| EGFR | EGFR | TK | 4i23 | A | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 870 | 0.48 | |
| AURKA (AurA) | Aur | Other | 2c6e | A | | n-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamide | Human | 1989 | 0.44 | |
| EGFR | EGFR | TK | 4hjo | A | | [6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amine | Human | 835 | 0.57 | |
| EGFR | EGFR | TK | 7a6j | A | B | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14124 | 0.42 | |
| EGFR | EGFR | TK | 4i24 | A | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 831 | 0.48 | |
| CDK2 | CDK | CMGC | 1di8 | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 4577 | 0.47 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe2 | A | B | 5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5519 | 0.41 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe2 | A | A | 5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5508 | 0.41 | |
| EGFR | EGFR | TK | 8f1y | A | | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14940 | 0.42 | |
| EGFR | EGFR | TK | 8f1w | A | | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14944 | 0.42 | |
| AURKA (AurA) | Aur | Other | 2c6e | B | | n-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamide | Human | 2046 | 0.44 | |
| EGFR | EGFR | TK | 1m17 | A | A | [6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amine | Human | 873 | 0.57 | |
| MAPK14 (p38a) | MAPK | CMGC | 1di9 | A | | 4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazoline | Human | 5251 | 0.42 | |
| TTBK1 | TTBK | CK1 | 4btk | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 771 | 0.47 | |
| EGFR | EGFR | TK | 4i24 | B | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 910 | 0.48 | |
| EGFR | EGFR | TK | 1m17 | A | B | [6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amine | Human | 905 | 0.57 | |
| EGFR | EGFR | TK | 7a6j | A | A | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14125 | 0.42 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12049 | 0.47 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12046 | 0.47 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12047 | 0.47 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12048 | 0.47 | |
| RET | Ret | TK | 5amn | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 6412 | 0.47 | |
Match: