Drugs and clinical candidates

This overview is powered by the PKIDB1,2 from the Bonnet lab and is complemented with in-house annotations.
INN / Name Brand name Synonyms Approval year Phase KLIFS links Structures
ASP4132 1

BI 2536BI-2536
BI2536
2


AMG-208 2


GSK-690693GSK690693 1


ENMD-2076 2


ASP5878 1

AZD4573 2


SAR125844 2


AT7519AT7519M 1


AMG319 2


SCR-1481B1BMS-817378 1

TAS-117 2

MK-8353SCH900353 1


BFH772 2

FN-1501 1

PRN1371 1


TG 100801TG100801 2

EOC317ACTB-1003 1

TP-3654 1

CEP-37440 1

ODM-203 1

AZD-8835AZD8835
AZD 8835
1

PF-06459988 2


AMG-337 2


PIM447LGH447 1


BAY1082439 1

ARRY-382 2

CC-115 1

ASP3026 1


XL019 1


JI-101 2

XL228 1

RGB-286638 1

GSK1059615 1

TAK-901 1

VS-5584SB2343 1

MRX-2843UNC2371 1

BGT226NVP-BGT226
BGT-226
BGT 226
2

AZD8330ARRY-424704
ARRY-704
1

ON123300ON 123300 2

SAR-260301SAR260301 1


PND-1186VS-4718
SR-2516
1

CP-547632 2


TAK-960 1


GDC-0349 1

MK-8033 1

TAK-593 1

Palomid529 1

JNJ-38877605 1

AZD1208 1

AZD-7762 1


PF-04217903 1


MK-2461MK2461 2

AZD-8055 1

MEN1611CH5132799
CH 5132799
CH-5132799
1


BMS-599626AC480 1

RO4987655CH4987655 1


TAK-285 1


CC-401 1

OSI-930 1

SGX-523 1


PHA-793887 1


VS-6766RG 7304
CKI27
CH5126766
RO5126766
1


XL092 1

AZD-8154AZD8154
AZD 8154
2


PF-06952229 1

LY-3200882 2

AR-13503Metabolite netarsudil 1

TT 00420TT-00420 1

CLN-081TAS6417 1/2

BTX-A51 1

IPN60130BLU-782 1

DAY101MLN-2480
MLN2480
TAK580
TAK-580
1

AZD4547AZD-4547
KB-74810
2

GDC-0134 1

JNJ-67856633JNJ67856633
JNJ 67856633
2

SHR0302SHR 0302 3

CFI-400945CFI400945
CFI 400945
1

LY3295668AK-01 1

KB-0742 1

PF-07104091 2

M4205 1

MAP855 0

RP-6306 1

GSK2982772 2

VIC 1911VIC-1911
TAS-119
TAS-2104
1.5

MEN1703SEL24 1.5

BLU-945BLU 945 1

RP-3500 1.5

AZD4604AZD-4604
Jak1-IN-7
1

AZD7624AZD-7624 2

CFI-402257CFI402257 1.5

MLI-2MLi-2 1


LUT014LUT-014 2

AZD1390 1

BIIB068BIIB-068 1

ARRY-371797ARRY-797
ARRY371797
ARRY797
2

GSK2292767GSK-2292767 1


AZD7648AZD-7648 1.5


MW150MW-150
MW01-18-150SRM
1


RG-1530R-1530
R1530
RG1530
1

AZD7451AZ12607092
AZD-7451
1

GR-389988GR389988
GZ389988
GZ389988A
2

RV6153RV-6153 1

RV1729RV-1729 1

GSK2646264 1

KX2-361KX-02
KX2 361
KX2361
1

AZD0156 1

TAK-733TAK733 1


BMS-986142BMS986142 2


PF-114PF114 1.5

CBS-3595 1

PF-06263276PF 0626327
PF0626327
1


GDC-0834GDC 0834 1


AC430AC-430 1

PLX8394PLX 8394
PLX-8394
1.5

LY3009120LY-3009120 1


PF-3758309PF-03758309
PF3758309
1


SAR407899HY-15687A
SAR-407899
2

CUDC-101CUDC101 1

SGI-1776SGI 1776
SGI1776
1

AZD8186AZD 8186
