20STE4zy5Bn~2~-[(trans-4-aminocyclohexyl)methyl]-n~4~-(3-cyclopropyl-1h-pyrazol-5-yl)pyrimidine-2,4-diamineHuman163
PAK1STE20STE4zy6AAn~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman138
PAK1STE20STE4zy6ABn~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman173
PAK1STE20STE4zy6BAn~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman156
PAK1STE20STE4zy6BBn~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman184
PAK1STE20STE5dewA8-[(trans-4-aminocyclohexyl)methyl]-6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-2-(ethylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman7408
PAK1STE20STE5dewB8-[(trans-4-aminocyclohexyl)methyl]-6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-2-(ethylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman7409
PAK1STE20STE5deyA8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6364
PAK1STE20STE5deyB8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6365
PAK1STE20STE5dfpAA6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-8-ethyl-2-{[2-(1-methylpiperidin-4-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6366
PAK1STE20STE5dfpAB6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-8-ethyl-2-{[2-(1-methylpiperidin-4-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6363
PAK1STE20STE5imeA8-(3-aminopropyl)-6-[2-chloro-4-(3-methyl-2-oxopyrazin-1(2h)-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6644
PAK1STE20STE5imeB8-(3-aminopropyl)-6-[2-chloro-4-(3-methyl-2-oxopyrazin-1(2h)-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6643
PAK1STE20STE5kbqA[4-methyl-3-[methyl-[2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]pyrimidin-4-yl]amino]phenyl]methanolHuman7081
PAK1STE20STE5kbqB-Human7082
PAK1STE20STE5kbrA(4-chlorophenyl)-[5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]methanoneHuman7080
PAK1STE20STE5kbrB(4-chlorophenyl)-[5-(1-piperidin-4-ylpyrazol-4-yl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]methanoneHuman7079
PAK1STE20STE6b16An~4~-(5-cyclopropyl-1h-pyrazol-3-yl)-n~2~-[(1s)-1-(1h-pyrrolo[3,2-b]pyridin-5-yl)ethyl]pyrimidine-2,4-diamineHuman8574
PAK1STE20STE6b16Bn~4~-(5-cyclopropyl-1h-pyrazol-3-yl)-n~2~-[(1s)-1-(1h-pyrrolo[3,2-b]pyridin-5-yl)ethyl]pyrimidine-2,4-diamineHuman8575
PAK1STE20STE7vtoAA4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman14483
PAK1STE20STE7vtoAB4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman14484
PAK1STE20STE8x5zAA-Human15049
PAK1STE20STE8x5zAB-Human15048
PAK3STE20STE6fd3AAadenosine-5'-diphosphateHuman9462
PAK3STE20STE6fd3ABadenosine-5'-diphosphateHuman9463
PAK4STE20STE2bvaA-Human1394
PAK4STE20STE2bvaB-Human1407
PAK4STE20STE2cdzAAn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman1378
PAK4STE20STE2cdzABn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman1374
PAK4STE20STE2j0iAA-Human1391
PAK4STE20STE2j0iAB-Human1377
PAK4STE20STE2q0nAA-Human1393
PAK4STE20STE2q0nAB-Human1401
PAK4STE20STE2x4zApf-3758309Human1387
PAK4STE20STE4appAAn-[6,6-dimethyl-5-[(2s)-4-methyl-2-(phenylmethyl)piperazin-1-yl]carbonyl-2,4-dihydropyrrolo[3,4-c]pyrazol-3-yl]-3-phenoxy-benzamideHuman1385
PAK4STE20STE4appABn-[6,6-dimethyl-5-[(2s)-4-methyl-2-(phenylmethyl)piperazin-1-yl]carbonyl-2,4-dihydropyrrolo[3,4-c]pyrazol-3-yl]-3-phenoxy-benzamideHuman1390
PAK4STE20STE4fieAphosphoaminophosphonic acid-adenylate esterHuman1405
PAK4STE20STE4fieBphosphoaminophosphonic acid-adenylate esterHuman1372
PAK4STE20STE4fifAAphosphoaminophosphonic acid-adenylate esterHuman1395
PAK4STE20STE4fifABphosphoaminophosphonic acid-adenylate esterHuman1370
PAK4STE20STE4fifBAphosphoaminophosphonic acid-adenylate esterHuman1381
PAK4STE20STE4fifBBphosphoaminophosphonic acid-adenylate esterHuman1379
PAK4STE20STE4figAphosphoaminophosphonic acid-adenylate esterHuman1392
PAK4STE20STE4figBphosphoaminophosphonic acid-adenylate esterHuman1373
PAK4STE20STE4fihAA-Human1399
PAK4STE20STE4fihAB-Human1402
PAK4STE20STE4fiiAA-Human1383
PAK4STE20STE4fiiAB-Human1396
PAK4STE20STE4fijA-Human1408
PAK4STE20STE4jdhAA-Human1371
PAK4STE20STE4jdhAB-Human1406
PAK4STE20STE4jdiAAphosphoaminophosphonic acid-adenylate esterHuman1403
PAK4STE20STE4jdiABphosphoaminophosphonic acid-adenylate esterHuman1380
PAK4STE20STE4jdjAA-Human1400
PAK4STE20STE4jdjAB-Human1397
PAK4STE20STE4jdkAA-Human1375
PAK4STE20STE4jdkAB-Human1398
PAK4STE20STE4l67A-Human1376
PAK4STE20STE4njdAAn-(1h-indazol-5-yl)-n'-[2-(1h-indol-3-yl)ethyl]-6-methoxy-1,3,5-triazine-2,4-diamineHuman1382
PAK4STE20STE4njdABn-(1h-indazol-5-yl)-n'-[2-(1h-indol-3-yl)ethyl]-6-methoxy-1,3,5-triazine-2,4-diamineHuman1384
PAK4STE20STE4o0vA1-({1-(2-aminopyrimidin-4-yl)-2-[(2-methoxyethyl)amino]-1h-benzimidazol-6-yl}ethynyl)cyclohexanolHuman1386
PAK4STE20STE4o0xA1-{[1-(4-amino-1,3,5-triazin-2-yl)-2-methyl-1h-benzimidazol-6-yl]ethynyl}cyclohexanolHuman1404
PAK4STE20STE4o0yA4-[1-(4-amino-1,3,5-triazin-2-yl)-2-(ethylamino)-1h-benzimidazol-6-yl]-2-methylbut-3-yn-2-olHuman1388
PAK4STE20STE4xbrAadenosine-5'-triphosphateHuman6257
PAK4STE20STE4xbuA-Human6256
PAK4STE20STE5bmsAn~2~-[(7-chloro-1h-benzimidazol-6-yl)methyl]-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)pyrimidine-2,4-diamineHuman1389
PAK4STE20STE5i0bA6-bromo-2-[1-methyl-3-(propan-2-yl)-1h-pyrazol-4-yl]-1h-imidazo[4,5-b]pyridineHuman7315
PAK4STE20STE5upkBphosphoaminophosphonic acid-adenylate esterHuman9435
PAK4STE20STE5uplA-Human9436
PAK4STE20STE5vedAstaurosporineHuman8570
PAK4STE20STE5veeA6-(2,4-dichlorophenyl)-8-ethyl-2-{[3-fluoro-4-(piperazin-1-yl)phenyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman8572
PAK4STE20STE5vefAA5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman8569
PAK4STE20STE5vefAB5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman8571
PAK4STE20STE5xvaA[6-chloranyl-4-[(5-methyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl]-[(3r)-3-methylpiperazin-1-yl]methanoneHuman9550
PAK4STE20STE5xvfA2-(4-azanylpiperidin-1-yl)-6-chloranyl-n-(1-methylimidazol-4-yl)quinazolin-4-amineHuman9549
PAK4STE20STE5xvgA[6-chloranyl-4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl]-[(3r)-3-methylpiperazin-1-yl]methanoneHuman9551
PAK4STE20STE5zjwAA(3z)-n-[(1s)-2-hydroxy-1-phenylethyl]-3-[(1h-imidazol-2-yl)(phenyl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamideHuman10999
PAK4STE20STE5zjwAB(3z)-n-[(1s)-2-hydroxy-1-phenylethyl]-3-[(1h-imidazol-2-yl)(phenyl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamideHuman11000
PAK4STE20STE6wlxAA-Human12399
PAK4STE20STE6wlxAB-Human12400
PAK4STE20STE6wlyAA-Human12397
PAK4STE20STE6wlyAB-Human12396
PAK4STE20STE6wlyAC-Human12398
PAK4STE20STE7cmbA1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indole-3-carboxamideHuman13818
PAK4STE20STE7cp3A[(3r)-3-azanylpiperidin-1-yl]-[1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]methanoneHuman13849
PAK4STE20STE7cp4A[1-(2-azanylpyrimidin-4-yl)-6-[2-(1-oxidanylcyclohexyl)ethynyl]indol-3-yl]-[(3s)-3-methylpiperazin-1-yl]methanoneHuman13850
PAK4STE20STE7s46Aphosphoaminophosphonic acid-adenylate esterHuman14495
PAK4STE20STE7s47AAphosphoaminophosphonic acid-adenylate esterHuman14493
PAK4STE20STE7s47ABphosphoaminophosphonic acid-adenylate esterHuman14494
PAK4STE20STE7s48AA-Human14492
PAK4STE20STE7s48AB-Human14491
PAK4STE20STE8ahgAA~{n}-methyl-3-propan-2-yl-1~{h}-pyrazolo[3,4-c]pyridine-4-carboxamideHuman14370
PAK4STE20STE8ahgAB~{n}-methyl-3-propan-2-yl-1~{h}-pyrazolo[3,4-c]pyridine-4-carboxamideHuman14368
PAK4STE20STE8ahhAA5-cyano-~{n}-methyl-pyrazolo[1,5-a]pyridine-3-carboxamideHuman14372
PAK4STE20STE8ahhAB5-cyano-~{n}-methyl-pyrazolo[1,5-a]pyridine-3-carboxamideHuman14371
PAK4STE20STE8ahiA~{n}-methyl-1,3-benzothiazole-6-carboxamideHuman14369
PAK5STE20STE2f57AA-Human200
PAK5STE20STE2f57AB-Human202
PAK5STE20STE2f57BAn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman199
PAK5STE20STE2f57BBn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman201
PAK5STE20STE8c12AA-Human14952
PAK5STE20STE8c12AB-Human14953
PAK6STE20STE2c30AA-Human4679
PAK6STE20STE2c30AB-Human4678
PAK6STE20STE4ks7AApf-3758309Human4682
PAK6STE20STE4ks7ABpf-3758309Human4681
PAK6STE20STE4ks8AAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4683
PAK6STE20STE4ks8ABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4680
PASKCAMKLCAMK3dlsAadenosine-5'-diphosphateHuman3382
PASKCAMKLCAMK3dlsBadenosine-5'-diphosphateHuman3381
PASKCAMKLCAMK3dlsCadenosine-5'-diphosphateHuman3377
PASKCAMKLCAMK3dlsDadenosine-5'-diphosphateHuman3378
PASKCAMKLCAMK3dlsEadenosine-5'-diphosphateHuman3379
PASKCAMKLCAMK3dlsFadenosine-5'-diphosphateHuman3380
PBKTOPKOther5j0aA-Human7083
PBKTOPKOther5j0aB-Human7084
PDGFRA (PDGFRa)PDGFRTK5grnAAn-[2-(dimethylamino)ethyl]-n-[[4-[[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methyl]pyridine-3-carboxamideHuman9479
PDGFRA (PDGFRa)PDGFRTK5grnABn-[2-(dimethylamino)ethyl]-n-[[4-[[4-methyl-3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methyl]pyridine-3-carboxamideHuman9478
PDGFRA (PDGFRa)PDGFRTK5k5xA-Human6962
PDGFRA (PDGFRa)PDGFRTK6a32A-Human11327
PDGFRA (PDGFRa)PDGFRTK6joiA1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amineHuman12102
PDGFRA (PDGFRa)PDGFRTK6jojA1-(2-{5-[(3-methyloxetan-3-yl)methoxy]-1h-benzimidazol-1-yl}quinolin-8-yl)piperidin-4-amineHuman12104
PDGFRA (PDGFRa)PDGFRTK6jokAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman12105
PDGFRA (PDGFRa)PDGFRTK6jolA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman12103
PDGFRA (PDGFRa)PDGFRTK8pqhA(1~{s})-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15107
PDGFRA (PDGFRa)PDGFRTK8pqiAA(1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15109
PDGFRA (PDGFRa)PDGFRTK8pqiAB(1~{s})-~{n}-ethyl-1-(4-fluorophenyl)-1-[2-[4-[6-(1-methylpyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]piperazin-1-yl]pyrimidin-5-yl]ethanamineHuman15104
PDGFRA (PDGFRa)PDGFRTK8pqjAA-Human15106
PDGFRA (PDGFRa)PDGFRTK8pqjAB-Human15105
PDGFRA (PDGFRa)PDGFRTK8pqkAA-Human15110
PDGFRA (PDGFRa)PDGFRTK8pqkAB-Human15108
PDPK1 (PDK1)PDK1AGC1h1wAAadenosine-5'-triphosphateHuman3186
PDPK1 (PDK1)PDK1AGC1h1wABadenosine-5'-triphosphateHuman3194
PDPK1 (PDK1)PDK1AGC1okyAAstaurosporineHuman3164
PDPK1 (PDK1)PDK1AGC1okyABstaurosporineHuman3195
PDPK1 (PDK1)PDK1AGC1okzA7-hydroxystaurosporineHuman3209
PDPK1 (PDK1)PDK1AGC1uu3AA(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHuman3180
PDPK1 (PDK1)PDK1AGC1uu3AB(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHuman3248
PDPK1 (PDK1)PDK1AGC1uu7A3-(1h-indol-3-yl)-4-(1-{2-[(2s)-1-methylpyrrolidinyl]ethyl}-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3224
PDPK1 (PDK1)PDK1AGC1uu8AA3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3239
PDPK1 (PDK1)PDK1AGC1uu8AB3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3237
PDPK1 (PDK1)PDK1AGC1uu9AA3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman6800
PDPK1 (PDK1)PDK1AGC1uu9AB3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman6799
PDPK1 (PDK1)PDK1AGC1uvrA3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3193
PDPK1 (PDK1)PDK1AGC1z5mAn-(3-{[5-bromo-2-({3-[(pyrrolidin-1-ylcarbonyl)amino]phenyl}amino)pyrimidin-4-yl]amino}propyl)-2,2-dimethylmalonamideHuman3152
PDPK1 (PDK1)PDK1AGC2biyAAadenosine-5'-triphosphateHuman3232
PDPK1 (PDK1)PDK1AGC2biyABadenosine-5'-triphosphateHuman3169
PDPK1 (PDK1)PDK1AGC2pe0A5-hydroxy-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-2-oneHuman3206
PDPK1 (PDK1)PDK1AGC2pe1A1-{2-oxo-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-5-yl}ureaHuman3167
PDPK1 (PDK1)PDK1AGC2pe2A3-[5-({5-[(aminocarbonyl)amino]-2-oxo-2h-indol-3-yl}methyl)-1h-pyrrol-3-yl]-n-(2-piperidin-1-ylethyl)benzamideHuman3163
PDPK1 (PDK1)PDK1AGC2r7bA10,11-dimethoxy-4-methyldibenzo[c,f]-2,7-naphthyridine-3,6-diamineHuman3215
PDPK1 (PDK1)PDK1AGC2xchA8-(cyclohexa-2,5-dien-1-ylideneamino)-1-(piperidin-4-ylmethyl)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman3220
PDPK1 (PDK1)PDK1AGC2xckA1-methyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-n-[(2-methylpyridin-4-yl)methyl]-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman3201
PDPK1 (PDK1)PDK1AGC3h9oA2-(1h-imidazol-1-yl)-9-methoxy-8-(2-methoxyethoxy)benzo[c][2,7]naphthyridin-4-amineHuman3226
PDPK1 (PDK1)PDK1AGC3hrcAAadenosine-5'-triphosphateHuman3172
PDPK1 (PDK1)PDK1AGC3hrcABadenosine-5'-triphosphateHuman3223
PDPK1 (PDK1)PDK1AGC3hrfAAadenosine-5'-triphosphateHuman3170
PDPK1 (PDK1)PDK1AGC3hrfABadenosine-5'-triphosphateHuman3247
PDPK1 (PDK1)PDK1AGC3ionA2-(5-{[(2s)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amineHuman3218
PDPK1 (PDK1)PDK1AGC3iopA2-(5-{[(2r)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amineHuman3204
PDPK1 (PDK1)PDK1AGC3naxA1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman3200
PDPK1 (PDK1)PDK1AGC3nayA4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-oneHuman3231
PDPK1 (PDK1)PDK1AGC3nayB4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-oneHuman3203
PDPK1 (PDK1)PDK1AGC3nunAA6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amineHuman3183
PDPK1 (PDK1)PDK1AGC3nunAB6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amineHuman3216
PDPK1 (PDK1)PDK1AGC3nusAA1h-indazol-3-amineHuman3233
PDPK1 (PDK1)PDK1AGC3nusAB1h-indazol-3-amineHuman3185
PDPK1 (PDK1)PDK1AGC3nuuAA3,4-dihydroisoquinolin-1(2h)-oneHuman3214
PDPK1 (PDK1)PDK1AGC3nuuAB3,4-dihydroisoquinolin-1(2h)-oneHuman3159
PDPK1 (PDK1)PDK1AGC3nuyAAquinazolin-4(1h)-oneHuman3236
PDPK1 (PDK1)PDK1AGC3nuyABquinazolin-4(1h)-oneHuman3242
PDPK1 (PDK1)PDK1AGC3orxA-Human3235
PDPK1 (PDK1)PDK1AGC3orxB-Human3178
PDPK1 (PDK1)PDK1AGC3orxC-Human3245
PDPK1 (PDK1)PDK1AGC3orxD-Human3210
PDPK1 (PDK1)PDK1AGC3orxE-Human3202
PDPK1 (PDK1)PDK1AGC3orxF-Human3228
PDPK1 (PDK1)PDK1AGC3orxG-Human3189
PDPK1 (PDK1)PDK1AGC3orxH-Human3177
PDPK1 (PDK1)PDK1AGC3orzAA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3197
PDPK1 (PDK1)PDK1AGC3orzAB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3181
PDPK1 (PDK1)PDK1AGC3orzBA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3160
PDPK1 (PDK1)PDK1AGC3orzBB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3198
PDPK1 (PDK1)PDK1AGC3orzCA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3150
PDPK1 (PDK1)PDK1AGC3orzCB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3243
PDPK1 (PDK1)PDK1AGC3orzDA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3192
PDPK1 (PDK1)PDK1AGC3orzDB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3184
PDPK1 (PDK1)PDK1AGC3otuA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3217
PDPK1 (PDK1)PDK1AGC3pwyAn-[2-({6-[(2-sulfanylethyl)amino]pyrimidin-4-yl}amino)ethyl]propanamideHuman3155
PDPK1 (PDK1)PDK1AGC3qc4AA1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman9254
PDPK1 (PDK1)PDK1AGC3qc4AB1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman9253
PDPK1 (PDK1)PDK1AGC3qc4BA1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman9255
PDPK1 (PDK1)PDK1AGC3qc4BB1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman9256
PDPK1 (PDK1)PDK1AGC3qcqAA6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamineHuman3205
PDPK1 (PDK1)PDK1AGC3qcqAB6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamineHuman3166
PDPK1 (PDK1)PDK1AGC3qcsAA6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amineHuman3179
PDPK1 (PDK1)PDK1AGC3qcsAB6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amineHuman3157
PDPK1 (PDK1)PDK1AGC3qcxAA6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amineHuman3187
PDPK1 (PDK1)PDK1AGC3qcxAB6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amineHuman3249
PDPK1 (PDK1)PDK1AGC3qcyAA(2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamideHuman3151
PDPK1 (PDK1)PDK1AGC3qcyAB(2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamideHuman3161
PDPK1 (PDK1)PDK1AGC3qd0AA(3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamideHuman3196
PDPK1 (PDK1)PDK1AGC3qd0AB(3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamideHuman3162
PDPK1 (PDK1)PDK1AGC3qd3AAtert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamateHuman3188
PDPK1 (PDK1)PDK1AGC3qd3ABtert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamateHuman3171
PDPK1 (PDK1)PDK1AGC3qd4AAtert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamateHuman3225
PDPK1 (PDK1)PDK1AGC3qd4ABtert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamateHuman3190
PDPK1 (PDK1)PDK1AGC3rcjA3-(1-benzyl-1h-1,2,3-triazol-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman3154
PDPK1 (PDK1)PDK1AGC3rwpAA[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanoneHuman3208
PDPK1 (PDK1)PDK1AGC3rwpAB[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanoneHuman3199
PDPK1 (PDK1)PDK1AGC3rwqA[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[2-(pyridin-3-yl)ethyl]amino}pyrazin-2-yl)methanoneHuman3213
PDPK1 (PDK1)PDK1AGC3sc1A6-[2-(hydroxymethyl)phenyl]isoquinolin-1(2h)-oneHuman3173
PDPK1 (PDK1)PDK1AGC4a06AAadenosine-5'-triphosphateHuman3207
PDPK1 (PDK1)PDK1AGC4a06ABadenosine-5'-triphosphateHuman3227
PDPK1 (PDK1)PDK1AGC4a07AAadenosine-5'-triphosphateHuman3234
PDPK1 (PDK1)PDK1AGC4a07ABadenosine-5'-triphosphateHuman3238
PDPK1 (PDK1)PDK1AGC4aw0AAadenosine-5'-triphosphateHuman3176
PDPK1 (PDK1)PDK1AGC4aw0ABadenosine-5'-triphosphateHuman3241
PDPK1 (PDK1)PDK1AGC4aw1AAadenosine-5'-triphosphateHuman3229
PDPK1 (PDK1)PDK1AGC4aw1ABadenosine-5'-triphosphateHuman3221
PDPK1 (PDK1)PDK1AGC4ct1AAadenosine-5'-triphosphateHuman3158
PDPK1 (PDK1)PDK1AGC4ct1ABadenosine-5'-triphosphateHuman3168
PDPK1 (PDK1)PDK1AGC4ct2AAadenosine-5'-triphosphateHuman3153
PDPK1 (PDK1)PDK1AGC4ct2ABadenosine-5'-triphosphateHuman3230
PDPK1 (PDK1)PDK1AGC4rqkAAadenosine-5'-triphosphateHuman3175
PDPK1 (PDK1)PDK1AGC4rqkABadenosine-5'-triphosphateHuman3156
PDPK1 (PDK1)PDK1AGC4rqkACadenosine-5'-triphosphateHuman3211
PDPK1 (PDK1)PDK1AGC4rqvAAadenosine-5'-triphosphateHuman3219
PDPK1 (PDK1)PDK1AGC4rqvABadenosine-5'-triphosphateHuman3182
PDPK1 (PDK1)PDK1AGC4rqvACadenosine-5'-triphosphateHuman3222
PDPK1 (PDK1)PDK1AGC4rrvAAadenosine-5'-triphosphateHuman3244
PDPK1 (PDK1)PDK1AGC4rrvABadenosine-5'-triphosphateHuman3212
PDPK1 (PDK1)PDK1AGC4rrvACadenosine-5'-triphosphateHuman3191
PDPK1 (PDK1)PDK1AGC4xx9AAadenosine-5'-triphosphateHuman6193
PDPK1 (PDK1)PDK1AGC4xx9ABadenosine-5'-triphosphateHuman6192
PDPK1 (PDK1)PDK1AGC5ackAAadenosine-5'-triphosphateHuman6191
PDPK1 (PDK1)PDK1AGC5ackABadenosine-5'-triphosphateHuman6194
PDPK1 (PDK1)PDK1AGC5hkmA4-ethyl-6-[5-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-2-amineHuman6670
PDPK1 (PDK1)PDK1AGC5hngA6-methoxy-2-(1h-pyrazol-5-yl)-1h-benzimidazoleHuman6675
PDPK1 (PDK1)PDK1AGC5ho7AA5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamideHuman6673
PDPK1 (PDK1)PDK1AGC5ho7AB5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamideHuman6671
PDPK1 (PDK1)PDK1AGC5ho8AA4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman6674
PDPK1 (PDK1)PDK1AGC5ho8AB4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman6672
PDPK1 (PDK1)PDK1AGC5lvlAA2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHuman7106
PDPK1 (PDK1)PDK1AGC5lvlAB2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHuman7110
PDPK1 (PDK1)PDK1AGC5lvmAAadenineHuman7112
PDPK1 (PDK1)PDK1AGC5lvmABadenineHuman7103
PDPK1 (PDK1)PDK1AGC5lvmACadenineHuman7138
PDPK1 (PDK1)PDK1AGC5lvnAAadenosineHuman7105
PDPK1 (PDK1)PDK1AGC5lvnABadenosineHuman7109
PDPK1 (PDK1)PDK1AGC5lvoAAadenosine-5'-triphosphateHuman7104
PDPK1 (PDK1)PDK1AGC5lvoABadenosine-5'-triphosphateHuman7114
PDPK1 (PDK1)PDK1AGC5lvpAadenosine-5'-triphosphateHuman7102
PDPK1 (PDK1)PDK1AGC5lvpBadenosine-5'-triphosphateHuman7113
PDPK1 (PDK1)PDK1AGC5lvpCadenosine-5'-triphosphateHuman7111
PDPK1 (PDK1)PDK1AGC5lvpDadenosine-5'-triphosphateHuman7108
PDPK1 (PDK1)PDK1AGC5mrdAAadenosine-5'-triphosphateHuman7395
PDPK1 (PDK1)PDK1AGC5mrdABadenosine-5'-triphosphateHuman7394
PDPK1 (PDK1)PDK1AGC8dqtA-Human14812
PEAK1 (SgK269)NKF3Other6bhcAA-Human9068
PEAK1 (SgK269)NKF3Other6bhcAB-Human9067
PHKG2 (PHKg2)PHKCAMK2y7jAAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1894
PHKG2 (PHKg2)PHKCAMK2y7jABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1893
PHKG2 (PHKg2)PHKCAMK2y7jBAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1897
PHKG2 (PHKg2)PHKCAMK2y7jBBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1895
PHKG2 (PHKg2)PHKCAMK2y7jCAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1896
PHKG2 (PHKg2)PHKCAMK2y7jCBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1900
PHKG2 (PHKg2)PHKCAMK2y7jDAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1898
PHKG2 (PHKg2)PHKCAMK2y7jDBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1899
PI4K2APIKAtypical4hndAadenosine-5'-diphosphateHuman9265
PI4K2APIKAtypical4hndBadenosine-5'-diphosphateHuman9261
PI4K2APIKAtypical4hneAadenosine-5'-diphosphateHuman9262
PI4K2APIKAtypical4hneBadenosine-5'-diphosphateHuman9263
PI4K2APIKAtypical4plaAadenosine-5'-triphosphateHuman9259
PI4K2APIKAtypical4yc4A[(1s,3s,4s)-3-(6-amino-9h-purin-9-yl)bicyclo[2.2.1]hept-1-yl]methanolHuman9258
PI4K2APIKAtypical5eutA-Human9264
PI4K2APIKAtypical5i0nAAadenosine-5'-triphosphateHuman9260
PI4K2APIKAtypical5i0nABadenosine-5'-triphosphateHuman9257
PI4K2BPIKAtypical4wtvAAadenosine-5'-triphosphateHuman9095
PI4K2BPIKAtypical4wtvABadenosine-5'-triphosphateHuman9098
PI4K2BPIKAtypical4wtvBAadenosine-5'-triphosphateHuman9097
PI4K2BPIKAtypical4wtvBBadenosine-5'-triphosphateHuman9096
PI4K2BPIKAtypical8a5xA4-azanyl-7-[3-(hydroxymethyl)phenyl]quinazoline-6-carboxamideHuman14384
PI4KAPIKAtypical6bq1A5-{2-amino-1-[4-(morpholin-4-yl)phenyl]-1h-benzimidazol-6-yl}-n-(2-fluorophenyl)-2-methoxypyridine-3-sulfonamideHuman9070
PI4KAPIKAtypical6bq1E5-{2-amino-1-[4-(morpholin-4-yl)phenyl]-1h-benzimidazol-6-yl}-n-(2-fluorophenyl)-2-methoxypyridine-3-sulfonamideHuman9069
PI4KBPIKAtypical4d0lAn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9152
PI4KBPIKAtypical4d0lCn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9143
PI4KBPIKAtypical4d0lEn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9139
PI4KBPIKAtypical4d0mAn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9136
PI4KBPIKAtypical4d0mcn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9148
PI4KBPIKAtypical4d0mCn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9153
PI4KBPIKAtypical4d0mgn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9146
PI4KBPIKAtypical4d0mGn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9134
PI4KBPIKAtypical4d0mIn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9151
PI4KBPIKAtypical4d0mMn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9138
PI4KBPIKAtypical4d0mOn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9154
PI4KBPIKAtypical4d0mQn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9145
PI4KBPIKAtypical4d0mSn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9142
PI4KBPIKAtypical4d0mWn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9155
PI4KBPIKAtypical4d0mYn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9133
PI4KBPIKAtypical4waeAadenosine-5'-triphosphateHuman9144
PI4KBPIKAtypical4wagA6-chloro-3-(3,4-dimethoxyphenyl)-2-methylimidazo[1,2-b]pyridazin-8-amineHuman9137
PI4KBPIKAtypical5c46E-Human9141
PI4KBPIKAtypical5c4gEn~2~-[7-(3,4-dimethoxyphenyl)quinoxalin-2-yl]-n-methylglycinamideHuman9135
PI4KBPIKAtypical5euqE~{n}-[5-[3-[[(4-hydroxyphenyl)amino]-bis(oxidanyl)-$l^{4}-sulfanyl]-4-methoxy-phenyl]-4-methyl-1,3-thiazol-2-yl]cyclopentanecarboxamideHuman9132
PI4KBPIKAtypical5fblA~{n}-[2-[[6-chloranyl-3-(4-methoxy-3-morpholin-4-ylsulfonyl-phenyl)-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9150
PI4KBPIKAtypical5fbqA~{n}-[2-[[6-chloranyl-3-[3-[4-(hydroxymethyl)piperidin-1-yl]sulfonyl-4-methoxy-phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9131
PI4KBPIKAtypical5fbrA~{n}-[2-[[3-[3-[(4-azanylcyclohexyl)sulfamoyl]-4-methoxy-phenyl]-6-chloranyl-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9140
PI4KBPIKAtypical5fbvA~{n}-[2-[[6-chloranyl-3-[3-(2-hydroxyethylsulfamoyl)-4-methoxy-phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9147
PI4KBPIKAtypical5fbwA~{n}-[2-[[6-chloranyl-3-[4-methoxy-3-[[(2~{r})-1-oxidanylbutan-2-yl]sulfamoyl]phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9149
PI4KBPIKAtypical6gl3A(3~{s})-4-(6-azanyl-1-methyl-pyrazolo[3,4-d]pyrimidin-4-yl)-~{n}-(4-methoxy-2-methyl-phenyl)-3-methyl-piperazine-1-carboxamideHuman10442
PI4KBPIKAtypical6gl3B-Human10443
PI4KBPIKAtypical8q6fAA3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidineHuman15018
PI4KBPIKAtypical8q6fAB3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidineHuman15013
PI4KBPIKAtypical8q6fAC3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidineHuman15011
PI4KBPIKAtypical8q6gAA3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15014
PI4KBPIKAtypical8q6gAB3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15012
PI4KBPIKAtypical8q6gAC3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15016
PI4KBPIKAtypical8q6hAA3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15015
PI4KBPIKAtypical8q6hAB3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15017
Pik3c2aPIPAtypical7bi2AA9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-oneMouse14153
Pik3c2aPIPAtypical7bi2AB9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-oneMouse14151
Pik3c2aPIPAtypical7bi4AA-Mouse14155
Pik3c2aPIPAtypical7bi4AB-Mouse14156
Pik3c2aPIPAtypical7bi6AAadenosine-5'-triphosphateMouse14154
Pik3c2aPIPAtypical7bi6ABadenosine-5'-triphosphateMouse14149
Pik3c2aPIPAtypical7bi9AAn-(2,3-dihydro-7,8-dimethoxyimidazo[1,2-c] quinazolin-5-yl)nicotinamideMouse14150
Pik3c2aPIPAtypical7bi9ABn-(2,3-dihydro-7,8-dimethoxyimidazo[1,2-c] quinazolin-5-yl)nicotinamideMouse14152
Pik3c2aPIPAtypical7z74AA~{n}-[4-(3-hydroxyphenyl)-1,3-thiazol-2-yl]-2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-ethanamideMouse14360
Pik3c2aPIPAtypical7z74AB~{n}-[4-(3-hydroxyphenyl)-1,3-thiazol-2-yl]-2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-ethanamideMouse14357
Pik3c2aPIPAtypical7z75A~{n}-[4-[3-(methylsulfonylamino)phenyl]-1,3-thiazol-2-yl]-2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-ethanamideMouse14359
Pik3c2aPIPAtypical8a9iAA2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-~{n}-(1,3-thiazol-2-yl)ethanamideMouse14361
Pik3c2aPIPAtypical8a9iAB2-[4-oxidanylidene-3-(2-phenylethyl)pteridin-2-yl]sulfanyl-~{n}-(1,3-thiazol-2-yl)ethanamideMouse14358
PIK3C3PIKAtypical3ihyA-Human9341
PIK3C3PIKAtypical3ihyB-Human9336
PIK3C3PIKAtypical3ihyC-Human9331
PIK3C3PIKAtypical3ihyD-Human9337
PIK3C3PIKAtypical3ihyE-Human9344
PIK3C3PIKAtypical3ls8AA-Human9340
PIK3C3PIKAtypical3ls8AB-Human9348
PIK3C3PIKAtypical3ls8BA-Human9333
PIK3C3PIKAtypical3ls8BB-Human9339
PIK3C3PIKAtypical4oysA(8s)-9-[(5-chloranylpyridin-3-yl)methyl]-2-[(3r)-3-methylmorpholin-4-yl]-8-(trifluoromethyl)-6,7,8,9a-tetrahydro-3h-pyrimido[1,2-a]pyrimidin-4-oneHuman9327
PIK3C3PIKAtypical4ph4BA-Human9326
PIK3C3PIKAtypical4ph4BB-Human9330
PIK3C3PIKAtypical4uwfA-Human9328
PIK3C3PIKAtypical4uwgAA-Human9347
PIK3C3PIKAtypical4uwgAB-Human9350
PIK3C3PIKAtypical4uwhAA-Human9346
PIK3C3PIKAtypical4uwhAB-Human9334
PIK3C3PIKAtypical4uwkAA-Human9342
PIK3C3PIKAtypical4uwkAB-Human9335
PIK3C3PIKAtypical4uwlA-Human9332
PIK3C3PIKAtypical5anlA(8s)-2-(morpholin-4-yl)-9-[2-(propan-2-yloxy)ethyl]-8-(trifluoromethyl)-6,7,8,9-tetrahydro-4h-pyrimido[1,2-a]pyrimidin-4-oneHuman9349
PIK3C3PIKAtypical5ennAA1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-olHuman9343
PIK3C3PIKAtypical5ennAB1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-olHuman9338
PIK3C3PIKAtypical5ennBA1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-olHuman9345
PIK3C3PIKAtypical5ennBB1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-olHuman9329
PIK3C3PIKAtypical6i3uA2-morpholin-4-yl-6-[7-[(2~{r})-1-morpholin-4-ylpropan-2-yl]oxy-9~{h}-thioxanthen-4-yl]pyran-4-oneHuman11292
PIK3C3PIKAtypical6ykgA4-morpholin-4-yl-6-[(2~{r})-2-(phenylmethyl)pyrrolidin-1-yl]-1~{h}-pyridin-2-oneHuman13509
PIK3C3PIKAtypical7bl1B-Human13361
PIK3C3PIKAtypical7rsjAAn-{4-[(7r,8r)-4-oxo-7-(propan-2-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]pyridin-2-yl}cyclopropanecarboxamideHuman13983
PIK3C3PIKAtypical7rsjABn-{4-[(7r,8r)-4-oxo-7-(propan-2-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]pyridin-2-yl}cyclopropanecarboxamideHuman13982
PIK3C3PIKAtypical7rspAA(7r,8r)-2-[(3r)-3-methylmorpholin-4-yl]-7-(propan-2-yl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5h)-oneHuman13981
PIK3C3PIKAtypical7rspAB(7r,8r)-2-[(3r)-3-methylmorpholin-4-yl]-7-(propan-2-yl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5h)-oneHuman13986
PIK3C3PIKAtypical7rsvAA(5as,8ar,9s)-2-[(3r)-3-methylmorpholin-4-yl]-5,5a,6,7,8,8a-hexahydro-4h-cyclopenta[e]pyrazolo[1,5-a]pyrazin-4-oneHuman13985
PIK3C3PIKAtypical7rsvAB(5as,8ar,9s)-2-[(3r)-3-methylmorpholin-4-yl]-5,5a,6,7,8,8a-hexahydro-4h-cyclopenta[e]pyrazolo[1,5-a]pyrazin-4-oneHuman13984
PIK3C3PIKAtypical8sorA-Human14803
Pik3ca (p110a)PIKAtypical4a55Apik-108Mouse9403
PIK3CA (p110a)PIKAtypical2rd0A-Human9287
PIK3CA (p110a)PIKAtypical3hhmA(1s,6br,9as,11r,11br)-9a,11b-dimethyl-1-[(methyloxy)methyl]-3,6,9-trioxo-1,6,6b,7,8,9,9a,10,11,11b-decahydro-3h-furo[4,3,2-de]indeno[4,5-h][2]benzopyran-11-yl acetateHuman9275
PIK3CA (p110a)PIKAtypical3hizA-Human9311
PIK3CA (p110a)PIKAtypical3zimA1-[4-[[2-(1h-indazol-4-yl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidin-6-yl]methyl]piperazin-1-yl]-6-methyl-hept-5-ene-1,4-dioneHuman9294
PIK3CA (p110a)PIKAtypical4jpsAA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman9317
PIK3CA (p110a)PIKAtypical4jpsAB(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman9314
PIK3CA (p110a)PIKAtypical4l1bA-Human9292
PIK3CA (p110a)PIKAtypical4l23A3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenolHuman9290
PIK3CA (p110a)PIKAtypical4l2yA3-amino-5-[4-(morpholin-4-yl)pyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl]phenolHuman9276
PIK3CA (p110a)PIKAtypical4ovuAA-Human9291
PIK3CA (p110a)PIKAtypical4ovuAB-Human9271
PIK3CA (p110a)PIKAtypical4ovvA-Human9307
PIK3CA (p110a)PIKAtypical4tuuA-Human9281
PIK3CA (p110a)PIKAtypical4tv3A2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman9278
PIK3CA (p110a)PIKAtypical4wafAAn,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamideHuman9288
PIK3CA (p110a)PIKAtypical4wafABn,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamideHuman9272
PIK3CA (p110a)PIKAtypical4yknAA3-(6-methoxypyridin-3-yl)-5-[({4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl}amino)methyl]benzoic acidHuman9283
PIK3CA (p110a)PIKAtypical4yknAB3-(6-methoxypyridin-3-yl)-5-[({4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl}amino)methyl]benzoic acidHuman9315
PIK3CA (p110a)PIKAtypical4zopAA(2s,3r)-n~1~-(8-tert-butyl-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-2-yl)-3-methylpyrrolidine-1,2-dicarboxamideHuman9298
PIK3CA (p110a)PIKAtypical4zopAB(2s,3r)-n~1~-(8-tert-butyl-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-2-yl)-3-methylpyrrolidine-1,2-dicarboxamideHuman9312
PIK3CA (p110a)PIKAtypical5dxhAmethyl {2-[4-(2-chlorophenyl)-4h-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl}carbamateHuman9310
PIK3CA (p110a)PIKAtypical5dxhDmethyl {2-[4-(2-chlorophenyl)-4h-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl}carbamateHuman9300
PIK3CA (p110a)PIKAtypical5dxtA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHuman9299
PIK3CA (p110a)PIKAtypical5fi4AA~{n}-[6-[5-azanyl-6-[(2~{s})-1,1,1-tris(fluoranyl)propan-2-yl]oxy-pyrazin-2-yl]imidazo[1,2-a]pyridin-2-yl]ethanamideHuman9302
PIK3CA (p110a)PIKAtypical5fi4AB~{n}-[6-[5-azanyl-6-[(2~{s})-1,1,1-tris(fluoranyl)propan-2-yl]oxy-pyrazin-2-yl]imidazo[1,2-a]pyridin-2-yl]ethanamideHuman9309
PIK3CA (p110a)PIKAtypical5itdA5-{4-[3-(4-acetylpiperazine-1-carbonyl)phenyl]quinazolin-6-yl}-2-methoxypyridine-3-carbonitrileHuman9313
PIK3CA (p110a)PIKAtypical5sw8A-Human9274
PIK3CA (p110a)PIKAtypical5swgA-Human9306
PIK3CA (p110a)PIKAtypical5swoA-Human9303
PIK3CA (p110a)PIKAtypical5swpA-Human9293
PIK3CA (p110a)PIKAtypical5swrA-Human9279
PIK3CA (p110a)PIKAtypical5swtA-Human9273
PIK3CA (p110a)PIKAtypical5sx8A-Human9269
PIK3CA (p110a)PIKAtypical5sx9A-Human9305
PIK3CA (p110a)PIKAtypical5sxaA-Human9285
PIK3CA (p110a)PIKAtypical5sxbA-Human9282
PIK3CA (p110a)PIKAtypical5sxcA-Human9297
PIK3CA (p110a)PIKAtypical5sxdA-Human9304
PIK3CA (p110a)PIKAtypical5sxeA-Human9280
PIK3CA (p110a)PIKAtypical5sxfA-Human9284
PIK3CA (p110a)PIKAtypical5sxiA-Human9270
PIK3CA (p110a)PIKAtypical5sxjA-Human9301
PIK3CA (p110a)PIKAtypical5sxkA-Human9296
PIK3CA (p110a)PIKAtypical5ubrA1-[4-(3-{4-amino-5-[1-(oxan-4-yl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)piperazin-1-yl]ethan-1-oneHuman9289
PIK3CA (p110a)PIKAtypical5uk8AA(r)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1h-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholineHuman9295
PIK3CA (p110a)PIKAtypical5uk8AB(r)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1h-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholineHuman9286
PIK3CA (p110a)PIKAtypical5ukjAn,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamideHuman9277
PIK3CA (p110a)PIKAtypical5ul1AA3-amino-6-(4-{[(2s)-1-(dimethylamino)propan-2-yl]sulfonyl}phenyl)-n-phenylpyrazine-2-carboxamideHuman9316
PIK3CA (p110a)PIKAtypical5ul1AB3-amino-6-(4-{[(2s)-1-(dimethylamino)propan-2-yl]sulfonyl}phenyl)-n-phenylpyrazine-2-carboxamideHuman9308
PIK3CA (p110a)PIKAtypical5xghA3-[(4-fluorophenyl)methylamino]-5-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenolHuman9864
PIK3CA (p110a)PIKAtypical5xgiA3-azanyl-5-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenolHuman9865
PIK3CA (p110a)PIKAtypical5xgjA3-(4-morpholin-4-ylfuro[3,2-d]pyrimidin-2-yl)-5-[(phenylmethyl)amino]phenolHuman9863
PIK3CA (p110a)PIKAtypical6gvfAA5-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11659
PIK3CA (p110a)PIKAtypical6gvfAB5-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11658
PIK3CA (p110a)PIKAtypical6gvgA5-(6-azanyl-4-methyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11655
PIK3CA (p110a)PIKAtypical6gvhAA5-(6-azanyl-4-chloranyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11657
PIK3CA (p110a)PIKAtypical6gvhAB5-(6-azanyl-4-chloranyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11653
PIK3CA (p110a)PIKAtypical6gviAA3-(2-azanyl-1,3-benzoxazol-5-yl)-1-propan-2-yl-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman11656
PIK3CA (p110a)PIKAtypical6gviAB3-(2-azanyl-1,3-benzoxazol-5-yl)-1-propan-2-yl-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman11654
PIK3CA (p110a)PIKAtypical6nctA-Human11221
PIK3CA (p110a)PIKAtypical6oacA4-(difluoromethyl)-5-{4-[(3s)-3-methylmorpholin-4-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}pyridin-2-amineHuman11381
PIK3CA (p110a)PIKAtypical6pysAA(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11575
PIK3CA (p110a)PIKAtypical6pysAB(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11576
PIK3CA (p110a)PIKAtypical7jiuAA(3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-oneHuman13760
PIK3CA (p110a)PIKAtypical7jiuAB(3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-oneHuman13761
PIK3CA (p110a)PIKAtypical7k6mAA2,2-difluoroethyl (3s)-3-{[2'-amino-5-fluoro-2-(morpholin-4-yl)[4,5'-bipyrimidin]-6-yl]amino}-3-(hydroxymethyl)pyrrolidine-1-carboxylateHuman13225
PIK3CA (p110a)PIKAtypical7k6mAB2,2-difluoroethyl (3s)-3-{[2'-amino-5-fluoro-2-(morpholin-4-yl)[4,5'-bipyrimidin]-6-yl]amino}-3-(hydroxymethyl)pyrrolidine-1-carboxylateHuman13227
PIK3CA (p110a)PIKAtypical7k6nAAtert-butyl (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-3-methylpyrrolidine-1-carboxylateHuman13226
PIK3CA (p110a)PIKAtypical7k6nABtert-butyl (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-3-methylpyrrolidine-1-carboxylateHuman13224
PIK3CA (p110a)PIKAtypical7k6oAA(3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-n-methylpyrrolidine-1-sulfonamideHuman13207
PIK3CA (p110a)PIKAtypical7k6oAB(3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-n-methylpyrrolidine-1-sulfonamideHuman13206
PIK3CA (p110a)PIKAtypical7k71A2-(morpholin-4-yl)[4,5'-bipyrimidin]-2'-amineHuman13219
PIK3CA (p110a)PIKAtypical7mlkAA4-[6-(3,4,5-trimethoxyanilino)pyrazin-2-yl]benzamideHuman14216
PIK3CA (p110a)PIKAtypical7mlkAB4-[6-(3,4,5-trimethoxyanilino)pyrazin-2-yl]benzamideHuman14217
PIK3CA (p110a)PIKAtypical7mynAA-Human13963
PIK3CA (p110a)PIKAtypical7mynAB-Human13964
PIK3CA (p110a)PIKAtypical7myoBA-Human13962
PIK3CA (p110a)PIKAtypical7myoBB-Human13965
