Search results (42 entries covering 26 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
CAMK2A (CaMK2a)CAMK2CAMK7uirAadenosine-5'-triphosphateHuman14173
CAMK2A (CaMK2a)CAMK2CAMK7kl1Badenosine-5'-triphosphateHuman13062
CAMK2B (CaMK2b)CAMK2CAMK3bhhD-Human1504
CAMK2B (CaMK2b)CAMK2CAMK3bhhB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1506
CAMK2B (CaMK2b)CAMK2CAMK3bhhC-Human1505
CAMK2B (CaMK2b)CAMK2CAMK3bhhA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1507
CAMK2A (CaMK2a)CAMK2CAMK6vzkA4'-hydroxycinnamic acidHuman12165
CAMK2D (CaMK2d)CAMK2CAMK8usoA-Human15247
CAMK2D (CaMK2d)CAMK2CAMK9blhAB7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman16000
CAMK2D (CaMK2d)CAMK2CAMK9blhAA7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman16001
CAMK2A (CaMK2a)CAMK2CAMK7kl0Amethyl 6-o-(heptylcarbamoyl)-beta-l-altropyranosideHuman13111
CAMK2A (CaMK2a)CAMK2CAMK7uisA-Human14174
CAMK2A (CaMK2a)CAMK2CAMK7ujrA-Human14191
CAMK2A (CaMK2a)CAMK2CAMK7kl2A-Human13064
CAMK2G (CaMK2g)CAMK2CAMK2v7oAB-Human7238
CAMK2G (CaMK2g)CAMK2CAMK2v7oAA-Human7239
CAMK2D (CaMK2d)CAMK2CAMK5vloAn-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideHuman8348
CAMK2A (CaMK2a)CAMK2CAMK3soaA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman2473
CAMK2A (CaMK2a)CAMK2CAMK6x5gAA-Human13061
CAMK2A (CaMK2a)CAMK2CAMK6w4oO-Human12485
CAMK2A (CaMK2a)CAMK2CAMK7ujtAadenosine-5'-triphosphateHuman14192
CAMK2A (CaMK2a)CAMK2CAMK2vz6AA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2472
CAMK2A (CaMK2a)CAMK2CAMK2vz6BA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2474
CAMK2A (CaMK2a)CAMK2CAMK7ujpAadenosine-5'-diphosphateHuman14193
CAMK2A (CaMK2a)CAMK2CAMK7kl1Aadenosine-5'-triphosphateHuman13059
CAMK2A (CaMK2a)CAMK2CAMK6w4pH-Human12484
CAMK2A (CaMK2a)CAMK2CAMK7kl0Bmethyl 6-o-(heptylcarbamoyl)-beta-l-altropyranosideHuman13114
CAMK2A (CaMK2a)CAMK2CAMK6x5qA-Human13056
CAMK2A (CaMK2a)CAMK2CAMK7ujsAadenosine-5'-diphosphateHuman14190
CAMK2A (CaMK2a)CAMK2CAMK6x5gAB-Human13068
CAMK2A (CaMK2a)CAMK2CAMK2vz6BB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2470
CAMK2A (CaMK2a)CAMK2CAMK2vz6AB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2471
CAMK2A (CaMK2a)CAMK2CAMK7ujqAmethyl 6-o-(heptylcarbamoyl)-beta-l-altropyranosideHuman14189
CAMK2D (CaMK2d)CAMK2CAMK6aywBn-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman8665
CAMK2A (CaMK2a)CAMK2CAMK7uiqA-Human14175
CAMK2D (CaMK2d)CAMK2CAMK2welAB(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2137
CAMK2D (CaMK2d)CAMK2CAMK6aywAn-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman8666
CAMK2D (CaMK2d)CAMK2CAMK2vn9A[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2140
CAMK2D (CaMK2d)CAMK2CAMK2vn9B[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2139
CAMK2D (CaMK2d)CAMK2CAMK5vloBn-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideHuman8347
CAMK2D (CaMK2d)CAMK2CAMK2welAC(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2136
CAMK2D (CaMK2d)CAMK2CAMK2welAA(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2138