| DDR1 | DDR | TK | 5sb0 | A | | n-{[(1r,2s)-2-{2-[(pyridin-3-yl)oxy]ethyl}cyclohexyl]methyl}-3-(trifluoromethoxy)benzamide | Human | 14264 | |
| DDR1 | DDR | TK | 5sav | A | A | n-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamide | Human | 14265 | |
| DDR1 | DDR | TK | 7feh | A | A | n-[(5-chloranyl-2-ethylsulfonyl-phenyl)methyl]-3-piperazin-1-yl-5-(trifluoromethyloxy)benzamide | Human | 14309 | |
| DDR1 | DDR | TK | 9sp9 | A | | ~{n}-(1-imidazo[1,2-a]pyridin-3-ylcarbonyl-2,3-dihydroindol-6-yl)-3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)benzamide | Human | 15544 | |
| DDR1 | DDR | TK | 5sb1 | A | A | 4-chloro-n-[(3s,4r)-4-phenylpyrrolidin-3-yl]-3-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | 14252 | |
| DDR1 | DDR | TK | 5sav | A | B | n-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamide | Human | 14261 | |
| DDR1 | DDR | TK | 4bkj | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 3263 | |
| DDR1 | DDR | TK | 5bvn | A | | n-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 3261 | |
| DDR1 | DDR | TK | 4bkj | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 3259 | |
| DDR1 | DDR | TK | 5saz | A | B | 2-chloro-5-{3-chloro-4-[(2-hydroxyethyl)amino]benzamido}-n-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamide | Human | 14260 | |
| DDR1 | DDR | TK | 6fil | A | A | 2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamide | Human | 10746 | |
| DDR1 | DDR | TK | 3zos | B | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3258 | |
| DDR1 | DDR | TK | 3zos | B | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3260 | |
| DDR1 | DDR | TK | 6few | A | B | 2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamide | Human | 10740 | |
| DDR1 | DDR | TK | 3zos | A | A | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3253 | |
| DDR1 | DDR | TK | 5fdp | A | | (4~{s})-4-methyl-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinoline-7-carboxamide | Human | 6676 | |
| DDR1 | DDR | TK | 4bkj | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 3255 | |
| DDR1 | DDR | TK | 5saw | A | B | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 14251 | |
| DDR1 | DDR | TK | 5fdx | B | | 3-[(4-methylpiperazin-1-yl)methyl]-~{n}-[(4~{r})-4-methyl-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinolin-7-yl]-5-(trifluoromethyl)benzamide | Human | 7130 | |
| DDR1 | DDR | TK | 7bcm | B | | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 13381 | |
| DDR1 | DDR | TK | 6gwr | B | B | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamide | Human | 10487 | |
| DDR1 | DDR | TK | 5sb2 | A | A | 3-chloro-n-[(1r,2s)-2-phenylcyclopropyl]-5-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | 14250 | |
| DDR1 | DDR | TK | 5bvo | A | | n-(5-{(1s)-1-[(5-fluoro-1,3-benzoxazol-2-yl)amino]ethyl}-2-methylphenyl)imidazo[1,2-a]pyridine-3-carboxamide | Human | 3250 | |
| DDR1 | DDR | TK | 5bvk | A | | 1-(2-chlorophenyl)-3-(pyridin-3-ylmethyl)urea | Human | 3251 | |
| DDR1 | DDR | TK | 4ckr | A | A | 4-[(4-ethylpiperazin-1-yl)methyl]-n-{4-methyl-3-[(2-oxo-2,3-dihydro-1h-indol-5-yl)oxy]phenyl}-3-(trifluoromethyl)benzamide | Human | 3257 | |
| DDR1 | DDR | TK | 4bkj | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 3256 | |