PIK3CA (p110a)PIKAtypical7pg5AA-Human14346
PIK3CA (p110a)PIKAtypical7pg5AB-Human14347
PIK3CA (p110a)PIKAtypical7pg6AA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14348
PIK3CA (p110a)PIKAtypical7pg6AB(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14349
PIK3CA (p110a)PIKAtypical7r9vAn-[2-(4-{4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethyl]-1-(prop-2-enoyl)piperidine-4-carboxamideHuman14178
PIK3CA (p110a)PIKAtypical7r9yAn-[2-(4-{4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethyl]-n-methyl-1-(prop-2-enoyl)piperidine-4-carboxamideHuman14179
PIK3CA (p110a)PIKAtypical7tz7AA(4s,5r)-3-[2'-amino-2-(morpholin-4-yl)-4'-(trifluoromethyl)[4,5'-bipyrimidin]-6-yl]-4-(hydroxymethyl)-5-methyl-1,3-oxazolidin-2-oneHuman14223
PIK3CA (p110a)PIKAtypical7tz7AB(4s,5r)-3-[2'-amino-2-(morpholin-4-yl)-4'-(trifluoromethyl)[4,5'-bipyrimidin]-6-yl]-4-(hydroxymethyl)-5-methyl-1,3-oxazolidin-2-oneHuman14222
PIK3CA (p110a)PIKAtypical8am0A(2r)-2-[[2-[(4s)-4-[bis(fluoranyl)methyl]-2-oxidanylidene-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl]amino]propanamideHuman15083
PIK3CA (p110a)PIKAtypical8bfuA-Human14613
PIK3CA (p110a)PIKAtypical8dcpAA-Human14380
PIK3CA (p110a)PIKAtypical8dcpAB-Human14376
PIK3CA (p110a)PIKAtypical8dcxA-Human14377
PIK3CA (p110a)PIKAtypical8dd4AA-Human14378
PIK3CA (p110a)PIKAtypical8dd4AB-Human14379
PIK3CA (p110a)PIKAtypical8dd8A-Human14375
PIK3CA (p110a)PIKAtypical8exlAA2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamideHuman14537
PIK3CA (p110a)PIKAtypical8exlAB2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamideHuman14536
PIK3CA (p110a)PIKAtypical8exoAA1-{(4s,11am)-2-[(4r)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-prolinamideHuman14541
PIK3CA (p110a)PIKAtypical8exoAB1-{(4s,11am)-2-[(4r)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-prolinamideHuman14534
PIK3CA (p110a)PIKAtypical8exuAA(2s)-2-cyclopropyl-2-({(4s,11am)-2-[(4s)-2-oxo-4-(trifluoromethyl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}amino)acetamideHuman14539
PIK3CA (p110a)PIKAtypical8exuAB(2s)-2-cyclopropyl-2-({(4s,11am)-2-[(4s)-2-oxo-4-(trifluoromethyl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}amino)acetamideHuman14544
PIK3CA (p110a)PIKAtypical8exvAAn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14542
PIK3CA (p110a)PIKAtypical8exvABn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14538
PIK3CA (p110a)PIKAtypical8guaA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14540
PIK3CA (p110a)PIKAtypical8gubA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14543
PIK3CA (p110a)PIKAtypical8gudAA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14535
PIK3CA (p110a)PIKAtypical8ilrABn-[(2s)-1-(ethylamino)-1-oxidanylidene-3-[4-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamideHuman14973
PIK3CA (p110a)PIKAtypical8ilsABn-[(2r)-1-(ethylamino)-1-oxidanylidene-3-[4-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamideHuman14968
PIK3CA (p110a)PIKAtypical8ilvAn-[(2r)-1-(ethylamino)-1-oxidanylidene-3-[3-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamideHuman14974
PIK3CA (p110a)PIKAtypical8ow2AA-Human14765
PIK3CA (p110a)PIKAtypical8ow2AB-Human14764
PIK3CA (p110a)PIKAtypical8sbcAA(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(pyridin-2-yl)-1h-imidazo[4,5-b]pyridineHuman14841
PIK3CA (p110a)PIKAtypical8sbcAB(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(pyridin-2-yl)-1h-imidazo[4,5-b]pyridineHuman14842
PIK3CA (p110a)PIKAtypical8sbjAA(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(1h-pyrazol-3-yl)-3h-imidazo[4,5-b]pyridineHuman14839
PIK3CA (p110a)PIKAtypical8sbjAB(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(1h-pyrazol-3-yl)-3h-imidazo[4,5-b]pyridineHuman14840
PIK3CA (p110a)PIKAtypical8tduAAn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14967
PIK3CA (p110a)PIKAtypical8tduABn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14969
PIK3CA (p110a)PIKAtypical8tgdAAn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14972
PIK3CA (p110a)PIKAtypical8tgdABn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14970
PIK3CA (p110a)PIKAtypical8ts7A-Human15088
PIK3CA (p110a)PIKAtypical8ts8A-Human15086
PIK3CA (p110a)PIKAtypical8ts9A-Human15089
PIK3CA (p110a)PIKAtypical8tsaA-Human15087
PIK3CA (p110a)PIKAtypical8tsbA-Human15085
PIK3CA (p110a)PIKAtypical8tscA-Human15084
PIK3CA (p110a)PIKAtypical8tsdA-Human15090
PIK3CA (p110a)PIKAtypical8tu6A-Human14971
Pik3cb (p110b)PIKAtypical2y3aA2-(1h-indazol-4-yl)-6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-yl-thieno[3,2-d]pyrimidineMouse9402
Pik3cb (p110b)PIKAtypical4bfrA2-[2-(2-methyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-6-morpholin-4-yl-3h-pyrimidin-4-oneMouse9400
Pik3cb (p110b)PIKAtypical4bfrB2-[2-(2-methyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-6-morpholin-4-yl-3h-pyrimidin-4-oneMouse9401
Pik3cd (p110d)PIKAtypical2wxfAA2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-oneMouse9355
Pik3cd (p110d)PIKAtypical2wxfAB2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-oneMouse9352
Pik3cd (p110d)PIKAtypical2wxgA2-{[4-amino-3-(3-fluoro-5-hydroxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-oneMouse9395
Pik3cd (p110d)PIKAtypical2wxhA2-{[4-amino-3-(3-fluoro-4-hydroxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-oneMouse9387
Pik3cd (p110d)PIKAtypical2wxiA2-{[4-amino-3-(3-hydroxyprop-1-yn-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-oneMouse9373
Pik3cd (p110d)PIKAtypical2wxjAn-[6-(4-amino-1-{[2-(4-methylpiperazin-1-yl)quinolin-3-yl]methyl}-1h-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzothiazol-2-yl]acetamideMouse9375
Pik3cd (p110d)PIKAtypical2wxkA3-(2-amino-1,3-benzothiazol-6-yl)-1-{[2-(4-methylpiperazin-1-yl)quinolin-3-yl]methyl}-1h-pyrazolo[3,4-d]pyrimidin-4-amineMouse9382
Pik3cd (p110d)PIKAtypical2wxlAA2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-1h-benzimidazoleMouse9376
Pik3cd (p110d)PIKAtypical2wxlAB2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-1h-benzimidazoleMouse9389
Pik3cd (p110d)PIKAtypical2wxmA1-(1-methylethyl)-3-(pyridin-3-ylethynyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineMouse9359
Pik3cd (p110d)PIKAtypical2wxnA3-{[4-amino-1-(1-methylethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]ethynyl}phenolMouse9365
Pik3cd (p110d)PIKAtypical2wxoAAn-(3-{[(1z)-3,5-dimethoxycyclohexa-2,4-dien-1-ylidene]amino}quinoxalin-2-yl)-4-fluorobenzenesulfonamideMouse9381
Pik3cd (p110d)PIKAtypical2wxoABn-(3-{[(1z)-3,5-dimethoxycyclohexa-2,4-dien-1-ylidene]amino}quinoxalin-2-yl)-4-fluorobenzenesulfonamideMouse9361
Pik3cd (p110d)PIKAtypical2wxpA2-(1h-indazol-4-yl)-6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-yl-thieno[3,2-d]pyrimidineMouse9366
Pik3cd (p110d)PIKAtypical2wxqA2-{[3-(2-methoxyphenyl)-4-oxo-3,4,5,6,7,8-hexahydroquinazolin-2-yl]sulfanyl}-n-quinoxalin-6-ylacetamideMouse9393
Pik3cd (p110d)PIKAtypical2wxrA-Mouse9385
Pik3cd (p110d)PIKAtypical2x38AA2-[(6-amino-9h-purin-9-yl)methyl]-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-oneMouse9369
Pik3cd (p110d)PIKAtypical2x38AB2-[(6-amino-9h-purin-9-yl)methyl]-5-methyl-3-(2-methylphenyl)quinazolin-4(3h)-oneMouse9380
Pik3cd (p110d)PIKAtypical4ajwA2-[(1-methyl-1h-benzimidazol-2-yl)methyl]-6-morpholin-4-ylpyrimidin-4(3h)-oneMouse9364
Pik3cd (p110d)PIKAtypical4ajwB2-[(1-methyl-1h-benzimidazol-2-yl)methyl]-6-morpholin-4-ylpyrimidin-4(3h)-oneMouse9360
Pik3cd (p110d)PIKAtypical4v0iA2-[2-(2-methyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-6-morpholin-4-yl-3h-pyrimidin-4-oneMouse9399
Pik3cd (p110d)PIKAtypical4v0iB2-[2-(2-methyl-2,3-dihydro-indol-1-yl)-2-oxo-ethyl]-6-morpholin-4-yl-3h-pyrimidin-4-oneMouse9384
Pik3cd (p110d)PIKAtypical4xe0A5-fluoro-3-phenyl-2-[(1s)-1-(7h-purin-6-ylamino)propyl]quinazolin-4(3h)-oneMouse9368
Pik3cd (p110d)PIKAtypical5ae8A6-(1h-indol-4-yl)-4-(5-{[4-(1-methylethyl)-1-piperazinyl]methyl}-1,3-oxazol-2-yl)-1h-indazoleMouse9390
Pik3cd (p110d)PIKAtypical5ae9An-[5-[4-(5-{[(2r,6s)-2,6-dimethyl-4-morpholinyl]methyl}-1,3-oxazol-2-yl)-1h-indazol-6-yl]-2-(methyloxy)-3-pyridinyl]methanesulfonamideMouse9372
Pik3cd (p110d)PIKAtypical5i4uA2,4-diamino-6-{[(1s)-1-(5-chloro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)ethyl]amino}pyrimidine-5-carbonitrileMouse9391
Pik3cd (p110d)PIKAtypical5i6uA2-[(1s)-1-({6-amino-5-[(1h-pyrazol-4-yl)ethynyl]pyrimidin-4-yl}amino)ethyl]-5-chloro-3-phenylquinazolin-4(3h)-oneMouse9370
Pik3cd (p110d)PIKAtypical5is5A5-{4-[3-(4-acetylpiperazine-1-carbonyl)phenyl]quinazolin-6-yl}-2-methoxypyridine-3-carbonitrileMouse9356
Pik3cd (p110d)PIKAtypical5l72An-[6-(5-methanesulfonamido-6-methoxypyridin-3-yl)-1,3-dihydro-2-benzofuran-4-yl]-2-(morpholin-4-yl)acetamideMouse9386
Pik3cd (p110d)PIKAtypical5ncyAA4-azanyl-6-[[(1~{s})-1-(3-methyl-5-oxidanylidene-6-phenyl-[1,3]thiazolo[3,2-a]pyridin-7-yl)ethyl]amino]pyrimidine-5-carbonitrileMouse9379
Pik3cd (p110d)PIKAtypical5ncyAB4-azanyl-6-[[(1~{s})-1-(3-methyl-5-oxidanylidene-6-phenyl-[1,3]thiazolo[3,2-a]pyridin-7-yl)ethyl]amino]pyrimidine-5-carbonitrileMouse9357
Pik3cd (p110d)PIKAtypical5nczAA4-azanyl-6-[[(1~{s})-1-[6-[3-[(dimethylamino)methyl]phenyl]-3-methyl-5-oxidanylidene-[1,3]thiazolo[3,2-a]pyridin-7-yl]ethyl]amino]pyrimidine-5-carbonitrileMouse9396
Pik3cd (p110d)PIKAtypical5nczAB4-azanyl-6-[[(1~{s})-1-[6-[3-[(dimethylamino)methyl]phenyl]-3-methyl-5-oxidanylidene-[1,3]thiazolo[3,2-a]pyridin-7-yl]ethyl]amino]pyrimidine-5-carbonitrileMouse9388
Pik3cd (p110d)PIKAtypical5ngbA3-[[4-(2-morpholin-4-yl-4-oxidanylidene-3~{h}-quinolin-8-yl)-1,2,3-triazol-1-yl]methyl]benzoic acidMouse9353
Pik3cd (p110d)PIKAtypical5o83AleniolisibMouse9351
Pik3cd (p110d)PIKAtypical5t27A3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{s})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amineMouse9383
Pik3cd (p110d)PIKAtypical5t28A3-(benzotriazol-1-yl)-5-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-amineMouse9398
Pik3cd (p110d)PIKAtypical5t2bA5-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]-3-(1~{h}-pyrazol-4-yl)pyrazin-2-amineMouse9374
Pik3cd (p110d)PIKAtypical5t2dA4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]-~{n},~{n}-dimethyl-pyrazole-1-sulfonamideMouse9397
Pik3cd (p110d)PIKAtypical5t2gA4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-1-carboxamideMouse9363
Pik3cd (p110d)PIKAtypical5t2iAA1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-4-carboxamideMouse9358
Pik3cd (p110d)PIKAtypical5t2iAB1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-4-carboxamideMouse9367
Pik3cd (p110d)PIKAtypical5t2lAA1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-3-carboxamideMouse9378
Pik3cd (p110d)PIKAtypical5t2lAB1-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-3-carboxamideMouse9394
Pik3cd (p110d)PIKAtypical5t2mA4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]benzamideMouse9371
Pik3cd (p110d)PIKAtypical5t7fA2,4-bis(azanyl)-6-[[(1~{s})-1-[5-chloranyl-3-(5-fluoranyl-4-methyl-pyridin-3-yl)-4-oxidanylidene-quinazolin-2-yl]ethyl]amino]pyrimidine-5-carbonitrileMouse9362
Pik3cd (p110d)PIKAtypical5t7fB2,4-bis(azanyl)-6-[[(1~{s})-1-[5-chloranyl-3-(5-fluoranyl-4-methyl-pyridin-3-yl)-4-oxidanylidene-quinazolin-2-yl]ethyl]amino]pyrimidine-5-carbonitrileMouse9354
Pik3cd (p110d)PIKAtypical5t8iAA2,4-diamino-6-{[(s)-[5-chloro-8-fluoro-4-oxo-3-(pyridin-3-yl)-3,4-dihydroquinazolin-2-yl](cyclopropyl)methyl]amino}pyrimidine-5-carbonitrileMouse9392
Pik3cd (p110d)PIKAtypical5t8iAB2,4-diamino-6-{[(s)-[5-chloro-8-fluoro-4-oxo-3-(pyridin-3-yl)-3,4-dihydroquinazolin-2-yl](cyclopropyl)methyl]amino}pyrimidine-5-carbonitrileMouse9377
Pik3cd (p110d)PIKAtypical6dgtA4-[1-(5,8-difluoroquinolin-4-yl)-2-methyl-4-(4h-1,2,4-triazol-3-yl)-1h-benzimidazol-6-yl]-3-fluoropyridin-2-amineMouse10603
Pik3cd (p110d)PIKAtypical6eyzA2-methoxy-5-[4-[5-[(4-propan-2-ylpiperazin-1-yl)methyl]-1,3-oxazol-2-yl]-2~{h}-indazol-6-yl]pyridine-3-carboxylic acidMouse9426
Pik3cd (p110d)PIKAtypical6ez6Amethyl 2-methoxy-5-[4-[5-[(4-propan-2-ylpiperazin-1-yl)methyl]-1,3-oxazol-2-yl]-2~{h}-indazol-6-yl]pyridine-3-carboxylateMouse9460
Pik3cd (p110d)PIKAtypical6ftnAA~{n}-[5-[2-[(1~{s})-1-cyclopropylethyl]-7-methyl-1-oxidanylidene-3~{h}-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamideMouse10010
Pik3cd (p110d)PIKAtypical6ftnAB~{n}-[5-[2-[(1~{s})-1-cyclopropylethyl]-7-methyl-1-oxidanylidene-3~{h}-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamideMouse10011
Pik3cd (p110d)PIKAtypical6gy0A~{n}-[4-methyl-5-(1-oxidanylidene-7-sulfamoyl-isoindol-5-yl)-1,3-thiazol-2-yl]ethanamideMouse11298
Pik3cd (p110d)PIKAtypical6hi1A3-(6-morpholin-4-ylpyridin-2-yl)phenolMouse11624
Pik3cd (p110d)PIKAtypical6hi2A3-[6-[(1~{s},6~{r})-3-oxabicyclo[4.1.0]heptan-6-yl]pyridin-2-yl]phenolMouse11623
Pik3cd (p110d)PIKAtypical6hi9AA3-[6-(oxan-4-yl)pyridin-2-yl]phenolMouse11625
Pik3cd (p110d)PIKAtypical6hi9AB3-[6-(oxan-4-yl)pyridin-2-yl]phenolMouse11622
Pik3cd (p110d)PIKAtypical6mulAA1-{1-[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]piperidin-4-yl}-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-oneMouse11300
Pik3cd (p110d)PIKAtypical6mulAB1-{1-[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]piperidin-4-yl}-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-oneMouse11297
Pik3cd (p110d)PIKAtypical6mulBA1-{1-[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]piperidin-4-yl}-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-oneMouse11301
Pik3cd (p110d)PIKAtypical6mulBB1-{1-[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]piperidin-4-yl}-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-oneMouse11293
Pik3cd (p110d)PIKAtypical6mumAA[(3s)-3-{[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]oxy}pyrrolidin-1-yl](oxan-4-yl)methanoneMouse11294
Pik3cd (p110d)PIKAtypical6mumAB[(3s)-3-{[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]oxy}pyrrolidin-1-yl](oxan-4-yl)methanoneMouse11296
Pik3cd (p110d)PIKAtypical6mumBA[(3s)-3-{[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]oxy}pyrrolidin-1-yl](oxan-4-yl)methanoneMouse11299
Pik3cd (p110d)PIKAtypical6mumBB[(3s)-3-{[8-(1-ethyl-5-methyl-1h-pyrazol-4-yl)-9-methyl-9h-purin-6-yl]oxy}pyrrolidin-1-yl](oxan-4-yl)methanoneMouse11295
Pik3cd (p110d)PIKAtypical6q6yA~{n}-(2-chloranyl-5-phenyl-pyridin-3-yl)benzenesulfonamideMouse10826
Pik3cd (p110d)PIKAtypical6q73A~{n}-[2-chloranyl-5-(3,6-dihydro-2~{h}-pyran-4-yl)pyridin-3-yl]methanesulfonamideMouse10825
Pik3cd (p110d)PIKAtypical6q74A~{n}-[5-(3,6-dihydro-2~{h}-pyran-4-yl)-2-methoxy-pyridin-3-yl]-2-methyl-1-(phenylmethyl)imidazole-4-sulfonamideMouse10824
Pik3cd (p110d)PIKAtypical6tnrAA~{n}-[2-methoxy-5-[7-[2-[4-(2-oxidanylpropan-2-yl)piperidin-1-yl]ethoxy]-1,3-dihydro-2-benzofuran-5-yl]pyridin-3-yl]methanesulfonamideMouse11911
Pik3cd (p110d)PIKAtypical6tnrAB~{n}-[2-methoxy-5-[7-[2-[4-(2-oxidanylpropan-2-yl)piperidin-1-yl]ethoxy]-1,3-dihydro-2-benzofuran-5-yl]pyridin-3-yl]methanesulfonamideMouse11910
Pik3cd (p110d)PIKAtypical6tnsA2-methoxy-~{n}-[2-methoxy-5-[7-[[(2~{r})-4-(oxetan-3-yl)morpholin-2-yl]methoxy]-1,3-dihydro-2-benzofuran-5-yl]pyridin-3-yl]ethanesulfonamideMouse11909
Pik3cd (p110d)PIKAtypical6zaaA4-[6-methoxy-5-(methylsulfamoyl)pyridin-3-yl]-~{n}-(1-methylpiperidin-4-yl)-2,3-dihydro-1,4-benzoxazine-6-carboxamideMouse12635
Pik3cd (p110d)PIKAtypical6zacAA~{n}-[5-[6-[(dimethylamino)methyl]-2,3-dihydro-1,4-benzoxazin-4-yl]-2-methoxy-pyridin-3-yl]methanesulfonamideMouse12633
Pik3cd (p110d)PIKAtypical6zacAB~{n}-[5-[6-[(dimethylamino)methyl]-2,3-dihydro-1,4-benzoxazin-4-yl]-2-methoxy-pyridin-3-yl]methanesulfonamideMouse12634
Pik3cd (p110d)PIKAtypical6zadAmethoxymethyloxathiatetraazatetracyclodocosahexaenedioneMouse12653
Pik3cd (p110d)PIKAtypical7oi4AAn-[5-[2-[(1s)-1-cyclopropylethyl]-7-[[4-[(dimethylamino)methyl]phenyl]sulfamoyl]-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamideMouse13800
Pik3cd (p110d)PIKAtypical7oi4ABn-[5-[2-[(1s)-1-cyclopropylethyl]-7-[[4-[(dimethylamino)methyl]phenyl]sulfamoyl]-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamideMouse13805
Pik3cd (p110d)PIKAtypical7oijAA6-[[5-[2-[(1s)-1-cyclopropylethyl]-7-(methylsulfamoyl)-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]amino]-n-[3-(dimethylamino)propyl]pyridine-2-carboxamideMouse13801
Pik3cd (p110d)PIKAtypical7oijAB6-[[5-[2-[(1s)-1-cyclopropylethyl]-7-(methylsulfamoyl)-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]amino]-n-[3-(dimethylamino)propyl]pyridine-2-carboxamideMouse13807
Pik3cd (p110d)PIKAtypical7oilAA2-[(1s)-1-cyclopropylethyl]-5-[4-methyl-2-[[6-(2-oxidanylidenepyrrolidin-1-yl)pyridin-2-yl]amino]-1,3-thiazol-5-yl]-7-methylsulfonyl-3h-isoindol-1-oneMouse13804
Pik3cd (p110d)PIKAtypical7oilAB2-[(1s)-1-cyclopropylethyl]-5-[4-methyl-2-[[6-(2-oxidanylidenepyrrolidin-1-yl)pyridin-2-yl]amino]-1,3-thiazol-5-yl]-7-methylsulfonyl-3h-isoindol-1-oneMouse13806
Pik3cd (p110d)PIKAtypical7oisAAn-[5-[2-[(1s)-1-cyclopropylethyl]-7-[(3-methylsulfonylphenyl)sulfamoyl]-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamideMouse13803
Pik3cd (p110d)PIKAtypical7oisABn-[5-[2-[(1s)-1-cyclopropylethyl]-7-[(3-methylsulfonylphenyl)sulfamoyl]-1-oxidanylidene-3h-isoindol-5-yl]-4-methyl-1,3-thiazol-2-yl]ethanamideMouse13802
Pik3cd (p110d)PIKAtypical7popA5-[3,6-dihydro-2h-pyran-4-yl]-2-methoxy-n-[2-methylpyridin-4-yl]pyridine-3-sulfonamideMouse13917
Pik3cd (p110d)PIKAtypical7porA~{n}-[2-[2-fluoranyl-4-[(4-propan-2-ylpiperazin-1-yl)methyl]phenyl]pyridin-4-yl]-2-methoxy-5-morpholin-4-yl-pyridine-3-sulfonamideMouse13915
Pik3cd (p110d)PIKAtypical7posA5-(3,6-dihydro-2~{h}-pyran-4-yl)-2-methoxy-~{n}-[5-[3-(4-propan-2-ylpiperazin-1-yl)prop-1-ynyl]pyridin-3-yl]pyridine-3-sulfonamideMouse13918
Pik3cd (p110d)PIKAtypical7potAn-[5-(3,6-dihydro-2h-pyran-4-yl)-2-methoxy-pyridin-3-yl]benzenesulfonamideMouse13916
Pik3cd (p110d)PIKAtypical7r26A5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amineMouse14231
Pik3cd (p110d)PIKAtypical7r2bA(4~{s})-3-[6-[2-azanyl-4-(trifluoromethyl)pyrimidin-5-yl]-2-morpholin-4-yl-pyrimidin-4-yl]-4-methyl-1,3-oxazolidin-2-oneMouse14230
PIK3CD (p110d)PIKAtypical5dxuA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHuman9091
PIK3CD (p110d)PIKAtypical5m6uA4-azanyl-6-[[(1~{s})-1-(4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]pyrimidine-5-carbonitrileHuman9094
PIK3CD (p110d)PIKAtypical5t8fA2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamideHuman9093
PIK3CD (p110d)PIKAtypical5ubtA1-[4-(3-{4-amino-5-[1-(oxan-4-yl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)piperazin-1-yl]ethan-1-oneHuman9092
PIK3CD (p110d)PIKAtypical5vlrA4-acetyl-1-(3-{4-amino-5-[1-(2,2,2-trifluoroethyl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)-3,3-dimethylpiperazin-2-oneHuman9090
PIK3CD (p110d)PIKAtypical6g6wAA~{n}-[3-[4-[[(1~{s})-1-(5-methyl-4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-5-oxidanyl-phenyl]methanesulfonamideHuman10673
PIK3CD (p110d)PIKAtypical6g6wAB~{n}-[3-[4-[[(1~{s})-1-(5-methyl-4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-5-oxidanyl-phenyl]methanesulfonamideHuman10674
PIK3CD (p110d)PIKAtypical6ocoA4-[(1s,4s)-5-(3-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carbonitrileHuman11865
PIK3CD (p110d)PIKAtypical6ocuA5-{(3r)-3-methyl-4-[(1r,2r)-2-methylcyclopropane-1-carbonyl]piperazin-1-yl}-3-(1-methyl-1h-pyrazol-4-yl)pyrazine-2-carbonitrileHuman11864
PIK3CD (p110d)PIKAtypical6pyrAA(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11547
PIK3CD (p110d)PIKAtypical6pyrAB(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11546
PIK3CD (p110d)PIKAtypical6pyuA(3s)-1'-(cyclopropanecarbonyl)-5-(quinoxalin-6-yl)spiro[indole-3,2'-pyrrolidin]-2(1h)-oneHuman11548
PIK3CD (p110d)PIKAtypical7jisA(3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-oneHuman13201
PIK3CD (p110d)PIKAtypical7lm2Acyclopropyl[(3s)-3-{[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]amino}pyrrolidin-1-yl]methanoneHuman13532
PIK3CD (p110d)PIKAtypical7lq1An-(5-(6-(2-((2s,6r)-2,6-dimethylmorpholino)pyridin-4-yl)-1-oxoisoindolin-4-yl)-2-methoxypyridin-3-yl)methanesulfonamideHuman14106
PIK3CD (p110d)PIKAtypical8bcyAA9-[2-(3,4-dichlorophenyl)ethyl]-2-(3-hydroxyphenyl)-8-oxidanylidene-7~{h}-purine-6-carboxamideHuman14735
PIK3CD (p110d)PIKAtypical8bcyAB9-[2-(3,4-dichlorophenyl)ethyl]-2-(3-hydroxyphenyl)-8-oxidanylidene-7~{h}-purine-6-carboxamideHuman14734
PIK3CG (p110g)PIKAtypical1e8yA-Human9248
PIK3CG (p110g)PIKAtypical1e8zAstaurosporineHuman9228
PIK3CG (p110g)PIKAtypical1he8A-Human9201
PIK3CG (p110g)PIKAtypical2a4zA(5e)-5-[(2,2-difluoro-1,3-benzodioxol-5-yl)methylene]-1,3-thiazolidine-2,4-dioneHuman9180
PIK3CG (p110g)PIKAtypical2a5uA(5e)-5-(quinoxalin-6-ylmethylene)-1,3-thiazolidine-2,4-dioneHuman9183
PIK3CG (p110g)PIKAtypical2chwA2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-oneHuman9182
PIK3CG (p110g)PIKAtypical2chxAn-(2,3-dihydro-7,8-dimethoxyimidazo[1,2-c] quinazolin-5-yl)nicotinamideHuman9247
PIK3CG (p110g)PIKAtypical2chzAn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9251
PIK3CG (p110g)PIKAtypical2v4lA3-[4-amino-1-(1-methylethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]phenolHuman9237
PIK3CG (p110g)PIKAtypical3apcA5-(7-methanesulfonyl-2-morpholin-4-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamineHuman9231
PIK3CG (p110g)PIKAtypical3apdA5-(2-morpholin-4-yl-7-pyridin-3-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamineHuman9205
PIK3CG (p110g)PIKAtypical3apfA3-[7-(1h-benzimidazol-5-yl)-2-(morpholin-4-yl)-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl]phenolHuman9250
PIK3CG (p110g)PIKAtypical3csfA-Human9215
PIK3CG (p110g)PIKAtypical3cstAmethylated ruthenium pyridocarbazoleHuman9220
PIK3CG (p110g)PIKAtypical3dbsA2-(1h-indazol-4-yl)-6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-yl-thieno[3,2-d]pyrimidineHuman9230
PIK3CG (p110g)PIKAtypical3dpdA5,5-dimethyl-2-morpholin-4-yl-5,6-dihydro-1,3-benzothiazol-7(4h)-oneHuman9159
PIK3CG (p110g)PIKAtypical3eneA1-methyl-3-naphthalen-2-yl-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9188
PIK3CG (p110g)PIKAtypical3ibeA1-(4-{4-morpholin-4-yl-1-[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-6-yl}phenyl)-3-pyridin-4-ylureaHuman9171
PIK3CG (p110g)PIKAtypical3l08AA2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamideHuman9217
PIK3CG (p110g)PIKAtypical3l08AB2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamideHuman9164
PIK3CG (p110g)PIKAtypical3l13A[3-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenyl]methanolHuman9167
PIK3CG (p110g)PIKAtypical3l16A5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyridin-2-amineHuman9233
PIK3CG (p110g)PIKAtypical3l17A4-methyl-5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyrimidin-2-amineHuman9185
PIK3CG (p110g)PIKAtypical3l54A6-(1h-pyrazolo[3,4-b]pyridin-5-yl)-4-pyridin-4-ylquinolineHuman9197
PIK3CG (p110g)PIKAtypical3lj3A(2z)-4,6-dihydroxy-2-{[1-methyl-4-(4-methylpiperazin-1-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methylidene}-1-benzofuran-3(2h)-oneHuman9214
PIK3CG (p110g)PIKAtypical3mjwA(2z)-4,6-dihydroxy-2-[(8-methoxy-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)methylidene]-1-benzofuran-3(2h)-oneHuman9229
PIK3CG (p110g)PIKAtypical3ml8A8-cyclopentyl-6-[3-(hydroxymethyl)phenyl]-4-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman9192
PIK3CG (p110g)PIKAtypical3ml9A2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman9187
PIK3CG (p110g)PIKAtypical3nzsA6-(1,1-dioxidothiomorpholin-4-yl)-n-(3-methoxyphenyl)-1-methyl-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9179
PIK3CG (p110g)PIKAtypical3nzuA6-(2h-indazol-4-yl)-1-methyl-n-[3-(methylsulfonyl)propyl]-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9177
PIK3CG (p110g)PIKAtypical3oawA2-amino-4-methyl-8-(1-methylethyl)-6-(1h-pyrazol-4-yl)pteridin-7(8h)-oneHuman9240
PIK3CG (p110g)PIKAtypical3p2bAA3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenolHuman9169
PIK3CG (p110g)PIKAtypical3p2bAB3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenolHuman9165
PIK3CG (p110g)PIKAtypical3preA2-amino-8-(trans-4-methoxycyclohexyl)-4-methyl-6-(1h-pyrazol-3-yl)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman9198
PIK3CG (p110g)PIKAtypical3przA4-amino-2-methyl-n-(1h-pyrazol-3-yl)quinazoline-8-carboxamideHuman9210
PIK3CG (p110g)PIKAtypical3ps6A4-amino-n-(6-methoxypyridin-3-yl)-2-methylquinazoline-8-carboxamideHuman9170
PIK3CG (p110g)PIKAtypical3qaqA[(4-{2-[(3-hydroxyphenyl)amino]-1h-benzimidazol-1-yl}-1,3,5-triazin-2-yl)amino]acetonitrileHuman9211
PIK3CG (p110g)PIKAtypical3qarA1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-3-yl)-1h-benzimidazol-2-amineHuman9178
PIK3CG (p110g)PIKAtypical3qjzAn-{6-[2-(methylsulfanyl)pyrimidin-4-yl]-1,3-benzothiazol-2-yl}acetamideHuman9181
PIK3CG (p110g)PIKAtypical3qk0An-[6-(6-chloro-5-{[(4-fluorophenyl)sulfonyl]amino}pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamideHuman9213
PIK3CG (p110g)PIKAtypical3r7qAn-(2-chlorophenyl)-n-methyl-4h-thieno[3,2-c]chromene-2-carboxamideHuman9227
PIK3CG (p110g)PIKAtypical3r7rA8-(acetylamino)-n-(2-chlorophenyl)-n-methyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2-carboxamideHuman9168
PIK3CG (p110g)PIKAtypical3s2aAn-{2-chloro-5-[4-(morpholin-4-yl)quinolin-6-yl]pyridin-3-yl}-4-fluorobenzenesulfonamideHuman9158
PIK3CG (p110g)PIKAtypical3sd5A5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amineHuman9243
PIK3CG (p110g)PIKAtypical3t8mAn~2~-{2-chloro-4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-n~2~,n~8~-dimethyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2,8-dicarboxamideHuman9186
PIK3CG (p110g)PIKAtypical3tjpAn~6~-(3,4-dimethoxyphenyl)-2-(morpholin-4-yl)-4,5'-bipyrimidine-2',6-diamineHuman9234
PIK3CG (p110g)PIKAtypical3tl5A(2s)-1-(4-{[2-(2-aminopyrimidin-5-yl)-7-methyl-4-(morpholin-4-yl)thieno[3,2-d]pyrimidin-6-yl]methyl}piperazin-1-yl)-2-hydroxypropan-1-oneHuman9160
PIK3CG (p110g)PIKAtypical3zvvA5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-amineHuman9172
PIK3CG (p110g)PIKAtypical3zw3An-{6-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]imidazo[1,2-a]pyridin-2-yl}acetamideHuman9207
PIK3CG (p110g)PIKAtypical4anuA3-amino-n-methyl-6-[3-(1h-tetrazol-5-yl)phenyl]pyrazine-2-carboxamideHuman9162
PIK3CG (p110g)PIKAtypical4anvAA2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazineHuman9195
PIK3CG (p110g)PIKAtypical4anvAB2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazineHuman9166
PIK3CG (p110g)PIKAtypical4anwAA3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamideHuman9174
PIK3CG (p110g)PIKAtypical4anwAB3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamideHuman9175
PIK3CG (p110g)PIKAtypical4anxA5-{3-[(4-{3-[4-(1-methylethyl)phenyl]pyrazin-2-yl}piperazin-1-yl)sulfonyl]phenyl}pyrimidin-2-amineHuman9252
PIK3CG (p110g)PIKAtypical4aofAn-[6-(5-methylsulfonylpyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]ethanamideHuman9245
PIK3CG (p110g)PIKAtypical4dk5A4-(2-[(6-methoxypyridin-3-yl)amino]-5-{[4-(methylsulfonyl)piperazin-1-yl]methyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amineHuman9232
PIK3CG (p110g)PIKAtypical4ezjA2-(1-{[2-(5-fluoro-1h-indol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-olHuman9222
PIK3CG (p110g)PIKAtypical4ezkA2-(1-{[2-(2h-indazol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-olHuman9176
PIK3CG (p110g)PIKAtypical4ezlA2-(1-{[2-(2-aminopyrimidin-5-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-olHuman9235
PIK3CG (p110g)PIKAtypical4f1sAn-(5-{[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-(tetrahydro-2h-pyran-4-yl)pyridin-2-yl]amino}-2-chloropyridin-3-yl)methanesulfonamideHuman9221
PIK3CG (p110g)PIKAtypical4fa6A2-amino-8-cyclopentyl-4-methyl-6-(1h-pyrazol-4-yl)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman9191
PIK3CG (p110g)PIKAtypical4fadA2-amino-6-(5-fluoro-6-methoxypyridin-3-yl)-4-methyl-8-(pyrrolidin-1-yl)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman9202
PIK3CG (p110g)PIKAtypical4fhjA3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-5-yl)imidazo[1,2-a]pyridin-2-amineHuman9209
PIK3CG (p110g)PIKAtypical4fhkA3-[2-methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]-n-(1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-2-amineHuman9204
PIK3CG (p110g)PIKAtypical4fjyA4-[3,3-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1h-indol-1-yl]-7-fluoro-3-methyl-2-(pyridin-3-yl)quinolineHuman9249
PIK3CG (p110g)PIKAtypical4fjzA1'-[7-fluoro-3-methyl-2-(pyridin-2-yl)quinolin-4-yl]-6'-(morpholin-4-yl)-1',2,2',3,5,6-hexahydrospiro[pyran-4,3'-pyrrolo[3,2-b]pyridine]Human9173
PIK3CG (p110g)PIKAtypical4flhA4-(2-[(5-fluoro-6-methoxypyridin-3-yl)amino]-5-{(1r)-1-[4-(methylsulfonyl)piperazin-1-yl]ethyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amineHuman9212
PIK3CG (p110g)PIKAtypical4fulA4-({4-[3-(piperidin-1-ylcarbonyl)phenyl]pyrimidin-2-yl}amino)benzenesulfonamideHuman9242
PIK3CG (p110g)PIKAtypical4g11A2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyrimidin-2-yl]-n-phenylacetamideHuman9223
PIK3CG (p110g)PIKAtypical4gb9A2-[1-({2-[2-(dimethylamino)-1h-benzimidazol-1-yl]-9-methyl-6-(morpholin-4-yl)-9h-purin-8-yl}methyl)piperidin-4-yl]propan-2-olHuman9218
PIK3CG (p110g)PIKAtypical4hleA2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepine-8-carboxamideHuman9219
PIK3CG (p110g)PIKAtypical4hvbA1-{1-[(2s)-2-hydroxypropanoyl]piperidin-4-yl}-3-methyl-8-(6-methylpyridin-3-yl)-1,3-dihydro-2h-imidazo[4,5-c][1,5]naphthyridin-2-oneHuman9225
PIK3CG (p110g)PIKAtypical4j6iA2-methyl-1-(4-{2-[1-(2,2,2-trifluoroethyl)-1h-1,2,4-triazol-5-yl]-4,5-dihydro[1]benzoxepino[5,4-d][1,3]thiazol-8-yl}-1h-pyrazol-1-yl)propan-2-olHuman9189
PIK3CG (p110g)PIKAtypical4kz0Amethyl 2-(acetylamino)-1,3-benzothiazole-6-carboxylateHuman9161
PIK3CG (p110g)PIKAtypical4kzcAn-{6-[6-amino-5-(trifluoromethyl)pyridin-3-yl]imidazo[1,2-a]pyridin-2-yl}acetamideHuman9224
PIK3CG (p110g)PIKAtypical4ps3A1-[6-(5-methoxypyridin-3-yl)-1,3-benzothiazol-2-yl]-3-[2-(1-propyl-1h-imidazol-4-yl)ethyl]ureaHuman9193
PIK3CG (p110g)PIKAtypical4ps7An-[6-(pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamideHuman9163
PIK3CG (p110g)PIKAtypical4ps8An-[6-(5,6-dimethoxypyridin-3-yl)-1,3-benzothiazol-2-yl]acetamideHuman9184
PIK3CG (p110g)PIKAtypical4urkA2-[[(1r)-1-(7-methyl-2-morpholin-4-yl-4-oxidanylidene-pyrido[1,2-a]pyrimidin-9-yl)ethyl]amino]benzoic acidHuman9196
PIK3CG (p110g)PIKAtypical4wwnAn-{(1s)-1-[7-fluoro-2-(pyridin-2-yl)quinolin-3-yl]ethyl}-9h-purin-6-amineHuman9226
PIK3CG (p110g)PIKAtypical4wwoAn-{(1s)-1-[8-chloro-2-(3-fluorophenyl)quinolin-3-yl]ethyl}-9h-purin-6-amineHuman9190
PIK3CG (p110g)PIKAtypical4wwpAn-{(1s)-1-[8-chloro-2-(2-methylpyridin-3-yl)quinolin-3-yl]ethyl}-9h-purin-6-amineHuman9200
PIK3CG (p110g)PIKAtypical4xx5An-[5-(5-methoxypyridin-3-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamideHuman9236
PIK3CG (p110g)PIKAtypical4xz4An-[5-(6-methoxypyrazin-2-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamideHuman9194
PIK3CG (p110g)PIKAtypical5edsA4-azanyl-6-[[(1~{s})-1-[6-fluoranyl-1-(3-methylsulfonylphenyl)benzimidazol-2-yl]ethyl]amino]pyrimidine-5-carbonitrileHuman9208
PIK3CG (p110g)PIKAtypical5g2nA2-azanyl-~{n}-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]pyrimidine-5-carboxamideHuman9206
PIK3CG (p110g)PIKAtypical5g55A6-cyano-4-[[(1r)-1-(4-methylphenyl)ethyl]amino]quinoline-3-carboxamideHuman9199
PIK3CG (p110g)PIKAtypical5jhaA[1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)pyrimidin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanolHuman9246
PIK3CG (p110g)PIKAtypical5jhbA[1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanolHuman9238
PIK3CG (p110g)PIKAtypical5kaeA4-azanyl-6-[[(1~{s})-1-(6-fluoranyl-3-phenyl-4-piperazin-1-ylcarbonyl-quinolin-2-yl)ethyl]amino]pyrimidine-5-carbonitrileHuman9241
PIK3CG (p110g)PIKAtypical5oq4AA5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amineHuman9244
PIK3CG (p110g)PIKAtypical5oq4AB5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amineHuman9203
PIK3CG (p110g)PIKAtypical5t23A3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{s})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amineHuman9157
PIK3CG (p110g)PIKAtypical6audAA10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepineHuman9239
PIK3CG (p110g)PIKAtypical6audAB10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepineHuman9216
PIK3CG (p110g)PIKAtypical6c1sA{4-[2-(5,6-dimethoxypyridin-3-yl)-5-oxo-5,7-dihydro-6h-pyrrolo[3,4-b]pyridin-6-yl]-1h-pyrazol-1-yl}acetonitrileHuman10037
PIK3CG (p110g)PIKAtypical6fh5A3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-oneHuman10883
PIK3CG (p110g)PIKAtypical6gq7A3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-oneHuman10009
PIK3CG (p110g)PIKAtypical6t3bA2-[(4-methoxy-2-methyl-phenyl)amino]-7-methyl-9-(4-oxidanylcyclohexyl)purin-8-oneHuman11906
PIK3CG (p110g)PIKAtypical6t3cA7-methyl-2-[(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(oxan-4-yl)purin-8-oneHuman11907
PIK3CG (p110g)PIKAtypical6xrlA2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman12774
PIK3CG (p110g)PIKAtypical6xrmA5-[2-amino-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-2-[(1s)-1-cyclopropylethyl]-7-(trifluoromethyl)-2,3-dihydro-1h-isoindol-1-oneHuman12775
PIK3CG (p110g)PIKAtypical6xrnA2-amino-5-{2-[(1s)-1-cyclopropylethyl]-7-methyl-1-oxo-2,3-dihydro-1h-isoindol-5-yl}-n-(trans-3-hydroxycyclobutyl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman13954
PIK3CG (p110g)PIKAtypical7jweAgedatolisibHuman13412
PIK3CG (p110g)PIKAtypical7jwzA2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman13410
PIK3CG (p110g)PIKAtypical7jx0An~3~-{[5-(4-acetylphenyl)-4-methyl-1,3-thiazol-2-yl]carbamoyl}-n-tert-butyl-beta-alaninamideHuman13411
PIK3CG (p110g)PIKAtypical7kkeAn-[2-(3,3-dimethylbutoxy)ethyl]-n'-{4-methyl-5-[(pyridin-4-yl)ethynyl]-1,3-thiazol-2-yl}ureaHuman13433
PIK3CG (p110g)PIKAtypical7mezA-Human13798
PIK3CG (p110g)PIKAtypical7z61A9-[(3~{r},4~{r})-4-fluoranylpyrrolidin-3-yl]-7-methyl-2-[(7-methylquinolin-6-yl)amino]purin-8-oneHuman14286
PIK3CG (p110g)PIKAtypical8dp0A-Human14838
PIK3R4VPS15Other7bl1C-Human13360
PIK3R4VPS15Other8sorD-Human14802
PIM1PIMCAMK1xqzA-Human2361
PIM1PIMCAMK1xr1Aphosphoaminophosphonic acid-adenylate esterHuman2406
PIM1PIMCAMK1xwsAA3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2343
PIM1PIMCAMK1xwsAB3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2441
PIM1PIMCAMK1yhsAstaurosporineHuman2444
PIM1PIMCAMK1yi3A2-morpholin-4-yl-7-phenyl-4h-chromen-4-oneHuman2398
PIM1PIMCAMK1yi4AadenosineHuman2403
PIM1PIMCAMK1ywvAA-Human2430
PIM1PIMCAMK1ywvAB-Human2397
PIM1PIMCAMK1yxsAA-Human2417
PIM1PIMCAMK1yxsAB-Human2461
PIM1PIMCAMK1yxtAAphosphoaminophosphonic acid-adenylate esterHuman2425
PIM1PIMCAMK1yxtABphosphoaminophosphonic acid-adenylate esterHuman2319
PIM1PIMCAMK1yxuAadenosine monophosphateHuman2438
PIM1PIMCAMK1yxuBadenosine monophosphateHuman2410
PIM1PIMCAMK1yxuCadenosine monophosphateHuman2408
PIM1PIMCAMK1yxuDadenosine monophosphateHuman2332
PIM1PIMCAMK1yxvAA3,4-dihydroxy-1-methylquinolin-2(1h)-oneHuman2367
PIM1PIMCAMK1yxvAB3,4-dihydroxy-1-methylquinolin-2(1h)-oneHuman2366
PIM1PIMCAMK1yxxAA(3e)-3-[(4-hydroxyphenyl)imino]-1h-indol-2(3h)-oneHuman2351
PIM1PIMCAMK1yxxAB(3e)-3-[(4-hydroxyphenyl)imino]-1h-indol-2(3h)-oneHuman2437
PIM1PIMCAMK2bikBA3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2341
PIM1PIMCAMK2bikBB3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2463
PIM1PIMCAMK2bilB3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2449
PIM1PIMCAMK2bzhBAruthenium-pyridocarbazole-1Human7230
PIM1PIMCAMK2bzhBBruthenium-pyridocarbazole-1Human7234
PIM1PIMCAMK2bziBA-Human7225
PIM1PIMCAMK2bziBB-Human7233
PIM1PIMCAMK2bzjAAruthenium-pyridocarbazole-3Human7224
PIM1PIMCAMK2bzjABruthenium-pyridocarbazole-3Human7228
PIM1PIMCAMK2bzkBphosphoaminophosphonic acid-adenylate esterHuman2330
PIM1PIMCAMK2c3iBA1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman2348
PIM1PIMCAMK2c3iBB1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman2374
PIM1PIMCAMK2j2iBA(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHuman2318
PIM1PIMCAMK2j2iBB(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHuman2434
PIM1PIMCAMK2o3pAA3,5,7,3',4'-pentahydroxyflavoneHuman2320
PIM1PIMCAMK2o3pAB3,5,7,3',4'-pentahydroxyflavoneHuman2409
PIM1PIMCAMK2o63A3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)-4h-chromen-4-oneHuman2453
