| AURKA (AurA) | Aur | Other | 2wtv | A | A | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2056 | 0.70 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | C | A | alisertib | Human | 7186 | 1.00 | |
| AURKA (AurA) | Aur | Other | 2wtv | B | A | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2037 | 0.70 | |
| FGFR1 | FGFR | TK | 5ur1 | B | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 7969 | 0.40 | |
| AURKA (AurA) | Aur | Other | 3h10 | D | | 9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amine | Human | 2059 | 0.63 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | C | B | alisertib | Human | 7175 | 1.00 | |
| AURKA (AurA) | Aur | Other | 2wtv | C | A | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2017 | 0.70 | |
| AURKA (AurA) | Aur | Other | 2wtv | B | B | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2057 | 0.70 | |
| EPHA2 (EphA2) | Eph | TK | 5ia1 | A | | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 7191 | 0.70 | |
| AURKA (AurA) | Aur | Other | 2wtw | A | | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 1956 | 0.70 | |
| AURKA (AurA) | Aur | Other | 3h10 | B | | 9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amine | Human | 1988 | 0.63 | |
| AURKA (AurA) | Aur | Other | 2wtv | D | B | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2076 | 0.70 | |
| AURKA (AurA) | Aur | Other | 3h10 | A | | 9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amine | Human | 2009 | 0.63 | |
| AURKA (AurA) | Aur | Other | 2wtv | C | B | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2016 | 0.70 | |
| AURKA (AurA) | Aur | Other | 2x81 | A | | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 1966 | 0.70 | |
| AURKA (AurA) | Aur | Other | 2wtv | A | B | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 1997 | 0.70 | |
| AURKA (AurA) | Aur | Other | 2wtv | D | A | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 2078 | 0.70 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | A | B | alisertib | Human | 7171 | 1.00 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | B | A | alisertib | Human | 7174 | 1.00 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | A | A | alisertib | Human | 7169 | 1.00 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | B | B | alisertib | Human | 7179 | 1.00 | |
| FGFR1 | FGFR | TK | 5ur1 | B | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 7971 | 0.40 | |
| FGFR1 | FGFR | TK | 5ur1 | A | B | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 7972 | 0.40 | |
| FGFR1 | FGFR | TK | 5ur1 | A | A | 3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 7970 | 0.40 | |
Match: