Drugs and clinical candidates

This overview is powered by in-house annotations and is complemented with data from the PKIDB1,2 (Bonnet lab).
INN / Name Brand name Synonyms Approval year Phase KLIFS links Structures
BAY1217389BAY-1217389
BAY 1217389
1


M4205 1

PF-07104091 2

KB-0742 1

LY3295668AK-01 1

JNJ-67856633JNJ67856633
JNJ 67856633
2

GDC-0134 1

AZD4547AZD-4547
KB-74810
2


BTX-A51 1

AR-13503Metabolite netarsudil 1

LY-3200882 2

PF-06952229 1

AZD-8154AZD8154
AZD 8154
2


PHA-793887 1


SGX-523 1


OSI-930 1

CC-401 1

TAK-285 1


RO4987655CH4987655 1


BMS-599626AC480 1

AZD-8055 1

MK-2461MK2461 2

PF-04217903 1


AZD-7762 1


AZD1208 1

JNJ-38877605 1

Palomid529 1

TAK-593 1

MK-8033 1

GDC-0349 1

TAK-960 1


CP-547632 2


PND-1186VS-4718
SR-2516
1

SAR-260301SAR260301 1


AZD8330ARRY-424704
ARRY-704
1

BGT226NVP-BGT226
BGT-226
BGT 226
2

MRX-2843UNC2371 1

VS-5584SB2343 1

TAK-901 1

GSK1059615 1

RGB-286638 1

XL228 1

JI-101 2

XL019 1


ASP3026 1


CC-115 1

ARRY-382 2

BAY1082439 1

PIM447LGH447 1


AMG-337 2


PF-06459988 2


AZD-8835AZD8835
AZD 8835
1

ODM-203 1

ASP4132 1

CEP-37440 1

TP-3654 1

EOC317ACTB-1003 1

TG 100801TG100801 2

PRN1371 1


FN-1501 1

BFH772 2

MK-8353SCH900353 1


SCR-1481B1BMS-817378 1

AMG319 2


AT7519AT7519M 1


SAR125844 2


AZD4573 2


ASP5878 1

ENMD-2076 2


GSK-690693GSK690693 1


AMG-208 2


BI 2536BI-2536
BI2536
2


AEE788AEE 788
NVP-AEE788
2


LY3214996 2

BAY1125976BAY-1125976 1

M2698MSC2363318A 1


CEP-40783RXDX-106 1

AV-412MP412 1

OMO-1OMO1
JNJ38877618
JNJ-38877618
1

TAS0728 2

GDC-0575ARRY-575
RG7741
1

KO-947 1

CC-90003 1

CG-806 2

T-1101TAI-95 1

IM156HL156A
HL271
1

FF10101FF-10101-01 1

GLPG0259GLPG-0259
GTPL9848
2

GSK2982772GSK772 2


GSK2983559 1

GSK3145095GSK095 2

BIIB-091BIIB091 1


ESK981CEP 11981
CEP11981
1

LY3405105 1

AUM-001ETC-1907206
ETC-206
2

Debio0123Debio 0123
Debio-01230
1

SY-5609SY-0005609
CDK7-IN-3
1

AS-0141 1

CC-90005 1

ASTX029ASTX-029 1.5

TAK-020 1

RVU120SEL120
SEL120-34A
1.5

CC-90001CC 90001 2

BMS-387032BMS 387032
BMS387032
SNS 032
SNS-032
1


CHIR-265CHIR 265
CHIR265
RAF 265
RAF-265
RAF265
2


CI-1040CI 1040
CI1040
PD-184352
PD184352
2

GSK-461364AGSK 461364
GSK-461364
GSK461364
GSK461364A
1

KW-2449KW 2449 1

SU-14813SU014813
SU14813
1

TG-100-115TG 100-115
TG 100115
TG100-115
1.5


VX-702I14-1965
VX 702
VX702
2

AZD6703AZ 12012199
AZ-12012199
AZ12012199
AZD 6703
AZD-6703
1


PH-797804 2


BMS-582949BMS 582949
BMS582949
PS 540446
PS-540446
PS540446
2


BMS-690514BMS 690514
BMS690514
2

CP-724714CP 724714
CP724714
2

7-hydroxystaurosporineKRX-0601
KRX0601
UCN 01
UCN-01
2


PF-04691502PF 04691502
PF04691502
2


MK-8776MK 8776
SCH-900776
SCH 900776
2

MK-2206MK 2206 2

AT-9283AT 9283
AT9283
2

BMS-754807BMS 754807
BMS754807
2


BMS-777607BMS 777607
BMS777607
2


BMS-911543BMS 911543
BMS911543
1.5


LY2090314LY-2090314 1.5

ZSTK474TCMDC-137004
ZSTK 474
ZSTK-474
1.5


AKN-028AKN 028
AKN028
1.5

PF-4708671PF4708671 0


GSK269962AGSK-269962A
GSK269962
0

BI-D1870 0

GSK650394GSK-650394 0


KU-60019 0

VE-821VE 821 0

PF-477736PF 477736
PF-00477736
1

AZD6482AZD 6482
AZD-6482
1


AMG-900AMG 900
AMG900
1

MK-5108MK5108
VX-689
VX689
1


P505-15BIIB057
PRT-062607
PRT062607
0


LY2874455LY-2874455 1


XL413BMS-863233
BMS863233
XL-413
1


CEP-1347CEP 1347
CEP1347
KT-7515
KT7515
3

LY2584702LY 2584702
LY-2584702
1

GSK1070916GSK-1070916 1

AZD5438AZD 5438
AZD-5438
1


AZD8186AZD 8186
AZD-8186
1

SGI-1776SGI 1776
SGI1776
1

CUDC-101CUDC101 1

SAR407899HY-15687A
SAR-407899
2

PF-3758309PF-03758309
PF3758309
1


LY3009120LY-3009120 1


PLX8394PLX 8394
PLX-8394
1.5

AC430AC-430 1

GDC-0834GDC 0834 1


PF-06263276PF 0626327
PF0626327
1


CBS-3595 1

BMS-986142BMS986142 2


TAK-733TAK733 1


AZD0156 1

KX2-361KX-02
KX2 361
KX2361
1

GSK2646264 1

RV1729RV-1729 1

RV6153RV-6153 1

GR-389988GR389988
GZ389988
GZ389988A
2

RG-1530R-1530
R1530
RG1530
1

MW150MW-150
MW01-18-150SRM
1


AZD7648AZD-7648 1.5


GSK2292767GSK-2292767 1


ARRY-371797ARRY-797
ARRY371797
ARRY797
2

BIIB068BIIB-068 1

AZD1390 1

LUT014LUT-014 2

MLI-2MLi-2 1


AZD7624AZD-7624 2

AZD4604AZD-4604
Jak1-IN-7
1

BLU-945BLU 945 1

MEN1703SEL24 1.5

VIC 1911VIC-1911
TAS-119
TAS-2104
1.5

RP-6306 1

MAP855 0

NVP-CLR457CLR457 1

IOA-244 1

APG-2449APG 2449 1

XL999 1

BMS-986176BMS986176
LX-9211
LX9211
2

KT-413 1

TL-895TL895 2

AEW-541AEW 541
Aew-541
NVP-AEW541
NVP-AEW 541
1

AG-13958AG 13958 2

AS-602868SPC-839 1

AST-487NVP-AST487
NVP-AST-487
1

AT-13148AT13148 1

AZD-1480AZD1480
AZD 1480
2


CEP-5214 1

CYC-116CYC 116
CYC-116
1


E-6201E6201
ER-806201
2


GS-9901GS 9901 1


GSK-2636771GSK2636771 2

GSK-3179106GSK3179106 1

H3B-6527H3b 6527
H3b-6527
1

JNJ-49095397RV568
RV-568
2

KRN-633K00589A
KRN633
KRN-633
1

LX-7101LX7101 1

MK-0941 2

MLN-8054MLN 8054
MLN8054
1


PD-0166285PD-0166285
TCMDC-140940
TCMDC-140940
1


PF-00562271Pf-00562271
PF 562271
PF-562271
1


PF-03715455PF 03715455 2


PF-06273340PF06273340 1


PKI-179PKI 179 1

R-1487 1


R-343 2

RG-547R 547
R-547
RG-547
RO4584820
RO-4584820
2


Senexin BBcd-115
BCD-115
1

SNS-314SNS 314 1


SU-014813SU-14813 2

TAK-715TAK 715
TAK-715
2


XL-281BMS-908662
EXEL-2819
Xl 281
Xl-281
2

Y-39983Y-39983
Y-39983
1

ZD-4190ZD4190 1

CEP-7055CEP7055 1

SU-9516SU9516 1


AZD-1080AZ-11548415
AZD1080
1

AZD-1656AZD1656 2

TOP-1288TOP1288 2

KA 2237KA2237 1

HKI-357HKI357 1

RO-3201195RO3201195 1


AMG-548AMG548 1

GLPG3970 2

TAK-279NDI-034858
NTX-973
2

GSK2256098 2

BI 853520IN10018 1.5

CC-99677 1

CHF-6297CHI 91040 1.5

GNE-0877DNL201 1

AMP945 1.5

EP0042 1.5

GSK3923868 1

KER-047 1

NXP900eCF506 1


JNJ-64264681JNJ64264681 1

SIR1-365SIR1365 1

CT-1578CT 1578
SB 1578
1

XL-418 1

XP-102 1.5


AbemaciclibVerzenio
Verzenios
LY-2835219
LY2835219
2017 4


AbivertinibA610
AC-0010
AC0010
ACEA100610
Avitinib
EX-ACEA0010
3

AbrocitinibCibinqoPF-049658422022 4


AcalabrutinibCalquenceACP-1962017 4


AcalisibCAL-120
CAL120
GS-9820
GS9820
2

AcrizanibLHA510 2

AcumapimodBCT 197
BCT-197
BCT197
2

AdavosertibAZD 1775
AZD-1775
AZD1775
MK-1775
MK1775
2


AfatinibGilotrif
Giotrif
BIBW-2992
BIBW2992
2013 4



AfuresertibASB-183
ASB183
GSK-2110183
GSK-2110183C
GSK2110183
GSK2110183C
LAE002
2

AgerafenibAB-024
AC-013773
CEP-32496
RXDX 105
RXDX-105
1

AlectinibAlecensaAF-802
AF802
CH-5424802
CH5424802
RO-5424802
RO5424802
2015 4


AlisertibMLN 8237
MLN-8237
MLN8237
3


AllitinibALL-3
AST-1306
2

Alofanib 1

AlpelisibPiqray
Vijoice
BYL-719
NVP-BYL719
2019 4


AltiratinibDCC-2701
DP-5164
1


AlvocidibFlavopiridol
HL 275
HL-275
HMR 1275
HMR-1275
L 86 8275
L-868275
L86-8275
MDL 107,826A
MDL-107826A
NSC-649890
TP-1287 (prodrug form)
3


AmcasertibBBI-503
BBI503
2

AmdizalisibHMPL-689 2

AmuvatinibHPK 56
HPK-56
HPK56
MP 470
MP-470
MP470
2

AnsornitinibANG-3070 2

ApilimodLAM-002A
LAM002A
STA 5326
STA-5326
STA5326
2

ApitolisibG-038390
G-038390.1
GDC-0980
GDC-0980.1
RG-7422
RG7422
2


AsciminibScemblixABL-001
ABL001
ABL001-NX
NVP-ABL001
2021 4


AsnuciclibSunaciclib
CDKI-73
1

AtuveciclibBAY 1143572
BAY-1143572
BAY1143572
1

AtuzabrutinibPRN473
SAR 444727
2

AumolertinibAmeileHS-10296
Almonertinib
2020 (NMPA) 4

AvapritinibAyvakit70C366
BLU-285
C-366
X-720776
X720776
2020 4


AvotaciclibBEY 1107
BEY1107
BEY-1107
1

AvutometinibVS-6766
RG 7304
CKI27
CH5126766
RO5126766
1


AxitinibInlytaAG-013736
AG-13736
2012 4


AzenosertibZN-c3
ZN c3
2

BafetinibCNS-9
INNO-406
NS-187
2


BalamapimodMKI-833 1

BarasertibAZD 1152
AZD-1152
AZD1152
3

BaricitinibOlumiantINCB-028050
INCB-28050
INCB028050
LY-3009104
LY3009104
2017 4


BefotertinibD-0316
D 0316
D0316
2

BelizatinibTSR-011
TSR011
2


BelumosudilRezurockKD025
SLx2119
2021 4


BelvarafenibHM95573
GDC-5573
2


BemcentinibBGB 324
BGB-324
BGB324
CS-1046
HY-15150
KB-80319
QC-11751
R 428
R-428
R428
SYN-1131
SYN1131
W-5845
2


BentamapimodAS-602801
PGL-5001
2

BerzosertibM-6620
M6620
VE-822
VX-970
VX970
2

BezuclastinibPLX9486
CGT 9486
2

BimiralisibNC-B5
NCB5
PI3K-IN-2
PQR-309
PQR309
2


BinimetinibMektoviARRY 438162
ARRY-162
ARRY-438162
MEK-162
MEK162
NVP-MEK162
2018 4


BoditrectinibAUM601
AUM-601
CHC 2014
CHC2014
HL5101
HL 5101
NOV-1601
NOV 1601
1

BosutinibBosulifBosutinib monohydrate
SK-606
SKI-606
2012 4


BranebrutinibBMS-986195 2


BrepocitinibPF-06700841 3


BriciclibON 014185 1

BrigatinibAlunbrigAP-26113
AP26113
2017 4


BrivanibBMS-540215 3

Brivanib alaninateBMS-582664
BMS-582664-02
Brivanib l-alanine ester
3

BuparlisibBKM-120
BKM-120NX
BKM120-NX
NVP-BKM-120
NVP-BKM120
3


CabozantinibCabometyx
Cometriq
BMS-907351
XL-184
XL184
2012 4

CamonsertibRP-3500
RP3500
2

CanertinibCI-1033 3

CapivasertibTruqapAZC5363
AZD 5363
AZD-5363
AZD5363
2023 4


CapmatinibTabrectaINC-280
INC280
INCB-28060
NVP-INC280
NVP-INC280-NX
NYP-INC280-NX
2020 4

CatequentinibFOCUS VAL3818
Anlotinib
Altn
2018 (NMPA) 4

CediranibRecentinAZD-2171
AZD2171
ZD-2171
3

CenisertibAS-703569
R-763
1

CeralasertibAZD6738 3

Cerdulatinib 2.5


CeritinibZykadiaLDK-378
LDK378
NVP-LDK-378-NX
NVP-LDK378-NX
2014 4


CevidoplenibSKI-O-703 2

CirtuvivintSM08502 1

CobimetinibCotellicGDC-0623
GDC-0973
RG 7420
RG-7420
RG-7421
RG7420
XL-518
2015 4


