| - | | Palomid
529 | | 1 |
|
|
| - | | AMG-337 | | 2 |
|
|
| - | | PIM447
LGH447 | | 1 |
|
|
| - | | BAY1082439 | | 1 |
|
|
| - | | ARRY-382 | | 2 |
|
|
| - | | CC-115 | | 1 |
|
|
| - | | ASP3026 | | 1 |
|
|
| - | | XL019 | | 1 |
|
|
| - | | JI-101 | | 2 |
|
|
| - | | XL228 | | 1 |
|
|
| - | | RGB-286638 | | 1 |
|
|
| - | | GSK1059615 | | 1 |
|
|
| - | | TAK-901 | | 1 |
|
|
| - | | VS-5584
SB2343 | | 1 |
|
|
| - | | MRX-2843
UNC2371 | | 1 |
|
|
| - | | BGT226
NVP-BGT226 | | 2 |
|
|
| - | | AZD8330
ARRY-424704
ARRY-704 | | 1 |
|
|
| - | | ON123300
ON 123300 | | 2 |
|
|
| - | | SAR-260301 | | 1 |
|
|
| - | | PND-1186
VS-4718
SR-2516 | | 1 |
|
|
| - | | CP-547632 | | 2 |
|
|
| - | | TAK-960 | | 1 |
|
|
| - | | GDC-0349 | | 1 |
|
|
| - | | MK-8033 | | 1 |
|
|
| - | | TAK-593 | | 1 |
|
|
| - | | KB-0742 | | 1 |
|
|
| - | | JNJ-38877605 | | 1 |
|
|
| - | | AZD1208 | | 1 |
|
|
| - | | AZD-7762 | | 1 |
|
|
| - | | PF-04217903 | | 1 |
|
|
| - | | MK-2461
MK2461 | | 2 |
|
|
| - | | AZD-8055 | | 1 |
|
|
| - | | CH5132799 | | 1 |
|
|
| - | | BMS-599626
AC480 | | 1 |
|
|
| - | | RO4987655
CH4987655 | | 1 |
|
|
| - | | TAK-285 | | 1 |
|
|
| - | | CC-401 | | 1 |
|
|
| - | | OSI-930 | | 1 |
|
|
| - | | SGX-523 | | 1 |
|
|
| - | | PHA-793887 | | 1 |
|
|
| - | | TPX-0022
TPX0022 | | 1 |
|
|
| - | | VS-6766
RG 7304
CKI27
CH5126766
RO5126766 | | 1 |
|
|
| - | | XL092 | | 1 |
|
|
| - | | PF-06873600 | | 2 |
|
|
| - | | AZD-8154
AZD8154
AZD 8154 | | 2 |
|
|
| - | | PF-06952229 | | 1 |
|
|
| - | | LY-3200882 | | 2 |
|
|
| - | | AR-13503
Metabolite netarsudil | | 1 |
|
|
| - | | TT 00420
TT-00420 | | 1 |
|
|
| - | | DZD4205
AZD-4205
DZD 4205
AZD4205 | | 1/2 |
|
|
| - | | CLN-081
TAS6417 | | 1/2 |
|
|
| - | | BDTX-189 | | 1 |
|
|
| - | | BTX-A51 | | 1 |
|
|
| - | | IPN60130
BLU-782 | | 1 |
|
|
| - | | DAY101
MLN-2480
MLN2480
TAK580
TAK-580 | | 1 |
|
|
| - | | AZD4547
AZD-4547
KB-74810 | | 2 |
|
|
| - | | CA-4948 | | 2 |
|
|
| - | | GDC-0134 | | 1 |
|
|
| - | | JNJ-67856633
JNJ67856633
JNJ 67856633 | | 2 |
|
|
| - | | SHR0302
SHR 0302 | | 3 |
|
|
| - | | CFI-400945
CFI400945
CFI 400945 | | 1 |
|
|
| - | | LY3295668
AK-01 | | 1 |
|
|
| - | | PF-07104091 | | 2 |
|
|
| - | | M4205 | | 1 |
|
|
| - | | LY3405105 | | 1 |
|
|
| - | | HM43239
HM-43239 | | 1.5 |
|
|
| - | | VIP152
BAY-1251152 | | 1 |
|
|
| - | | ESK981
CEP 11981
CEP11981 | | 1 |
|
|
| - | | BIIB091 | | 1 |
|
|
| - | | GSK3145095 | | 2 |
|
|
| - | | GSK2983559 | | 1 |
|
|
| - | | GSK2982772 | | 2 |
|
|
| - | | GLPG0259
GLPG-0259
GTPL9848 | | 2 |
|
|
| - | | FF10101
FF-10101-01 | | 1 |
|
|
| - | | IM156
HL156A
HL271 | | 1 |
|
|
| - | | T-1101
TAI-95 | | 1 |
