Search results (296 entries covering 132 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
EPHA2 (EphA2)EphTK6q7dAB3-[[4-imidazol-1-yl-6-(4-oxidanylpiperidin-1-yl)-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11928
EPHA2 (EphA2)EphTK4p2kA-Human2091
EPHA2 (EphA2)EphTK4trlA-Human2090
EPHA3 (EphA3)EphTK2qodAC-Human2866
EPHA2 (EphA2)EphTK5i9zABn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman7181
EPHA2 (EphA2)EphTK5i9yAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7194
EPHA2 (EphA2)EphTK5ia2AB7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman7172
EPHB4 (EphB4)EphTK6fnjBA4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10340
EPHB4 (EphB4)EphTK2vwyAAn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-methylsulfonylphenyl)pyrimidine-2,4-diamineHuman353
EPHA2 (EphA2)EphTK6hesAB4-methyl-3-[(2-pyridin-3-ylquinazolin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11566
EPHB4 (EphB4)EphTK2yn8BstaurosporineHuman349
EPHA2 (EphA2)EphTK5ia0CAalisertibHuman7186
EPHB4 (EphB4)EphTK2vwyABn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-methylsulfonylphenyl)pyrimidine-2,4-diamineHuman355
EPHA3 (EphA3)EphTK4twnAB1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman2865
EPHA2 (EphA2)EphTK6hewAC-Human11553
EPHA7 (EphA7)EphTK2reiAA-Human4
EPHA7 (EphA7)EphTK7eecAB-Human13790
EPHA7 (EphA7)EphTK7eedA-Human13791
EPHA7 (EphA7)EphTK7eecAA-Human13792
EPHA7 (EphA7)EphTK3dkoAA5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamideHuman1
EPHA7 (EphA7)EphTK2reiAB-Human2
EPHA7 (EphA7)EphTK7eefA-Human13793
EPHA7 (EphA7)EphTK3dkoAB5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamideHuman3
EPHA2 (EphA2)EphTK5nk9AA(2~{z})-~{n}-(2-chloranyl-6-methyl-phenyl)-2-[3-[(4-methyl-4-oxidanyl-cyclohexyl)carbamoyl]phenyl]imino-1,3-thiazolidine-5-carboxamideHuman8073
EPHA2 (EphA2)EphTK5nk6AB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(4-oxidanylcyclohexyl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8061
EPHA2 (EphA2)EphTK6q7eAB3-[[4-imidazol-1-yl-6-[(3~{r})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11932
EPHA2 (EphA2)EphTK5nkaAA4-[[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylamino]cyclohexane-1-carboxylic acidHuman8075
EPHA2 (EphA2)EphTK6hexAC-Human11551
EPHA2 (EphA2)EphTK6q7bAB3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11935
EPHB4 (EphB4)EphTK6fniAB4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10333
EPHB4 (EphB4)EphTK6fnjBB4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10341
EPHB4 (EphB4)EphTK6fnkAA1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10344
EPHB4 (EphB4)EphTK2vwzAAn-[3-[[4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl]amino]phenyl]methanesulfonamideHuman360
EPHA2 (EphA2)EphTK8bofAB4-methyl-~{n}-(3-methylphenyl)-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14652
EPHA8 (EphA8)EphTK3kulBA-Human1249
EPHA8 (EphA8)EphTK3kulBB-Human1250
EPHA8 (EphA8)EphTK3kulAB-Human1252
EPHA8 (EphA8)EphTK3kulAA-Human1251
EPHA2 (EphA2)EphTK8bogAA~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamideHuman14650
EPHB1 (EphB1)EphTK6umwAA7-chlorotetracyclineHuman12924
EPHB4 (EphB4)EphTK2xvdAA{4-methyl-3-[(1-methylethyl)(2-{[3-(methylsulfonyl)-5-morpholin-4-ylphenyl]amino}pyrimidin-4-yl)amino]phenyl}methanolHuman363
EPHB4 (EphB4)EphTK2x9fAAn^4^-1h-indazol-4-yl-n^2^-[3-(methylsulfonyl)phenyl]pyrimidine-2,4-diamineHuman354
EPHB4 (EphB4)EphTK2vwvABn'-(3-chloro-4-methoxy-phenyl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazine-2,4-diamineHuman369
EPHA3 (EphA3)EphTK2qoqAAphosphoaminophosphonic acid-adenylate esterHuman2890
EPHB4 (EphB4)EphTK4aw5AB(3z)-5-[(1-ethylpiperidin-4-yl)amino]-3-[(5-methoxy-1h-benzimidazol-2-yl)(phenyl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman376
EPHB4 (EphB4)EphTK6fnjAA4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10336
EPHA3 (EphA3)EphTK4gk2AA7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2841
EPHB4 (EphB4)EphTK6fniAA4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10338
EPHA2 (EphA2)EphTK7kjaBAphosphomethylphosphonic acid adenylate esterHuman13249
EPHA2 (EphA2)EphTK6hesAA4-methyl-3-[(2-pyridin-3-ylquinazolin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11550
EPHA3 (EphA3)EphTK4gk4AA8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2854
EPHA3 (EphA3)EphTK2qofAC-Human2870
EPHA3 (EphA3)EphTK2qolAB-Human2836
EPHA3 (EphA3)EphTK4gk2AB7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2858
EPHA3 (EphA3)EphTK2qo7AAphosphoaminophosphonic acid-adenylate esterHuman2874
EPHA3 (EphA3)EphTK2qoqACphosphoaminophosphonic acid-adenylate esterHuman2879
EPHA3 (EphA3)EphTK4p5zA2-amino-1-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenyl]-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman2887
EPHA3 (EphA3)EphTK4p4cA2-amino-1-(3-methoxyphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman2875
EPHA3 (EphA3)EphTK2qo9AAphosphoaminophosphonic acid-adenylate esterHuman2862
EPHA3 (EphA3)EphTK2qobAA-Human2889
EPHA3 (EphA3)EphTK2qo7ACphosphoaminophosphonic acid-adenylate esterHuman2839
EPHA3 (EphA3)EphTK4twoAB5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acidHuman2848
EPHA3 (EphA3)EphTK2qodAA-Human2869
EPHA3 (EphA3)EphTK3dzqAAn-[2-methyl-5-({[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamideHuman2852
EPHA3 (EphA3)EphTK6in0AA1,4,7,10,13,16-hexaoxacyclooctadecaneHuman11792
EPHA3 (EphA3)EphTK2qobAC-Human2850
EPHA3 (EphA3)EphTK6in0AB1,4,7,10,13,16-hexaoxacyclooctadecaneHuman11793
EPHA3 (EphA3)EphTK2qocAB-Human2856
EPHA3 (EphA3)EphTK2qonAA-Human2867
EPHA3 (EphA3)EphTK2qo7ABphosphoaminophosphonic acid-adenylate esterHuman2857
EPHA3 (EphA3)EphTK3fxxABphosphoaminophosphonic acid-adenylate esterHuman2860
EPHA3 (EphA3)EphTK4gk3AB8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2885
EPHA3 (EphA3)EphTK2qooAB-Human2881
EPHA3 (EphA3)EphTK2qonAB-Human2853
EPHA3 (EphA3)EphTK4g2fAB1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-oneHuman2838
EPHA2 (EphA2)EphTK5ek7B-Human6321
EPHA2 (EphA2)EphTK5nk6AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(4-oxidanylcyclohexyl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8094
EPHA2 (EphA2)EphTK5nkaAB4-[[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylamino]cyclohexane-1-carboxylic acidHuman8086
EPHA2 (EphA2)EphTK6fnhAA1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10422
EPHA2 (EphA2)EphTK7kjaBBphosphomethylphosphonic acid adenylate esterHuman13251
EPHA2 (EphA2)EphTK5nkaAC-Human8083
EPHA2 (EphA2)EphTK6hesAC-Human11554
EPHA2 (EphA2)EphTK5nkfAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)-5-(trifluoromethyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8087
EPHA2 (EphA2)EphTK6q7cAB3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpiperidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11930
EPHA2 (EphA2)EphTK5nkgAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-ethyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8079
EPHA2 (EphA2)EphTK5ia0CBalisertibHuman7175
