| STK11 (LKB1) | CAMKL | CAMK | 8vsu | B | | adenosine-5'-diphosphate | Human | 15343 | |
| MARK3 | CAMKL | CAMK | 7p1l | A | | 5-bromo-4-n-[2-(1h-imidazol-5-yl)ethyl]-2-n-[3-(morpholin-4-ylmethyl)phenyl]pyrimidine-2,4-diamine | Human | 13799 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | B | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1633 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | A | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | 1576 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ywp | A | | 1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea | Human | 1658 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | B | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1623 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | A | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | 1563 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | A | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | 9503 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hxl | A | | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrile | Human | 1552 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgx | A | | 2-[(6-amino-7h-purin-8-yl)thio]acetamide | Human | 1595 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | C | A | staurosporine | Human | 9847 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | B | - | Human | 1666 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | B | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | 1583 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op4 | A | | [4-[[4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-fluoranyl-5-methoxy-phenyl]-morpholin-4-yl-methanone | Human | 8613 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmv | A | | 1-[(2s)-4-(7h-purin-6-yl)morpholin-2-yl]methanamine | Human | 1562 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6bx6 | A | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 9878 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | A | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | 1608 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | B | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | 1535 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | B | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 1681 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | B | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | 1659 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8601 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | A | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1541 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmw | A | | 1-[(2s)-4-(5-bromo-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | 1594 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1zlt | A | | (4z)-4-(2-amino-5-oxo-3,5-dihydro-4h-imidazol-4-ylidene)-2,3-dichloro-4,5,6,7-tetrahydropyrrolo[2,3-c]azepin-8(1h)-one | Human | 1596 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq6 | A | | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 8610 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydk | A | | 2-(carbamoylamino)-5-phenyl-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | 1646 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | A | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | 8602 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brn | A | | (2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-ol | Human | 1631 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | A | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | 1695 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opv | A | | 4-(3-methylphenyl)-6-[(1-methylpyrazol-3-yl)amino]-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | 8608 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | B | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | 1615 | |
| MARK2 | CAMKL | CAMK | 3iec | A | | - | Human | 3045 | |
| MARK2 | CAMKL | CAMK | 5kz7 | A | | 7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-one | Human | 7967 | |
| MARK2 | CAMKL | CAMK | 5kz8 | A | | 5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-one | Human | 7965 | |
| MARK2 | CAMKL | CAMK | 5eak | A | | n-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide | Human | 6410 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | B | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 1687 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | B | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 13779 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | B | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1560 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmq | A | | n-(4-oxo-5,6,7,8-tetrahydro-4h-[1,3]thiazolo[5,4-c]azepin-2-yl)acetamide | Human | 1647 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4rer | A | | staurosporine | Human | 121 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4red | A | | - | Human | 122 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4rew | A | | staurosporine | Human | 124 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jhg | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 13816 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9h | A | | staurosporine | Human | 10714 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jhh | A | | - | Human | 13817 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7m74 | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 14017 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jij | B | | - | Human | 13819 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9j | A | | staurosporine | Human | 10717 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | B | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | 8604 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | A | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13772 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | A | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | 13775 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | B | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13768 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk1 | A | | 4-amino-2-[(1,3-dimethyl-1h-pyrazol-4-yl)amino]-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13763 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjo | A | | 4-amino-6-(2,3-difluorophenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13780 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sui | A | | (3r,4r)-4-{(3s,4s)-4-[6-chloro-2-({5-chloro-1-[(1r)-2,2-difluorocyclopropyl]-1h-pyrazol-4-yl}amino)quinazolin-7-yl]-3-fluoropiperidin-1-yl}oxolan-3-ol | Human | 14045 | |
| MARK2 | CAMKL | CAMK | 5kz8 | B | | 5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-one | Human | 7968 | |