| DDR1 | DDR | TK | 5fdx | A | | 3-[(4-methylpiperazin-1-yl)methyl]-~{n}-[(4~{r})-4-methyl-2-pyrimidin-5-yl-3,4-dihydro-1~{h}-isoquinolin-7-yl]-5-(trifluoromethyl)benzamide | Human | 7131 | |
| DDR1 | DDR | TK | 5sau | A | A | 3-[(6-aminopyridin-3-yl)ethynyl]-n-[3-(trifluoromethyl)phenyl]benzamide | Human | 14253 | |
| DDR1 | DDR | TK | 6fin | A | B | 3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-8-(1~{h}-indazol-5-ylcarbonyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one | Human | 10747 | |
| DDR1 | DDR | TK | 7be6 | A | A | 5-amino-n-(4-(((2s)-4-cyclohexyl-1-((1-(methylsulfonyl)piperidin-3-yl)amino)-1-oxobutan-2-yl)carbamoyl)benzyl)-1-phenyl-1h-pyrazole-4-carboxamide | Human | 13378 | |
| DDR1 | DDR | TK | 5sb2 | A | B | 3-chloro-n-[(1r,2s)-2-phenylcyclopropyl]-5-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | 14254 | |
| DDR1 | DDR | TK | 5sb1 | A | B | 4-chloro-n-[(3s,4r)-4-phenylpyrrolidin-3-yl]-3-{[(1h-pyrrolo[2,3-b]pyridin-5-yl)oxy]methyl}benzamide | Human | 14257 | |
| DDR1 | DDR | TK | 6fio | A | B | 2-[1'-(1~{h}-indazol-5-ylcarbonyl)-4-methyl-2-oxidanylidene-spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10749 | |
| DDR1 | DDR | TK | 5sau | A | B | 3-[(6-aminopyridin-3-yl)ethynyl]-n-[3-(trifluoromethyl)phenyl]benzamide | Human | 14258 | |
| DDR1 | DDR | TK | 5saw | A | A | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 14259 | |
| DDR1 | DDR | TK | 6gwr | A | B | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamide | Human | 10484 | |
| DDR1 | DDR | TK | 6bsd | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 10761 | |
| DDR1 | DDR | TK | 6hp9 | A | | (2~{r})-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-2-(pyrimidin-5-ylamino)-2,3-dihydro-1~{h}-indene-5-carboxamide | Human | 10885 | |
| DDR1 | DDR | TK | 6fin | A | A | 3-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-8-(1~{h}-indazol-5-ylcarbonyl)-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one | Human | 10743 | |
| DDR1 | DDR | TK | 5sax | A | A | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 14262 | |
| DDR1 | DDR | TK | 7feh | A | B | n-[(5-chloranyl-2-ethylsulfonyl-phenyl)methyl]-3-piperazin-1-yl-5-(trifluoromethyloxy)benzamide | Human | 14308 | |
| DDR1 | DDR | TK | 6fil | A | B | 2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamide | Human | 10739 | |
| DDR1 | DDR | TK | 6fiq | A | | 1-(1~{h}-indazol-5-ylcarbonyl)-5'-methoxy-1'-[2-oxidanylidene-2-[(2~{s})-2-(trifluoromethyl)pyrrolidin-1-yl]ethyl]spiro[piperidine-4,3'-pyrrolo[3,2-b]pyridine]-2'-one | Human | 10742 | |
| DDR1 | DDR | TK | 7be6 | A | B | 5-amino-n-(4-(((2s)-4-cyclohexyl-1-((1-(methylsulfonyl)piperidin-3-yl)amino)-1-oxobutan-2-yl)carbamoyl)benzyl)-1-phenyl-1h-pyrazole-4-carboxamide | Human | 13380 | |
| DDR1 | DDR | TK | 6fex | A | A | 2-[4-bromanyl-2-oxidanylidene-1'-(1~{h}-pyrazolo[4,3-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10741 | |
| DDR1 | DDR | TK | 6few | A | A | 2-[8-(2~{h}-indazol-5-ylcarbonyl)-4-oxidanylidene-1-phenyl-1,3,8-triazaspiro[4.5]decan-3-yl]-~{n}-methyl-ethanamide | Human | 10738 | |
| DDR1 | DDR | TK | 3zos | A | B | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 3262 | |
| DDR1 | DDR | TK | 6y23 | C | | - | Human | 12743 | |
| DDR1 | DDR | TK | 6fio | A | A | 2-[1'-(1~{h}-indazol-5-ylcarbonyl)-4-methyl-2-oxidanylidene-spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10748 | |