EPHA2 (EphA2)EphTK6fnfAA4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10417
EPHA2 (EphA2)EphTK6q7dAA3-[[4-imidazol-1-yl-6-(4-oxidanylpiperidin-1-yl)-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11937
EPHA2 (EphA2)EphTK5i9zAAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman7180
EPHA2 (EphA2)EphTK1mqbAphosphoaminophosphonic acid-adenylate esterHuman2088
EPHA2 (EphA2)EphTK5ia4AAn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman7189
EPHA2 (EphA2)EphTK8bokAA~{n}-(3,5-dimethoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14648
EPHA2 (EphA2)EphTK6heuAB3-[(4,6-dipyridin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11552
EPHA2 (EphA2)EphTK5i9xAA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman7182
EPHA2 (EphA2)EphTK6q7eAA3-[[4-imidazol-1-yl-6-[(3~{r})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11926
EPHB3 (EphB3)EphTK3zfyAB-Human538
EPHA2 (EphA2)EphTK5nkeAB2-[[3-bromanyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8063
EPHA2 (EphA2)EphTK6heyAB3-[(4,6-dipyridin-3-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11558
EPHA2 (EphA2)EphTK8bioAB8-(4-azanylbutyl)-6-[2-chloranyl-5-(trifluoromethyl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14513
EPHA2 (EphA2)EphTK6fngAB4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10416
EPHA2 (EphA2)EphTK8bogAB~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamideHuman14649
EPHA2 (EphA2)EphTK6fnfAB4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10420
EPHA2 (EphA2)EphTK5nkeAA2-[[3-bromanyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8078
EPHA2 (EphA2)EphTK6hevAB4-methyl-3-[(2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11565
EPHA2 (EphA2)EphTK5nk5AC-Human8091
EPHA2 (EphA2)EphTK6q7bAA3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11927
EPHA2 (EphA2)EphTK5nk4AA2-[[3-[[(4~{r})-3,3-bis(fluoranyl)piperidin-4-yl]carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8070
EPHA2 (EphA2)EphTK6fnhBB1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10413
EPHA2 (EphA2)EphTK8bocAB~{n}-[3,5-bis(trifluoromethyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman15002
EPHA2 (EphA2)EphTK5nk7AB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8081
EPHA2 (EphA2)EphTK5i9wABphosphoaminophosphonic acid-adenylate esterHuman7178
EPHA2 (EphA2)EphTK5nk0AB2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8096
EPHA2 (EphA2)EphTK5nkdAB2-[(3~{r})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidin-3-yl]ethanoic acidHuman8082
EPHA2 (EphA2)EphTK6fnhCB1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10419
EPHA2 (EphA2)EphTK5nkhAB2-[[3-(2-aminophenyl)-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8077
EPHA2 (EphA2)EphTK7kjaABphosphomethylphosphonic acid adenylate esterHuman13255
EPHA2 (EphA2)EphTK6hewAA4-methyl-3-[(1-methyl-6-pyrimidin-5-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11549
EPHA2 (EphA2)EphTK6fnhBA1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10421
EPHA2 (EphA2)EphTK5nkhAA2-[[3-(2-aminophenyl)-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8074
EPHA2 (EphA2)EphTK5nk1AA2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8064
EPHA2 (EphA2)EphTK6q7gAA3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11933
EPHA2 (EphA2)EphTK5ia4ABn-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamideHuman7168
EPHA2 (EphA2)EphTK8bk0AB~{n}-(2-chlorophenyl)-6-piperidin-4-yl-imidazo[1,2-a]pyridine-3-carboxamideHuman14503