AZD-8186
1

AZD5438AZD 5438
AZD-5438
1


GSK1070916GSK-1070916 1

LY2584702LY 2584702
LY-2584702
1

CEP-1347CEP 1347
CEP1347
KT-7515
KT7515
3

XL413BMS-863233
BMS863233
XL-413
1


LY2874455LY-2874455 1


P505-15BIIB057
PRT-062607
PRT062607
0


MK-5108MK5108
VX-689
VX689
1


AMG-900AMG 900
AMG900
1

AZD6482AZD 6482
AZD-6482
1


PF-477736PF 477736
PF-00477736
1

VE-821VE 821 0

KU-60019 0

GSK650394GSK-650394 0


BI-D1870 0

GSK269962AGSK-269962A
GSK269962
0

PF-4708671PF4708671 0


AKN-028AKN 028
AKN028
1.5

ZSTK474TCMDC-137004
ZSTK 474
ZSTK-474
1.5


LY2090314LY-2090314 1.5

BMS-911543BMS 911543
BMS911543
1.5

BMS-777607BMS 777607
BMS777607
2


BMS-754807BMS 754807
BMS754807
2


AT-9283AT 9283
AT9283
2

MK-2206MK 2206 2

MK-8776MK 8776
SCH 900776
2

PF-04691502PF 04691502
PF04691502
2


7-hydroxystaurosporineKRX-0601
KRX0601
UCN 01
UCN-01
2


CP-724714CP 724714
CP724714
2

BMS-690514BMS 690514
BMS690514
2

BMS-582949BMS 582949
BMS582949
PS 540446
PS-540446
PS540446
2


PH-797804 2


AZD6703AZ 12012199
AZ-12012199
AZ12012199
AZD 6703
AZD-6703
1


VX-702I14-1965
VX 702
VX702
2

TG-100-115TG 100-115
TG 100115
TG100-115
1.5


SU-14813SU014813
SU14813
1

KW-2449KW 2449 1

GSK-461364AGSK 461364
GSK-461364
GSK461364
GSK461364A
1

CI-1040CI 1040
CI1040
PD-184352
PD184352
2

CHIR-265CHIR 265
CHIR265
RAF 265
RAF-265
RAF265
2


BMS-387032BMS 387032
BMS387032
SNS 032
SNS-032
1


CC-90001CC 90001 2

HMPL-523HMPL523
HMPL 523
3

RVU120SEL120
SEL120-34A
1.5

TAK-020 1

ZN-c3ZN c3 2

ASTX029ASTX-029 1.5

CC-90005 1

AS-0141 1

SY-5609SY-0005609
CDK7-IN-3
1

Debio0123Debio 0123
Debio-01230
1

AUM-001ETC-1907206
ETC-206
2

LY3405105 1

HM43239HM-43239 1.5

ESK981CEP 11981
CEP11981
1

BIIB091 1

GSK3145095 2

GSK2983559 1

GLPG0259GLPG-0259
GTPL9848
2

FF10101FF-10101-01 1

IM156HL156A
HL271
1

T-1101TAI-95 1

ONO-7475 2

CG-806 2

CC-90003 1

KO-947 1

GDC-0575ARRY-575
RG7741
1

TAS0728 2

OMO-1OMO1
JNJ38877618
JNJ-38877618
1

AV-412MP412 1

CEP-40783RXDX-106 1

M2698MSC2363318A 1

BAY1125976BAY-1125976 1

LY3214996 2

AEE788AEE 788
NVP-AEE788
2


AbemaciclibVerzenio
Verzenios
LY-2835219
LY2835219
2017 4


AbivertinibA610
AC-0010
AC0010
ACEA100610
Avitinib
EX-ACEA0010
3

AbrocitinibCibinqoPF-049658422022 4


AcalabrutinibCalquenceACP-1962017 4

AcalisibCAL-120
CAL120
GS-9820
GS9820
2

AcumapimodBCT 197
BCT-197
BCT197
2

AdavosertibAZD 1775
AZD-1775
AZD1775
MK-1775
MK1775
2


AfatinibGilotrif
Giotrif
BIBW-2992
BIBW2992
2013 4



AfuresertibASB-183
ASB183
GSK-2110183
GSK-2110183C
GSK2110183
GSK2110183C
LAE002
2

