Search results (1251 entries covering 663 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
CDK2CDKCMGC9espAB4-bromo-1-(2-methoxyethyl)-1h-pyrazoleHuman15901
CDK2CDKCMGC2wxvCn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4504
CDK2CDKCMGC5anoA-Human6537
CDK2CDKCMGC4eopAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4258
CDK2CDKCMGC3rakAB4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4331
CDK2CDKCMGC9et2AB~{n}-(4-bromophenyl)ethanamideHuman15902
CDK2CDKCMGC8ru8AA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman15329
CDK2CDKCMGC3unkA4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman4374
CDK2CDKCMGC2vu3AB4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman3884
CDK2CDKCMGC1r78AA4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman4253
CDK2CDKCMGC1h00AB(2r)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4428
CDK2CDKCMGC2ds1A(13r,15s)-13-methyl-16-oxa-8,9,12,22,24-pentaazahexacyclo[15.6.2.16,9.1,12,15.0,2,7.0,21,25]heptacosa-1(24),2,4,6,17(25),18,20-heptaene-23,26-dioneHuman4513
CDK2CDKCMGC4ek5ABn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHuman4145
CDK2CDKCMGC9eszAD5-iodanylpyrimidineHuman15903
CDK1 (CDC2)CDKCMGC6gu6A3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman10774
CDK2CDKCMGC2wevCA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4503
CDK2CDKCMGC6q4fABpyridine-2,6-diamineHuman11211
CDK2CDKCMGC2uzoA4-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3862
CDK1 (CDC2)CDKCMGC4yc6EA-Human4612
CDK1 (CDC2)CDKCMGC6gu4A~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10777
CDK2CDKCMGC3s0oAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHuman4123
CDK2CDKCMGC3qhwCBadenosine-5'-diphosphateHuman4143
CDK2CDKCMGC4fx3AB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman3931
CDK2CDKCMGC3qhwABadenosine-5'-diphosphateHuman4156
CDK2CDKCMGC4cfxAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4086
CDK2CDKCMGC3qqhAA2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenolHuman4393
CDK2CDKCMGC3raiAA4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4441
CDK2CDKCMGC3sqqAB4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3925
CDK2CDKCMGC6gueC4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10772
CDK2CDKCMGC1fvvA4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman4065
CDK2CDKCMGC1pxoAB-Human3860
CDK2CDKCMGC3r9hAB4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4336
CDK2CDKCMGC1e1vA6-o-cyclohexylmethyl guanineHuman3886
CDK2CDKCMGC4bcnCA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4436
CDK2CDKCMGC4eolAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4089
CDK2CDKCMGC4kd1AA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman4585
CDK2CDKCMGC4bcpCA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman3872
CDK2CDKCMGC4bcnAB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4298
CDK2CDKCMGC1h1sCo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4572
CDK2CDKCMGC3ti1AAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4201
CDK1 (CDC2)CDKCMGC5hq0AB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman6421
CDK2CDKCMGC4cfmAA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4207
CDK2CDKCMGC5ievABroniciclibHuman6570
CDK2CDKCMGC4eosCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4008
CDK2CDKCMGC1pxkAB-Human3980
CDK2CDKCMGC3tnwCB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman4493
CDK2CDKCMGC4fksAAn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4412
CDK8CDKCMGC6qtjA~{n},~{n}-dimethyl-2-[4-[4-(2,6-naphthyridin-4-yl)phenyl]pyrazol-1-yl]ethanamideHuman12093
CDK8CDKCMGC5hvyABn-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}ureaHuman6552
CDK2CDKCMGC1urcCA-Human4006
CDK2CDKCMGC1pxoAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4512
CDK2CDKCMGC6guhAB4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10769
CDK2CDKCMGC2c5xCBhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4418
CDK2CDKCMGC2cchCC-Human4431
CDK2CDKCMGC1ke9A3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4250
CDK2CDKCMGC2b54A6-(3,4-dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4(5h)-oneHuman4292
CDK2CDKCMGC2iw8ABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4377
CDK2CDKCMGC2bhhA(2e,3s)-3-hydroxy-5'-[(4-hydroxypiperidin-1-yl)sulfonyl]-3-methyl-1,3-dihydro-2,3'-biindol-2'(1'h)-oneHuman4417
CDK2CDKCMGC3r8vAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3938
CDK2CDKCMGC3bhuAB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4446
CDK2CDKCMGC4fkoAB2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHuman4534
CDK2CDKCMGC4eoiCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4011
CDK2CDKCMGC2c5vAA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4012
CDK2CDKCMGC4fx3CA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4349
CDK2CDKCMGC3qqkAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4568
CDK2CDKCMGC1oiuCB3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4049
CDK2CDKCMGC1h1qC2-anilino-6-cyclohexylmethoxypurineHuman4053
CDK2CDKCMGC1e9hA2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHuman4302
CDK4CDKCMGC7sj3An-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman14485
CDK2CDKCMGC2r3qAA3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman4038
CDK5CDKCMGC4au8AB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2786
CDK2CDKCMGC2c5nCBn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman3903
CDK2CDKCMGC7ackCA8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13450
CDK2CDKCMGC2xnbAA3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHuman4217
CDK2CDKCMGC6q49AC-Human11193
CDK2CDKCMGC2wfyAA-Human4324
CDK2CDKCMGC4bcpAB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4304
CDK2CDKCMGC4i3zCadenosine-5'-diphosphateHuman3961
CDK2CDKCMGC2r3nAB3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4046
CDK2CDKCMGC3qtqAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4103
CDK2CDKCMGC9esuAC-Human15904
CDK2CDKCMGC6q4aAB5-iodanylpyrimidineHuman11200
CDK2CDKCMGC2fvdA(4-amino-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrimidin-5-yl)(2,3-difluoro-6-methoxyphenyl)methanoneHuman4408
CDK2CDKCMGC6ylkABmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12494
CDK2CDKCMGC3qx4AA4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4409
CDK2CDKCMGC1e1xA6-cyclohexylmethyloxy-5-nitroso-pyrimidine-2,4-diamineHuman4114
CDK2CDKCMGC4cfvAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman4328
CDK2CDKCMGC2bpmC(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHuman4128
CDK5CDKCMGC1h4lA-Human2788
CDK5CDKCMGC7vdrA(1r)-1-[7-[(2-fluoranyl-4-pyrazol-1-yl-phenyl)amino]-1,6-naphthyridin-2-yl]-1-(1-methylpiperidin-4-yl)ethanolHuman14146
CDK2CDKCMGC3eidCA-Human4072
CDK2CDKCMGC2r3kAA3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman3953
CDK2CDKCMGC3s1hAA4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4068
CDK2CDKCMGC3ddqCAr-roscovitineHuman4364
CDK2CDKCMGC3ralAB4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3984
CDK2CDKCMGC2vttA4-{[(2,6-difluorophenyl)carbonyl]amino}-n-[(3s)-piperidin-3-yl]-1h-pyrazole-3-carboxamideHuman4100
CDK1 (CDC2)CDKCMGC4yc6GA-Human4613
CDK2CDKCMGC1giiA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHuman4448
CDK2CDKCMGC6q4bAB5-bromanylpyrimidineHuman11210
CDK1 (CDC2)CDKCMGC6gu2AB2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10776
CDK2CDKCMGC2r3hAB3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman3970
CDK2CDKCMGC5nevA4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHuman8020
CDK2CDKCMGC5mhqAB(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHuman9408
CDK2CDKCMGC2c5vCA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4384
CDK2CDKCMGC3rprAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanoneHuman4241
CDK8CDKCMGC4f7jAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)ureaHuman3842
CDK2CDKCMGC7rwfA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHuman14344
CDK2CDKCMGC4ek4AC4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman4369
CDK2CDKCMGC2c5yABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman6777
CDK2CDKCMGC2wmbC-Human4474
CDK2CDKCMGC3qtuAA4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4009
CDK2CDKCMGC3dogCA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4382
CDK2CDKCMGC2cjmAadenosine-5'-triphosphateHuman4406
CDK2CDKCMGC4eokAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3913
CDK2CDKCMGC2vtrAA5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4391
CDK2CDKCMGC3eidCB-Human4467
CDK2CDKCMGC3pj8AB(2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-olHuman4454
CDK2CDKCMGC2c5vAB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4338
CDK2CDKCMGC4bcmAA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4290
CDK2CDKCMGC2r3rAB3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4215
CDK2CDKCMGC7m2fAB[(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acidHuman13796
CDK2CDKCMGC3tnwCA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3940
CDK2CDKCMGC3qhwCAadenosine-5'-diphosphateHuman4129
CDK2CDKCMGC2wfyCB-Human4096
CDK2CDKCMGC2wevCC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4288
CDK2CDKCMGC3ddpCB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6778
CDK2CDKCMGC1jsvA4-[(6-amino-4-pyrimidinyl)amino]benzenesulfonamideHuman4171
CDK2CDKCMGC3qtzAA4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4109
CDK2CDKCMGC1pxnAA4-[4-(4-methyl-2-methylamino-thiazol-5-yl)-pyrimidin-2-ylamino]-phenolHuman4383
CDK2CDKCMGC1h0wAB1-amino-6-cyclohex-3-enylmethyloxypurineHuman4016
CDK2CDKCMGC3r9dAA4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4562
CDK1 (CDC2)CDKCMGC6gu7G-Human10779
CDK2CDKCMGC2cchAAadenosine-5'-triphosphateHuman4303
CDK2CDKCMGC2cchCAadenosine-5'-triphosphateHuman3932
CDK2CDKCMGC1fvvC4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman4461
CDK2CDKCMGC6q4dAB2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11215
CDK2CDKCMGC4eoqCBadenosine-5'-triphosphateHuman3912
CDK2CDKCMGC1ol1C-Human3951
CDK2CDKCMGC3rzbAB4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamideHuman4395
CDK16 (PCTAIRE1)CDKCMGC3mtlAB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human1702
CDK2CDKCMGC6q4kAA-Human11179
CDK2CDKCMGC1h27C-Human4030
CDK2CDKCMGC1oiuAB3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4556
CDK2CDKCMGC4eorABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3934
CDK2CDKCMGC4bcmCB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4124
CDK2CDKCMGC3pxqA8-anilino-1-naphthalene sulfonateHuman3947
CDK2CDKCMGC1h0vAB5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHuman3933
CDK2CDKCMGC1w8cAA6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHuman4332
CDK2CDKCMGC4eokCo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4385
CDK2CDKCMGC3qtwAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman3890
CDK2CDKCMGC4bckAB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman3960
CDK2CDKCMGC4eooAAadenosine-5'-triphosphateHuman4403
CDK2CDKCMGC2c6mA4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6782
CDK2CDKCMGC3qwjAB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamideHuman4182
CDK1 (CDC2)CDKCMGC6gu7A4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10781
CDK16 (PCTAIRE1)CDKCMGC5g6vB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman7274
CDK2CDKCMGC7ackAA8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13451
CDK2CDKCMGC7s4tAA2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHuman14374