| MARK2 | CAMKL | CAMK | 5kz7 | B | | 7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-one | Human | 7966 | |
| MARK2 | CAMKL | CAMK | 3iec | C | | - | Human | 3046 | |
| MARK2 | CAMKL | CAMK | 5eak | B | | n-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide | Human | 6411 | |
| MARK2 | CAMKL | CAMK | 3iec | B | | - | Human | 3044 | |
| MARK2 | CAMKL | CAMK | 3iec | D | | - | Human | 3043 | |
| MARK1 | CAMKL | CAMK | 2hak | D | | - | Human | 257 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4q | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 15241 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4o | A | | 2-[bis(fluoranyl)methoxy]-4-[6-(2-cyanopropan-2-yl)pyrazolo[1,5-a]pyridin-3-yl]-~{n}-[(1~{r},2~{s})-2-fluoranylcyclopropyl]-6-methoxy-benzamide | Human | 15242 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4u | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 15240 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4v | A | | 1-(2,4-dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]urea | Human | 15243 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 10ia | A | | (10as,13as)-3-cyclopropyl-1-methyl-8-(trifluoromethyl)-3,4,10a,11,13a,14-hexahydro-10h,13h-9,5-(azeno)furo[3,4-k]pyrazolo[4,3-b][1,4,6,10]oxatriazacyclotridecine | Human | 15693 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 10hz | A | | (10as,13as)-3-cyclobutyl-1-methyl-8-(trifluoromethyl)-3,4,10a,11,13a,14-hexahydro-10h,13h-9,5-(azeno)furo[3,4-k]pyrazolo[4,3-b][1,4,6,10]oxatriazacyclotridecine | Human | 15694 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 10hy | A | | (11r)-8-chloro-3,11-dimethyl-2-(oxan-4-yl)-2,4,10,11,12,13-hexahydro-9,5-(azeno)pyrazolo[3,4-b][1,4,6,10]oxatriazacyclotridecine | Human | 15695 | |
| MARK3 | CAMKL | CAMK | 8uoh | A | B | - | Human | 15733 | |
| MARK3 | CAMKL | CAMK | 9vir | A | | ~{n}-[5-[[4-[[(3~{r},3~{a}~{r},6~{a}~{s})-3-methoxy-2,3,3~{a},6~{a}-tetrahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[[(2~{r},8~{r})-2-fluoranyl-1,2,3,5,6,7-hexahydropyrrolizin-8-yl]methoxy]phenyl]-1-methyl-pyrazole-4-carboxamide | Human | 15734 | |
| MARK3 | CAMKL | CAMK | 8uoh | A | A | - | Human | 15735 | |
| MELK | CAMKL | CAMK | 9f31 | A | | n-[4-(1h-indazol-5-yl)phenyl]propanamide | Human | 15787 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | B | staurosporine | Human | 13495 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | B | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1652 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hog | A | | (5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanol | Human | 1653 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | B | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | 1598 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8595 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyf | A | | 4-[3-amino-6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | 1622 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brg | A | | (5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-acetic | Human | 1589 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 7myj | A | | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 14273 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | B | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | 13774 | |
| MARK1 | CAMKL | CAMK | 2hak | G | | - | Human | 256 | |
| MARK1 | CAMKL | CAMK | 2hak | F | | - | Human | 254 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 2yza | A | | - | Human | 189 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | B | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | 1559 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6bx6 | A | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 9877 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5iso | A | | staurosporine | Human | 7981 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | C | B | staurosporine | Human | 9850 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5iso | C | | staurosporine | Human | 7980 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | C | B | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6423 | |
| SNRK | CAMKL | CAMK | 5yks | A | | - | Human | 8660 | |
| MARK1 | CAMKL | CAMK | 6c9d | B | B | - | Human | 10050 | |
| MARK1 | CAMKL | CAMK | 6c9d | B | A | - | Human | 10049 | |
| MARK1 | CAMKL | CAMK | 2hak | H | | - | Human | 261 | |
| MARK1 | CAMKL | CAMK | 6c9d | A | A | - | Human | 10052 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cfe | C | | staurosporine | Human | 192 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cff | A | | staurosporine | Human | 191 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | A | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | 1664 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | B | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1543 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | B | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1602 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | B | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | 1550 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk3 | A | | 4-amino-7-methyl-2-({5-methyl-1-[(3s)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13764 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | B | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1590 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgv | A | | (2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-ol | Human | 1545 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | B | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | 6652 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4jik | A | | 2-(4-chlorophenyl)-8-[(3s)-piperidin-3-ylamino]imidazo[1,2-c]pyrimidine-5-carboxamide | Human | 1698 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | A | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | 1564 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | A | staurosporine | Human | 13492 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | B | - | Human | 13493 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | A | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1651 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | B | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | 1648 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | A | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1600 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8594 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3l | A | | 3-(1h-benzimidazol-2-yl)-1h-indazole | Human | 1612 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siv | A | | n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)cyclopropanecarboxamide | Human | 14886 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | B | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | 1607 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8611 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | A | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | 1547 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | A | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | 9500 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bkn | A | | adenine | Human | 13769 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tki | A | | n-(2-aminoethyl)-5-(2-{[4-(morpholin-4-yl)pyridin-2-yl]amino}-1,3-thiazol-5-yl)pyridine-3-carboxamide | Human | 1599 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgu | A | | 2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acid | Human | 1697 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq5 | A | | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 8597 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8596 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjm | A | | 4-amino-6-{[(2-fluorophenyl)methyl]amino}-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13770 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | A | - | Human | 13494 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | B | n,n-dimethyl-7h-purin-6-amine | Human | 13771 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e80 | A | | 2-[(1r,4r)-2-{(6p)-6-[(6m)-6-(1h-pyrazol-5-yl)-1h-indazol-1-yl]pyrimidin-4-yl}-2-azabicyclo[2.1.1]hexan-4-yl]propan-2-ol | Human | 14621 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3j | A | | debromohymenialdisine | Human | 1551 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | A | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 1538 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | B | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1567 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvk | A | | n-[3-(6-cyano-9h-pyrrolo[2,3-b:5,4-c']dipyridin-3-yl)phenyl]acetamide | Human | 1549 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | A | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | 1603 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | A | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1689 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | B | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | 1537 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tkh | A | | 1-(morpholin-4-yl)-2-[4-(2-{[5-(pyridin-3-yl)-1,3-thiazol-2-yl]amino}pyridin-4-yl)piperazin-1-yl]ethanone | Human | 1665 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvl | A | | 3-(2-hydroxyphenyl)-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1634 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | B | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1640 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | B | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | 14044 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | A | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | 1540 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | A | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1673 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | B | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | 1613 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | 1566 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wms | A | | [4-amino-2-(tert-butylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 1657 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | B | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | 1575 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | A | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | 1593 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9u | A | | 18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-one | Human | 1584 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | A | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | 1611 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | B | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | 1693 | |
| MARK2 | CAMKL | CAMK | 8txy | A | | n-[(5p,8r)-5-(2-cyano-5-{[(3r)-1-methylpyrrolidin-3-yl]methoxy}pyridin-4-yl)pyrazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide | Human | 15136 | |
| SIK3 (QSK) | CAMKL | CAMK | 8oku | A | | ~{n}-ethyl-4-[5-[1-(2-hydroxyethyl)pyrazol-4-yl]benzimidazol-1-yl]-2,6-dimethoxy-benzamide | Human | 15169 | |
| MARK1 | CAMKL | CAMK | 2hak | C | | - | Human | 260 | |
| MELK | CAMKL | CAMK | 5m5a | A | A | k-252a | Human | 8735 | |
| MELK | CAMKL | CAMK | 5mai | A | A | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 8728 | |
| MELK | CAMKL | CAMK | 5twy | B | | 2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 8669 | |
| MELK | CAMKL | CAMK | 4d2p | D | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2486 | |
| MELK | CAMKL | CAMK | 6vxr | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 12644 | |
| MELK | CAMKL | CAMK | 5k00 | A | A | 4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamide | Human | 7497 | |
| MELK | CAMKL | CAMK | 4d2w | A | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2515 | |
| MELK | CAMKL | CAMK | 4ump | C | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2479 | |
| MELK | CAMKL | CAMK | 4d2v | D | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2502 | |
| MELK | CAMKL | CAMK | 6vxr | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 12645 | |
| MELK | CAMKL | CAMK | 4d2p | A | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2513 | |
| MELK | CAMKL | CAMK | 4d2p | C | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2501 | |
| MELK | CAMKL | CAMK | 4ump | D | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2525 | |
| MELK | CAMKL | CAMK | 5twz | A | | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 8675 | |
| MELK | CAMKL | CAMK | 5m5a | A | B | k-252a | Human | 8733 | |
| MELK | CAMKL | CAMK | 4ump | B | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2504 | |
| MELK | CAMKL | CAMK | 5tx3 | B | | 7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-one | Human | 8674 | |
| MELK | CAMKL | CAMK | 4d2v | D | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2506 | |
| MELK | CAMKL | CAMK | 4d2v | A | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2522 | |
| MELK | CAMKL | CAMK | 4umq | A | B | 3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminium | Human | 2523 | |
| MELK | CAMKL | CAMK | 5tvt | A | | 9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3-methyl-3,4-dihydropyrimido[5,4-c][1,5]naphthyridin-2(1h)-one | Human | 8667 | |
| MELK | CAMKL | CAMK | 4d2w | C | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2503 | |
| MELK | CAMKL | CAMK | 6gvx | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11139 | |
| MELK | CAMKL | CAMK | 5iha | A | A | 1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazine | Human | 6663 | |