|
|
| - | | ONO-7475 | | 2 |
|
|
| - | | CG-806 | | 2 |
|
|
| - | | CC-90003 | | 1 |
|
|
| - | | KO-947 | | 1 |
|
|
| - | | GDC-0575
ARRY-575
RG7741 | | 1 |
|
|
| - | | TAS0728 | | 2 |
|
|
| - | | JNJ-38877618 | | 1 |
|
|
| - | | AV-412
MP412 | | 1 |
|
|
| - | | INCB053914 | | 2 |
|
|
| - | | CEP-40783
RXDX-106 | | 1 |
|
|
| - | | M2698
MSC2363318A | | 1 |
|
|
| - | | BAY1125976
BAY-1125976 | | 1 |
|
|
| - | | LY3214996 | | 2 |
|
|
| - | | AEE788
AEE 788
NVP-AEE788 | | 2 |
|
|
| - | | BI 2536 | | 2 |
|
|
| - | | AMG-208 | | 2 |
|
|
| - | | GSK-690693
GSK690693 | | 1 |
|
|
| - | | 9-ING-41 | | 2 |
|
|
| - | | ENMD-2076 | | 2 |
|
|
| - | | ASP5878 | | 1 |
|
|
| - | | AZD4573 | | 2 |
|
|
| - | | SAR125844 | | 2 |
|
|
| - | | AT7519
AT7519M | | 1 |
|
|
| - | | AMG319 | | 2 |
|
|
| - | | SCR-1481B1
BMS-817378 | | 1 |
|
|
| - | | TAS-117 | | 2 |
|
|
| - | | MK-8353
SCH900353 | | 1 |
|
|
| - | | BFH772 | | 2 |
|
|
| - | | FN-1501 | | 1 |
|
|
| - | | PRN1371 | | 1 |
|
|
| - | | BLZ945 | | 2 |
|
|
| - | | TG 100801
TG100801 | | 2 |
|
|
| - | | EOC317
ACTB-1003 | | 1 |
|
|
| - | | TP-3654 | | 1 |
|
|
| - | | CEP-37440 | | 1 |
|
|
| - | | ASP4132 | | 1 |
|
|
| - | | ODM-203 | | 1 |
|
|
| - | | AZD-8835 | | 1 |
|
|
| - | | PF-06459988 | | 2 |
|
|
| Abemaciclib | Verzenio
Verzenios | LY-2835219
LY2835219 | 2017 | 4 |
|
|
| Abivertinib | | A610
AC-0010
AC0010
ACEA100610
Avitinib
EX-ACEA0010 | | 3 |
|
|
| Abrocitinib | | PF-04965842 | | 3 |
|
|
| Acalabrutinib | Calquence | ACP-196 | 2017 | 4 |
|
|
| Acalisib | | CAL-120
CAL120
GS-9820
GS9820 | | 2 |
|
|
| Acumapimod | | | | 2 |
|
|
| Adavosertib | | AZD 1775
AZD-1775
AZD1775
MK-1775
MK1775 | | 2 |
|
|
| Afatinib | Gilotrif
Giotrif | BIBW-2992
BIBW2992 | 2013 | 4 |
|
|
| Afuresertib | | ASB-183
ASB183
GSK-2110183
GSK-2110183C
GSK2110183
GSK2110183C
LAE002 | | 2 |
|
|
| Agerafenib | | AB-024
AC-013773
CEP-32496
RXDX 105
RXDX-105 | | 1 |
|
|
| Alectinib | Alecensa | AF-802
AF802
CH-5424802
CH5424802
RO-5424802
RO5424802 | 2015 | 4 |
|
|
| Alisertib | | MLN 8237
MLN-8237
MLN8237 | | 3 |
|
|
| Allitinib | | ALL-3
AST-1306 | | 2 |
|
|
| Alofanib | | | | 1 |
|
|
| Alpelisib | Piqray | BYL-719
NVP-BYL719 | 2019 | 4 |
|
|
| Altiratinib | | DCC-2701
DP-5164 | | 1 |
|
|
| Alvocidib | | Flavopiridol
HL 275
HL-275
HMR 1275
HMR-1275
L 86 8275
L-868275
L86-8275
MDL 107,826A
MDL-107826A
NSC-649890 | | 3 |
|
|
| Amcasertib | | BBI-503
BBI503 | | 2 |
|
|
| Amuvatinib | | HPK 56
HPK-56
HPK56
MP 470
MP-470
MP470 | | 2 |
|
|
| Apatinib | Aitan | Rivoceranib
Albumin paclitaxel
Capecitabine
Carboplatin
Cryoablation
Docetaxel
Egafur
Emozolomide
H20140103
NAVELBINE+AITAN
NO.
Oxaliplatin
Paclitaxol
Pemetrexed
SHR-1210
VP-16
Xelox
YN968D1 | 2014 | 4 |
|
|
| Apilimod | | LAM-002A
LAM002A
STA 5326
STA-5326
STA5326 | | 2 |
|
|
| Apitolisib | | G-038390
G-038390.1
GDC-0980
GDC-0980.1
RG-7422
RG7422 | | 2 |
|
|
| Asciminib | Scemblix | ABL-001
ABL001
ABL001-NX
NVP-ABL001 | 2021 | 4 |
|
|
| Atuveciclib | | BAY 1143572
BAY-1143572
BAY1143572 | | 1 |
|
|
| Aumolertinib | Ameile | HS-10296
Almonertinib | | 4 (NMPA) |
|
|
| Avapritinib | Ayvakit | 70C366
BLU-285
C-366
X-720776
X720776 | 2020 | 4 |
|
|
| Axitinib | Inlyta | AG-013736
AG-13736 | 2012 | 4 |
|
|
| Bafetinib | | CNS-9
INNO-406
NS-187 | | 2 |
|
|
| Balamapimod | | MKI-833 | | 1 |
|
|
| Barasertib | | AZD 1152
AZD-1152
AZD1152 | | 3 |
|
|
| Baricitinib | Olumiant | INCB-028050
INCB-28050
INCB028050
LY-3009104
LY3009104 | 2017 | 4 |
|
|
| Belizatinib | | TSR-011
TSR011 | | 2 |
|
|
| Belumosudil | Rezurock | KD025
SLx2119 | 2021 | 4 |
|
|
| Belvarafenib | | HM95573
GDC-5573 | | 2 |
|
|
| Bemcentinib | | BGB 324
BGB-324
BGB324
CS-1046
HY-15150
KB-80319
QC-11751
R 428
R-428
R428
SYN-1131
SYN1131
W-5845 | | 2 |
|
|
| Bentamapimod | | AS-602801
PGL-5001 | | 2 |
|
|
| Berzosertib | | M-6620
M6620
VE-822
VX-970
VX970 | | 2 |
|
|
| Bezuclastinib | | PLX9486
CGT 9486 | | 2 |
|
|
| Bimiralisib | | NC-B5
NCB5
PI3K-IN-2
PQR-309
PQR309 | | 2 |
|
|
| Binimetinib | Mektovi | ARRY 438162
ARRY-162
ARRY-438162
MEK-162
MEK162
NVP-MEK162 | 2018 | 4 |
|
|
| Bosutinib | Bosulif | Bosutinib monohydrate
SK-606
SKI-606 | 2012 | 4 |
|
|
| Branebrutinib | | BMS-986195 | | 2 |
|
|
| Brepocitinib | | PF-06700841 | | 2 |
|
|
| Briciclib | | ON 014185 | | 1 |
|
|
| Brigatinib | Alunbrig | AP-26113
AP26113 | 2017 | 4 |
|
|
| Brivanib | | BMS-540215 | | 3 |
|
|
| Brivanib alaninate | | BMS-582664
BMS-582664-02
Brivanib l-alanine ester | | 3 |
|
|
| Buparlisib | | BKM-120
BKM-120NX
BKM120-NX
NVP-BKM-120
NVP-BKM120 | | 3 |
|
|
| Cabozantinib | Cabometyx
Cometriq | BMS-907351
XL-184
XL184 | 2012 | 4 |
|
|
| Canertinib | | CI-1033 | | 3 |
|
|
| Capivasertib | | AZC5363
AZD 5363
AZD-5363
AZD5363 | | 3 |
|
|
| Capmatinib | Tabrecta | INC-280
INC280
INCB-28060
NVP-INC280
NVP-INC280-NX
NYP-INC280-NX | 2020 | 4 |
|
|
| Catequentinib | FOCUS V | AL3818
Anlotinib
Altn | | 4 |
|
|
| Cediranib | Recentin | AZD-2171
AZD2171
ZD-2171 | | 3 |
|
|
| Cenisertib | | AS-703569
R-763 | | 1 |
|
|
| Ceralasertib | | AZD6738 | | 2 |
|
|
| Cerdulatinib | | | | 2.5 |
|
|
| Ceritinib | Zykadia | LDK-378
LDK378
NVP-LDK-378-NX
NVP-LDK378-NX | 2014 | 4 |
|
|
| Chiauranib | | CS-2164
CS2164 | | 3 |
|
|
| Cobimetinib | Cotellic | GDC-0623
GDC-0973
RG 7420
RG-7420
RG-7421
RG7420
XL-518 | 2015 | 4 |
|
|
| Conteltinib | | CT-707
CT707 | | 1 |
|
|
| Copanlisib | Aliqopa | BAY 80-6946
BAY-80-6946
BAY80-6946 | 2017 | 4 |
|
|
| Crenolanib | | ARO 002
ARO-002
CP 868596
CP-868,596
CP-868596 | | 3 |
|
|
| Crizotinib | Xalkori | PF-02341066
PF-2341066 | 2011 | 4 |
|
|
| Dabrafenib | Tafinlar | GSK-2118436
GSK-2118436A
GSK2118436
GSK2118436A | 2013 | 4 |
|
|
| Dacomitinib | Vizimpro | Dacomitinib hydrate
