Search results (418 entries covering 242 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
STK11 (LKB1)CAMKLCAMK8vsuBadenosine-5'-diphosphateHuman15343
MARK3CAMKLCAMK7p1lA5-bromo-4-n-[2-(1h-imidazol-5-yl)ethyl]-2-n-[3-(morpholin-4-ylmethyl)phenyl]pyrimidine-2,4-diamineHuman13799
CHEK1 (CHK1)CAMKLCAMK4ft5AB1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1633
CHEK1 (CHK1)CAMKLCAMK2wmtAA2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-olHuman1576
CHEK1 (CHK1)CAMKLCAMK2ywpA1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)ureaHuman1658
CHEK1 (CHK1)CAMKLCAMK4fswAB8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1623
CHEK1 (CHK1)CAMKLCAMK2ym6AA1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamineHuman1563
CHEK1 (CHK1)CAMKLCAMK6fcfAA4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamideHuman9503
CHEK1 (CHK1)CAMKLCAMK2hxlA3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrileHuman1552
CHEK1 (CHK1)CAMKLCAMK2cgxA2-[(6-amino-7h-purin-8-yl)thio]acetamideHuman1595
PRKAA2 (AMPKa2)CAMKLCAMK6b1uCAstaurosporineHuman9847
CHEK1 (CHK1)CAMKLCAMK3f9nAB-Human1666
CHEK1 (CHK1)CAMKLCAMK2yerAB5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-oneHuman1583
CHEK1 (CHK1)CAMKLCAMK5op4A[4-[[4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-fluoranyl-5-methoxy-phenyl]-morpholin-4-yl-methanoneHuman8613
CHEK1 (CHK1)CAMKLCAMK2wmvA1-[(2s)-4-(7h-purin-6-yl)morpholin-2-yl]methanamineHuman1562
PRKAA2 (AMPKa2)CAMKLCAMK6bx6AA2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman9878
CHEK1 (CHK1)CAMKLCAMK4ftkAA3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-olHuman1608
CHEK1 (CHK1)CAMKLCAMK4ftrAB2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamideHuman1535
CHEK1 (CHK1)CAMKLCAMK4hyiAB2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman1681
CHEK1 (CHK1)CAMKLCAMK4ftiABmethyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylateHuman1659
CHEK1 (CHK1)CAMKLCAMK5oq7AA5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8601
CHEK1 (CHK1)CAMKLCAMK4fswAA8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1541
CHEK1 (CHK1)CAMKLCAMK2wmwA1-[(2s)-4-(5-bromo-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamineHuman1594
CHEK1 (CHK1)CAMKLCAMK1zltA(4z)-4-(2-amino-5-oxo-3,5-dihydro-4h-imidazol-4-ylidene)-2,3-dichloro-4,5,6,7-tetrahydropyrrolo[2,3-c]azepin-8(1h)-oneHuman1596
CHEK1 (CHK1)CAMKLCAMK5oq6A2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman8610
CHEK1 (CHK1)CAMKLCAMK2ydkA2-(carbamoylamino)-5-phenyl-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamideHuman1646
CHEK1 (CHK1)CAMKLCAMK5opbAA(2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholineHuman8602
CHEK1 (CHK1)CAMKLCAMK2brnA(2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-olHuman1631
CHEK1 (CHK1)CAMKLCAMK4ftnAA4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-olHuman1695
CHEK1 (CHK1)CAMKLCAMK5opvA4-(3-methylphenyl)-6-[(1-methylpyrazol-3-yl)amino]-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrileHuman8608
CHEK1 (CHK1)CAMKLCAMK4fsuAB4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrileHuman1615
MARK2CAMKLCAMK3iecA-Human3045
MARK2CAMKLCAMK5kz7A7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-oneHuman7967
MARK2CAMKLCAMK5kz8A5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-oneHuman7965
MARK2CAMKLCAMK5eakAn-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHuman6410
CHEK1 (CHK1)CAMKLCAMK2ydjB5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman1687
CHEK1 (CHK1)CAMKLCAMK7bjjAB1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman13779
CHEK1 (CHK1)CAMKLCAMK2ym4ABethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1560
CHEK1 (CHK1)CAMKLCAMK2wmqAn-(4-oxo-5,6,7,8-tetrahydro-4h-[1,3]thiazolo[5,4-c]azepin-2-yl)acetamideHuman1647
PRKAA1 (AMPKa1)CAMKLCAMK4rerAstaurosporineHuman121
PRKAA1 (AMPKa1)CAMKLCAMK4redA-Human122
PRKAA1 (AMPKa1)CAMKLCAMK4rewAstaurosporineHuman124
PRKAA1 (AMPKa1)CAMKLCAMK7jhgA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman13816
PRKAA1 (AMPKa1)CAMKLCAMK6c9hAstaurosporineHuman10714
PRKAA1 (AMPKa1)CAMKLCAMK7jhhA-Human13817
PRKAA1 (AMPKa1)CAMKLCAMK7m74A6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman14017
PRKAA1 (AMPKa1)CAMKLCAMK7jijB-Human13819
PRKAA1 (AMPKa1)CAMKLCAMK6c9jAstaurosporineHuman10717
CHEK1 (CHK1)CAMKLCAMK5opbAB(2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholineHuman8604
CHEK1 (CHK1)CAMKLCAMK7bjxAA4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13772
CHEK1 (CHK1)CAMKLCAMK7bjdAA2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrileHuman13775
CHEK1 (CHK1)CAMKLCAMK7bjxAB4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13768
CHEK1 (CHK1)CAMKLCAMK7bk1A4-amino-2-[(1,3-dimethyl-1h-pyrazol-4-yl)amino]-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13763
CHEK1 (CHK1)CAMKLCAMK7bjoA4-amino-6-(2,3-difluorophenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13780
CHEK1 (CHK1)CAMKLCAMK7suiA(3r,4r)-4-{(3s,4s)-4-[6-chloro-2-({5-chloro-1-[(1r)-2,2-difluorocyclopropyl]-1h-pyrazol-4-yl}amino)quinazolin-7-yl]-3-fluoropiperidin-1-yl}oxolan-3-olHuman14045
MARK2CAMKLCAMK5kz8B5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-oneHuman7968
MARK2CAMKLCAMK5kz7B7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-oneHuman7966
MARK2CAMKLCAMK3iecC-Human3046
MARK2CAMKLCAMK5eakBn-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHuman6411
MARK2CAMKLCAMK3iecB-Human3044
MARK2CAMKLCAMK3iecD-Human3043
MARK1CAMKLCAMK2hakD-Human257
SIK3 (QSK)CAMKLCAMK8r4qA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman15241
SIK3 (QSK)CAMKLCAMK8r4oA2-[bis(fluoranyl)methoxy]-4-[6-(2-cyanopropan-2-yl)pyrazolo[1,5-a]pyridin-3-yl]-~{n}-[(1~{r},2~{s})-2-fluoranylcyclopropyl]-6-methoxy-benzamideHuman15242
SIK3 (QSK)CAMKLCAMK8r4uA8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman15240
SIK3 (QSK)CAMKLCAMK8r4vA1-(2,4-dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]ureaHuman15243
CHEK1 (CHK1)CAMKLCAMK10iaA(10as,13as)-3-cyclopropyl-1-methyl-8-(trifluoromethyl)-3,4,10a,11,13a,14-hexahydro-10h,13h-9,5-(azeno)furo[3,4-k]pyrazolo[4,3-b][1,4,6,10]oxatriazacyclotridecineHuman15693
CHEK1 (CHK1)CAMKLCAMK10hzA(10as,13as)-3-cyclobutyl-1-methyl-8-(trifluoromethyl)-3,4,10a,11,13a,14-hexahydro-10h,13h-9,5-(azeno)furo[3,4-k]pyrazolo[4,3-b][1,4,6,10]oxatriazacyclotridecineHuman15694
CHEK1 (CHK1)CAMKLCAMK10hyA(11r)-8-chloro-3,11-dimethyl-2-(oxan-4-yl)-2,4,10,11,12,13-hexahydro-9,5-(azeno)pyrazolo[3,4-b][1,4,6,10]oxatriazacyclotridecineHuman15695
MARK3CAMKLCAMK8uohAB-Human15733
MARK3CAMKLCAMK9virA~{n}-[5-[[4-[[(3~{r},3~{a}~{r},6~{a}~{s})-3-methoxy-2,3,3~{a},6~{a}-tetrahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[[(2~{r},8~{r})-2-fluoranyl-1,2,3,5,6,7-hexahydropyrrolizin-8-yl]methoxy]phenyl]-1-methyl-pyrazole-4-carboxamideHuman15734
MARK3CAMKLCAMK8uohAA-Human15735
MELKCAMKLCAMK9f31An-[4-(1h-indazol-5-yl)phenyl]propanamideHuman15787
CHEK1 (CHK1)CAMKLCAMK7akoABstaurosporineHuman13495
CHEK1 (CHK1)CAMKLCAMK4gh2AB3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1652
CHEK1 (CHK1)CAMKLCAMK2hogA(5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanolHuman1653
CHEK1 (CHK1)CAMKLCAMK4fsqAB4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-olHuman1598
CHEK1 (CHK1)CAMKLCAMK5op2AA5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8595
CHEK1 (CHK1)CAMKLCAMK4qyfA4-[3-amino-6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acidHuman1622
CHEK1 (CHK1)CAMKLCAMK2brgA(5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-aceticHuman1589
PRKAA2 (AMPKa2)CAMKLCAMK7myjA(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman14273
CHEK1 (CHK1)CAMKLCAMK7bjdAB2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrileHuman13774
MARK1CAMKLCAMK2hakG-Human256
MARK1CAMKLCAMK2hakF-Human254
PRKAA2 (AMPKa2)CAMKLCAMK2yzaA-Human189
CHEK1 (CHK1)CAMKLCAMK2ym6AB1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamineHuman1559
PRKAA2 (AMPKa2)CAMKLCAMK6bx6AB2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman9877
PRKAA2 (AMPKa2)CAMKLCAMK5isoAstaurosporineHuman7981
PRKAA2 (AMPKa2)CAMKLCAMK6b1uCBstaurosporineHuman9850
PRKAA2 (AMPKa2)CAMKLCAMK5isoCstaurosporineHuman7980
PRKAA2 (AMPKa2)CAMKLCAMK4zhxCB(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6423
SNRKCAMKLCAMK5yksA-Human8660
MARK1CAMKLCAMK6c9dBB-Human10050
MARK1CAMKLCAMK6c9dBA-Human10049
MARK1CAMKLCAMK2hakH-Human261
MARK1CAMKLCAMK6c9dAA-Human10052
PRKAA2 (AMPKa2)CAMKLCAMK4cfeCstaurosporineHuman192
PRKAA2 (AMPKa2)CAMKLCAMK4cffAstaurosporineHuman191
CHEK1 (CHK1)CAMKLCAMK4ftqAA5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrileHuman1664
CHEK1 (CHK1)CAMKLCAMK2ym3ABethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1543
CHEK1 (CHK1)CAMKLCAMK3ot3AB5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amineHuman1602
CHEK1 (CHK1)CAMKLCAMK4ftqAB5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrileHuman1550
CHEK1 (CHK1)CAMKLCAMK7bk3A4-amino-7-methyl-2-({5-methyl-1-[(3s)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13764
CHEK1 (CHK1)CAMKLCAMK3ot8ABn-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amineHuman1590