AgerafenibAB-024
AC-013773
CEP-32496
RXDX 105
RXDX-105
1

AlectinibAlecensaAF-802
AF802
CH-5424802
CH5424802
RO-5424802
RO5424802
2015 4


AlisertibMLN 8237
MLN-8237
MLN8237
3


AllitinibALL-3
AST-1306
2

Alofanib 1

AlpelisibPiqrayBYL-719
NVP-BYL719
2019 4


AltiratinibDCC-2701
DP-5164
1

AlvocidibFlavopiridol
HL 275
HL-275
HMR 1275
HMR-1275
L 86 8275
L-868275
L86-8275
MDL 107,826A
MDL-107826A
NSC-649890
3


AmcasertibBBI-503
BBI503
2

AmdizalisibHMPL-689 2

AmuvatinibHPK 56
HPK-56
HPK56
MP 470
MP-470
MP470
2

ApilimodLAM-002A
LAM002A
STA 5326
STA-5326
STA5326
2

ApitolisibG-038390
G-038390.1
GDC-0980
GDC-0980.1
RG-7422
RG7422
2


AsciminibScemblixABL-001
ABL001
ABL001-NX
NVP-ABL001
2021 4


AtuveciclibBAY 1143572
BAY-1143572
BAY1143572
1

AumolertinibAmeileHS-10296
Almonertinib
4 (NMPA)

AvapritinibAyvakit70C366
BLU-285
C-366
X-720776
X720776
2020 4

AvotaciclibBEY 1107
BEY1107
BEY-1107
1

AxitinibInlytaAG-013736
AG-13736
2012 4


BafetinibCNS-9
INNO-406
NS-187
2


BalamapimodMKI-833 1

BarasertibAZD 1152
AZD-1152
AZD1152
3

BaricitinibOlumiantINCB-028050
INCB-28050
INCB028050
LY-3009104
LY3009104
2017 4


BefotertinibD-0316
D 0316
D0316
2

BelizatinibTSR-011
TSR011
2


BelumosudilRezurockKD025
SLx2119
2021 4

BelvarafenibHM95573
GDC-5573
2


BemcentinibBGB 324
BGB-324
BGB324
CS-1046
HY-15150
KB-80319
QC-11751
R 428
R-428
R428
SYN-1131
SYN1131
W-5845
2

BentamapimodAS-602801
PGL-5001
2

BerzosertibM-6620
M6620
VE-822
VX-970
VX970
2

BezuclastinibPLX9486
CGT 9486
2

BimiralisibNC-B5
NCB5
PI3K-IN-2
PQR-309
PQR309
2


BinimetinibMektoviARRY 438162
ARRY-162
ARRY-438162
MEK-162
MEK162
NVP-MEK162
2018 4


BosutinibBosulifBosutinib monohydrate
SK-606
SKI-606
2012 4


BranebrutinibBMS-986195 2


BrepocitinibPF-06700841 2


BriciclibON 014185 1

BrigatinibAlunbrigAP-26113
AP26113
2017 4


BrivanibBMS-540215 3

Brivanib alaninateBMS-582664
BMS-582664-02
Brivanib l-alanine ester
3

BuparlisibBKM-120
BKM-120NX
BKM120-NX
NVP-BKM-120
NVP-BKM120
3


CabozantinibCabometyx
Cometriq
BMS-907351
XL-184
XL184
2012 4

CanertinibCI-1033 3

CapivasertibAZC5363
AZD 5363
AZD-5363
AZD5363
3


CapmatinibTabrectaINC-280
INC280
INCB-28060
NVP-INC280
NVP-INC280-NX
NYP-INC280-NX
2020 4

CatequentinibFOCUS VAL3818
Anlotinib
Altn
4

CediranibRecentinAZD-2171
AZD2171
ZD-2171
3

CenisertibAS-703569
R-763
1

CeralasertibAZD6738 2

Cerdulatinib 2.5

CeritinibZykadiaLDK-378
LDK378
NVP-LDK-378-NX
NVP-LDK378-NX
2014 4


ChiauranibCS-2164
CS2164
3

CobimetinibCotellicGDC-0623
GDC-0973
RG 7420
RG-7420
RG-7421
RG7420
XL-518
2015 4


ConteltinibCT-707
CT707
1

CopanlisibAliqopaBAY 80-6946
BAY-80-6946
BAY80-6946
2017 4


Cotosudil 0

CrenolanibARO 002
ARO-002
CP 868596
CP-868,596
CP-868596
3


CrizotinibXalkoriPF-02341066
PF-2341066
2011 4


DabrafenibTafinlarGSK-2118436
GSK-2118436A
GSK2118436
GSK2118436A
2013 4


DacomitinibVizimproDacomitinib hydrate
PF-00299804
2018 4


DactolisibBEZ-235
BEZ235
NVP-BEZ235
NVP-BEZ235-NX
3

DalpiciclibSHR 6390
SHR-6390
SHR6390
3

DanusertibPHA-739358 2


DarovasertibIDE-196
IDE196
LXS-196
LXS196
1

DasatinibDasatinib
Sprycel
BMS-354825
BMS-354825 HYDRATE
BMS-354825-03
Dasatinib hydrate
Dasatinib monohydrate
2006 4


DecernotinibAdelatinib
VRT-831509
VX-509
2


DefactinibPF-04554878
VS-6063
2


DefosbarasertibBarasertib-hqpa
AZD-1152HQPA
AZD-2811
AZD2811
AZD 2811
2

Delgocitinib 2


DerazantinibARQ 087
ARQ-087
ARQ087
2

DeucravacitinibBMS-986165
BMS986165
3


DeuruxolitinibCTP-543
CTP543
D8-ruxolitinib
3

DezapelisibINCB040093 0

DilmapimodGW-681323
SB-681323
SB681323
2

DinaciclibMK-7965
SCH 727965
SCH-727965
3


DonafenibZepsunSorafenib (D3)
CM-4307
2021 (NMPA) 4

DoramapimodBIRB 796 BS
BIRB-796
BIRB-796 BS
2


DovitinibCHIR-258
GFKI-258
NVP-TKI258
TKI-258
3


DubermatinibHCL-2084
TP 0903
TP-0903
TP0903
1.5

DuvelisibCopiktraINK-1147
INK-1197
IPI-145
2018 4

EbvaciclibPF-06873600 2


EclitasertibDNL758
SAR443122
2

EdicotinibJNJ-40346527 2

EdralbrutinibSHR-1459
SHR1459
TG-1701
TG1701
1

EganelisibIPI-549
IPI549
2


ElimusertibBAY 1895344
BAY-1895344
BAY1895344
1.5

Elraglusib9-ING-41 2

ElsubrutinibABBV 105 2

ElzovantinibTPX-0022
TPX0022
CSF1R-IN-2
1

EmavusertibCA-4948
AU-4948
AU4948
CA4948
2

Empesertib(-)-BAY-1161909
BAY 1161909
MPS1-IN-5
1


EncorafenibBraftoviLGX-818
NVP-LGX-818-NXA
NVP-LGX818
NVP-LGX818-NXA
2018 4

EnitociclibVIP152
BAY-1251152
1

EnsartinibX-396 3

EntospletinibGS-9973
SYK INHIBITOR GS-9973
2


EntrectinibRozlytrekNMS-E628
RXDX-101
2019 4


EnzastaurinKinenzaLY-317615
LY317615
DB102
DB-102
3

EpertinibS-222611 1

EpitinibHMPL-813 1

ErdafitinibBalversaJNJ-427564932019 4


ErlotinibTarcevaCP-358,774
CP-358774
CP-35877401
OSI-774
R-1415
RG-1415
RO-508231
2004 4


EvobrutinibM-2951 3


FadraciclibCYC-065
CYC065
1

FalnidamolBIBX 1382 1

FamitinibSHR-1020 3

FasudilAT 877
AT-877
HA 1077
HA-1077
ZK-258594
4


FedratinibInrebicSAR-302503
SAR302503
TG-101348
TG101348
2019 4


FenebrutinibG-02599853
G02599853
GDC-0853
RG-7845
RG7845
RO-7010939
RO7010939
3


FilgotinibJyselecaG-146034
G146034
GLPG-0634
GLPG0634
GS-6034
2020 (EMA, MHLW) 4


FimepinostatCUDC 907
CUDC-907
2

FisogatinibBLU-554
BLU 554
BLU111362
2


Flonoltinib 1

FlumbatinibXinfuFlumatinib
HH-GV678
HHGV-678
2019 (NMPA) 4

ForetinibEXEL-2880
GSK-089
GSK-1363089
GSK-1363089G
GSK089
GSK1363089G
XL-880
XL880
2


Fosifidancitinib I-538 ?

