| MERTK (MER) | Axl | TK | 7ab2 | A | A | 4-[2-(butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | Human | 12934 | 0.85 | |
| MERTK (MER) | Axl | TK | 5k0k | B | B | 15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-one | Human | 7346 | 0.41 | |
| MERTK (MER) | Axl | TK | 5k0k | A | B | 15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-one | Human | 7347 | 0.41 | |
| MERTK (MER) | Axl | TK | 5k0k | A | A | 15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-one | Human | 7345 | 0.41 | |
| MERTK (MER) | Axl | TK | 6mep | A | | cis-4-[(2-[(4-{[4-(1,3-dioxolan-2-yl)pyridin-2-yl]ethynyl}phenyl)amino]-5-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}pyrimidin-4-yl)amino]cyclohexan-1-ol | Human | 11602 | 0.40 | |
| MERTK (MER) | Axl | TK | 5k0k | B | A | 15-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}-4,5,6,7,9,10,11,12-octahydro-2,16-(azenometheno)pyrrolo[2,1-d][1,3,5,9]tetraazacyclotetradecin-8(3h)-one | Human | 7348 | 0.41 | |
| MERTK (MER) | Axl | TK | 7ab2 | A | B | 4-[2-(butylamino)-5-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexan-1-ol | Human | 12936 | 0.85 | |
| MERTK (MER) | Axl | TK | 6mep | B | | cis-4-[(2-[(4-{[4-(1,3-dioxolan-2-yl)pyridin-2-yl]ethynyl}phenyl)amino]-5-{4-[(4-methylpiperazin-1-yl)methyl]phenyl}pyrimidin-4-yl)amino]cyclohexan-1-ol | Human | 11601 | 0.40 | |
| PAK1 | STE20 | STE | 5dfp | A | A | 6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-8-ethyl-2-{[2-(1-methylpiperidin-4-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6366 | 0.43 | |
| PAK1 | STE20 | STE | 5dfp | A | B | 6-[2-chloro-4-(6-methylpyrazin-2-yl)phenyl]-8-ethyl-2-{[2-(1-methylpiperidin-4-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6363 | 0.43 | |