CHEK1 (CHK1)CAMKLCAMK2cgvA(2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-olHuman1545
CHEK1 (CHK1)CAMKLCAMK5f4nABmethyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylateHuman6652
CHEK1 (CHK1)CAMKLCAMK4jikA2-(4-chlorophenyl)-8-[(3s)-piperidin-3-ylamino]imidazo[1,2-c]pyrimidine-5-carboxamideHuman1698
CHEK1 (CHK1)CAMKLCAMK4ft9AA1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylureaHuman1564
CHEK1 (CHK1)CAMKLCAMK7akoBAstaurosporineHuman13492
CHEK1 (CHK1)CAMKLCAMK7akmBB-Human13493
CHEK1 (CHK1)CAMKLCAMK2yexAA5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1651
CHEK1 (CHK1)CAMKLCAMK4ft9AB1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylureaHuman1648
CHEK1 (CHK1)CAMKLCAMK4gh2AA3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1600
CHEK1 (CHK1)CAMKLCAMK5oq7AB5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8594
CHEK1 (CHK1)CAMKLCAMK2c3lA3-(1h-benzimidazol-2-yl)-1h-indazoleHuman1612
CHEK1 (CHK1)CAMKLCAMK8sivAn-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)cyclopropanecarboxamideHuman14886
CHEK1 (CHK1)CAMKLCAMK4qygB3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acidHuman1607
CHEK1 (CHK1)CAMKLCAMK5op2AB5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8611
CHEK1 (CHK1)CAMKLCAMK4fsyAA2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamideHuman1547
CHEK1 (CHK1)CAMKLCAMK6fc8AA2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamideHuman9500
CHEK1 (CHK1)CAMKLCAMK7bknAadenineHuman13769
CHEK1 (CHK1)CAMKLCAMK3tkiAn-(2-aminoethyl)-5-(2-{[4-(morpholin-4-yl)pyridin-2-yl]amino}-1,3-thiazol-5-yl)pyridine-3-carboxamideHuman1599
CHEK1 (CHK1)CAMKLCAMK2cguA2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acidHuman1697
CHEK1 (CHK1)CAMKLCAMK5oq5A2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman8597
CHEK1 (CHK1)CAMKLCAMK5oq7BB5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8596
CHEK1 (CHK1)CAMKLCAMK7bjmA4-amino-6-{[(2-fluorophenyl)methyl]amino}-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13770
CHEK1 (CHK1)CAMKLCAMK7akmBA-Human13494
CHEK1 (CHK1)CAMKLCAMK7bjhABn,n-dimethyl-7h-purin-6-amineHuman13771
CHEK1 (CHK1)CAMKLCAMK8e80A2-[(1r,4r)-2-{(6p)-6-[(6m)-6-(1h-pyrazol-5-yl)-1h-indazol-1-yl]pyrimidin-4-yl}-2-azabicyclo[2.1.1]hexan-4-yl]propan-2-olHuman14621
CHEK1 (CHK1)CAMKLCAMK2c3jAdebromohymenialdisineHuman1551
CHEK1 (CHK1)CAMKLCAMK4hyiAA2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman1538
CHEK1 (CHK1)CAMKLCAMK2yexAB5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1567
CHEK1 (CHK1)CAMKLCAMK4rvkAn-[3-(6-cyano-9h-pyrrolo[2,3-b:5,4-c']dipyridin-3-yl)phenyl]acetamideHuman1549
CHEK1 (CHK1)CAMKLCAMK4ftjAAtrans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanolHuman1603
CHEK1 (CHK1)CAMKLCAMK4qyhA3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1689
CHEK1 (CHK1)CAMKLCAMK4fsyAB2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamideHuman1537
CHEK1 (CHK1)CAMKLCAMK3tkhA1-(morpholin-4-yl)-2-[4-(2-{[5-(pyridin-3-yl)-1,3-thiazol-2-yl]amino}pyridin-4-yl)piperazin-1-yl]ethanoneHuman1665
CHEK1 (CHK1)CAMKLCAMK4rvlA3-(2-hydroxyphenyl)-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1634
CHEK1 (CHK1)CAMKLCAMK4ftuABmethyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1640
CHEK1 (CHK1)CAMKLCAMK7sufAB8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amineHuman14044
CHEK1 (CHK1)CAMKLCAMK4ftaAA6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acidHuman1540
CHEK1 (CHK1)CAMKLCAMK2x8dAA5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1673
CHEK1 (CHK1)CAMKLCAMK4ftjABtrans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanolHuman1613
CHEK1 (CHK1)CAMKLCAMK3pa4AB2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamideHuman1566
CHEK1 (CHK1)CAMKLCAMK2wmsA[4-amino-2-(tert-butylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman1657
CHEK1 (CHK1)CAMKLCAMK4fsrAB6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazoleHuman1575
CHEK1 (CHK1)CAMKLCAMK4ftcAA1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)ureaHuman1593
CHEK1 (CHK1)CAMKLCAMK2e9uA18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-oneHuman1584
CHEK1 (CHK1)CAMKLCAMK2yerAA5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-oneHuman1611
CHEK1 (CHK1)CAMKLCAMK4ft0AB2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acidHuman1693
MARK2CAMKLCAMK8txyAn-[(5p,8r)-5-(2-cyano-5-{[(3r)-1-methylpyrrolidin-3-yl]methoxy}pyridin-4-yl)pyrazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamideHuman15136
SIK3 (QSK)CAMKLCAMK8okuA~{n}-ethyl-4-[5-[1-(2-hydroxyethyl)pyrazol-4-yl]benzimidazol-1-yl]-2,6-dimethoxy-benzamideHuman15169