PF-00299804 | 2018 | 4 |
|
|
| Dactolisib | | BEZ-235
BEZ235
NVP-BEZ235
NVP-BEZ235-NX | | 3 |
|
|
| Danusertib | | PHA-739358 | | 2 |
|
|
| Darovasertib | | IDE-196
IDE196
LXS-196
LXS196 | | 1 |
|
|
| Dasatinib | Dasatinib
Sprycel | BMS-354825
BMS-354825 HYDRATE
BMS-354825-03
Dasatinib hydrate
Dasatinib monohydrate | 2006 | 4 |
|
|
| Decernotinib | | Adelatinib
VRT-831509
VX-509 | | 2 |
|
|
| Defactinib | | PF-04554878
VS-6063 | | 2 |
|
|
| Delgocitinib | | | | 2 |
|
|
| Derazantinib | | ARQ 087
ARQ-087
ARQ087 | | 2 |
|
|
| Deucravacitinib | | BMS-986165
BMS986165 | | 3 |
|
|
| Dezapelisib | | INCB040093 | | 0 |
|
|
| Dilmapimod | | GW-681323
SB-681323
SB681323 | | 2 |
|
|
| Dinaciclib | | MK-7965
SCH 727965
SCH-727965 | | 3 |
|
|
| Donafenib | Zepsun | Sorafenib (D3)
CM-4307 | 2021 (NMPA) | 4 |
|
|
| Doramapimod | | BIRB 796 BS
BIRB-796
BIRB-796 BS | | 2 |
|
|
| Dovitinib | | CHIR-258
GFKI-258
NVP-TKI258
TKI-258 | | 3 |
|
|
| Dubermatinib | | HCL-2084
TP 0903
TP-0903
TP0903 | | 1.5 |
|
|
| Duvelisib | Copiktra | INK-1147
INK-1197
IPI-145 | 2018 | 4 |
|
|
| Ebvaciclib | | PF-06873600 | | 2 |
|
|
| Edicotinib | | JNJ-40346527 | | 2 |
|
|
| Edralbrutinib | | SHR-1459
SHR1459
TG-1701
TG1701 | | 1 |
|
|
| Eganelisib | | IPI-549
IPI549 | | 2 |
|
|
| Elimusertib | | BAY 1895344
BAY-1895344
BAY1895344 | | 1.5 |
|
|
| Elsubrutinib | | ABBV 105 | | 2 |
|
|
| Empesertib | | (-)-BAY-1161909
BAY 1161909
MPS1-IN-5 | | 1 |
|
|
| Encorafenib | Braftovi | LGX-818
NVP-LGX-818-NXA
NVP-LGX818
NVP-LGX818-NXA | 2018 | 4 |
|
|
| Ensartinib | | X-396 | | 3 |
|
|
| Entospletinib | | GS-9973
SYK INHIBITOR GS-9973 | | 2 |
|
|
| Entrectinib | Rozlytrek | NMS-E628
RXDX-101 | 2019 | 4 |
|
|
| Enzastaurin | Kinenza | LY-317615
LY317615
DB102
DB-102 | | 3 |
|
|
| Epertinib | | S-222611 | | 1 |
|
|
| Epitinib | | HMPL-813 | | 1 |
|
|
| Erdafitinib | Balversa | JNJ-42756493 | 2019 | 4 |
|
|
| Erlotinib | Tarceva | CP-358,774
CP-358774
CP-35877401
OSI-774
R-1415
RG-1415
RO-508231 | 2004 | 4 |
|
|
| Evobrutinib | | M-2951 | | 3 |
|
|
| Fadraciclib | | CYC-065
CYC065 | | 1 |
|
|
| Falnidamol | | BIBX 1382 | | 1 |
|
|
| Famitinib | | SHR-1020 | | 3 |
|
|
| Fasudil | | AT 877
AT-877
HA 1077
HA-1077
ZK-258594 | | 4 |
|
|
| Fedratinib | Inrebic | SAR-302503
SAR302503
TG-101348
TG101348 | 2019 | 4 |
|
|
| Fenebrutinib | | G-02599853
G02599853
GDC-0853
RG-7845
RG7845
RO-7010939
RO7010939 | | 3 |
|
|
| Filgotinib | Jyseleca | G-146034
G146034
GLPG-0634
GLPG0634
GS-6034 | 2020 (EMA, MHLW) | 4 |
|
|
| Fisogatinib | | BLU-554
BLU 554
BLU111362 | | 2 |
|
|
| Flumatinib | | HH-GV678
HHGV-678 | | 4 |
|
|
| Foretinib | | EXEL-2880
GSK-089
GSK-1363089
GSK-1363089G
GSK089
GSK1363089G
XL-880
XL880 | | 2 |
|
|
| Fosifidancitinib | | I-538 | | ? |
|
|
| Foslinanib | | CVM-1118
TRX 818
TRX-818 | | 2 |
|
|
| Fostamatinib | Tavalisse | R-788
R-935788
R788
R935788 | 2018 | 4 |
|
|
| Fruquintinib | | HMP-013
HMPL-013 | | 3 |
|
|
| Furmonertinib | | Alflutinib
AST-2818
AST2818 | | 3 |
|
|
| Futibatinib | | | | 3 |
|
|
| Galunisertib | | LY-2157299
LY2157299 | | 2 |