FoslinanibCVM-1118
TRX 818
TRX-818
2

FostamatinibTavalisseR-788
R-935788
R788
R935788
2018 4


FruquintinibHMP-013
HMPL-013
3

FurmonertinibAlflutinib
AST-2818
AST2818
3

Futibatinib 3


GalunisertibLY-2157299
LY2157299
2

GandotinibLY-2784544
LY2784544
2

GartisertibM-4344
M4344
VX-803
VX803
1

GedatolisibPF-05212384
PKI-587
2


GefitinibIressaZD-1839
ZD1839
2003 4


GilteritinibXospataASP-2215
ASP2215
2018 4


GlesatinibMG-90265
MG-90265X
MG90265
MG90265GLY
MG90265H9
MG90265X
MGCD-265
MGCD265
2

Glumetinib 1

GolidocitinibDZD4205
AZD-4205
DZD 4205
AZD4205
1/2

GolvatinibE-7050
E7050
2


GusacitinibASN-002
ASN002
EN-3351
EN3351
2

Henatinib 1

IbrutinibImbruvicaCRA-032765
PC-32765
PCI 32765
PCI-32765
PCI-32765-00
2013 4



IcotinibConmanaBPI-2009H2011 (CFDA) 4

IdelalisibZydeligCAL-101
GS-1101
GS-11CAL-101
2014 4


IfidancitinibA 301
A-301
A301
R2010
2

IlginatinibNS-018 2

IlorasertibA-968660
A-968660.0
ABBOTT-968660
ABT-348
ABT-348, A-968660
2

ImatinibGleevecSTI-5712001 4


InavolisibGDC-0077
GDC0077
RO7113755
RG6114
2

InfigratinibTruseltiqBGJ-398
BGJ398
MVP-BGJ398
NVP-BGJ398
2021 4


IpatasertibGDC-0068
RG-7440
RG7440
3


ItacitinibINCB-039110
INCB-39110
INCB039110
3

ItacnosertibTP-0184
TP0184
1

IzencitinibTD 1473
TD1473
TD-1473
3

LanraplenibGS-9876 2


LapatinibTykerb
Tyverb
GSK-572016
GW-2016
GW-572016
GW-572016X
GW572016
2007 4


LarotrectinibVitrakviARRY-470
BAY-2757556
BAY2757556
LOXO-101
2018 4

LazertinibGNS-1480
GNS1480
JNJ-73841937
YH-25448
YH25448
C-18112003-G
4 (MFDS)

LeniolisibCDZ173-NX 2


LenvatinibKisplyx
Lenvima
E-7080
ER-203492-00
2015 4


LerociclibG1T38 1.5

LestaurtinibA-154475
A-154475.0
CEP-701
KT-555
KT-5555
KT5555
SP-924
SP924
SPM-924
3