MARK1CAMKLCAMK2hakC-Human260
MELKCAMKLCAMK5m5aAAk-252aHuman8735
MELKCAMKLCAMK5maiAA3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman8728
MELKCAMKLCAMK5twyB2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman8669
MELKCAMKLCAMK4d2pDA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2486
MELKCAMKLCAMK6vxrAB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman12644
MELKCAMKLCAMK5k00AA4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamideHuman7497
MELKCAMKLCAMK4d2wAA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2515
MELKCAMKLCAMK4umpCA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2479
MELKCAMKLCAMK4d2vDA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2502
MELKCAMKLCAMK6vxrAA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman12645
MELKCAMKLCAMK4d2pAA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2513
MELKCAMKLCAMK4d2pCB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2501
MELKCAMKLCAMK4umpDB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2525
MELKCAMKLCAMK5twzA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman8675
MELKCAMKLCAMK5m5aABk-252aHuman8733
MELKCAMKLCAMK4umpBB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2504
MELKCAMKLCAMK5tx3B7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-oneHuman8674
MELKCAMKLCAMK4d2vDB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2506
MELKCAMKLCAMK4d2vAB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2522
MELKCAMKLCAMK4umqAB3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminiumHuman2523
MELKCAMKLCAMK5tvtA9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3-methyl-3,4-dihydropyrimido[5,4-c][1,5]naphthyridin-2(1h)-oneHuman8667
MELKCAMKLCAMK4d2wCB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2503
MELKCAMKLCAMK6gvxAB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11139
MELKCAMKLCAMK5ihaAA1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazineHuman6663
MELKCAMKLCAMK5twlA9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3,4-dihydropyrimido[5,4-c]quinolin-2(1h)-oneHuman8668
MELKCAMKLCAMK4d2tAB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2489
MELKCAMKLCAMK5magAApf-3758309Human8736
MELKCAMKLCAMK4bkyAB3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamideHuman2490
MELKCAMKLCAMK4d2vBB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2507
MELKCAMKLCAMK4bkzABn-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamideHuman2484
MELKCAMKLCAMK4umpAA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2497
MELKCAMKLCAMK5mafAmethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman8732
MELKCAMKLCAMK5ihcAA4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridineHuman6660
MELKCAMKLCAMK4ixpA-Human2528
MELKCAMKLCAMK4d2wDB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2495
MELKCAMKLCAMK5ih8An-[(pyridin-2-yl)methyl]-4-[4-(pyridin-4-yl)-1h-pyrazol-1-yl]benzamideHuman6661
CHEK1 (CHK1)CAMKLCAMK4ftlAB4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-olHuman1573
CHEK1 (CHK1)CAMKLCAMK2e9nA3-(4'-hydroxybiphenyl-4-yl)-n-(4-hydroxycyclohexyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamideHuman1690
PASKCAMKLCAMK3dlsBadenosine-5'-diphosphateHuman3381
PASKCAMKLCAMK3dlsAadenosine-5'-diphosphateHuman3382
CHEK1 (CHK1)CAMKLCAMK3ot8AAn-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amineHuman1569
CHEK1 (CHK1)CAMKLCAMK6fcfAB4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamideHuman9498
PRKAA2 (AMPKa2)CAMKLCAMK4zhxAA(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6425
MARK1CAMKLCAMK6c9dAB-Human10051
MARK1CAMKLCAMK2hakE-Human255
MARK1CAMKLCAMK2hakA-Human258
MARK1CAMKLCAMK2hakB-Human259
MARK4CAMKLCAMK5es1A~{n}-[(1~{r},6~{r})-6-azanyl-2,2-bis(fluoranyl)cyclohexyl]-5-ethyl-4-[6-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHuman6260
MARK4CAMKLCAMK8xflA-Human15101
CHEK1 (CHK1)CAMKLCAMK3ot3AA5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amineHuman1696
CHEK1 (CHK1)CAMKLCAMK5opuA6-azanyl-4-(3-methylphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrileHuman8615
CHEK1 (CHK1)CAMKLCAMK2ym3AAethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1644
CHEK1 (CHK1)CAMKLCAMK8siwA(1s,2s)-n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)-2-(1-methyl-1h-pyrazol-4-yl)cyclopropane-1-carboxamideHuman14885
CHEK1 (CHK1)CAMKLCAMK5dlsA1-benzyl-n-(5-{5-[3-(dimethylamino)-2,2-dimethylpropoxy]-1h-indol-2-yl}-6-oxo-1,6-dihydropyridin-3-yl)-1h-pyrazole-4-carboxamideHuman6151
CHEK1 (CHK1)CAMKLCAMK1zysAn-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamideHuman1655