|
|
| Gandotinib | | LY-2784544
LY2784544 | | 2 |
|
|
| Gedatolisib | | PF-05212384
PKI-587 | | 2 |
|
|
| Gefitinib | Iressa | ZD-1839
ZD1839 | 2003 | 4 |
|
|
| Gilteritinib | Xospata | ASP-2215
ASP2215 | 2018 | 4 |
|
|
| Glesatinib | | MG-90265
MG-90265X
MG90265
MG90265GLY
MG90265H9
MG90265X
MGCD-265
MGCD265 | | 2 |
|
|
| Glumetinib | | | | 1 |
|
|
| Golvatinib | | E-7050
E7050 | | 2 |
|
|
| Gusacitinib | | ASN-002
ASN002
EN-3351
EN3351 | | 2 |
|
|
| Henatinib | | | | 1 |
|
|
| Ibrutinib | Imbruvica | CRA-032765
PC-32765
PCI 32765
PCI-32765
PCI-32765-00 | 2013 | 4 |
|
|
| Icotinib | Conmana | BPI-2009H | 2011 (CFDA) | 4 |
|
|
| Idelalisib | Zydelig | CAL-101
GS-1101
GS-11CAL-101 | 2014 | 4 |
|
|
| Ifidancitinib | | A 301
A-301
A301
R2010 | | 2 |
|
|
| Ilginatinib | | NS-018 | | 2 |
|
|
| Ilorasertib | | A-968660
A-968660.0
ABBOTT-968660
ABT-348
ABT-348, A-968660 | | 2 |
|
|
| Imatinib | Gleevec | STI-571 | 2001 | 4 |
|
|
| Inavolisib | | GDC-0077
GDC0077
RO7113755
RG6114 | | 2 |
|
|
| Infigratinib | Truseltiq | BGJ-398
BGJ398
MVP-BGJ398
NVP-BGJ398 | 2021 | 4 |
|
|
| Ipatasertib | | GDC-0068
RG-7440
RG7440 | | 3 |
|
|
| Itacitinib | | INCB-039110
INCB-39110
INCB039110 | | 3 |
|
|
| Itacnosertib | | TP-0184
TP0184 | | 1 |
|
|
| Izencitinib | | TD 1473
TD1473
TD-1473 | | 3 |
|
|
| Lanraplenib | | GS-9876 | | 2 |
|
|
| Lapatinib | Tykerb
Tyverb | GSK-572016
GW-2016
GW-572016
GW-572016X
GW572016 | 2007 | 4 |
|
|
| Larotrectinib | Vitrakvi | ARRY-470
BAY-2757556
BAY2757556
LOXO-101 | 2018 | 4 |
|
|
| Lazertinib | | GNS-1480
GNS1480
JNJ-73841937
YH-25448
YH25448
C-18112003-G | | 4 (MFDS) |
|
|
| Leniolisib | | CDZ173-NX | | 2 |
|
|
| Lenvatinib | Kisplyx
Lenvima | E-7080
ER-203492-00 | 2015 | 4 |
|
|
| Lerociclib | | G1T38 | | 1.5 |
|
|
| Lestaurtinib | | A-154475
A-154475.0
CEP-701
KT-555
KT-5555
KT5555
SP-924
SP924
SPM-924 | | 3 |
|
|
| Lifirafenib | | BGB 283
BGB-283 | | 1 |
|
|
| Linifanib | | A-741439
ABT-869
AL-39324
RG-3635 | | 3 |
|
|
| Linperlisib | | YY-20394
YY20394 | | 3 |
|
|
| Linsitinib | | ASP-7487
OSI-906
OSI-906AA | | 3 |
|
|
| Lorecivivint | | Adavivint
SM0-4690
SM04690 | | 2 |
|
|
| Lorlatinib | Lorbrena | PF-06463922 | 2018 | 4 |
|
|
| Lorpucitinib | | | | 1 |
|
|
| Losmapimod | | FTX-1821
FTX1821
Gsk-ahab
Gskahab
GW-856553
GW-856553X
GW856553X | | 3 |
|
|
| Lucitanib | | AL-3810
CO-3810
E-3810
S 80881
S-80881 | | 2 |
|
|
| Luxeptinib | | CG026806
CG-806 | | 1 |
|
|
| Maribavir | Livtencity | TAK-620
1263W94 | 2021 | 4 |
|
|
| Masitinib | Kinavet
Masivet | AB-1010 | | 3 |
|
|
| Mavelertinib | | PF-06747775 | | 2 |
|
|
| Merestinib | | LY-2801653
LY2801653 | | 2 |
|
|
| Mevociclib | | SY-1365
SY1365 | | 1 |
|
|
| Midostaurin | Rydapt | CGP 41251
CGP-41251
NVP-PKC412
PKC 412
PKC-412 | 2017 | 4 |
|
|
| Milciclib | | PHA 848125
PHA-848125 | | 2 |
|
|
| Miransertib | | ARQ 092
ARQ-092 | | 2 |
|
|
| Mirdametinib | | PD 0325901
PD-0325901
PD0325901 | | 2 |
|
|
| Mivavotinib | | TAK-659F | | 2 |
|
|
| Mobocertinib | Exkivity | TAK788
TAK-788
AP32788 | 2021 | 4 |
|
|
| Momelotinib | | CYT-0387