EPHA2 (EphA2)EphTK8bk0AA~{n}-(2-chlorophenyl)-6-piperidin-4-yl-imidazo[1,2-a]pyridine-3-carboxamideHuman14504
EPHB4 (EphB4)EphTK6fnjAB4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10334
EPHB4 (EphB4)EphTK6fnlAA-Human10343
EPHB4 (EphB4)EphTK2vx0AAn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-morpholin-4-ylphenyl)pyrimidine-2,4-diamineHuman375
EPHB4 (EphB4)EphTK4bb4AAn-(2-methoxyethyl)-4-[(6-pyridin-4-ylquinazolin-2-yl)amino]benzamideHuman364
EPHB4 (EphB4)EphTK2yn8AstaurosporineHuman352
EPHA3 (EphA3)EphTK3fy2AB-Human2837
EPHA2 (EphA2)EphTK5i9yABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman7176
EPHB3 (EphB3)EphTK5l6pA~{n}-(4-phenylazanylquinazolin-7-yl)ethanamideHuman6937
EPHB3 (EphB3)EphTK3zfyBB-Human536
EPHB3 (EphB3)EphTK3zfyAA-Human537
EPHB3 (EphB3)EphTK3zfyBA-Human539
EPHB3 (EphB3)EphTK5l6oA1-(4-phenylazanylquinazolin-7-yl)ethanoneHuman6938
EPHB1 (EphB1)EphTK5mjbA2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamideHuman7584
EPHB1 (EphB1)EphTK7kplAA-Human13384
EPHB1 (EphB1)EphTK3zfxG-Human554
EPHB1 (EphB1)EphTK3zfxA-Human560
EPHB1 (EphB1)EphTK5mjaB2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamideHuman7583
EPHB1 (EphB1)EphTK7kplAB-Human13383
EPHB4 (EphB4)EphTK2vwwABn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3,4,5- trimethoxyphenyl)pyrimidine-2,4-diamineHuman358
EPHB4 (EphB4)EphTK2vwxAA3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamideHuman361
EPHB4 (EphB4)EphTK6fnmABn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman10339
EPHB4 (EphB4)EphTK2vwzABn-[3-[[4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl]amino]phenyl]methanesulfonamideHuman362
EPHB4 (EphB4)EphTK6fnmAAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman10342
EPHB4 (EphB4)EphTK2xvdAB{4-methyl-3-[(1-methylethyl)(2-{[3-(methylsulfonyl)-5-morpholin-4-ylphenyl]amino}pyrimidin-4-yl)amino]phenyl}methanolHuman372
EPHB4 (EphB4)EphTK2vx1AB3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzamideHuman374
EPHB4 (EphB4)EphTK4aw5AA(3z)-5-[(1-ethylpiperidin-4-yl)amino]-3-[(5-methoxy-1h-benzimidazol-2-yl)(phenyl)methylidene]-1,3-dihydro-2h-indol-2-oneHuman367
EPHA2 (EphA2)EphTK8qqyAB6-(4-fluoranyl-3-methoxy-phenyl)-13$l^{6}-thia-2,4,8,12,19-pentazatricyclo[12.3.1.1^{3,7}]nonadeca-1(18),3,5,7(19),14,16-hexaene 13,13-dioxideHuman15000
EPHB4 (EphB4)EphTK3zewBAstaurosporineHuman351
EPHA2 (EphA2)EphTK8bocAA~{n}-[3,5-bis(trifluoromethyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman15003
EPHA2 (EphA2)EphTK5ia1A4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman7191
EPHB4 (EphB4)EphTK2vx0ABn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-morpholin-4-ylphenyl)pyrimidine-2,4-diamineHuman368
EPHA2 (EphA2)EphTK8bogAC~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamideHuman14654
EPHA2 (EphA2)EphTK8bofAA4-methyl-~{n}-(3-methylphenyl)-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14656
EPHA2 (EphA2)EphTK8bohAA4-methyl-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14647
EPHA2 (EphA2)EphTK8boiAB4-methyl-~{n}-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14655
EPHA2 (EphA2)EphTK8bohAB4-methyl-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14651
EPHB4 (EphB4)EphTK6fnlAB-Human10335
EPHB4 (EphB4)EphTK6fnkAB1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10337
EPHB4 (EphB4)EphTK4bb4ABn-(2-methoxyethyl)-4-[(6-pyridin-4-ylquinazolin-2-yl)amino]benzamideHuman366
EPHB4 (EphB4)EphTK3zewAAstaurosporineHuman373