PIM1PIMCAMK2o64A3,5,6,7-tetrahydroxy-2-(3,4-dihydroxyphenyl)-4h-chromen-4-oneHuman2421
PIM1PIMCAMK2o65A5,7-dihydroxy-2-(3,4,5-trihydroxyphenyl)-4h-chromen-4-oneHuman2324
PIM1PIMCAMK2objA6-(5-bromo-2-hydroxyphenyl)-2-oxo-4-phenyl-1,2-dihydropyridine-3-carbonitrileHuman2336
PIM1PIMCAMK2oi4XA-Human7236
PIM1PIMCAMK2oi4XB-Human7226
PIM1PIMCAMK2xixAA3,5-diamino-1h-[1,2,4]triazoleHuman2468
PIM1PIMCAMK2xixAB3,5-diamino-1h-[1,2,4]triazoleHuman2433
PIM1PIMCAMK2xiyAA2-hydroxymethyl-benzoimidazoleHuman2415
PIM1PIMCAMK2xiyAB2-hydroxymethyl-benzoimidazoleHuman2363
PIM1PIMCAMK2xizAA(e)-pyridin-4-yl-acrylic acidHuman2436
PIM1PIMCAMK2xizAB(e)-pyridin-4-yl-acrylic acidHuman2373
PIM1PIMCAMK2xj0AA(e)-3-(2-amino-pyridine-5yl)-acrylic acidHuman2435
PIM1PIMCAMK2xj0AB(e)-3-(2-amino-pyridine-5yl)-acrylic acidHuman2395
PIM1PIMCAMK2xj1AA(2e)-3-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}phenyl)prop-2-enoic acidHuman2469
PIM1PIMCAMK2xj1AB(2e)-3-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}phenyl)prop-2-enoic acidHuman2422
PIM1PIMCAMK2xj2AA(2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acidHuman2334
PIM1PIMCAMK2xj2AB(2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acidHuman2418
PIM1PIMCAMK3a99Aphosphoaminophosphonic acid-adenylate esterHuman2322
PIM1PIMCAMK3bgpA4-[3-(4-chlorophenyl)-2,1-benzisoxazol-5-yl]pyrimidin-2-amineHuman2359
PIM1PIMCAMK3bgqAn-cyclohexyl-3-[3-(trifluoromethyl)phenyl][1,2,4]triazolo[4,3-b]pyridazin-6-amineHuman2465
PIM1PIMCAMK3bgzA2,3-diphenyl-1h-indole-7-carboxylic acidHuman2462
PIM1PIMCAMK3bwfAA-Human7231
PIM1PIMCAMK3bwfAB-Human7235
PIM1PIMCAMK3c4eAn-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amineHuman2413
PIM1PIMCAMK3c4eBn-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amineHuman2423
PIM1PIMCAMK3c4eCn-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amineHuman2440
PIM1PIMCAMK3c4eDn-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amineHuman2378
PIM1PIMCAMK3cxwAA(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman2464
PIM1PIMCAMK3cxwAB(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman2392
PIM1PIMCAMK3cy2AA(4r)-7-chloro-9-methyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman2333
PIM1PIMCAMK3cy2AB(4r)-7-chloro-9-methyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman2459
PIM1PIMCAMK3cy3A(2s)-1,3-benzothiazol-2-yl{2-[(2-pyridin-3-ylethyl)amino]pyrimidin-4-yl}ethanenitrileHuman2443
PIM1PIMCAMK3dcvA4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHuman2372
PIM1PIMCAMK3f2aA(2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acidHuman2460
PIM1PIMCAMK3jpvA1,10-dihydropyrrolo[2,3-a]carbazole-3-carbaldehydeHuman2431
PIM1PIMCAMK3jxwA8-[(e)-2-cyclopropylethenyl]-2-[(dimethylamino)methyl][1]benzothieno[3,2-d]pyrimidin-4(3h)-oneHuman2393
PIM1PIMCAMK3jy0AA8-chloro-2-{[(3s)-3-hydroxypyrrolidin-1-yl]methyl}[1]benzothieno[3,2-d]pyrimidin-4(3h)-oneHuman2405
PIM1PIMCAMK3jyaAA6,9-dichloro[1]benzothieno[3,2-d]pyrimidin-4(3h)-oneHuman2371
PIM1PIMCAMK3ma3AAnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman2368
PIM1PIMCAMK3ma3ABnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman2347
PIM1PIMCAMK3qf9AA6-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}naphthalene-1-carboxamideHuman2329
PIM1PIMCAMK3qf9AB6-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}naphthalene-1-carboxamideHuman2331
PIM1PIMCAMK3r00A5-bromo-1-benzofuran-2-carboxylic acidHuman2467
PIM1PIMCAMK3r01A5-bromo-7-methoxy-1-benzofuran-2-carboxylic acidHuman2407
PIM1PIMCAMK3r02AA7-[(cis-4-aminocyclohexyl)amino]-5-bromo-1-benzofuran-2-carboxylic acidHuman2420
PIM1PIMCAMK3r02AB7-[(cis-4-aminocyclohexyl)amino]-5-bromo-1-benzofuran-2-carboxylic acidHuman2338
PIM1PIMCAMK3r04AA5-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}-1-benzofuran-2-carboxylic acidHuman2353
PIM1PIMCAMK3r04AB5-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}-1-benzofuran-2-carboxylic acidHuman2335
PIM1PIMCAMK3t9iA2-methoxy-4-(3-phenyl-2h-pyrazolo[3,4-b]pyridin-6-yl)phenolHuman2450
PIM1PIMCAMK3uixAA2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHuman2456
PIM1PIMCAMK3uixAB2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHuman2387
PIM1PIMCAMK3umwAA(2z)-2-(1h-indazol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3(2h)-oneHuman2411
PIM1PIMCAMK3umwAB(2z)-2-(1h-indazol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3(2h)-oneHuman2414
PIM1PIMCAMK3umxAA(2z)-7-(azepan-1-ylmethyl)-6-hydroxy-2-(1h-indol-3-ylmethylidene)-1-benzofuran-3(2h)-oneHuman2432
PIM1PIMCAMK3umxAB(2z)-7-(azepan-1-ylmethyl)-6-hydroxy-2-(1h-indol-3-ylmethylidene)-1-benzofuran-3(2h)-oneHuman2375
PIM1PIMCAMK3vbqAA5-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}benzyl)-2h-1lambda~4~,3-thiazole-2,4(3h)-dioneHuman2354
PIM1PIMCAMK3vbqAB5-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}benzyl)-2h-1lambda~4~,3-thiazole-2,4(3h)-dioneHuman2454
PIM1PIMCAMK3vbtA4-chloro-2-(1h-pyrazol-3-yl)phenolHuman2349
PIM1PIMCAMK3vbvA8-hydroxyquinoline-2-carboxamideHuman2399
PIM1PIMCAMK3vbwA1,3-dioxo-2,3-dihydro-1h-indene-2-carbonitrileHuman2390
PIM1PIMCAMK3vbxAA6-bromo-4-hydroxy-2h-chromen-2-oneHuman2427
PIM1PIMCAMK3vbxAB6-bromo-4-hydroxy-2h-chromen-2-oneHuman2448
PIM1PIMCAMK3vbyAfuran-2-yl(1h-indol-3-yl)methanoneHuman2466
PIM1PIMCAMK3vc4A(5z)-5-[3-(trifluoromethyl)benzylidene]-1,3-thiazolidine-2,4-dioneHuman2356
PIM1PIMCAMK3we8AAcyclopentadienyl(carbon monoxide)(7-oxo-7,10-dihydro-1,8-phenanthrolin-10-yl-kappa~2~c~10~,n~1~)rutheniumHuman7237
PIM1PIMCAMK3we8ABcyclopentadienyl(carbon monoxide)(7-oxo-7,10-dihydro-1,8-phenanthrolin-10-yl-kappa~2~c~10~,n~1~)rutheniumHuman7232
PIM1PIMCAMK4a7cAn-(piperidin-4-ylmethyl)-3-[3-(trifluoromethyloxy)phenyl]-[1,2,3]triazolo[4,5-b]pyridin-5-amineHuman2321
PIM1PIMCAMK4aluAA8-bromo-2-(2-chlorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman2452
PIM1PIMCAMK4aluAB8-bromo-2-(2-chlorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman2384
PIM1PIMCAMK4alvAA8-bromo-2-{2-chloro-4-[(piperidin-4-ylmethyl)amino]phenyl}[1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman2323
PIM1PIMCAMK4alvAB8-bromo-2-{2-chloro-4-[(piperidin-4-ylmethyl)amino]phenyl}[1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman2396
PIM1PIMCAMK4alwAA8-bromanyl-2-[(4-methylpiperazin-1-yl)methyl]-3h-[1]benzofuro[3,2-d]pyrimidin-4-oneHuman2419
PIM1PIMCAMK4alwAB8-bromanyl-2-[(4-methylpiperazin-1-yl)methyl]-3h-[1]benzofuro[3,2-d]pyrimidin-4-oneHuman2350
PIM1PIMCAMK4as0AAphtalimide-ruthenium complexHuman7227
PIM1PIMCAMK4as0ABphtalimide-ruthenium complexHuman7229
PIM1PIMCAMK4bznAn-(2,2-dimethylpropyl)-2-[1-oxo-7-(thiophen-3-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamideHuman2402
PIM1PIMCAMK4bzoAn-[(1s)-2-amino-1-phenylethyl]-2-[(4s)-7-(2-fluoro-4-pyridinyl)-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamideHuman2339
PIM1PIMCAMK4dtkAA(5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dioneHuman2344
PIM1PIMCAMK4dtkAB(5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dioneHuman2451
PIM1PIMCAMK4enxA(2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-nitrobenzylidene)-1,3-thiazolidin-4-oneHuman2352
PIM1PIMCAMK4enyAA(2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-oneHuman2342
PIM1PIMCAMK4enyAB(2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-oneHuman2424
PIM1PIMCAMK4gw8AA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman2428
PIM1PIMCAMK4gw8AB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman2391
PIM1PIMCAMK4i41A1,4-dihydroxy-5,8-bis({2-[(2-hydroxyethyl)amino]ethyl}amino)-9,10-anthracenedioneHuman2326
PIM1PIMCAMK4iaaA10-{2-[(2r)-1-methylpiperidin-2-yl]ethyl}-2-(methylsulfanyl)-10h-phenothiazineHuman2325
PIM1PIMCAMK4jx3A-Human2380
PIM1PIMCAMK4jx7A2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6h)-oneHuman2340
PIM1PIMCAMK4k0yAAn-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2455
PIM1PIMCAMK4k0yABn-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2445
PIM1PIMCAMK4k18A5-(4-cyanobenzyl)-n-(4-fluorophenyl)-7-hydroxypyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2377
PIM1PIMCAMK4k1bAn-[5-(2-fluorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-5-({[(3r,4r)-3-fluoropiperidin-4-yl]methyl}amino)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2362
PIM1PIMCAMK4ll5AA6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazoleHuman2365
PIM1PIMCAMK4ll5AB6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazoleHuman2382
PIM1PIMCAMK4lm5AA2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHuman2400
PIM1PIMCAMK4lm5AB2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHuman2327
PIM1PIMCAMK4lmuAA3,5,7,3',4'-pentahydroxyflavoneHuman2376
PIM1PIMCAMK4lmuAB3,5,7,3',4'-pentahydroxyflavoneHuman2404
PIM1PIMCAMK4mbiAn,n-dimethyl-n'-[3-(1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]ethane-1,2-diamineHuman2447
PIM1PIMCAMK4mblA(1r,2r)-n-[3-(naphthalen-2-yl)pyrazolo[1,5-a]pyrimidin-5-yl]cyclohexane-1,2-diamineHuman2381
PIM1PIMCAMK4mtaA2-methyl-5-phenylfuran-3-carboxylic acidHuman2370
PIM1PIMCAMK4n6yA2-(acetylamino)-n-[2-(piperidin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman2383
PIM1PIMCAMK4n6zA3-amino-n-{4-[(3s)-3-aminopiperidin-1-yl]pyridin-3-yl}pyrazine-2-carboxamideHuman2442
PIM1PIMCAMK4n70AAn-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamideHuman2388
PIM1PIMCAMK4n70ABn-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamideHuman2357
PIM1PIMCAMK4rblA1,4,5,8-tetrahydroxyanthracene-9,10-dioneHuman2385
PIM1PIMCAMK4rc2A1-amino-5,8-dihydroxy-4-({2-[(2-hydroxyethyl)amino]ethyl}amino)anthracene-9,10-dioneHuman2346
PIM1PIMCAMK4rc3A1,4-dihydroxy-5,8-bis{[2-(2-hydroxyethoxy)ethyl]amino}anthracene-9,10-dioneHuman2412
PIM1PIMCAMK4rc4A1,4-bis[(2-aminoethyl)amino]-5,8-dihydroxyanthracene-9,10-dioneHuman2369
PIM1PIMCAMK4rpvA(3s)-1-{6-[5-(2,6-difluorophenyl)-2h-indazol-3-yl]pyrazin-2-yl}piperidin-3-amineHuman2364
PIM1PIMCAMK4ty1An-tert-butyl-5-[3-(4-cyclopropylpyrimidin-2-yl)-1h-indol-5-yl]-1,3,4-oxadiazol-2-amineHuman2394
PIM1PIMCAMK4wrsA3-{6-[(4r)-6-azaspiro[2.5]oct-4-yloxy]pyrazin-2-yl}-5-(2,6-difluorophenyl)-1h-indazoleHuman2439
PIM1PIMCAMK4wsyA5-[3-(quinolin-3-yl)-2h-indazol-5-yl]-1,3-thiazol-2-amineHuman2429
PIM1PIMCAMK4wt6A6-[5-(5-amino-1,3,4-thiadiazol-2-yl)-1h-indol-3-yl]-n-cyclopentylpyridin-2-amineHuman2386
PIM1PIMCAMK4xh6A5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4h-chromen-4-oneHuman5975
PIM1PIMCAMK4xhkBA2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHuman2446
PIM1PIMCAMK4xhkBB2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHuman2355
PIM1PIMCAMK5c1qB3-methoxy[1]benzothieno[2,3-c]quinolin-6(5h)-oneHuman6288
PIM1PIMCAMK5dgzA(2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amineHuman6209
PIM1PIMCAMK5dhjAA3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridineHuman6212
PIM1PIMCAMK5dhjAB3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridineHuman6211
PIM1PIMCAMK5diaA(1s,3s)-n-{6-[5-(pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridin-3-yl]pyridin-2-yl}cyclohexane-1,3-diamineHuman6210
PIM1PIMCAMK5dwrAn-{4-[(1r,3s,5s)-3-amino-5-methylcyclohexyl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamideHuman6238
PIM1PIMCAMK5eolA macrocyclic quinoxaline-pyrrolodihydropiperidinoneHuman6601
PIM1PIMCAMK5iisA3-amino-n-(2'-amino-6'-methyl[4,4'-bipyridin]-3-yl)-6-(2-fluorophenyl)pyridine-2-carboxamideHuman6504
PIM1PIMCAMK5ipjA2-(tert-butylamino)-3-methyl-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-oneHuman6703
PIM1PIMCAMK5kcxAA4-chloranyl-1-methyl-2-[4-(4-methylpiperazin-1-yl)phenyl]pyrrolo[2,3-b]pyridine-6-carboxamideHuman8247
PIM1PIMCAMK5kcxAB4-chloranyl-1-methyl-2-[4-(4-methylpiperazin-1-yl)phenyl]pyrrolo[2,3-b]pyridine-6-carboxamideHuman8248
PIM1PIMCAMK5kgdA2-pyridin-3-yl-1~{h}-benzimidazoleHuman8309
PIM1PIMCAMK5kgeA5-(3,4-dichlorophenyl)-1~{h}-pyrazol-3-amineHuman8310
PIM1PIMCAMK5kggA2-(5-chloranyl-1~{h}-indol-3-yl)ethanamineHuman8308
PIM1PIMCAMK5kgiA2-[3,4-bis(chloranyl)phenoxy]ethanamineHuman8306
PIM1PIMCAMK5kgkA3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amineHuman8307
PIM1PIMCAMK5kziA~{n}-[4-[(3~{s})-3-azanylpiperidin-1-yl]pyridin-3-yl]-2-[2,6-bis(fluoranyl)phenyl]imidazo[1,5-b]pyridazin-7-amineHuman7195
PIM1PIMCAMK5mzlAA~{n}-quinolin-5-ylpyridine-3-carboxamideHuman9562
PIM1PIMCAMK5mzlAB~{n}-quinolin-5-ylpyridine-3-carboxamideHuman9563
PIM1PIMCAMK5n4nAA3,4-dimethyl-5-(1~{h}-1,2,4-triazol-3-yl)thiophene-2-carbonitrileHuman9579
PIM1PIMCAMK5n4nAB3,4-dimethyl-5-(1~{h}-1,2,4-triazol-3-yl)thiophene-2-carbonitrileHuman9595
PIM1PIMCAMK5n4oAA(~{e})-3-(4-methylphenyl)prop-2-enoic acidHuman9580
PIM1PIMCAMK5n4oAB(~{e})-3-(4-methylphenyl)prop-2-enoic acidHuman9582
PIM1PIMCAMK5n4rAA2-(azepan-1-yl)-1-(1~{h}-indol-3-yl)propan-1-oneHuman9584
PIM1PIMCAMK5n4rAB2-(azepan-1-yl)-1-(1~{h}-indol-3-yl)propan-1-oneHuman9583
PIM1PIMCAMK5n4uAA5-(2-azanyl-1,3-thiazol-4-yl)-1,3-dihydrobenzimidazol-2-oneHuman9588
PIM1PIMCAMK5n4uAB5-(2-azanyl-1,3-thiazol-4-yl)-1,3-dihydrobenzimidazol-2-oneHuman9590
PIM1PIMCAMK5n4vAA2-cyclopropyl-4,5-dimethyl-thieno[2,3-d]pyrimidine-6-carboxylic acidHuman9592
PIM1PIMCAMK5n4vAB2-cyclopropyl-4,5-dimethyl-thieno[2,3-d]pyrimidine-6-carboxylic acidHuman9594
PIM1PIMCAMK5n4xAA4,5-bis(bromanyl)thiophene-2-carbohydrazideHuman9600
PIM1PIMCAMK5n4xAB4,5-bis(bromanyl)thiophene-2-carbohydrazideHuman9593
PIM1PIMCAMK5n4yAA2,5-dihydro-1~{h}-isothiochromeno[4,3-c]pyrazol-3-oneHuman9589
PIM1PIMCAMK5n4yAB2,5-dihydro-1~{h}-isothiochromeno[4,3-c]pyrazol-3-oneHuman9597
PIM1PIMCAMK5n4zAA(~{e})-4-(4-hydroxyphenyl)but-3-en-2-oneHuman9587
PIM1PIMCAMK5n4zAB(~{e})-4-(4-hydroxyphenyl)but-3-en-2-oneHuman9599
PIM1PIMCAMK5n50AA2-(4-chlorophenyl)sulfanylethanehydrazideHuman9585
PIM1PIMCAMK5n50AB2-(4-chlorophenyl)sulfanylethanehydrazideHuman9598
PIM1PIMCAMK5n51AA3,4-bis(bromanyl)thiophene-2-carboxylic acidHuman9596
PIM1PIMCAMK5n51AB3,4-bis(bromanyl)thiophene-2-carboxylic acidHuman9591
PIM1PIMCAMK5n52AA(~{e})-3-(2,3-dimethoxyphenyl)prop-2-enoic acidHuman9581
PIM1PIMCAMK5n52AB(~{e})-3-(2,3-dimethoxyphenyl)prop-2-enoic acidHuman9586
PIM1PIMCAMK5n5lAA5-bromanyl-1~{h}-indole-3-carboxylic acidHuman9703
PIM1PIMCAMK5n5lAB5-bromanyl-1~{h}-indole-3-carboxylic acidHuman9704
PIM1PIMCAMK5n5mAA~{n}-(isoquinolin-5-ylmethyl)-~{n}-methyl-2-[(3~{r})-pyrrolidin-3-yl]benzamideHuman9702
PIM1PIMCAMK5n5mAB~{n}-(isoquinolin-5-ylmethyl)-~{n}-methyl-2-[(3~{r})-pyrrolidin-3-yl]benzamideHuman9705
PIM1PIMCAMK5ndtAA3-(2-thiophen-2-ylethenyl)-1~{h}-quinoxalin-2-oneHuman9907
PIM1PIMCAMK5ndtAB3-(2-thiophen-2-ylethenyl)-1~{h}-quinoxalin-2-oneHuman9906
PIM1PIMCAMK5o11AA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman8656
PIM1PIMCAMK5o11AB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman8657
PIM1PIMCAMK5o12A(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman8654
PIM1PIMCAMK5o13AA(3~{e})-5-chloranyl-3-[[5-[3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl]furan-2-yl]methylidene]-1~{h}-indol-2-oneHuman8653
PIM1PIMCAMK5o13AB(3~{e})-5-chloranyl-3-[[5-[3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl]furan-2-yl]methylidene]-1~{h}-indol-2-oneHuman8655
PIM1PIMCAMK5telAA4-chloro-2-{5,6-dimethoxy-1-[2-(4-methylpiperazin-1-yl)ethyl]-1h-indol-3-yl}-1h-pyrrolo[2,3-b]pyridineHuman8564
PIM1PIMCAMK5telAB4-chloro-2-{5,6-dimethoxy-1-[2-(4-methylpiperazin-1-yl)ethyl]-1h-indol-3-yl}-1h-pyrrolo[2,3-b]pyridineHuman8562
PIM1PIMCAMK5texA(4-{4-chloro-1-methyl-2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)methanolHuman8566
PIM1PIMCAMK5toeA2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrileHuman8563
PIM1PIMCAMK5turA1-methyl-2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrileHuman8565
PIM1PIMCAMK5v80A1-methyl-4-{3-[6-(piperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[3,4-c]pyridin-5-yl}piperazin-2-oneHuman9828
PIM1PIMCAMK5v82A1-{6-[(3r)-4,4-difluoropiperidin-3-yl]pyridin-2-yl}-6-(6-methylpyrazin-2-yl)-1h-pyrazolo[4,3-c]pyridineHuman7581
PIM1PIMCAMK5vuaBA(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9074
PIM1PIMCAMK5vuaBB(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9077
PIM1PIMCAMK5vubBA(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9073
PIM1PIMCAMK5vubBB(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9076
PIM1PIMCAMK5vubBC(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9072
PIM1PIMCAMK5vucBA(2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-oneHuman9071
PIM1PIMCAMK5vucBB(2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-oneHuman9075
PIM1PIMCAMK6aydAAn-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamideHuman9442
PIM1PIMCAMK6aydABn-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamideHuman9443
PIM1PIMCAMK6bskA4-{6-[6-(propan-2-ylamino)-1h-indazol-1-yl]pyrazin-2-yl}benzoic acidHuman9758
PIM1PIMCAMK6kziA4-(2-chloro-10h-phenoxazin-10-yl)-n,n-diethylbutan-1-amineHuman12019
PIM1PIMCAMK6l11A5-(2-chloranylphenoxazin-10-yl)-~{n},~{n}-diethyl-pentan-1-amineHuman12336
PIM1PIMCAMK6l12A4-[(2-chloranylphenoxazin-10-yl)methyl]cyclohexan-1-amineHuman12340
PIM1PIMCAMK6l13A2-chloranyl-10-(2-piperidin-4-ylethyl)phenoxazineHuman12337
PIM1PIMCAMK6l14A2-chloranyl-10-[3-[(3~{s})-piperidin-3-yl]propyl]phenoxazineHuman12338
PIM1PIMCAMK6l15A7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazineHuman12339
PIM1PIMCAMK6l16A2-[4-[2-(7-chloranylpyrido[3,4-b][1,4]benzoxazin-5-yl)ethyl]piperidin-1-yl]ethanamineHuman12335
PIM1PIMCAMK6l17A7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazin-8-amineHuman12740
PIM1PIMCAMK6mt0A3-(1-methylcyclopropyl)-2-[(1-methylcyclopropyl)amino]-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-oneHuman10850
PIM1PIMCAMK6no8A5-amino-n-{5-[(4s)-4-aminoazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamideHuman11832
PIM1PIMCAMK6no9A5-amino-n-{5-[(4r,5r)-4-amino-5-fluoroazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamideHuman10936
PIM1PIMCAMK6pcwA4-[5-(cyclopropylcarbamoyl)thiophen-2-yl]-1-benzothiophene-2-carboxamideHuman11455
PIM1PIMCAMK6pdiA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11459
PIM1PIMCAMK6pdnAA4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acidHuman11456
PIM1PIMCAMK6pdnAB4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acidHuman11458
PIM1PIMCAMK6pdoAA4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamideHuman11461
PIM1PIMCAMK6pdoAB4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamideHuman11460
PIM1PIMCAMK6pdpAA5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamideHuman11454
PIM1PIMCAMK6pdpAB5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamideHuman11457
PIM1PIMCAMK6qxkBA2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-oneHuman11035
PIM1PIMCAMK6qxkBB2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-oneHuman11036
PIM1PIMCAMK6vruAA3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamideHuman13127
PIM1PIMCAMK6vruAB3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamideHuman13128
PIM1PIMCAMK6vrvA4-chloro-1-{(1s)-1-[(3s)-3-fluoropyrrolidin-3-yl]ethyl}-3-methyl-1h-pyrrolo[2,3-b]pyridine-6-carboxamideHuman13129
PIM1PIMCAMK6ykdAA~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamideHuman12402
PIM1PIMCAMK6ykdAB~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamideHuman12401
PIM1PIMCAMK7oovA~{n}-[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-[[(2~{r})-1-azanyl-5-[[$l^{1}-azanyl($l^{2}-azanylidene)methyl]-$l^{2}-azanyl]-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]amino]-5-carbamimidamido-1-oxidanylidene-pentan-2-yl]-9-oxidanylidene-9-[4-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]nonanamideHuman13824
PIM1PIMCAMK7oowA-Human13826
PIM1PIMCAMK7ooxAA-Human13825
PIM1PIMCAMK7ooxAB-Human13823
PIM1PIMCAMK7qb2A4-[(e)-(6-azanyl-1-methyl-2-oxidanylidene-indol-3-ylidene)methyl]benzoic acidHuman14518
PIM1PIMCAMK7qfmAA4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHuman14561
PIM1PIMCAMK7qfmAB4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHuman14560
PIM1PIMCAMK7vsyA-Human15098
PIM1PIMCAMK7xsvAA8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaeneHuman14287
PIM1PIMCAMK7xsvAB8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaeneHuman14288
PIM1PIMCAMK7z6uAA4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHuman14602
PIM1PIMCAMK7z6uAB4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHuman14600
PIM1PIMCAMK7zunA(4~{s})-4-(2-azanylethyl)-6-phenyl-7-[3-(trifluoromethyloxy)phenyl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1-olHuman14383
PIM1PIMCAMK8afrAA4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acidHuman14603
PIM1PIMCAMK8afrAB4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acidHuman14601
PIM2PIMCAMK2iwiAruthenium-pyridocarbazole-1Human7217
PIM2PIMCAMK2iwiBruthenium-pyridocarbazole-1Human7216
PIM2PIMCAMK4x7qA2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHuman1415
PIM2PIMCAMK4x7qB2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHuman1416
PKMYT1 (MYT1)WEEOther3p1aAA-Human1216
PKMYT1 (MYT1)WEEOther3p1aAB-Human1217
PKMYT1 (MYT1)WEEOther5vcvAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman8339
PKMYT1 (MYT1)WEEOther5vcwA(2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamideHuman8335
PKMYT1 (MYT1)WEEOther5vcwB(2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-3-cyano-7-ethoxyquinolin-6-yl}-4-(dimethylamino)but-2-enamideHuman8346
PKMYT1 (MYT1)WEEOther5vcxAn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman8341
PKMYT1 (MYT1)WEEOther5vcyAA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8345
PKMYT1 (MYT1)WEEOther5vcyAB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8338
PKMYT1 (MYT1)WEEOther5vczAA4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8342
PKMYT1 (MYT1)WEEOther5vczAB4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8336
PKMYT1 (MYT1)WEEOther5vd0A1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman8344
PKMYT1 (MYT1)WEEOther5vd1AAn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman8337
PKMYT1 (MYT1)WEEOther5vd1ABn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman8340
PKMYT1 (MYT1)WEEOther5vd3An-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman8343
PKMYT1 (MYT1)WEEOther8d6cA(1p)-2-amino-6-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman14296
PKMYT1 (MYT1)WEEOther8d6dA(1p)-2-amino-5-bromo-1-(3-hydroxy-2,6-dimethylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman14294
PKMYT1 (MYT1)WEEOther8d6eAA(1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamideHuman14295
PKMYT1 (MYT1)WEEOther8d6eAB(1p)-2-amino-1-(3-hydroxy-2,6-dimethylphenyl)-5,6-dimethyl-1h-pyrrolo[2,3-b]pyridine-3-carboxamideHuman14293
PKMYT1 (MYT1)WEEOther8d6fA(1m)-2-amino-1-(5-hydroxy-2-methylphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman14297
PKMYT1 (MYT1)WEEOther8wjyAA[6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanoneHuman15008
PKMYT1 (MYT1)WEEOther8wjyAB[6-azanyl-5-(2,6-dimethyl-3-oxidanyl-phenyl)-2,3-dimethyl-pyrrolo[2,3-b]pyrazin-7-yl]-(6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazin-5-yl)methanoneHuman15007
PKN1PKNAGC4otdAA-Human545
PKN1PKNAGC4otdAB-Human546
PKN1PKNAGC4otgAAlestaurtinibHuman548
PKN1PKNAGC4otgABlestaurtinibHuman549
PKN1PKNAGC4othAA-Human7203
PKN1PKNAGC4othAB-Human7204
PKN1PKNAGC4otiAA3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHuman551
PKN1PKNAGC4otiAB3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHuman547
PKN2PKNAGC4crsAphosphothiophosphoric acid-adenylate esterHuman535
PLK1PLKOther2ou7AAphosphoaminophosphonic acid-adenylate esterHuman4956
PLK1PLKOther2ou7ABphosphoaminophosphonic acid-adenylate esterHuman4973
PLK1PLKOther2owbAA4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHuman4974
PLK1PLKOther2owbAB4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHuman4958
PLK1PLKOther2rkuAA4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman4969
PLK1PLKOther2rkuAB4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman4966
PLK1PLKOther2v5qAA-Human4970
PLK1PLKOther2v5qAB-Human4960
PLK1PLKOther2v5qBA-Human4959
PLK1PLKOther2v5qBB-Human4961
PLK1PLKOther2yacA1-(2-hydroxyethyl)-8-[[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)phenyl]amino]-4,5-dihydropyrimido[5,4-g]indazole-3-carboxamideHuman4957
PLK1PLKOther3fc2AAn-{trans-4-[4-(cyclopropylmethyl)piperazin-1-yl]cyclohexyl}-4-{[(7r)-7-ethyl-5-methyl-8-(1-methylethyl)-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxybenzamideHuman4964
PLK1PLKOther3fc2ABn-{trans-4-[4-(cyclopropylmethyl)piperazin-1-yl]cyclohexyl}-4-{[(7r)-7-ethyl-5-methyl-8-(1-methylethyl)-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxybenzamideHuman4967
PLK1PLKOther3kb7A8-{[2-methoxy-5-(4-methylpiperazin-1-yl)phenyl]amino}-1-methyl-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4962
PLK1PLKOther3thbA9-chloro-2-({5-[3-(dimethylamino)propyl]-2-methylpyridin-3-yl}amino)-5,7-dihydro-6h-pyrimido[5,4-d][1]benzazepine-6-thioneHuman4968
PLK1PLKOther4a4lA1-methyl-5-(2-{[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)phenyl]amino}pyrimidin-4-yl)-1h-pyrrole-3-carboxamideHuman4971
PLK1PLKOther4a4oA1-methyl-2-(2-{[5-(4-methylpiperazin-1-yl)-2-(trifluoromethoxy)phenyl]amino}pyrimidin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4965
PLK1PLKOther4j52AA4-{[(7r)-9-cyclopentyl-7-ethenyl-7-fluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl]amino}-3-methoxy-n-(4-methylpiperazin-1-yl)benzamideHuman4955
PLK1PLKOther4j52AB4-{[(7r)-9-cyclopentyl-7-ethenyl-7-fluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl]amino}-3-methoxy-n-(4-methylpiperazin-1-yl)benzamideHuman4976
PLK1PLKOther4j53AA4-[(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-2-fluoro-5-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman4975
PLK1PLKOther4j53AB4-[(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-2-fluoro-5-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman4972
PLK1PLKOther4j53AC4-[(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-2-fluoro-5-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman4963
PLK1PLKOther5ta6AA4-{[(6r)-7-cyano-5-cyclopentyl-6-ethyl-5,6-dihydroimidazo[1,5-f]pteridin-3-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman7465
PLK1PLKOther5ta6AB4-{[(6r)-7-cyano-5-cyclopentyl-6-ethyl-5,6-dihydroimidazo[1,5-f]pteridin-3-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman7462
PLK1PLKOther5ta6AC4-{[(6r)-7-cyano-5-cyclopentyl-6-ethyl-5,6-dihydroimidazo[1,5-f]pteridin-3-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman7463
PLK1PLKOther5ta8AA4-[(9-cyclopentyl-7,7-difluoro-5-methyl-6-oxo-6,7,8,9-tetrahydro-5h-pyrimido[4,5-b][1,4]diazepin-2-yl)amino]-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman7464
PLK1PLKOther8bjtA1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman14712
PLK1PLKOther8x72Aphosphoaminophosphonic acid-adenylate esterHuman15097
PLK2PLKOther4i5mA4-{[(7r)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,7,8-tetrahydropteridin-2-yl]amino}-3-methoxy-n-(1-methylpiperidin-4-yl)benzamideHuman5557
PLK2PLKOther4i5pAA(7r)-8-cyclopentyl-7-ethyl-5-methyl-2-(1h-pyrrol-2-yl)-7,8-dihydropteridin-6(5h)-oneHuman5559
PLK2PLKOther4i5pAB(7r)-8-cyclopentyl-7-ethyl-5-methyl-2-(1h-pyrrol-2-yl)-7,8-dihydropteridin-6(5h)-oneHuman5560
PLK2PLKOther4i6bAA(7r)-8-cyclopentyl-7-ethyl-5-methyl-7,8-dihydropteridin-6(5h)-oneHuman5565
PLK2PLKOther4i6bAB(7r)-8-cyclopentyl-7-ethyl-5-methyl-7,8-dihydropteridin-6(5h)-oneHuman5562
PLK2PLKOther4i6fAA(7r)-8-cyclopentyl-7-ethyl-5-methyl-2-(2-phenyl-1h-imidazol-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman5564
PLK2PLKOther4i6fAB(7r)-8-cyclopentyl-7-ethyl-5-methyl-2-(2-phenyl-1h-imidazol-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman5563
PLK2PLKOther4i6hAA(7r)-8-cyclopentyl-7-ethyl-5-methyl-2-[2-(1,3-thiazol-4-yl)-1h-imidazol-1-yl]-7,8-dihydropteridin-6(5h)-oneHuman5558
PLK2PLKOther4i6hAB(7r)-8-cyclopentyl-7-ethyl-5-methyl-2-[2-(1,3-thiazol-4-yl)-1h-imidazol-1-yl]-7,8-dihydropteridin-6(5h)-oneHuman5561
PLK3PLKOther4b6lA4-[[(4r)-5-cyclopentyl-4-ethyl-3a,4-dihydro-3h-[1,2,4]triazolo[4,3-f]pteridin-7-yl]amino]-n-cyclopropyl-3-methoxy-benzamideHuman3797
PLK4PLKOther3cokAAphosphoaminophosphonic acid-adenylate esterHuman1814
PLK4PLKOther3cokABphosphoaminophosphonic acid-adenylate esterHuman1818
PLK4PLKOther3cokBAphosphoaminophosphonic acid-adenylate esterHuman1815
PLK4PLKOther3cokBBphosphoaminophosphonic acid-adenylate esterHuman1817
PLK4PLKOther4jxfA(1r,2s)-2-{3-[(e)-2-{4-[(dimethylamino)methyl]phenyl}ethenyl]-2h-indazol-6-yl}-5'-methoxyspiro[cyclopropane-1,3'-indol]-2'(1'h)-oneHuman1816
PLK4PLKOther4yurA2-({2-fluoro-4-[(2-fluoro-3-nitrobenzyl)sulfonyl]phenyl}sulfanyl)-5-methoxy-n-(3-methyl-1h-pyrazol-5-yl)-6-(morpholin-4-yl)pyrimidin-4-amineHuman1813
Pomk (SGK196)Other-UniqueOther5gz8A-Mouse8033
Pomk (SGK196)Other-UniqueOther5gz9Aphosphoaminophosphonic acid-adenylate esterMouse8034
PRAG1 (SgK223)NKF3Other5ve6A-Human8573
Prkaa1 (AMPKa1)CAMKLCAMK5ufuAstaurosporineMouse7590
PRKAA1 (AMPKa1)CAMKLCAMK4redA-Human122
PRKAA1 (AMPKa1)CAMKLCAMK4redB-Human123
PRKAA1 (AMPKa1)CAMKLCAMK4rerAstaurosporineHuman121
PRKAA1 (AMPKa1)CAMKLCAMK4rewAstaurosporineHuman124
PRKAA1 (AMPKa1)CAMKLCAMK6c9fAstaurosporineHuman10716
PRKAA1 (AMPKa1)CAMKLCAMK6c9gAstaurosporineHuman10715
PRKAA1 (AMPKa1)CAMKLCAMK6c9hAstaurosporineHuman10714
PRKAA1 (AMPKa1)CAMKLCAMK6c9jAstaurosporineHuman10717
PRKAA1 (AMPKa1)CAMKLCAMK7jhgA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman13816
PRKAA1 (AMPKa1)CAMKLCAMK7jhhA-Human13817
PRKAA1 (AMPKa1)CAMKLCAMK7jijB-Human13819
PRKAA1 (AMPKa1)CAMKLCAMK7m74A6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman14017
PRKAA2 (AMPKa2)CAMKLCAMK2h6dAA-Human196
PRKAA2 (AMPKa2)CAMKLCAMK2h6dAB-Human194
PRKAA2 (AMPKa2)CAMKLCAMK2yzaA-Human189
PRKAA2 (AMPKa2)CAMKLCAMK3aqvA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman193
PRKAA2 (AMPKa2)CAMKLCAMK4cfeAstaurosporineHuman195
PRKAA2 (AMPKa2)CAMKLCAMK4cfeCstaurosporineHuman192
PRKAA2 (AMPKa2)CAMKLCAMK4cffAstaurosporineHuman191
PRKAA2 (AMPKa2)CAMKLCAMK4cffCstaurosporineHuman190
PRKAA2 (AMPKa2)CAMKLCAMK4zhxAA(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6425
PRKAA2 (AMPKa2)CAMKLCAMK4zhxAB(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6429
PRKAA2 (AMPKa2)CAMKLCAMK4zhxCA(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6427
PRKAA2 (AMPKa2)CAMKLCAMK4zhxCB(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6423
PRKAA2 (AMPKa2)CAMKLCAMK5ezvAAstaurosporineHuman6424
PRKAA2 (AMPKa2)CAMKLCAMK5ezvABstaurosporineHuman6428
PRKAA2 (AMPKa2)CAMKLCAMK5ezvCAstaurosporineHuman6430
PRKAA2 (AMPKa2)CAMKLCAMK5ezvCBstaurosporineHuman6426
PRKAA2 (AMPKa2)CAMKLCAMK5isoAstaurosporineHuman7981
PRKAA2 (AMPKa2)CAMKLCAMK5isoCstaurosporineHuman7980
PRKAA2 (AMPKa2)CAMKLCAMK6b1uAAstaurosporineHuman9848
PRKAA2 (AMPKa2)CAMKLCAMK6b1uABstaurosporineHuman9849
PRKAA2 (AMPKa2)CAMKLCAMK6b1uCAstaurosporineHuman9847
PRKAA2 (AMPKa2)CAMKLCAMK6b1uCBstaurosporineHuman9850
PRKAA2 (AMPKa2)CAMKLCAMK6b2eAstaurosporineHuman9851
PRKAA2 (AMPKa2)CAMKLCAMK6bx6AA2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman9878
PRKAA2 (AMPKa2)CAMKLCAMK6bx6AB2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman9877
PRKAA2 (AMPKa2)CAMKLCAMK7myjA(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman14273
Prkaca (PKACa)PKAAGC1apmEA-Mouse5972
Prkaca (PKACa)PKAAGC1apmEB-Mouse5949
Prkaca (PKACa)PKAAGC1atpEadenosine-5'-triphosphateMouse5902
Prkaca (PKACa)PKAAGC1bkxAadenosine-5'-monophosphateMouse5957
Prkaca (PKACa)PKAAGC1bx6AbalanolMouse5955
Prkaca (PKACa)PKAAGC1fmoEadenosineMouse5932
Prkaca (PKACa)PKAAGC1j3hA-Mouse5926
Prkaca (PKACa)PKAAGC1j3hB-Mouse5873
Prkaca (PKACa)PKAAGC1jbpEadenosine-5'-diphosphateMouse5914
Prkaca (PKACa)PKAAGC1jluE-Mouse5924
Prkaca (PKACa)PKAAGC1l3rEadenosine-5'-diphosphateMouse5950
Prkaca (PKACa)PKAAGC1rdqEAadenosine-5'-diphosphateMouse5964
Prkaca (PKACa)PKAAGC1rdqEBadenosine-5'-triphosphateMouse5927
Prkaca (PKACa)PKAAGC1re8A3-[(4-hydroxybenzoyl)amino]azepan-4-yl 4-(2-hydroxybenzoyl)benzoateMouse5923
Prkaca (PKACa)PKAAGC1rejA3-[(4-hydroxybenzoyl)amino]azepan-4-yl 4-hydroxybenzoateMouse5931
Prkaca (PKACa)PKAAGC1rekA3-[(3-sec-butyl-4-hydroxybenzoyl)amino]azepan-4-yl 4-(2-hydroxy-5-methoxybenzoyl)benzoateMouse5969
Prkaca (PKACa)PKAAGC1sykA-Mouse5891
Prkaca (PKACa)PKAAGC1sykB-Mouse5948
Prkaca (PKACa)PKAAGC2cpkE-Mouse5959
Prkaca (PKACa)PKAAGC2erzE1-(1-hydroxy-5-isoquinolinesulfonyl)homopiperazineMouse5895
Prkaca (PKACa)PKAAGC2qcsAAphosphoaminophosphonic acid-adenylate esterMouse5945
Prkaca (PKACa)PKAAGC2qcsABphosphoaminophosphonic acid-adenylate esterMouse5956
Prkaca (PKACa)PKAAGC2qurA-Mouse5896
Prkaca (PKACa)PKAAGC2qvsE-Mouse5922
Prkaca (PKACa)PKAAGC3fhiAphosphoaminophosphonic acid-adenylate esterMouse5951
Prkaca (PKACa)PKAAGC3fjqEadenosine-5'-triphosphateMouse5875
Prkaca (PKACa)PKAAGC3idbAphosphoaminophosphonic acid-adenylate esterMouse5939
Prkaca (PKACa)PKAAGC3idcAphosphoaminophosphonic acid-adenylate esterMouse5933
Prkaca (PKACa)PKAAGC3j4qDA-Mouse5888
Prkaca (PKACa)PKAAGC3j4qDB-Mouse5943
Prkaca (PKACa)PKAAGC3j4qEA-Mouse5937
Prkaca (PKACa)PKAAGC3j4qEB-Mouse5913
Prkaca (PKACa)PKAAGC3j4rDA-Mouse5928
Prkaca (PKACa)PKAAGC3j4rDB-Mouse5967
Prkaca (PKACa)PKAAGC3j4rEA-Mouse5877
Prkaca (PKACa)PKAAGC3j4rEB-Mouse5940
Prkaca (PKACa)PKAAGC3o7lBphosphoaminophosphonic acid-adenylate esterMouse5908
Prkaca (PKACa)PKAAGC3o7lD-Mouse5958
Prkaca (PKACa)PKAAGC3ow3A(2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amineMouse5941
Prkaca (PKACa)PKAAGC3pvbAphosphoaminophosphonic acid-adenylate esterMouse5880
Prkaca (PKACa)PKAAGC3qalEadenosine-5'-triphosphateMouse5921
Prkaca (PKACa)PKAAGC3qamEadenosine-5'-triphosphateMouse5906
Prkaca (PKACa)PKAAGC3tnpC-Mouse5889
Prkaca (PKACa)PKAAGC3tnpF-Mouse5893
Prkaca (PKACa)PKAAGC3x2uAAadenosine-5'-triphosphateMouse6294
Prkaca (PKACa)PKAAGC3x2uABadenosine-5'-triphosphateMouse6298
Prkaca (PKACa)PKAAGC3x2vAAadenosine-5'-triphosphateMouse6299
Prkaca (PKACa)PKAAGC3x2vABadenosine-5'-triphosphateMouse6297
Prkaca (PKACa)PKAAGC3x2wAAadenosine-5'-triphosphateMouse6296
Prkaca (PKACa)PKAAGC3x2wABadenosine-5'-triphosphateMouse6295
Prkaca (PKACa)PKAAGC4dfxEAphosphoaminophosphonic acid-adenylate esterMouse5925
Prkaca (PKACa)PKAAGC4dfxEBphosphoaminophosphonic acid-adenylate esterMouse5885
Prkaca (PKACa)PKAAGC4dfyA-Mouse5886
Prkaca (PKACa)PKAAGC4dfyE-Mouse5960
Prkaca (PKACa)PKAAGC4dfzEA-Mouse5874
Prkaca (PKACa)PKAAGC4dfzEB-Mouse5966
Prkaca (PKACa)PKAAGC4dfzEC-Mouse5971
Prkaca (PKACa)PKAAGC4dg0EAphosphoaminophosphonic acid-adenylate esterMouse5929
Prkaca (PKACa)PKAAGC4dg0EBphosphoaminophosphonic acid-adenylate esterMouse5892
Prkaca (PKACa)PKAAGC4dg2EA-Mouse5952
Prkaca (PKACa)PKAAGC4dg2EB-Mouse5962
Prkaca (PKACa)PKAAGC4dg3Ephosphoaminophosphonic acid-adenylate esterMouse5898
Prkaca (PKACa)PKAAGC4dh1Aadenosine-5'-triphosphateMouse5907
Prkaca (PKACa)PKAAGC4dh3Aadenosine-5'-triphosphateMouse5965
Prkaca (PKACa)PKAAGC4dh5Aadenosine-5'-diphosphateMouse5917
Prkaca (PKACa)PKAAGC4dh7Aphosphoaminophosphonic acid-adenylate esterMouse5934
Prkaca (PKACa)PKAAGC4dh8Aphosphoaminophosphonic acid-adenylate esterMouse5904
Prkaca (PKACa)PKAAGC4dinAadenosine-5'-triphosphateMouse5919
Prkaca (PKACa)PKAAGC4hptEAphosphoaminophosphonic acid-adenylate esterMouse5899
Prkaca (PKACa)PKAAGC4hptEBphosphoaminophosphonic acid-adenylate esterMouse5884
Prkaca (PKACa)PKAAGC4hpuEAphosphoaminophosphonic acid-adenylate esterMouse5963
Prkaca (PKACa)PKAAGC4hpuEB-Mouse5882
Prkaca (PKACa)PKAAGC4iacAphosphomethylphosphonic acid adenylate esterMouse5936
Prkaca (PKACa)PKAAGC4iadAadenosine-5'-diphosphateMouse5883
Prkaca (PKACa)PKAAGC4iafAadenosine-5'-diphosphateMouse5876
Prkaca (PKACa)PKAAGC4iaiAAadenosine-5'-diphosphateMouse5881
Prkaca (PKACa)PKAAGC4iaiABadenosine-5'-diphosphateMouse5901
Prkaca (PKACa)PKAAGC4iaiACadenosine-5'-diphosphateMouse5912
Prkaca (PKACa)PKAAGC4iakAAadenosine-5'-diphosphateMouse5903
Prkaca (PKACa)PKAAGC4iakABadenosine-5'-diphosphateMouse5918
Prkaca (PKACa)PKAAGC4iayAadenosine-5'-diphosphateMouse5911
Prkaca (PKACa)PKAAGC4iazAAadenosine-5'-diphosphateMouse5900
Prkaca (PKACa)PKAAGC4iazABadenosine-5'-diphosphateMouse5938
Prkaca (PKACa)PKAAGC4ib0AAadenosine-5'-diphosphateMouse5947
Prkaca (PKACa)PKAAGC4ib0ABadenosine-5'-diphosphateMouse5910
Prkaca (PKACa)PKAAGC4ib1AAadenosine-5'-diphosphateMouse5968
Prkaca (PKACa)PKAAGC4ib1ABadenosine-5'-diphosphateMouse5961
Prkaca (PKACa)PKAAGC4ib3Aadenosine-5'-diphosphateMouse5944
Prkaca (PKACa)PKAAGC4ntsA-Mouse5920
Prkaca (PKACa)PKAAGC4ntsB-Mouse5879