CYT-11387
CYT-387
CYT387
GS-0387 | | 3 |
|
|
| Motesanib | | AMG 706
AMG-706 | | 3 |
|
|
| Mubritinib | | TAK-165 | | 1 |
|
|
| Naporafenib | | LXH 254
LXH-254
LXH254
PAN-RAF INHIBITOR LXH254 | | 2 |
|
|
| Naquotinib | | ASP-8273
ASP8273 | | 3 |
|
|
| Nazartinib | | EGF-816
EGF816
NVP-EGF816-NX | | 3 |
|
|
| Neflamapimod | | 745
VD-31
VD-31,745
VD-31745
VRT-031745
VX-745 | | 2 |
|
|
| Nemiralisib | | GSK-2269557
GSK-2269557A
GSK2269557A | | 2 |
|
|
| Nemtabrutinib | | ARQ 531
K-1026 | | 1.5 |
|
|
| Neratinib | Nerlynx | CDP-820
HKI-272
WAY-179272 | 2017 | 4 |
|
|
| Netarsudil | Rhopressa | AR-13324 | 2017 | 4 |
|
|
| Nilotinib | Tasigna | AMN 107
AMN-107
AMN107 | 2007 | 4 |
|
|
| Ningetinib | | | | 1.5 |
|
|
| Nintedanib | Ofev
Vargatef | BIBF 1120
BIBF-1120
BIBF1120
Intedanib | 2014 | 4 |
|
|
| Oclacitinib | | Jaki
PF-03394197 | | 0 |
|
|
| Olafertinib | | CK101
CK‐101
RX-518
RX518 | | 1 |
|
|
| Olmutinib | | BI 1482694
BI-1482694
HM-61713
HM61713 | | 2 |
|
|
| Olverembatinib | | HQP1351 GZD824 | | 1.5 |
|
|
| Omipalisib | | GSK-2126458
GSK2126458 | | 1 |
|
|
| Onatasertib | | ATG-008
CC 223
CC-223 | | 2 |
|
|
| Onvansertib | | NMS-1286937
NMS-P937
PCM-075 | | 2 |
|
|
| Opaganib | | ABC 294640
ABC-294640 | | 2.5 |
|
|
| Orantinib | | NSC-702827
SU-6668
TSU-68 | | 3 |
|
|
| Orelabrutinib | | ICP022
ICP-022 | | 2 |
|
|
| Osimertinib | Tagrisso | AZD-9291
AZD9291
Mereletinib | 2015 | 4 |
|
|
| Pacritinib | | ONX-0803
SB-1518
SB1518 | | 3 |
|
|
| Palbociclib | Ibrance | PD-0332991 | 2015 | 4 |
|
|
| Pamapimod | | R-1503
R1503
RO 4402257
RO-4402257 | | 2 |
|
|
| Pamufetinib | | TAS-115 | | 2 |
|
|
| Panulisib | | | | 1 |
|
|
| Parsaclisib | | INCB-050465
INCB050465 | | 3 |
|
|
| Paxalisib | | GDC-0084
GDC0084
G02441729
G-02441729
RG-7666 | | 2 |
|
|
| Pazopanib | Votrient | GW786034 | 2009 | 4 |
|
|
| Peficitinib | | ASP-015K
ASP015K
JNJ-54781532 | | 3 |
|
|
| Pegcantratinib | | CT327
CT-327
SNA-120 | | 2 |
|
|
| Pelitinib | | EKB-569
WAY-EKB-569 | | 2 |
|
|
| Pemigatinib | Pemazyre | INCB054828 | 2020 | 4 |
|
|
| Peposertib | | M-3814
Nedisertib
M3814
MSC 2490484A
MSC-2490484A
MSC2490484A | | 1.5 |
|
|
| Pexidartinib | Turalio | CML-261
PLX-3397
PLX3397 | 2019 | 4 |
|
|
| Pexmetinib | | | | 1 |
|
|
| Pictilisib | | CDC-0941
GDC 0941
GDC-0941
RG-7321 | | 2 |
|
|
| Pilaralisib | | SAR-245408
SAR245408
XL-147
XL147 | | 2 |
|
|
| Pimasertib | | AS 703026
AS-703026
AS703026
EMD 1036239
EMD-1036239
G-02443714
MSC-1936369A
MSC-1936369B
MSC1936369A
MSC1936369A
AS703026
EMD 1036239 | | 2 |
|
|
| Pirtobrutinib | | LOXO-305 | | 3 |
|
|
| Ponatinib | Iclusig | AP-24534
AP24534 | 2012 | 4 |
|
|
| Poseltinib | | HM71224
LY3337641 | | 2 |
|
|
| Poziotinib | | HM 781-36
HM 781-36B
HM-781-36
HM-781-36B
NOV-120101 | | 2 |
|
|
| Pralsetinib | Gavreto | BLU-123244
BLU-667
BLU123244
X-581238
X581238 | 2020 | 4 |
|
|
| Prexasertib | | LY2606368 | | 2 |
|
|
| Puquitinib | | | | 1 |
|
|
| Pyrotinib | | | | 3 |
|
|
| Quizartinib | | AC-010220
AC-220
AC010220
AC220
ASP-2689 | | 3 |
|
|
| Rabusertib | | IC-83
LY-2603618
LY2603618 | | 2 |