CDK2CDKCMGC2r3lAC3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4496
CDK2CDKCMGC7s4tAB2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHuman14373
CDK2CDKCMGC8h6pA(7s,10r)-11-oxa-2,4,5,13,17,23-hexaazatetracyclo[17.3.1.1~3,6~.1~7,10~]pentacosa-1(23),3(25),5,19,21-pentaene-12,18-dioneHuman14625
CDK2CDKCMGC5nevC4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHuman8019
CDK2CDKCMGC3rm6AB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamideHuman4357
CDK2CDKCMGC8h6tA(1r,3s)-3-{3-[(pyridin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl propan-2-ylcarbamateHuman14626
CDK2CDKCMGC4fktABn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4322
CDK2CDKCMGC6p3wAA-Human11515
CDK2CDKCMGC2c5nAAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4063
CDK2CDKCMGC7m2fAA[(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acidHuman13797
CDK2CDKCMGC1urcAA-Human4334
CDK2CDKCMGC6p3wCA-Human11514
CDK2CDKCMGC7ra5AB4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman13959
CDK2CDKCMGC3qtzAB4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4337
CDK2CDKCMGC6rijAA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12623
CDK2CDKCMGC4ez7AstaurosporineHuman4240
CDK2CDKCMGC1di8A4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman4577
CDK2CDKCMGC3rahAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman4438
CDK2CDKCMGC2uzlA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHuman3917
CDK2CDKCMGC3lfsAn-(6-chloro-5-phenyl-1h-indazol-3-yl)butanamideHuman4069
CDK2CDKCMGC4fklAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4134
CDK2CDKCMGC1oiqAn-[4-(2-methylimidazo[1,2-a]pyridin-3-yl)-2-pyrimidinyl]acetamideHuman4379
CDK2CDKCMGC4eomAAadenosine-5'-triphosphateHuman4528
CDK2CDKCMGC2w05ABn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHuman4256
CDK2CDKCMGC2vu3AA4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman4582
CDK2CDKCMGC6q4eAB6-iodanyl-7~{h}-purin-2-amineHuman11205
CDK2CDKCMGC1h00AA(2s)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4484
CDK9CDKCMGC7nwkAn-((1r,3r)-3-(7-(4-fluoro-2-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-2-yl)cyclopentyl)acetamideHuman13951
CDK2CDKCMGC2c5xABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman3892
CDK2CDKCMGC3ddqAAr-roscovitineHuman4477
CDK2CDKCMGC1vywCn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamideHuman4133
CDK2CDKCMGC2c5oCA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4414
CDK2CDKCMGC7zpcAA~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamideHuman14606
CDK2CDKCMGC7s85A2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethoxy)benzoic acidHuman14425
CDK2CDKCMGC4i3zAadenosine-5'-diphosphateHuman4148
CDK2CDKCMGC7ug1AA8-(4-chloroanilino)naphthalene-1-sulfonic acidHuman14700
CDK2CDKCMGC7ug1AB8-(4-chloroanilino)naphthalene-1-sulfonic acidHuman14701
CDK2CDKCMGC4fkrAA(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman4149
CDK2CDKCMGC1h26A-Human4122
CDK2CDKCMGC5ieyAA4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHuman6566
CDK2CDKCMGC6gubA2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10764
CDK2CDKCMGC3qzhA4-methoxy-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3954
CDK2CDKCMGC2wmbA-Human4060
CDK2CDKCMGC3rmfAA4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3873
CDK2CDKCMGC6q4iAA2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHuman11183
CDK2CDKCMGC6rijCA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12625
CDK2CDKCMGC3r6xAB4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4107
CDK2CDKCMGC1e9hC2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHuman4570
CDK2CDKCMGC1b39Aadenosine-5'-triphosphateHuman4407
CDK2CDKCMGC5oo3AA1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHuman10569
CDK2CDKCMGC2v22C-Human4255
CDK2CDKCMGC3py1AB(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman4444
CDK2CDKCMGC2bpmA(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHuman4042
CDK12 (CRK7)CDKCMGC7nxkA(e)-n-[4-[(1r,3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]cyclohexyl]oxyphenyl]-4-(dimethylamino)but-2-enamideHuman13547
CDK2CDKCMGC2cciAadenosine-5'-triphosphateHuman4373
CDK2CDKCMGC1ke6An-methyl-{4-[2-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)hydrazino]phenyl}methanesulfonamideHuman4219
CDK2CDKCMGC1oguAB4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3935
CDK2CDKCMGC7b7sAA7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxideHuman13833
CDK2CDKCMGC2r3lAA3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4200
CDK9CDKCMGC8i0lA2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman15170
CDK2CDKCMGC6gukAA~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10773
CDK2CDKCMGC2w1hAn-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamideHuman4228
CDK2CDKCMGC4cfwAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4557
CDK2CDKCMGC3my5CC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3929
CDK2CDKCMGC2uznA4-{5-[(1z)-1-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)ethyl]-2-furyl}benzenesulfonamideHuman4064
CDK2CDKCMGC3sw7AAn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHuman4198
CDK2CDKCMGC4bcoAB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4051
CDK2CDKCMGC3lfnAn-[6-(4-hydroxyphenyl)-5-phenyl-1h-indazol-3-yl]butanamideHuman4330
CDK2CDKCMGC5ankA2,4,6-trioxo-1-phenyl-hexahydropyrimidine-5-carboxamideHuman6538
CDK2CDKCMGC3rmfAB4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4014
CDK2CDKCMGC3qtxAA4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4339
CDK2CDKCMGC1h1rAA6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman3906
CDK2CDKCMGC4cfnAB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4437
CDK2CDKCMGC4eomCAadenosine-5'-triphosphateHuman4481
CDK2CDKCMGC2wevAB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4580
CDK2CDKCMGC7kjsA6-(difluoromethyl)-8-[(1r,2r)-2-hydroxy-2-methylcyclopentyl]-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman13740
CDK2CDKCMGC7b7sAB7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxideHuman13834
CDK2CDKCMGC1pxlAB-Human4074
CDK2CDKCMGC3eocA5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman4390
CDK2CDKCMGC4bckCD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4080
CDK2CDKCMGC7mkxA2-[(5-bromo-2-{4-[(cyanomethyl)sulfamoyl]anilino}pyrimidin-4-yl)amino]-6-fluorobenzamideHuman14490
CDK2CDKCMGC1jvpP13-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazoleHuman3919
CDK2CDKCMGC2vtoABn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHuman3946
CDK2CDKCMGC3rniAA3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman3993
CDK2CDKCMGC3ralAA4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4017
CDK2CDKCMGC4eojABadenosine-5'-triphosphateHuman4015
CDK2CDKCMGC3py1AA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman4361
CDK1 (CDC2)CDKCMGC4y72AA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4610
CDK2CDKCMGC6q4iAB2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHuman11197
CDK2CDKCMGC1oiuCA3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4524
CDK16 (PCTAIRE1)CDKCMGC9r2iCphosphothiophosphoric acid-adenylate esterHuman15481
CDK2CDKCMGC3r7yAA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamideHuman4476
CDK2CDKCMGC4ii5CAadenosine-5'-diphosphateHuman4530
CDK2CDKCMGC1oiyCA4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4465
CDK2CDKCMGC1pxiAB-Human3924
CDK2CDKCMGC5andA2-imidazol-1-yl-1h-benzimidazoleHuman6543
CDK2CDKCMGC4bcoCB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4018
CDK7CDKCMGC8p4zAA2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHuman14796
CDK7CDKCMGC8p4zAB2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHuman14797
CDK2CDKCMGC8uv0AA1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-olHuman15238
CDK2CDKCMGC3r9nAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3885
CDK2CDKCMGC8uv0AB1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-olHuman15239
CDK1 (CDC2)CDKCMGC4yc6AA-Human4607
CDK2CDKCMGC4fkvAB(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHuman3939
CDK2CDKCMGC3qx2AB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamideHuman4297
CDK2CDKCMGC1gy3Cadenosine-5'-triphosphateHuman4445
CDK2CDKCMGC5jq8A(3s,4s)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman7417
CDK2CDKCMGC3rm6AA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamideHuman4262
CDK2CDKCMGC7qhlAA5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidineHuman14275
CDK2CDKCMGC3qqjAB2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4204
CDK2CDKCMGC3qqgAB4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4310
CDK2CDKCMGC3qqfAA5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4211
CDK2CDKCMGC2iw8CBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4350
CDK7CDKCMGC8pyrAB-Human15253
CDK2CDKCMGC2c4gC(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHuman4453
CDK2CDKCMGC1okwA-Human4314
CDK2CDKCMGC1w0xCAolomoucineHuman4537
CDK2CDKCMGC6gukAB~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10768
CDK2CDKCMGC2vtnA4-(acetylamino)-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4027
CDK2CDKCMGC2c6tC4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman3994
CDK2CDKCMGC2xmyAB4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHuman3985
CDK2CDKCMGC9qjjBots964Human15914
CDK2CDKCMGC13gkAC-Human15915
CDK2CDKCMGC9nyrAB-Human15916
CDK2CDKCMGC9et1AA4-iodanylbenzamideHuman15917
CDK2CDKCMGC9glaAA7-dimethylphosphoryl-3-[2-[[(3~{s})-6,6-dimethylpiperidin-3-yl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]-1~{h}-indole-6-carbonitrileHuman15918
CDK2CDKCMGC9fr2A4-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]benzenesulfonyl fluorideHuman15919
CDK2CDKCMGC9eswAD-Human15920
CDK2CDKCMGC9eskAB(4-bromo-2-oxopyridin-1(2h)-yl)acetic acidHuman15913
CDK2CDKCMGC9esjAA2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman15953
CDK2CDKCMGC9eswAB(4-bromanylpyridin-2-yl)methanolHuman15954
CDK2CDKCMGC9esuAB4-bromanyl-2-(methoxymethyl)pyridineHuman15955
CDK2CDKCMGC9esoAB-Human15956
CDK2CDKCMGC7s7aAA2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14427
CDK2CDKCMGC9esyAA4-bromanyl-1,8-naphthyridineHuman15930
CDK2CDKCMGC9et1AB4-iodanylbenzamideHuman15951
CDK2CDKCMGC9etpAA4-bromo-1h-pyrazoleHuman15952
CDK2CDKCMGC2r3kAB3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman3876
CDK2CDKCMGC7sa0AA2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acidHuman14428
CDK2CDKCMGC7sa0AB2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acidHuman14429
CDK2CDKCMGC7s84AB2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14432
CDK2CDKCMGC9nyqA4-({4-[(1s,4s)-4-hydroxy-4-methylcyclohexyl]-5-(trifluoromethyl)pyrimidin-2-yl}amino)-n,3-dimethylbenzene-1-sulfonamideHuman15957
CDK2CDKCMGC9gp3A(3~{s})-~{n}-ethyl-3-[[9-ethyl-2-[[(2~{r},3~{s})-2-oxidanylpentan-3-yl]amino]purin-6-yl]amino]pyrrolidine-1-sulfonamideHuman15958
CDK2CDKCMGC9esqAA4-bromanyl-2-oxidanyl-benzoic acidHuman15959
CDK2CDKCMGC7s9xAA2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acidHuman14430
CDK9CDKCMGC32awA4-[[[6-[5-chloranyl-2-[[4-[[(2~{r})-1-methoxypropan-2-yl]amino]phenyl]amino]pyridin-4-yl]pyridin-2-yl]amino]methyl]oxane-4-carbonitrileHuman15994
CDK13 (CHED)CDKCMGC7nxjAn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman13544
CDK2CDKCMGC3pxrAA-Human3941
CDK2CDKCMGC7s7aAB2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14426
CDK2CDKCMGC2clxAA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3909