CHEK1 (CHK1)CAMKLCAMK4fttABmethyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1670
CHEK1 (CHK1)CAMKLCAMK2wmtAB2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-olHuman1685
CHEK1 (CHK1)CAMKLCAMK3pa4AA2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamideHuman1592
CHEK1 (CHK1)CAMKLCAMK2ydiAA5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamideHuman1684
CHEK1 (CHK1)CAMKLCAMK6fckAA2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamideHuman9501
CHEK1 (CHK1)CAMKLCAMK1nvsArel-(9r,12s)-9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2h)-dioneHuman1591
CHEK1 (CHK1)CAMKLCAMK4rvmA3-[4-(piperidin-1-ylmethyl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1624
CHEK1 (CHK1)CAMKLCAMK4ft0AA2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acidHuman1637
CHEK1 (CHK1)CAMKLCAMK2e9vB18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrileHuman1638
CHEK1 (CHK1)CAMKLCAMK2ghgA5-{5-[(s)-2-amino-3-(1h-indol-3-yl)-propoxyl]-pyridin-3-yl}-3-[1-(1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman1581
CHEK1 (CHK1)CAMKLCAMK2e9pA1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}ureaHuman1618
CHEK1 (CHK1)CAMKLCAMK4hyhAB2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamideHuman1626
CHEK1 (CHK1)CAMKLCAMK4fttAAmethyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1565
CHEK1 (CHK1)CAMKLCAMK4ftoAB4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrileHuman1605
CHEK1 (CHK1)CAMKLCAMK4fstAA4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenolHuman1619
CHEK1 (CHK1)CAMKLCAMK7bkoA1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman13765
CHEK1 (CHK1)CAMKLCAMK4ftkAB3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-olHuman1536
CHEK1 (CHK1)CAMKLCAMK5op7A[4-[[5-chloranyl-4-(methylamino)-7~{h}-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-phenyl]-morpholin-4-yl-methanoneHuman8609
CHEK1 (CHK1)CAMKLCAMK4fszAA(3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acidHuman1553
CHEK1 (CHK1)CAMKLCAMK2c3kA4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenolHuman1674
CHEK1 (CHK1)CAMKLCAMK4ftmAB4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenolHuman1556
CHEK1 (CHK1)CAMKLCAMK4ftcAB1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)ureaHuman1680
CHEK1 (CHK1)CAMKLCAMK7akmAAphosphothiophosphoric acid-adenylate esterHuman13489
CHEK1 (CHK1)CAMKLCAMK2e9vA18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrileHuman1574
CHEK1 (CHK1)CAMKLCAMK2hxqA3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-oneHuman1587
CHEK1 (CHK1)CAMKLCAMK1nvrAstaurosporineHuman1585
CHEK1 (CHK1)CAMKLCAMK2wmuAA6-morpholin-4-yl-9h-purineHuman1662
CHEK1 (CHK1)CAMKLCAMK4ftnAB4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-olHuman1678
CHEK1 (CHK1)CAMKLCAMK4fsuAA4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrileHuman1539
CHEK1 (CHK1)CAMKLCAMK2gdoA4-[(3s)-1-azabicyclo[2.2.2]oct-3-ylamino]-3-(1h-benzimidazol-2-yl)-6-chloroquinolin-2(1h)-oneHuman1606
CHEK1 (CHK1)CAMKLCAMK2broA(2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diolHuman1686
CHEK1 (CHK1)CAMKLCAMK2ydjA5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman1649
CHEK1 (CHK1)CAMKLCAMK2ym4AAethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1572
CHEK1 (CHK1)CAMKLCAMK2ym8A(r)-5-(8-chloroisoquinolin-3-ylamino)-3-(1-(dimethylamino)propan-2-yloxy)pyrazine-2-carbonitrileHuman1588
CHEK1 (CHK1)CAMKLCAMK7bk2A4-amino-7-methyl-2-({5-methyl-1-[(3r)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13766
CHEK1 (CHK1)CAMKLCAMK3nlbA3-methyl-5-[5-(1-methylethyl)-1h-benzimidazol-2-yl]-n-(1-methylpiperidin-4-yl)-1h-pyrazole-4-carboxamideHuman1641
CHEK1 (CHK1)CAMKLCAMK4qyeA4-[6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acidHuman1601
CHEK1 (CHK1)CAMKLCAMK7bjeAAadenineHuman13767
CHEK1 (CHK1)CAMKLCAMK4qyhB3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1586
CHEK1 (CHK1)CAMKLCAMK2ym5A(3-{4-[(2s)-2-(aminomethyl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}phenyl)methanolHuman1627
CHEK1 (CHK1)CAMKLCAMK8e81A(1s)-1-[(1p)-1-{6-[(3r)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}-1h-indazol-6-yl]spiro[2.2]pentane-1-carbonitrileHuman14620
CHEK1 (CHK1)CAMKLCAMK2wmxA1-[(2s)-4-(5-phenyl-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamineHuman1636
CHEK1 (CHK1)CAMKLCAMK7akoAAstaurosporineHuman13490
CHEK1 (CHK1)CAMKLCAMK2brbA2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanolHuman1582
CHEK1 (CHK1)CAMKLCAMK4ftaAB6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acidHuman1660
