| EGFR | EGFR | TK | 4i23 | A | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 870 | 0.43 | |
| EGFR | EGFR | TK | 4lrm | B | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 867 | 0.44 | |
| EGFR | EGFR | TK | 4ll0 | A | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 804 | 0.44 | |
| EGFR | EGFR | TK | 4ll0 | B | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 796 | 0.44 | |
| EGFR | EGFR | TK | 1xkk | A | | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamine | Human | 844 | 0.57 | |
| JAK3 | JakA | TK | 4z16 | C | | n-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamide | Human | 6397 | 0.40 | |
| EGFR | EGFR | TK | 4i24 | A | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 831 | 0.43 | |
| CDK2 | CDK | CMGC | 1di8 | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 4577 | 0.41 | |
| EGFR | EGFR | TK | 2j5f | A | | n-[4-(3-bromo-phenylamino)-quinazolin-6-yl]-acrylamide | Human | 862 | 0.59 | |
| EGFR | EGFR | TK | 8hy7 | A | | ~{n}-[3-[[6-fluoranyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]quinazolin-4-yl]amino]phenyl]prop-2-enamide | Human | 14941 | 0.44 | |
| JAK3 | JakA | TK | 4z16 | D | | n-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamide | Human | 6394 | 0.40 | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbt | B | | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamine | Human | 2825 | 0.57 | |
| EGFR | EGFR | TK | 4lrm | E | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 825 | 0.44 | |
| JAK3 | JakA | TK | 4z16 | B | | n-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamide | Human | 6396 | 0.40 | |
| JAK3 | JakA | TK | 4z16 | A | | n-(3-{[(5-chloro-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]methyl}phenyl)prop-2-enamide | Human | 6395 | 0.40 | |
| EGFR | EGFR | TK | 4lqm | A | | n-[4-(3-bromo-phenylamino)-quinazolin-6-yl]-acrylamide | Human | 785 | 0.59 | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | B | A | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | 2818 | 0.56 | |
| ERBB4 (ErbB4) | EGFR | TK | 3bbt | D | | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-[5-({[2-(methylsulfonyl)ethyl]amino}methyl)-2-furyl]-4-quinazolinamine | Human | 2819 | 0.57 | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | B | B | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | 2823 | 0.56 | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | A | B | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | 2827 | 0.56 | |
| ERBB4 (ErbB4) | EGFR | TK | 2r4b | A | A | n-{3-chloro-4-[(3-fluorobenzyl)oxy]phenyl}-6-ethylthieno[3,2-d]pyrimidin-4-amine | Human | 2822 | 0.56 | |
| PRKACA (PKACa) | PKA | AGC | 6frx | A | | ~{n}-[3-[(5-chloranyl-2-phenylazanyl-pyrimidin-4-yl)amino]phenyl]prop-2-enamide | Human | 11261 | 0.43 | |
| TTBK1 | TTBK | CK1 | 4btk | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 771 | 0.41 | |
| EGFR | EGFR | TK | 4lrm | D | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 786 | 0.44 | |
| EGFR | EGFR | TK | 4lrm | A | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 901 | 0.44 | |
| EGFR | EGFR | TK | 4i24 | B | | (2e)-n-{4-[(3-chloro-4-fluorophenyl)amino]-7-methoxyquinazolin-6-yl}-4-(piperidin-1-yl)but-2-enamide | Human | 910 | 0.43 | |
| EGFR | EGFR | TK | 4lrm | C | | n-{4-[(3-bromophenyl)amino]quinazolin-6-yl}propanamide | Human | 781 | 0.44 | |
| EGFR | EGFR | TK | 8kfq | A | | ~{n}-[3-[[6-chloranyl-2-[(1-ethylpyrazol-4-yl)amino]quinazolin-4-yl]amino]phenyl]prop-2-enamide | Human | 15367 | 0.42 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12049 | 0.41 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12046 | 0.41 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12047 | 0.41 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12048 | 0.41 | |
| RET | Ret | TK | 5amn | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 6412 | 0.41 | |