| EGFR | EGFR | TK | 7u9a | A | | 4-(5-chloro-4-fluoro-2-hydroxyanilino)-7-methoxyquinazolin-6-ol | Human | 14527 | 0.41 | |
| EGFR | EGFR | TK | 4i23 | A | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 870 | 0.40 | |
| EGFR | EGFR | TK | 7a6j | A | B | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14124 | 0.46 | |
| MERTK (MER) | Axl | TK | 7avy | A | | n-(2-(2-cyclopropylethoxy)pyrimidin-5-yl)-7-methoxy-6-(piperidin-4-ylmethoxy)quinazolin-4-amine | Human | 13369 | 0.47 | |
| EGFR | EGFR | TK | 3ug2 | A | A | gefitinib | Human | 898 | 0.47 | |
| GAK | NAK | Other | 5y80 | A | A | gefitinib | Human | 10329 | 0.47 | |
| GAK | NAK | Other | 5y7z | A | | gefitinib | Human | 10332 | 0.47 | |
| EGFR | EGFR | TK | 4i24 | A | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 831 | 0.40 | |
| CDK2 | CDK | CMGC | 1di8 | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 4577 | 0.41 | |
| GAK | NAK | Other | 5y7z | B | | gefitinib | Human | 10331 | 0.47 | |
| EGFR | EGFR | TK | 8f1w | A | | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14944 | 0.46 | |
| EGFR | EGFR | TK | 8f1y | A | | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14940 | 0.46 | |
| EGFR | EGFR | TK | 3ug2 | A | B | gefitinib | Human | 819 | 0.47 | |
| EGFR | EGFR | TK | 2ito | A | | gefitinib | Human | 783 | 0.47 | |
| EGFR | EGFR | TK | 2itz | A | | gefitinib | Human | 789 | 0.47 | |
| GAK | NAK | Other | 5y80 | A | B | gefitinib | Human | 10330 | 0.47 | |
| EPHB4 (EphB4) | Eph | TK | 2vwu | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin-4-amine | Human | 370 | 0.40 | |
| MAPK14 (p38a) | MAPK | CMGC | 1di9 | A | | 4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazoline | Human | 5251 | 0.42 | |
| KSR2 | RAF | TKL | 5kkr | B | | 6,7-dimethoxy-~{n}-(2-methyl-4-phenoxy-phenyl)quinazolin-4-amine | Human | 7027 | 0.42 | |
| TTBK1 | TTBK | CK1 | 4btk | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 771 | 0.41 | |
| RET | Ret | TK | 2ivu | A | | 4-bromo-2-fluoro-n-[(4e)-6-methoxy-7-[(1-methylpiperidin-4-yl)methoxy]quinazolin-4(1h)-ylidene]aniline | Human | 3364 | 1.00 | |
| EGFR | EGFR | TK | 4i22 | A | | gefitinib | Human | 823 | 0.47 | |
| EGFR | EGFR | TK | 4wkq | A | A | gefitinib | Human | 889 | 0.47 | |
| EGFR | EGFR | TK | 4wkq | A | B | gefitinib | Human | 837 | 0.47 | |
| EGFR | EGFR | TK | 4i24 | B | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 910 | 0.40 | |
| EGFR | EGFR | TK | 2ity | A | | gefitinib | Human | 790 | 0.47 | |
| EGFR | EGFR | TK | 7a6j | A | A | 1-[4-[4-[[3,4-bis(chloranyl)-2-fluoranyl-phenyl]amino]-7-methoxy-quinazolin-6-yl]oxypiperidin-1-yl]propan-1-one | Human | 14125 | 0.46 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12049 | 0.41 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12046 | 0.41 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12047 | 0.41 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12048 | 0.41 | |
| RET | Ret | TK | 5amn | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 6412 | 0.41 | |