CHEK1 (CHK1)CAMKLCAMK4qygA3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acidHuman1568
CHEK1 (CHK1)CAMKLCAMK7akmABphosphothiophosphoric acid-adenylate esterHuman13491
CHEK1 (CHK1)CAMKLCAMK7sugAA1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrileHuman14039
CHEK1 (CHK1)CAMKLCAMK2br1AA2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanolHuman1677
CHEK1 (CHK1)CAMKLCAMK7bjeABadenineHuman13773
CHEK1 (CHK1)CAMKLCAMK3pa3AA2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamideHuman1691
CHEK1 (CHK1)CAMKLCAMK2brmAB3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-oneHuman1643
CHEK1 (CHK1)CAMKLCAMK4ft5AA1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1617
CHEK1 (CHK1)CAMKLCAMK2ydiAB5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamideHuman1579
CHEK1 (CHK1)CAMKLCAMK8sixA(1s)-n-(7-chloro-6-{4-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperazin-1-yl}isoquinolin-3-yl)-6-oxaspiro[2.5]octane-1-carboxamideHuman14887
CHEK1 (CHK1)CAMKLCAMK4fsqAA4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-olHuman1688
CHEK1 (CHK1)CAMKLCAMK2ym7AB5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrileHuman1645
CHEK1 (CHK1)CAMKLCAMK2x8iAA7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1699
CHEK1 (CHK1)CAMKLCAMK5f4nAAmethyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylateHuman6651
CHEK1 (CHK1)CAMKLCAMK5op5A3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrileHuman8600
CHEK1 (CHK1)CAMKLCAMK2ym7AA5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrileHuman1650
CHEK1 (CHK1)CAMKLCAMK4ftlAA4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-olHuman1614
CHEK1 (CHK1)CAMKLCAMK4fsrAA6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazoleHuman1629
CHEK1 (CHK1)CAMKLCAMK4ftmAC4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenolHuman1616
CHEK1 (CHK1)CAMKLCAMK2brmAA3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-oneHuman1621
CHEK1 (CHK1)CAMKLCAMK4ftmAA4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenolHuman1546
CHEK1 (CHK1)CAMKLCAMK2e9oA4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHuman1667
CHEK1 (CHK1)CAMKLCAMK5opsA4-(3-hydroxyphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrileHuman8598
CHEK1 (CHK1)CAMKLCAMK4fsnAA4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHuman1542
CHEK1 (CHK1)CAMKLCAMK2r0uA6-(3-aminopropyl)-4-(3-hydroxyphenyl)-9-(1h-pyrazol-4-yl)benzo[h]isoquinolin-1(2h)-oneHuman1632
CHEK1 (CHK1)CAMKLCAMK2xf0A3-phenyl-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazineHuman1534
CHEK1 (CHK1)CAMKLCAMK7bjhAAn,n-dimethyl-7h-purin-6-amineHuman13776
CHEK1 (CHK1)CAMKLCAMK4ftiAAmethyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylateHuman1577
CHEK1 (CHK1)CAMKLCAMK7sufAA8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amineHuman14040
CHEK1 (CHK1)CAMKLCAMK5oorAstaurosporineHuman8603
CHEK1 (CHK1)CAMKLCAMK4ftrAA2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamideHuman1692
CHEK1 (CHK1)CAMKLCAMK4ft7AB1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1557
CHEK1 (CHK1)CAMKLCAMK2hy0A3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-pyrazol-4-yl)quinolin-2(1h)-oneHuman1555
CHEK1 (CHK1)CAMKLCAMK6fckAB2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamideHuman9499
CHEK1 (CHK1)CAMKLCAMK2qhnA5-ethyl-3-methyl-1,5-dihydro-4h-pyrazolo[4,3-c]quinolin-4-oneHuman1675
CHEK1 (CHK1)CAMKLCAMK5oq8A5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8606
CHEK1 (CHK1)CAMKLCAMK6fc8AB2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamideHuman9502
CHEK1 (CHK1)CAMKLCAMK2xezA6-(1h-pyrazol-3-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazineHuman1580
CHEK1 (CHK1)CAMKLCAMK2x8eA5-methyl-8-pyridin-4-yl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1548
CHEK1 (CHK1)CAMKLCAMK5oq7BA5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8605
CHEK1 (CHK1)CAMKLCAMK3pa5AB2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamideHuman1544
CHEK1 (CHK1)CAMKLCAMK7bjjAA1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman13777
CHEK1 (CHK1)CAMKLCAMK7sujA(3r,4r)-4-{4-[6-chloro-2-({1-[(1r)-2,2-difluorocyclopropyl]-5-methyl-1h-pyrazol-4-yl}amino)quinazolin-7-yl]piperidin-1-yl}-4-methyloxolan-3-olHuman14041
CHEK1 (CHK1)CAMKLCAMK3jvsA-Human1630
CHEK1 (CHK1)CAMKLCAMK4ft3AB1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylureaHuman1672
CHEK1 (CHK1)CAMKLCAMK2brhAAn-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycineHuman1694
CHEK1 (CHK1)CAMKLCAMK7sugAB1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrileHuman14042