| MELK | CAMKL | CAMK | 5twl | A | | 9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3,4-dihydropyrimido[5,4-c]quinolin-2(1h)-one | Human | 8668 | |
| MELK | CAMKL | CAMK | 4d2t | A | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2489 | |
| MELK | CAMKL | CAMK | 5mag | A | A | pf-3758309 | Human | 8736 | |
| MELK | CAMKL | CAMK | 4bky | A | B | 3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamide | Human | 2490 | |
| MELK | CAMKL | CAMK | 4d2v | B | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2507 | |
| MELK | CAMKL | CAMK | 4bkz | A | B | n-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 2484 | |
| MELK | CAMKL | CAMK | 4ump | A | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2497 | |
| MELK | CAMKL | CAMK | 5maf | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 8732 | |
| MELK | CAMKL | CAMK | 5ihc | A | A | 4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridine | Human | 6660 | |
| MELK | CAMKL | CAMK | 4ixp | A | | - | Human | 2528 | |
| MELK | CAMKL | CAMK | 4d2w | D | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2495 | |
| MELK | CAMKL | CAMK | 5ih8 | A | | n-[(pyridin-2-yl)methyl]-4-[4-(pyridin-4-yl)-1h-pyrazol-1-yl]benzamide | Human | 6661 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | B | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | 1573 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9n | A | | 3-(4'-hydroxybiphenyl-4-yl)-n-(4-hydroxycyclohexyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamide | Human | 1690 | |
| PASK | CAMKL | CAMK | 3dls | B | | adenosine-5'-diphosphate | Human | 3381 | |
| PASK | CAMKL | CAMK | 3dls | A | | adenosine-5'-diphosphate | Human | 3382 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | A | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1569 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | B | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | 9498 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | A | A | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6425 | |
| MARK1 | CAMKL | CAMK | 6c9d | A | B | - | Human | 10051 | |
| MARK1 | CAMKL | CAMK | 2hak | E | | - | Human | 255 | |
| MARK1 | CAMKL | CAMK | 2hak | A | | - | Human | 258 | |
| MARK1 | CAMKL | CAMK | 2hak | B | | - | Human | 259 | |
| MARK4 | CAMKL | CAMK | 5es1 | A | | ~{n}-[(1~{r},6~{r})-6-azanyl-2,2-bis(fluoranyl)cyclohexyl]-5-ethyl-4-[6-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide | Human | 6260 | |
| MARK4 | CAMKL | CAMK | 8xfl | A | | - | Human | 15101 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | A | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1696 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opu | A | | 6-azanyl-4-(3-methylphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | 8615 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | A | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1644 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siw | A | | (1s,2s)-n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)-2-(1-methyl-1h-pyrazol-4-yl)cyclopropane-1-carboxamide | Human | 14885 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5dls | A | | 1-benzyl-n-(5-{5-[3-(dimethylamino)-2,2-dimethylpropoxy]-1h-indol-2-yl}-6-oxo-1,6-dihydropyridin-3-yl)-1h-pyrazole-4-carboxamide | Human | 6151 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1zys | A | | n-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamide | Human | 1655 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | B | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1670 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | B | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | 1685 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | 1592 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | A | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | 1684 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | A | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | 9501 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvs | A | | rel-(9r,12s)-9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2h)-dione | Human | 1591 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvm | A | | 3-[4-(piperidin-1-ylmethyl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1624 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | A | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | 1637 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | B | | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | 1638 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ghg | A | | 5-{5-[(s)-2-amino-3-(1h-indol-3-yl)-propoxyl]-pyridin-3-yl}-3-[1-(1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one | Human | 1581 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9p | A | | 1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}urea | Human | 1618 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | B | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | 1626 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | A | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1565 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | B | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | 1605 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | A | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | 1619 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bko | A | | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 13765 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | B | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | 1536 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op7 | A | | [4-[[5-chloranyl-4-(methylamino)-7~{h}-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-phenyl]-morpholin-4-yl-methanone | Human | 8609 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | A | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | 1553 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3k | A | | 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenol | Human | 1674 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | B | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | 1556 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | B | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | 1680 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | A | phosphothiophosphoric acid-adenylate ester | Human | 13489 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | A | | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | 1574 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hxq | A | | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-one | Human | 1587 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvr | A | | staurosporine | Human | 1585 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | A | 6-morpholin-4-yl-9h-purine | Human | 1662 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | B | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | 1678 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | A | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | 1539 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2gdo | A | | 4-[(3s)-1-azabicyclo[2.2.2]oct-3-ylamino]-3-(1h-benzimidazol-2-yl)-6-chloroquinolin-2(1h)-one | Human | 1606 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2bro | A | | (2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diol | Human | 1686 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | A | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 1649 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | A | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1572 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym8 | A | | (r)-5-(8-chloroisoquinolin-3-ylamino)-3-(1-(dimethylamino)propan-2-yloxy)pyrazine-2-carbonitrile | Human | 1588 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk2 | A | | 4-amino-7-methyl-2-({5-methyl-1-[(3r)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13766 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3nlb | A | | 3-methyl-5-[5-(1-methylethyl)-1h-benzimidazol-2-yl]-n-(1-methylpiperidin-4-yl)-1h-pyrazole-4-carboxamide | Human | 1641 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qye | A | | 4-[6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | 1601 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | A | adenine | Human | 13767 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | B | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1586 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym5 | A | | (3-{4-[(2s)-2-(aminomethyl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}phenyl)methanol | Human | 1627 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e81 | A | | (1s)-1-[(1p)-1-{6-[(3r)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}-1h-indazol-6-yl]spiro[2.2]pentane-1-carbonitrile | Human | 14620 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmx | A | | 1-[(2s)-4-(5-phenyl-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | 1636 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | A | staurosporine | Human | 13490 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brb | A | | 2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanol | Human | 1582 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | B | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | 1660 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | A | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | 1568 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | B | phosphothiophosphoric acid-adenylate ester | Human | 13491 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | A | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | 14039 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | A | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | 1677 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | B | adenine | Human | 13773 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | 1691 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | B | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | 1643 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | A | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1617 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | B | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | 1579 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8six | A | | (1s)-n-(7-chloro-6-{4-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperazin-1-yl}isoquinolin-3-yl)-6-oxaspiro[2.5]octane-1-carboxamide | Human | 14887 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | A | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | 1688 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | B | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | 1645 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | A | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1699 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | A | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | 6651 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op5 | A | | 3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | 8600 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | A | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | 1650 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | A | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | 1614 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | A | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | 1629 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | C | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | 1616 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | A | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | 1621 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | A | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | 1546 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9o | A | | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | 1667 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5ops | A | | 4-(3-hydroxyphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | 8598 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | A | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | 1542 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2r0u | A | | 6-(3-aminopropyl)-4-(3-hydroxyphenyl)-9-(1h-pyrazol-4-yl)benzo[h]isoquinolin-1(2h)-one | Human | 1632 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xf0 | A | | 3-phenyl-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | 1534 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | A | n,n-dimethyl-7h-purin-6-amine | Human | 13776 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | A | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | 1577 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | A | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | 14040 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oor | A | | staurosporine | Human | 8603 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | A | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | 1692 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | B | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1557 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hy0 | A | | 3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-pyrazol-4-yl)quinolin-2(1h)-one | Human | 1555 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | B | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | 9499 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2qhn | A | | 5-ethyl-3-methyl-1,5-dihydro-4h-pyrazolo[4,3-c]quinolin-4-one | Human | 1675 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq8 | A | | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8606 