CDK2CDKCMGC4eojAAadenosine-5'-triphosphateHuman4271
CDK2CDKCMGC4eomCBadenosine-5'-triphosphateHuman4423
CDK2CDKCMGC3r71AA4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3962
CDK2CDKCMGC1pxoAC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4546
CDK2CDKCMGC4eopCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4061
CDK2CDKCMGC3r8lAB(5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4523
CDK2CDKCMGC6athAB-Human10570
CDK2CDKCMGC3qqgAA4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4130
CDK2CDKCMGC4bckCC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4029
CDK2CDKCMGC7qhlAB5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidineHuman14276
CDK2CDKCMGC4eolCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4521
CDK2CDKCMGC6q4kAC-Human11189
CDK1 (CDC2)CDKCMGC4yc6EB-Human4614
CDK7CDKCMGC1ua2Cadenosine-5'-triphosphateHuman542
CDK7CDKCMGC7b5oJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13278
CDK2CDKCMGC7zpcAB~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamideHuman14607
CDK7CDKCMGC7nvr8-Human13543
CDK2CDKCMGC1fq1Badenosine-5'-triphosphateHuman4266
CDK2CDKCMGC4cfvAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman4180
CDK8CDKCMGC5hnbAB[6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanoneHuman6563
CDK5CDKCMGC7vdqA2-[[7-[[2-fluoranyl-4-[3-(hydroxymethyl)pyrazol-1-yl]phenyl]amino]-1,6-naphthyridin-2-yl]-(1-methylpiperidin-4-yl)amino]ethanoic acidHuman14144
CDK5CDKCMGC7vdsAA5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHuman14148
CDK5CDKCMGC1unhA(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2780
CDK5CDKCMGC3o0gA-Human2782
CDK5CDKCMGC1unlB-Human2790
CDK2CDKCMGC7rxoAB2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acidHuman14351
CDK2CDKCMGC7uxkA-Human14570
CDK2CDKCMGC7uxiAA-Human14571
CDK2CDKCMGC7rxoAA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acidHuman14352
CDK2CDKCMGC7uxiAB-Human14572
CDK2CDKCMGC7vduAB[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14137
CDK2CDKCMGC1gz8AB1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHuman3956
CDK2CDKCMGC4eojCAadenosine-5'-triphosphateHuman4041
CDK2CDKCMGC4fkrAB(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman4535
CDK2CDKCMGC3eidAA(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4386
CDK2CDKCMGC6p3wAB-Human11517
CDK2CDKCMGC4bcmAB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4203
CDK2CDKCMGC1h24A-Human4199
CDK2CDKCMGC1oguCB4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman4560
CDK2CDKCMGC4bghAB4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHuman4509
CDK16 (PCTAIRE1)CDKCMGC5g6vA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman7273
CDK2CDKCMGC2c6iA4-{[5-(cyclohexylmethoxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6774
CDK2CDKCMGC2wfyCA-Human4329
CDK2CDKCMGC3r8lAA(5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4186
CDK2CDKCMGC1gihA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHuman3922
CDK2CDKCMGC1f5qCA-Human4281
CDK2CDKCMGC8erdAA(2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanoneHuman14949
CDK2CDKCMGC8ernAAn,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamideHuman14948
CDK2CDKCMGC8ernABn,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamideHuman14950
CDK2CDKCMGC3pxfAA8-anilino-1-naphthalene sulfonateHuman4047
CDK2CDKCMGC8erdAB(2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanoneHuman14951
CDK2CDKCMGC4eoqCAadenosine-5'-triphosphateHuman4004
CDK2CDKCMGC5fp5A4-fluorobenzoic acidHuman6285
CDK2CDKCMGC2vtjA4-[(6-chloropyrazin-2-yl)amino]benzenesulfonamideHuman3959
CDK2CDKCMGC7s9xAB2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acidHuman14431
CDK2CDKCMGC6gufCn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman10762
CDK2CDKCMGC2uzbAD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman3866
CDK2CDKCMGC6gvaAB5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman11204
CDK2CDKCMGC2c6kA4-{[5-(cyclohexylamino)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6773
CDK2CDKCMGC1pkdA7-hydroxystaurosporineHuman4170
CDK2CDKCMGC6q48AC4-iodanyl-3~{h}-pyridin-2-oneHuman11196
CDK2CDKCMGC6q3bAA4-iodopyrazoleHuman11177
CDK2CDKCMGC1h25C-Human4112
CDK2CDKCMGC3pj8AA(2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-olHuman4375
CDK2CDKCMGC2c5xAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4312
CDK2CDKCMGC3sw7ABn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHuman4584
CDK2CDKCMGC3rahAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman4206
CDK2CDKCMGC1pxmAA3-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-ylamino]-phenolHuman3944
CDK2CDKCMGC4bghAA4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHuman4073
CDK2CDKCMGC3bhvCA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4353
CDK2CDKCMGC2x1nCB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4062
CDK8CDKCMGC5fgkAB8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6388
CDK2CDKCMGC3qrtAA(5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4586
CDK2CDKCMGC3rakAA4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4574
CDK8CDKCMGC4f70A1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[2-(morpholin-4-yl)ethyl]ureaHuman3852
CDK6CDKCMGC3nuxA4-[5-chloro-3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineHuman2807
CDK8CDKCMGC5xqxAn-methyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHuman8313
CDK6CDKCMGC5l2tA7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman6992
CDK2CDKCMGC5ievAAroniciclibHuman6567
CDK2CDKCMGC3qqhAB2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenolHuman4533
CDK2CDKCMGC3rkbAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4039
CDK2CDKCMGC4ek6ABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHuman4056
CDK2CDKCMGC4eorCAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4221
CDK2CDKCMGC3r83AA4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4234
CDK2CDKCMGC2clxAB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3880
CDK2CDKCMGC5uq2A-Human8221
CDK2CDKCMGC3r1sAB2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4358
CDK2CDKCMGC3pxyAB2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenolHuman3904
CDK2CDKCMGC6q3fAA-Human11181
CDK2CDKCMGC3qx4AB4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3990
CDK2CDKCMGC5cyiAA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6052
CDK2CDKCMGC4cfxAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4485
CDK2CDKCMGC3r6xAA4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4398
CDK2CDKCMGC2g9xA3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-olHuman3883
CDK2CDKCMGC3r8vAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman4191
CDK2CDKCMGC2a4lAr-roscovitineHuman4238
CDK2CDKCMGC3s00AB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHuman4248
CDK2CDKCMGC1ke5An-methyl-4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4376
CDK2CDKCMGC4nj3AA6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman4075
CDK2CDKCMGC1gy3Aadenosine-5'-triphosphateHuman3978
CDK2CDKCMGC1jstCadenosine-5'-triphosphateHuman4356
CDK2CDKCMGC1h1pA6-o-cyclohexylmethyl guanineHuman4309
CDK2CDKCMGC9esjAB2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman15905
CDK2CDKCMGC9esyAB4-bromanyl-1,8-naphthyridineHuman15906
CDK2CDKCMGC6rijCB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12622
CDK2CDKCMGC7s84AA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14424
CDK2CDKCMGC6q4jAA2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHuman11209
CDK2CDKCMGC2bheA(2z)-5'-bromo-2,3'-biindole-2',3(1h,1'h)-dione ammoniateHuman4184
CDK2CDKCMGC1ol2C-Human4497
CDK2CDKCMGC6q4cAB4-bromanyl-1,8-naphthyridineHuman11207
CDK2CDKCMGC4rj3AB1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4127
CDK2CDKCMGC1pf8A(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3861
CDK2CDKCMGC1hclAA-Human4545
CDK2CDKCMGC1b38Aadenosine-5'-triphosphateHuman4483
CDK2CDKCMGC1g5sA2-[trans-(4-aminocyclohexyl)amino]-6-(benzyl-amino)-9-cyclopentylpurineHuman3888
CDK2CDKCMGC4ek3AA-Human3971
CDK2CDKCMGC3r8uAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman3926
CDK2CDKCMGC4eoiAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4307
CDK2CDKCMGC1h1rAB6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman4494
CDK2CDKCMGC4eonAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4326
CDK2CDKCMGC3qtxAB4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4419
CDK2CDKCMGC4cfuAB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman4308
CDK2CDKCMGC6q4cAC4-bromanyl-1,8-naphthyridineHuman11201
CDK2CDKCMGC5anjAn-(9h-purin-6-yl)thiophene-2-carboxamideHuman6541
CDK8CDKCMGC6tpaA1-[4-chloranyl-3-(trifluoromethyl)phenyl]-3-(5-oxidanylidene-6-pyridin-4-yl-pyrido[2,3-b][1,5]benzoxazepin-9-yl)ureaHuman13160
CDK2CDKCMGC2v22A-Human4077
CDK2CDKCMGC7b5rL-Human13265
CDK2CDKCMGC4fkiABn-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamideHuman4272
CDK8CDKCMGC5xs2AB3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHuman8314
CDK2CDKCMGC2iw6A[(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrileHuman4019
CDK8CDKCMGC4crlAcortistatin aHuman6096
CDK8CDKCMGC4g6lA-Human3851
CDK2CDKCMGC4eonCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4153
CDK8CDKCMGC5idpAA(3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanoneHuman7317
CDK8CDKCMGC5fgkAA8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6391
CDK8CDKCMGC6r3sAB6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman12141
CDK8CDKCMGC5hvyAAn-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}ureaHuman6553
CDK2CDKCMGC8byaA-Human14814
CDK2CDKCMGC8bzoA-Human14815
CDK2CDKCMGC3rniAB3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4420
CDK2CDKCMGC3qhrAadenosine-5'-diphosphateHuman4458
CDK2CDKCMGC2v0dA2-imino-5-(1-pyridin-2-yl-meth-(e)-ylidene)-1,3-thiazolidin-4-oneHuman4327
CDK2CDKCMGC2wihAn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4163
CDK2CDKCMGC5oo1A~{n}-(4-pyrimidin-2-ylphenyl)propanamideHuman10566
CDK8CDKCMGC5hbjAA8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6390
CDK8CDKCMGC4f6uAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]ureaHuman3849
CDK8CDKCMGC4f7jAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)ureaHuman3843
CDK8CDKCMGC4f7sABn-(2-phenylethyl)quinazolin-4-amineHuman3853
CDK8CDKCMGC5bnjA8-{3-chloro-5-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]pyridin-4-yl}-2,8-diazaspiro[4.5]decan-1-oneHuman6152
CDK9CDKCMGC6cytA-Human10797
CDK9CDKCMGC4bciA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman2243
CDK9CDKCMGC3miaAphosphoaminophosphonic acid-adenylate esterHuman2242
CDK9CDKCMGC3mi9A-Human2239
CDK2CDKCMGC3ddpAB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6780
CDK2CDKCMGC5aneA6-methoxy-9h-purineHuman6542
CDK2CDKCMGC1h1qA2-anilino-6-cyclohexylmethoxypurineHuman4195
CDK2CDKCMGC3ezvA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman4083
CDK8CDKCMGC3rgfAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3841
CDK9CDKCMGC4ogrIadenosineHuman2241
CDK8CDKCMGC5hnbAA[6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanoneHuman6562
CDK8CDKCMGC6qtgA2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]-~{n},~{n}-dimethyl-ethanamideHuman12094
CDK2CDKCMGC1h1sAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4400
CDK8CDKCMGC4f7nA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(5-hydroxypentyl)ureaHuman3847
CDK9CDKCMGC3tn8A4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman2240