CHEK1 (CHK1)CAMKLCAMK7suhA1-[5-chloro-4-({6-chloro-7-[1-(oxetan-3-yl)piperidin-4-yl]quinazolin-2-yl}amino)-1h-pyrazol-1-yl]-2-methylpropan-2-olHuman14043
CHEK1 (CHK1)CAMKLCAMK4ft3AA1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylureaHuman1554
CHEK1 (CHK1)CAMKLCAMK3jvrA-Human1625
CHEK1 (CHK1)CAMKLCAMK3pa3AB2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamideHuman1635
CHEK1 (CHK1)CAMKLCAMK4fstAB4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenolHuman1663
CHEK1 (CHK1)CAMKLCAMK2aypA(3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-oneHuman1682
CHEK1 (CHK1)CAMKLCAMK2wmuAB6-morpholin-4-yl-9h-purineHuman1578
CHEK1 (CHK1)CAMKLCAMK2x8dAB5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1620
CHEK1 (CHK1)CAMKLCAMK4ftoAA4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrileHuman1661
CHEK1 (CHK1)CAMKLCAMK5ootA2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman8599
CHEK1 (CHK1)CAMKLCAMK1ia8A-Human1656
CHEK1 (CHK1)CAMKLCAMK4fsmAB4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenolHuman1671
CHEK1 (CHK1)CAMKLCAMK3f9nAA-Human1700
CHEK1 (CHK1)CAMKLCAMK4fsnAB4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHuman1679
CHEK1 (CHK1)CAMKLCAMK4fsmAA4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenolHuman1570
CHEK1 (CHK1)CAMKLCAMK2qhmA(3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylateHuman1669
CHEK1 (CHK1)CAMKLCAMK7bjrA4-amino-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13778
CHEK1 (CHK1)CAMKLCAMK4fszAB(3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acidHuman1628
CHEK1 (CHK1)CAMKLCAMK7mckAn-{5-[(3s)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl}-6-(1-methyl-1h-pyrazol-4-yl)pyridine-2-carboxamideHuman13622
CHEK1 (CHK1)CAMKLCAMK5oopAAphosphoaminophosphonic acid-adenylate esterHuman8612
CHEK1 (CHK1)CAMKLCAMK4ftuAAmethyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1639
CHEK1 (CHK1)CAMKLCAMK4hyhAA2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamideHuman1561
CHEK1 (CHK1)CAMKLCAMK4ft7AA1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1610
CHEK1 (CHK1)CAMKLCAMK2brhABn-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycineHuman1654
CHEK1 (CHK1)CAMKLCAMK2cgwA4,4'-(1-propyl-1h-1,2,4-triazole-3,5-diyl)bis(2,5-dihydro-1,2,5-oxadiazol-3-amine)Human1683
CHEK1 (CHK1)CAMKLCAMK2br1AB2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanolHuman1571
CHEK1 (CHK1)CAMKLCAMK2x8iAB7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1558
CHEK1 (CHK1)CAMKLCAMK2wmrAB5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-oneHuman1604
CHEK1 (CHK1)CAMKLCAMK3pa5AA2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamideHuman1676
CHEK1 (CHK1)CAMKLCAMK5oopABphosphoaminophosphonic acid-adenylate esterHuman8607
CHEK1 (CHK1)CAMKLCAMK2xeyA3-(1h-indol-3-yl)-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazineHuman1668
CHEK1 (CHK1)CAMKLCAMK3u9nA2-(2,3-dihydro-1-benzofuran-5-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman1597
CHEK1 (CHK1)CAMKLCAMK7akoBBstaurosporineHuman13496
CHEK1 (CHK1)CAMKLCAMK1nvqA7-hydroxystaurosporineHuman1642
CHEK1 (CHK1)CAMKLCAMK5oprA5-[4-(morpholin-4-ylmethyl)phenyl]-3-(1-propan-2-yl-1,2,3-triazol-4-yl)pyridin-2-amineHuman8614
MARK3CAMKLCAMK3fe3AA-Human3267
MARK3CAMKLCAMK2qnjA-Human3269
MARK3CAMKLCAMK3fe3BB-Human3265
MARK3CAMKLCAMK2qnjB-Human3264
MARK3CAMKLCAMK9vgrAn-[5-[[4-[[(3r,3ar,6r,6ar)-3-methoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]-1-methyl-pyrazole-4-carboxamideHuman15736
MARK3CAMKLCAMK9ysqA3-({5-chloro-2-[2-(difluoromethoxy)-4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl}amino)thiophene-2-carboxamideHuman15737
MARK3CAMKLCAMK9vfoAn-[5-[[4-[[(3r,3ar,6r,6ar)-3-methoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]-2-azanyl-ethanamideHuman15738
MARK3CAMKLCAMK3fe3AB-Human3266
MARK3CAMKLCAMK3fe3BA-Human3268
MELKCAMKLCAMK4d2tBB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2512
MELKCAMKLCAMK6gvxBB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11138
MELKCAMKLCAMK5ih9AB1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazineHuman6657
MELKCAMKLCAMK4bkzAAn-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamideHuman2505
MELKCAMKLCAMK5mahAA~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamideHuman8729
MELKCAMKLCAMK4d2wBB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2482
MELKCAMKLCAMK4umpCB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2508
MELKCAMKLCAMK4d2pCA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2496
MELKCAMKLCAMK5ihaAB1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazineHuman6658
MELKCAMKLCAMK4umrA4-fluoro-n-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamideHuman2521