LifirafenibBGB 283
BGB-283
1


LinifanibA-741439
ABT-869
AL-39324
RG-3635
3

LinperlisibYY-20394
YY20394
3

LinsitinibASP-7487
OSI-906
OSI-906AA
3

LorecivivintAdavivint
SM0-4690
SM04690
2

LorlatinibLorbrena
Lorviqua
PF-064639222018 4


Lorpucitinib 1

LosmapimodFTX-1821
FTX1821
Gsk-ahab
Gskahab
GW-856553
GW-856553X
GW856553X
3

LucitanibAL-3810
CO-3810
E-3810
S 80881
S-80881
2


LuxeptinibCG026806
CG-806
1

MaribavirLivtencityTAK-620
1263W94
2021 4

MasitinibKinavet
Masivet
AB-1010 3


MavelertinibPF-06747775 2


MerestinibLY-2801653
LY2801653
2


MevociclibSY-1365
SY1365
1

MidostaurinRydaptCGP 41251
CGP-41251
NVP-PKC412
PKC 412
PKC-412
2017 4


MilciclibPHA 848125
PHA-848125
2


MiransertibARQ 092
ARQ-092
2


MirdametinibPD 0325901
PD-0325901
PD0325901
2


MivavotinibTAK-659F 2


MobocertinibExkivityTAK788
TAK-788
AP32788
2021 4

MomelotinibCYT-0387
CYT-11387
CYT-387
CYT387
GS-0387
3


MotesanibAMG 706
AMG-706
3


MubritinibTAK-165 1

NaporafenibLXH 254
LXH-254
LXH254
PAN-RAF INHIBITOR LXH254
2


NaquotinibASP-8273
ASP8273
3


NazartinibEGF-816
EGF816
NVP-EGF816-NX
3


Neflamapimod745
VD-31
VD-31,745
VD-31745
VRT-031745
VX-745
2


NemiralisibGSK-2269557
GSK-2269557A
GSK2269557A
2


NemtabrutinibARQ 531
K-1026
1.5

NeratinibNerlynxCDP-820
HKI-272
WAY-179272
2017 4


NetarsudilRhopressaAR-133242017 4

NezulcitinibTD-0903
TD 0903
TD0903
2

NilotinibTasignaAMN 107
AMN-107
AMN107
2007 4


Ningetinib 1.5

NintedanibOfev
Vargatef
BIBF 1120
BIBF-1120
BIBF1120
Intedanib
2014 4


OclacitinibJaki
PF-03394197
0

OlafertinibCK101
CK‐101
RX-518
RX518
1

OlmutinibBI 1482694
BI-1482694
HM-61713
HM61713
2

OlverembatinibHQP1351 GZD824 1.5

OmipalisibGSK-2126458
GSK2126458
1


OnatasertibATG-008
CC 223
CC-223
2

OnvansertibNMS-1286937
NMS-P937
PCM-075
2


OpaganibABC 294640
ABC-294640
2.5

OrantinibNSC-702827
SU-6668
TSU-68
3


OrelabrutinibICP022
ICP-022
2

OsimertinibTagrissoAZD-9291
AZD9291
Mereletinib
2015 4



PacritinibVonjoONX-0803
SB-1518
SB1518
2022 4


PalbociclibIbrancePD-03329912015 4


PamapimodR-1503
R1503
RO 4402257
RO-4402257
2


PamufetinibTAS-115 2

Panulisib 1

ParsaclisibINCB-050465
INCB050465
3

PaxalisibGDC-0084
GDC0084
G02441729
G-02441729
RG-7666
2

PazopanibVotrientGW7860342009 4

PeficitinibASP-015K
ASP015K
JNJ-54781532
3


PegcantratinibCT327
CT-327
SNA-120
2

PelitinibEKB-569
WAY-EKB-569
2


PemigatinibPemazyreINCB0548282020 4

PeposertibM-3814
Nedisertib
M3814
MSC 2490484A
MSC-2490484A
MSC2490484A
1.5


PexidartinibTuralioCML-261
PLX-3397
PLX3397
2019 4


Pexmetinib 1

PictilisibCDC-0941
GDC 0941
GDC-0941
RG-7321
2


PilaralisibSAR-245408
SAR245408
XL-147
XL147
2

PimasertibAS 703026
AS-703026
AS703026
EMD 1036239
EMD-1036239
G-02443714
MSC-1936369A
MSC-1936369B
MSC1936369A
MSC1936369A
AS703026
EMD 1036239
2


PirtobrutinibLOXO-305
RXC-005
LY-3527727
LY3527727
3

PonatinibIclusigAP-24534
AP24534
2012 4


PoseltinibHM71224
LY3337641
2

PoziotinibHM 781-36
HM 781-36B
HM-781-36
HM-781-36B
NOV-120101
2

PralsetinibGavretoBLU-123244
BLU-667
BLU123244
X-581238
X581238
2020 4


PrexasertibLY2606368 2

Puquitinib 1

Pyrotinib 3

QuizartinibAC-010220
AC-220
AC010220
AC220
ASP-2689
3


RabusertibIC-83
LY-2603618
LY2603618
2

RadotinibIY5511 3

RalimetinibLSN-2322600
LSN2322600
LY-2228820
LY2228820
LY22288220
2

RavoxertinibGDC-0994
GDC0994
RG-7842
1


RebastinibDCC-2036
DP-1919
2


RecilisibEx-rad
ON 01210
ON 01210.NA
ON-01210
1

RefametinibBAY 869766
BAY 8697661
BAY-86-9766
BAY-869766
BAY-8697661
BAY86-9766
RDEA 119
RDEA-119
2