EPHA2 (EphA2)EphTK8xpvAB1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman15135
EPHB1 (EphB1)EphTK3zfxD-Human552
EPHB1 (EphB1)EphTK7kpmABadenosine-5'-diphosphateHuman13382
EPHA3 (EphA3)EphTK4p5qAA2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman2892
EPHA2 (EphA2)EphTK8boiAA4-methyl-~{n}-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14645
EPHA2 (EphA2)EphTK5nkcAB(3~{s})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidine-3-carboxylic acidHuman8072
EPHA2 (EphA2)EphTK8bodAB~{n}-[3,5-bis(chloranyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14646
EPHA2 (EphA2)EphTK8binAC8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14512
EPHA2 (EphA2)EphTK7kjaAAphosphomethylphosphonic acid adenylate esterHuman13250
EPHA2 (EphA2)EphTK5nkiAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]-1,3-thiazole-5-carboxamideHuman8084
EPHA2 (EphA2)EphTK6hetAC-Human11562
EPHA2 (EphA2)EphTK8xpvAA1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}ureaHuman15134
EPHA2 (EphA2)EphTK5i9xAB4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman7177
EPHA2 (EphA2)EphTK5ia0ABalisertibHuman7171
EPHA2 (EphA2)EphTK6fnhCA1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10415
EPHA2 (EphA2)EphTK5nkfAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)-5-(trifluoromethyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8071
EPHA2 (EphA2)EphTK5nk4AB2-[[3-[[(4~{r})-3,3-bis(fluoranyl)piperidin-4-yl]carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8076
EPHA2 (EphA2)EphTK6q7cAA3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpiperidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11931
EPHA2 (EphA2)EphTK5nkgAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-ethyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8090
EPHA2 (EphA2)EphTK6q7fAA3-[(4-imidazol-1-yl-6-piperazin-1-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11929
EPHA2 (EphA2)EphTK6hexAB4-methyl-3-[(1-methyl-6-pyrazin-2-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11555
EPHA2 (EphA2)EphTK5i9wAAphosphoaminophosphonic acid-adenylate esterHuman7187
EPHB4 (EphB4)EphTK2x9fABn^4^-1h-indazol-4-yl-n^2^-[3-(methylsulfonyl)phenyl]pyrimidine-2,4-diamineHuman359
EPHB4 (EphB4)EphTK2vwuAn-(5-chloro-1,3-benzodioxol-4-yl)-6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin-4-amineHuman370
EPHA2 (EphA2)EphTK8bodAA~{n}-[3,5-bis(chloranyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14657
EPHA2 (EphA2)EphTK8bomAA~{n}-(3-methoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14658
EPHA2 (EphA2)EphTK5ia3AB6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-oneHuman7184
EPHA2 (EphA2)EphTK5nk9AB(2~{z})-~{n}-(2-chloranyl-6-methyl-phenyl)-2-[3-[(4-methyl-4-oxidanyl-cyclohexyl)carbamoyl]phenyl]imino-1,3-thiazolidine-5-carboxamideHuman8067
EPHA2 (EphA2)EphTK8bokAB~{n}-(3,5-dimethoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14659
EPHA2 (EphA2)EphTK5nk5AA2-[[3-[(3-aminophenyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8068
EPHA2 (EphA2)EphTK7kjcBAphosphomethylphosphonic acid adenylate esterHuman13252
EPHA2 (EphA2)EphTK5i9uAA-Human7190
EPHA2 (EphA2)EphTK7kjbA-Human13253
EPHA2 (EphA2)EphTK5ia0BBalisertibHuman7179
EPHA2 (EphA2)EphTK5nk3AB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8080
EPHB1 (EphB1)EphTK7kpmAAadenosine-5'-diphosphateHuman13385
EPHA3 (EphA3)EphTK2qofAA-Human2888
EPHA3 (EphA3)EphTK2qo2AA-Human2880
EPHA3 (EphA3)EphTK3fy2AA-Human2851
EPHA3 (EphA3)EphTK4p5qAB2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamideHuman2878