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | B | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | 9502 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xez | A | | 6-(1h-pyrazol-3-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | 1580 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8e | A | | 5-methyl-8-pyridin-4-yl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1548 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8605 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | B | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | 1544 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | A | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 13777 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suj | A | | (3r,4r)-4-{4-[6-chloro-2-({1-[(1r)-2,2-difluorocyclopropyl]-5-methyl-1h-pyrazol-4-yl}amino)quinazolin-7-yl]piperidin-1-yl}-4-methyloxolan-3-ol | Human | 14041 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvs | A | | - | Human | 1630 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | B | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | 1672 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | A | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | 1694 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | B | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | 14042 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suh | A | | 1-[5-chloro-4-({6-chloro-7-[1-(oxetan-3-yl)piperidin-4-yl]quinazolin-2-yl}amino)-1h-pyrazol-1-yl]-2-methylpropan-2-ol | Human | 14043 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | A | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | 1554 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvr | A | | - | Human | 1625 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | 1635 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | B | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | 1663 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ayp | A | | (3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-one | Human | 1682 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | B | 6-morpholin-4-yl-9h-purine | Human | 1578 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | B | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1620 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | A | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | 1661 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oot | A | | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 8599 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1ia8 | A | | - | Human | 1656 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | B | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | 1671 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | A | - | Human | 1700 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | B | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | 1679 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | A | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | 1570 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2qhm | A | | (3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylate | Human | 1669 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjr | A | | 4-amino-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13778 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | B | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | 1628 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7mck | A | | n-{5-[(3s)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl}-6-(1-methyl-1h-pyrazol-4-yl)pyridine-2-carboxamide | Human | 13622 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 8612 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | A | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1639 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | A | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | 1561 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | A | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1610 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | B | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | 1654 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgw | A | | 4,4'-(1-propyl-1h-1,2,4-triazole-3,5-diyl)bis(2,5-dihydro-1,2,5-oxadiazol-3-amine) | Human | 1683 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | B | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | 1571 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | B | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1558 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | B | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | 1604 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | A | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | 1676 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 8607 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xey | A | | 3-(1h-indol-3-yl)-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | 1668 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3u9n | A | | 2-(2,3-dihydro-1-benzofuran-5-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 1597 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | B | staurosporine | Human | 13496 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvq | A | | 7-hydroxystaurosporine | Human | 1642 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opr | A | | 5-[4-(morpholin-4-ylmethyl)phenyl]-3-(1-propan-2-yl-1,2,3-triazol-4-yl)pyridin-2-amine | Human | 8614 | |
| MARK3 | CAMKL | CAMK | 3fe3 | A | A | - | Human | 3267 | |
| MARK3 | CAMKL | CAMK | 2qnj | A | | - | Human | 3269 | |
| MARK3 | CAMKL | CAMK | 3fe3 | B | B | - | Human | 3265 | |
| MARK3 | CAMKL | CAMK | 2qnj | B | | - | Human | 3264 | |
| MARK3 | CAMKL | CAMK | 9vgr | A | | n-[5-[[4-[[(3r,3ar,6r,6ar)-3-methoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]-1-methyl-pyrazole-4-carboxamide | Human | 15736 | |
| MARK3 | CAMKL | CAMK | 9ysq | A | | 3-({5-chloro-2-[2-(difluoromethoxy)-4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl}amino)thiophene-2-carboxamide | Human | 15737 | |
| MARK3 | CAMKL | CAMK | 9vfo | A | | n-[5-[[4-[[(3r,3ar,6r,6ar)-3-methoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]-2-azanyl-ethanamide | Human | 15738 | |
| MARK3 | CAMKL | CAMK | 3fe3 | A | B | - | Human | 3266 | |
| MARK3 | CAMKL | CAMK | 3fe3 | B | A | - | Human | 3268 | |
| MELK | CAMKL | CAMK | 4d2t | B | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2512 | |
| MELK | CAMKL | CAMK | 6gvx | B | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11138 | |
| MELK | CAMKL | CAMK | 5ih9 | A | B | 1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazine | Human | 6657 | |
| MELK | CAMKL | CAMK | 4bkz | A | A | n-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 2505 | |