RegorafenibStivargaBAY 73-4506
BAY 73-4506 MONOHYDRATE
BAY-73-4506
BAY-734506
2012 4

RemibrutinibLOU064 2

RepotrectinibEXP-6
TPX-0005
TRX-0005
1.5


RezivertinibBPI 7711 3

RibociclibKisqaliLEE-011
LEE-011A
LEE011
LEE011A
NVP-LEE011
2017 4


RigosertibON 01910 3


RilzabrutinibPRN-1008
PRN1008
3

RimacalibSMP-114 2

RineterkibERK-IN-1
LTT-462
LTT462
2

Ripasudil 2

RipretinibQinlockDCC-26182020 4

RitlecitinibPF-06651600
PF06651600
3


Riviciclib 2

RivoceranibAitanApatinib
Albumin paclitaxel
Capecitabine
Carboplatin
Cryoablation
Docetaxel
Egafur
Emozolomide
H20140103
NAVELBINE+AITAN
NO.
Oxaliplatin
Paclitaxol
Pemetrexed
SHR-1210
VP-16
Xelox
YN968D1
2014 4

RoblitinibFGF-401
FGF401
NVP-FGF401
2


RociletinibAVL-301
CNX-419
CO-1686
CS-1631
3


RogaratinibBAY-1163877 2

Roniciclib 2


RopsacitinibPF-06826647 2


RuboxistaurinArxxantLY-333531 3


RuxolitinibJakafi
Jakavi
Opzelura
INC-424
INC424
INCB-018424
INCB-18424
INCB018424
2011 4


SamotolisibLY 3023414
LY-3023414
LY3023414
2

SamuraciclibCT7001
ICEC-0942
ICEC0942
PPDA-001
1


SapanisertibINK-128
INK128
MLN-0128
MLN0128
TAK-228
2


SapitinibAZD-8931
AZD8931
2

SaracatinibAZ-10353926
AZD-0530
AZD0530
3


SavolitinibOrpathysAZD-6094
AZD6094
HMPL-504
Volitinib
2021 (NMPA) 4


Selatinib 1

SeletalisibUCB-5857
UCB5857
2

SeliciclibAL-39256
CYC-202
NSC-701554
2


SelitrectinibLOXO-195 1.5

SelonsertibGS-4997 3


SelpercatinibRetevmoLOXO-292
LY-3527723
LY3527723
WHO 10967
2020 4


SelumetinibKoselugoARRY-142886
ARRY-886
AZD-6244
AZD6244
2020 4


SemaxanibNSC-696819
Semaxinib
SU-5416
SU005416
SU5416
3


SerabelisibAGN-PC-0DB6FL
INK1117
MLN-1117
MLN1117
TAK-117
2

SeralutinibGB-002
Gb002
PK-10571
PK10571
2

SilmitasertibCX 4945
CX-4945
CX4945
2


SimotinibSIM-6802 3

SimurosertibTAK-931 2

SitravatinibMG-516
MG-91516
MGCD-516
MGCD516
3

SolcitinibG-154578
G154578
GLPG-0778
GLPG-0788
GLPG0778
GSK-2586184
GSK-2586184A
GSK2586184A
2