CDK9CDKCMGC4ec9A-Human2234
CDK9CDKCMGC4imyABadenosine monophosphateHuman2252
CDK9CDKCMGC5l1zA-Human7121
CDK9CDKCMGC6w9eAA(4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13859
CDK8CDKCMGC5i5zAn-methyl-8-(1-methyl-2,2-dioxo-2,3-dihydro-1h-2lambda~6~,1-benzothiazol-5-yl)-1,6-naphthyridine-2-carboxamideHuman6536
CDK8CDKCMGC5idnAA[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanoneHuman7322
CDK9CDKCMGC6z45A(1~{s},3~{r})-3-acetamido-~{n}-[5-chloranyl-4-(5,5-dimethyl-4,6-dihydropyrrolo[1,2-b]pyrazol-3-yl)pyridin-2-yl]cyclohexane-1-carboxamideHuman13115
CDK9CDKCMGC3blrA2-(2-chloro-phenyl)-5,7-dihydroxy-8-(3-hydroxy-1-methyl-piperidin-4-yl)-4h-benzopyran-4-oneHuman2236
CDK2CDKCMGC3r8zAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanoneHuman4137
CDK8CDKCMGC5hbhA5-[5-chloranyl-4-[1-(2-methoxyethyl)-1,8-diazaspiro[4.5]decan-8-yl]pyridin-3-yl]-1-methyl-3~{h}-2,1-benzothiazole 2,2-dioxideHuman6387
CDK8CDKCMGC5icpAB[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanoneHuman7321
CDK8CDKCMGC6y0aAA6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman13306
CDK8CDKCMGC5hbeAA8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-oneHuman6389
CDK2CDKCMGC1vyzAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzamideHuman4325
CDK9CDKCMGC4imyEBadenosine monophosphateHuman2256
CDK9CDKCMGC6gzhA[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHuman10427
CDK9CDKCMGC3blqAadenosine-5'-triphosphateHuman2248
CDK9CDKCMGC6w9eAC(4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13861
CDK2CDKCMGC2x1nAB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4078
CDK1 (CDC2)CDKCMGC5lqfAAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7364
CDK1 (CDC2)CDKCMGC4yc6AB-Human4616
CDK1 (CDC2)CDKCMGC5lqfDBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7367
CDK1 (CDC2)CDKCMGC6gu7C-Human10775
CDK1 (CDC2)CDKCMGC4yc3AB-Human6554
CDK2CDKCMGC4ii5AAadenosine-5'-diphosphateHuman3930
CDK2CDKCMGC4eosCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4181
CDK2CDKCMGC2r3iAC-Human4317
CDK2CDKCMGC3ql8AB3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrileHuman4306
CDK2CDKCMGC3r8uAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman3864
CDK2CDKCMGC3tizA1-{(e)-[(4-hydroxyphenyl)imino]methyl}naphthalen-2-olHuman4136
CDK2CDKCMGC4eosAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4340
CDK2CDKCMGC3qtuAB4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4323
CDK1 (CDC2)CDKCMGC4yc6CB-Human4611
CDK2CDKCMGC3ej1Cn-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHuman4092
CDK2CDKCMGC3qqkAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4514
CDK5CDKCMGC1unhB(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2787
CDK2CDKCMGC2vtiAn-(4-sulfamoylphenyl)-1h-indazole-3-carboxamideHuman4177
CDK2CDKCMGC3r8pAA(5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4232
CDK8CDKCMGC4f6sA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman3848
CDK2CDKCMGC3bhuAA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4105
CDK2CDKCMGC1f5qAA-Human4194
CDK2CDKCMGC1ol1A-Human4429
CDK2CDKCMGC6q4hAB2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHuman11190
CDK2CDKCMGC2c6oAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman6783
CDK2CDKCMGC5osmABmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHuman9740
CDK7CDKCMGC7b5qJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13277
CDK5CDKCMGC3o0gB{4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanoneHuman2783
CDK2CDKCMGC3qu0AA4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4427
CDK2CDKCMGC2r3mAAn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHuman4286
CDK2CDKCMGC5oo0AA-Human9744
CDK2CDKCMGC3ig7An-{1-[cis-3-(acetylamino)cyclobutyl]-1h-imidazol-4-yl}-2-(4-methoxyphenyl)acetamideHuman4021
CDK2CDKCMGC3qx2AA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamideHuman4031
CDK2CDKCMGC4eojCBadenosine-5'-triphosphateHuman4311
CDK2CDKCMGC4fkpAB3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4313
CDK2CDKCMGC3qruAB(5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4516
CDK2CDKCMGC2wmaA-Human4435
CDK2CDKCMGC6gucA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman10767
CDK2CDKCMGC2r3gAB6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman3923
CDK2CDKCMGC3r28AB4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamideHuman4293
CDK2CDKCMGC3r1qAB4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4507
CDK2CDKCMGC4bzdAB6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHuman4490
CDK2CDKCMGC4eorAAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4205
CDK2CDKCMGC3rpoAB4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acidHuman4098
CDK2CDKCMGC2wipC1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHuman4190
CDK1 (CDC2)CDKCMGC4yc3AA-Human6555
CDK2CDKCMGC3bhuCA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4087
CDK2CDKCMGC3rjcAB{4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanoneHuman4469
CDK2CDKCMGC1y8yA(5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-(4-methanesulfonylphenyl)amineHuman3914
CDK2CDKCMGC6gubC2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10763
CDK2CDKCMGC4fkjAAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHuman4387
CDK2CDKCMGC4fksABn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4489
CDK2CDKCMGC1h27A-Human4116
CDK2CDKCMGC3r7vAA5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamideHuman4380
CDK2CDKCMGC2c6lA4-({5-[(4-aminocyclohexyl)amino][1,2,4]triazolo[1,5-a]pyrimidin-7-yl}amino)benzenesulfonamideHuman6779
CDK2CDKCMGC1oi9AA6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4033
CDK2CDKCMGC5lmkAB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7398
CDK2CDKCMGC4cfuCA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman3967
CDK2CDKCMGC4cfvCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman3999
CDK2CDKCMGC5uq3A-Human8222
CDK2CDKCMGC6q3cAA4-bromo-1h-pyrazoleHuman11191
CDK2CDKCMGC4erwAstaurosporineHuman4370
CDK2CDKCMGC2i40AB5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4470
CDK2CDKCMGC4ek5AAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHuman4037
CDK2CDKCMGC3eidAB(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4424
CDK2CDKCMGC3rprAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanoneHuman4452
CDK2CDKCMGC5fp6AA3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHuman6302
CDK2CDKCMGC3r1sAA2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4263
CDK2CDKCMGC3qqjAA2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4113
CDK2CDKCMGC3s0oAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHuman3898
CDK2CDKCMGC2g9xC3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-olHuman4082
CDK2CDKCMGC3rjcAA{4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanoneHuman4032
CDK2CDKCMGC2iw6C[(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrileHuman4108
CDK2CDKCMGC6athAA-Human10567
CDK2CDKCMGC1pyeA[2-amino-6-(2,6-difluoro-benzoyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl-methanoneHuman4284
CDK2CDKCMGC2uueC4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHuman4321
CDK2CDKCMGC2r3jAA3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4185
CDK2CDKCMGC1pxiAA4-(2,5-dichlorothien-3-yl)pyrimidin-2-amineHuman4381
CDK2CDKCMGC1okwC-Human3896
CDK2CDKCMGC1pxpAAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4316
CDK2CDKCMGC1pxlAA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4233
CDK2CDKCMGC3le6A5-(2-chlorophenyl)-3-methyl-7-nitropyrazolo[3,4-b][1,4]benzodiazepineHuman4125
CDK8CDKCMGC3rgfAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3846
CDK2CDKCMGC3ns9A(2s,3s)-3-{[7-(benzylamino)-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-5-yl]amino}butane-1,2,4-triolHuman4575
CDK8CDKCMGC5ceiAB4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamideHuman6403
CDK2CDKCMGC5cyiCB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6053
CDK2CDKCMGC3qxpAB4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4482
CDK2CDKCMGC4ek8AA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amineHuman4079
CDK2CDKCMGC3rm7AA2-[(4-hydroxybenzyl)amino]-5-nitrobenzamideHuman3893
CDK2CDKCMGC2uzbAC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4099
CDK2CDKCMGC3pxyAA2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenolHuman4057
CDK2CDKCMGC4cfwAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4280
CDK2CDKCMGC1oi9AB6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4492
CDK2CDKCMGC3qziAA4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamideHuman4094
CDK2CDKCMGC3qrtAB(5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4536
CDK2CDKCMGC5uq1C-Human8223
CDK2CDKCMGC3r7iAA4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acidHuman4450
CDK2CDKCMGC4fklAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4583
CDK2CDKCMGC6yl6AA-Human12498
CDK2CDKCMGC2r3lAB3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4085
CDK2CDKCMGC8fp0ABr-roscovitineHuman14756
CDK2CDKCMGC8fp5ABadenosine-5'-triphosphateHuman14757
CDK2CDKCMGC8fp0AAr-roscovitineHuman14758
CDK2CDKCMGC8fowAA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman14759
CDK2CDKCMGC8fowAB3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman14760
CDK2CDKCMGC8fp5AAadenosine-5'-triphosphateHuman14761
CDK2CDKCMGC3f5xA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman3882
CDK2CDKCMGC3qhrCadenosine-5'-diphosphateHuman3879
CDK2CDKCMGC4bcqCB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4120
CDK2CDKCMGC3bhtAA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman3950
CDK2CDKCMGC2r3rAA3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4040
CDK2CDKCMGC1oguAA4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3965
CDK2CDKCMGC2wevCB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman3859
CDK2CDKCMGC3r8mAA1h-indazole-3-carbohydrazideHuman4111
CDK2CDKCMGC1oiyAA4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4225
CDK2CDKCMGC2j9mAA6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxideHuman4154
CDK1 (CDC2)CDKCMGC5lqfABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7366
CDK2CDKCMGC3py0AA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3995
CDK2CDKCMGC2vv9AB2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHuman3881
CDK2CDKCMGC3qzgAA2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenolHuman4144
CDK2CDKCMGC2vv9AA2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHuman3989
CDK2CDKCMGC1h25A-Human4273
CDK2CDKCMGC3r7eAA5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamideHuman4159
CDK2CDKCMGC2r3nAA3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4101
CDK2CDKCMGC1fvtA4-(5-bromo-2-oxo-2h-indol-3-ylazo)-benzenesulfonamideHuman4480
CDK1 (CDC2)CDKCMGC4y72AB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4609
CDK2CDKCMGC2vtoAAn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHuman4421
CDK2CDKCMGC1ke7A3-{[(2,2-dioxido-1,3-dihydro-2-benzothien-5-yl)amino]methylene}-5-(1,3-oxazol-5-yl)-1,3-dihydro-2h-indol-2-oneHuman4295
CDK2CDKCMGC3bhvCB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4529
CDK2CDKCMGC1h24C-Human4296
CDK2CDKCMGC3bhtCA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4151
CDK2CDKCMGC4ek6AAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHuman4359
CDK2CDKCMGC4fkwAB2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHuman4277
CDK2CDKCMGC3tiyAB2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHuman4488
CDK2CDKCMGC1ol2A-Human4305
CDK2CDKCMGC6q4hAA2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHuman11194
CDK2CDKCMGC2cciCadenosine-5'-triphosphateHuman4532
CDK2CDKCMGC1finCadenosine-5'-triphosphateHuman4479
CDK2CDKCMGC2r3oAC(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4229
CDK5CDKCMGC7vdsAB5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHuman14147
CDK9CDKCMGC4imyAAadenosine monophosphateHuman2238
CDK9CDKCMGC8k5rA(1s,3s)-n3-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamineHuman15081
CDK5CDKCMGC1ungB6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2789
CDK9CDKCMGC4ogrEadenosineHuman2235
CDK2CDKCMGC1gijA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-(5-pyrrolidin-2-yl-1h-pyrazol-3-yl)-ureaHuman4542
CDK2CDKCMGC4eooCBadenosine-5'-triphosphateHuman4139
CDK2CDKCMGC2r3kAC3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman4022
CDK2CDKCMGC4eorCBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4487
CDK2CDKCMGC2vtqA{[(2,6-difluorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman3891
CDK2CDKCMGC9essAA(4-bromo-2-methoxyphenyl)methanolHuman15908
CDK2CDKCMGC4eonAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman3902
CDK2CDKCMGC3s00AA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHuman4208
CDK2CDKCMGC3dogAA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4541
CDK2CDKCMGC4fkqAA4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHuman3972
CDK2CDKCMGC9esjAC2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman15909
CDK2CDKCMGC1dm2AB4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHuman4024
CDK2CDKCMGC2r3pAB5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHuman4392
CDK2CDKCMGC2i40AA5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4363
CDK13 (CHED)CDKCMGC5efqCadenosine-5'-diphosphateHuman6324
CDK2CDKCMGC3eocC5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman3969
CDK2CDKCMGC9essAB(4-bromo-2-methoxyphenyl)methanolHuman15911
CDK2CDKCMGC5d1jAn-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamideHuman4058
CDK2CDKCMGC6q4eAC6-iodanyl-7~{h}-purin-2-amineHuman11219
CDK2CDKCMGC3qtwAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4397
CDK2CDKCMGC2w05AAn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHuman4547
CDK2CDKCMGC5oo3AB1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHuman10568
CDK2CDKCMGC3f5xC4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman3894
CDK2CDKCMGC3ti1ABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4213
CDK2CDKCMGC6q49AB-Human11220
CDK2CDKCMGC2bkzA1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHuman3942
CDK2CDKCMGC4acmAA3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman4247
CDK2CDKCMGC3wblAn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman3895
CDK2CDKCMGC3rm7AB2-[(4-hydroxybenzyl)amino]-5-nitrobenzamideHuman4499
CDK2CDKCMGC4cfxCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4442
CDK2CDKCMGC3pxrAB-Human4173
CDK2CDKCMGC2r3hAA3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman4152
CDK2CDKCMGC6q4eAA6-iodanyl-7~{h}-purin-2-amineHuman11199
CDK2CDKCMGC2r3jAB3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4544
CDK2CDKCMGC3s1hAB4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4226
CDK2CDKCMGC5if1AA-Human6568
CDK2CDKCMGC2iw9CBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3858
CDK2CDKCMGC5lmkCB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7397
CDK2CDKCMGC4cfwCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4549
CDK2CDKCMGC8curAB6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman14692
CDK9CDKCMGC4imyCAadenosine monophosphateHuman2237
CDK2CDKCMGC2cchABadenosine-5'-triphosphateHuman4553
CDK2CDKCMGC8oy2A(1s,2s,11as)-1-methoxy-1,4,7,10-tetramethyl-2,9-bis(oxidanyl)-2,11a-dihydrobenzo[b][1,4]benzodioxepine-3,6-dioneHuman15078
CDK13 (CHED)CDKCMGC5efqAadenosine-5'-diphosphateHuman6323
CDK7CDKCMGC1ua2Dadenosine-5'-triphosphateHuman543
CDK2CDKCMGC3qwkAB4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4155
CDK6CDKCMGC8i0mA2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman15164
CDK4CDKCMGC3g33A-Human3387
CDK6CDKCMGC2f2cB(2s)-2-({6-[(3-amino-5-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHuman2795
CDK6CDKCMGC4auaA1h-benzimidazol-2-yl(1h-pyrrol-2-yl)methanoneHuman2801
CDK2CDKCMGC6yl6AB-Human12495
CDK2CDKCMGC1pxmAB-Human3936
CDK2CDKCMGC8curAA6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman14693
CDK2CDKCMGC4cfmCA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4260
CDK2CDKCMGC4d1xA(4s)-2-(6-hydroxy-1,3-benzothiazol-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHuman4344
CDK2CDKCMGC8ru8AB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman15328
CDK2CDKCMGC4bckAC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4433
CDK2CDKCMGC4cfxAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman3963
CDK2CDKCMGC1oiyAB4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman3945
CDK2CDKCMGC4cfwAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4141
CDK2CDKCMGC2vthA5-hydroxynaphthalene-1-sulfonamideHuman4274
CDK2CDKCMGC2x1nAA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4579
CDK2CDKCMGC4bckAA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4095
CDK2CDKCMGC1hclAB-Human4540
CDK2CDKCMGC4bcnAA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4084
CDK2CDKCMGC3r9nAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3867
CDK2CDKCMGC3qqlAB(5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4378
CDK2CDKCMGC7nvqAstaurosporineHuman13627
CDK2CDKCMGC1h07AB((2-bromo-4-methylphenyl){6-[(4-{[(2s)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHuman3908
CDK2CDKCMGC5uq1A-Human8220
CDK2CDKCMGC2uueA4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHuman4515
CDK2CDKCMGC4fkiAAn-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamideHuman4430
CDK2CDKCMGC4cfmAB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman3986
CDK2CDKCMGC2c6tA4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman4371
CDK2CDKCMGC6guhAA4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10765
CDK2CDKCMGC2xnbAB3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHuman4034
CDK2CDKCMGC4bcqCA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman3996
CDK2CDKCMGC5osjAB-Human9742
CDK2CDKCMGC6yl1ABmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12496
CDK2CDKCMGC3rzbAA4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamideHuman4264
CDK2CDKCMGC2xmyAA4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHuman4526
CDK2CDKCMGC2cchAC-Human4566
CDK2CDKCMGC3raiAB4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4002
CDK12 (CRK7)CDKCMGC8bu6B~{n}-(1~{h}-benzimidazol-2-ylmethyl)-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman14921
CDK12 (CRK7)CDKCMGC9fmrB~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman15854
CDK6CDKCMGC6oqoAn-[5-(6-ethyl-2,6-diazaspiro[3.3]heptan-2-yl)pyridin-2-yl]-5-fluoro-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12646
CDK6CDKCMGC9d8uAatirmociclibHuman15857
CDK6CDKCMGC1g3nA-Human2806
CDK6CDKCMGC1bi7A-Human2798
CDK6CDKCMGC1blxA-Human2802
CDK6CDKCMGC1bi8A-Human2796
CDK6CDKCMGC6oqlA5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12647
CDK6CDKCMGC9pe7A(3r,4r)-4-({(4m)-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-1,3-benzimidazol-6-yl]pyrimidin-2-yl}amino)-1-(methanesulfonyl)piperidin-3-olHuman15858
CDK6CDKCMGC1jowB-Human2793
CDK6CDKCMGC1bi8C-Human2799
CDK6CDKCMGC4ez5A{5-[4-(dimethylamino)piperidin-1-yl]-1h-imidazo[4,5-b]pyridin-2-yl}[2-(isoquinolin-4-yl)pyridin-4-yl]methanoneHuman2800
CDK6CDKCMGC2eufB6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman2804
CDK6CDKCMGC1xo2B3,7,3',4'-tetrahydroxyflavoneHuman2794
CDK2CDKCMGC1w0xCBolomoucineHuman4478
CDK2CDKCMGC1h01AA(2r)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman3974
CDK2CDKCMGC6p3wCB-Human11516
CDK2CDKCMGC1h07AA((2-bromo-4-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHuman3918
CDK2CDKCMGC1pxjAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman3927
CDK2CDKCMGC2iw9CAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4218
CDK2CDKCMGC4bcpAA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4552
CDK2CDKCMGC2b55A2-(4-(aminomethyl)piperidin-1-yl)-n-(3_cyclohexyl-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)acetamideHuman4216
CDK2CDKCMGC6q4dAA2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11184
CDK2CDKCMGC3royAA4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4131
CDK2CDKCMGC4ii5ABadenosine-5'-diphosphateHuman4456
CDK2CDKCMGC3uliAA1-(aminomethyl)-n-(3-{[6-bromo-2-(4-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-7-yl]amino}propyl)cyclopropanecarboxamideHuman4115
CDK2CDKCMGC3bhtAB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4491
CDK2CDKCMGC3r8mAB1h-indazole-3-carbohydrazideHuman4451
CDK2CDKCMGC2w06A4-{[4-(1-cyclopropyl-2-methyl-1h-imidazol-5-yl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman3982
CDK2CDKCMGC2uzdA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3877
CDK2CDKCMGC5angA7-hydroxy-4-(morpholinomethyl)chromen-2-oneHuman6540
CDK2CDKCMGC5k4jAA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6751
CDK2CDKCMGC2c5oCB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4050
CDK2CDKCMGC4fksACn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4315
CDK2CDKCMGC2iw9AAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4174
CDK2CDKCMGC3r71AB4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4345
CDK2CDKCMGC2btrAn-(5-isopropyl-thiazol-2-yl)-2-pyridin-3-yl-acetamideHuman3998
CDK2CDKCMGC9d0wC-Human15925
CDK2CDKCMGC2r3fAB5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4291
CDK2CDKCMGC1p2aA5-[(2-aminoethyl)amino]-6-fluoro-3-(1h-pyrrol-2-yl)benzo[cd]indol-2(1h)-oneHuman4422
CDK2CDKCMGC3rpoAA4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acidHuman3966
CDK2CDKCMGC1urcCB-Human3937
CDK2CDKCMGC4cfwCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4102
CDK2CDKCMGC2r3pAA5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHuman4176
CDK2CDKCMGC5oo0AC-Human9745
CDK2CDKCMGC1v1kAB(2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-olHuman3928
CDK2CDKCMGC1jsuA-Human4146
CDK1 (CDC2)CDKCMGC6gu7E-Human10782
CDK1 (CDC2)CDKCMGC6gu2AA2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10780
CDK1 (CDC2)CDKCMGC6gu3A4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10778
CDK2CDKCMGC6oqiA5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4s)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12648
CDK12 (CRK7)CDKCMGC6ckxAn-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamideHuman10578
CDK6CDKCMGC5l2sAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman6990
CDK2CDKCMGC2wpaCn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHuman4162
CDK2CDKCMGC9et7AB4-bromanyl-1~{h}-pyridin-2-oneHuman15907
CDK2CDKCMGC2exmAn-(3-methylbut-2-en-1-yl)-9h-purin-6-amineHuman4055
CDK2CDKCMGC1h1rCB6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman4081
CDK2CDKCMGC1pxoAD[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4167
CDK2CDKCMGC3bhvAB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4001
CDK2CDKCMGC4fkuAA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman3863
CDK2CDKCMGC6q4aAA5-iodanylpyrimidineHuman11195
CDK2CDKCMGC4ek8AB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amineHuman3871
CDK2CDKCMGC9d0xB-Human15910
CDK2CDKCMGC4bcoAA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman3988
CDK2CDKCMGC5iexAA(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHuman6565