MELKCAMKLCAMK6gvxAA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11137
MELKCAMKLCAMK5twuB-Human8672
MELKCAMKLCAMK4d2tBA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2520
MELKCAMKLCAMK4d2tAA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2487
MELKCAMKLCAMK4d2pDB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2518
MELKCAMKLCAMK4umpDA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2516
MELKCAMKLCAMK4d2wCA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2527
MELKCAMKLCAMK5k00AB4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamideHuman7498
MELKCAMKLCAMK4d2wDA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2481
MELKCAMKLCAMK4bl1ABphosphoaminophosphonic acid-adenylate esterHuman2519
MELKCAMKLCAMK5ihcAB4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridineHuman6662
MELKCAMKLCAMK4d2tDA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2530
MELKCAMKLCAMK4d2vAA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2493
MELKCAMKLCAMK4d2pBB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2498
MELKCAMKLCAMK4d2wBA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2500
MELKCAMKLCAMK5ih9AA1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazineHuman6659
MELKCAMKLCAMK4umuA(2-ethoxy-4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}phenyl)methanaminiumHuman2517
MELKCAMKLCAMK4d2pBA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2494
MELKCAMKLCAMK5maiAB3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman8730
MELKCAMKLCAMK6gvxBA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11136
MELKCAMKLCAMK5twyA2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman8671
MELKCAMKLCAMK4d2vBA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2483
MELKCAMKLCAMK4umqAA3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminiumHuman2488
MELKCAMKLCAMK4d2tCA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2491
MELKCAMKLCAMK5mahAB~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamideHuman8734
MELKCAMKLCAMK4bkyAA3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamideHuman2480
MELKCAMKLCAMK4d2tCB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2526
MELKCAMKLCAMK4d2wAB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2509
MELKCAMKLCAMK4umpAB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2485
MELKCAMKLCAMK5twuA-Human8670
MELKCAMKLCAMK5tx3A7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-oneHuman8673
MELKCAMKLCAMK4bl1AAphosphoaminophosphonic acid-adenylate esterHuman2514
MELKCAMKLCAMK4d2vCB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2492
MELKCAMKLCAMK4umtA1-(4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}-2-methoxybenzyl)piperazinediiumHuman2510
MELKCAMKLCAMK5magABpf-3758309Human8731
MELKCAMKLCAMK4umpBA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2524
MELKCAMKLCAMK4d2vCA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2529
MELKCAMKLCAMK4d2pAB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2499
MELKCAMKLCAMK4d2tDB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2511
CHEK1 (CHK1)CAMKLCAMK2wmrAA5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-oneHuman1609
STK11 (LKB1)CAMKLCAMK2wtkFphosphoaminophosphonic acid-adenylate esterHuman1869
STK11 (LKB1)CAMKLCAMK2wtkCphosphoaminophosphonic acid-adenylate esterHuman1868
PASKCAMKLCAMK3dlsFadenosine-5'-diphosphateHuman3380
PASKCAMKLCAMK3dlsCadenosine-5'-diphosphateHuman3377
PASKCAMKLCAMK3dlsEadenosine-5'-diphosphateHuman3379
PASKCAMKLCAMK3dlsDadenosine-5'-diphosphateHuman3378
PRKAA1 (AMPKa1)CAMKLCAMK6c9gAstaurosporineHuman10715
PRKAA1 (AMPKa1)CAMKLCAMK4redB-Human123
PRKAA1 (AMPKa1)CAMKLCAMK6c9fAstaurosporineHuman10716
SNRKCAMKLCAMK5yksB-Human8661
PRKAA2 (AMPKa2)CAMKLCAMK2h6dAB-Human194
PRKAA2 (AMPKa2)CAMKLCAMK5ezvABstaurosporineHuman6428
PRKAA2 (AMPKa2)CAMKLCAMK6b1uABstaurosporineHuman9849
PRKAA2 (AMPKa2)CAMKLCAMK3aqvA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman193
PRKAA2 (AMPKa2)CAMKLCAMK4cfeAstaurosporineHuman195
PRKAA2 (AMPKa2)CAMKLCAMK4zhxCA(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6427
PRKAA2 (AMPKa2)CAMKLCAMK6b1uAAstaurosporineHuman9848
PRKAA2 (AMPKa2)CAMKLCAMK5ezvCAstaurosporineHuman6430
PRKAA2 (AMPKa2)CAMKLCAMK4cffCstaurosporineHuman190
PRKAA2 (AMPKa2)CAMKLCAMK2h6dAA-Human196
PRKAA2 (AMPKa2)CAMKLCAMK5ezvCBstaurosporineHuman6426
PRKAA2 (AMPKa2)CAMKLCAMK5ezvAAstaurosporineHuman6424
PRKAA2 (AMPKa2)CAMKLCAMK6b2eAstaurosporineHuman9851
PRKAA2 (AMPKa2)CAMKLCAMK4zhxAB(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6429