| MELK | CAMKL | CAMK | 5mah | A | A | ~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide | Human | 8729 | |
| MELK | CAMKL | CAMK | 4d2w | B | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2482 | |
| MELK | CAMKL | CAMK | 4ump | C | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2508 | |
| MELK | CAMKL | CAMK | 4d2p | C | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2496 | |
| MELK | CAMKL | CAMK | 5iha | A | B | 1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazine | Human | 6658 | |
| MELK | CAMKL | CAMK | 4umr | A | | 4-fluoro-n-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamide | Human | 2521 | |
| MELK | CAMKL | CAMK | 6gvx | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11137 | |
| MELK | CAMKL | CAMK | 5twu | B | | - | Human | 8672 | |
| MELK | CAMKL | CAMK | 4d2t | B | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2520 | |
| MELK | CAMKL | CAMK | 4d2t | A | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2487 | |
| MELK | CAMKL | CAMK | 4d2p | D | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2518 | |
| MELK | CAMKL | CAMK | 4ump | D | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2516 | |
| MELK | CAMKL | CAMK | 4d2w | C | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2527 | |
| MELK | CAMKL | CAMK | 5k00 | A | B | 4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamide | Human | 7498 | |
| MELK | CAMKL | CAMK | 4d2w | D | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2481 | |
| MELK | CAMKL | CAMK | 4bl1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2519 | |
| MELK | CAMKL | CAMK | 5ihc | A | B | 4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridine | Human | 6662 | |
| MELK | CAMKL | CAMK | 4d2t | D | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2530 | |
| MELK | CAMKL | CAMK | 4d2v | A | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2493 | |
| MELK | CAMKL | CAMK | 4d2p | B | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2498 | |
| MELK | CAMKL | CAMK | 4d2w | B | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2500 | |
| MELK | CAMKL | CAMK | 5ih9 | A | A | 1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazine | Human | 6659 | |
| MELK | CAMKL | CAMK | 4umu | A | | (2-ethoxy-4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}phenyl)methanaminium | Human | 2517 | |
| MELK | CAMKL | CAMK | 4d2p | B | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2494 | |
| MELK | CAMKL | CAMK | 5mai | A | B | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 8730 | |
| MELK | CAMKL | CAMK | 6gvx | B | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11136 | |
| MELK | CAMKL | CAMK | 5twy | A | | 2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 8671 | |
| MELK | CAMKL | CAMK | 4d2v | B | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2483 | |
| MELK | CAMKL | CAMK | 4umq | A | A | 3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminium | Human | 2488 | |
| MELK | CAMKL | CAMK | 4d2t | C | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2491 | |
| MELK | CAMKL | CAMK | 5mah | A | B | ~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide | Human | 8734 | |
| MELK | CAMKL | CAMK | 4bky | A | A | 3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamide | Human | 2480 | |
| MELK | CAMKL | CAMK | 4d2t | C | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2526 | |
| MELK | CAMKL | CAMK | 4d2w | A | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2509 | |
| MELK | CAMKL | CAMK | 4ump | A | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2485 | |
| MELK | CAMKL | CAMK | 5twu | A | | - | Human | 8670 | |
| MELK | CAMKL | CAMK | 5tx3 | A | | 7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-one | Human | 8673 | |
| MELK | CAMKL | CAMK | 4bl1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2514 | |
| MELK | CAMKL | CAMK | 4d2v | C | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2492 | |
| MELK | CAMKL | CAMK | 4umt | A | | 1-(4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}-2-methoxybenzyl)piperazinediium | Human | 2510 | |
| MELK | CAMKL | CAMK | 5mag | A | B | pf-3758309 | Human | 8731 | |
| MELK | CAMKL | CAMK | 4ump | B | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2524 | |
| MELK | CAMKL | CAMK | 4d2v | C | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2529 | |
| MELK | CAMKL | CAMK | 4d2p | A | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2499 | |
| MELK | CAMKL | CAMK | 4d2t | D | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2511 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | A | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | 1609 | |
| STK11 (LKB1) | CAMKL | CAMK | 2wtk | F | | phosphoaminophosphonic acid-adenylate ester | Human | 1869 | |
| STK11 (LKB1) | CAMKL | CAMK | 2wtk | C | | phosphoaminophosphonic acid-adenylate ester | Human | 1868 | |
| PASK | CAMKL | CAMK | 3dls | F | | adenosine-5'-diphosphate | Human | 3380 | |
| PASK | CAMKL | CAMK | 3dls | C | | adenosine-5'-diphosphate | Human | 3377 | |
| PASK | CAMKL | CAMK | 3dls | E | | adenosine-5'-diphosphate | Human | 3379 | |
| PASK | CAMKL | CAMK | 3dls | D | | adenosine-5'-diphosphate | Human | 3378 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9g | A | | staurosporine | Human | 10715 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4red | B | | - | Human | 123 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9f | A | | staurosporine | Human | 10716 | |
| SNRK | CAMKL | CAMK | 5yks | B | | - | Human | 8661 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 2h6d | A | B | - | Human | 194 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | A | B | staurosporine | Human | 6428 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | A | B | staurosporine | Human | 9849 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 3aqv | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 193 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cfe | A | | staurosporine | Human | 195 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | C | A | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6427 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | A | A | staurosporine | Human | 9848 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | C | A | staurosporine | Human | 6430 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cff | C | | staurosporine | Human | 190 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 2h6d | A | A | - | Human | 196 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | C | B | staurosporine | Human | 6426 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | A | A | staurosporine | Human | 6424 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b2e | A | | staurosporine | Human | 9851 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | A | B | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6429 | |