CDK2CDKCMGC8b54AB~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman14680
CDK2CDKCMGC1urcAB-Human4010
CDK2CDKCMGC3r28AA4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamideHuman4052
CDK2CDKCMGC4bcpCB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4501
CDK2CDKCMGC9hiuB-Human15912
CDK2CDKCMGC2b52A1-(3-(2,4-dimethylthiazol-5-yl)-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)-3-(4-methylpiperazin-1-yl)ureaHuman3997
CDK2CDKCMGC6gvaAA5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman11206
CDK2CDKCMGC3r1yAA2-[(pyridin-3-ylmethyl)amino]benzamideHuman4319
CDK2CDKCMGC6yl1AAmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12497
CDK2CDKCMGC4cfuAA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman3905
CDK2CDKCMGC2c4gA(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHuman4088
CDK2CDKCMGC4rj3AA1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4244
CDK2CDKCMGC1h26C-Human4179
CDK2CDKCMGC6q4bAC5-bromanylpyrimidineHuman11180
CDK2CDKCMGC9eslAB4-bromanyl-1-(2-methoxyethyl)pyridin-2-oneHuman15931
CDK2CDKCMGC3r7uAA2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamideHuman4510
CDK2CDKCMGC4eomABadenosine-5'-triphosphateHuman4472
CDK2CDKCMGC3qwkAA4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4091
CDK2CDKCMGC1pxjAB-Human3911
CDK2CDKCMGC2whbCA-Human4132
CDK2CDKCMGC4fkpAA3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4035
CDK2CDKCMGC6inlA2,2'-{[6-{[(4-methoxyphenyl)methyl]amino}-9-(propan-2-yl)-9h-purin-2-yl]azanediyl}di(ethan-1-ol)Human11794
CDK2CDKCMGC4eolAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4270
CDK2CDKCMGC3dogCB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4121
CDK2CDKCMGC3r7iAB4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acidHuman4070
CDK2CDKCMGC9esqAB4-bromanyl-2-oxidanyl-benzoic acidHuman15933
CDK2CDKCMGC3rpvAA4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4348
CDK2CDKCMGC3qziAB4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamideHuman4500
CDK2CDKCMGC4fkqAB4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHuman4026
CDK2CDKCMGC4eopCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4463
CDK2CDKCMGC2btsA4-[(5-isopropyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4443
CDK2CDKCMGC3tnwAA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman4254
CDK2CDKCMGC1h08AB(2s)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHuman4411
CDK2CDKCMGC3r1qAA4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4224
CDK2CDKCMGC3pxzA8-anilino-1-naphthalene sulfonateHuman4251
CDK2CDKCMGC1qmzCadenosine-5'-triphosphateHuman4527
CDK2CDKCMGC1pxkAAn-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n'-hydroxyimidoformamideHuman3915
CDK2CDKCMGC4cfxCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4166
CDK2CDKCMGC3my5CA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4473
CDK2CDKCMGC3sw4ABn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHuman4439
CDK2CDKCMGC2r3gAA6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman4276
CDK2CDKCMGC9esuAD-Human15934
CDK2CDKCMGC4eosAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4028
CDK2CDKCMGC2c5yAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman6785
CDK2CDKCMGC4eolCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4235
CDK2CDKCMGC9esnAB4-bromo-1-(2-hydroxyethyl)pyridin-2(1h)-oneHuman15923
CDK2CDKCMGC3bhvAA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4531
CDK2CDKCMGC3my5AB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3887
CDK2CDKCMGC6q4fAApyridine-2,6-diamineHuman11202
CDK2CDKCMGC5if1CB-Human6571
CDK2CDKCMGC6sg4AA-Human13246
CDK2CDKCMGC4eoqAAadenosine-5'-triphosphateHuman4402
CDK2CDKCMGC5a14AB1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHuman3901
CDK2CDKCMGC5cyiCA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6055
CDK2CDKCMGC3sw4AAn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHuman4076
CDK2CDKCMGC4bckCB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4506
CDK2CDKCMGC2vtsA5-[(4-aminocyclohexyl)amino]-7-(propan-2-ylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4300
CDK2CDKCMGC9et2AA~{n}-(4-bromophenyl)ethanamideHuman15924
CDK2CDKCMGC1f5qCB-Human3952
CDK2CDKCMGC3r1yAB2-[(pyridin-3-ylmethyl)amino]benzamideHuman4405
CDK2CDKCMGC1ckpABpurvalanol bHuman4214
CDK2CDKCMGC4kd1AB3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman4525
CDK2CDKCMGC3iggAn-[1-(cis-3-hydroxycyclobutyl)-1h-imidazol-4-yl]-2-(4-methoxyphenyl)acetamideHuman4360
CDK2CDKCMGC3qxpAA4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4343
CDK2CDKCMGC3r9dAB4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4565
CDK2CDKCMGC2r3iAB5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4059
CDK2CDKCMGC1h28C-Human4351
CDK2CDKCMGC2whbAB-Human4457
CDK2CDKCMGC1v1kAA(2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-olHuman4189
CDK2CDKCMGC11gvAA(1r,3s)-3-{3-[(1-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl bicyclo[1.1.1]pentan-1-ylcarbamateHuman15932
CDK2CDKCMGC6q4fACpyridine-2,6-diamineHuman11212
CDK2CDKCMGC3r8zAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanoneHuman4140
CDK2CDKCMGC5lmkAA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7399
CDK2CDKCMGC3bhuCB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4464
CDK2CDKCMGC2uzbCD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4502
CDK2CDKCMGC6q4dAC2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11188
CDK2CDKCMGC2w17ABn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman4165
CDK2CDKCMGC3qhwAAadenosine-5'-diphosphateHuman4346
CDK2CDKCMGC2uzeC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHuman4071
CDK2CDKCMGC1oi9CA6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4571
CDK2CDKCMGC3rk7A4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzamideHuman4236
CDK2CDKCMGC1f5qAB-Human4517
CDK2CDKCMGC3r8pAB(5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4538
CDK2CDKCMGC3rk9AA[4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4158
CDK2CDKCMGC3tnwAB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3948
CDK2CDKCMGC9nyrAA-Human15939
CDK2CDKCMGC3s2pA(3s,4s)-1-{3-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-4-hydroxyphenyl}pyrrolidine-3,4-diolHuman4404
CDK2CDKCMGC5jq5A(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman7416
CDK2CDKCMGC4eopAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4044
CDK2CDKCMGC2vtpAA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4511
CDK2CDKCMGC2cjmCadenosine-5'-triphosphateHuman4126
CDK2CDKCMGC9et7AA4-bromanyl-1~{h}-pyridin-2-oneHuman15940
CDK2CDKCMGC2c5nCAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4161
CDK2CDKCMGC3my5AA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4554
CDK2CDKCMGC4cfuCB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman4539
CDK2CDKCMGC9eskAA(4-bromo-2-oxopyridin-1(2h)-yl)acetic acidHuman15945
CDK2CDKCMGC2duvA2-(3,4-dihydroxyphenyl)-8-(1,1-dioxidoisothiazolidin-2-yl)-3-hydroxy-6-methyl-4h-chromen-4-oneHuman4193
CDK2CDKCMGC3qqlAA(5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4341
CDK2CDKCMGC1pkdC7-hydroxystaurosporineHuman3973
CDK2CDKCMGC3r9hAA4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman3958
CDK2CDKCMGC4fx3CB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4495
CDK2CDKCMGC7ra5AA4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman13960
CDK2CDKCMGC9etpAB4-bromo-1h-pyrazoleHuman15949
CDK2CDKCMGC6q3fAB-Human11187
CDK2CDKCMGC2c5nABn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4223
CDK2CDKCMGC4fkwAA2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHuman4252
CDK2CDKCMGC5if1CA-Human6564
CDK2CDKCMGC4acmAB3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman3983
CDK2CDKCMGC2whbAA-Human4471
CDK2CDKCMGC1okvC-Human4093
CDK2CDKCMGC4bcoCA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4333
CDK2CDKCMGC2c68A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydropyrazolo[1,5-a]pyrimidin-7-amineHuman6776
CDK2CDKCMGC2vtmApyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4283
CDK2CDKCMGC1oitA4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]benzenesulfonamideHuman4025
CDK2CDKCMGC4gcjAB4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4362
CDK2CDKCMGC3qtsAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanoneHuman4275
CDK2CDKCMGC3fz1A(3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-oneHuman4335
CDK2CDKCMGC4fkuAB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4573
CDK2CDKCMGC2uzeA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHuman3949
CDK2CDKCMGC2vtpAB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4401
CDK2CDKCMGC6q4cAA4-bromanyl-1,8-naphthyridineHuman11182
CDK8CDKCMGC4f6wAn-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-4-[2-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)ethyl]piperazine-1-carboxamideHuman3845
CDK8CDKCMGC4f7lAtert-butyl [3-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)propyl]carbamateHuman3840
CDK8CDKCMGC4f6uAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]ureaHuman3844
CDK2CDKCMGC2wipA1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHuman4520
CDK2CDKCMGC2i40CA5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4222
CDK2CDKCMGC4cfmCB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4005
CDK2CDKCMGC6q4jAB2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHuman11213
CDK2CDKCMGC4bcqAB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4415
CDK2CDKCMGC2j9mAB6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxideHuman4246
CDK2CDKCMGC1p5eC4,5,6,7-tetrabromobenzotriazoleHuman4434
CDK2CDKCMGC2iw8AAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4142
CDK2CDKCMGC3ddqABr-roscovitineHuman4269
CDK2CDKCMGC1w8cAB6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHuman4197
CDK2CDKCMGC3rk5A4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzoic acidHuman4160
CDK2CDKCMGC9eswAA(4-bromanylpyridin-2-yl)methanolHuman15935
CDK2CDKCMGC1h1pC6-o-cyclohexylmethyl guanineHuman4581
CDK2CDKCMGC3rk9AB[4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4259
CDK2CDKCMGC9eswAC-Human15936
CDK2CDKCMGC1buhA-Human4178
CDK2CDKCMGC3sqqAA4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4231
CDK2CDKCMGC2wxvAn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4318
CDK2CDKCMGC4fkvAA(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHuman4299
CDK2CDKCMGC9hj1B-Human15937
CDK2CDKCMGC3bhtCB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman3889
CDK2CDKCMGC9esuAA4-bromanyl-2-(methoxymethyl)pyridineHuman15938
CDK2CDKCMGC4bcnCB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4150
CDK2CDKCMGC4eooCAadenosine-5'-triphosphateHuman4188
CDK2CDKCMGC3r7eAB5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamideHuman4447
CDK2CDKCMGC9ob3A(1r,3r)-3-{3-[(pyrazine-2-carbonyl)amino]-1h-pyrazol-5-yl}cyclopentyl [(1s)-1-cyclopropylethyl]carbamateHuman15941
CDK2CDKCMGC5osmAAmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHuman9741
CDK2CDKCMGC2r3mABn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHuman4576
CDK2CDKCMGC2c5xCAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4466
CDK2CDKCMGC4bcqAA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4396
CDK2CDKCMGC3r73AB4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3899
CDK2CDKCMGC5fp6AB3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHuman6301
CDK2CDKCMGC2wmaC-Human4410