Prkaca (PKACa)PKAAGC4nttAadenosine-5'-diphosphateMouse5942
Prkaca (PKACa)PKAAGC4nttBadenosine-5'-diphosphateMouse5905
Prkaca (PKACa)PKAAGC4o21AAadenosine-5'-diphosphateMouse5954
Prkaca (PKACa)PKAAGC4o21ABadenosine-5'-diphosphateMouse5909
Prkaca (PKACa)PKAAGC4o22AA-Mouse5953
Prkaca (PKACa)PKAAGC4o22AB-Mouse5970
Prkaca (PKACa)PKAAGC4wbbB-Mouse5930
Prkaca (PKACa)PKAAGC4x6qC-Mouse5916
Prkaca (PKACa)PKAAGC4x6rAAadenosine-5'-triphosphateMouse5897
Prkaca (PKACa)PKAAGC4x6rABadenosine-5'-triphosphateMouse5887
Prkaca (PKACa)PKAAGC4xw4AAphosphoaminophosphonic acid-adenylate esterMouse5946
Prkaca (PKACa)PKAAGC4xw4ABphosphoaminophosphonic acid-adenylate esterMouse5935
Prkaca (PKACa)PKAAGC4xw5AAadenosine-5'-triphosphateMouse5890
Prkaca (PKACa)PKAAGC4xw5ABadenosine-5'-triphosphateMouse5894
Prkaca (PKACa)PKAAGC4xw6AAadenosine-5'-diphosphateMouse5878
Prkaca (PKACa)PKAAGC4xw6ABadenosine-5'-diphosphateMouse5915
Prkaca (PKACa)PKAAGC5jr7Aadenosine-5'-diphosphateMouse7509
Prkaca (PKACa)PKAAGC5jr7Cadenosine-5'-diphosphateMouse7510
Prkaca (PKACa)PKAAGC5x3fB-Mouse8191
Prkaca (PKACa)PKAAGC6e21AAadenosine-5'-diphosphateMouse11316
Prkaca (PKACa)PKAAGC6e21ABadenosine-5'-diphosphateMouse11323
Prkaca (PKACa)PKAAGC6mm5EA-Mouse11319
Prkaca (PKACa)PKAAGC6mm5EBphosphoaminophosphonic acid-adenylate esterMouse11315
Prkaca (PKACa)PKAAGC6mm6CA-Mouse11326
Prkaca (PKACa)PKAAGC6mm6CBphosphoaminophosphonic acid-adenylate esterMouse11310
Prkaca (PKACa)PKAAGC6mm6CCphosphoaminophosphonic acid-adenylate esterMouse11321
Prkaca (PKACa)PKAAGC6mm6EA-Mouse11311
Prkaca (PKACa)PKAAGC6mm6EBphosphoaminophosphonic acid-adenylate esterMouse11314
Prkaca (PKACa)PKAAGC6mm6ECphosphoaminophosphonic acid-adenylate esterMouse11320
Prkaca (PKACa)PKAAGC6mm7AA-Mouse11325
Prkaca (PKACa)PKAAGC6mm7ABphosphoaminophosphonic acid-adenylate esterMouse11322
Prkaca (PKACa)PKAAGC6mm7DA-Mouse11312
Prkaca (PKACa)PKAAGC6mm7DBphosphoaminophosphonic acid-adenylate esterMouse11318
Prkaca (PKACa)PKAAGC6mm8CA-Mouse11317
Prkaca (PKACa)PKAAGC6mm8CBphosphoaminophosphonic acid-adenylate esterMouse11324
Prkaca (PKACa)PKAAGC6mm8CCphosphoaminophosphonic acid-adenylate esterMouse11313
Prkaca (PKACa)PKAAGC7e0zAphosphoaminophosphonic acid-adenylate esterMouse14205
Prkaca (PKACa)PKAAGC7e11Aphosphoaminophosphonic acid-adenylate esterMouse14206
PRKACA (PKACa)PKAAGC2gu8An-[(1s)-2-amino-1-(2,4-dichlorobenzyl)ethyl]-5-[2-(methylamino)pyrimidin-4-yl]thiophene-2-carboxamideHuman5295
PRKACA (PKACa)PKAAGC3aglA(10r,20r,23r)-1-[(2s,3s,4r,5r)-5-(6-amino-9h-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]-20,23-bis(3-carbamimidamidopropyl)-10-methyl-1,8,11,18,21-pentaoxo-2,9,12,19,22-pentaazatetracosan-24-amideHuman5267
PRKACA (PKACa)PKAAGC3aglB(10r,20r,23r)-1-[(2s,3s,4r,5r)-5-(6-amino-9h-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]-20,23-bis(3-carbamimidamidopropyl)-10-methyl-1,8,11,18,21-pentaoxo-2,9,12,19,22-pentaazatetracosan-24-amideHuman5283
PRKACA (PKACa)PKAAGC3agmA-Human5282
PRKACA (PKACa)PKAAGC3amaA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman5284
PRKACA (PKACa)PKAAGC3ambAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman5276
PRKACA (PKACa)PKAAGC3l9lA5-[2-({(2s)-2-amino-3-[4-(trifluoromethyl)phenyl]propyl}amino)-1,3-thiazol-5-yl]-1,3-dihydro-2h-indol-2-oneHuman5305
PRKACA (PKACa)PKAAGC3l9lB5-[2-({(2s)-2-amino-3-[4-(trifluoromethyl)phenyl]propyl}amino)-1,3-thiazol-5-yl]-1,3-dihydro-2h-indol-2-oneHuman5302
PRKACA (PKACa)PKAAGC3l9mA(2s)-n~1~-[5-(3-methyl-1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamineHuman5270
PRKACA (PKACa)PKAAGC3l9mB(2s)-n~1~-[5-(3-methyl-1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamineHuman5278
PRKACA (PKACa)PKAAGC3l9nA(2s)-n~1~-[5-(1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamineHuman5292
PRKACA (PKACa)PKAAGC3mvjA(3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amineHuman5289
PRKACA (PKACa)PKAAGC3mvjB-Human5288
PRKACA (PKACa)PKAAGC3mvjE(3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amineHuman5291
PRKACA (PKACa)PKAAGC3nx8AA-Human5277
PRKACA (PKACa)PKAAGC3nx8AB-Human5294
PRKACA (PKACa)PKAAGC3oogAA1-(4-hydroxy-3-methylphenyl)ethanoneHuman5281
PRKACA (PKACa)PKAAGC3oogAB1-(4-hydroxy-3-methylphenyl)ethanoneHuman5272
PRKACA (PKACa)PKAAGC3ovvAAn'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazideHuman5266
PRKACA (PKACa)PKAAGC3ovvABn'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazideHuman5269
PRKACA (PKACa)PKAAGC3owpAA(2s)-2-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylethanehydrazideHuman5273
PRKACA (PKACa)PKAAGC3owpAB(2s)-2-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylethanehydrazideHuman5296
PRKACA (PKACa)PKAAGC3oxtA(2s)-2-amino-n'-[(1e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-phenylethanehydrazideHuman5268
PRKACA (PKACa)PKAAGC3p0mAA(2r)-4-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylbutanehydrazideHuman5297
PRKACA (PKACa)PKAAGC3p0mAB(2r)-4-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylbutanehydrazideHuman5279
PRKACA (PKACa)PKAAGC3pooAAn'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazideHuman5300
PRKACA (PKACa)PKAAGC3pooABn'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazideHuman5285
PRKACA (PKACa)PKAAGC3vqhAAn-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamideHuman5271
PRKACA (PKACa)PKAAGC3vqhABn-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamideHuman5275
PRKACA (PKACa)PKAAGC4ae6AA-Human5274
PRKACA (PKACa)PKAAGC4ae6AB-Human5301
PRKACA (PKACa)PKAAGC4ae6BA-Human5290
PRKACA (PKACa)PKAAGC4ae6BB-Human5298
PRKACA (PKACa)PKAAGC4ae9AA-Human5265
PRKACA (PKACa)PKAAGC4ae9AB-Human5307
PRKACA (PKACa)PKAAGC4ae9BA-Human5299
PRKACA (PKACa)PKAAGC4ae9BB-Human5286
PRKACA (PKACa)PKAAGC4uj1A7-[(3s,4r)-4-(3-chlorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6548
PRKACA (PKACa)PKAAGC4uj2AA7-[(3s,4r)-4-(3-iodanylphenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6550
PRKACA (PKACa)PKAAGC4uj2AB7-[(3s,4r)-4-(3-iodanylphenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6551
PRKACA (PKACa)PKAAGC4uj9A7-[(3s,4r)-4-[4-(trifluoromethyl)phenyl]carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6544
PRKACA (PKACa)PKAAGC4ujaAA7-{(3s,4r)-4-[(5-bromothiophen-2-yl)carbonyl]pyrrolidin-3-yl}quinazolin-4(3h)-oneHuman6549
PRKACA (PKACa)PKAAGC4ujaAB7-{(3s,4r)-4-[(5-bromothiophen-2-yl)carbonyl]pyrrolidin-3-yl}quinazolin-4(3h)-oneHuman6547
PRKACA (PKACa)PKAAGC4ujbAA7-[(3s,4r)-4-(3-fluorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6546
PRKACA (PKACa)PKAAGC4ujbAB7-[(3s,4r)-4-(3-fluorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-oneHuman6545
PRKACA (PKACa)PKAAGC4wb5AAadenosine-5'-triphosphateHuman5280
PRKACA (PKACa)PKAAGC4wb5ABadenosine-5'-triphosphateHuman5306
PRKACA (PKACa)PKAAGC4wb6Aadenosine-5'-triphosphateHuman5303
PRKACA (PKACa)PKAAGC4wb6Badenosine-5'-triphosphateHuman5293
PRKACA (PKACa)PKAAGC4wb7AAadenosine-5'-triphosphateHuman6876
PRKACA (PKACa)PKAAGC4wb7ABadenosine-5'-triphosphateHuman6878
PRKACA (PKACa)PKAAGC4wb7BAadenosine-5'-triphosphateHuman6875
PRKACA (PKACa)PKAAGC4wb7BBadenosine-5'-triphosphateHuman6877
PRKACA (PKACa)PKAAGC4wb8AAadenosine-5'-triphosphateHuman5304
PRKACA (PKACa)PKAAGC4wb8ABadenosine-5'-triphosphateHuman5287
PRKACA (PKACa)PKAAGC5bx6AA4-chlorophthalazin-1(2h)-oneHuman7075
PRKACA (PKACa)PKAAGC5bx6AB4-chlorophthalazin-1(2h)-oneHuman7078
PRKACA (PKACa)PKAAGC5bx7AA1-benzothiophen-3-ylmethanolHuman7076
PRKACA (PKACa)PKAAGC5bx7AB1-benzothiophen-3-ylmethanolHuman7077
PRKACA (PKACa)PKAAGC5izfA-Human6854
PRKACA (PKACa)PKAAGC5izjAA-Human6857
PRKACA (PKACa)PKAAGC5izjAB-Human6855
PRKACA (PKACa)PKAAGC5izjBA-Human6851
PRKACA (PKACa)PKAAGC5izjBB-Human6858
PRKACA (PKACa)PKAAGC5j5xAA-Human6853
PRKACA (PKACa)PKAAGC5j5xAB-Human6856
PRKACA (PKACa)PKAAGC5j5xAC-Human6852
PRKACA (PKACa)PKAAGC5n23AA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman9747
PRKACA (PKACa)PKAAGC5n23AB1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman9746
PRKACA (PKACa)PKAAGC5uzkAA2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(1h-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideHuman9726
PRKACA (PKACa)PKAAGC6byrAadenosine-5'-triphosphateHuman11256
PRKACA (PKACa)PKAAGC6byrCadenosine-5'-triphosphateHuman11258
PRKACA (PKACa)PKAAGC6bysA-Human11259
PRKACA (PKACa)PKAAGC6bysC-Human11257
PRKACA (PKACa)PKAAGC6bysE-Human11262
PRKACA (PKACa)PKAAGC6bysG-Human11260
PRKACA (PKACa)PKAAGC6c0uAn-[(3r,4r)-4-{[4-(2-fluoro-3-methoxy-6-propoxybenzene-1-carbonyl)benzene-1-carbonyl]amino}pyrrolidin-3-yl]-1h-indazole-5-carboxamideHuman9974
PRKACA (PKACa)PKAAGC6frxA~{n}-[3-[(5-chloranyl-2-phenylazanyl-pyrimidin-4-yl)amino]phenyl]prop-2-enamideHuman11261
PRKACA (PKACa)PKAAGC6no7A-Human11465
PRKACA (PKACa)PKAAGC6no7C-Human11466
PRKACA (PKACa)PKAAGC6no7Eadenosine-5'-triphosphateHuman11463
PRKACA (PKACa)PKAAGC6no7Gadenosine-5'-triphosphateHuman11464
PRKACA (PKACa)PKAAGC6qj7AA~{n}'-[(2~{s})-2-[3,5-bis(fluoranyl)phenyl]-2-oxidanyl-ethanoyl]-2-ethyl-3-methyl-4-oxidanyl-benzohydrazideHuman11990
PRKACA (PKACa)PKAAGC6qj7AB~{n}'-[(2~{s})-2-[3,5-bis(fluoranyl)phenyl]-2-oxidanyl-ethanoyl]-2-ethyl-3-methyl-4-oxidanyl-benzohydrazideHuman11991
PRKACA (PKACa)PKAAGC6wjfA-Human13008
PRKACA (PKACa)PKAAGC6wjfB-Human13009
PRKACA (PKACa)PKAAGC6wjgA-Human13006
PRKACA (PKACa)PKAAGC6wjgB-Human13007
PRKACA (PKACa)PKAAGC7y1gAA1-chloranyl-~{n}-[(~{s})-(3-chloranyl-4-cyano-phenyl)-[(2~{r},4~{s})-4-oxidanylpyrrolidin-2-yl]methyl]-7-methoxy-isoquinoline-6-carboxamideHuman14422
PRKACA (PKACa)PKAAGC7y1gAB1-chloranyl-~{n}-[(~{s})-(3-chloranyl-4-cyano-phenyl)-[(2~{r},4~{s})-4-oxidanylpyrrolidin-2-yl]methyl]-7-methoxy-isoquinoline-6-carboxamideHuman14423
PRKACA (PKACa)PKAAGC8fe2A6-[(6m)-6-(1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-9h-purineHuman14889
PRKACA (PKACa)PKAAGC8fe5A6-[(6p)-6-(1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-7,9-dihydro-8h-purin-8-oneHuman14888
PRKACA (PKACa)PKAAGC8fecA6-[(6p)-6-(4-bromo-1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-7h-purineHuman14890
PRKACA (PKACa)PKAAGC8x5lA(2s)-2-(4-chlorophenyl)-2-hydroxy-2-[4-(1h-pyrazol-4-yl)phenyl]ethanaminiumHuman15111
PRKCA (PKCa)PKCAGC3iw4A3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dioneHuman3041
PRKCA (PKCa)PKCAGC3iw4B3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dioneHuman3039
PRKCA (PKCa)PKCAGC3iw4C3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dioneHuman3042
PRKCA (PKCa)PKCAGC4ra4A(1r)-9-[(3s,4s)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman3040
PRKCA (PKCa)PKCAGC8u37AA(6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamideHuman15159
PRKCA (PKCa)PKCAGC8u37AB(6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamideHuman15162
PRKCA (PKCa)PKCAGC8uakAA(6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamideHuman15161
PRKCA (PKCa)PKCAGC8uakAB(6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamideHuman15160
PRKCB (PKCb)PKCAGC2i0eA3-{1-[3-(dimethylamino)propyl]-2-methyl-1h-indol-3-yl}-4-(2-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2550
PRKCB (PKCb)PKCAGC2i0eB3-{1-[3-(dimethylamino)propyl]-2-methyl-1h-indol-3-yl}-4-(2-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2549
PRKCH (PKCh)PKCAGC3txoA2-methyl-n~1~-[3-(pyridin-4-yl)-2,6-naphthyridin-1-yl]propane-1,2-diamineHuman2316
PRKCH (PKCh)PKCAGC8fp1A(3p)-3-[6-chloro-4-(9-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrileHuman14694
PRKCH (PKCh)PKCAGC8fp3AA(3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrileHuman14696
PRKCH (PKCh)PKCAGC8fp3AB(3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrileHuman14695
Prkci (PKCi)PKCAGC4dc2AAadenineMouse5830
Prkci (PKCi)PKCAGC4dc2ABadenineMouse5829
PRKCI (PKCi)PKCAGC1zrzA3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3354
PRKCI (PKCi)PKCAGC3a8wAadenosine-5'-triphosphateHuman3353
PRKCI (PKCi)PKCAGC3a8wBadenosine-5'-triphosphateHuman3346
PRKCI (PKCi)PKCAGC3a8xA-Human3351
PRKCI (PKCi)PKCAGC3a8xB-Human3348
PRKCI (PKCi)PKCAGC3zh8AA(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3349
PRKCI (PKCi)PKCAGC3zh8AB(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3350
PRKCI (PKCi)PKCAGC3zh8BA(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3356
PRKCI (PKCi)PKCAGC3zh8BB(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3347
PRKCI (PKCi)PKCAGC3zh8CA(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3355
PRKCI (PKCi)PKCAGC3zh8CB(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3352
PRKCI (PKCi)PKCAGC5li1AAphosphoaminophosphonic acid-adenylate esterHuman7072
PRKCI (PKCi)PKCAGC5li1ABphosphoaminophosphonic acid-adenylate esterHuman7067
PRKCI (PKCi)PKCAGC5li9AAphosphomethylphosphonic acid adenylate esterHuman7068
PRKCI (PKCi)PKCAGC5li9ABphosphomethylphosphonic acid adenylate esterHuman7074
PRKCI (PKCi)PKCAGC5lihAAadenosine-5'-diphosphateHuman7071
PRKCI (PKCi)PKCAGC5lihABadenosine-5'-diphosphateHuman7070
PRKCI (PKCi)PKCAGC5lihBAadenosine-5'-diphosphateHuman7069
PRKCI (PKCi)PKCAGC5lihBBadenosine-5'-diphosphateHuman7073
PRKCI (PKCi)PKCAGC6ilzA2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamideHuman11358
PRKCI (PKCi)PKCAGC6ilzC2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamideHuman11357
PRKCI (PKCi)PKCAGC6ilzE2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamideHuman11356
PRKCI (PKCi)PKCAGC6ilzG2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamideHuman11355
PRKCQ (PKCt)PKCAGC1xjdAstaurosporineHuman5357
PRKCQ (PKCt)PKCAGC2jedA3-(8-dimethylaminomethyl-6,7,8,9-tetrahydro-pyrido[1,2-a]indol-10-yl)-4-(1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman5352
PRKCQ (PKCt)PKCAGC2jedB3-(8-dimethylaminomethyl-6,7,8,9-tetrahydro-pyrido[1,2-a]indol-10-yl)-4-(1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman5358
PRKCQ (PKCt)PKCAGC4q9zAA(1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5356
PRKCQ (PKCt)PKCAGC4q9zAB(1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5353
PRKCQ (PKCt)PKCAGC4q9zBA(1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5355
PRKCQ (PKCt)PKCAGC4q9zBB(1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5362
PRKCQ (PKCt)PKCAGC4ra5AA(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5354
PRKCQ (PKCt)PKCAGC4ra5AB(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5359
PRKCQ (PKCt)PKCAGC4ra5BA(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5361
PRKCQ (PKCt)PKCAGC4ra5BB(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5360
PRKCQ (PKCt)PKCAGC5f9eAA2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHuman6630
PRKCQ (PKCt)PKCAGC5f9eAB2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHuman6629
PRKCQ (PKCt)PKCAGC5f9eBA2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHuman6631
PRKCQ (PKCt)PKCAGC5f9eBB2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHuman6628
PRKG1 (PKG1)PKGAGC6bdlAA-Human10641
PRKG1 (PKG1)PKGAGC6bdlAB-Human10644
PRKG1 (PKG1)PKGAGC6bdlBA-Human10643
PRKG1 (PKG1)PKGAGC6bdlBB-Human10642
PRKG1 (PKG1)PKGAGC6bg2AAphosphoaminophosphonic acid-adenylate esterHuman10670
PRKG1 (PKG1)PKGAGC6bg2ABphosphoaminophosphonic acid-adenylate esterHuman10667
PRKG1 (PKG1)PKGAGC6bg2BAphosphoaminophosphonic acid-adenylate esterHuman10668
PRKG1 (PKG1)PKGAGC6bg2BBphosphoaminophosphonic acid-adenylate esterHuman10666
PRKG1 (PKG1)PKGAGC6bg2CAphosphoaminophosphonic acid-adenylate esterHuman10669
PRKG1 (PKG1)PKGAGC6bg2CBphosphoaminophosphonic acid-adenylate esterHuman10672
PRKG1 (PKG1)PKGAGC6bg2DAphosphoaminophosphonic acid-adenylate esterHuman10671
PRKG1 (PKG1)PKGAGC6bg2DBphosphoaminophosphonic acid-adenylate esterHuman10665
PRKG1 (PKG1)PKGAGC6c0tAn-[(3r,4r)-4-{[4-(2-fluoro-3-methoxy-6-propoxybenzene-1-carbonyl)benzene-1-carbonyl]amino}pyrrolidin-3-yl]-1h-indazole-5-carboxamideHuman9975
PRKG1 (PKG1)PKGAGC7lv3Aphosphoaminophosphonic acid-adenylate esterHuman14343
PRKG1 (PKG1)PKGAGC7t4tAAadenosine-5'-triphosphateHuman14791
PRKG1 (PKG1)PKGAGC7t4tABadenosine-5'-triphosphateHuman14795
PRKG1 (PKG1)PKGAGC7t4uAA-Human14788
PRKG1 (PKG1)PKGAGC7t4uAB-Human14789
PRKG1 (PKG1)PKGAGC7t4vAA-Human14790
PRKG1 (PKG1)PKGAGC7t4vAB-Human14792
PRKG1 (PKG1)PKGAGC7t4wAA-Human14794
PRKG1 (PKG1)PKGAGC7t4wAB-Human14793
PRPF4B (PRP4)DYRKCMGC4ianA-Human5543
PRPF4B (PRP4)DYRKCMGC4ianB-Human5546
PRPF4B (PRP4)DYRKCMGC4ifcAAadenosine-5'-diphosphateHuman5538
PRPF4B (PRP4)DYRKCMGC4ifcABadenosine-5'-diphosphateHuman5544
PRPF4B (PRP4)DYRKCMGC4ifcBAadenosine-5'-diphosphateHuman5542
PRPF4B (PRP4)DYRKCMGC4ifcBBadenosine-5'-diphosphateHuman5540
PRPF4B (PRP4)DYRKCMGC4iirAAphosphoaminophosphonic acid-adenylate esterHuman5545
PRPF4B (PRP4)DYRKCMGC4iirABphosphoaminophosphonic acid-adenylate esterHuman5539
PRPF4B (PRP4)DYRKCMGC4iirBAphosphoaminophosphonic acid-adenylate esterHuman5536
PRPF4B (PRP4)DYRKCMGC4iirBBphosphoaminophosphonic acid-adenylate esterHuman5537
PRPF4B (PRP4)DYRKCMGC4ijpAA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5547
PRPF4B (PRP4)DYRKCMGC4ijpAB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5535
PRPF4B (PRP4)DYRKCMGC4ijpBA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5541
PRPF4B (PRP4)DYRKCMGC4ijpBB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5534
PRPF4B (PRP4)DYRKCMGC6cnhAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman9776
PRPF4B (PRP4)DYRKCMGC6cnhAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman9775
PRPF4B (PRP4)DYRKCMGC6pjjAA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11585
PRPF4B (PRP4)DYRKCMGC6pjjAB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11577
PRPF4B (PRP4)DYRKCMGC6pjjBA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11583
PRPF4B (PRP4)DYRKCMGC6pjjBB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11581
PRPF4B (PRP4)DYRKCMGC6pjjCA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11578
PRPF4B (PRP4)DYRKCMGC6pjjCB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11586
PRPF4B (PRP4)DYRKCMGC6pjjDA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11580
PRPF4B (PRP4)DYRKCMGC6pjjDB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11579
PRPF4B (PRP4)DYRKCMGC6pk6AA4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11582
PRPF4B (PRP4)DYRKCMGC6pk6AB4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11584
PTK2 (FAK)FAKTK1mp8Aadenosine-5'-diphosphateHuman217
PTK2 (FAK)FAKTK2etmA7-pyridin-2-yl-n-(3,4,5-trimethoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-2-amineHuman246
PTK2 (FAK)FAKTK2etmB7-pyridin-2-yl-n-(3,4,5-trimethoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-2-amineHuman225
PTK2 (FAK)FAKTK2ijmAAadenosine-5'-triphosphateHuman215
PTK2 (FAK)FAKTK2ijmABadenosine-5'-triphosphateHuman243
PTK2 (FAK)FAKTK2ijmBAadenosine-5'-diphosphateHuman220
PTK2 (FAK)FAKTK2ijmBBadenosine-5'-diphosphateHuman249
PTK2 (FAK)FAKTK3bz3AAn-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamideHuman228
PTK2 (FAK)FAKTK3bz3ABn-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamideHuman227
PTK2 (FAK)FAKTK3pxkA6-(4,4-dimethylpent-2-yn-1-yl)-1lambda~4~-pyrrolo[2,3-d][1,3]thiazoleHuman241
PTK2 (FAK)FAKTK3pxkB6-(4,4-dimethylpent-2-yn-1-yl)-1lambda~4~-pyrrolo[2,3-d][1,3]thiazoleHuman236
PTK2 (FAK)FAKTK4ebvAA-Human237
PTK2 (FAK)FAKTK4ebvAB-Human231
PTK2 (FAK)FAKTK4ebvAC-Human224
PTK2 (FAK)FAKTK4ebwAA-Human218
PTK2 (FAK)FAKTK4ebwAB-Human219
PTK2 (FAK)FAKTK4ebwAC-Human235
PTK2 (FAK)FAKTK4gu6AAn-(3-{[(5-cyano-2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)amino]methyl}pyridin-2-yl)-n-methylmethanesulfonamideHuman252
PTK2 (FAK)FAKTK4gu6ABn-(3-{[(5-cyano-2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)amino]methyl}pyridin-2-yl)-n-methylmethanesulfonamideHuman226
PTK2 (FAK)FAKTK4gu6BAn-(3-{[(5-cyano-2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)amino]methyl}pyridin-2-yl)-n-methylmethanesulfonamideHuman240
PTK2 (FAK)FAKTK4gu6BBn-(3-{[(5-cyano-2-phenyl-1h-pyrrolo[2,3-b]pyridin-4-yl)amino]methyl}pyridin-2-yl)-n-methylmethanesulfonamideHuman223
PTK2 (FAK)FAKTK4gu9An-(2-fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman222
PTK2 (FAK)FAKTK4gu9Bn-(2-fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman221
PTK2 (FAK)FAKTK4i4eAA[4-(2-hydroxyethyl)piperidin-1-yl][4-(5-methyl-4,4-dioxido-1,5-dihydropyrazolo[4,3-c][2,1]benzothiazin-8-yl)phenyl]methanoneHuman245
PTK2 (FAK)FAKTK4i4eAB[4-(2-hydroxyethyl)piperidin-1-yl][4-(5-methyl-4,4-dioxido-1,5-dihydropyrazolo[4,3-c][2,1]benzothiazin-8-yl)phenyl]methanoneHuman216
PTK2 (FAK)FAKTK4i4eAC[4-(2-hydroxyethyl)piperidin-1-yl][4-(5-methyl-4,4-dioxido-1,5-dihydropyrazolo[4,3-c][2,1]benzothiazin-8-yl)phenyl]methanoneHuman234
PTK2 (FAK)FAKTK4i4fAA-Human238
PTK2 (FAK)FAKTK4i4fAB-Human251
PTK2 (FAK)FAKTK4i4fAC-Human232
PTK2 (FAK)FAKTK4k8aA3-bromo-5-(2h-tetrazol-5-yl)pyridineHuman244
PTK2 (FAK)FAKTK4k8aB3-bromo-5-(2h-tetrazol-5-yl)pyridineHuman239
PTK2 (FAK)FAKTK4k9yAA1-[4-(6-amino-9h-purin-9-yl)phenyl]-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman230
PTK2 (FAK)FAKTK4k9yAB1-[4-(6-amino-9h-purin-9-yl)phenyl]-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman233
PTK2 (FAK)FAKTK4k9yAC1-[4-(6-amino-9h-purin-9-yl)phenyl]-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman229
PTK2 (FAK)FAKTK4kabA3-methyl-1,5-dihydropyrazolo[4,3-c]pyrazoleHuman242
PTK2 (FAK)FAKTK4kabB3-methyl-1,5-dihydropyrazolo[4,3-c]pyrazoleHuman250
PTK2 (FAK)FAKTK4kaoA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(pyridin-3-yl)phenyl]ureaHuman248
PTK2 (FAK)FAKTK4kaoB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(pyridin-3-yl)phenyl]ureaHuman253
PTK2 (FAK)FAKTK4q9sA3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman247
PTK2 (FAK)FAKTK6i8zA3-methoxy-~{n}-(1-methylpiperidin-1-ium-4-yl)-4-[[4-[(3-oxidanylidene-1,2-dihydroinden-4-yl)oxy]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamideHuman10904
PTK2 (FAK)FAKTK6yojAA6-[[4-[(3-methylsulfonylphenyl)methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3,4-dihydro-1~{h}-quinolin-2-oneHuman13319
PTK2 (FAK)FAKTK6yojAB6-[[4-[(3-methylsulfonylphenyl)methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]-3,4-dihydro-1~{h}-quinolin-2-oneHuman13316
PTK2 (FAK)FAKTK6yq1AA~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13332
PTK2 (FAK)FAKTK6yq1AB~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13327
PTK2 (FAK)FAKTK6yq1BA~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13317
PTK2 (FAK)FAKTK6yq1BB~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13312
PTK2 (FAK)FAKTK6yq1CA~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13315
PTK2 (FAK)FAKTK6yq1CB~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13324
PTK2 (FAK)FAKTK6yq1DA~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13330
PTK2 (FAK)FAKTK6yq1DB~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-3,4-dihydro-1~{h}-quinolin-6-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13333
PTK2 (FAK)FAKTK6yr9AAn-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamideHuman13325
PTK2 (FAK)FAKTK6yr9ABn-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamideHuman13313
PTK2 (FAK)FAKTK6yr9BAn-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamideHuman13326
PTK2 (FAK)FAKTK6yr9BBn-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamideHuman13328
PTK2 (FAK)FAKTK6yr9CAn-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamideHuman13311
PTK2 (FAK)FAKTK6yr9CBn-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamideHuman13334
PTK2 (FAK)FAKTK6yr9DAn-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamideHuman13321
PTK2 (FAK)FAKTK6yr9DBn-methyl-n-(2-{[2-(2-oxo-2,3-dihydro-1h-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-phenyl)-methanesulfonamideHuman13314
PTK2 (FAK)FAKTK6yt6BA~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-1,3-dihydroindol-5-yl)amino]pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13271
PTK2 (FAK)FAKTK6yt6BB~{n}-methyl-~{n}-[3-[[[2-[(2-oxidanylidene-1,3-dihydroindol-5-yl)amino]pyrimidin-4-yl]amino]methyl]pyridin-2-yl]methanesulfonamideHuman13272
PTK2 (FAK)FAKTK6yvsAA5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-oneHuman13323
PTK2 (FAK)FAKTK6yvsAB5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-oneHuman13310
PTK2 (FAK)FAKTK6yvsBA5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-oneHuman13335
PTK2 (FAK)FAKTK6yvsBB5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-oneHuman13331
PTK2 (FAK)FAKTK6yvsCA5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-oneHuman13320
PTK2 (FAK)FAKTK6yvsCB5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-oneHuman13307
PTK2 (FAK)FAKTK6yvsDA5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-oneHuman13318
PTK2 (FAK)FAKTK6yvsDB5-[[4-(pyridin-3-ylmethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-1,3-dihydroindol-2-oneHuman13309
PTK2 (FAK)FAKTK6yvyAA4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman13275
PTK2 (FAK)FAKTK6yvyAB4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman13270
PTK2 (FAK)FAKTK6yvyBA4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman13276
PTK2 (FAK)FAKTK6yvyBB4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman13267
PTK2 (FAK)FAKTK6yvyCA4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman13269
PTK2 (FAK)FAKTK6yvyCB4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman13268
PTK2 (FAK)FAKTK6yvyDA4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman13273
PTK2 (FAK)FAKTK6yvyDB4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman13274
PTK2 (FAK)FAKTK6yxvA~{n}-methyl-~{n}-[3-[(~{e})-[2-phenylazanyl-5-(trifluoromethyl)pyrimidin-4-yl]iminomethyl]pyridin-2-yl]methanesulfonamideHuman13336
PTK2 (FAK)FAKTK6yxvB~{n}-methyl-~{n}-[3-[(~{e})-[2-phenylazanyl-5-(trifluoromethyl)pyrimidin-4-yl]iminomethyl]pyridin-2-yl]methanesulfonamideHuman13329
PTK2 (FAK)FAKTK6yxvC~{n}-methyl-~{n}-[3-[(~{e})-[2-phenylazanyl-5-(trifluoromethyl)pyrimidin-4-yl]iminomethyl]pyridin-2-yl]methanesulfonamideHuman13322
PTK2 (FAK)FAKTK6yxvD~{n}-methyl-~{n}-[3-[(~{e})-[2-phenylazanyl-5-(trifluoromethyl)pyrimidin-4-yl]iminomethyl]pyridin-2-yl]methanesulfonamideHuman13308
PTK2 (FAK)FAKTK7pi4DA-Human13913
PTK2 (FAK)FAKTK7pi4DB-Human13914
PTK2B (PYK2)FAKTK3cc6AA-Human93
PTK2B (PYK2)FAKTK3cc6AB-Human92
PTK2B (PYK2)FAKTK3et7A5-{[4-{[2-(pyrrolidin-1-ylsulfonyl)benzyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,3-dihydro-2h-indol-2-oneHuman90
PTK2B (PYK2)FAKTK3fzoA-Human95
PTK2B (PYK2)FAKTK3fzpAphosphothiophosphoric acid-adenylate esterHuman88
PTK2B (PYK2)FAKTK3fzrAn-methyl-n-{2-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]phenyl}methanesulfonamideHuman87
PTK2B (PYK2)FAKTK3fzsA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman94
PTK2B (PYK2)FAKTK3fztA1-[5-tert-butyl-2-(4-methylphenyl)-1,2-dihydro-3h-pyrazol-3-ylidene]-3-{3-[(pyridin-3-yloxy)methyl]-1h-pyrazol-5-yl}ureaHuman86
PTK2B (PYK2)FAKTK3h3cA4-{[4-{[(1r,2r)-2-(dimethylamino)cyclopentyl]amino}-5-(trifluoromethyl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman96
PTK2B (PYK2)FAKTK4h1jA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(4-methoxy-2-methylphenyl)-1h-pyrazol-5-yl]ureaHuman91
PTK2B (PYK2)FAKTK4h1mA7-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)-n-(propan-2-yl)-1h-indole-2-carboxamideHuman89
PTK2B (PYK2)FAKTK5to8A25-(methylsulfonyl)-8-(trifluoromethyl)-5,17,18,21,22,23,24,25-octahydro-12h-7,11-(azeno)-16,13-(metheno)pyrido[3,2-i]pyrrolo[1,2-q][1,3,7,11,17]pentaazacyclohenicosin-20(6h)-oneHuman7316
PTK2B (PYK2)FAKTK5tobAn-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamideHuman8686
PTK2B (PYK2)FAKTK8xoxAAn-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamideHuman15171
PTK2B (PYK2)FAKTK8xoxABn-methyl-n-{3-[({2-[(2-oxo-2,3-dihydro-1h-indol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl}amino)methyl]pyridin-2-yl}methanesulfonamideHuman15172
PTK6 (BRK)SrcTK5d7vAA-Human6953
PTK6 (BRK)SrcTK5d7vAB-Human6950
PTK6 (BRK)SrcTK5d7vBA-Human6955
PTK6 (BRK)SrcTK5d7vBB-Human6951
PTK6 (BRK)SrcTK5d7vCA-Human6949
PTK6 (BRK)SrcTK5d7vCB-Human6954
PTK6 (BRK)SrcTK5d7vDA-Human6948
PTK6 (BRK)SrcTK5d7vDB-Human6952
PTK6 (BRK)SrcTK5da3AA(2-chloro-4-{[6-cyclopropyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanoneHuman6989
PTK6 (BRK)SrcTK5da3AB(2-chloro-4-{[6-cyclopropyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanoneHuman6988
PTK6 (BRK)SrcTK5h2uAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7338
PTK6 (BRK)SrcTK5h2uABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7343
PTK6 (BRK)SrcTK5h2uBAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7339
PTK6 (BRK)SrcTK5h2uBBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7337
PTK6 (BRK)SrcTK5h2uCAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7341
PTK6 (BRK)SrcTK5h2uCBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7342
PTK6 (BRK)SrcTK5h2uDAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7344
PTK6 (BRK)SrcTK5h2uDBn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7340
PTK6 (BRK)SrcTK6cz2AA-Human10030
PTK6 (BRK)SrcTK6cz2AB-Human10031
PTK6 (BRK)SrcTK6cz3AA(3-fluoro-4-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanoneHuman10001
PTK6 (BRK)SrcTK6cz3AB(3-fluoro-4-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanoneHuman9999
PTK6 (BRK)SrcTK6cz4AA2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamideHuman9998
PTK6 (BRK)SrcTK6cz4AB2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamideHuman10000
PTK7 (CCK4)CCK4TK6vg3A-Human12292
PTK7 (CCK4)CCK4TK6vg3B-Human12293
PTK7 (CCK4)CCK4TK6vg3C-Human12291
RAF1RAFTKL3omvA(1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oximeHuman937
RAF1RAFTKL3omvB(1e)-5-(1-piperidin-4-yl-3-pyridin-4-yl-1h-pyrazol-4-yl)-2,3-dihydro-1h-inden-1-one oximeHuman936
RAF1RAFTKL8gaeD-Human14715
RAF1RAFTKL8gftD-Human14725
RETRetTK2ivsAA(3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxideHuman3372
RETRetTK2ivsAB(3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxideHuman3369
RETRetTK2ivsBA(3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxideHuman3357
RETRetTK2ivsBB(3ar,4r,6r,6ar)-4-(6-amino-9h-purin-9-yl)-6-(hydroxymethyl)tetrahydrofuro[3,4-d][1,3,2]dioxaphosphol-2-ol 2-oxideHuman3374
RETRetTK2ivtAAadenosine monophosphateHuman3361
RETRetTK2ivtABadenosine monophosphateHuman3365
RETRetTK2ivuA4-bromo-2-fluoro-n-[(4e)-6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4(1h)-ylidene]anilineHuman3364
RETRetTK2ivvA1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamineHuman3373
RETRetTK2x2kAA(3z)-5-amino-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman3360
RETRetTK2x2kAB(3z)-5-amino-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman3358
RETRetTK2x2lAA(3z)-5-amino-3-[(4-methoxyphenyl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman3363
RETRetTK2x2lAB(3z)-5-amino-3-[(4-methoxyphenyl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman3371
RETRetTK2x2lAC(3z)-5-amino-3-[(4-methoxyphenyl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman3367
RETRetTK2x2mA(3z)-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman3366
RETRetTK2x2mB(3z)-3-[(3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman3375
RETRetTK4ckiAAadenosineHuman3362
RETRetTK4ckiABadenosineHuman3370
RETRetTK4ckiACadenosineHuman3368
RETRetTK4ckjAAadenosineHuman3359
RETRetTK4ckjABadenosineHuman3376
RETRetTK5amnA4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman6412
RETRetTK5fm2A1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamineHuman7328
RETRetTK5fm3A1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamineHuman7327
RETRetTK6fekAAadenosineHuman9604
RETRetTK6fekABadenosineHuman9603
RETRetTK6i82AA~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamineHuman12050
RETRetTK6i82AB~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamineHuman12054
RETRetTK6i82BA~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamineHuman12052
RETRetTK6i82BB~{n}-[3-(1,3-benzodioxol-5-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-~{n}',~{n}'-dimethyl-propane-1,3-diamineHuman12053
RETRetTK6i83A4-[5-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl]benzamideHuman12051
RETRetTK6ne7AAadenosine monophosphateHuman11149
RETRetTK6ne7ABadenosine monophosphateHuman11148
RETRetTK6ne7ACadenosine monophosphateHuman11152
RETRetTK6necAAmethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman11151
RETRetTK6necABmethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman11150
RETRetTK6necCAmethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman11147
RETRetTK6necCBmethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman11153
RETRetTK6njaAAadenineHuman11146
RETRetTK6njaABadenineHuman11145
RETRetTK6vhgAA3-(3,4-dimethoxyphenyl)-n~5~-(1-methylpiperidin-4-yl)-6-phenylpyrazolo[1,5-a]pyrimidine-5,7-diamineHuman11997
RETRetTK6vhgAB3-(3,4-dimethoxyphenyl)-n~5~-(1-methylpiperidin-4-yl)-6-phenylpyrazolo[1,5-a]pyrimidine-5,7-diamineHuman11998
RETRetTK7du8AAselpercatinibHuman14096
RETRetTK7du8ABselpercatinibHuman14095
RETRetTK7du9AApralsetinibHuman14050
RETRetTK7du9ABpralsetinibHuman14047
RETRetTK7duaAA4-azanyl-7-(1-methylcyclopropyl)-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamideHuman14048
RETRetTK7duaAB4-azanyl-7-(1-methylcyclopropyl)-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamideHuman14049
RETRetTK7duaAC4-azanyl-7-(1-methylcyclopropyl)-~{n}-(5-methyl-1~{h}-pyrazol-3-yl)pyrrolo[2,3-d]pyrimidine-5-carboxamideHuman14046
RETRetTK7ju5AApralsetinibHuman13106
RETRetTK7ju5ABpralsetinibHuman13109
RETRetTK7ju5BApralsetinibHuman13105
RETRetTK7ju5BBpralsetinibHuman13108
RETRetTK7ju6AAselpercatinibHuman13103
RETRetTK7ju6ABselpercatinibHuman13107
RETRetTK7ju6BAselpercatinibHuman13110
RETRetTK7ju6BBselpercatinibHuman13104
RETRetTK7nznA2-[4-[[4-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]-6-[(3-methyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]-~{n}-(3-fluorophenyl)ethanamideHuman14105
RETRetTK7runA1-(4-{(1s,3s)-3-[4-amino-5-(3-amino-4-chlorophenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl]cyclobutyl}piperazin-1-yl)ethan-1-oneHuman14072
RIOK1RIOAtypical4otpAadenosine-5'-diphosphateHuman9156
RIOK1RIOAtypical6g5iz-Human10004
RIOK1RIOAtypical6zv6IA-Human13546
RIOK1RIOAtypical6zv6IB-Human13545
RIOK1RIOAtypical6zxdz-Human13013
RIOK1RIOAtypical6zxez-Human13011
RIOK1RIOAtypical6zxfzadenosine-5'-triphosphateHuman13010
RIOK1RIOAtypical6zxgzadenosine-5'-triphosphateHuman13012
RIOK1RIOAtypical6zxhzadenosine-5'-triphosphateHuman13073
RIOK2RIOAtypical6fdmAAphosphoaminophosphonic acid-adenylate esterHuman10875
RIOK2RIOAtypical6fdmABphosphoaminophosphonic acid-adenylate esterHuman10877
RIOK2RIOAtypical6fdmBA-Human10869
RIOK2RIOAtypical6fdmBB-Human10871
RIOK2RIOAtypical6fdmCAphosphoaminophosphonic acid-adenylate esterHuman10874
RIOK2RIOAtypical6fdmCBphosphoaminophosphonic acid-adenylate esterHuman10876
RIOK2RIOAtypical6fdmDA-Human10868
RIOK2RIOAtypical6fdmDB-Human10872
RIOK2RIOAtypical6fdnA-Human10873
RIOK2RIOAtypical6fdnB-Human10867
RIOK2RIOAtypical6fdoA-Human10878
RIOK2RIOAtypical6fdoB-Human10870
RIOK2RIOAtypical6g18v-Human9986
RIOK2RIOAtypical6g51v-Human9985
RIOK2RIOAtypical6hk6A2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10638
RIOK2RIOAtypical6hk6B2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10636
RIOK2RIOAtypical6hk6C2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10639
RIOK2RIOAtypical6hk6D2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10634
RIOK2RIOAtypical6hk6E2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10633
RIOK2RIOAtypical6hk6F2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10637
RIOK2RIOAtypical6hk6G2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10640
RIOK2RIOAtypical6hk6H2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10632
RIOK2RIOAtypical6hk6I2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10631
RIOK2RIOAtypical6hk6J2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10635
RIOK2RIOAtypical7vbtA8-(6-methoxypyridin-3-yl)-1-[4-piperazin-1-yl-3-(trifluoromethyl)phenyl]-5h-[1,2,3]triazolo[4,5-c]quinolin-4-oneHuman14274
RIPK1RIPKTKL4ithAA(5r)-5-[(7-chloro-1h-indol-3-yl)methyl]-3-methylimidazolidine-2,4-dioneHuman566
RIPK1RIPKTKL4ithAB(5r)-5-[(7-chloro-1h-indol-3-yl)methyl]-3-methylimidazolidine-2,4-dioneHuman567
RIPK1RIPKTKL4ithBA(5r)-5-[(7-chloro-1h-indol-3-yl)methyl]-3-methylimidazolidine-2,4-dioneHuman564
RIPK1RIPKTKL4ithBB(5r)-5-[(7-chloro-1h-indol-3-yl)methyl]-3-methylimidazolidine-2,4-dioneHuman571
RIPK1RIPKTKL4itiAA1-{(3s,3as)-3-[3-fluoro-4-(trifluoromethoxy)phenyl]-8-methoxy-3,3a,4,5-tetrahydro-2h-benzo[g]indazol-2-yl}-2-hydroxyethanoneHuman570