ConteltinibCT-707
CT707
1

CopanlisibAliqopaBAY 80-6946
BAY-80-6946
BAY80-6946
2017 4


Cotosudil 0

CrenolanibARO 002
ARO-002
CP 868596
CP-868,596
CP-868596
3


CrizotinibXalkoriPF-02341066
PF-2341066
2011 4


DabrafenibTafinlarGSK-2118436
GSK-2118436A
GSK2118436
GSK2118436A
2013 4


DacomitinibVizimproDacomitinib hydrate
PF-00299804
2018 4


DactolisibBEZ-235
BEZ235
NVP-BEZ235
NVP-BEZ235-NX
3

DalpiciclibSHR 6390
SHR-6390
SHR6390
3

DanusertibPHA-739358 2


DarovasertibIDE-196
IDE196
LXS-196
LXS196
2

DasatinibDasatinib
Sprycel
BMS-354825
BMS-354825 HYDRATE
BMS-354825-03
Dasatinib hydrate
Dasatinib monohydrate
2006 4


DecernotinibAdelatinib
VRT-831509
VX-509
2


DefactinibPF-04554878
VS-6063
2


DefosbarasertibBarasertib-hqpa
AZD-1152HQPA
AZD-2811
AZD2811
AZD 2811
2

DelgocitinibCorectimJTE-052
JTE-052A
LEO 124249
LEO-124249
LEO 124249A
LEO-124249A
2020 (PMDA) 4


DenfivontinibG-749
G-801
SKI-G-801
1

DerazantinibARQ 087
ARQ-087
ARQ087
2

DeucravacitinibSotyktuBMS-986165
BMS986165
2022 4


DeuruxolitinibLeqselviCTP-543
CTP543
D8-ruxolitinib
2024 4

DezapelisibINCB040093 0

DilmapimodGW-681323
SB-681323
SB681323
2

DinaciclibMK-7965
SCH 727965
SCH-727965
3


DonafenibZepsunSorafenib (D3)
CM-4307
2021 (NMPA) 4

DoramapimodBIRB 796 BS
BIRB-796
BIRB-796 BS
2


DorzagliatinHMS-5552
HMS5552
RO-5305552
RO5305552
Sinogliatin
3

DovitinibCHIR-258
GFKI-258
NVP-TKI258
TKI-258
3


DubermatinibHCL-2084
TP 0903
TP-0903
TP0903
1.5

DuvelisibCopiktraINK-1147
INK-1197
IPI-145
2018 4

EbvaciclibPF-06873600 2


EclitasertibDNL758
SAR443122
2

EdecesertibGS-5718
GS 5718
2

EdicotinibJNJ-40346527 2

EdralbrutinibSHR-1459
SHR1459
TG-1701
TG1701
1

EganelisibIPI-549
IPI549
2


ElimusertibBAY 1895344
BAY-1895344
BAY1895344
1.5

Elraglusib9-ING-41 2

ElsubrutinibABBV 105
ABBV-105
2

ElzovantinibTPX-0022
TPX0022
CSF1R-IN-2
1

EmavusertibCA-4948
AU-4948
AU4948
CA4948
2


Empesertib(-)-BAY-1161909
BAY 1161909
MPS1-IN-5
1


EmprumapimodPF-06802861
PF-07265803
0

EnbezotinibTPX-0046 1.5

EncorafenibBraftoviLGX-818
NVP-LGX-818-NXA
NVP-LGX818
NVP-LGX818-NXA
2018 4

EnitociclibVIP152
BAY-1251152
1

EnsartinibX-396 3

EntospletinibGS-9973
SYK INHIBITOR GS-9973
3


EntrectinibRozlytrekNMS-E628
RXDX-101
2019 4


EnzastaurinKinenzaLY-317615
LY317615
DB102
DB-102
AR101
3

EpertinibS-222611 1

EpitinibHMPL-813 1

ErdafitinibBalversaJNJ-427564932019 4


ErlotinibTarcevaCP-358,774
CP-358774
CP-35877401
OSI-774
R-1415
RG-1415
RO-508231
2004 4


EvobrutinibM-2951 3


ExarafenibKIN-2787 1


FadraciclibCYC-065
CYC065
1.5

FalnidamolBIBX 1382 1

FamitinibSHR-1020 3

FasudilErilAT 877
AT-877
HA 1077
HA-1077
ZK-258594
1995 (PMDA), 2010 (NMPA) 4


FedratinibInrebicSAR-302503
SAR302503
TG-101348
TG101348
2019 4


FenebrutinibG-02599853
G02599853
GDC-0853
RG-7845
RG7845
RO-7010939
RO7010939
3


FidrisertibIPN60130
BLU-782
1

FilgotinibJyselecaG-146034
G146034
GLPG-0634
GLPG0634
GS-6034
2020 (EMA, PMDA) 4


FimepinostatCUDC 907
CUDC-907
2

FisogatinibBLU-554
BLU 554
BLU111362
2


Flonoltinib 1


FlumbatinibXinfuFlumatinib
HH-GV678
HHGV-678
2019 (NMPA) 4

ForetinibEXEL-2880
GSK-089
GSK-1363089
GSK-1363089G
GSK089
GSK1363089G
XL-880
XL880
2


Fosifidancitinib I-538 ?