CDK2CDKCMGC9jj5A~{n}-(4-azanylcyclohexyl)-4-[[2,6-bis(fluoranyl)-3-[4-(methylcarbamoyl)phenyl]phenyl]carbonylamino]-1~{h}-pyrazole-3-carboxamideHuman15942
CDK2CDKCMGC3ql8AA3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrileHuman3916
CDK2CDKCMGC2c5oAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4388
CDK2CDKCMGC5iexAB(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHuman6572
CDK2CDKCMGC3qzfA2-(4,6-diamino-1,3,5-triazin-2-yl)benzene-1,4-diolHuman4569
CDK2CDKCMGC2a0cXA2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHuman4157
CDK2CDKCMGC5a14AA1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHuman3977
CDK2CDKCMGC4gcjAA4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4138
CDK2CDKCMGC1urwAB2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]-Human4196
CDK2CDKCMGC8b54AA~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman14681
CDK2CDKCMGC9hiwB-Human15943
CDK2CDKCMGC4bckAD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4563
CDK2CDKCMGC5aniA6-chloro-9h-purineHuman6539
CDK9CDKCMGC4ec8A-Human2244
CDK2CDKCMGC2c69A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-7-amineHuman6775
CDK2CDKCMGC1pw2A-Human4432
CDK2CDKCMGC1wccAB2-amino-6-chloropyrazineHuman3897
CDK2CDKCMGC3lfqAn-(6,7-difluoro-5-phenyl-1h-indazol-3-yl)butanamideHuman4320
CDK2CDKCMGC4ek4AB4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman3957
CDK2CDKCMGC4cfnCB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4567
CDK2CDKCMGC4eoiAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4342
CDK2CDKCMGC6ylkAAmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12499
CDK2CDKCMGC2x1nCA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman3991
CDK2CDKCMGC2c5oAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4440
CDK2CDKCMGC3pxfAB8-anilino-1-naphthalene sulfonateHuman4301
CDK8CDKCMGC6t41A~{n}-[(4-chlorophenyl)methyl]quinazolin-4-amineHuman11908
CDK2CDKCMGC3r7yAB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamideHuman3975
CDK2CDKCMGC1pxnAB-Human4172
CDK2CDKCMGC3tiyAA2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHuman4413
CDK2CDKCMGC6q3bAB4-iodopyrazoleHuman11208
CDK2CDKCMGC1hckABadenosine-5'-triphosphateHuman4416
CDK2CDKCMGC1h01AB(2s)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4561
CDK2CDKCMGC5lmkCA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7396
CDK2CDKCMGC1qmzAadenosine-5'-triphosphateHuman4242
CDK8CDKCMGC5idpAB(3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanoneHuman7320
CDK8CDKCMGC5icpAA[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanoneHuman7318
CDK8CDKCMGC8tqcCB-Human15963
CDK8CDKCMGC5xs2AA3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHuman8315
CDK8CDKCMGC8tq2CB-Human15964
CDK8CDKCMGC5idnAB[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanoneHuman7319
CDK8CDKCMGC5hbjAB8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6385
CDK8CDKCMGC6y0aAB6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman13305
CDK8CDKCMGC8tq2CA-Human15965
CDK8CDKCMGC8tqcCA-Human15966
CDK8CDKCMGC6r3sAA6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman12140
CDK8CDKCMGC5ceiAA4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamideHuman6404
CDK16 (PCTAIRE1)CDKCMGC3mtlAA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human1701
CDK2CDKCMGC3qxoA5-nitro-2-[(4-sulfamoylbenzyl)amino]benzamideHuman4282
CDK1 (CDC2)CDKCMGC4yc6CA-Human4608
CDK1 (CDC2)CDKCMGC4yc6GB-Human4615
CDK1 (CDC2)CDKCMGC5lqfDAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7365
CDK1 (CDC2)CDKCMGC5hq0AA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman6422
CDK1 (CDC2)CDKCMGC7nj0B-Human13827
CDK12 (CRK7)CDKCMGC8buqB(2~{r})-2-[[6-[[1-(3-chlorophenyl)pyrazol-3-yl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14917
CDK12 (CRK7)CDKCMGC6td3H(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12370
CDK12 (CRK7)CDKCMGC8bu2B~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-propan-2-yl-purin-6-amineHuman14918
CDK12 (CRK7)CDKCMGC5acbCn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman6701
CDK12 (CRK7)CDKCMGC6b3eA2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-olHuman9452
CDK12 (CRK7)CDKCMGC8bufB2-(6,7-dihydro-4~{h}-thieno[3,2-c]pyridin-5-ylmethyl)-6,7-dimethoxy-3~{h}-quinazolin-4-oneHuman14919
CDK12 (CRK7)CDKCMGC4un0C-Human4854
CDK12 (CRK7)CDKCMGC9jk1An-[5-[[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-[(phenylmethyl)carbamoyl]amino]-2-[4-(dimethylamino)piperidin-1-yl]phenyl]propanamideHuman15853
CDK12 (CRK7)CDKCMGC8burBB~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamideHuman14920
CDK12 (CRK7)CDKCMGC6td3B(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12371
CDK12 (CRK7)CDKCMGC8buhB6-[[[2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-9-propan-2-yl-purin-6-yl]amino]methyl]-3-pyridin-2-yl-1~{h}-pyridin-2-oneHuman14922
CDK12 (CRK7)CDKCMGC4cxaC-Human4853
CDK12 (CRK7)CDKCMGC8bupB(2~{r})-2-[[6-[3-(3-methylphenyl)propylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14923
CDK12 (CRK7)CDKCMGC8bumB(2r)-2-[[6-(5-naphthalen-1-ylpentylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14924
CDK12 (CRK7)CDKCMGC8buiB(2~{r})-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)amino]purin-2-yl]amino]butan-1-olHuman14925
CDK12 (CRK7)CDKCMGC8bu5B~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman14926
CDK12 (CRK7)CDKCMGC8bukB(2~{r})-2-[[6-(naphthalen-2-ylmethylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14927
CDK12 (CRK7)CDKCMGC8bubB~{n}-(5-methyl-2,3-dihydro-1,3-thiazol-2-yl)-3-(5-methylfuran-2-yl)carbonyl-1,3-thiazolidine-4-carboxamideHuman14928
CDK12 (CRK7)CDKCMGC9x26AB(2s)-n-[2-[4-(dimethylamino)piperidin-1-yl]-5-[[(1s)-1-(4-fluorophenyl)ethyl]carbamoyl-[4-(quinazolin-2-ylamino)cyclohexyl]amino]pyridin-3-yl]-2-fluoranyl-propanamideHuman15855
CDK12 (CRK7)CDKCMGC8budB~{n}-(5-bromanylpyridin-2-yl)-3-(4-oxidanylidenequinazolin-3-yl)propanamideHuman14929
CDK12 (CRK7)CDKCMGC9x26AA(2s)-n-[2-[4-(dimethylamino)piperidin-1-yl]-5-[[(1s)-1-(4-fluorophenyl)ethyl]carbamoyl-[4-(quinazolin-2-ylamino)cyclohexyl]amino]pyridin-3-yl]-2-fluoranyl-propanamideHuman15856
CDK12 (CRK7)CDKCMGC8p81AB~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman15061
CDK12 (CRK7)CDKCMGC4nstCadenosine-5'-diphosphateHuman4851
CDK12 (CRK7)CDKCMGC6ckxCn-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamideHuman10579
CDK12 (CRK7)CDKCMGC8bu1B(2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-olHuman14930
CDK12 (CRK7)CDKCMGC6b3eC2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-olHuman9453
CDK12 (CRK7)CDKCMGC4un0D-Human4855
CDK12 (CRK7)CDKCMGC8bu3B2-morpholin-4-yl-9-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]purin-6-amineHuman14931
CDK12 (CRK7)CDKCMGC8buaB(2~{r})-~{n}-(1~{h}-benzimidazol-2-yl)-2-(3-oxidanylidene-1~{h}-isoindol-2-yl)propanamideHuman14932
CDK12 (CRK7)CDKCMGC8bujB(2~{r})-2-[[6-(octylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14933
CDK12 (CRK7)CDKCMGC8buoB(2~{r})-2-[[6-[(3-fluoranyl-4-pyridin-2-yl-phenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14934
CDK12 (CRK7)CDKCMGC4cxaAphosphoaminophosphonic acid-adenylate esterHuman4856
CDK12 (CRK7)CDKCMGC8bugB2-[2-[(6-methylpyridin-2-yl)amino]-1,3-thiazol-4-yl]-~{n}-(5-methyl-1,3-thiazol-2-yl)ethanamideHuman14935
CDK12 (CRK7)CDKCMGC8p81AA~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman15062
CDK12 (CRK7)CDKCMGC8butB2-[[6-[[4-(2-hydroxyethyloxy)phenyl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14936
CDK4CDKCMGC5fwmK-Human6749
CDK4CDKCMGC5fwkK-Human6747
CDK4CDKCMGC6p8fB-Human11892
CDK4CDKCMGC3g33C-Human3384
CDK4CDKCMGC6p8eB-Human11891
CDK4CDKCMGC2w9zBB-Human3383
CDK12 (CRK7)CDKCMGC8busB1,3-dimethyl-5-[[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]methyl]pyrazole-4-sulfonamideHuman14908
CDK12 (CRK7)CDKCMGC8bucB2-(1~{h}-benzimidazol-2-ylsulfanyl)-~{n}-(5-chloranylpyridin-2-yl)ethanamideHuman14909
CDK12 (CRK7)CDKCMGC8bu4B(2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-olHuman14910
CDK12 (CRK7)CDKCMGC8bulB(2~{r})-2-[[6-(3-phenylpropylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14911
CDK12 (CRK7)CDKCMGC6td3E(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12369
CDK12 (CRK7)CDKCMGC8bueB~{n}-(1~{h}-benzimidazol-2-yl)-1-(2-methoxy-5-methyl-phenyl)-5-oxidanylidene-pyrrolidine-3-carboxamideHuman14912
CDK12 (CRK7)CDKCMGC8bu7B-Human14913
CDK12 (CRK7)CDKCMGC8bu9Br-roscovitineHuman14914
CDK12 (CRK7)CDKCMGC5acbDn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman6702
CDK12 (CRK7)CDKCMGC8burBA~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamideHuman14915
CDK12 (CRK7)CDKCMGC8bunB(2~{r})-2-[[6-[(4-phenylphenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14916
CDK12 (CRK7)CDKCMGC4nstAadenosine-5'-diphosphateHuman4852
CDK6CDKCMGC1g3nE-Human2805
CDK6CDKCMGC3nupA4-[3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(1-methylpiperidin-4-yl)pyrimidin-2-amineHuman2797
CDK6CDKCMGC4tthB9-cyclopentyl-n-(5-piperazin-1-ylpyridin-2-yl)pyrido[4,5]pyrrolo[1,2-d]pyrimidin-2-amineHuman2803
CDK6CDKCMGC5l2iA6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6991
CDK2CDKCMGC2r3iAA5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4135
CDK2CDKCMGC3r7uAB2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamideHuman4023
CDK2CDKCMGC1h08AA(2r)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHuman4220
CDK2CDKCMGC2whbCB-Human4352
CDK2CDKCMGC4eoiCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4522
CDK2CDKCMGC1ckpAApurvalanol bHuman4066
CDK2CDKCMGC2uzdC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3900
CDK2CDKCMGC4fkjABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHuman4164
CDK2CDKCMGC1pxpAB-Human3943
CDK2CDKCMGC2wfyAB-Human4426
CDK2CDKCMGC2wevAC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4007
CDK2CDKCMGC2b53A6-(3-aminophenyl)-n-(tert-butyl)-2-(trifluoromethyl)quinazolin-4-amineHuman3875
CDK2CDKCMGC4fkpAC3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4468
CDK2CDKCMGC4d1zA(4s)-2-(8-hydroxyquinolin-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHuman4486
CDK2CDKCMGC1h0wAA1-amino-6-cyclohex-3-enylmethyloxypurineHuman3987
CDK2CDKCMGC1oirA1-(dimethylamino)-3-(4-{{4-(2-methylimidazo[1,2-a]pyridin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4389
CDK2CDKCMGC3ezrA3-methoxy-4-{3-[4-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman4475
CDK2CDKCMGC5l2wA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman6993
CDK2CDKCMGC1h1rCA6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman3920
CDK2CDKCMGC3qqfAB5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4287
CDK2CDKCMGC6q3cAB4-bromo-1h-pyrazoleHuman11203
CDK2CDKCMGC5ieyAB4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHuman6573
CDK2CDKCMGC4nj3AB6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman4366
CDK2CDKCMGC9glaAB7-dimethylphosphoryl-3-[2-[[(3~{s})-6,6-dimethylpiperidin-3-yl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]-1~{h}-indole-6-carbonitrileHuman15921
CDK2CDKCMGC2iw8CAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4294
CDK2CDKCMGC6sg4CB-Human13245
CDK2CDKCMGC2vtlAn-phenyl-1h-pyrazole-3-carboxamideHuman3870
CDK2CDKCMGC4cfwCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4508
CDK2CDKCMGC1w98A-Human4013
CDK2CDKCMGC7vduAA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14136
CDK2CDKCMGC9esnAA4-bromo-1-(2-hydroxyethyl)pyridin-2(1h)-oneHuman15922
CDK2CDKCMGC2r3oAB(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4354
