| MET | Met | TK | 3dkf | A | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 3030 | 0.46 | |
| MET | Met | TK | 3qti | A | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | 2994 | 0.41 | |
| MET | Met | TK | 3qti | B | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | 3024 | 0.41 | |
| MET | Met | TK | 3dkg | A | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 3019 | 0.46 | |
| MET | Met | TK | 3zc5 | A | | 6-{(1s)-1-[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]ethyl}quinoline | Human | 3003 | 0.43 | |
| DYRK1A | DYRK | CMGC | 6s11 | A | A | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11361 | 0.42 | |
| DYRK1A | DYRK | CMGC | 6s11 | B | B | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11372 | 0.42 | |
| DYRK1A | DYRK | CMGC | 6s11 | B | A | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11378 | 0.42 | |
| DYRK1A | DYRK | CMGC | 6s11 | A | B | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11364 | 0.42 | |
| MET | Met | TK | 5eob | A | A | 6-[bis(fluoranyl)-[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinoline | Human | 7100 | 0.67 | |
| MET | Met | TK | 3zbx | A | | 6-[[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinoline | Human | 3036 | 0.44 | |
| MET | Met | TK | 5eob | A | B | 6-[bis(fluoranyl)-[6-(4-fluorophenyl)-[1,2,4]triazolo[4,3-b][1,2,4]triazin-3-yl]methyl]quinoline | Human | 7101 | 0.67 | |
| MET | Met | TK | 3dkf | A | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 3029 | 0.46 | |
| MET | Met | TK | 3qti | A | B | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | 3028 | 0.41 | |
| MET | Met | TK | 3dkf | A | C | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 2984 | 0.46 | |
| MET | Met | TK | 3dkg | A | C | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 3006 | 0.46 | |
| MET | Met | TK | 3qti | B | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)imidazo[1,2-b]pyridazin-3-yl]methyl}quinoline | Human | 3017 | 0.41 | |
| MET | Met | TK | 3dkg | A | A | 6-{[6-(1-methyl-1h-pyrazol-4-yl)[1,2,4]triazolo[4,3-b]pyridazin-3-yl]sulfanyl}quinoline | Human | 2993 | 0.46 | |