FoslinanibCVM-1118
TRX 818
TRX-818
2

FostamatinibTavalisseR-788
R-935788
R788
R935788
2018 4


FruquintinibFruzaqla
Elunate
HMP-013
HMPL-013
2018 (NMPA) 4

FurmonertinibIvesaAlflutinib
AST-2818
AST2818
2021 (NMPA) 4

FutibatinibLytgobi2022 4


GalunisertibLY-2157299
LY2157299
2

GandotinibLY-2784544
LY2784544
2


GartisertibM-4344
M4344
VX-803
VX803
1

GedatolisibPF-05212384
PKI-587
2


GefitinibIressaZD-1839
ZD1839
2003 4


GilteritinibXospataASP-2215
ASP2215
2018 4


GlesatinibMG-90265
MG-90265X
MG90265
MG90265GLY
MG90265H9
MG90265X
MGCD-265
MGCD265
2

GolidocitinibDZD4205
AZD-4205
DZD 4205
AZD4205
1/2

GolvatinibE-7050
E7050
2


GumarontinibGlumetinib
SCC244
SCC-244
1

GunagratinibICP-192 2

GusacitinibASN-002
ASN002
EN-3351
EN3351
2

Henatinib 1

IbcasertibChiauranib
CS-2164
CS2164
3

IbrutinibImbruvicaCRA-032765
PC-32765
PCI 32765
PCI-32765
PCI-32765-00
2013 4



IcotinibConmanaBPI-2009H2011 (NMPA) 4

IdelalisibZydeligCAL-101
GS-1101
GS-11CAL-101
2014 4


IfidancitinibA 301
A-301
A301
R2010
2

IlginatinibNS-018 2

IlorasertibA-968660
A-968660.0
ABBOTT-968660
ABT-348
ABT-348, A-968660
2

IlunocitinibLY-3411067
LY3411067
Veterinary development

ImatinibGleevecSTI-5712001 4


InavolisibItovebiGDC-0077
GDC0077
RO7113755
RG6114
2024 4


InfigratinibTruseltiqBGJ-398
BGJ398
MVP-BGJ398
NVP-BGJ398
2021 4


IpatasertibGDC-0068
RG-7440
RG7440
3


ItacitinibINCB-039110
INCB-39110
INCB039110
3


ItacnosertibTP-0184
TP0184
1

IvarmacitinibSHR0302
SHR 0302
3

IzencitinibTD 1473
TD1473
TD-1473
3

IzorlisibMEN1611
CH5132799
CH 5132799
CH-5132799
1


LanraplenibGS-9876 2


LapatinibTykerb
Tyverb
GSK-572016
GW-2016
GW-572016
GW-572016X
GW572016
2007 4


Larotinib 1

LarotrectinibVitrakviARRY-470
BAY-2757556
BAY2757556
LOXO-101
2018 4

LazertinibLeclaza
Lazcluze
GNS-1480
GNS1480
JNJ-73841937
YH-25448
YH25448
C-18112003-G
2021 (MFDS) 4

LeniolisibJoenjaCDZ173-NX2023 4


LenvatinibKisplyx
Lenvima
E-7080
ER-203492-00
2015 4


LerociclibG1T38 3

LestaurtinibA-154475
A-154475.0
CEP-701
KT-555
KT-5555
KT5555
SP-924
SP924
SPM-924
3


LifirafenibBGB 283
BGB-283
1


LinifanibA-741439
ABT-869
AL-39324
RG-3635
3

LinperlisibYY-20394
YY20394
3

LinsitinibASP-7487
OSI-906
OSI-906AA
3

LirafugratinibRLY-4008 2

LisaftoclaxAPG-2575
APG 2575
1.5

LorecivivintAdavivint
SM0-4690
SM04690
3

LorlatinibLorbrena
Lorviqua
PF-064639222018 4


Lorpucitinib 1

LosmapimodFTX-1821
FTX1821
Gsk-ahab
Gskahab
GW-856553
GW-856553X
GW856553X
3

LucitanibAL-3810
CO-3810
E-3810
S 80881
S-80881
2


LuvixasertibCFI-402257
CFI402257
1.5

LuxeptinibCG026806
CG-806
1

MaribavirLivtencityTAK-620
1263W94
2021 4

MasitinibKinavet
Masivet
AB-10102008 (EMA-veterinary);2010-15 (FDA-veterinary) 3


MavelertinibPF-06747775 2


MerestinibLY-2801653
LY2801653
2


MevociclibSY-1365
SY1365
1

MidostaurinRydaptCGP 41251
CGP-41251
NVP-PKC412
PKC 412
PKC-412
2017 4


MilciclibPHA 848125
PHA-848125
2


MiransertibARQ 092
ARQ-092
2


MirdametinibPD 0325901
PD-0325901
PD0325901
2


MivavotinibTAK-659
CB-659
2


MobocertinibExkivityTAK788
TAK-788
AP32788
2021 4

MomelotinibOjjaaraCYT-0387
CYT-11387
CYT-387
CYT387
GS-0387
2023 4


MotesanibAMG 706
AMG-706
3


MubritinibTAK-165 1

NaporafenibLXH 254
LXH-254
LXH254
PAN-RAF INHIBITOR LXH254
2


NaquotinibASP-8273
ASP8273
3


NarazaciclibON123300
ON 123300
2

NazartinibEGF-816
EGF816
NVP-EGF816-NX
3


Neflamapimod745
VD-31
VD-31,745
VD-31745
VRT-031745
VX-745
2


NemiralisibGSK-2269557
GSK-2269557A
GSK2269557A
2


NemtabrutinibARQ 531
K-1026
2

NeratinibNerlynxCDP-820
HKI-272
WAY-179272
2017 4


NetarsudilRhopressaAR-133242017 4

NezulcitinibTD-0903
TD 0903
TD0903
2

NilotinibTasignaAMN 107
AMN-107
AMN107
2007 4


Ningetinib 1.5

NintedanibOfev
Vargatef
BIBF 1120
BIBF-1120
BIBF1120
Intedanib
2014 4


OcifisertibCFI-400945
CFI400945
CFI 400945
1

OclacitinibJaki
PF-03394197
0

OlafertinibCK101
CK‐101
RX-518
RX518
1

OlmutinibOlitaBI 1482694
BI-1482694
HM-61713
HM61713
2016 (MFDS) 4

OlverembatinibNailikeHQP1351 GZD8242021 (NMPA) 4


OmipalisibGSK-2126458
GSK2126458
1


OnatasertibATG-008
CC 223
CC-223
2

OnvansertibNMS-1286937
NMS-P937
PCM-075
2


OpaganibABC 294640
ABC-294640
2.5

OrantinibNSC-702827
SU-6668
TSU-68
3


OrelabrutinibHibrukaICP022
ICP-022
2020 (NMPA) 4

OsimertinibTagrissoAZD-9291
AZD9291
Mereletinib
2015 4



PacritinibVonjoONX-0803
SB-1518
SB1518
2022 4


PadnarsertibKPT-9274
KPT9274
PAK4-IN-1
1


PalbociclibIbrancePD-03329912015 4


PaltimatrectinibPBI-200 1.5

PamapimodR-1503
R1503
RO 4402257
RO-4402257
2


PamufetinibTAS-115 2

Panulisib 1

ParsaclisibINCB-050465
INCB050465
3

PaxalisibGDC-0084
GDC0084
G02441729
G-02441729
RG-7666
2

PazopanibVotrientGW7860342009 4

PeficitinibSmyrafASP-015K
ASP015K
JNJ-54781532
2021 (PMDA) 4


PegcantratinibCT327
CT-327
SNA-120
2

PelitinibEKB-569
WAY-EKB-569
2


PemigatinibPemazyreINCB0548282020 4


PeposertibM-3814
Nedisertib
M3814
MSC 2490484A
MSC-2490484A
MSC2490484A
1.5


PexidartinibTuralioCML-261
PLX-3397
PLX3397
2019 4


Pexmetinib 1

PictilisibCDC-0941
GDC 0941
GDC-0941
RG-7321
2


PifusertibTAS117
TAS-117
2

PilaralisibSAR-245408
SAR245408
XL-147
XL147
2

PimasertibAS 703026
AS-703026
AS703026
EMD 1036239
EMD-1036239
G-02443714
MSC-1936369A
MSC-1936369B
MSC1936369A
AS703026
EMD 1036239
2


PirotinibKBP-5209 2

PirtobrutinibJaypircaLOXO-305
RXC-005
LY-3527727
LY3527727
2023 4


PlogosertibCYC140 1.5

PonatinibIclusigAP-24534
AP24534
2012 4


PoseltinibHM71224
LY3337641
2

PovorcitinibINCB 54707
INCB054707
2

PoziotinibHM 781-36
HM 781-36B
HM-781-36
HM-781-36B
NOV-120101
3

PralsetinibGavretoBLU-123244
BLU-667
BLU123244
X-581238
X581238
2020 4


PrexasertibLY2606368 2

Puquitinib 1

PyrotinibIreneSHR-12582020 (NMPA) 4

QuizartinibVanflytaAC-010220
AC-220
AC010220
AC220
ASP-2689
2023 4


RabusertibIC-83
LY-2603618
LY2603618
2

RadotinibSupectIY55112015 (MFDS) 4

RalimetinibLSN-2322600
LSN2322600
LY-2228820
LY2228820
LY22288220
2


RavoxertinibGDC-0994
GDC0994
RG-7842
1


RebastinibDCC-2036
DP-1919
2


RecilisibEx-rad
ON 01210
ON 01210.NA
ON-01210
1

RefametinibBAY 869766
BAY 8697661
BAY-86-9766
BAY-869766
BAY-8697661
BAY86-9766
RDEA 119
RDEA-119
2