RIPK1RIPKTKL4itiAB1-{(3s,3as)-3-[3-fluoro-4-(trifluoromethoxy)phenyl]-8-methoxy-3,3a,4,5-tetrahydro-2h-benzo[g]indazol-2-yl}-2-hydroxyethanoneHuman563
RIPK1RIPKTKL4itiBA1-{(3s,3as)-3-[3-fluoro-4-(trifluoromethoxy)phenyl]-8-methoxy-3,3a,4,5-tetrahydro-2h-benzo[g]indazol-2-yl}-2-hydroxyethanoneHuman562
RIPK1RIPKTKL4itiBB1-{(3s,3as)-3-[3-fluoro-4-(trifluoromethoxy)phenyl]-8-methoxy-3,3a,4,5-tetrahydro-2h-benzo[g]indazol-2-yl}-2-hydroxyethanoneHuman569
RIPK1RIPKTKL4itjAAn-[(1s)-1-(2-chloro-6-fluorophenyl)ethyl]-5-cyano-1-methyl-1h-pyrrole-2-carboxamideHuman575
RIPK1RIPKTKL4itjABn-[(1s)-1-(2-chloro-6-fluorophenyl)ethyl]-5-cyano-1-methyl-1h-pyrrole-2-carboxamideHuman572
RIPK1RIPKTKL4itjBAn-[(1s)-1-(2-chloro-6-fluorophenyl)ethyl]-5-cyano-1-methyl-1h-pyrrole-2-carboxamideHuman565
RIPK1RIPKTKL4itjBBn-[(1s)-1-(2-chloro-6-fluorophenyl)ethyl]-5-cyano-1-methyl-1h-pyrrole-2-carboxamideHuman574
RIPK1RIPKTKL4neuAA1-[4-(1-aminoisoquinolin-5-yl)phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)ureaHuman576
RIPK1RIPKTKL4neuAB1-[4-(1-aminoisoquinolin-5-yl)phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)ureaHuman561
RIPK1RIPKTKL4neuBA1-[4-(1-aminoisoquinolin-5-yl)phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)ureaHuman568
RIPK1RIPKTKL4neuBB1-[4-(1-aminoisoquinolin-5-yl)phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)ureaHuman573
RIPK1RIPKTKL5hx6A5-benzyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-1,2-oxazole-3-carboxamideHuman6417
RIPK1RIPKTKL5hx6B5-benzyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-1,2-oxazole-3-carboxamideHuman6418
RIPK1RIPKTKL5tx5AAgsk2982772Human8214
RIPK1RIPKTKL5tx5ABgsk2982772Human8217
RIPK1RIPKTKL5tx5BAgsk2982772Human8216
RIPK1RIPKTKL5tx5BBgsk2982772Human8215
RIPK1RIPKTKL6c3eAA2-benzyl-5-nitro-1h-benzimidazoleHuman9750
RIPK1RIPKTKL6c3eAB2-benzyl-5-nitro-1h-benzimidazoleHuman9751
RIPK1RIPKTKL6c3eBA2-benzyl-5-nitro-1h-benzimidazoleHuman9755
RIPK1RIPKTKL6c3eBB2-benzyl-5-nitro-1h-benzimidazoleHuman9757
RIPK1RIPKTKL6c4dA(3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrileHuman9754
RIPK1RIPKTKL6c4dB(3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrileHuman9752
RIPK1RIPKTKL6c4dC(3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrileHuman9756
RIPK1RIPKTKL6c4dD(3s)-3-(2-benzyl-3-chloro-7-oxo-2,4,5,7-tetrahydro-6h-pyrazolo[3,4-c]pyridin-6-yl)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepine-8-carbonitrileHuman9753
RIPK1RIPKTKL6hhoA6-[4-[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]carbonylpiperidin-1-yl]pyrimidine-4-carbonitrileHuman10783
RIPK1RIPKTKL6hhoB6-[4-[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]carbonylpiperidin-1-yl]pyrimidine-4-carbonitrileHuman10784
RIPK1RIPKTKL6nw2AA(5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman11040
RIPK1RIPKTKL6nw2AB(5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman11041
RIPK1RIPKTKL6nw2BA(5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman11039
RIPK1RIPKTKL6nw2BB(5r)-5-methyl-n-[(3s)-5-methyl-4-oxo-2,3,4,5-tetrahydro-1,5-benzoxazepin-3-yl]-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman11043
RIPK1RIPKTKL6nyhA(5s)-n-[(3s)-7-methoxy-1-methyl-2-oxo-2,3,4,5-tetrahydro-1h-pyrido[3,4-b]azepin-3-yl]-5-phenyl-6,7-dihydro-5h-pyrrolo[1,2-b][1,2,4]triazole-2-carboxamideHuman11057
RIPK1RIPKTKL6nyhB(5s)-n-[(3s)-7-methoxy-1-methyl-2-oxo-2,3,4,5-tetrahydro-1h-pyrido[3,4-b]azepin-3-yl]-5-phenyl-6,7-dihydro-5h-pyrrolo[1,2-b][1,2,4]triazole-2-carboxamideHuman11056
RIPK1RIPKTKL6ocqAA1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-oneHuman11046
RIPK1RIPKTKL6ocqAB1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-oneHuman11047
RIPK1RIPKTKL6ocqBA1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-oneHuman11048
RIPK1RIPKTKL6ocqBB1-[(2s)-2-(3-fluorophenyl)pyrrolidin-1-yl]-2,2-dimethylpropan-1-oneHuman11045
RIPK1RIPKTKL6r5fA[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanoneHuman11038
RIPK1RIPKTKL6r5fB[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanoneHuman11044
RIPK1RIPKTKL6r5fC[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanoneHuman11042
RIPK1RIPKTKL6r5fD[(5~{s})-5-[3,5-bis(fluoranyl)phenyl]pyrazolidin-1-yl]-[1-(5-methyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]methanoneHuman11037
RIPK1RIPKTKL6rlnA~{n}-[(3~{s})-7,9-bis(fluoranyl)-2-oxidanylidene-1,3,4,5-tetrahydro-1-benzazepin-3-yl]-3-(phenylmethyl)-1~{h}-1,2,4-triazole-5-carboxamideHuman11383
RIPK1RIPKTKL6rlnB~{n}-[(3~{s})-7,9-bis(fluoranyl)-2-oxidanylidene-1,3,4,5-tetrahydro-1-benzazepin-3-yl]-3-(phenylmethyl)-1~{h}-1,2,4-triazole-5-carboxamideHuman11382
RIPK1RIPKTKL7fczAn-[(3s)-7-(2-cyclopropylethynyl)-5-methyl-4-oxidanylidene-2,3-dihydro-1,5-benzoxazepin-3-yl]-5-(phenylmethyl)-4h-1,2,4-triazole-3-carboxamideHuman14071
RIPK1RIPKTKL7fd0An-[(3s)-5-methyl-7-[2-(oxan-4-yl)ethynyl]-4-oxidanylidene-2,3-dihydro-1,5-benzoxazepin-3-yl]-5-(phenylmethyl)-4h-1,2,4-triazole-3-carboxamideHuman14070
RIPK1RIPKTKL7xmkA5-[2-(cyclopropylcarbonylamino)-[1,2,4]triazolo[1,5-a]pyridin-7-yl]-n-[(1s)-1-(3-fluorophenyl)ethyl]-1-methyl-indole-3-carboxamideHuman14716
RIPK1RIPKTKL7ydxAA1-methyl-5-[2-(2-methylpropanoylamino)-[1,2,4]triazolo[1,5-a]pyridin-7-yl]-n-[(1s)-1-phenylethyl]indole-3-carboxamideHuman14711
RIPK1RIPKTKL7ydxAB1-methyl-5-[2-(2-methylpropanoylamino)-[1,2,4]triazolo[1,5-a]pyridin-7-yl]-n-[(1s)-1-phenylethyl]indole-3-carboxamideHuman14710
RIPK1RIPKTKL8i2nA~{n}-methyl-1-[4-[[[1-methyl-5-(phenylmethyl)pyrazol-3-yl]carbonylamino]methyl]phenyl]benzimidazole-5-carboxamideHuman15186
RIPK2RIPKTKL4c8bA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman1254
RIPK2RIPKTKL4c8bB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman1253
RIPK2RIPKTKL5ar2AA-Human6183
RIPK2RIPKTKL5ar2AB-Human6173
RIPK2RIPKTKL5ar2BA-Human6185
RIPK2RIPKTKL5ar2BB-Human6181
RIPK2RIPKTKL5ar3AAphosphomethylphosphonic acid adenylate esterHuman6184
RIPK2RIPKTKL5ar3ABphosphomethylphosphonic acid adenylate esterHuman6186
RIPK2RIPKTKL5ar3BAphosphomethylphosphonic acid adenylate esterHuman6177
RIPK2RIPKTKL5ar3BBphosphomethylphosphonic acid adenylate esterHuman6190
RIPK2RIPKTKL5ar4A4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman6180
RIPK2RIPKTKL5ar4B4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman6187
RIPK2RIPKTKL5ar5AA2-(2-(4-chlorophenyl)-1h-imidazol-5-yl)-n,1-bis(2-methoxyethyl)-1h-benzo[d]imidazole-5-carboxamideHuman6189
RIPK2RIPKTKL5ar5AB2-(2-(4-chlorophenyl)-1h-imidazol-5-yl)-n,1-bis(2-methoxyethyl)-1h-benzo[d]imidazole-5-carboxamideHuman6175
RIPK2RIPKTKL5ar5BA2-(2-(4-chlorophenyl)-1h-imidazol-5-yl)-n,1-bis(2-methoxyethyl)-1h-benzo[d]imidazole-5-carboxamideHuman6171
RIPK2RIPKTKL5ar5BB2-(2-(4-chlorophenyl)-1h-imidazol-5-yl)-n,1-bis(2-methoxyethyl)-1h-benzo[d]imidazole-5-carboxamideHuman6172
RIPK2RIPKTKL5ar7AA1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-pyridin-4-yloxyphenyl)ureaHuman6174
RIPK2RIPKTKL5ar7AB1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-pyridin-4-yloxyphenyl)ureaHuman6182
RIPK2RIPKTKL5ar7BA1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-pyridin-4-yloxyphenyl)ureaHuman6178
RIPK2RIPKTKL5ar7BB1-(5-tert-butyl-1,2-oxazol-3-yl)-3-(4-pyridin-4-yloxyphenyl)ureaHuman6188
RIPK2RIPKTKL5ar8A2,6-bis(fluoranyl)-n-[3-[5-[2-[(3-methylsulfonylphenyl)amino]pyrimidin-4-yl]-2-morpholin-4-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamideHuman6176
RIPK2RIPKTKL5ar8B2,6-bis(fluoranyl)-n-[3-[5-[2-[(3-methylsulfonylphenyl)amino]pyrimidin-4-yl]-2-morpholin-4-yl-1,3-thiazol-4-yl]phenyl]benzenesulfonamideHuman6179
RIPK2RIPKTKL5j79AA4-methyl-3-{[6-(methylsulfonyl)quinolin-4-yl]amino}phenolHuman6634
RIPK2RIPKTKL5j79AB4-methyl-3-{[6-(methylsulfonyl)quinolin-4-yl]amino}phenolHuman6636
RIPK2RIPKTKL5j79BA4-methyl-3-{[6-(methylsulfonyl)quinolin-4-yl]amino}phenolHuman6633
RIPK2RIPKTKL5j79BB4-methyl-3-{[6-(methylsulfonyl)quinolin-4-yl]amino}phenolHuman6635
RIPK2RIPKTKL5j7bA6-(tert-butylsulfonyl)-n-(5-fluoro-2h-indazol-3-yl)quinolin-4-amineHuman6637
RIPK2RIPKTKL5j7bB6-(tert-butylsulfonyl)-n-(5-fluoro-2h-indazol-3-yl)quinolin-4-amineHuman6632
RIPK2RIPKTKL5ng0AAphosphomethylphosphonic acid adenylate esterHuman8054
RIPK2RIPKTKL5ng0ABphosphomethylphosphonic acid adenylate esterHuman8051
RIPK2RIPKTKL5ng0BAphosphomethylphosphonic acid adenylate esterHuman8057
RIPK2RIPKTKL5ng0BBphosphomethylphosphonic acid adenylate esterHuman8055
RIPK2RIPKTKL5ng2AAstaurosporineHuman8050
RIPK2RIPKTKL5ng2ABstaurosporineHuman8056
RIPK2RIPKTKL5ng2BAstaurosporineHuman8053
RIPK2RIPKTKL5ng2BBstaurosporineHuman8052
RIPK2RIPKTKL5ng3A-Human8169
RIPK2RIPKTKL5ng3B-Human8170
RIPK2RIPKTKL5ng3C-Human8171
RIPK2RIPKTKL5ng3D-Human8172
RIPK2RIPKTKL5w5jAn-(2-chlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamideHuman8593
RIPK2RIPKTKL5w5jBn-(2-chlorophenyl)pyrazolo[1,5-a]pyridine-3-carboxamideHuman8591
RIPK2RIPKTKL5w5oA4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8579
RIPK2RIPKTKL5w5oB4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8587
RIPK2RIPKTKL5w5oC4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8577
RIPK2RIPKTKL5w5oD4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8576
RIPK2RIPKTKL5w5oE4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8592
RIPK2RIPKTKL5w5oF4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8582
RIPK2RIPKTKL5w5oG4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8580
RIPK2RIPKTKL5w5oH4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8588
RIPK2RIPKTKL5w5oI4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8590
RIPK2RIPKTKL5w5oJ4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8586
RIPK2RIPKTKL5w5oK4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8583
RIPK2RIPKTKL5w5oL4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8585
RIPK2RIPKTKL5w5oM4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8589
RIPK2RIPKTKL5w5oN4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8578
RIPK2RIPKTKL5w5oO4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8584
RIPK2RIPKTKL5w5oP4-{6-(tert-butylsulfonyl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]imidazo[1,2-a]pyridin-3-yl}-6-chloropyridin-2-amineHuman8581
RIPK2RIPKTKL6es0A2-[2-fluoranyl-4-[[2-fluoranyl-4-[2-(methylcarbamoyl)pyridin-4-yl]oxy-phenyl]carbamoylamino]phenyl]sulfanylethanoic acidHuman9574
RIPK2RIPKTKL6es0B2-[2-fluoranyl-4-[[2-fluoranyl-4-[2-(methylcarbamoyl)pyridin-4-yl]oxy-phenyl]carbamoylamino]phenyl]sulfanylethanoic acidHuman9573
RIPK2RIPKTKL6fu5A~{n}-[5-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methoxy-phenyl]propane-1-sulfonamideHuman9852
RIPK2RIPKTKL6fu5B~{n}-[5-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methoxy-phenyl]propane-1-sulfonamideHuman9853
RIPK2RIPKTKL6hmxA6-~{tert}-butylsulfonyl-~{n}-(3,4-dimethyl-1~{h}-pyrazol-5-yl)-7-methoxy-quinolin-4-amineHuman10676
RIPK2RIPKTKL6hmxB6-~{tert}-butylsulfonyl-~{n}-(3,4-dimethyl-1~{h}-pyrazol-5-yl)-7-methoxy-quinolin-4-amineHuman10675
RIPK2RIPKTKL6rn8A2-[4-(1,3-benzothiazol-5-ylamino)-6-~{tert}-butylsulfonyl-quinazolin-7-yl]oxyethyl dihydrogen phosphateHuman11434
RIPK2RIPKTKL6rn8B2-[4-(1,3-benzothiazol-5-ylamino)-6-~{tert}-butylsulfonyl-quinazolin-7-yl]oxyethyl dihydrogen phosphateHuman11431
RIPK2RIPKTKL6rnaA2-[4-(1,3-benzothiazol-5-ylamino)-6-~{tert}-butylsulfonyl-quinazolin-7-yl]oxyethanolHuman11433
RIPK2RIPKTKL6rnaB2-[4-(1,3-benzothiazol-5-ylamino)-6-~{tert}-butylsulfonyl-quinazolin-7-yl]oxyethanolHuman11432
RIPK2RIPKTKL6s1fA~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamideHuman11733
RIPK2RIPKTKL6s1fB~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamideHuman11730
RIPK2RIPKTKL6s1fC~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamideHuman11731
RIPK2RIPKTKL6s1fD~{n}-[3-[2-azanyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxy-phenyl]methanesulfonamideHuman11732
RIPK2RIPKTKL6szeAA5-amino-1-phenylpyrazole-4-carboxamideHuman11759
RIPK2RIPKTKL6szeAB5-amino-1-phenylpyrazole-4-carboxamideHuman11761
RIPK2RIPKTKL6szeBA5-amino-1-phenylpyrazole-4-carboxamideHuman11760
RIPK2RIPKTKL6szeBB5-amino-1-phenylpyrazole-4-carboxamideHuman11758
RIPK2RIPKTKL6szjAA5-amino-1-~{tert}-butyl-3-(3-methoxyphenyl)pyrazole-4-carboxamideHuman11848
RIPK2RIPKTKL6szjAB5-amino-1-~{tert}-butyl-3-(3-methoxyphenyl)pyrazole-4-carboxamideHuman11853
RIPK2RIPKTKL6szjBA5-amino-1-~{tert}-butyl-3-(3-methoxyphenyl)pyrazole-4-carboxamideHuman11846
RIPK2RIPKTKL6szjBB5-amino-1-~{tert}-butyl-3-(3-methoxyphenyl)pyrazole-4-carboxamideHuman11851
RIPK2RIPKTKL6ul8AA(5s,6s,8r)-2-(1,3-benzothiazol-5-yl)-6-hydroxy-4,5,6,7,8,9-hexahydro-5,8-methanopyrazolo[1,5-a][1,3]diazocine-3-carboxamideHuman11847
RIPK2RIPKTKL6ul8AB(5s,6s,8r)-2-(1,3-benzothiazol-5-yl)-6-hydroxy-4,5,6,7,8,9-hexahydro-5,8-methanopyrazolo[1,5-a][1,3]diazocine-3-carboxamideHuman11849
RIPK2RIPKTKL6ul8BA(5s,6s,8r)-2-(1,3-benzothiazol-5-yl)-6-hydroxy-4,5,6,7,8,9-hexahydro-5,8-methanopyrazolo[1,5-a][1,3]diazocine-3-carboxamideHuman11852
RIPK2RIPKTKL6ul8BB(5s,6s,8r)-2-(1,3-benzothiazol-5-yl)-6-hydroxy-4,5,6,7,8,9-hexahydro-5,8-methanopyrazolo[1,5-a][1,3]diazocine-3-carboxamideHuman11850
RIPK2RIPKTKL8azaB-Human14473
Ripk3 (RIPK3)RIPKTKL4m66AA-Mouse5825
Ripk3 (RIPK3)RIPKTKL4m66AB-Mouse5826
Ripk3 (RIPK3)RIPKTKL4m66BA-Mouse5821
Ripk3 (RIPK3)RIPKTKL4m66BB-Mouse5823
Ripk3 (RIPK3)RIPKTKL4m69AAphosphoaminophosphonic acid-adenylate esterMouse5824
Ripk3 (RIPK3)RIPKTKL4m69ABphosphoaminophosphonic acid-adenylate esterMouse5822
Ripk3 (RIPK3)RIPKTKL6okoAA1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamideMouse11438
Ripk3 (RIPK3)RIPKTKL6okoAB1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamideMouse11439
Ripk3 (RIPK3)RIPKTKL6okoBA1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamideMouse11440
Ripk3 (RIPK3)RIPKTKL6okoBB1-(4-fluorophenyl)-n-[3-fluoro-4-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamideMouse11441
RIPK3RIPKTKL7monBn-[4-({2-[(cyclopropanecarbonyl)amino]pyridin-4-yl}oxy)-3-fluorophenyl]-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamideHuman13979
RIPK3RIPKTKL7mx3A3-(1,3-benzothiazol-5-yl)-7-(1,3-dimethyl-1h-pyrazol-5-yl)thieno[3,2-c]pyridin-4-amineHuman13995
Ripk4 (ANKRD3)RIPKTKL5wniAadenosine-5'-triphosphateMouse9889
Ripk4 (ANKRD3)RIPKTKL5wnjAlestaurtinibMouse9893
Ripk4 (ANKRD3)RIPKTKL5wnkA3,3'-(2,4-diaminopteridine-6,7-diyl)diphenolMouse9892
Ripk4 (ANKRD3)RIPKTKL5wnlAstaurosporineMouse9891
Ripk4 (ANKRD3)RIPKTKL5wnmAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideMouse9890
RNASEL (RNAseL)Other-UniqueOther4oauCadenosine-5'-diphosphateHuman468
RNASEL (RNAseL)Other-UniqueOther4oavBphosphomethylphosphonic acid adenylate esterHuman467
RNASEL (RNAseL)Other-UniqueOther4oavDphosphomethylphosphonic acid adenylate esterHuman466
ROCK1DMPKAGC2esmA5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman2726
ROCK1DMPKAGC2esmB5-(1,4-diazepan-1-sulfonyl)isoquinolineHuman2714
ROCK1DMPKAGC2etkA1-(1-hydroxy-5-isoquinolinesulfonyl)homopiperazineHuman2707
ROCK1DMPKAGC2etkB1-(1-hydroxy-5-isoquinolinesulfonyl)homopiperazineHuman2723
ROCK1DMPKAGC2etrA(r)-trans-4-(1-aminoethyl)-n-(4-pyridyl) cyclohexanecarboxamideHuman2700
ROCK1DMPKAGC2etrB(r)-trans-4-(1-aminoethyl)-n-(4-pyridyl) cyclohexanecarboxamideHuman2704
ROCK1DMPKAGC2v55Aphosphoaminophosphonic acid-adenylate esterHuman2694
ROCK1DMPKAGC2v55Cphosphoaminophosphonic acid-adenylate esterHuman2711
ROCK1DMPKAGC3d9vA(s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazineHuman2696
ROCK1DMPKAGC3d9vB(s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazineHuman2701
ROCK1DMPKAGC3nczAcis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamideHuman2699
ROCK1DMPKAGC3nczBcis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamideHuman2720
ROCK1DMPKAGC3nczCcis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamideHuman2719
ROCK1DMPKAGC3nczDcis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamideHuman2724
ROCK1DMPKAGC3ndmA-Human2695
ROCK1DMPKAGC3ndmB(3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamideHuman2698
ROCK1DMPKAGC3ndmC(3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamideHuman2722
ROCK1DMPKAGC3ndmD(3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamideHuman2705
ROCK1DMPKAGC3tv7A1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHuman2697
ROCK1DMPKAGC3tv7B1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHuman2703
ROCK1DMPKAGC3tv7C1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHuman2717
ROCK1DMPKAGC3tv7D1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHuman2725
ROCK1DMPKAGC3twjA1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHuman2710
ROCK1DMPKAGC3twjB-Human2718
ROCK1DMPKAGC3twjC1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)ureaHuman2689
ROCK1DMPKAGC3twjD-Human2690
ROCK1DMPKAGC3v8sA1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHuman2716
ROCK1DMPKAGC3v8sB1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHuman2709
ROCK1DMPKAGC3v8sC1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHuman2702
ROCK1DMPKAGC3v8sD1-(1h-indazol-5-yl)-3-(2-phenylethyl)ureaHuman2692
ROCK1DMPKAGC4w7pAn~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamineHuman2721
ROCK1DMPKAGC4w7pBn~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamineHuman2708
ROCK1DMPKAGC4w7pCn~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamineHuman2688
ROCK1DMPKAGC4w7pDn~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamineHuman2712
ROCK1DMPKAGC4yvcA2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamideHuman2715
ROCK1DMPKAGC4yvcB2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamideHuman2727
ROCK1DMPKAGC4yveA2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamideHuman2693
ROCK1DMPKAGC4yveB2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamideHuman2706
ROCK1DMPKAGC5bmlAn-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-{3-[(methylsulfonyl)amino]phenyl}acetamideHuman2713
ROCK1DMPKAGC5bmlBn-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-{3-[(methylsulfonyl)amino]phenyl}acetamideHuman2691
ROCK1DMPKAGC5hvuA2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamideHuman7414
ROCK1DMPKAGC5hvuB2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamideHuman7415
ROCK1DMPKAGC5kksA2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamideHuman8183
ROCK1DMPKAGC5kksB2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamideHuman8181
ROCK1DMPKAGC5kktA2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamideHuman8182
ROCK1DMPKAGC5kktB2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamideHuman8184
ROCK1DMPKAGC5uzjAn-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamideHuman9706
ROCK1DMPKAGC5uzjBn-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamideHuman9707
ROCK1DMPKAGC5wneA3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamideHuman10446
ROCK1DMPKAGC5wneB3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamideHuman10453
ROCK1DMPKAGC5wneC3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamideHuman10462
ROCK1DMPKAGC5wneD3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamideHuman10445
ROCK1DMPKAGC5wnfAA1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHuman10447
ROCK1DMPKAGC5wnfAB1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHuman10444
ROCK1DMPKAGC5wnfBA1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHuman10463
ROCK1DMPKAGC5wnfBB1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHuman10450
ROCK1DMPKAGC5wnfCA1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHuman10455
ROCK1DMPKAGC5wnfCB1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHuman10460
ROCK1DMPKAGC5wnfDA1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHuman10451
ROCK1DMPKAGC5wnfDB1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamideHuman10452
ROCK1DMPKAGC5wngA(2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamideHuman10459
ROCK1DMPKAGC5wngB(2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamideHuman10461
ROCK1DMPKAGC5wngC(2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamideHuman10458
ROCK1DMPKAGC5wngD(2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamideHuman10457
ROCK1DMPKAGC5wnhA(2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamideHuman10448
ROCK1DMPKAGC5wnhB(2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamideHuman10449
ROCK1DMPKAGC5wnhC(2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamideHuman10456
ROCK1DMPKAGC5wnhD(2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamideHuman10454
ROCK1DMPKAGC6e9wAn-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamideHuman10691
ROCK1DMPKAGC6e9wBn-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamideHuman10690
ROCK1DMPKAGC7jouAn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHuman12768
ROCK1DMPKAGC7s25AA2-[3-(methoxymethyl)phenyl]-n-[4-(1h-pyrazol-4-yl)phenyl]acetamideHuman14435
ROCK1DMPKAGC7s25AB2-[3-(methoxymethyl)phenyl]-n-[4-(1h-pyrazol-4-yl)phenyl]acetamideHuman14436
ROCK1DMPKAGC7s26A2-[methyl(phenyl)amino]-1-[4-(1h-pyrrolo[2,3-b]pyridin-3-yl)-3,6-dihydropyridin-1(2h)-yl]ethan-1-oneHuman14437
ROCK2DMPKAGC4l6qA6-[4-(aminomethyl)-2-fluorophenoxy]-2,1-benzoxaborol-1(3h)-olHuman1811
ROCK2DMPKAGC4l6qB6-[4-(aminomethyl)-2-fluorophenoxy]-2,1-benzoxaborol-1(3h)-olHuman1810
ROCK2DMPKAGC4wotAmethyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoateHuman6827
ROCK2DMPKAGC4wotBmethyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoateHuman6829
ROCK2DMPKAGC4wotCmethyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoateHuman6828
ROCK2DMPKAGC4wotDmethyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoateHuman6830
ROCK2DMPKAGC5u7qA-Human7988
ROCK2DMPKAGC5u7qB-Human7990
ROCK2DMPKAGC5u7qC-Human7987
ROCK2DMPKAGC5u7qD-Human7986
ROCK2DMPKAGC5u7rA(1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-oneHuman7989
ROCK2DMPKAGC5u7rB(1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-oneHuman7984
ROCK2DMPKAGC5u7rC(1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-oneHuman7983
ROCK2DMPKAGC5u7rD(1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-oneHuman7985
ROCK2DMPKAGC6ed6An-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamideHuman10689
ROCK2DMPKAGC6ed6Bn-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamideHuman10688
ROCK2DMPKAGC6p5mAA6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-oneHuman11920
ROCK2DMPKAGC6p5mAB6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-oneHuman11915
ROCK2DMPKAGC6p5mBA6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-oneHuman11921
ROCK2DMPKAGC6p5mBB6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-oneHuman11924
ROCK2DMPKAGC6p5mCA-Human11917
ROCK2DMPKAGC6p5mCB-Human11916
ROCK2DMPKAGC6p5mDA-Human11925
ROCK2DMPKAGC6p5mDB-Human11922
ROCK2DMPKAGC6p5pA2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-oneHuman11914
ROCK2DMPKAGC6p5pB2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-oneHuman11923
ROCK2DMPKAGC6p5pC2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-oneHuman11919
ROCK2DMPKAGC6p5pD2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-oneHuman11918
ROCK2DMPKAGC7jntAAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12744
ROCK2DMPKAGC7jntABn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12754
ROCK2DMPKAGC7jntBAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12756
ROCK2DMPKAGC7jntBBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12766
ROCK2DMPKAGC7jntCAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12752
ROCK2DMPKAGC7jntCBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12745
ROCK2DMPKAGC7jntDAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12755
ROCK2DMPKAGC7jntDBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12750
ROCK2DMPKAGC7jntEAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12746
ROCK2DMPKAGC7jntEBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12747
ROCK2DMPKAGC7jntFAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12749
ROCK2DMPKAGC7jntFBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12758
ROCK2DMPKAGC7jntGAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12761
ROCK2DMPKAGC7jntGBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12767
ROCK2DMPKAGC7jntHAn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12760
ROCK2DMPKAGC7jntHBn-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamideHuman12753
ROCK2DMPKAGC7jovAn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHuman12757
ROCK2DMPKAGC7jovBn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHuman12765
ROCK2DMPKAGC7jovCn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHuman12748
ROCK2DMPKAGC7jovDn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHuman12764
ROCK2DMPKAGC7jovEn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHuman12762
ROCK2DMPKAGC7jovFn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHuman12759
ROCK2DMPKAGC7jovGn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHuman12763
ROCK2DMPKAGC7jovHn-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamideHuman12751
ROCK2DMPKAGC7p6nA~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-yl-piperidine-1-carboxamideHuman14314
ROCK2DMPKAGC8gdsA4-{4-[2-(2,3-dihydro-1h-indol-1-yl)-2-oxoethyl]phenyl}phthalazin-1(2h)-oneHuman14736
ROR1RorTK6tu9A3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman11944
ROR1RorTK6tu9B3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman11945
ROR2RorTK3zzwAA-Human410
ROR2RorTK3zzwAB-Human412
ROR2RorTK3zzwBA-Human415
ROR2RorTK3zzwBB-Human411
ROR2RorTK4gt4AA-Human414
ROR2RorTK4gt4AB-Human409
ROR2RorTK4gt4BA-Human413
ROR2RorTK4gt4BB-Human408
ROS1 (ROS)SevTK3zbfA3-[(1r)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1h-pyrazol-4-yl)pyridin-2-amineHuman197
ROS1 (ROS)SevTK4uxlA(10r)-7-amino-12-fluoro-2,10,16-trimethyl-15-oxo-10,15,16,17-tetrahydro-2h-8,4-(metheno)pyrazolo[4,3-h][2,5,11]benzoxadiazacyclotetradecine-3-carbonitrileHuman198
ROS1 (ROS)SevTK7z5wA~{n}-[6-methyl-2-[(2~{s})-2-[3-(3-methylpyrazin-2-yl)-1,2-oxazol-5-yl]pyrrolidin-1-yl]pyrimidin-4-yl]-1,3-thiazol-2-amineHuman14326
ROS1 (ROS)SevTK7z5xA(2r)-2-[5-(6-amino-5-{(1r)-1-[2-(1,3-dihydro-2h-1,2,3-triazol-2-yl)-5-fluorophenyl]ethoxy}pyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]propane-1,2-diolHuman14325
RPS6KA1 (RSK3)RSKAGC2z7qAphosphomethylphosphonic acid adenylate esterHuman2778
RPS6KA1 (RSK3)RSKAGC2z7rAstaurosporineHuman2777
RPS6KA1 (RSK3)RSKAGC2z7sA2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHuman2776
RPS6KA1-b (RSK3-b)RSKbCAMK2wntAA-Human6862
RPS6KA1-b (RSK3-b)RSKbCAMK2wntAB-Human6859
RPS6KA1-b (RSK3-b)RSKbCAMK2wntBA-Human6860
RPS6KA1-b (RSK3-b)RSKbCAMK2wntBB-Human6861
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyAA-Human5568
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyAB-Human5569
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyBA-Human5573
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyBB-Human5574
RPS6KA1-b (RSK3-b)RSKbCAMK4nifAA-Human5572
RPS6KA1-b (RSK3-b)RSKbCAMK4nifAB-Human5570
RPS6KA1-b (RSK3-b)RSKbCAMK4nifDA-Human5571
RPS6KA1-b (RSK3-b)RSKbCAMK4nifDB-Human5575
RPS6KA2-b (RSK1-b)RSKbCAMK8wf4A-Human15082
Rps6ka3 (RSK2)RSKAGC3g51Aphosphoaminophosphonic acid-adenylate esterMouse5695
Rps6ka3 (RSK2)RSKAGC3ubdAA5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4h-chromen-3-yl 3,4-di-o-acetyl-6-deoxy-alpha-l-mannopyranosideMouse5693
Rps6ka3 (RSK2)RSKAGC3ubdAB5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4h-chromen-3-yl 3,4-di-o-acetyl-6-deoxy-alpha-l-mannopyranosideMouse5691
Rps6ka3 (RSK2)RSKAGC4el9A5,7-dihydroxy-2-(4-hydroxyphenyl)-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranosideMouse5692
Rps6ka3 (RSK2)RSKAGC4gueAA2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranosideMouse5696
Rps6ka3 (RSK2)RSKAGC4gueAB2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranosideMouse5694
RPS6KA3 (RSK2)RSKAGC4nusAA2,6-difluoro-4-{4-[4-(4-methylpiperazin-1-yl)phenyl]pyridin-3-yl}phenolHuman133
RPS6KA3 (RSK2)RSKAGC4nusAB2,6-difluoro-4-{4-[4-(4-methylpiperazin-1-yl)phenyl]pyridin-3-yl}phenolHuman131
RPS6KA3 (RSK2)RSKAGC4nw5AA7-(2-fluoro-6-methoxyphenyl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineHuman134
RPS6KA3 (RSK2)RSKAGC4nw5AB7-(2-fluoro-6-methoxyphenyl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineHuman135
RPS6KA3 (RSK2)RSKAGC4nw6AA7-(1h-benzimidazol-7-yl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineHuman132
RPS6KA3 (RSK2)RSKAGC4nw6AB7-(1h-benzimidazol-7-yl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amineHuman136
RPS6KA3 (RSK2)RSKAGC5d9kA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman5988
RPS6KA3 (RSK2)RSKAGC5d9kB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman5987
RPS6KA3 (RSK2)RSKAGC5d9lAA4,4'-(1h-pyrazole-3,4-diyl)diphenolHuman5986
RPS6KA3 (RSK2)RSKAGC5d9lAB4,4'-(1h-pyrazole-3,4-diyl)diphenolHuman5989
RPS6KA3 (RSK2)RSKAGC7opoAphosphoaminophosphonic acid-adenylate esterHuman14079
RPS6KA3 (RSK2)RSKAGC8eq5AA2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranosideHuman14713
RPS6KA3 (RSK2)RSKAGC8eq5AB2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranosideHuman14714
Rps6ka3-b (RSK2-b)RSKbCAMK2qr7AA-Mouse5759
Rps6ka3-b (RSK2-b)RSKbCAMK2qr7AB-Mouse5757
Rps6ka3-b (RSK2-b)RSKbCAMK2qr8AA-Mouse5760
Rps6ka3-b (RSK2-b)RSKbCAMK2qr8AB-Mouse5755
Rps6ka3-b (RSK2-b)RSKbCAMK4m8tA(2e)-2-cyano-3-[3-(1h-pyrazol-4-yl)phenyl]prop-2-enamideMouse5756
Rps6ka3-b (RSK2-b)RSKbCAMK4maoA(2z)-2-(1h-1,2,4-triazol-1-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]prop-2-enenitrileMouse5758
Rps6ka3-b (RSK2-b)RSKbCAMK5o1sAdimethyl fumarateMouse9976
RPS6KA3-b (RSK2-b)RSKbCAMK4d9tAmethyl (2s)-3-{4-amino-7-[(1e)-3-hydroxyprop-1-en-1-yl]-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl}-2-cyanopropanoateHuman1493
RPS6KA3-b (RSK2-b)RSKbCAMK4d9uAtert-butyl (2s)-3-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl]-2-cyanopropanoateHuman1499
RPS6KA3-b (RSK2-b)RSKbCAMK4jg6A(2s)-2-cyano-3-(1h-indazol-5-yl)propanamideHuman1495
RPS6KA3-b (RSK2-b)RSKbCAMK4jg7AA(2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamideHuman1496
RPS6KA3-b (RSK2-b)RSKbCAMK4jg7AB(2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamideHuman1494
RPS6KA3-b (RSK2-b)RSKbCAMK4jg8AA(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman1497
RPS6KA3-b (RSK2-b)RSKbCAMK4jg8AB(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman1498
RPS6KA5 (MSK1)RSKAGC1vzoAA-Human108
RPS6KA5 (MSK1)RSKAGC1vzoAB-Human107
RPS6KA5-b (MSK1-b)RSKbCAMK3kn5Aphosphoaminophosphonic acid-adenylate esterHuman4603
RPS6KA5-b (MSK1-b)RSKbCAMK3kn5Bphosphoaminophosphonic acid-adenylate esterHuman4600
RPS6KA5-b (MSK1-b)RSKbCAMK3kn6A-Human4602
RPS6KA5-b (MSK1-b)RSKbCAMK3kn6B-Human4601
RPS6KA5-b (MSK1-b)RSKbCAMK7up4AA(5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14277
RPS6KA5-b (MSK1-b)RSKbCAMK7up4AB(5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14279
RPS6KA5-b (MSK1-b)RSKbCAMK7up5AA(2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrileHuman14280
RPS6KA5-b (MSK1-b)RSKbCAMK7up5AB(2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrileHuman14278
RPS6KA5-b (MSK1-b)RSKbCAMK7up6AA(e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound formHuman14353
RPS6KA5-b (MSK1-b)RSKbCAMK7up6AB(e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound formHuman14354
RPS6KA5-b (MSK1-b)RSKbCAMK7up7AA(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman14318
RPS6KA5-b (MSK1-b)RSKbCAMK7up7AB(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman14317
RPS6KA5-b (MSK1-b)RSKbCAMK7up8AA(5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14282
RPS6KA5-b (MSK1-b)RSKbCAMK7up8AB(5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14281
RPS6KA6 (RSK4)RSKAGC6g76Aphosphoaminophosphonic acid-adenylate esterHuman11006
RPS6KA6 (RSK4)RSKAGC6g76Bphosphoaminophosphonic acid-adenylate esterHuman11008
RPS6KA6 (RSK4)RSKAGC6g77Aphosphoaminophosphonic acid-adenylate esterHuman11005
RPS6KA6 (RSK4)RSKAGC6g77Bphosphoaminophosphonic acid-adenylate esterHuman11009
RPS6KA6 (RSK4)RSKAGC6g78Aphosphoaminophosphonic acid-adenylate esterHuman11010
RPS6KA6 (RSK4)RSKAGC6g78Bphosphoaminophosphonic acid-adenylate esterHuman11007
RPS6KB1 (p70S6K)RSKAGC3a60AstaurosporineHuman1852
RPS6KB1 (p70S6K)RSKAGC3a60BstaurosporineHuman1856
RPS6KB1 (p70S6K)RSKAGC3a61AstaurosporineHuman1846
RPS6KB1 (p70S6K)RSKAGC3a62AstaurosporineHuman1867
RPS6KB1 (p70S6K)RSKAGC3we4A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHuman1860
RPS6KB1 (p70S6K)RSKAGC3wf5AA4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidineHuman1857
RPS6KB1 (p70S6K)RSKAGC3wf5AB4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidineHuman1845
RPS6KB1 (p70S6K)RSKAGC3wf6AA4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidineHuman1864
RPS6KB1 (p70S6K)RSKAGC3wf6AB4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidineHuman1859
RPS6KB1 (p70S6K)RSKAGC3wf7AA1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamideHuman1854
RPS6KB1 (p70S6K)RSKAGC3wf7AB1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamideHuman1851
RPS6KB1 (p70S6K)RSKAGC3wf8A2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl 7,8,9,10-tetrahydro-6h-cyclohepta[b]quinoline-11-carboxylateHuman1848
RPS6KB1 (p70S6K)RSKAGC3wf9A(2s)-1-oxo-1-[(4-sulfamoylphenyl)amino]propan-2-yl (2s)-2-methyl-1,2,3,4-tetrahydroacridine-9-carboxylateHuman1866
RPS6KB1 (p70S6K)RSKAGC4l3jA2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHuman1858
RPS6KB1 (p70S6K)RSKAGC4l3lA2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHuman1863
RPS6KB1 (p70S6K)RSKAGC4l42A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHuman1865
RPS6KB1 (p70S6K)RSKAGC4l43A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHuman1861
RPS6KB1 (p70S6K)RSKAGC4l44A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHuman1849
RPS6KB1 (p70S6K)RSKAGC4l45A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHuman1850
RPS6KB1 (p70S6K)RSKAGC4l46A2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazoleHuman1847
RPS6KB1 (p70S6K)RSKAGC4rloA[(amino-kappan)methanethiolato](3-fluoro-9-hydroxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(1,4,7-trithionane-kappa~3~s~1~,s~4~,s~7~)rutheniumHuman7218
RPS6KB1 (p70S6K)RSKAGC4rloBstaurosporineHuman7220
RPS6KB1 (p70S6K)RSKAGC4rlpA[(amino-kappan)methanethiolato](3-fluoro-9-methoxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(n-methyl-1,4,7-trithiecan-9-amine-kappa~3~s~1~,s~4~,s~7~)rutheniumHuman7219
RPS6KB1 (p70S6K)RSKAGC7n91A4-{[(1s)-1-(3-fluorophenyl)-2-(methylamino)ethyl]amino}quinazoline-8-carboxamideHuman14284
RPS6KB1 (p70S6K)RSKAGC7n93AA4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamideHuman14285
RPS6KB1 (p70S6K)RSKAGC7n93AB4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamideHuman14283
RYKRykTK6tuaA-Human11943
SGK1SGKAGC2r5tAphosphoaminophosphonic acid-adenylate esterHuman6849
SGK1SGKAGC3hdmA4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acidHuman3271
SGK1SGKAGC3hdnA[4-(5-naphthalen-2-yl-1h-pyrrolo[2,3-b]pyridin-3-yl)phenyl]acetic acidHuman3270
SGK1SGKAGC7pueA6-[4-[[2,3-bis(chloranyl)phenyl]sulfonylamino]phenyl]-~{n}-[(3~{r})-pyrrolidin-3-yl]-2~{h}-pyrazolo[3,4-b]pyridine-4-carboxamideHuman14012
SIK3 (QSK)CAMKLCAMK8okuA~{n}-ethyl-4-[5-[1-(2-hydroxyethyl)pyrazol-4-yl]benzimidazol-1-yl]-2,6-dimethoxy-benzamideHuman15169
SLKSTE20STE2j51A5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman1833
SLKSTE20STE2jflA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman1838
SLKSTE20STE2jfmAA-Human1836
SLKSTE20STE2jfmAB-Human1841
SLKSTE20STE2uv2AA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman1834
SLKSTE20STE2uv2AB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman1837
SLKSTE20STE4usfAA4-[4-(6-methoxynaphthalen-2-yl)-1h-imidazol-5-yl]pyridineHuman1839
SLKSTE20STE4usfAB4-[4-(6-methoxynaphthalen-2-yl)-1h-imidazol-5-yl]pyridineHuman1832
SLKSTE20STE4usfBA4-[4-(6-methoxynaphthalen-2-yl)-1h-imidazol-5-yl]pyridineHuman1835
SLKSTE20STE4usfBB4-[4-(6-methoxynaphthalen-2-yl)-1h-imidazol-5-yl]pyridineHuman1840
SLKSTE20STE6hvdAA3-(1,3-benzothiazol-2-ylamino)-4-(2-methoxyphenyl)pyrrole-2,5-dioneHuman10625
SLKSTE20STE6hvdAB3-(1,3-benzothiazol-2-ylamino)-4-(2-methoxyphenyl)pyrrole-2,5-dioneHuman10624
SLKSTE20STE8bemAAtivozanibHuman14487
SLKSTE20STE8bemABtivozanibHuman14486
SMG1PIKKAtypical6l53A-Human12156
SMG1PIKKAtypical6l54A-Human12155
SMG1PIKKAtypical6sytA-Human11866
SMG1PIKKAtypical6z3rAphosphoaminophosphonic acid-adenylate esterHuman12630
SMG1PIKKAtypical7pw4A1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-ureaHuman14003
SMG1PIKKAtypical7pw5A1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-ureaHuman14002
SMG1PIKKAtypical7pw6A1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-ureaHuman14001
SMG1PIKKAtypical7pw7A1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-ureaHuman14005
SMG1PIKKAtypical7pw8Aphosphoaminophosphonic acid-adenylate esterHuman14004
SMG1PIKKAtypical7pw9Aphosphoaminophosphonic acid-adenylate esterHuman14000
SNRKCAMKLCAMK5yksA-Human8660
SNRKCAMKLCAMK5yksB-Human8661
Src (SRC)SrcTK6f3fAadenosine-5'-diphosphateMouse9461
Src (SRC)SrcTK8xn8AAadenosine-5'-diphosphateMouse15182
Src (SRC)SrcTK8xn8ABadenosine-5'-diphosphateMouse15183
SRCSrcTK1fmkA-Human981
SRCSrcTK1kswAn6-benzyl adenosine-5'-diphosphateHuman985
SRCSrcTK1y57A4-[(4-methylpiperazin-1-yl)methyl]-n-{3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl}benzamideHuman986
SRCSrcTK1yi6A-Human967
SRCSrcTK1yi6B-Human991
SRCSrcTK1yojA-Human984
SRCSrcTK1yojB-Human974
SRCSrcTK1yolA1-{4-[4-amino-5-(3-methoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl]benzyl}piperidin-4-olHuman968
SRCSrcTK1yolB1-{4-[4-amino-5-(3-methoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl]benzyl}piperidin-4-olHuman966
SRCSrcTK1yomA2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHuman973
SRCSrcTK1yomB2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHuman987
SRCSrcTK2bdfA{[(4-{[2-(4-aminocyclohexyl)-9-ethyl-9h-purin-6-yl]amino}phenyl)(hydroxy)phosphoryl]methyl}phosphonic acidHuman980
SRCSrcTK2bdfB{[(4-{[2-(4-aminocyclohexyl)-9-ethyl-9h-purin-6-yl]amino}phenyl)(hydroxy)phosphoryl]methyl}phosphonic acidHuman975
SRCSrcTK2bdjA3-[2-(2-cyclopentyl-6-{[4-(dimethylphosphoryl)phenyl]amino}-9h-purin-9-yl)ethyl]phenolHuman971
SRCSrcTK2h8hAAn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman970
SRCSrcTK2h8hABn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman992
SRCSrcTK2srcAphosphoaminophosphonic acid-adenylate esterHuman979
SRCSrcTK4k11AA1-tert-butyl-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman983
SRCSrcTK4k11AB1-tert-butyl-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman977
SRCSrcTK4mxoA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman990
SRCSrcTK4mxoB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman978
SRCSrcTK4mxxA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman989
SRCSrcTK4mxxB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman976
SRCSrcTK4mxyA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman982
SRCSrcTK4mxyB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman972
SRCSrcTK4mxzA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman969
SRCSrcTK4mxzB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman988
SRCSrcTK6ateAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10920
SRCSrcTK6e6eAAn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11485
SRCSrcTK6e6eABn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11482
SRCSrcTK6e6eACn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11491
SRCSrcTK6e6eBAn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11480
SRCSrcTK6e6eBBn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11476
SRCSrcTK6e6eBCn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11484
SRCSrcTK6e6eCAn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11471
SRCSrcTK6e6eCBn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11492
SRCSrcTK6e6eCCn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11488
SRCSrcTK6e6eDAn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11489
SRCSrcTK6e6eDBn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11494
SRCSrcTK6e6eDCn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11473
SRCSrcTK6e6eEAn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11479
SRCSrcTK6e6eEBn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11490
SRCSrcTK6e6eECn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11478
SRCSrcTK6e6eFAn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11487
SRCSrcTK6e6eFBn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11472
SRCSrcTK6e6eFCn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11486
SRCSrcTK6e6eGAn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11493
SRCSrcTK6e6eGBn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11474
SRCSrcTK6e6eGCn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11477
SRCSrcTK6e6eHAn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11475
SRCSrcTK6e6eHBn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11483
SRCSrcTK6e6eHCn-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamideHuman11481
SRCSrcTK7ng7Atert-butyl (4-(4-amino-1-(2-(4-(dimethylamino)piperidin-1-yl)ethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)carbamateHuman13900
SRCSrcTK7oteA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman14240
SRCSrcTK8haqA4-[(~{e})-(7-oxidanyl-6~{h}-pyrrolo[2,3-g][1,3]benzothiazol-8-yl)methylideneamino]-~{n}-pyridin-2-yl-benzenesulfonamideHuman14883
SRPK1SRPKCMGC1wakA-Human120
SRPK1SRPKCMGC1wbpAadenosine-5'-diphosphateHuman119
SRPK1SRPKCMGC3begAphosphoaminophosphonic acid-adenylate esterHuman9472
SRPK1SRPKCMGC4wuaAAn-[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamideHuman9471
SRPK1SRPKCMGC4wuaABn-[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamideHuman9469
SRPK1SRPKCMGC5mxxAA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman9470
SRPK1SRPKCMGC5mxxAB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman9467
SRPK1SRPKCMGC5my8AAsphinx31Human9466
SRPK1SRPKCMGC5my8ABsphinx31Human9468
SRPK1SRPKCMGC5xv7A9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrileHuman9727
SRPK1SRPKCMGC6fadA-Human11638
SRPK1SRPKCMGC6fadB-Human11640
SRPK1SRPKCMGC6fadC-Human11639
SRPK1SRPKCMGC6fadD-Human11637
SRPK1SRPKCMGC7dd1A-Human13510
SRPK1SRPKCMGC7pqsAA~{n}-[3-[[[2-(6-chloranyl-7-fluoranyl-1~{h}-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-~{n}-methyl-methanesulfonamideHuman14014
SRPK1SRPKCMGC7pqsAB~{n}-[3-[[[2-(6-chloranyl-7-fluoranyl-1~{h}-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-~{n}-methyl-methanesulfonamideHuman14015
SRPK1SRPKCMGC7zksAAn-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamideHuman14619
SRPK1SRPKCMGC7zksABn-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamideHuman14618
SRPK2SRPKCMGC2x7gApurvalanol bHuman1409
SRPK2SRPKCMGC5myvAA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7579
SRPK2SRPKCMGC5myvAB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7575
SRPK2SRPKCMGC5myvBA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7576
SRPK2SRPKCMGC5myvBB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7573
SRPK2SRPKCMGC5myvCA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7580
SRPK2SRPKCMGC5myvCB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7571
SRPK2SRPKCMGC5myvDA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7578
SRPK2SRPKCMGC5myvDB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7572
SRPK2SRPKCMGC7zkxAAn-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamideHuman14617
SRPK2SRPKCMGC7zkxABn-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamideHuman14616
STK10 (LOK)STE20STE2j7tAA(3z)-n-(3-chlorophenyl)-3-({3,5-dimethyl-4-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-2-yl}methylene)-n-methyl-2-oxoindoline-5-sulfonamideHuman946
STK10 (LOK)STE20STE2j7tAB(3z)-n-(3-chlorophenyl)-3-({3,5-dimethyl-4-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-2-yl}methylene)-n-methyl-2-oxoindoline-5-sulfonamideHuman960
STK10 (LOK)STE20STE4aotAA1-(4-{methyl[2-({4-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]amino}phenyl)-3-{3-[(4-methylpiperazin-1-yl)carbonyl]phenyl}ureaHuman947
STK10 (LOK)STE20STE4aotAB1-(4-{methyl[2-({4-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]amino}phenyl)-3-{3-[(4-methylpiperazin-1-yl)carbonyl]phenyl}ureaHuman944
STK10 (LOK)STE20STE4aotBA1-(4-{methyl[2-({4-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]amino}phenyl)-3-{3-[(4-methylpiperazin-1-yl)carbonyl]phenyl}ureaHuman945
STK10 (LOK)STE20STE4aotBB1-(4-{methyl[2-({4-[(methylsulfonyl)methyl]phenyl}amino)pyrimidin-4-yl]amino}phenyl)-3-{3-[(4-methylpiperazin-1-yl)carbonyl]phenyl}ureaHuman943
STK10 (LOK)STE20STE4bc6AA4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman942
STK10 (LOK)STE20STE4bc6AB4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman961
STK10 (LOK)STE20STE4equAAn-{3-[(3-{4-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}pyridin-2-yl)amino]-4-methylphenyl}-3-(trifluoromethyl)benzamideHuman957
STK10 (LOK)STE20STE4equABn-{3-[(3-{4-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}pyridin-2-yl)amino]-4-methylphenyl}-3-(trifluoromethyl)benzamideHuman938
STK10 (LOK)STE20STE4equBAn-{3-[(3-{4-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}pyridin-2-yl)amino]-4-methylphenyl}-3-(trifluoromethyl)benzamideHuman941
STK10 (LOK)STE20STE4equBBn-{3-[(3-{4-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}pyridin-2-yl)amino]-4-methylphenyl}-3-(trifluoromethyl)benzamideHuman959
STK10 (LOK)STE20STE4usdAA4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridineHuman953
STK10 (LOK)STE20STE4usdAB4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridineHuman949
STK10 (LOK)STE20STE4usdBA4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridineHuman939
STK10 (LOK)STE20STE4usdBB4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridineHuman956
STK10 (LOK)STE20STE4useAA4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridineHuman952
STK10 (LOK)STE20STE4useAB4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridineHuman951
STK10 (LOK)STE20STE4useBA4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridineHuman958
STK10 (LOK)STE20STE4useBB4-{5-(6-methoxynaphthalen-2-yl)-1-methyl-2-[2-methyl-4-(methylsulfonyl)phenyl]-1h-imidazol-4-yl}pyridineHuman954
STK10 (LOK)STE20STE5ajqAA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman950
STK10 (LOK)STE20STE5ajqAB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman955
STK10 (LOK)STE20STE5ajqBA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman940
STK10 (LOK)STE20STE5ajqBB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman948
STK10 (LOK)STE20STE5owqAA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman8385
STK10 (LOK)STE20STE5owqAB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman8386
STK10 (LOK)STE20STE5owqBA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman8387
STK10 (LOK)STE20STE5owqBB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman8389
STK10 (LOK)STE20STE5owrAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman8384
STK10 (LOK)STE20STE5owrABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman8388
STK10 (LOK)STE20STE6eimAA~{n}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-1~{h}-benzimidazol-2-yl]furan-2-carboxamideHuman8626
STK10 (LOK)STE20STE6eimAB~{n}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-1~{h}-benzimidazol-2-yl]furan-2-carboxamideHuman8625
STK10 (LOK)STE20STE6eimBA~{n}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-1~{h}-benzimidazol-2-yl]furan-2-carboxamideHuman8623
STK10 (LOK)STE20STE6eimBB~{n}-[5-[4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]phenoxy]-1~{h}-benzimidazol-2-yl]furan-2-carboxamideHuman8624
STK10 (LOK)STE20STE6gttAA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman10026
STK10 (LOK)STE20STE6gttAB1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman10025
STK10 (LOK)STE20STE6hxfAA3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dioneHuman10656
STK10 (LOK)STE20STE6hxfAB3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dioneHuman10654
STK10 (LOK)STE20STE6hxfBA3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dioneHuman10651
STK10 (LOK)STE20STE6hxfBB3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dioneHuman10652
STK10 (LOK)STE20STE6hxfCA3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dioneHuman10649
STK10 (LOK)STE20STE6hxfCB3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dioneHuman10655
STK10 (LOK)STE20STE6hxfDA3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dioneHuman10650
STK10 (LOK)STE20STE6hxfDB3-(2-methoxyphenyl)-4-[[4-(phenylcarbonyl)phenyl]amino]pyrrole-2,5-dioneHuman10653
STK10 (LOK)STE20STE6i2yAn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman10787
STK10 (LOK)STE20STE6i2yBn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman10788
STK10 (LOK)STE20STE7qgpA1-[(4-chloranyl-2-methyl-phenyl)methyl]-3-(7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaen-5-yl)ureaHuman14075
STK11 (LKB1)CAMKLCAMK2wtkCphosphoaminophosphonic acid-adenylate esterHuman1868
STK11 (LKB1)CAMKLCAMK2wtkFphosphoaminophosphonic acid-adenylate esterHuman1869
STK16 (MPSK1)NAKOther2bujAstaurosporineHuman2229
STK16 (MPSK1)NAKOther2bujBstaurosporineHuman2230
STK17A (DRAK1)DAPKCAMK7queA~{n}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamideHuman14094
STK17A (DRAK1)DAPKCAMK7qufA~{n}-~{tert}-butyl-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamideHuman14093
STK17B (DRAK2)DAPKCAMK3lm0AA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-5-methylpyrimidin-2-yl}amino)phenyl]acetonitrileHuman6796
STK17B (DRAK2)DAPKCAMK3lm0AB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-5-methylpyrimidin-2-yl}amino)phenyl]acetonitrileHuman6797
STK17B (DRAK2)DAPKCAMK3lm5AA3,5,7,3',4'-pentahydroxyflavoneHuman6795
STK17B (DRAK2)DAPKCAMK3lm5AB3,5,7,3',4'-pentahydroxyflavoneHuman6798
STK17B (DRAK2)DAPKCAMK6qf4AAadenosine-5'-diphosphateHuman11397
STK17B (DRAK2)DAPKCAMK6qf4ABadenosine-5'-diphosphateHuman11396
STK17B (DRAK2)DAPKCAMK6y6fAA2-[6-(4-methylsulfanylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12045
STK17B (DRAK2)DAPKCAMK6y6fAB2-[6-(4-methylsulfanylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12042
STK17B (DRAK2)DAPKCAMK6y6hAA2-[6-(1-benzothiophen-2-yl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12043
STK17B (DRAK2)DAPKCAMK6y6hAB2-[6-(1-benzothiophen-2-yl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12044
STK17B (DRAK2)DAPKCAMK6zjfAA2-[6-(4-cyclopropylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12642
STK17B (DRAK2)DAPKCAMK6zjfAB2-[6-(4-cyclopropylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12643
STK17B (DRAK2)DAPKCAMK7akgAA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman13005
STK17B (DRAK2)DAPKCAMK7akgAB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman13004
STK17B (DRAK2)DAPKCAMK7q7cAAadenosine-5'-diphosphateHuman14510
STK17B (DRAK2)DAPKCAMK7q7cABadenosine-5'-diphosphateHuman14508
STK17B (DRAK2)DAPKCAMK7q7dAAadenosine-5'-triphosphateHuman14519
STK17B (DRAK2)DAPKCAMK7q7dABadenosine-5'-triphosphateHuman14509
STK17B (DRAK2)DAPKCAMK7q7eAAadenosine-5'-triphosphateHuman14520
STK17B (DRAK2)DAPKCAMK7q7eABadenosine-5'-triphosphateHuman14507
STK24 (MST3)STE20STE3a7fA-Human5596
STK24 (MST3)STE20STE3a7gA-Human5612
STK24 (MST3)STE20STE3a7gB-Human5598
STK24 (MST3)STE20STE3a7hAadenosine-5'-triphosphateHuman5600
STK24 (MST3)STE20STE3a7hBadenosine-5'-triphosphateHuman5576
STK24 (MST3)STE20STE3a7iAadenineHuman5611
STK24 (MST3)STE20STE3a7jAadenosine-5'-diphosphateHuman5594
STK24 (MST3)STE20STE3ckwAA-Human5580
STK24 (MST3)STE20STE3ckwAB-Human5601
STK24 (MST3)STE20STE3ckxAstaurosporineHuman5599
STK24 (MST3)STE20STE3zhpC-Human5593
STK24 (MST3)STE20STE3zhpD-Human5588
STK24 (MST3)STE20STE4o27Badenosine-5'-diphosphateHuman5602
STK24 (MST3)STE20STE4qmlAphosphoaminophosphonic acid-adenylate esterHuman5605
STK24 (MST3)STE20STE4qmmA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman5583
STK24 (MST3)STE20STE4qmnAA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman5587
STK24 (MST3)STE20STE4qmnAB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman5604
STK24 (MST3)STE20STE4qmoAA(8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman5585
STK24 (MST3)STE20STE4qmoAB(8z)-8-(1h-imidazol-5-ylmethylidene)-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman5597
STK24 (MST3)STE20STE4qmpA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman5584
STK24 (MST3)STE20STE4qmqAA1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amineHuman5607
STK24 (MST3)STE20STE4qmqAB1-{2-[5-(2-methoxyethoxy)-1h-benzimidazol-1-yl]quinolin-8-yl}piperidin-4-amineHuman5595
STK24 (MST3)STE20STE4qmsAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman5590
STK24 (MST3)STE20STE4qmsABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman5608
STK24 (MST3)STE20STE4qmtAn-[2-oxo-3-((e)-phenyl{[4-(piperidin-1-ylmethyl)phenyl]imino}methyl)-2,6-dihydro-1h-indol-5-yl]ethanesulfonamideHuman5613
STK24 (MST3)STE20STE4qmuAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman5606
STK24 (MST3)STE20STE4qmuAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman5603
STK24 (MST3)STE20STE4qmvAn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman5581
STK24 (MST3)STE20STE4qmwAA1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman5577
STK24 (MST3)STE20STE4qmwAB1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman5582
STK24 (MST3)STE20STE4qmxAn-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amineHuman5609
STK24 (MST3)STE20STE4qmyAstaurosporineHuman5592
STK24 (MST3)STE20STE4qmzAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman5578
STK24 (MST3)STE20STE4qnaA2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman5579
STK24 (MST3)STE20STE4qo9An-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman5586
STK24 (MST3)STE20STE4qo9Bn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman5591
STK24 (MST3)STE20STE4u8zA3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrileHuman5610
STK24 (MST3)STE20STE4w8dA5-(1-methyl-1h-pyrazol-4-yl)-4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidineHuman5614
STK24 (MST3)STE20STE4w8eA3-{4-[(2r)-2-(5-methyl-1,2,4-oxadiazol-3-yl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrileHuman5589
STK24 (MST3)STE20STE7b30A8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman13047
STK24 (MST3)STE20STE7b31AA1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-oneHuman13045
STK24 (MST3)STE20STE7b31AB1-[(5-azanyl-1,3-dioxan-2-yl)methyl]-3-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-7-(methylamino)-1,6-naphthyridin-2-oneHuman13050
STK24 (MST3)STE20STE7b32A8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[(2-methoxyphenyl)amino]pyrido[2,3-d]pyrimidin-7-oneHuman13049
STK24 (MST3)STE20STE7b33A8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[4-[6-[bis(fluoranyl)methyl]pyridin-2-yl]-2-chloranyl-phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman13048
STK24 (MST3)STE20STE7b34A8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranyl-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman13051
STK24 (MST3)STE20STE7b35A8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman13052
STK24 (MST3)STE20STE7b35B8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-methoxy-6-methyl-pyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman13046
STK24 (MST3)STE20STE8bziAA8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14585
STK24 (MST3)STE20STE8bziAB8-(4-azanylbutyl)-6-[2,5-bis(fluoranyl)-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14584
STK24 (MST3)STE20STE8bzjAA8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14586
STK24 (MST3)STE20STE8bzjAB8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14583
STK24 (MST3)STE20STE8qlqAAmacrocyclic inhibitorHuman14873
STK24 (MST3)STE20STE8qlqABmacrocyclic inhibitorHuman14870
STK24 (MST3)STE20STE8qlrA8-(4-azanylbutyl)-2-[1,3-bis(oxidanyl)propan-2-ylamino]-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]pyrido[2,3-d]pyrimidin-7-oneHuman14875
STK24 (MST3)STE20STE8qlsAA8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14872
STK24 (MST3)STE20STE8qlsAB8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14876
STK24 (MST3)STE20STE8qlsAC8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-(3-morpholin-4-ylpropylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14871
STK24 (MST3)STE20STE8qltAA8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-oneHuman14874
STK24 (MST3)STE20STE8qltAB8-(4-azanylbutyl)-6-[2-chloranyl-4-(6-methylpyridin-2-yl)phenyl]-2-[3-(2-oxidanylidenepyrrolidin-1-yl)propylamino]pyrido[2,3-d]pyrimidin-7-oneHuman14869
STK25 (YSK1)STE20STE2xikAA5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman463
STK25 (YSK1)STE20STE2xikAB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman465
STK25 (YSK1)STE20STE4nzwB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman464
STK25 (YSK1)STE20STE7z4vAA~{n}-(5-~{tert}-butyl-1~{h}-pyrazol-3-yl)-4-pyrrolidin-1-ylsulfonyl-benzamideHuman14176
STK25 (YSK1)STE20STE7z4vAB~{n}-(5-~{tert}-butyl-1~{h}-pyrazol-3-yl)-4-pyrrolidin-1-ylsulfonyl-benzamideHuman14177
STK26 (MST4)STE20STE3ggfAA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman1807
STK26 (MST4)STE20STE3ggfAB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman1808
STK26 (MST4)STE20STE3ggfBA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman1805
STK26 (MST4)STE20STE3ggfBB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman1804
STK26 (MST4)STE20STE4fzaB-Human1806
STK26 (MST4)STE20STE4fzdB-Human1809
STK26 (MST4)STE20STE4fzfB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman1803
STK26 (MST4)STE20STE7b36A8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman13044
STK26 (MST4)STE20STE7b36C8-[(trans-5-amino-1,3-dioxan-2-yl)methyl]-6-[2-chloro-4-(6-methylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman13043
STK3 (MST2)STE20STE4lg4AA-Human1442
STK3 (MST2)STE20STE4lg4AB-Human1438
STK3 (MST2)STE20STE4lg4BA-Human1433
STK3 (MST2)STE20STE4lg4BB-Human1427
STK3 (MST2)STE20STE4lg4CA-Human1432
STK3 (MST2)STE20STE4lg4CB-Human1440
STK3 (MST2)STE20STE4lg4DA-Human1435
STK3 (MST2)STE20STE4lg4DB-Human1434
STK3 (MST2)STE20STE4lg4EA-Human1439
STK3 (MST2)STE20STE4lg4EB-Human1441
STK3 (MST2)STE20STE4lg4FA-Human1431
STK3 (MST2)STE20STE4lg4FB-Human1436
STK3 (MST2)STE20STE4lgdAphosphoaminophosphonic acid-adenylate esterHuman1437
STK3 (MST2)STE20STE4lgdBphosphoaminophosphonic acid-adenylate esterHuman1428
STK3 (MST2)STE20STE4lgdCphosphoaminophosphonic acid-adenylate esterHuman1429
STK3 (MST2)STE20STE4lgdDphosphoaminophosphonic acid-adenylate esterHuman1430
STK3 (MST2)STE20STE5dh3AA4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman7031
STK3 (MST2)STE20STE5dh3AB4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman7028
STK3 (MST2)STE20STE5dh3BA4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman7029
STK3 (MST2)STE20STE5dh3BB4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman7030
STK3 (MST2)STE20STE6ao5Aphosphoaminophosphonic acid-adenylate esterHuman8662
STK3 (MST2)STE20STE8a66AA4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman14323
STK3 (MST2)STE20STE8a66AB4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman14324
STK32A (YANK1)YANKAGC4fr4AAstaurosporineHuman4693
STK32A (YANK1)YANKAGC4fr4ABstaurosporineHuman4690
STK32A (YANK1)YANKAGC4fr4BAstaurosporineHuman4692
STK32A (YANK1)YANKAGC4fr4BBstaurosporineHuman4695
STK32A (YANK1)YANKAGC4fr4CAstaurosporineHuman4684
STK32A (YANK1)YANKAGC4fr4CBstaurosporineHuman4694
STK32A (YANK1)YANKAGC4fr4DAstaurosporineHuman4688
STK32A (YANK1)YANKAGC4fr4DBstaurosporineHuman4687
STK32A (YANK1)YANKAGC4fr4EAstaurosporineHuman4689
STK32A (YANK1)YANKAGC4fr4EBstaurosporineHuman4685
STK32A (YANK1)YANKAGC4fr4FAstaurosporineHuman4691
STK32A (YANK1)YANKAGC4fr4FBstaurosporineHuman4686
STK38 (NDR1)NDRAGC6bxiAphosphoaminophosphonic acid-adenylate esterHuman10326
STK38 (NDR1)NDRAGC6bxiBphosphoaminophosphonic acid-adenylate esterHuman10325
Stk39 (STLK3)STE20STE5d9hAadenosine-5'-triphosphateMouse6025
Stk39 (STLK3)STE20STE5d9hBadenosine-5'-triphosphateMouse6024
Stk39 (STLK3)STE20STE5dbxAAphosphoaminophosphonic acid-adenylate esterMouse6109
Stk39 (STLK3)STE20STE5dbxABphosphoaminophosphonic acid-adenylate esterMouse6107
Stk39 (STLK3)STE20STE5dbxBAphosphoaminophosphonic acid-adenylate esterMouse6106
Stk39 (STLK3)STE20STE5dbxBBphosphoaminophosphonic acid-adenylate esterMouse6108
STK4 (MST1)STE20STE3comA-Human2828
STK4 (MST1)STE20STE3comB-Human2829
STK4 (MST1)STE20STE6yatA4-[5-(3-chlorophenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]morpholineHuman12241
STK4 (MST1)STE20STE6yatB4-[5-(3-chlorophenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl]morpholineHuman12242
STK4 (MST1)STE20STE8a5jAA4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman14290
STK4 (MST1)STE20STE8a5jAB4-[(5,10-dimethyl-6-oxo-6,10-dihydro-5h-pyrimido[5,4-b]thieno[3,2-e][1,4]diazepin-2-yl)amino]benzenesulfonamideHuman14291
STK40 (SgK495)SgK495CAMK5l2qAA-Human8015
STK40 (SgK495)SgK495CAMK5l2qAB-Human8014
STK40 (SgK495)SgK495CAMK5l2qBA-Human8011
STK40 (SgK495)SgK495CAMK5l2qBB-Human8017
STK40 (SgK495)SgK495CAMK5l2qCA-Human8018
STK40 (SgK495)SgK495CAMK5l2qCB-Human8016
STK40 (SgK495)SgK495CAMK5l2qDA-Human8012
STK40 (SgK495)SgK495CAMK5l2qDB-Human8013
STRADA (STLK5)STE20STE2wtkBphosphoaminophosphonic acid-adenylate esterHuman3485
STRADA (STLK5)STE20STE2wtkEphosphoaminophosphonic acid-adenylate esterHuman3484
STRADA (STLK5)STE20STE3gniBadenosine-5'-triphosphateHuman3486
SYKSykTK1xbaA-Human1193
SYKSykTK1xbbAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1184
SYKSykTK1xbbAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman1196
SYKSykTK1xbcAAstaurosporineHuman1165
SYKSykTK1xbcABstaurosporineHuman1207
SYKSykTK3emgA2-{2-[(3,5-dimethylphenyl)amino]pyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-methylethyl]-4-methyl-1,3-thiazole-5-carboxamideHuman1183
SYKSykTK3fqeA2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(3-methylphenyl)amino]pyrimidine-5-carboxamideHuman1155
SYKSykTK3fqhAn-(2-hydroxy-1,1-dimethylethyl)-1-methyl-3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indole-5-carboxamideHuman1203
SYKSykTK3fqhBn-(2-hydroxy-1,1-dimethylethyl)-1-methyl-3-(1h-pyrrolo[2,3-b]pyridin-2-yl)-1h-indole-5-carboxamideHuman1171
SYKSykTK3fqsAA6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-oneHuman1169
SYKSykTK3fqsAB6-({5-fluoro-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}amino)-2,2-dimethyl-2h-pyrido[3,2-b][1,4]oxazin-3(4h)-oneHuman1202
SYKSykTK3srvAA2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamideHuman1154
SYKSykTK3srvAB2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamideHuman1162
SYKSykTK3srvBA2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamideHuman1181
SYKSykTK3srvBB2-{[(3r,4r)-3-aminotetrahydro-2h-pyran-4-yl]amino}-4-[(4-methylphenyl)amino]pyrimidine-5-carboxamideHuman1206
SYKSykTK3tubA1-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-3-[(1r,2s)-2-phenylcyclopropyl]ureaHuman1179
SYKSykTK3tucA1-benzyl-n-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-2-oxo-1,2-dihydropyridine-3-carboxamideHuman1195
SYKSykTK3tudAn-{4-methyl-3-[8-methyl-7-oxo-2-(phenylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]phenyl}-3-(trifluoromethyl)benzamideHuman1176
SYKSykTK3vf8A3-[5-(5-ethoxy-6-fluoro-1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]-1,1-diethylureaHuman1187
SYKSykTK3vf9A3-{2-[5-(difluoromethyl)-2h-thieno[3,2-c]pyrazol-3-yl]-1h-indol-6-yl}pentan-3-olHuman1159
SYKSykTK4dflA3-amino-6-{3-[(methylsulfonyl)amino]phenyl}-n-(piperidin-4-ylmethyl)pyrazine-2-carboxamideHuman1152
SYKSykTK4dfnAA3-amino-6-[3-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-[(1r,2r,3s,5s,7s)-5-hydroxyadamantan-2-yl]pyrazine-2-carboxamideHuman1201
SYKSykTK4dfnAB3-amino-6-[3-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-[(1r,2r,3s,5s,7s)-5-hydroxyadamantan-2-yl]pyrazine-2-carboxamideHuman1199
SYKSykTK4f4pAAn-{6-[3-(piperazin-1-yl)phenyl]pyridin-2-yl}-4-(trifluoromethyl)pyridin-2-amineHuman1178
SYKSykTK4f4pABn-{6-[3-(piperazin-1-yl)phenyl]pyridin-2-yl}-4-(trifluoromethyl)pyridin-2-amineHuman1156
SYKSykTK4fl1AAphosphoaminophosphonic acid-adenylate esterHuman1160
SYKSykTK4fl1ABphosphoaminophosphonic acid-adenylate esterHuman1167
SYKSykTK4fl2Aphosphoaminophosphonic acid-adenylate esterHuman1191
SYKSykTK4fl3AAphosphoaminophosphonic acid-adenylate esterHuman1170
SYKSykTK4fl3ABphosphoaminophosphonic acid-adenylate esterHuman1172
SYKSykTK4fynAA3-[8-({4-[ethyl(2-hydroxyethyl)amino]phenyl}amino)imidazo[1,2-a]pyrazin-5-yl]phenolHuman1174
SYKSykTK4fynAB3-[8-({4-[ethyl(2-hydroxyethyl)amino]phenyl}amino)imidazo[1,2-a]pyrazin-5-yl]phenolHuman1197
SYKSykTK4fyoAA4-{[(3s)-1-{7-[(3,4-dimethoxyphenyl)amino][1,3]thiazolo[5,4-d]pyrimidin-5-yl}pyrrolidin-3-yl]carbamoyl}benzoic acidHuman1180
SYKSykTK4fyoAB4-{[(3s)-1-{7-[(3,4-dimethoxyphenyl)amino][1,3]thiazolo[5,4-d]pyrimidin-5-yl}pyrrolidin-3-yl]carbamoyl}benzoic acidHuman1205
SYKSykTK4fz6AAn-{6-[(2s)-2-methylpyrrolidin-1-yl]pyridin-2-yl}-6-phenylimidazo[1,2-b]pyridazin-8-amineHuman1173
SYKSykTK4fz6ABn-{6-[(2s)-2-methylpyrrolidin-1-yl]pyridin-2-yl}-6-phenylimidazo[1,2-b]pyridazin-8-amineHuman1185
SYKSykTK4fz7AA6-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(6-ethylpyridin-2-yl)amino]pyridazine-3-carboxamideHuman1186
SYKSykTK4fz7AB6-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(6-ethylpyridin-2-yl)amino]pyridazine-3-carboxamideHuman1177
SYKSykTK4gfgA6-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(5,6-dimethylpyridin-2-yl)amino]pyridazine-3-carboxamideHuman1188
SYKSykTK4i0rAAn-(propan-2-yl)-2-(3,4,5-trimethoxyphenyl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman1192
SYKSykTK4i0rABn-(propan-2-yl)-2-(3,4,5-trimethoxyphenyl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman1175
SYKSykTK4i0sAA2-(6-chloro-1-methyl-1h-indazol-3-yl)-n-(propan-2-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman1157
SYKSykTK4i0sAB2-(6-chloro-1-methyl-1h-indazol-3-yl)-n-(propan-2-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman1166
SYKSykTK4i0tAAn-tert-butyl-2-(5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-1-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman1198
SYKSykTK4i0tABn-tert-butyl-2-(5,6,7,8-tetrahydroimidazo[1,5-a]pyridin-1-yl)-5h-pyrrolo[2,3-b]pyrazine-7-carboxamideHuman1164
SYKSykTK4puzA6-(1h-indazol-6-yl)-n-[4-(morpholin-4-yl)phenyl]imidazo[1,2-a]pyrazin-8-amineHuman1163
SYKSykTK4puzB6-(1h-indazol-6-yl)-n-[4-(morpholin-4-yl)phenyl]imidazo[1,2-a]pyrazin-8-amineHuman1153
SYKSykTK4pv0A4-[(3-{8-[(3,4-dimethoxyphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzoyl)amino]benzoic acidHuman1161
SYKSykTK4px6AA7-{[(1r,2s)-2-aminocyclohexyl]amino}-5-(1h-indol-7-ylamino)pyrido[4,3-d]pyrimidin-4(3h)-oneHuman1200
SYKSykTK4px6AB7-{[(1r,2s)-2-aminocyclohexyl]amino}-5-(1h-indol-7-ylamino)pyrido[4,3-d]pyrimidin-4(3h)-oneHuman1204
SYKSykTK4rssAA1-[(3-methyl-1-{2-[(1,2,3-trimethyl-1h-indol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-olHuman6169
SYKSykTK4rssAB1-[(3-methyl-1-{2-[(1,2,3-trimethyl-1h-indol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-olHuman6170
SYKSykTK4rx7AA3-{[(1r,2s)-2-aminocyclohexyl]amino}-5-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}-1,2,4-triazine-6-carboxamideHuman1189
SYKSykTK4rx7AB3-{[(1r,2s)-2-aminocyclohexyl]amino}-5-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}-1,2,4-triazine-6-carboxamideHuman1182
SYKSykTK4rx8AA3-{[(1r,2s)-2-aminocyclohexyl]amino}-5-(1h-indol-7-ylamino)-1,2,4-triazine-6-carboxamideHuman1158
SYKSykTK4rx8AB3-{[(1r,2s)-2-aminocyclohexyl]amino}-5-(1h-indol-7-ylamino)-1,2,4-triazine-6-carboxamideHuman1168
SYKSykTK4rx9AA2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamideHuman1190
SYKSykTK4rx9AB2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamideHuman1194
SYKSykTK4wnmAn~3~-(tetrahydro-2h-pyran-4-yl)-n~6~-[5-(tetrahydro-2h-pyran-4-ylmethyl)[1,2,4]triazolo[1,5-a]pyridin-2-yl]-1h-indazole-3,6-diamineHuman6358
SYKSykTK4xg2A-Human6309
SYKSykTK4xg3A4-{[5-fluoro-4-(3-{[(3r)-3-hydroxypyrrolidin-1-yl]methyl}-4-methyl-1h-pyrrol-1-yl)pyrimidin-2-yl]amino}-2,6-dimethylphenyl methanesulfonateHuman6308
SYKSykTK4xg3B4-{[5-fluoro-4-(3-{[(3r)-3-hydroxypyrrolidin-1-yl]methyl}-4-methyl-1h-pyrrol-1-yl)pyrimidin-2-yl]amino}-2,6-dimethylphenyl methanesulfonateHuman6314
SYKSykTK4xg4A(3r)-1-{[1-(5-fluoro-2-{[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]amino}pyrimidin-4-yl)-4-methyl-1h-pyrrol-3-yl]methyl}pyrrolidin-3-olHuman6319
SYKSykTK4xg6A1-[(1-{2-[(3,5-dimethylphenyl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-olHuman6312
SYKSykTK4xg7AA1-[(3-methyl-1-{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-olHuman6316
SYKSykTK4xg7AB1-[(3-methyl-1-{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-1h-pyrazol-4-yl)methyl]azetidin-3-olHuman6318
SYKSykTK4xg8A1-[(1-{2-[(3-chloro-1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-olHuman6317
SYKSykTK4xg8C1-[(1-{2-[(3-chloro-1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-olHuman6310
SYKSykTK4xg9A1-[(1-{2-[(3-chloro-1,2-dimethyl-1h-indol-5-yl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-olHuman6311
SYKSykTK4xg9B1-[(1-{2-[(3-chloro-1,2-dimethyl-1h-indol-5-yl)amino]pyrimidin-4-yl}-3-methyl-1h-pyrazol-4-yl)methyl]azetidin-3-olHuman6315
SYKSykTK4yjoAA5-chloro-n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamineHuman6120
SYKSykTK4yjoAB5-chloro-n~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamineHuman6119
SYKSykTK4yjpA2-[{2-[(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)amino]pyrimidin-4-yl}(1h-indazol-4-yl)amino]ethanolHuman6115
SYKSykTK4yjqAA3-[1h-indazol-4-yl(2-{[3-(4-methyl-1,3-oxazol-5-yl)phenyl]amino}pyrimidin-4-yl)amino]propan-1-olHuman6114
SYKSykTK4yjqAB3-[1h-indazol-4-yl(2-{[3-(4-methyl-1,3-oxazol-5-yl)phenyl]amino}pyrimidin-4-yl)amino]propan-1-olHuman6123
SYKSykTK4yjrAA3-(1h-indazol-4-yl{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-olHuman6113
SYKSykTK4yjrAB3-(1h-indazol-4-yl{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-olHuman6116
SYKSykTK4yjrAC3-(1h-indazol-4-yl{2-[(1-methyl-1h-indazol-5-yl)amino]pyrimidin-4-yl}amino)propan-1-olHuman6122
SYKSykTK4yjsA3-[{2-[(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)amino]pyrimidin-4-yl}(1h-indazol-4-yl)amino]propan-1-olHuman6117
SYKSykTK4yjtAAn~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-5-fluoro-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamineHuman6125
SYKSykTK4yjtABn~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-5-fluoro-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamineHuman6118
SYKSykTK4yjtACn~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-n~4~-ethyl-5-fluoro-n~4~-(1h-indazol-4-yl)pyrimidine-2,4-diamineHuman6124
SYKSykTK4yjuAAn~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-5-fluoro-n~4~-(1h-indazol-4-yl)-n~4~-methylpyrimidine-2,4-diamineHuman6112
SYKSykTK4yjuABn~2~-(1,1-dioxido-2,3-dihydro-1,2-benzothiazol-6-yl)-5-fluoro-n~4~-(1h-indazol-4-yl)-n~4~-methylpyrimidine-2,4-diamineHuman6121
SYKSykTK4yjvAA3-[6-({4-[ethyl(1h-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1h-indazol-1-yl]propan-1-olHuman6150
SYKSykTK4yjvAB3-[6-({4-[ethyl(1h-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1h-indazol-1-yl]propan-1-olHuman6148
SYKSykTK4yjvAC3-[6-({4-[ethyl(1h-indazol-4-yl)amino]-5-fluoropyrimidin-2-yl}amino)-2,4-dihydro-1h-indazol-1-yl]propan-1-olHuman6149
SYKSykTK5c26A3-{8-[(3,4-dimethoxyphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzamideHuman6131
SYKSykTK5c27A3-{8-[(3,4-dimethoxyphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}-n-[4-(methylcarbamoyl)phenyl]benzamideHuman6132
SYKSykTK5cxhA(4r)-4-[(1r)-1-{[6-(3,4-dimethoxyphenyl)[1,3]thiazolo[5,4-c]pyridin-4-yl]oxy}ethyl]pyrrolidin-2-oneHuman6057
SYKSykTK5cxzAAn-{7-[4-(dimethylamino)phenyl]-1,6-naphthyridin-5-yl}propane-1,3-diamineHuman6040
SYKSykTK5cxzABn-{7-[4-(dimethylamino)phenyl]-1,6-naphthyridin-5-yl}propane-1,3-diamineHuman6041
SYKSykTK5cy3AA(5r)-5-[(1r)-1-{[6-(1-methyl-1h-pyrazol-4-yl)-2,1-benzothiazol-4-yl]oxy}ethyl]-1,3-oxazolidin-2-oneHuman6058
SYKSykTK5cy3AB(5r)-5-[(1r)-1-{[6-(1-methyl-1h-pyrazol-4-yl)-2,1-benzothiazol-4-yl]oxy}ethyl]-1,3-oxazolidin-2-oneHuman6056
SYKSykTK5ghvA1-({1-[2-({3,5-dimethyl-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}amino)pyrimidin-4-yl]-4-methyl-1h-pyrrol-3-yl}methyl)azetidin-3-olHuman6743
SYKSykTK5ghvB1-({1-[2-({3,5-dimethyl-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}amino)pyrimidin-4-yl]-4-methyl-1h-pyrrol-3-yl}methyl)azetidin-3-olHuman6742
SYKSykTK5lmaAA~{n}'-[7-(4-methylphenyl)pyrido[3,4-b]pyrazin-5-yl]butane-1,4-diamineHuman7047
SYKSykTK5lmaAB~{n}'-[7-(4-methylphenyl)pyrido[3,4-b]pyrazin-5-yl]butane-1,4-diamineHuman7049
SYKSykTK5lmaAC~{n}'-[7-(4-methylphenyl)pyrido[3,4-b]pyrazin-5-yl]butane-1,4-diamineHuman7044