SonolisibPX-866 2

SorafenibNexavarBAY 43-9006
BAY-43-9006
2005 4


SotrastaurinAEB-071
AEB071
NVP-AEB071
2


SotuletinibBLZ 945
BLZ-945
BLZ945
2

SovesudilAMA 0076
AMA-0076
AMA0076
PHP-201
PHP201
3

SpebrutinibAVL-292
CC-292
2


SunitinibSutentSU-011248
SU-11248
SU011248
2006 4


SurufatinibHMPL-012
Sulfatinib
KDR-IN-1
3

TafetinibSIM 010603
SIM-010603
1

TaletrectinibDS-6051b
AB-106
2

TalmapimodSCIO 469
SCIO-469
2


TamatinibR-406 2


TandutinibCT 53518
CT-53518
CT53518
MLN-0518
MLN-518
2

TanzisertibCC-930
JNK 930
JNK-930
2


TarloxotinibPR610
TH-4000
2

TaselisibGDC-0032
RG-7604
3


TasurgratinibE-7090
E7090
2

TelatinibBAY 57-9352
BAY-57-9352
BAY-579352
2

Tenalisib 2

TepotinibTepmetkoEMD 1214063
EMD-1214063
EMD1214063
MSC-2156119
MSC-2156119J
MSC2156119
2021 4


TesevatinibEXEL-7647
KD-019
KD-020
KD019
XL-647
XL647
3

TheliatinibHMPL-309
Xiliertinib
1

TideglusibNP031112 2

TilpisertibGS-4875
GS 4875
GS4875
2

TirabrutinibVelexbruGS-4059
ONO-4059
2


TirbanibulinKX2-391
KX-01
3


TivantinibARQ 197
ARQ-197
3



TivozanibFotivdaASP-4130
AV-951
KIL-8951
KIL8951
KRN-951
2021 4


TizaterkibATG-017
AZD0364
1


ToceranibPHA-291639 0


TofacitinibXeljanz550
CP 690550
CP- 690 550
CP-690
CP-690,550
CP-690-550
CP-690550
CP690,550
CP690550
Tasocitinib
2012 4


TolebrutinibBTK'168
PRN-2246
PRN2246
SAR442168
3

TolimidoneCP-26154
MLR-1023
2

TomivosertibEFT 508
EFT-508
EFT508
2


TozasertibMK-045
MK-0457
VX-68
VX-680
2


TrametinibMekinistGSK-1120212
GSK1120212
JTP 74057
JTP-74057
TMT-212
TMT212
2013 4


TrilaciclibCoselaG1T282021 4

TucatinibTukysaARRY-380
ONT-380
2020 4

TuxobertinibBDTX-189
BDTX189
1

UlixertinibBVD-523
Bvd-erk
VRT-752271
2


UmbralisibUkoniqRP-5264
RP5264
TGR 1202
TGR-1202
2021 4

UpadacitinibRinvoqABT-4942019 4

UprosertibGSK-2141795
GSK-2141795C
GSK2141795
GSK2141795C
2

UzansertibINCB053914
INCB-053914
2

VactosertibTEW 7197
TEW-7197
2

VandetanibCaprelsa
Zactima
GNF-PF-2188
ZD-64
ZD-6474
ZD6474
2011 4


VarlitinibAR-00334543
ARRY-334543
ARRY-543
ASLAN-001
ASLAN001
2.5

VatalanibBAY-86-5127
CGP-79787
K-222584
NVP-PTK787
PTK-787
PTK787
ZK-222584
3

VebreltinibAPL-101
CBI-3103
PLB-1001
1

VecabrutinibBIIB-062
BSK-4841
FP-0182
FP0182
SNS-062
1

VemurafenibZelborafPLX-4032
PLX4032
RG 7204
RG-7204
RO 5185426
RO-51-85426
RO-5185426
2011 4


VerosudilAR-12286 2

VevorisertibARQ 751 1

VimseltinibDCC-3014
DCC3014
2

VistusertibAZD-2014
AZD2014
2

VodobatinibK0706 2

VolasertibBI 6727
BI-6727
3


VorolanibX-82 2

Voruciclib 2

VoxtalisibSAR-245409
SAR245409
XL-765
2

XiliertinibHMPL-309
HMPL309
Theliatinib
1

ZabedosertibBAY-1834845
BAY1834845
1

ZandelisibACC-524
ME-401
PW-143
PWT-143
PWT143
ME401
3

ZanubrutinibBrukinsaBGB-31112019 4


Zeteletinib 1

ZimlovisertibPF-06650833 2


ZoligratinibDEBIO-1347
DEBIO1347
1

ZorifertinibAZD-3759
AZD3759
AZD 3759
2

ZotiraciclibEX45
SB-1317
SB1317
TG-02
TG02
1