RegorafenibStivargaBAY 73-4506
BAY 73-4506 MONOHYDRATE
BAY-73-4506
BAY-734506
2012 4

RemibrutinibLOU064 2

RepotrectinibAugtyroEXP-6
TPX-0005
TRX-0005
2023 4


RezivertinibBPI 7711 3

RibociclibKisqaliLEE-011
LEE-011A
LEE011
LEE011A
NVP-LEE011
2017 4


RigosertibON 01910 3


RilzabrutinibPRN-1008
PRN1008
3


RimacalibSMP-114 2

RineterkibERK-IN-1
LTT-462
LTT462
2

RipasudilGlanatecK-1152014 (PMDA) 4

RipretinibQinlockDCC-26182020 4

RisvodetinibIkT-148009 2

RitlecitinibLitfuloPF-06651600
PF06651600
2023 4


Riviciclib 2

RivoceranibAitanApatinib
Albumin paclitaxel
Capecitabine
Carboplatin
Cryoablation
Docetaxel
Egafur
Emozolomide
H20140103
NAVELBINE+AITAN
NO.
Oxaliplatin
Paclitaxol
Pemetrexed
SHR-1210
VP-16
Xelox
YN968D1
2014 (NMPA) 4

RoblitinibFGF-401
FGF401
NVP-FGF401
2


RociletinibAVL-301
CNX-419
CO-1686
CS-1631
3


RogaratinibBAY-1163877 2

Roniciclib 2


RopsacitinibPF-06826647 2


RuboxistaurinArxxantLY-333531 3


RuserontinibSKLB-1028
SKLB1028
3


RuxolitinibJakafi
Jakavi
Opzelura
INC-424
INC424
INCB-018424
INCB-18424
INCB018424
2011 4


SamotolisibLY 3023414
LY-3023414
LY3023414
2

SamuraciclibCT7001
ICEC-0942
ICEC0942
PPDA-001
1


SapanisertibINK-128
INK128
MLN-0128
MLN0128
TAK-228
CB-228
2


SapitinibAZD-8931
AZD8931
2

SaracatinibAZ-10353926
AZD-0530
AZD0530
3


SavolitinibOrpathysAZD-6094
AZD6094
HMPL-504
Volitinib
2021 (NMPA) 4


Selatinib 1

SeletalisibUCB-5857
UCB5857
2

SeliciclibAL-39256
CYC-202
NSC-701554
2


SelitrectinibLOXO-195 1.5

SelonsertibGS-4997 3


SelpercatinibRetevmoLOXO-292
LY-3527723
LY3527723
WHO 10967
2020 4


SelumetinibKoselugoARRY-142886
ARRY-886
AZD-6244
AZD6244
2020 4


SemaxanibNSC-696819
Semaxinib
SU-5416
SU005416
SU5416
3


SerabelisibAGN-PC-0DB6FL
INK1117
MLN-1117
MLN1117
TAK-117
2

SeralutinibGB-002
Gb002
PK-10571
PK10571
2

SilmitasertibCX 4945
CX-4945
CX4945
2


SimotinibXimotiniSIM-68022018 (NMPA) 4

SimurosertibTAK-931 2

SitravatinibMG-516
MG-91516
MGCD-516
MGCD516
3

SolcitinibG-154578
G154578
GLPG-0778
GLPG-0788
GLPG0778
GSK-2586184
GSK-2586184A
GSK2586184A
2

SonolisibPX-866 2

SorafenibNexavarBAY 43-9006
BAY-43-9006
2005 4


SotrastaurinAEB-071
AEB071
NVP-AEB071
2


SotuletinibBLZ 945
BLZ-945
BLZ945
2

SovesudilAMA 0076
AMA-0076
AMA0076
PHP-201
PHP201
3

SovleplenibHMPL-523
HMPL523
HMPL 523
3

SpebrutinibAVL-292
CC-292
2


SunitinibSutentSU-011248
SU-11248
SU011248
2006 4


SunvozertinibDZD9008 1.5

SurufatinibSulandaHMPL-012
Sulfatinib
KDR-IN-1
2021 (NMPA) 4

TafetinibSIM 010603
SIM-010603
1

TaletrectinibDS-6051b
AB-106
2

TalmapimodSCIO 469
SCIO-469
2


TamatinibR-406 2


TamnorzatinibONO-7475 2

TandutinibCT 53518
CT-53518
CT53518
MLN-0518
MLN-518
2

TanzisertibCC-930
JNK 930
JNK-930
2


TarloxotinibPR610
TH-4000
2

TaselisibGDC-0032
RG-7604
3


TasurgratinibE-7090
E7090
2

TelatinibBAY 57-9352
BAY-57-9352
BAY-579352
2

Tenalisib 2

TepotinibTepmetkoEMD 1214063
EMD-1214063
EMD1214063
MSC-2156119
MSC-2156119J
MSC2156119
2021 4