|
|
| Radotinib | | IY5511 | | 3 |
|
|
| Ralimetinib | | LSN-2322600
LSN2322600
LY-2228820
LY2228820
LY22288220 | | 2 |
|
|
| Ravoxertinib | | GDC-0994
GDC0994
RG-7842 | | 1 |
|
|
| Rebastinib | | DCC-2036
DP-1919 | | 2 |
|
|
| Recilisib | | Ex-rad
ON 01210
ON 01210.NA
ON-01210 | | 1 |
|
|
| Refametinib | | BAY 869766
BAY 8697661
BAY-86-9766
BAY-869766
BAY-8697661
BAY86-9766
RDEA 119
RDEA-119 | | 2 |
|
|
| Regorafenib | Stivarga | BAY 73-4506
BAY 73-4506 MONOHYDRATE
BAY-73-4506
BAY-734506 | 2012 | 4 |
|
|
| Remibrutinib | | LOU064 | | 2 |
|
|
| Repotrectinib | | TPX-0005
TRX-0005 | | 1.5 |
|
|
| Rezivertinib | | BPI 7711 | | 3 |
|
|
| Ribociclib | Kisqali | LEE-011
LEE-011A
LEE011
LEE011A
NVP-LEE011 | 2017 | 4 |
|
|
| Rigosertib | | ON 01910 | | 3 |
|
|
| Rilzabrutinib | | PRN-1008
PRN1008 | | 3 |
|
|
| Rimacalib | | SMP-114 | | 2 |
|
|
| Ripasudil | | | | 2 |
|
|
| Ripretinib | Qinlock | DCC-2618 | 2020 | 4 |
|
|
| Ritlecitinib | | PF-06651600
PF06651600 | | 3 |
|
|
| Riviciclib | | | | 2 |
|
|
| Roblitinib | | FGF-401
FGF401
NVP-FGF401 | | 2 |
|
|
| Rociletinib | | AVL-301
CNX-419
CO-1686
CS-1631 | | 3 |
|
|
| Rogaratinib | | BAY-1163877 | | 2 |
|
|
| Roniciclib | | | | 2 |
|
|
| Ropsacitinib | | PF-06826647 | | 2 |
|
|
| Ruboxistaurin | Arxxant | LY-333531 | | 3 |
|
|
| Ruxolitinib | Jakafi
Jakavi
Opzelura | INC-424
INC424
INCB-018424
INCB-18424
INCB018424 | 2011 | 4 |
|
|
| Samotolisib | | LY 3023414
LY-3023414
LY3023414 | | 2 |
|
|
| Samuraciclib | | CT7001
ICEC-0942
ICEC0942
PPDA-001 | | 1 |
|
|
| Sapanisertib | | INK-128
INK128
MLN-0128
MLN0128
TAK-228 | | 2 |
|
|
| Sapitinib | | AZD-8931
AZD8931 | | 2 |
|
|
| Saracatinib | | AZ-10353926
AZD-0530
AZD0530 | | 3 |
|
|
| Savolitinib | Orpathys | AZD-6094
AZD6094
HMPL-504
Volitinib | 2021 (NMPA) | 4 |
|
|
| Selatinib | | | | 1 |
|
|
| Seletalisib | | UCB-5857
UCB5857 | | 2 |
|
|
| Seliciclib | | AL-39256
CYC-202
NSC-701554 | | 2 |
|
|
| Selitrectinib | | LOXO-195 | | 1.5 |
|
|
| Selonsertib | | GS-4997 | | 3 |
|
|
| Selpercatinib | Retevmo | LOXO-292
LY-3527723
LY3527723
WHO 10967 | 2020 | 4 |
|
|
| Selumetinib | Koselugo | ARRY-142886
ARRY-886
AZD-6244
AZD6244 | 2020 | 4 |
|
|
| Semaxanib | | NSC-696819
Semaxinib
SU-5416
SU005416
SU5416 | | 3 |
|
|
| Serabelisib | | AGN-PC-0DB6FL
INK1117
MLN-1117
MLN1117
TAK-117 | | 2 |
|
|
| Seralutinib | | GB-002
Gb002
PK-10571
PK10571 | | 2 |
|
|
| Silmitasertib | | CX 4945
CX-4945
CX4945 | | 2 |
|
|
| Simotinib | | SIM-6802 | | 3 |
|
|
| Simurosertib | | TAK-931 | | 2 |
|
|
| Sitravatinib | | MG-516
MG-91516
MGCD-516
MGCD516 | | 3 |
|
|
| Solcitinib | | G-154578
G154578
GLPG-0778
GLPG-0788
GLPG0778
GSK-2586184
GSK-2586184A
GSK2586184A | | 2 |
|
|
| Sonolisib | | PX-866 | | 2 |
|
|
| Sorafenib | Nexavar | BAY 43-9006
BAY-43-9006 | 2005 | 4 |
|
|
| Sotrastaurin | | AEB-071
AEB071
NVP-AEB071 | | 2 |
|
|
| Spebrutinib | | AVL-292
CC-292 | | 2 |
|
|
| Sunitinib | Sutent | SU-011248
SU-11248
SU011248 | 2006 | 4 |
|
|
| Surufatinib | | HMPL-012
Sulfatinib
KDR-IN-1 | | 3 |
|
|
| Tafetinib | | SIM 010603
SIM-010603 | | 1 |