CDK2CDKCMGC2vtaA1h-indazoleHuman4118
CDK2CDKCMGC4fkoAA2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHuman4449
CDK2CDKCMGC3qtrAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman3874
CDK2CDKCMGC4bckCA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4268
CDK2CDKCMGC3ej1An-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHuman4168
CDK2CDKCMGC6q4gAA2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHuman11214
CDK2CDKCMGC2uzlC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHuman4106
CDK2CDKCMGC1dm2AA4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHuman4104
CDK2CDKCMGC3rpyAA4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4261
CDK2CDKCMGC3royAB4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4239
CDK2CDKCMGC3py0AB(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3869
CDK2CDKCMGC3ddqCBr-roscovitineHuman4289
CDK2CDKCMGC4cfnAA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4285
CDK2CDKCMGC4eoqABadenosine-5'-triphosphateHuman4230
CDK2CDKCMGC6q4bAA5-bromanylpyrimidineHuman11198
CDK2CDKCMGC2a0cXB2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHuman3868
CDK2CDKCMGC9esoAA-Human15926
CDK2CDKCMGC4lynA(2s)-n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)-2-phenylpropanamideHuman4550
CDK2CDKCMGC3qtrAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4243
CDK2CDKCMGC2r3fAA5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4175
CDK2CDKCMGC1oiuAA3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4110
CDK2CDKCMGC6rijAB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12624
CDK2CDKCMGC4ek4AA4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman4212
CDK2CDKCMGC3rpyAB4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4519
CDK2CDKCMGC5osjAA-Human9743
CDK2CDKCMGC5cyiAB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6054
CDK2CDKCMGC1jstAadenosine-5'-triphosphateHuman4455
CDK2CDKCMGC4fkgAA4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acidHuman4020
CDK2CDKCMGC2w17AAn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman3968
CDK2CDKCMGC2r64An-[5-(1,1-dioxidoisothiazolidin-2-yl)-1h-indazol-3-yl]-2-(4-piperidin-1-ylphenyl)acetamideHuman4425
CDK2CDKCMGC6gufAn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman10770
CDK2CDKCMGC2r3oAA(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4147
CDK2CDKCMGC13gkAA4-[(1m)-1-{4-[(azetidin-1-yl)methyl]-2-chlorophenyl}-1h-imidazol-4-yl]-n-[1-(methanesulfonyl)piperidin-4-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman15927
CDK2CDKCMGC1aq1AstaurosporineHuman4267
CDK2CDKCMGC2vtrAB5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman3907
CDK2CDKCMGC8ypwAmethyl 3-[4-[3-[[3-[(1-ethylsulfonylpiperidin-4-yl)carbamoyl]-1~{h}-pyrazol-4-yl]carbamoyl]-2,4-bis(fluoranyl)phenyl]piperidin-1-yl]-3-oxidanylidene-propanoateHuman15928
CDK2CDKCMGC3my5CB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4003
CDK2CDKCMGC2uzbCC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4045
CDK2CDKCMGC1urwAA2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]-Human4054
CDK2CDKCMGC1h28A-Human4169
CDK2CDKCMGC9espAA4-bromo-1-(2-methoxyethyl)-1h-pyrazoleHuman15929
CDK2CDKCMGC5if1AB-Human6569
CDK2CDKCMGC2bkzC1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHuman4555
CDK2CDKCMGC1r78AB4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman4249
CDK2CDKCMGC2wevAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4067
CDK2CDKCMGC3rkbAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4460
CDK2CDKCMGC4fkgAB4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acidHuman4559
CDK2CDKCMGC3unjA4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acidHuman4498
CDK2CDKCMGC4ez3A4-[(e)-(6-hydroxy-2-oxo-1,2-dihydropyridin-3-yl)diazenyl]benzenesulfonamideHuman4551
CDK2CDKCMGC4bcmCA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4227
CDK2CDKCMGC6q49AA-Human11185
CDK2CDKCMGC5k4jAB1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6750
CDK2CDKCMGC1ykrA4-{[6-(2,6-dichlorobenzoyl)imidazo[1,2-a]pyridin-2-yl]amino}benzenesulfonamideHuman4578
CDK2CDKCMGC6q4kAB-Human11186
CDK2CDKCMGC2i40CB5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4043
CDK2CDKCMGC1ke8A4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}-n-(1,3-thiazol-2-yl)benzenesulfonamideHuman4048
CDK2CDKCMGC2cchCBadenosine-5'-triphosphateHuman4000
CDK2CDKCMGC2wihCn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4119
CDK2CDKCMGC2c5vCB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4209
CDK2CDKCMGC2r3qAC3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman3976
CDK2CDKCMGC3r83AB4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4543
CDK2CDKCMGC3r7vAB5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamideHuman4183
CDK2CDKCMGC4cfxCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4257
CDK2CDKCMGC3r73AA4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4187
CDK2CDKCMGC5mhqAA(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHuman9409
CDK2CDKCMGC9eszAA-Human15944
CDK2CDKCMGC4cfnCA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4355
CDK2CDKCMGC3qzgAB2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenolHuman4347
CDK2CDKCMGC2jgzA-Human4117
CDK2CDKCMGC7ackCB8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13452
CDK2CDKCMGC6jgmA4-{[6-(cyclohexylmethoxy)-7h-purin-2-yl]amino}-n,n-diethylbenzamideHuman12008
CDK2CDKCMGC4fx3AA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4518
CDK2CDKCMGC1gz8AA1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHuman3981
CDK2CDKCMGC3qtqAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4210
CDK2CDKCMGC2iw9ABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3955
CDK2CDKCMGC1oguCA4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3964
CDK2CDKCMGC3qu0AB4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4558
CDK2CDKCMGC7rweA5-nitro-2-[(3-phenylpropyl)amino]benzoic acidHuman14345
CDK2CDKCMGC9eszAB5-iodanylpyrimidineHuman15946
CDK2CDKCMGC1p5eA4,5,6,7-tetrabromobenzotriazoleHuman4090
CDK2CDKCMGC2r3qAB3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman4459
CDK2CDKCMGC3rpvAB4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4372
CDK2CDKCMGC4fktAAn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4548
CDK2CDKCMGC1finAadenosine-5'-triphosphateHuman4367
CDK2CDKCMGC3dogAB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4365
CDK2CDKCMGC3ddpAA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6781
CDK2CDKCMGC1wccAA2-amino-6-chloropyrazineHuman4394
CDK2CDKCMGC6q48AB4-iodanyl-3~{h}-pyridin-2-oneHuman11218
CDK2CDKCMGC1oi9CB6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4036
CDK2CDKCMGC7ackAB8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13453
CDK2CDKCMGC13gkAB4-[(1m)-1-{4-[(azetidin-1-yl)methyl]-2-chlorophenyl}-1h-imidazol-4-yl]-n-[1-(methanesulfonyl)piperidin-4-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman15947
CDK2CDKCMGC1jvpP23-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazoleHuman4097
CDK2CDKCMGC4eooABadenosine-5'-triphosphateHuman4278
CDK2CDKCMGC3ddpCA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6784
CDK2CDKCMGC11gvAB(1r,3s)-3-{3-[(1-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl bicyclo[1.1.1]pentan-1-ylcarbamateHuman15948
CDK2CDKCMGC6gueA4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10771
CDK2CDKCMGC6sg4AB-Human13247
CDK2CDKCMGC6gucC(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman10766
CDK2CDKCMGC7e34A-Human13497
CDK2CDKCMGC2wpaAn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHuman4399
CDK2CDKCMGC1okvA-Human3921
CDK2CDKCMGC3qtsAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanoneHuman4564
CDK2CDKCMGC1hckAAadenosine-5'-triphosphateHuman3878
CDK2CDKCMGC6q4gAB2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHuman11217
CDK2CDKCMGC3my5AC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3910
CDK2CDKCMGC6sg4CA-Human13248
CDK2CDKCMGC9eslAA4-bromanyl-1-(2-methoxyethyl)pyridin-2-oneHuman15950
CDK2CDKCMGC6q3cAC-Human11178
CDK2CDKCMGC4ii5CBadenosine-5'-diphosphateHuman4462
CDK2CDKCMGC6q4aAC5-iodanylpyrimidineHuman11216
CDK2CDKCMGC3qwjAA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamideHuman4265
CDK2CDKCMGC3r9oA4-amino-n-(3,5-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4279
CDK2CDKCMGC3qruAA(5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4237
CDK2CDKCMGC1h0vAA5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHuman4368
CDK2CDKCMGC4eonCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4192
CDK2CDKCMGC4ek3AB-Human4202
CDK2CDKCMGC4cfvCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman3979
CDK2CDKCMGC1oiyCB4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4245
CDK2CDKCMGC6q48AA4-iodanyl-3~{h}-pyridin-2-oneHuman11192
CDK2CDKCMGC4bzdAA6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHuman3865
CDK2CDKCMGC1vywAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamideHuman3992
CDK2CDKCMGC1y91A4-[5-(trans-4-aminocyclohexylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-7-ylamino]-n,n-dimethylbenzenesulfonamideHuman4505
CDK2CDKCMGC7b5lL-Human13266
CDK8CDKCMGC4f7sAAn-(2-phenylethyl)quinazolin-4-amineHuman3850
CDK8CDKCMGC5hbeAB8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-oneHuman6386
CDK9CDKCMGC3tniA-Human2250
CDK9CDKCMGC4imyEAadenosine monophosphateHuman2258
CDK9CDKCMGC4imyCBadenosine monophosphateHuman2245
CDK9CDKCMGC4bchA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman2246
CDK9CDKCMGC4bcgA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman2255
CDK9CDKCMGC4ogrAadenosineHuman2254
CDK9CDKCMGC4bcjA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman2247
CDK9CDKCMGC6w9eAB(4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13858
CDK9CDKCMGC4or5A-Human2233
CDK9CDKCMGC6w9eAD(4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13860
CDK9CDKCMGC3blhA-Human2251
CDK9CDKCMGC3my1A5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman2249
CDK9CDKCMGC3lq5A(2s)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman2253
CDK9CDKCMGC4or5F-Human2231
CDK9CDKCMGC3tnhA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman2232
CDK9CDKCMGC4bcfA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman2257
CDK7CDKCMGC6xd3Jn-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamideHuman12772
CDK7CDKCMGC8byqI-Human14732
CDK7CDKCMGC6o9l8-Human11055
CDK7CDKCMGC8pyrAA-Human15254
CDK7CDKCMGC6xbzJphosphothiophosphoric acid-adenylate esterHuman12773
CDK7CDKCMGC1ua2Badenosine-5'-triphosphateHuman541
CDK7CDKCMGC1ua2Aadenosine-5'-triphosphateHuman540
CDK7CDKCMGC29wdI-Human16031
CDK7CDKCMGC8bvwI-Human14733
CDK7CDKCMGC7b5oJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13279
CDK7CDKCMGC7b5qJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13280
CDK4CDKCMGC5fwpK-Human7132
CDK4CDKCMGC6p8hB-Human11894
CDK4CDKCMGC2w9zBA-Human3388
CDK4CDKCMGC2w9fB-Human3386
CDK4CDKCMGC6p8gB-Human11893
CDK4CDKCMGC2w96BA-Human3390
CDK4CDKCMGC2w96BB-Human3389
CDK4CDKCMGC5fwlK-Human6748
CDK4CDKCMGC2w99B-Human3385
CDK5CDKCMGC1ungA6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2792
CDK5CDKCMGC1h4lB-Human2779
CDK5CDKCMGC4au8BB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2781
CDK5CDKCMGC7vdpA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14145
CDK5CDKCMGC4au8AA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2784
CDK5CDKCMGC1unlAr-roscovitineHuman2785
CDK5CDKCMGC4au8BA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2791