TesevatinibEXEL-7647
KD-019
KD-020
KD019
XL-647
XL647
3

TheliatinibHMPL-309
Xiliertinib
1

TideglusibNP031112 2

TilpisertibGS-4875
GS 4875
GS4875
2

TinengotinibTTT00420
TT 00420
TT-00420
1

TinlorafenibARRY-461
ARRY461
PF-07284890
PF07284890
1


TirabrutinibVelexbruGS-4059
ONO-4059
2020 (PMDA) 4


TirbanibulinKX2-391
KX-01
3


TivantinibARQ 197
ARQ-197
3



TivozanibFotivdaASP-4130
AV-951
KIL-8951
KIL8951
KRN-951
2021 4


TizaterkibATG-017
AZD0364
1


ToceranibPalladiaPHA-2916392009 (FDA-Veterinary) 0


TofacitinibXeljanz550
CP 690550
CP- 690 550
CP-690
CP-690,550
CP-690-550
CP-690550
CP690,550
CP690550
Tasocitinib
2012 4


TolebrutinibBTK'168
PRN-2246
PRN2246
SAR442168
3

TolimidoneCP-26154
MLR-1023
2

TomivosertibEFT 508
EFT-508
EFT508
2


TovorafenibDAY101
MLN-2480
MLN2480
TAK580
TAK-580
1

TozasertibMK-045
MK-0457
VX-68
VX-680
2


TrametinibMekinistGSK-1120212
GSK1120212
JTP 74057
JTP-74057
TMT-212
TMT212
2013 4


TrilaciclibCoselaG1T282021 4

TucatinibTukysaARRY-380
ONT-380
2020 4

TunlametinibHL-085
HL085
2

TuspetinibHM43239
HM-43239
1.5

TuvusertibM1774
M-1774
M 1774
2

TuxobertinibBDTX-189
BDTX189
1

UlecaciclibAuceliciclib
AU3-14
1.5

UlixertinibBVD-523
Bvd-erk
VRT-752271
2


UmbralisibUkoniqRP-5264
RP5264
TGR 1202
TGR-1202
2021 4

UnecritinibTQ-B3101 2

UpadacitinibRinvoqABT-4942019 4

UprosertibGSK-2141795
GSK-2141795C
GSK2141795
GSK2141795C
2

UtatrectinibAZD7451
AZ12607092
AZD-7451
1

UzansertibINCB053914
INCB-053914
2

VactosertibTEW 7197
TEW-7197
2

VamotinibPF-114
PF114
1.5

VandetanibCaprelsa
Zactima
GNF-PF-2188
ZD-64
ZD-6474
ZD6474
2011 4


VarlitinibAR-00334543
ARRY-334543
ARRY-543
ASLAN-001
ASLAN001
2.5

VatalanibBAY-86-5127
CGP-79787
K-222584
NVP-PTK787
PTK-787
PTK787
ZK-222584
3

VebreltinibAPL-101
CBI-3103
PLB-1001
1

VecabrutinibBIIB-062
BSK-4841
FP-0182
FP0182
SNS-062
1

VemurafenibZelborafPLX-4032
PLX4032
RG 7204
RG-7204
RO 5185426
RO-51-85426
RO-5185426
2011 4


VepafestinibTAS0953
HM06
1.5

VerosudilAR-12286 2

VevorisertibARQ 751 1

VimseltinibDCC-3014
DCC3014
2

VistusertibAZD-2014
AZD2014
2

VodobatinibK0706 2

VolasertibBI 6727
BI-6727
3


VorolanibEYP-1901
X-82
2

Voruciclib 2

VoxtalisibSAR-245409
SAR245409
XL-765
2

XiliertinibHMPL-309
HMPL309
Theliatinib
1

ZabedosertibBAY-1834845
BAY1834845
1

ZandelisibACC-524
ME-401
PW-143
PWT-143
PWT143
ME401
3

ZanubrutinibBrukinsaBGB-31112019 4


ZanzalintinibXL-091
XL092
1

ZapnometinibATR-002
ATR002
PD-0184264
PD0184264
2

Zeteletinib 1

ZilurgisertibINCB00928 1.5

ZimlovisertibPF-06650833 2


ZipalertinibCLN-081
TAS6417
1/2

ZoligratinibDEBIO-1347
DEBIO1347
1


ZorifertinibAZD-3759
AZD3759
AZD 3759
2

ZotiraciclibEX45
SB-1317
SB1317
TG-02
TG02
1

ZunsemetinibATI-450
ATI450
CDD-450
CDD450
2

ZurletrectinibICP-723 2