EPHA3 (EphA3)EphTK4g2fAA1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-oneHuman2843
EPHA3 (EphA3)EphTK4twoAA5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acidHuman2893
EPHA3 (EphA3)EphTK2qolAD-Human2877
EPHA3 (EphA3)EphTK2qo2AB-Human2886
EPHA3 (EphA3)EphTK2qo9ABphosphoaminophosphonic acid-adenylate esterHuman2864
EPHA3 (EphA3)EphTK2qokAA-Human2873
EPHA3 (EphA3)EphTK2qocAC-Human2871
EPHA3 (EphA3)EphTK2qoiAB-Human2891
EPHA3 (EphA3)EphTK2qocAAphosphoaminophosphonic acid-adenylate esterHuman2882
EPHA3 (EphA3)EphTK2qokAC-Human2884
EPHA3 (EphA3)EphTK2qooAA-Human2847
EPHA3 (EphA3)EphTK2qokAB-Human2876
EPHA3 (EphA3)EphTK3dzqABn-[2-methyl-5-({[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamideHuman2868
EPHA3 (EphA3)EphTK2qofAB-Human2859
EPHA3 (EphA3)EphTK4twnAA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman2846
EPHA3 (EphA3)EphTK4gk4AB8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2840
EPHA3 (EphA3)EphTK2qoqABphosphoaminophosphonic acid-adenylate esterHuman2849
EPHA3 (EphA3)EphTK2qoiAA-Human2855
EPHA3 (EphA3)EphTK2qobAB-Human2872
EPHA3 (EphA3)EphTK4gk3AA8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman2844
EPHA3 (EphA3)EphTK2gsfA-Human2861
EPHA3 (EphA3)EphTK3fxxAAphosphoaminophosphonic acid-adenylate esterHuman2883
EPHA3 (EphA3)EphTK2qolAA-Human2863
EPHA3 (EphA3)EphTK2qolAC-Human2845
EPHA3 (EphA3)EphTK2qodAB-Human2842
EPHA2 (EphA2)EphTK6hetAA~{n}-(3-chlorophenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman11564
EPHA2 (EphA2)EphTK6q7gAC3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11934
EPHA2 (EphA2)EphTK6q7gAB3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11938
EPHA2 (EphA2)EphTK6hexAA4-methyl-3-[(1-methyl-6-pyrazin-2-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11559
EPHA2 (EphA2)EphTK5nk2AB-Human8060
EPHA2 (EphA2)EphTK5nk8AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(2,2,6,6-tetramethyl-1-oxidanyl-piperidin-4-yl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8062
EPHA2 (EphA2)EphTK4pdoB-Human2087
EPHA2 (EphA2)EphTK5ia5AAgolvatinibHuman7192
EPHA2 (EphA2)EphTK6fngAA4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman10414
EPHA2 (EphA2)EphTK5njzAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8093
EPHA2 (EphA2)EphTK5nk3AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8092
EPHA2 (EphA2)EphTK8qqyAA6-(4-fluoranyl-3-methoxy-phenyl)-13$l^{6}-thia-2,4,8,12,19-pentazatricyclo[12.3.1.1^{3,7}]nonadeca-1(18),3,5,7(19),14,16-hexaene 13,13-dioxideHuman15001
EPHA2 (EphA2)EphTK5nk2AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8100
EPHA2 (EphA2)EphTK5nk2AC~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8065
EPHA2 (EphA2)EphTK1mqbBphosphoaminophosphonic acid-adenylate esterHuman2089
EPHA2 (EphA2)EphTK8bomAB~{n}-(3-methoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman14653
EPHA2 (EphA2)EphTK5i9vAAphosphothiophosphoric acid-adenylate esterHuman7188
EPHA2 (EphA2)EphTK5i9uAB-Human7185
EPHA2 (EphA2)EphTK5ia2AA7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dioneHuman7170
EPHA2 (EphA2)EphTK5ia0BAalisertibHuman7174
EPHA2 (EphA2)EphTK6heuAA3-[(4,6-dipyridin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11563
EPHA2 (EphA2)EphTK6hevAA4-methyl-3-[(2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11561
EPHA2 (EphA2)EphTK6heyAA3-[(4,6-dipyridin-3-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11557
EPHA2 (EphA2)EphTK7kjcBBphosphomethylphosphonic acid adenylate esterHuman13254