SYKSykTK5lmbAA7-[6-(dimethylamino)pyridin-3-yl]-~{n}-[[(3~{s})-piperidin-3-yl]methyl]pyrido[3,4-b]pyrazin-5-amineHuman7050
SYKSykTK5lmbAB7-[6-(dimethylamino)pyridin-3-yl]-~{n}-[[(3~{s})-piperidin-3-yl]methyl]pyrido[3,4-b]pyrazin-5-amineHuman7046
SYKSykTK5lmbBA7-[6-(dimethylamino)pyridin-3-yl]-~{n}-[[(3~{s})-piperidin-3-yl]methyl]pyrido[3,4-b]pyrazin-5-amineHuman7045
SYKSykTK5lmbBB7-[6-(dimethylamino)pyridin-3-yl]-~{n}-[[(3~{s})-piperidin-3-yl]methyl]pyrido[3,4-b]pyrazin-5-amineHuman7048
SYKSykTK5t68An~4~-cyclopropyl-n~2~-(3-methyl-1h-indazol-6-yl)furo[3,2-d]pyrimidine-2,4-diamineHuman7119
SYKSykTK5t68Bn~4~-cyclopropyl-n~2~-(3-methyl-1h-indazol-6-yl)furo[3,2-d]pyrimidine-2,4-diamineHuman7120
SYKSykTK5tiuAA5-{[(2s)-2-aminopropyl]amino}-3-(1h-indol-2-yl)pyrazine-2-carboxamideHuman7350
SYKSykTK5tiuAB5-{[(2s)-2-aminopropyl]amino}-3-(1h-indol-2-yl)pyrazine-2-carboxamideHuman7349
SYKSykTK5tr6AA6-{[(1r,2s)-2-aminocyclohexyl]amino}-7-fluoro-4-(1-methyl-1h-pyrazol-4-yl)-1,2-dihydro-3h-pyrrolo[3,4-c]pyridin-3-oneHuman7282
SYKSykTK5tr6AB6-{[(1r,2s)-2-aminocyclohexyl]amino}-7-fluoro-4-(1-methyl-1h-pyrazol-4-yl)-1,2-dihydro-3h-pyrrolo[3,4-c]pyridin-3-oneHuman7284
SYKSykTK5tt7AA2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(3-methylphenyl)amino]-6,7-dihydro-5h-pyrrolo[3,4-d]pyrimidin-5-oneHuman7281
SYKSykTK5tt7AB2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-[(3-methylphenyl)amino]-6,7-dihydro-5h-pyrrolo[3,4-d]pyrimidin-5-oneHuman7283
SYKSykTK5y5tA2-[[(1s,2s)-2-azanylcyclohexyl]amino]-4-[(4-methylsulfonylphenyl)amino]-6h-pyrido[4,3-d]pyrimidin-5-oneHuman10028
SYKSykTK5y5uA4-[(1-methylindazol-5-yl)amino]-2-(4-oxidanylpiperidin-1-yl)-8h-pyrido[4,3-d]pyrimidin-5-oneHuman10027
SYKSykTK5y5uB4-[(1-methylindazol-5-yl)amino]-2-(4-oxidanylpiperidin-1-yl)-8h-pyrido[4,3-d]pyrimidin-5-oneHuman10029
SYKSykTK6hm6AA2-(4-methylphenyl)-3-(pyridin-2-ylmethoxy)pyridineHuman10614
SYKSykTK6hm6AB2-(4-methylphenyl)-3-(pyridin-2-ylmethoxy)pyridineHuman10613
SYKSykTK6hm7AA7-[2-methoxy-6-[(4-methylpyridin-2-yl)methoxy]phenyl]-2,3,4,5-tetrahydro-1~{h}-3-benzazepineHuman10612
SYKSykTK6hm7AB7-[2-methoxy-6-[(4-methylpyridin-2-yl)methoxy]phenyl]-2,3,4,5-tetrahydro-1~{h}-3-benzazepineHuman10615
SYKSykTK6ssbA~{n}-[4-[5-[(dimethylamino)methyl]-1-methyl-pyrazol-3-yl]pyrimidin-2-yl]-3-methyl-1-(5-methyl-1,3,4-oxadiazol-2-yl)imidazo[1,5-a]pyridin-7-amineHuman12817
SYKSykTK6vovA6-(6-aminopyrazin-2-yl)-n-{4-[4-(oxetan-3-yl)piperazin-1-yl]phenyl}imidazo[1,2-a]pyrazin-8-amineHuman12041
SYKSykTK6vovB6-(6-aminopyrazin-2-yl)-n-{4-[4-(oxetan-3-yl)piperazin-1-yl]phenyl}imidazo[1,2-a]pyrazin-8-amineHuman12040
SYKSykTK6zc0A~{n},~{n}-dimethyl-1-[1-[2-(1-methylindol-4-yl)-3~{h}-imidazo[4,5-b]pyridin-7-yl]pyrazol-4-yl]methanamineHuman13636
SYKSykTK6zcpA7-[[4-[4-[(dimethylamino)methyl]pyrazol-1-yl]pyrimidin-2-yl]amino]-~{n},3-dimethyl-imidazo[1,5-a]pyridine-1-carboxamideHuman13632
SYKSykTK6zcqA7-[[4-[4-[[(3~{r},4~{r})-3-azanyloxan-4-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]-~{n},3-dimethyl-imidazo[1,5-a]pyridine-1-carboxamideHuman13633
SYKSykTK6zcrAA6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amineHuman13630
SYKSykTK6zcrAB6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amineHuman13631
SYKSykTK6zcsAA(3~{r},4~{r})-~{n}4-[1-[2-(1-methylindol-4-yl)-3~{h}-imidazo[4,5-b]pyridin-7-yl]pyrazol-4-yl]oxane-3,4-diamineHuman13639
SYKSykTK6zcsAB(3~{r},4~{r})-~{n}4-[1-[2-(1-methylindol-4-yl)-3~{h}-imidazo[4,5-b]pyridin-7-yl]pyrazol-4-yl]oxane-3,4-diamineHuman13641
SYKSykTK6zcuAA6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amineHuman13640
SYKSykTK6zcuAB6-chloro-2-(2-fluoro-4,5-dimethoxyphenyl)-n-(piperidin-4-ylmethyl)-3h-imidazo[4,5-b]pyridin-7-amineHuman13635
SYKSykTK6zcxAA~{n},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{r})-piperidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamideHuman13642
SYKSykTK6zcxAB~{n},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{r})-piperidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamideHuman13637
SYKSykTK6zcyAA~{n},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{r})-pyrrolidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamideHuman13634
SYKSykTK6zcyAB~{n},1-dimethyl-5-[[4-[3-methyl-4-[[(3~{r})-pyrrolidin-3-yl]amino]pyrazol-1-yl]pyrimidin-2-yl]amino]indazole-3-carboxamideHuman13638
SYKSykTK8bi2A10,13,23-trimethyl-16-oxa-2,4,8,9,13,19,23,30-octazapentacyclo[19.5.2.1^{3,7}.1^{8,11}.0^{24,28}]triaconta-1(27),3,5,7(30),9,11(29),21,24(28),25-nonaen-20-oneHuman14779
SYKSykTK8x5kAA2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamideHuman15103
SYKSykTK8x5kAB2-{[(1r,2s)-2-aminocyclohexyl]amino}-4-{[3-(2h-1,2,3-triazol-2-yl)phenyl]amino}pyrimidine-5-carboxamideHuman15102
TAOK3 (TAO3)STE20STE6bdnAAadenosine-5'-diphosphateHuman11004
TAOK3 (TAO3)STE20STE6bdnABadenosine-5'-diphosphateHuman11003
Tbk1 (TBK1)IKKOther4jl9An-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse5697
Tbk1 (TBK1)IKKOther4jlcA3-{2,4-dimethyl-5-[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-1h-pyrrol-3-yl}propanoic acidMouse5698
Tbk1 (TBK1)IKKOther6o8cAAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse11303
Tbk1 (TBK1)IKKOther6o8cABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse11302
Tbk1 (TBK1)IKKOther6o8cBAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse11305
Tbk1 (TBK1)IKKOther6o8cBBn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse11304
TBK1IKKOther4eutAAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman609
TBK1IKKOther4eutABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman621
TBK1IKKOther4eutBAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman618
TBK1IKKOther4eutBBn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman617
TBK1IKKOther4euuAAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman615
TBK1IKKOther4euuABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman611
TBK1IKKOther4euuBAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman606
TBK1IKKOther4euuBBn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman616
TBK1IKKOther4im0AAn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman610
TBK1IKKOther4im0ABn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman607
TBK1IKKOther4im2AAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman620
TBK1IKKOther4im2ABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman613
TBK1IKKOther4im3AAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman619
TBK1IKKOther4im3ABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman622
TBK1IKKOther4iw0An-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman608
TBK1IKKOther4iwoAn-{3-[(5-cyclopropyl-2-{[3-(2-oxopyrrolidin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman614
TBK1IKKOther4iwpAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman612
TBK1IKKOther4iwqAn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman605
TBK1IKKOther5w5vA2-amino-7-(1-methylethyl)-5-oxo-5h-chromeno[2,3-b]pyridine-3-carboxylic acidHuman10024
TBK1IKKOther6bnyA2-amino-7-(propan-2-yl)-3-(1h-tetrazol-5-yl)-5h-[1]benzopyrano[2,3-b]pyridin-5-oneHuman10369
TBK1IKKOther6bodAethyl 2-amino-5-oxo-7-(propan-2-yl)-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylateHuman10370
TBK1IKKOther6boeA2-amino-5-oxo-7-(propan-2-yl)-n-(1h-tetrazol-5-yl)-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxamideHuman10371
TBK1IKKOther6cq0A2-amino-7-[3-(dimethylamino)propyl]-5-oxo-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acidHuman10756
TBK1IKKOther6cq4A2-amino-7-(4,4-difluorocyclohexyl)-5-oxo-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acidHuman10757
TBK1IKKOther6cq5A2-amino-7-(1,1-dioxo-1lambda~6~-thian-4-yl)-5-oxo-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acidHuman10758
TBK1IKKOther6nt9A-Human10940
TBK1IKKOther6nt9B-Human10941
TBK1IKKOther6o8bAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman11053
TBK1IKKOther6o8bBn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman11054
TBK1IKKOther6rsrA~{n}-(cyclopropen-1-ylmethyl)-2-[[4-[[4-[3,3,3-tris(fluoranyl)propanoyl]piperazin-1-yl]methyl]pyridin-2-yl]amino]-1~{h}-benzimidazole-5-carboxamideHuman11903
TBK1IKKOther6rstA1-[4-[(1~{r})-1-[2-[[5-[1-(cyclopropylmethyl)pyrazol-4-yl]-1~{h}-benzimidazol-2-yl]amino]pyridin-4-yl]ethyl]piperazin-1-yl]-3,3,3-tris(fluoranyl)propan-1-oneHuman11902
TBK1IKKOther6rsuA3,3,3-tris(fluoranyl)-1-[4-[(1~{r})-1-[2-[[(2~{s})-5-(5-propan-2-yloxypyrimidin-4-yl)-2,3-dihydro-1~{h}-benzimidazol-2-yl]amino]pyridin-4-yl]ethyl]piperazin-1-yl]propan-1-oneHuman12126
TEK (TIE2)TieTK1fvrA-Human5551
TEK (TIE2)TieTK1fvrB-Human5554
TEK (TIE2)TieTK2oo8Xn-{3-[3-(dimethylamino)propyl]-5-(trifluoromethyl)phenyl}-4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]benzamideHuman5556
TEK (TIE2)TieTK2oscAn-{4-methyl-3-[(3-pyrimidin-4-ylpyridin-2-yl)amino]phenyl}-3-(trifluoromethyl)benzamideHuman5555
TEK (TIE2)TieTK2p4iA4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)-n-[2-morpholin-4-yl-5-(trifluoromethyl)phenyl]benzamideHuman5549
TEK (TIE2)TieTK2p4iB4-methyl-3-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)-n-[2-morpholin-4-yl-5-(trifluoromethyl)phenyl]benzamideHuman5550
TEK (TIE2)TieTK2wqbA2-[3-(cyclohexylmethyl)-5-phenyl-imidazol-4-yl]-[1,3]thiazolo[4,5-e]pyrimidin-7-amineHuman5553
TEK (TIE2)TieTK3l8pA2-methyl-11-(1-methylethyl)-8-[(2s)-tetrahydro-2h-pyran-2-yl]-2,11,12,13-tetrahydro-4h-indazolo[5,4-a]pyrrolo[3,4-c]carbazol-4-oneHuman5548
TEK (TIE2)TieTK4x3jA1-[4-(4-amino-5-oxopyrido[2,3-d]pyrimidin-8(5h)-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]ureaHuman5552
TEK (TIE2)TieTK6mweAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman10710
TEK (TIE2)TieTK6mweAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman10711
TEK (TIE2)TieTK6mweBA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman10712
TEK (TIE2)TieTK6mweBB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman10713
TGFBR1 (TGFbR1)STKRTKL1b6cB-Human2133
TGFBR1 (TGFbR1)STKRTKL1b6cD-Human2126
TGFBR1 (TGFbR1)STKRTKL1b6cF-Human2103
TGFBR1 (TGFbR1)STKRTKL1b6cH-Human2099
TGFBR1 (TGFbR1)STKRTKL1iasA-Human2113
TGFBR1 (TGFbR1)STKRTKL1iasB-Human2102
TGFBR1 (TGFbR1)STKRTKL1iasC-Human2117
TGFBR1 (TGFbR1)STKRTKL1iasD-Human2131
TGFBR1 (TGFbR1)STKRTKL1iasE-Human2134
TGFBR1 (TGFbR1)STKRTKL1py5A4-(3-pyridin-2-yl-1h-pyrazol-4-yl)quinolineHuman2094
TGFBR1 (TGFbR1)STKRTKL1rw8A3-(4-fluorophenyl)-2-(6-methylpyridin-2-yl)-5,6-dihydro-4h-pyrrolo[1,2-b]pyrazoleHuman2100
TGFBR1 (TGFbR1)STKRTKL1vjyA2-[5-(6-methylpyridin-2-yl)-2,3-dihydro-1h-pyrazol-4-yl]-1,5-naphthyridineHuman2096
TGFBR1 (TGFbR1)STKRTKL2wotAA4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amineHuman2120
TGFBR1 (TGFbR1)STKRTKL2wotAB4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amineHuman2092
TGFBR1 (TGFbR1)STKRTKL2wouA4-({4-[(2,6-dimethylpyridin-3-yl)oxy]pyridin-2-yl}amino)benzenesulfonamideHuman2125
TGFBR1 (TGFbR1)STKRTKL2x7oA(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2127
TGFBR1 (TGFbR1)STKRTKL2x7oB(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2128
TGFBR1 (TGFbR1)STKRTKL2x7oC(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2104
TGFBR1 (TGFbR1)STKRTKL2x7oD(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2107
TGFBR1 (TGFbR1)STKRTKL2x7oE(3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamideHuman2097
TGFBR1 (TGFbR1)STKRTKL3faaAn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2118
TGFBR1 (TGFbR1)STKRTKL3faaBn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2108
TGFBR1 (TGFbR1)STKRTKL3faaCn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2130
TGFBR1 (TGFbR1)STKRTKL3faaDn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2132
TGFBR1 (TGFbR1)STKRTKL3faaEn-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamideHuman2098
TGFBR1 (TGFbR1)STKRTKL3gxlAn-1h-indazol-5-yl-2-(6-methylpyridin-2-yl)quinazolin-4-amineHuman2116
TGFBR1 (TGFbR1)STKRTKL3hmmA2-(6-methylpyridin-2-yl)-n-pyridin-4-ylquinazolin-4-amineHuman2111
TGFBR1 (TGFbR1)STKRTKL3kcfA4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2112
TGFBR1 (TGFbR1)STKRTKL3kcfB4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2106
TGFBR1 (TGFbR1)STKRTKL3kcfC4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2093
TGFBR1 (TGFbR1)STKRTKL3kcfD4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2119
TGFBR1 (TGFbR1)STKRTKL3kcfE4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-oneHuman2105
TGFBR1 (TGFbR1)STKRTKL3tzmAA4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamideHuman2095
TGFBR1 (TGFbR1)STKRTKL3tzmAB4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamideHuman2110
TGFBR1 (TGFbR1)STKRTKL4x0mAA4-aminopyrido[2,3-d]pyrimidin-5(8h)-oneHuman2122
TGFBR1 (TGFbR1)STKRTKL4x0mAB4-aminopyrido[2,3-d]pyrimidin-5(8h)-oneHuman2121
TGFBR1 (TGFbR1)STKRTKL4x2fAA4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-oneHuman6207
TGFBR1 (TGFbR1)STKRTKL4x2fAB4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-oneHuman6208
TGFBR1 (TGFbR1)STKRTKL4x2gAA4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-oneHuman2123
TGFBR1 (TGFbR1)STKRTKL4x2gAB4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-oneHuman2114
TGFBR1 (TGFbR1)STKRTKL4x2jAA4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-oneHuman2124
TGFBR1 (TGFbR1)STKRTKL4x2jAB4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-oneHuman2115
TGFBR1 (TGFbR1)STKRTKL4x2kAA4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-oneHuman2135
TGFBR1 (TGFbR1)STKRTKL4x2kAB4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-oneHuman2101
TGFBR1 (TGFbR1)STKRTKL4x2nAA-Human2129
TGFBR1 (TGFbR1)STKRTKL4x2nAB-Human2109
TGFBR1 (TGFbR1)STKRTKL5e8sAA-Human6619
TGFBR1 (TGFbR1)STKRTKL5e8sAB-Human6609
TGFBR1 (TGFbR1)STKRTKL5e8tAA-Human6608
TGFBR1 (TGFbR1)STKRTKL5e8tAB-Human6613
TGFBR1 (TGFbR1)STKRTKL5e8uA-Human6616
TGFBR1 (TGFbR1)STKRTKL5e8wAAstaurosporineHuman6611
TGFBR1 (TGFbR1)STKRTKL5e8wABstaurosporineHuman6614
TGFBR1 (TGFbR1)STKRTKL5e8xAAstaurosporineHuman6615
TGFBR1 (TGFbR1)STKRTKL5e8xABstaurosporineHuman6617
TGFBR1 (TGFbR1)STKRTKL5e8zAA3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamideHuman6618
TGFBR1 (TGFbR1)STKRTKL5e8zAB3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamideHuman6612
TGFBR1 (TGFbR1)STKRTKL5e90AA3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamideHuman6610
TGFBR1 (TGFbR1)STKRTKL5e90AB3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamideHuman6607
TGFBR1 (TGFbR1)STKRTKL5friAAn-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamideHuman6894
TGFBR1 (TGFbR1)STKRTKL5friABn-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamideHuman6893
TGFBR1 (TGFbR1)STKRTKL5qikAAn-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamideHuman10657
TGFBR1 (TGFbR1)STKRTKL5qikABn-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamideHuman10662
TGFBR1 (TGFbR1)STKRTKL5qilAAn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10659
TGFBR1 (TGFbR1)STKRTKL5qilABn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10660
TGFBR1 (TGFbR1)STKRTKL5qimAAn-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10658
TGFBR1 (TGFbR1)STKRTKL5qimABn-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10661
TGFBR1 (TGFbR1)STKRTKL5qtzAA6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridineHuman11965
TGFBR1 (TGFbR1)STKRTKL5qtzAB6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridineHuman11966
TGFBR1 (TGFbR1)STKRTKL5qu0AA6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrileHuman11967
TGFBR1 (TGFbR1)STKRTKL5qu0AB6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrileHuman11964
TGFBR1 (TGFbR1)STKRTKL5usqAAn-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amineHuman7558
TGFBR1 (TGFbR1)STKRTKL5usqABn-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amineHuman7557
TGFBR1 (TGFbR1)STKRTKL6b8yAAn-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman9553
TGFBR1 (TGFbR1)STKRTKL6b8yABn-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman9552
TGFBR2 (TGFbR2)STKRTKL5e8vAA-Human6626
TGFBR2 (TGFbR2)STKRTKL5e8vAB-Human6622
TGFBR2 (TGFbR2)STKRTKL5e8yAstaurosporineHuman6627
TGFBR2 (TGFbR2)STKRTKL5e91A3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamideHuman6625
TGFBR2 (TGFbR2)STKRTKL5e92AAphosphoaminophosphonic acid-adenylate esterHuman6624
TGFBR2 (TGFbR2)STKRTKL5e92ABphosphoaminophosphonic acid-adenylate esterHuman6623
TGFBR2 (TGFbR2)STKRTKL5qinAAn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10664
TGFBR2 (TGFbR2)STKRTKL5qinABn-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamideHuman10663
TGFBR2 (TGFbR2)STKRTKL7dv6AA5-[(3s)-5,5-dimethyloxolan-3-yl]-6-methoxy-3-(2-methoxypyridin-4-yl)pyrazolo[1,5-a]pyrimidineHuman13629
TGFBR2 (TGFbR2)STKRTKL7dv6AB5-[(3s)-5,5-dimethyloxolan-3-yl]-6-methoxy-3-(2-methoxypyridin-4-yl)pyrazolo[1,5-a]pyrimidineHuman13628
TLK2TLKOther5o0yAphosphothiophosphoric acid-adenylate esterHuman9943
TNIKSTE20STE2x7fAA9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1943
TNIKSTE20STE2x7fAB9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1951
TNIKSTE20STE2x7fBA9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1950
TNIKSTE20STE2x7fBB9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1947
TNIKSTE20STE2x7fCA9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1942
TNIKSTE20STE2x7fCB9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1948
TNIKSTE20STE2x7fDA9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1944
TNIKSTE20STE2x7fDB9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1945
TNIKSTE20STE2x7fEA9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1946
TNIKSTE20STE2x7fEB9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman1949
TNIKSTE20STE5ax9A4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrileHuman6887
TNIKSTE20STE5ax9B4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrileHuman6892
TNIKSTE20STE5ax9C4-methoxy-3-[2-[(3-methoxy-4-morpholin-4-yl-phenyl)amino]pyridin-4-yl]benzenecarbonitrileHuman6889
TNIKSTE20STE5cwzA-Human6891
TNIKSTE20STE5cwzB-Human6890
TNIKSTE20STE5cwzC-Human6888
TNIKSTE20STE5d7aAcis-4-{[2-(1h-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanolHuman6963
TNIKSTE20STE5d7aBcis-4-{[2-(1h-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanolHuman6964
TNIKSTE20STE5d7aCcis-4-{[2-(1h-benzimidazol-5-ylamino)quinazolin-8-yl]oxy}cyclohexanolHuman6965
TNIKSTE20STE6ra5A5-bromanyl-2-(2-fluoranylpyridin-4-yl)-1,7-naphthyridin-8-amineHuman12238
TNIKSTE20STE6ra5B-Human12237
TNIKSTE20STE6ra7AA2-[8-azanyl-2-(2-fluoranylpyridin-4-yl)-1,7-naphthyridin-5-yl]propan-2-olHuman11801
TNIKSTE20STE6ra7AB2-[8-azanyl-2-(2-fluoranylpyridin-4-yl)-1,7-naphthyridin-5-yl]propan-2-olHuman11800
TNIKSTE20STE7xzqA-Human14474
TNIKSTE20STE7xzrAAphosphoaminophosphonic acid-adenylate esterHuman14476
TNIKSTE20STE7xzrABphosphoaminophosphonic acid-adenylate esterHuman14475
TNIKSTE20STE8x88A-Human15060
TNK2 (ACK)AckTK1u46A-Human3411
TNK2 (ACK)AckTK1u46B-Human3408
TNK2 (ACK)AckTK1u4dAdebromohymenialdisineHuman3398
TNK2 (ACK)AckTK1u4dBdebromohymenialdisineHuman3392
TNK2 (ACK)AckTK1u54Aphosphomethylphosphonic acid adenylate esterHuman3409
TNK2 (ACK)AckTK1u54Bphosphomethylphosphonic acid adenylate esterHuman3397
TNK2 (ACK)AckTK3eqpAn-(2,6-dimethylphenyl)-4-(2-ethoxyphenoxy)-2-({4-[4-(2-hydroxyethyl)piperazin-1-yl]phenyl}amino)pyrimidine-5-carboxamideHuman3403
TNK2 (ACK)AckTK3eqpBn-(2,6-dimethylphenyl)-4-(2-ethoxyphenoxy)-2-({4-[4-(2-hydroxyethyl)piperazin-1-yl]phenyl}amino)pyrimidine-5-carboxamideHuman3402
TNK2 (ACK)AckTK3eqrAn~3~-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl)-n~6~-(4-piperazin-1-ylphenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,6-diamineHuman3395
TNK2 (ACK)AckTK3eqrBn~3~-(2,6-dimethylphenyl)-1-(3-methoxy-3-methylbutyl)-n~6~-(4-piperazin-1-ylphenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,6-diamineHuman3406
TNK2 (ACK)AckTK4ewhA6-{4-[2-(dimethylamino)ethoxy]phenyl}-n-(1,3-dithiolan-2-ylmethyl)-5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman3410
TNK2 (ACK)AckTK4ewhB6-{4-[2-(dimethylamino)ethoxy]phenyl}-n-(1,3-dithiolan-2-ylmethyl)-5-phenyl-7h-pyrrolo[2,3-d]pyrimidin-4-amineHuman3405
TNK2 (ACK)AckTK4hzrAA-Human3394
TNK2 (ACK)AckTK4hzrAB-Human3399
TNK2 (ACK)AckTK4hzrBA-Human3396
TNK2 (ACK)AckTK4hzrBB-Human3391
TNK2 (ACK)AckTK4hzsA-Human3407
TNK2 (ACK)AckTK4hzsB-Human3400
TNK2 (ACK)AckTK4hzsC-Human3393
TNK2 (ACK)AckTK4hzsD-Human3404
TNK2 (ACK)AckTK4id7Acis-3-[8-amino-1-(4-phenoxyphenyl)imidazo[1,5-a]pyrazin-3-yl]cyclobutanolHuman3401
TNK2 (ACK)AckTK5zxbAAn-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamideHuman10492
TNK2 (ACK)AckTK5zxbABn-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamideHuman10494
TNK2 (ACK)AckTK5zxbBAn-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamideHuman10493
TNK2 (ACK)AckTK5zxbBBn-{3-[7-{[6-(4-acetylpiperazin-1-yl)pyridin-3-yl]amino}-1-methyl-2-oxo-1,4-dihydropyrimido[4,5-d]pyrimidin-3(2h)-yl]-4-methylphenyl}-3-(trifluoromethyl)benzamideHuman10495
TNK2 (ACK)AckTK6vqmA2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6h-pyrimido[5,4-d][1,3]benzodiazepin-6-oneHuman13289
TNK2 (ACK)AckTK6vqmB2-({4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]-2-methoxyphenyl}amino)-9-methyl-5,7-dihydro-6h-pyrimido[5,4-d][1,3]benzodiazepin-6-oneHuman13290
TNK2 (ACK)AckTK7kp6AA5-chloro-n~2~-[4-(4-methylpiperazin-1-yl)phenyl]-n~4~-{[(2r)-oxolan-2-yl]methyl}pyrimidine-2,4-diamineHuman14104
TNK2 (ACK)AckTK7kp6AB5-chloro-n~2~-[4-(4-methylpiperazin-1-yl)phenyl]-n~4~-{[(2r)-oxolan-2-yl]methyl}pyrimidine-2,4-diamineHuman14103
TNK2 (ACK)AckTK8fe9An-[(1s)-1-benzyl-2-[(6-chloro-2-oxo-1h-quinolin-4-yl)methylamino]-2-oxo-ethyl]-4-hydroxy-2-oxo-1h-quinoline-6-carboHuman14676
TNK2 (ACK)AckTK8hmtAA6-(2-bromophenyl)-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[[(2s)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-7-oneHuman15009
TNK2 (ACK)AckTK8hmtAB6-(2-bromophenyl)-2-[[3-methyl-4-(4-methylpiperazin-1-yl)phenyl]amino]-8-[[(2s)-oxolan-2-yl]methyl]pyrido[2,3-d]pyrimidin-7-oneHuman15010
TNNI3K (HH498)MLKTKL4yffAA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6068
TNNI3K (HH498)MLKTKL4yffAB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6062
TNNI3K (HH498)MLKTKL4yffBA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6065
TNNI3K (HH498)MLKTKL4yffBB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6063
TNNI3K (HH498)MLKTKL4yffCA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6069
TNNI3K (HH498)MLKTKL4yffCB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6067
TNNI3K (HH498)MLKTKL4yffDA3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6066
TNNI3K (HH498)MLKTKL4yffDB3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamideHuman6074
TNNI3K (HH498)MLKTKL4yfiAAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6059
TNNI3K (HH498)MLKTKL4yfiABn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6071
TNNI3K (HH498)MLKTKL4yfiBAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6061
TNNI3K (HH498)MLKTKL4yfiBBn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6060
TNNI3K (HH498)MLKTKL4yfiCAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6070
TNNI3K (HH498)MLKTKL4yfiCBn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6073
TNNI3K (HH498)MLKTKL4yfiDAn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6072
TNNI3K (HH498)MLKTKL4yfiDBn-methyl-3-(9h-purin-6-ylamino)benzenesulfonamideHuman6064
TNNI3K (HH498)MLKTKL6b5jAAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9791
TNNI3K (HH498)MLKTKL6b5jABn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9800
TNNI3K (HH498)MLKTKL6b5jACn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9798
TNNI3K (HH498)MLKTKL6b5jBAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9802
TNNI3K (HH498)MLKTKL6b5jBBn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9794
TNNI3K (HH498)MLKTKL6b5jBCn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9797
TNNI3K (HH498)MLKTKL6b5jCAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9799
TNNI3K (HH498)MLKTKL6b5jCBn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9793
TNNI3K (HH498)MLKTKL6b5jCCn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9796
TNNI3K (HH498)MLKTKL6b5jDAn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9792
TNNI3K (HH498)MLKTKL6b5jDBn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9801
TNNI3K (HH498)MLKTKL6b5jDCn-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamideHuman9795
TNNI3K (HH498)MLKTKL7mgjAn-methyl-4-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]pyridine-2-carboxamideHuman13969
TNNI3K (HH498)MLKTKL7mgkAAn-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]ureaHuman13968
TNNI3K (HH498)MLKTKL7mgkABn-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]ureaHuman13970
TP53RK (PRPK)Bud32Other6wqxCphosphoaminophosphonic acid-adenylate esterHuman13338
TP53RK (PRPK)Bud32Other6wqxDphosphoaminophosphonic acid-adenylate esterHuman13339
TP53RK (PRPK)Bud32Other7szaAA4-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dioneHuman14597
TP53RK (PRPK)Bud32Other7szaAB4-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dioneHuman14599
TP53RK (PRPK)Bud32Other7szbA5-amino-2-[(3r)-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dioneHuman14598
TP53RK (PRPK)Bud32Other7szcA4-hydroxy-2-[(3r)-3-methyl-2,6-dioxopiperidin-3-yl]-1h-isoindole-1,3(2h)-dioneHuman14559
TP53RK (PRPK)Bud32Other7szdA2-[(3r)-3-methyl-2,6-dioxopiperidin-3-yl]-1,3-dioxo-2,3-dihydro-1h-isoindole-5-carboxylic acidHuman14558
TRIB1 (Trb1)TrblCAMK5cekA-Human6241
TRIB1 (Trb1)TrblCAMK5cemAA-Human6242
TRIB1 (Trb1)TrblCAMK5cemAB-Human6243
TRIB1 (Trb1)TrblCAMK6dc0AA-Human10622
TRIB1 (Trb1)TrblCAMK6dc0AB-Human10623
TRIB1 (Trb1)TrblCAMK6dc0BA-Human10620
TRIB1 (Trb1)TrblCAMK6dc0BB-Human10621
TRIB2 (Trb2)TrblCAMK7upmA-Human14365
TRRAPPIKKAtypical8h7gA-Human14556
TTBK1TTBKCK14btjAadenosine-5'-diphosphateHuman769
TTBK1TTBKCK14btjBadenosine-5'-triphosphateHuman767
TTBK1TTBKCK14btkA4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman771
TTBK1TTBKCK14btmAmethyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoateHuman772
TTBK1TTBKCK14btmBmethyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoateHuman774
TTBK1TTBKCK14nfmA-Human768
TTBK1TTBKCK14nfnAA3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenolHuman773
TTBK1TTBKCK14nfnAB3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenolHuman770
TTBK1TTBKCK17jxxAA4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHuman13579
TTBK1TTBKCK17jxxAB4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHuman13578
TTBK1TTBKCK17jxyA(3s)-1-[1-(2-aminopyrimidin-4-yl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-methylpent-1-yn-3-olHuman13580
TTBK1TTBKCK17q8vA~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14133
TTBK1TTBKCK17q8wAA~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14134
TTBK1TTBKCK17q8wAB~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14135
TTBK1TTBKCK17qhwA~{n}-[4-(4-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14477
TTBK1TTBKCK17zhnAA4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHuman14721
TTBK1TTBKCK17zhnAB4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHuman14717
TTBK1TTBKCK17zhoAA4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-olHuman14718
TTBK1TTBKCK17zhoAB4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-olHuman14722
TTBK1TTBKCK17zhpAA1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-olHuman14724
TTBK1TTBKCK17zhpAB1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-olHuman14719
TTBK1TTBKCK17zhqAA(3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-olHuman14720
TTBK1TTBKCK17zhqAB(3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-olHuman14723
TTBK1TTBKCK18xpzA-Human15163
TTBK2TTBKCK16u0kAA4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman12046
TTBK2TTBKCK16u0kAB4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman12048
TTBK2TTBKCK16u0kBA4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman12049
TTBK2TTBKCK16u0kBB4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman12047
TTBK2TTBKCK16vrfAAadenosine-5'-diphosphateHuman12344
TTBK2TTBKCK16vrfABadenosine-5'-diphosphateHuman12343
TTBK2TTBKCK16vrfBAadenosine-5'-diphosphateHuman12345
TTBK2TTBKCK16vrfBBadenosine-5'-diphosphateHuman12342
TTBK2TTBKCK17q8yAA~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14141
TTBK2TTBKCK17q8yAB~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14138
TTBK2TTBKCK17q8zAA~{n}-(4-phenoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14142
TTBK2TTBKCK17q8zAB~{n}-(4-phenoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14140
TTBK2TTBKCK17q90AA~{n}-[4-(4-methoxyphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14139
TTBK2TTBKCK17q90AB~{n}-[4-(4-methoxyphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14143
TTKTTKOther2x9eAn-(2,6-diethylphenyl)-1-methyl-8-({4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(trifluoromethoxy)phenyl}amino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4729
TTKTTKOther2zmcA-Human4696
TTKTTKOther2zmdA2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHuman4731
TTKTTKOther3cekA-Human4716
TTKTTKOther3dbqA-Human4710
TTKTTKOther3gfwA1-(4-(4-(2-(isopropylsulfonyl)phenylamino)-1h-pyrrolo[2,3-b]pyridin-6-ylamino)-3-methoxyphenyl)piperidin-4-olHuman4714
TTKTTKOther3h9fAA9-cyclopentyl-2-(4-(4-hydroxypiperidin-1-yl)-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5h-pyrimido[4,5-b][1,4]diazepin-6(7h)-oneHuman4701
TTKTTKOther3h9fAB9-cyclopentyl-2-(4-(4-hydroxypiperidin-1-yl)-2-methoxyphenylamino)-5-methyl-8,9-dihydro-5h-pyrimido[4,5-b][1,4]diazepin-6(7h)-oneHuman4712
TTKTTKOther3hmnAadenosine-5'-triphosphateHuman4719
TTKTTKOther3hmoAstaurosporineHuman4707
TTKTTKOther3hmpA7-chloro-n-(cyclopropylmethyl)quinazolin-4-amineHuman4728
TTKTTKOther3vquA4-[(4-amino-5-cyano-6-ethoxypyridin-2-yl)amino]benzamideHuman4718
TTKTTKOther3w1fA5-[5-ethoxy-6-(1-methyl-1h-pyrazol-4-yl)-1h-indazol-3-yl]-2-methylbenzenesulfonamideHuman4722
TTKTTKOther3wyxA6-{[3-(cyanomethoxy)-4-(1-methyl-1h-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrileHuman4721
TTKTTKOther3wyyA(2e)-3-[4-({4-amino-5-cyano-6-[(3s,5s,7s)-tricyclo[3.3.1.1~3,7~]dec-1-ylamino]pyridin-2-yl}amino)-2-(cyanomethoxy)phenyl]-n-(2-methoxyethyl)prop-2-enamideHuman4711
TTKTTKOther3wzjA4-{6-(cyclohexylamino)-8-[(tetrahydro-2h-pyran-4-ylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}-n-cyclopropylbenzamideHuman4704
TTKTTKOther3wzkAn-cyclopropyl-4-{8-[(thiophen-2-ylmethyl)amino]imidazo[1,2-a]pyrazin-3-yl}benzamideHuman4703
TTKTTKOther4bhzAthieno[2,3-c][2,6]naphthyridineHuman4709
TTKTTKOther4bi0A5h-pyrimido[5,4-b]indoleHuman4702
TTKTTKOther4bi1Athieno[3,2-c][2,6]naphthyridineHuman4699
TTKTTKOther4bi2Athieno[2,3-c][2,7]naphthyridineHuman4700
TTKTTKOther4c4eAAn-(3,4-dimethoxyphenyl)-2-(1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4708
TTKTTKOther4c4eAB-Human4726
TTKTTKOther4c4fAn-(2-methoxyphenyl)-2-(1,3-oxazol-5-yl)-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4715
TTKTTKOther4c4gAtert-butyl 6-((2-chloro-4-(dimethylcarbamoyl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylateHuman4697
TTKTTKOther4c4hAtert-butyl 6-((2-chloro-4-(dimethylcarbamoyl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylateHuman4725
TTKTTKOther4c4iAtert-butyl 6-{[2-chloro-4-(dimethylcarbamoyl)phenyl]amino}-2-(1,3-oxazol-5-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylateHuman4698
TTKTTKOther4c4jAtert-butyl 6-{[2-chloro-4-(1-methyl-1h-imidazol-5-yl)phenyl]amino}-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylateHuman4723
TTKTTKOther4cv8A3-amino-5-(1-methyl-1h-pyrazol-4-yl)pyridin-2(1h)-oneHuman4706
TTKTTKOther4cv9A4-(4-methylpiperazin-1-yl)-n-(2-oxo-5-(pyridin-4-yl)-1,2-dihydropyridin-3-yl)benzamideHuman4705
TTKTTKOther4cvaAn-(6-oxo-1,6-dihydro-3,4'-bipyridin-5-yl)-4-(piperidin-1-yl)benzamideHuman4713
TTKTTKOther4d2sAn-{2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]phenyl}-4-(1h-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman4717
TTKTTKOther4js8A4-(cyclohexylmethoxy)-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-2h-indazoleHuman4724
TTKTTKOther4jt3A2-phenyl-n-[3-(3-sulfamoylphenyl)-2h-indazol-5-yl]acetamideHuman4727
TTKTTKOther4o6lAn-[(1r)-1-(2-chlorophenyl)propyl]-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1h-indazole-5-carboxamideHuman4730
TTKTTKOther4o6lBn-[(1r)-1-(2-chlorophenyl)propyl]-3-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1h-indazole-5-carboxamideHuman4720
TTKTTKOther4zegAn-cyclopropyl-2-methyl-4-(7-{[2-(morpholin-4-yl)ethyl]amino}-5-phenoxypyrazolo[1,5-a]pyrimidin-3-yl)benzamideHuman6574
TTKTTKOther5ap0A9-cyclopentyl-2-[[2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-phenyl]amino]-7-methyl-7,9-dihydro-8h-purin-8-oneHuman6101
TTKTTKOther5ap1A6-{[3-(cyanomethoxy)-4-(1-methyl-1h-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrileHuman6103
TTKTTKOther5ap2Aisopropyl 6-((4-(1,2-dimethyl-1h-imidazol-5-yl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylateHuman6105
TTKTTKOther5ap3A9-cyclopentyl-2-[[2-methoxy-4-[(1-methylpiperidin-4-yl)oxy]-phenyl]amino]-7-methyl-7,9-dihydro-8h-purin-8-oneHuman6099
TTKTTKOther5ap4A6-{[3-(cyanomethoxy)-4-(1-methyl-1h-pyrazol-4-yl)phenyl]amino}-2-(cyclohexylamino)pyridine-3-carbonitrileHuman6097
TTKTTKOther5ap5Atert-butyl 6-((2-chloro-4-(dimethylcarbamoyl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylateHuman6104
TTKTTKOther5ap6AAisopropyl 6-((4-(1,2-dimethyl-1h-imidazol-5-yl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylateHuman6098
TTKTTKOther5ap6ABisopropyl 6-((4-(1,2-dimethyl-1h-imidazol-5-yl)phenyl)amino)-2-(1-methyl-1h-pyrazol-4-yl)-1h-pyrrolo[3,2-c]pyridine-1-carboxylateHuman6102
TTKTTKOther5ap7An-(2,6-diethylphenyl)-1-methyl-8-({4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(trifluoromethoxy)phenyl}amino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman6100
TTKTTKOther5eh0An2-(2-methoxy-4-(1-methyl-1h-pyrazol-4-yl)phenyl)-n8-neopentylpyrido[3,4-d]pyrimidine-2,8-diamineHuman6850
TTKTTKOther5ehlA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman7256
TTKTTKOther5ehoA~{n}8-cyclohexyl-~{n}2-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]pyrido[3,4-d]pyrimidine-2,8-diamineHuman7257
TTKTTKOther5ehyA4-(furan-3-yl)-3-phenyl-2~{h}-pyrazolo[4,3-c]pyridineHuman6556
TTKTTKOther5ei2A~{n}-(2,4-dimethoxyphenyl)-8-(1-methylpyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amineHuman6559
TTKTTKOther5ei6A~{n}-(2,4-dimethoxyphenyl)-5-(1-methylpyrazol-4-yl)isoquinolin-3-amineHuman6558
TTKTTKOther5ei8A~{n}-[2-methoxy-4-(1-methylpyrazol-4-yl)phenyl]-8-(1-methylpyrazol-4-yl)pyrido[3,4-d]pyrimidin-2-amineHuman6557
TTKTTKOther5ljjAn~6~-cyclohexyl-n~2~-(4-morpholin-4-ylphenyl)-9h-purine-2,6-diamineHuman7092
TTKTTKOther5mrbA~{n}-(2,6-diethylphenyl)-8-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideHuman8270
TTKTTKOther5n7vA~{n}6-cyclohexyl-~{n}2-(2-methyl-4-morpholin-4-yl-phenyl)-7~{h}-purine-2,6-diamineHuman7978
TTKTTKOther5n84A~{n}-cyclopropyl-4-[8-(2-methylpropylamino)imidazo[1,2-a]pyrazin-3-yl]benzamideHuman7973
TTKTTKOther5n87A~{n}-(2,6-diethylphenyl)-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamideHuman7977
TTKTTKOther5n93A4-[[4-azanyl-6-(~{tert}-butylamino)-5-cyano-pyridin-2-yl]amino]benzamideHuman7976
TTKTTKOther5n9sA(2~{r})-2-(4-fluorophenyl)-~{n}-[4-[2-[(2-methoxy-4-methylsulfonyl-phenyl)amino]-[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl]propanamideHuman7979
TTKTTKOther5na0A~{n}-[3,5-diethyl-1-[2-[2-(2-methoxyethoxy)ethoxy]ethyl]pyrazol-4-yl]-2-[[2-methoxy-4-[4-(2-methoxyethanoyl)piperazin-1-yl]phenyl]amino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamideHuman7974
TTKTTKOther5nadAbay 1217389Human7975
TTKTTKOther5nttAAn-(2,6-diethylphenyl)-1-methyl-8-({4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(trifluoromethoxy)phenyl}amino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman8268
TTKTTKOther5nttABn-(2,6-diethylphenyl)-1-methyl-8-({4-[(1-methylpiperidin-4-yl)carbamoyl]-2-(trifluoromethoxy)phenyl}amino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman8267
TTKTTKOther5o91A~{n}-(2,6-diethylphenyl)-8-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideHuman8269
TTKTTKOther6b4wA4-{[4-(cyclopentyloxy)-5-(2-methyl-1,3-benzoxazol-6-yl)-7h-pyrrolo[2,3-d]pyrimidin-2-yl]amino}-3-methoxy-n-methylbenzamideHuman8616