|
|
| Taletrectinib | | DS-6051b
AB-106 | | 2 |
|
|
| Talmapimod | | SCIO 469
SCIO-469 | | 2 |
|
|
| Tamatinib | | R-406 | | 2 |
|
|
| Tandutinib | | CT 53518
CT-53518
CT53518
MLN-0518
MLN-518 | | 2 |
|
|
| Tanzisertib | | CC-930
JNK 930
JNK-930 | | 2 |
|
|
| Tarloxotinib | | Tarloxotinib bromide | | 2 |
|
|
| Taselisib | | GDC-0032
RG-7604 | | 3 |
|
|
| Tasurgratinib | | E-7090
E7090 | | 2 |
|
|
| Telatinib | | BAY 57-9352
BAY-57-9352
BAY-579352 | | 2 |
|
|
| Tenalisib | | | | 2 |
|
|
| Tepotinib | Tepmetko | EMD 1214063
EMD-1214063
EMD1214063
MSC-2156119
MSC-2156119J
MSC2156119 | 2021 | 4 |
|
|
| Tesevatinib | | EXEL-7647
KD-019
KD-020
KD019
XL-647
XL647 | | 3 |
|
|
| Theliatinib | | HMPL-309
Xiliertinib | | 1 |
|
|
| Tirabrutinib | | GS-4059
ONO-4059 | | 2 |
|
|
| Tirbanibulin | | KX2-391
KX-01 | | 3 |
|
|
| Tivantinib | | ARQ 197
ARQ-197 | | 3 |
|
|
| Tivozanib | Fotivda | ASP-4130
AV-951
KIL-8951
KIL8951
KRN-951 | 2021 | 4 |
|
|
| Tizaterkib | | ATG-017
AZD0364 | | 1 |
|
|
| Toceranib | | PHA-291639 | | 0 |
|
|
| Tofacitinib | Xeljanz | 550
CP 690550
CP- 690 550
CP-690
CP-690,550
CP-690-550
CP-690550
CP690,550
CP690550
Tasocitinib | 2012 | 4 |
|
|
| Tolebrutinib | | BTK'168
PRN-2246
PRN2246
SAR442168 | | 3 |
|
|
| Tomivosertib | | EFT 508
EFT-508
EFT508 | | 2 |
|
|
| Tozasertib | | MK-045
MK-0457
VX-68
VX-680 | | 2 |
|
|
| Trametinib | Mekinist | GSK-1120212
GSK1120212
JTP 74057
JTP-74057
TMT-212
TMT212 | 2013 | 4 |
|
|
| Trilaciclib | Cosela | G1T28 | 2021 | 4 |
|
|
| Tucatinib | Tukysa | ARRY-380
ONT-380 | 2020 | 4 |
|
|
| Ulixertinib | | BVD-523
Bvd-erk
VRT-752271 | | 2 |
|
|
| Umbralisib | Ukoniq | RP-5264
RP5264
TGR 1202
TGR-1202 | 2021 | 4 |
|
|
| Upadacitinib | Rinvoq | ABT-494 | 2019 | 4 |
|
|
| Uprosertib | | GSK-2141795
GSK-2141795C
GSK2141795
GSK2141795C | | 2 |
|
|
| Vactosertib | | TEW 7197
TEW-7197 | | 2 |
|
|
| Vandetanib | Caprelsa
Zactima | GNF-PF-2188
ZD-64
ZD-6474
ZD6474 | 2011 | 4 |
|
|
| Varlitinib | | AR-00334543
ARRY-334543
ARRY-543
ASLAN-001
ASLAN001 | | 2.5 |
|
|
| Vatalanib | | BAY-86-5127
CGP-79787
K-222584
NVP-PTK787
PTK-787
PTK787
ZK-222584 | | 3 |
|
|
| Vebreltinib | | APL-101
CBI-3103
PLB-1001 | | 1 |
|
|
| Vecabrutinib | | BIIB-062
BSK-4841
FP-0182
FP0182
SNS-062 | | 1 |
|
|
| Vemurafenib | Zelboraf | PLX-4032
PLX4032
RG 7204
RG-7204
RO 5185426
RO-51-85426
RO-5185426 | 2011 | 4 |
|
|
| Verosudil | | AR-12286 | | 2 |
|
|
| Vimseltinib | | DCC-3014
DCC3014 | | 2 |
|
|
| Vistusertib | | AZD-2014
AZD2014 | | 2 |
|
|
| Vodobatinib | | K0706 | | 2 |
|
|
| Volasertib | | BI 6727
BI-6727 | | 3 |
|
|
| Vorolanib | | X-82 | | 2 |
|
|
| Voruciclib | | | | 2 |
|
|
| Voxtalisib | | SAR-245409
SAR245409
XL-765 | | 2 |
|
|
| Xiliertinib | | HMPL-309
HMPL309
Theliatinib | | 1 |
|
|
| Zandelisib | | ACC-524
ME-401
PW-143
PWT-143
PWT143
ME401 | | 3 |
|
|
| Zanubrutinib | Brukinsa | BGB-3111 | 2019 | 4 |
|
|
| Zoligratinib | | DEBIO-1347
DEBIO1347 | | 1 |
|
|
| Zorifertinib | | AZD-3759
AZD3759
AZD 3759 | | 2 |
|
|
| Zotiraciclib | | EX45
SB-1317
SB1317
TG-02
TG02 | | 1 |
|
|