EPHA2 (EphA2)EphTK5ia3AA6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-oneHuman7193
EPHA2 (EphA2)EphTK5njzAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamideHuman8085
EPHA2 (EphA2)EphTK8binAA8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14514
EPHA2 (EphA2)EphTK6fnhAB1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amineHuman10418
EPHA2 (EphA2)EphTK5ia5ABgolvatinibHuman7183
EPHA2 (EphA2)EphTK8binAB8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman14515
EPHA2 (EphA2)EphTK6hewAB4-methyl-3-[(1-methyl-6-pyrimidin-5-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11556
EPHA2 (EphA2)EphTK5ia0AAalisertibHuman7169
EPHA2 (EphA2)EphTK5nkiAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]-1,3-thiazole-5-carboxamideHuman8069
EPHA2 (EphA2)EphTK5nkbAB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3,5-dimorpholin-4-ylphenyl)amino]-1,3-thiazole-5-carboxamideHuman8097
EPHA2 (EphA2)EphTK5nkdAA2-[(3~{r})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidin-3-yl]ethanoic acidHuman8058
EPHA2 (EphA2)EphTK5i9vABphosphothiophosphoric acid-adenylate esterHuman7173
EPHA2 (EphA2)EphTK7kjcABphosphomethylphosphonic acid adenylate esterHuman13256
EPHA2 (EphA2)EphTK5nkbAA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3,5-dimorpholin-4-ylphenyl)amino]-1,3-thiazole-5-carboxamideHuman8098
EPHA2 (EphA2)EphTK5nk8AB~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(2,2,6,6-tetramethyl-1-oxidanyl-piperidin-4-yl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8088
EPHA2 (EphA2)EphTK5ek7A-Human6322
EPHA2 (EphA2)EphTK6q7fAB3-[(4-imidazol-1-yl-6-piperazin-1-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamideHuman11936
EPHA2 (EphA2)EphTK6hetAB~{n}-(3-chlorophenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman11560
EPHA2 (EphA2)EphTK5nk5AB2-[[3-[(3-aminophenyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8066
EPHA2 (EphA2)EphTK5nkcAA(3~{s})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidine-3-carboxylic acidHuman8099
EPHA2 (EphA2)EphTK5nk1AB2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8059
EPHA2 (EphA2)EphTK7kjcAAphosphomethylphosphonic acid adenylate esterHuman13257
EPHA2 (EphA2)EphTK5nk7AA~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamideHuman8089
EPHA2 (EphA2)EphTK4pdoA-Human2086
EPHA2 (EphA2)EphTK5nk0AA2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamideHuman8095
EPHB4 (EphB4)EphTK2vwxAB3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamideHuman350
EPHB4 (EphB4)EphTK3zewABstaurosporineHuman377
EPHB4 (EphB4)EphTK2vwvAAn'-(3-chloro-4-methoxy-phenyl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazine-2,4-diamineHuman365
EPHB4 (EphB4)EphTK3zewBBstaurosporineHuman357
EPHB4 (EphB4)EphTK2vx1AA3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzamideHuman371
EPHB4 (EphB4)EphTK2vwwAAn'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3,4,5- trimethoxyphenyl)pyrimidine-2,4-diamineHuman356
EPHB1 (EphB1)EphTK3zfxI-Human559
EPHB1 (EphB1)EphTK6umwAB7-chlorotetracyclineHuman12923
EPHB1 (EphB1)EphTK3zfxC-Human557
EPHB1 (EphB1)EphTK5mjbB2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamideHuman7585
EPHB1 (EphB1)EphTK5mjaA2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamideHuman7582
EPHB1 (EphB1)EphTK3zfxH-Human556
EPHB1 (EphB1)EphTK3zfxB-Human558
EPHB1 (EphB1)EphTK3zfxE-Human555
EPHB1 (EphB1)EphTK3zfxF-Human553
EPHA5 (EphA5)EphTK2r2pAB-Human3413
EPHA5 (EphA5)EphTK2r2pAA-Human3412
EPHB2 (EphB2)EphTK3zfmA-Human2731