TTKTTKOther6gvjA-Human10847
TTKTTKOther6h3kA~{n}8-(2,2-dimethylpropyl)-~{n}2-[2-ethoxy-4-(4-methyl-1,2,4-triazol-3-yl)phenyl]-6-methyl-pyrido[3,4-d]pyrimidine-2,8-diamineHuman10571
TTKTTKOther6n6oA4-({5-chloro-4-[(cis-4-hydroxy-4-methylcyclohexyl)oxy]-7h-pyrrolo[2,3-d]pyrimidin-2-yl}amino)-n,n-dimethyl-3-{[(2r)-1,1,1-trifluoropropan-2-yl]oxy}benzamideHuman11240
TTKTTKOther6tn9AA[4-[[6-(3,5-dimethyl-4-oxidanyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]amino]phenyl]-morpholin-4-yl-methanoneHuman12271
TTKTTKOther6tn9AB[4-[[6-(3,5-dimethyl-4-oxidanyl-phenyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]amino]phenyl]-morpholin-4-yl-methanoneHuman12269
TTKTTKOther6tnbA(2~{r})-2-(4-fluorophenyl)-~{n}-[4-[2-[(2-methoxy-4-methylsulfonyl-phenyl)amino]-[1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl]propanamideHuman12267
TTKTTKOther6tncAn-cyclopropyl-4-{8-[(thiophen-2-ylmethyl)amino]imidazo[1,2-a]pyrazin-3-yl}benzamideHuman12270
TTKTTKOther6tndAAbay 1217389Human12268
TTKTTKOther6tndABbay 1217389Human12272
TTKTTKOther7chmA4-(cyclohexylamino)-2-[(2-methoxy-4-morpholin-4-ylcarbonyl-phenyl)amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13550
TTKTTKOther7chnA4-(cyclohexylamino)-2-[[2-methoxy-4-(2-oxidanylidenepyrrolidin-1-yl)phenyl]amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13552
TTKTTKOther7chtA2-[[2-methoxy-4-(2-oxidanylidenepyrrolidin-1-yl)phenyl]amino]-4-(oxan-4-ylamino)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13554
TTKTTKOther7cilAA4-(cyclohexylamino)-2-[(1-methylpyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13549
TTKTTKOther7cilAB4-(cyclohexylamino)-2-[(1-methylpyrazol-4-yl)amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13555
TTKTTKOther7cjaA4-(cyclopentylmethylamino)-2-[[2-methoxy-4-(2-oxidanylidenepyrrolidin-1-yl)phenyl]amino]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13551
TTKTTKOther7clhA2-[[2-methoxy-4-(2-oxidanylidenepyrrolidin-1-yl)phenyl]amino]-4-(methylamino)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13553
TTKTTKOther7lqdA~{n}-(2,6-diethylphenyl)-2-[[4-(4-methylpiperazin-1-yl)-2-(propanoylamino)phenyl]amino]-5,6-dihydropyrimido[4,5-e]indolizine-7-carboxamideHuman14108
TTNMLCKCAMK1tkiA-Human130
TTNMLCKCAMK1tkiB-Human126
TTNMLCKCAMK4jnwAA-Human127
TTNMLCKCAMK4jnwAB-Human129
TTNMLCKCAMK4jnwBA-Human125
TTNMLCKCAMK4jnwBB-Human128
TTNMLCKCAMK6ygnA-Human13488
TTNMLCKCAMK6ygnB-Human13487
Tyk2 (TYK2)JakATK4e1zAn-[5-(4-{[(3-chlorophenyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]furan-2-carboxamideMouse5828
Tyk2 (TYK2)JakATK4e20An-[4-(3-amino-1h-indazol-5-yl)phenyl]-3-chlorobenzenesulfonamideMouse5827
TYK2JakATK3lxnA3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrileHuman3337
TYK2JakATK3lxpA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman3340
TYK2JakATK3nyxAAn-{5-[(7-chloroquinolin-4-yl)sulfanyl]-1,3,4-thiadiazol-2-yl}thiophene-2-carboxamideHuman3341
TYK2JakATK3nyxABn-{5-[(7-chloroquinolin-4-yl)sulfanyl]-1,3,4-thiadiazol-2-yl}thiophene-2-carboxamideHuman3343
TYK2JakATK3nz0AA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman3342
TYK2JakATK3nz0AB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman3335
TYK2JakATK4gfoAA2,6-dichloro-n-(2-oxo-2,5-dihydropyridin-4-yl)benzamideHuman3336
TYK2JakATK4gfoAB2,6-dichloro-n-(2-oxo-2,5-dihydropyridin-4-yl)benzamideHuman3338
TYK2JakATK4gihAA2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman3339
TYK2JakATK4gihAB2,6-dichloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman3332
TYK2JakATK4giiA2,6-dichloro-4-cyano-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman3331
TYK2JakATK4gj2A2,6-dichloro-n-[2-({[(1r,2r)-2-fluorocyclopropyl]carbonyl}amino)pyridin-4-yl]benzamideHuman3344
TYK2JakATK4gj3A2,6-dichloro-4-cyano-n-[2-({[(1r,2r)-2-fluorocyclopropyl]carbonyl}amino)pyridin-4-yl]benzamideHuman3345
TYK2JakATK4gvjAadenosine-5'-diphosphateHuman3334
TYK2JakATK4py1A6-[(2,5-dimethoxyphenyl)sulfanyl]-3-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazineHuman3333
TYK2JakATK5f1zAA3-azanyl-5-[(2~{s})-3-methylbutan-2-yl]-7-[1-methyl-5-(2-oxidanylpropan-2-yl)pyrazol-3-yl]-1~{h}-pyrazolo[4,3-c]pyridin-4-oneHuman6356
TYK2JakATK5f1zAB3-azanyl-5-[(2~{s})-3-methylbutan-2-yl]-7-[1-methyl-5-(2-oxidanylpropan-2-yl)pyrazol-3-yl]-1~{h}-pyrazolo[4,3-c]pyridin-4-oneHuman6357
TYK2JakATK5f20A3-azanyl-5-(2-methylphenyl)-7-(1-methylpyrazol-3-yl)-1~{h}-pyrazolo[4,3-c]pyridin-4-oneHuman6355
TYK2JakATK5walAAn-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamideHuman8375
TYK2JakATK5walABn-[2-(2,6-dichlorophenyl)-1h-imidazo[4,5-c]pyridin-4-yl]cyclopropanecarboxamideHuman8374
TYK2JakATK6aamA4-[[(1s,3r)-5-oxidanyl-2-adamantyl]amino]-1h-pyrrolo[2,3-b]pyridine-5-carboxamideHuman10489
TYK2JakATK6dbkA4-({4-[(1s,4s)-5-(cyanoacetyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]pyrimidin-2-yl}amino)-n-ethylbenzamideHuman10490
TYK2JakATK6dbmAA[(1s)-2,2-difluorocyclopropyl][(1r,5s)-3-{2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octan-8-yl]methanoneHuman10491
TYK2JakATK6dbmAB[(1s)-2,2-difluorocyclopropyl][(1r,5s)-3-{2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-3,8-diazabicyclo[3.2.1]octan-8-yl]methanoneHuman10488
TYK2JakATK6ovaAA6-({4-[(3s)-3-cyano-3-cyclopropyl-2-oxopyrrolidin-1-yl]pyridin-2-yl}amino)-n,n-dimethylpyridine-3-carboxamideHuman11980
TYK2JakATK6ovaAB6-({4-[(3s)-3-cyano-3-cyclopropyl-2-oxopyrrolidin-1-yl]pyridin-2-yl}amino)-n,n-dimethylpyridine-3-carboxamideHuman11981
TYK2JakATK6vnsAA(1r,2r)-2-cyano-n-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropane-1-carboxamideHuman12139
TYK2JakATK6vnsAB(1r,2r)-2-cyano-n-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropane-1-carboxamideHuman12137
TYK2JakATK6vnvA(1s,2s)-2-cyano-n-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropane-1-carboxamideHuman12138
TYK2JakATK6vnxA(1s)-2,2-difluoro-n-[(1s,5r,6r)-3-{5-fluoro-2-[(1-methyl-1h-pyrazol-4-yl)amino]pyrimidin-4-yl}-6-methyl-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropane-1-carboxamideHuman12136
TYK2JakATK6vnyAn-[(1s,5r)-3-(5-fluoro-2-{[1-(2-hydroxyethyl)-1h-pyrazol-4-yl]amino}pyrimidin-4-yl)-3-azabicyclo[3.1.0]hexan-1-yl]cyclopropanecarboxamideHuman12135
TYK2JakATK6x8fAA[3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrileHuman13157
TYK2JakATK6x8fAB[3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrileHuman13159
TYK2JakATK6x8fCA[3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrileHuman13156
TYK2JakATK6x8fCB[3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}-1-(2,2,2-trifluoroethyl)azetidin-3-yl]acetonitrileHuman13158
TYK2JakATK6x8gAAtrans-3-(cyanomethyl)-3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}cyclobutane-1-carbonitrileHuman12992
TYK2JakATK6x8gABtrans-3-(cyanomethyl)-3-{4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]-1h-pyrazol-1-yl}cyclobutane-1-carbonitrileHuman12993
TYK2JakATK7uyrAA2-(4-{[2-(2,6-difluorophenyl)-5-oxo-5h-pyrrolo[3,4-d]pyrimidin-4-yl]amino}phenyl)-n-ethylacetamideHuman14338
TYK2JakATK7uyrAB2-(4-{[2-(2,6-difluorophenyl)-5-oxo-5h-pyrrolo[3,4-d]pyrimidin-4-yl]amino}phenyl)-n-ethylacetamideHuman14335
TYK2JakATK7uysAA2-(2,6-difluorophenyl)-4-(4-methoxyanilino)-5h-pyrrolo[3,4-d]pyrimidin-5-oneHuman14339
TYK2JakATK7uysAB2-(2,6-difluorophenyl)-4-(4-methoxyanilino)-5h-pyrrolo[3,4-d]pyrimidin-5-oneHuman14336
TYK2JakATK7uytAA6-{[(2m)-2-(2-chloro-6-fluorophenyl)-5-oxo-5h-pyrrolo[3,4-b]pyridin-4-yl]amino}-n-ethylpyridine-3-carboxamideHuman14342
TYK2JakATK7uytAB6-{[(2m)-2-(2-chloro-6-fluorophenyl)-5-oxo-5h-pyrrolo[3,4-b]pyridin-4-yl]amino}-n-ethylpyridine-3-carboxamideHuman14340
TYK2JakATK7uyuAA2-(2,6-difluorophenyl)-4-[4-(pyrrolidine-1-carbonyl)anilino]-5h-pyrrolo[3,4-b]pyridin-5-oneHuman14337
TYK2JakATK7uyuAB2-(2,6-difluorophenyl)-4-[4-(pyrrolidine-1-carbonyl)anilino]-5h-pyrrolo[3,4-b]pyridin-5-oneHuman14341
TYK2-bJakBTK3zonA5-phenyl-2-ureidothiophene-3-carboxamideHuman2200
TYK2-bJakBTK4oliA2-chloro-n-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamideHuman2198
TYK2-bJakBTK4wovAA2-methoxy-n-({6-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]pyridin-2-yl}methyl)acetamideHuman2196
TYK2-bJakBTK4wovAB2-methoxy-n-({6-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]pyridin-2-yl}methyl)acetamideHuman2199
TYK2-bJakBTK4wovBA2-methoxy-n-({6-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]pyridin-2-yl}methyl)acetamideHuman2195
TYK2-bJakBTK4wovBB2-methoxy-n-({6-[1-methyl-4-(methylamino)-1,6-dihydroimidazo[4,5-d]pyrrolo[2,3-b]pyridin-7-yl]pyridin-2-yl}methyl)acetamideHuman2197
TYK2-bJakBTK5c01Aunknown ligandHuman7222
TYK2-bJakBTK5c01Bunknown ligandHuman7223
TYK2-bJakBTK5c03AAphosphothiophosphoric acid-adenylate esterHuman6043
TYK2-bJakBTK5c03ABphosphothiophosphoric acid-adenylate esterHuman6044
TYK2-bJakBTK5c03BAphosphothiophosphoric acid-adenylate esterHuman6042
TYK2-bJakBTK5c03BBphosphothiophosphoric acid-adenylate esterHuman6045
TYK2-bJakBTK5tkdAA6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamideHuman7323
TYK2-bJakBTK5tkdAB6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamideHuman7326
TYK2-bJakBTK5tkdBA6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamideHuman7325
TYK2-bJakBTK5tkdBB6-[(3,5-dimethylphenyl)amino]-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamideHuman7324
TYK2-bJakBTK6nslAA6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamideHuman11952
TYK2-bJakBTK6nslAB6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamideHuman11954
TYK2-bJakBTK6nslBA6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamideHuman11955
TYK2-bJakBTK6nslBB6-{[1-(4-cyanophenyl)-2-oxo-1,2-dihydropyridin-3-yl]amino}-n-cyclopropyl-8-(methylamino)imidazo[1,2-b]pyridazine-3-carboxamideHuman11953
TYK2-bJakBTK6nzeAA4-[(2-carbamoylphenyl)amino]-6-[(5-fluoropyridin-2-yl)amino]-n-methylpyridine-3-carboxamideHuman11453
TYK2-bJakBTK6nzeAB4-[(2-carbamoylphenyl)amino]-6-[(5-fluoropyridin-2-yl)amino]-n-methylpyridine-3-carboxamideHuman11444
TYK2-bJakBTK6nzeBA4-[(2-carbamoylphenyl)amino]-6-[(5-fluoropyridin-2-yl)amino]-n-methylpyridine-3-carboxamideHuman11448
TYK2-bJakBTK6nzeBB4-[(2-carbamoylphenyl)amino]-6-[(5-fluoropyridin-2-yl)amino]-n-methylpyridine-3-carboxamideHuman11443
TYK2-bJakBTK6nzfAA6-[(5-fluoropyridin-2-yl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamideHuman11446
TYK2-bJakBTK6nzfAB6-[(5-fluoropyridin-2-yl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamideHuman11449
TYK2-bJakBTK6nzfBA6-[(5-fluoropyridin-2-yl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamideHuman11451
TYK2-bJakBTK6nzfBB6-[(5-fluoropyridin-2-yl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamideHuman11445
TYK2-bJakBTK6nzhAA6-[(cyclopropanecarbonyl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamideHuman11450
TYK2-bJakBTK6nzhAB6-[(cyclopropanecarbonyl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamideHuman11442
TYK2-bJakBTK6nzhBA6-[(cyclopropanecarbonyl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamideHuman11447
TYK2-bJakBTK6nzhBB6-[(cyclopropanecarbonyl)amino]-n-methyl-4-{[2-(methylsulfonyl)phenyl]amino}pyridine-3-carboxamideHuman11452
TYK2-bJakBTK6nzpAA6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl]amino}-n-methylpyridazine-3-carboxamideHuman11504
TYK2-bJakBTK6nzpAB6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl]amino}-n-methylpyridazine-3-carboxamideHuman11501
TYK2-bJakBTK6nzpBA6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl]amino}-n-methylpyridazine-3-carboxamideHuman11496
TYK2-bJakBTK6nzpBB6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(1-methyl-1h-1,2,4-triazol-3-yl)phenyl]amino}-n-methylpyridazine-3-carboxamideHuman11497
TYK2-bJakBTK6nzqAA6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[(2-methoxy-3-{[(pyridin-2-yl)methyl]carbamoyl}phenyl)amino]-n-methylpyridine-3-carboxamideHuman11502
TYK2-bJakBTK6nzqAB6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[(2-methoxy-3-{[(pyridin-2-yl)methyl]carbamoyl}phenyl)amino]-n-methylpyridine-3-carboxamideHuman11499
TYK2-bJakBTK6nzqBA6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[(2-methoxy-3-{[(pyridin-2-yl)methyl]carbamoyl}phenyl)amino]-n-methylpyridine-3-carboxamideHuman11495
TYK2-bJakBTK6nzqBB6-[(5-fluoro-4-methylpyridin-2-yl)amino]-4-[(2-methoxy-3-{[(pyridin-2-yl)methyl]carbamoyl}phenyl)amino]-n-methylpyridine-3-carboxamideHuman11506
TYK2-bJakBTK6nzrAAn-methyl-4-{[2-(methylsulfonyl)phenyl]amino}-6-[(pyridin-2-yl)amino]pyridazine-3-carboxamideHuman11505
TYK2-bJakBTK6nzrABn-methyl-4-{[2-(methylsulfonyl)phenyl]amino}-6-[(pyridin-2-yl)amino]pyridazine-3-carboxamideHuman11503
TYK2-bJakBTK6nzrBAn-methyl-4-{[2-(methylsulfonyl)phenyl]amino}-6-[(pyridin-2-yl)amino]pyridazine-3-carboxamideHuman11498
TYK2-bJakBTK6nzrBBn-methyl-4-{[2-(methylsulfonyl)phenyl]amino}-6-[(pyridin-2-yl)amino]pyridazine-3-carboxamideHuman11500
TYK2-bJakBTK7ax4A2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamideHuman13499
TYK2-bJakBTK7ax4B2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamideHuman13498
TYK2-bJakBTK7k7oAA6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(pyrimidin-2-yl)phenyl]amino}-n-methylpyridazine-3-carboxamideHuman13835
TYK2-bJakBTK7k7oAB6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(pyrimidin-2-yl)phenyl]amino}-n-methylpyridazine-3-carboxamideHuman13837
TYK2-bJakBTK7k7qAA6-[(cyclopropanecarbonyl)amino]-4-({3-[6-(dimethylcarbamoyl)pyridazin-3-yl]-2-methoxyphenyl}amino)-n-methylpyridazine-3-carboxamideHuman13838
TYK2-bJakBTK7k7qAB6-[(cyclopropanecarbonyl)amino]-4-({3-[6-(dimethylcarbamoyl)pyridazin-3-yl]-2-methoxyphenyl}amino)-n-methylpyridazine-3-carboxamideHuman13836
TYK2-bJakBTK8s98AA(8s)-n-cyclopropyl-5-[(2-methoxypyridin-3-yl)amino]-7-(methylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman14849
TYK2-bJakBTK8s98AB(8s)-n-cyclopropyl-5-[(2-methoxypyridin-3-yl)amino]-7-(methylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman14846
TYK2-bJakBTK8s99AA(8s)-n-[(1r,2s)-2-fluorocyclopropyl]-5-{[(1m,2'm)-3'-fluoro-2-oxo-2h-[1,2'-bipyridin]-3-yl]amino}-7-(methylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman14847
TYK2-bJakBTK8s99AB(8s)-n-[(1r,2s)-2-fluorocyclopropyl]-5-{[(1m,2'm)-3'-fluoro-2-oxo-2h-[1,2'-bipyridin]-3-yl]amino}-7-(methylamino)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman14850
TYK2-bJakBTK8s9aAA(8s)-n-[(1r,2r)-2-methoxycyclobutyl]-7-(methylamino)-5-{[(1p,2'p)-2-oxo-2h-[1,2'-bipyridin]-3-yl]amino}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman14848
TYK2-bJakBTK8s9aAB(8s)-n-[(1r,2r)-2-methoxycyclobutyl]-7-(methylamino)-5-{[(1p,2'p)-2-oxo-2h-[1,2'-bipyridin]-3-yl]amino}pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman14851
TYK2-bJakBTK8tb5AAn-{(3p)-3-[3-(dimethylsulfamoyl)phenyl]-1h-pyrrolo[2,3-c]pyridin-5-yl}cyclopropanecarboxamideHuman14958
TYK2-bJakBTK8tb5ABn-{(3p)-3-[3-(dimethylsulfamoyl)phenyl]-1h-pyrrolo[2,3-c]pyridin-5-yl}cyclopropanecarboxamideHuman14955
TYK2-bJakBTK8tb6AAn-[(3m)-3-{6-[(3r)-3-methoxyoxolan-3-yl]pyridin-2-yl}-1-methyl-1h-pyrrolo[2,3-c]pyridin-5-yl]ureaHuman14956
TYK2-bJakBTK8tb6ABn-[(3m)-3-{6-[(3r)-3-methoxyoxolan-3-yl]pyridin-2-yl}-1-methyl-1h-pyrrolo[2,3-c]pyridin-5-yl]ureaHuman14957
Tyro3 (TYRO3)AxlTK3qupA(5-fluoro-1h-indol-2-yl)[(3r)-1'-[(3r)-piperidin-3-yl]spiro[indole-3,3'-pyrrolidin]-1(2h)-yl]methanoneMouse5799
Tyro3 (TYRO3)AxlTK4feqA4-(cyclopentylamino)-n-[3-(2-oxopyrrolidin-1-yl)propyl]-2-{[2-(pyridin-4-yl)ethyl]amino}pyrimidine-5-carboxamideMouse5801
Tyro3 (TYRO3)AxlTK4ff8A4-(cyclopentylamino)-2-[(2-methoxybenzyl)amino]-n-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamideMouse5800
ULK1ULKOther4wnoAAn~2~-(4-aminophenyl)-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1881
ULK1ULKOther4wnoABn~2~-(4-aminophenyl)-n~4~-(5-cyclopropyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1876
ULK1ULKOther4wnpAAn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1878
ULK1ULKOther4wnpABn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1874
ULK1ULKOther4wnpBAn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1872
ULK1ULKOther4wnpBBn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1879
ULK1ULKOther4wnpCAn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1877
ULK1ULKOther4wnpCBn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1873
ULK1ULKOther4wnpDAn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1875
ULK1ULKOther4wnpDBn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman1880
ULK1ULKOther5ci7AAn-[3-({4-[(3-aminopropyl)amino]-5-iodopyrimidin-2-yl}amino)phenyl]pyrrolidine-1-carboxamideHuman5974
ULK1ULKOther5ci7ABn-[3-({4-[(3-aminopropyl)amino]-5-iodopyrimidin-2-yl}amino)phenyl]pyrrolidine-1-carboxamideHuman5973
ULK1ULKOther6mnhAAn-[(2r)-3-methylbutan-2-yl]-1h-benzotriazole-6-carboxamideHuman10979
ULK1ULKOther6mnhABn-[(2r)-3-methylbutan-2-yl]-1h-benzotriazole-6-carboxamideHuman10980
ULK1ULKOther6qasAAn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman10930
ULK1ULKOther6qasABn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman10931
ULK1ULKOther6qasBAn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman10932
ULK1ULKOther6qasBBn-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman10933
ULK2ULKOther6qatAn-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamideHuman11227
ULK2ULKOther6qatBn-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamideHuman11226
ULK2ULKOther6qatCn-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamideHuman11232
ULK2ULKOther6qatDn-{(3z)-2-oxo-3-[phenyl({4-[(piperidin-1-yl)methyl]phenyl}amino)methylidene]-2,3-dihydro-1h-indol-5-yl}ethanesulfonamideHuman11230
ULK2ULKOther6qauAAn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman11235
ULK2ULKOther6qauABn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman11225
ULK2ULKOther6qauBAn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman11222
ULK2ULKOther6qauBBn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman11236
ULK2ULKOther6qauCAn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman11229
ULK2ULKOther6qauCBn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman11233
ULK2ULKOther6qavAA~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamideHuman11231
ULK2ULKOther6qavAB~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamideHuman11239
ULK2ULKOther6qavBA~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamideHuman11224
ULK2ULKOther6qavBB~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamideHuman11237
ULK2ULKOther6qavCA~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamideHuman11223
ULK2ULKOther6qavCB~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamideHuman11228
ULK2ULKOther6qavDA~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamideHuman11234
ULK2ULKOther6qavDB~{n}-[3-[[5-cyclopropyl-2-[(2-methyl-3,4-dihydro-1~{h}-isoquinolin-6-yl)amino]pyrimidin-4-yl]amino]propyl]cyclobutanecarboxamideHuman11238
ULK2ULKOther6yidAA2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman12385
ULK2ULKOther6yidAB2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman12382
ULK2ULKOther6yidBA2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman12381
ULK2ULKOther6yidBB2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman12387
ULK2ULKOther6yidCA2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman12384
ULK2ULKOther6yidCB2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman12386
ULK2ULKOther6yidDA2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman12388
ULK2ULKOther6yidDB2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman12383
ULK3ULKOther6fdyU4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman10389
ULK3ULKOther6fdzUmomelotinibHuman10390
ULK4ULKOther6tszUphosphothiophosphoric acid-adenylate esterHuman11904
ULK4ULKOther6u5lAAn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman11890
ULK4ULKOther6u5lABn~2~-(1h-benzimidazol-6-yl)-n~4~-(5-cyclobutyl-1h-pyrazol-3-yl)quinazoline-2,4-diamineHuman11889
VRK1VRKCK12ktyA1-Human4877
VRK1VRKCK12ktyA10-Human4932
VRK1VRKCK12ktyA11-Human4917
VRK1VRKCK12ktyA12-Human4897
VRK1VRKCK12ktyA13-Human4922
VRK1VRKCK12ktyA14-Human4926
VRK1VRKCK12ktyA15-Human4953
VRK1VRKCK12ktyA16-Human4937
VRK1VRKCK12ktyA17-Human4920
VRK1VRKCK12ktyA18-Human4904
VRK1VRKCK12ktyA19-Human4875
VRK1VRKCK12ktyA2-Human4947
VRK1VRKCK12ktyA20-Human4890
VRK1VRKCK12ktyA3-Human4874
VRK1VRKCK12ktyA4-Human4938
VRK1VRKCK12ktyA5-Human4900
VRK1VRKCK12ktyA6-Human4929
VRK1VRKCK12ktyA7-Human4880
VRK1VRKCK12ktyA8-Human4939
VRK1VRKCK12ktyA9-Human4885
VRK1VRKCK12kulA1-Human4919
VRK1VRKCK12kulA10-Human4901
VRK1VRKCK12kulA11-Human4923
VRK1VRKCK12kulA12-Human4883
VRK1VRKCK12kulA13-Human4941
VRK1VRKCK12kulA14-Human4909
VRK1VRKCK12kulA15-Human4876
VRK1VRKCK12kulA16-Human4924
VRK1VRKCK12kulA17-Human4893
VRK1VRKCK12kulA18-Human4896
VRK1VRKCK12kulA19-Human4906
VRK1VRKCK12kulA2-Human4921
VRK1VRKCK12kulA20-Human4915
VRK1VRKCK12kulA3-Human4895
VRK1VRKCK12kulA4-Human4948
VRK1VRKCK12kulA5-Human4954
VRK1VRKCK12kulA6-Human4949
VRK1VRKCK12kulA7-Human4908
VRK1VRKCK12kulA8-Human4887
VRK1VRKCK12kulA9-Human4869
VRK1VRKCK12lavA1-Human4930
VRK1VRKCK12lavA10-Human4882
VRK1VRKCK12lavA11-Human4916
VRK1VRKCK12lavA12-Human4946
VRK1VRKCK12lavA13-Human4872
VRK1VRKCK12lavA14-Human4898
VRK1VRKCK12lavA15-Human4931
VRK1VRKCK12lavA16-Human4888
VRK1VRKCK12lavA17-Human4950
VRK1VRKCK12lavA18-Human4927
VRK1VRKCK12lavA19-Human4940
VRK1VRKCK12lavA2-Human4903
VRK1VRKCK12lavA20-Human4933
VRK1VRKCK12lavA3-Human4912
VRK1VRKCK12lavA4-Human4884
VRK1VRKCK12lavA5-Human4891
VRK1VRKCK12lavA6-Human4871
VRK1VRKCK12lavA7-Human4936
VRK1VRKCK12lavA8-Human4881
VRK1VRKCK12lavA9-Human4945
VRK1VRKCK12rsvA1-Human4910
VRK1VRKCK12rsvA10-Human4873
VRK1VRKCK12rsvA11-Human4902
VRK1VRKCK12rsvA12-Human4952
VRK1VRKCK12rsvA13-Human4935
VRK1VRKCK12rsvA14-Human4925
VRK1VRKCK12rsvA15-Human4911
VRK1VRKCK12rsvA16-Human4905
VRK1VRKCK12rsvA17-Human4951
VRK1VRKCK12rsvA18-Human4934
VRK1VRKCK12rsvA2-Human4914
VRK1VRKCK12rsvA3-Human4913
VRK1VRKCK12rsvA4-Human4907
VRK1VRKCK12rsvA5-Human4899
VRK1VRKCK12rsvA6-Human4943
VRK1VRKCK12rsvA7-Human4889
VRK1VRKCK12rsvA8-Human4918
VRK1VRKCK12rsvA9-Human4928
VRK1VRKCK13op5AA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4870
VRK1VRKCK13op5AB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4942
VRK1VRKCK13op5BA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4894
VRK1VRKCK13op5BB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4944
VRK1VRKCK13op5CA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4886
VRK1VRKCK13op5CB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4879
VRK1VRKCK13op5DA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4878
VRK1VRKCK13op5DB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4892
VRK1VRKCK15ukfA4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamideHuman8030
VRK1VRKCK15ukfB4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamideHuman8029
VRK1VRKCK15ukfC4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamideHuman8027
VRK1VRKCK15ukfD4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamideHuman8028
VRK1VRKCK15uvfA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman7521
VRK1VRKCK15uvfB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman7523
VRK1VRKCK15uvfC(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman7520
VRK1VRKCK15uvfD(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman7522
VRK1VRKCK16ac9AAphosphoaminophosphonic acid-adenylate esterHuman10816
VRK1VRKCK16ac9ABphosphoaminophosphonic acid-adenylate esterHuman10817
VRK1VRKCK16ac9BAphosphoaminophosphonic acid-adenylate esterHuman10818
VRK1VRKCK16ac9BBphosphoaminophosphonic acid-adenylate esterHuman10823
VRK1VRKCK16ac9CAphosphoaminophosphonic acid-adenylate esterHuman10822
VRK1VRKCK16ac9CBphosphoaminophosphonic acid-adenylate esterHuman10819
VRK1VRKCK16ac9DAphosphoaminophosphonic acid-adenylate esterHuman10821
VRK1VRKCK16ac9DBphosphoaminophosphonic acid-adenylate esterHuman10820
VRK1VRKCK16bp0AA-Human8744
VRK1VRKCK16bp0AB-Human8738
VRK1VRKCK16bp0BA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman8740
VRK1VRKCK16bp0BB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman8741
VRK1VRKCK16bp0CA-Human8743
VRK1VRKCK16bp0CB-Human8742
VRK1VRKCK16bp0DA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman8745
VRK1VRKCK16bp0DB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman8739
VRK1VRKCK16bruAA-Human9085
VRK1VRKCK16bruAB-Human9082
VRK1VRKCK16bruBA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman9088
VRK1VRKCK16bruBB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman9087
VRK1VRKCK16bruCA-Human9089
VRK1VRKCK16bruCB-Human9086
VRK1VRKCK16bruDA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman9084
VRK1VRKCK16bruDB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-oneHuman9083
VRK1VRKCK16btwAA2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9418
VRK1VRKCK16btwAB2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9425
VRK1VRKCK16btwBA2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9424
VRK1VRKCK16btwBB2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9411
VRK1VRKCK16btwCA-Human9419
VRK1VRKCK16btwCB-Human9416
VRK1VRKCK16btwDA2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9415
VRK1VRKCK16btwDB2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-oneHuman9420
VRK1VRKCK16bu6AA4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9423
VRK1VRKCK16bu6AB4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9417
VRK1VRKCK16bu6BA4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9421
VRK1VRKCK16bu6BB4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9422
VRK1VRKCK16bu6CA-Human9412
VRK1VRKCK16bu6CB-Human9414
VRK1VRKCK16bu6DA4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9413
VRK1VRKCK16bu6DB4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol)Human9410
VRK1VRKCK16cfmAA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9723
VRK1VRKCK16cfmAB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9718
VRK1VRKCK16cfmBA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9724
VRK1VRKCK16cfmBB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9725
VRK1VRKCK16cfmCA-Human9719
VRK1VRKCK16cfmCB-Human9720
VRK1VRKCK16cfmDA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9721
VRK1VRKCK16cfmDB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9722
VRK1VRKCK16cmmAA-Human9763
VRK1VRKCK16cmmAB-Human9760
VRK1VRKCK16cmmBA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9766
VRK1VRKCK16cmmBB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9761
VRK1VRKCK16cmmCA-Human9765
VRK1VRKCK16cmmCB-Human9762
VRK1VRKCK16cmmDA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9764
VRK1VRKCK16cmmDB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9759
VRK1VRKCK16cnxAA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9815
VRK1VRKCK16cnxAB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9810
VRK1VRKCK16cnxBA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9803
VRK1VRKCK16cnxBB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9806
VRK1VRKCK16cnxCA(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9805
VRK1VRKCK16cnxCB(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9804
VRK1VRKCK16cnxDA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9814
VRK1VRKCK16cnxDB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9807
VRK1VRKCK16cqhAA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9774
VRK1VRKCK16cqhAB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9768
VRK1VRKCK16cqhBA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9769
VRK1VRKCK16cqhBB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9770
VRK1VRKCK16cqhCA-Human9772
VRK1VRKCK16cqhCB-Human9773
VRK1VRKCK16cqhDA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9771
VRK1VRKCK16cqhDB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman9767
VRK1VRKCK16cswAA-Human9818
VRK1VRKCK16cswAB-Human9813
VRK1VRKCK16cswBA(7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-oneHuman9812
VRK1VRKCK16cswBB(7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-oneHuman9808
VRK1VRKCK16cswCA-Human9816
VRK1VRKCK16cswCB-Human9811
VRK1VRKCK16cswDA(7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-oneHuman9817
VRK1VRKCK16cswDB(7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-oneHuman9809
VRK1VRKCK16dd4AA-Human9935
VRK1VRKCK16dd4AB-Human9939
VRK1VRKCK16dd4BA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-oneHuman9937
VRK1VRKCK16dd4BB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-oneHuman9933
VRK1VRKCK16dd4CA-Human9940
VRK1VRKCK16dd4CB-Human9936
VRK1VRKCK16dd4DA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-oneHuman9938
VRK1VRKCK16dd4DB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-oneHuman9934
VRK1VRKCK16npnA(7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman11243
VRK1VRKCK16npnB(7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman11244
VRK1VRKCK16npnC(7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman11241
VRK1VRKCK16npnD(7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman11242
VRK1VRKCK16vxuB(7r)-8-(cyclopropylmethyl)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman13362
VRK1VRKCK16vzhA-Human12057
VRK1VRKCK16vzhB(7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-oneHuman12056
VRK1VRKCK16vzhC-Human12058
VRK1VRKCK16vzhD(7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-oneHuman12055
VRK2VRKCK12v62AA-Human2628
VRK2VRKCK12v62AB-Human2629
VRK2VRKCK12v62BA-Human2630
VRK2VRKCK12v62BB-Human2631
VRK2VRKCK15uu1A(7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-oneHuman7499
VRK2VRKCK16ncgA4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamideHuman10852
VRK2VRKCK16ncgB4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamideHuman10851
VRK2VRKCK18q1zAA2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrileHuman14899
VRK2VRKCK18q1zAB2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrileHuman14898
VRK3VRKCK12jiiAA-Human2939
VRK3VRKCK12jiiAB-Human2938
VRK3VRKCK12jiiBA-Human2936
VRK3VRKCK12jiiBB-Human2937
WEE1 (Wee1)WEEOther1x8bA9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman209
WEE1 (Wee1)WEEOther2in6A3-(9-hydroxy-1,3-dioxo-4-phenyl-2,3-dihydropyrrolo[3,4-c]carbazol-6(1h)-yl)propanoic acidHuman207
WEE1 (Wee1)WEEOther2io6A9-hydroxy-6-(3-hydroxypropyl)-4-(2-methoxyphenyl)pyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman214
WEE1 (Wee1)WEEOther2z2wAn-[4-(2-chlorophenyl)-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-c]carbazol-9-yl]formamideHuman203
WEE1 (Wee1)WEEOther3bi6AA4-(2-chlorophenyl)-9-hydroxy-6-methyl-1,3-dioxo-n-(2-pyrrolidin-1-ylethyl)pyrrolo[3,4-g]carbazole-8-carboxamideHuman213
WEE1 (Wee1)WEEOther3bi6AB4-(2-chlorophenyl)-9-hydroxy-6-methyl-1,3-dioxo-n-(2-pyrrolidin-1-ylethyl)pyrrolo[3,4-g]carbazole-8-carboxamideHuman205
WEE1 (Wee1)WEEOther3bizAA4-(2-chlorophenyl)-8-[3-(dimethylamino)propoxy]-9-hydroxy-6-methylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman210
WEE1 (Wee1)WEEOther3bizAB4-(2-chlorophenyl)-8-[3-(dimethylamino)propoxy]-9-hydroxy-6-methylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman204
WEE1 (Wee1)WEEOther3cqeAA8-bromo-4-(2-chlorophenyl)-n-(2-hydroxyethyl)-6-methyl-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-e]indole-7-carboxamideHuman206
WEE1 (Wee1)WEEOther3cqeAB8-bromo-4-(2-chlorophenyl)-n-(2-hydroxyethyl)-6-methyl-1,3-dioxo-1,2,3,6-tetrahydropyrrolo[3,4-e]indole-7-carboxamideHuman211
WEE1 (Wee1)WEEOther3cr0AA4-(2-chlorophenyl)-8-(2-hydroxyethyl)-6-methylpyrrolo[3,4-e]indole-1,3(2h,6h)-dioneHuman208
WEE1 (Wee1)WEEOther3cr0AB4-(2-chlorophenyl)-8-(2-hydroxyethyl)-6-methylpyrrolo[3,4-e]indole-1,3(2h,6h)-dioneHuman212
WEE1 (Wee1)WEEOther5v5yA1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman8328
WEE1 (Wee1)WEEOther5vc3A4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8329
WEE1 (Wee1)WEEOther5vc4A4-[(3,5-dichloro-4-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman8334
WEE1 (Wee1)WEEOther5vc5AA6-(2,6-dichlorophenyl)-2-({4-[2-(diethylamino)ethoxy]phenyl}amino)-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman8332
WEE1 (Wee1)WEEOther5vc5AB6-(2,6-dichlorophenyl)-2-({4-[2-(diethylamino)ethoxy]phenyl}amino)-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman8333
WEE1 (Wee1)WEEOther5vc6An,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman8331
WEE1 (Wee1)WEEOther5vd2An-{2-[(1s,4r)-6-{[4-(cyclobutylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1,2,3,4-tetrahydro-1,4-epiminonaphthalen-9-yl]-2-oxoethyl}acetamideHuman8330
WEE1 (Wee1)WEEOther5vd4A6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1-{6-[(1s)-2,2,2-trifluoro-1-hydroxyethyl]pyridin-2-yl}-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman9780
WEE1 (Wee1)WEEOther5vd5A1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(morpholin-4-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman9778
WEE1 (Wee1)WEEOther5vd7A6-{[3-fluoro-4-(4-methylpiperazin-1-yl)phenyl]amino}-1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman9782
WEE1 (Wee1)WEEOther5vd8A6-{[3-chloro-4-(4-methylpiperazin-1-yl)phenyl]amino}-1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman9777
WEE1 (Wee1)WEEOther5vd9A1-{6-[(1r)-1-hydroxyethyl]pyridin-2-yl}-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman9781
WEE1 (Wee1)WEEOther5vdaA1-{6-[(1s)-1-hydroxyethyl]pyridin-2-yl}-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman9779
WEE1 (Wee1)WEEOther7n3uA1-[(7r)-7-ethyl-7-hydroxy-7h-cyclopenta[b]pyridin-2-yl]-6-[4-(4-methylpiperazin-1-yl)anilino]-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman13857
WEE1 (Wee1)WEEOther8bjuAA2-(2-methoxyphenyl)-6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1-[6-(2-oxidanylpropan-2-yl)pyridin-2-yl]pyrazolo[3,4-d]pyrimidin-3-oneHuman14755
WEE1 (Wee1)WEEOther8bjuAB2-(2-methoxyphenyl)-6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1-[6-(2-oxidanylpropan-2-yl)pyridin-2-yl]pyrazolo[3,4-d]pyrimidin-3-oneHuman14754
WEE2 (Wee1B)WEEOther5vdkA1-[6-(2-hydroxypropan-2-yl)pyridin-2-yl]-6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-(prop-2-en-1-yl)-1,2-dihydro-3h-pyrazolo[3,4-d]pyrimidin-3-oneHuman8349
WNK1 (Wnk1)WNKOther4pwnA-Human1831
WNK1 (Wnk1)WNKOther5tf9A{2-[(4-chlorophenyl)methoxy]phenyl}{5-[2-(methylamino)-1,3-thiazol-4-yl]-2,3-dihydro-1h-indol-1-yl}methanoneHuman7099
WNK1 (Wnk1)WNKOther5tf9B{2-[(4-chlorophenyl)methoxy]phenyl}{5-[2-(methylamino)-1,3-thiazol-4-yl]-2,3-dihydro-1h-indol-1-yl}methanoneHuman7098
WNK1 (Wnk1)WNKOther5wdyAAphosphoaminophosphonic acid-adenylate esterHuman8326
WNK1 (Wnk1)WNKOther5wdyABphosphoaminophosphonic acid-adenylate esterHuman8321
WNK1 (Wnk1)WNKOther5wdyBAphosphoaminophosphonic acid-adenylate esterHuman8323
WNK1 (Wnk1)WNKOther5wdyBBphosphoaminophosphonic acid-adenylate esterHuman8322
WNK1 (Wnk1)WNKOther5we8AAphosphoaminophosphonic acid-adenylate esterHuman8324
WNK1 (Wnk1)WNKOther5we8ABphosphoaminophosphonic acid-adenylate esterHuman8325
WNK1 (Wnk1)WNKOther5we8BAphosphoaminophosphonic acid-adenylate esterHuman8327
WNK1 (Wnk1)WNKOther5we8BBphosphoaminophosphonic acid-adenylate esterHuman8320
WNK3 (Wnk3)WNKOther5o1vAA-Human8157
WNK3 (Wnk3)WNKOther5o1vAB-Human8165
WNK3 (Wnk3)WNKOther5o1vBA-Human8152
WNK3 (Wnk3)WNKOther5o1vBB-Human8150
WNK3 (Wnk3)WNKOther5o21A-Human8160
WNK3 (Wnk3)WNKOther5o21B-Human8158
WNK3 (Wnk3)WNKOther5o23AA-Human8151
WNK3 (Wnk3)WNKOther5o23AB-Human8155
WNK3 (Wnk3)WNKOther5o23BA-Human8159
WNK3 (Wnk3)WNKOther5o23BB-Human8166
WNK3 (Wnk3)WNKOther5o26AAphosphoaminophosphonic acid-adenylate esterHuman8164
WNK3 (Wnk3)WNKOther5o26ABphosphoaminophosphonic acid-adenylate esterHuman8149
WNK3 (Wnk3)WNKOther5o26BAphosphoaminophosphonic acid-adenylate esterHuman8162
WNK3 (Wnk3)WNKOther5o26BBphosphoaminophosphonic acid-adenylate esterHuman8156
WNK3 (Wnk3)WNKOther5o2bAA1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman8163
WNK3 (Wnk3)WNKOther5o2bAB1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman8153
WNK3 (Wnk3)WNKOther5o2bBA1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman8154
WNK3 (Wnk3)WNKOther5o2bBB1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman8161
WNK3 (Wnk3)WNKOther5o2cA-Human8148
WNK3 (Wnk3)WNKOther8edhAethyl 1-(5,7-dimethoxy-4-methylquinolin-2-yl)piperidine-4-carboxylateHuman14631
ZAP70SykTK1u59AAstaurosporineHuman2734
ZAP70SykTK1u59ABstaurosporineHuman2733
ZAP70SykTK2ozoAphosphoaminophosphonic acid-adenylate esterHuman2735
ZAP70SykTK4k2rAphosphoaminophosphonic acid-adenylate esterHuman2732