| DDR1 | DDR | TK | 6y23 | A | | - | Human | 12741 | |
| DDR1 | DDR | TK | 6y23 | B | | - | Human | 12742 | |
| DDR1 | DDR | TK | 6hp9 | B | | (2~{r})-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-2-(pyrimidin-5-ylamino)-2,3-dihydro-1~{h}-indene-5-carboxamide | Human | 10884 | |
| DDR1 | DDR | TK | 6brj | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 10760 | |
| DDR1 | DDR | TK | 5saz | A | A | 2-chloro-5-{3-chloro-4-[(2-hydroxyethyl)amino]benzamido}-n-(1h-pyrrolo[2,3-b]pyridin-5-yl)benzamide | Human | 14255 | |
| DDR1 | DDR | TK | 7bcm | A | | ~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[[(3~{s})-1-methylsulfonylpiperidin-3-yl]amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 13379 | |
| DDR1 | DDR | TK | 5say | A | | n-(2-{3-[(2-aminopyrimidin-5-yl)oxy]phenyl}ethyl)-3-(trifluoromethoxy)benzamide | Human | 14256 | |
| DDR2 | DDR | TK | 6fer | F | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10732 | |
| DDR1 | DDR | TK | 6fex | A | B | 2-[4-bromanyl-2-oxidanylidene-1'-(1~{h}-pyrazolo[4,3-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10744 | |
| DDR1 | DDR | TK | 5bvw | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 3254 | |
| DDR1 | DDR | TK | 6gwr | B | A | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamide | Human | 10486 | |
| DDR1 | DDR | TK | 4ckr | A | B | 4-[(4-ethylpiperazin-1-yl)methyl]-n-{4-methyl-3-[(2-oxo-2,3-dihydro-1h-indol-5-yl)oxy]phenyl}-3-(trifluoromethyl)benzamide | Human | 3252 | |
| DDR1 | DDR | TK | 5sax | A | B | 2-{3-[(pyridin-3-yl)ethynyl]phenyl}-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 14263 | |
| DDR1 | DDR | TK | 6gwr | A | A | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-~{n}-[3-[(4-methylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl]-4-propan-2-yl-benzamide | Human | 10485 | |
| DDR2 | DDR | TK | 7aym | A | A | n-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 13071 | |
| DDR2 | DDR | TK | 6fer | C | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10731 | |
| DDR2 | DDR | TK | 6fer | B | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10736 | |
| DDR2 | DDR | TK | 6fer | D | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10730 | |
| DDR2 | DDR | TK | 6fer | K | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10725 | |
| DDR2 | DDR | TK | 6fer | I | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10735 | |
| DDR2 | DDR | TK | 6fer | A | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10729 | |
| DDR2 | DDR | TK | 6fer | J | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10728 | |
| DDR2 | DDR | TK | 6fer | H | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10727 | |
| DDR2 | DDR | TK | 7aym | A | B | n-[5-({[(3-fluorophenyl)carbamoyl]amino}methyl)-2-methylphenyl]imidazo[1,2-a]pyridine-3-carboxamide | Human | 13072 | |
| DDR2 | DDR | TK | 6fer | E | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10726 | |
| DDR2 | DDR | TK | 6fer | L | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10733 | |
| DDR2 | DDR | TK | 6fer | G | | 2-[4,5-bis(fluoranyl)-2-oxidanylidene-1'-(1~{h}-pyrazolo[3,4-b]pyridin-5-ylcarbonyl)spiro[indole-3,4'-piperidine]-1-yl]-~{n}-[2,2,2-tris(fluoranyl)ethyl]ethanamide | Human | 10734 | |
