Search results (28 entries covering 13 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
CAMK1D (CaMK1d)CAMK1CAMK8bfsAA3~{h}-pyrrolo[2,3-c]isoquinolin-5-amineHuman14506
CAMK1 (CaMK1a)CAMK1CAMK4fg7Aadenosine-5'-triphosphateHuman4848
CAMK1D (CaMK1d)CAMK1CAMK8bfmApyrazolo[5,1-a]phthalazin-6-amineHuman14516
CAMK1D (CaMK1d)CAMK1CAMK6qp5AA-Human12028
CAMK1D (CaMK1d)CAMK1CAMK6t6fBA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11941
CAMK1D (CaMK1d)CAMK1CAMK6t29AB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamideHuman13203
CAMK1D (CaMK1d)CAMK1CAMK6t6fAB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11940
CAMK1D (CaMK1d)CAMK1CAMK6t6fBB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11942
CAMK1 (CaMK1a)CAMK1CAMK4fg9Aadenosine-5'-triphosphateHuman4846
CAMK1 (CaMK1a)CAMK1CAMK4fg9Badenosine-5'-triphosphateHuman4845
CAMK1 (CaMK1a)CAMK1CAMK4fgbA-Human4847
CAMK1 (CaMK1a)CAMK1CAMK4fg8Badenosine-5'-triphosphateHuman4849
CAMK1 (CaMK1a)CAMK1CAMK4fg8Aadenosine-5'-triphosphateHuman4850
CAMK1G (CaMK1g)CAMK1CAMK2jamAB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1221
CAMK1G (CaMK1g)CAMK1CAMK2jamAA5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1218
CAMK1G (CaMK1g)CAMK1CAMK2jamBA5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1220
CAMK1G (CaMK1g)CAMK1CAMK2jamBB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1219
CAMK1D (CaMK1d)CAMK1CAMK6t28AA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamideHuman13202
CAMK1D (CaMK1d)CAMK1CAMK2jc6CAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4832
CAMK1D (CaMK1d)CAMK1CAMK2jc6CBn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4831
CAMK1D (CaMK1d)CAMK1CAMK6t6fAA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11939
CAMK1D (CaMK1d)CAMK1CAMK2jc6ABn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4830
CAMK1D (CaMK1d)CAMK1CAMK8bfsAB3~{h}-pyrrolo[2,3-c]isoquinolin-5-amineHuman14505
CAMK1D (CaMK1d)CAMK1CAMK6t29AA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamideHuman13204
CAMK1D (CaMK1d)CAMK1CAMK2jc6AAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4829
CAMK1D (CaMK1d)CAMK1CAMK6qp5AB-Human12029
CAMK1D (CaMK1d)CAMK1CAMK6t28AB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamideHuman13205
CAMK4 (CaMK4)CAMK1CAMK2w4oA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman2687