| EPHA2 (EphA2) | Eph | TK | 6q7d | A | B | 3-[[4-imidazol-1-yl-6-(4-oxidanylpiperidin-1-yl)-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11928 | |
| EPHA2 (EphA2) | Eph | TK | 4p2k | A | | - | Human | 2091 | |
| EPHA2 (EphA2) | Eph | TK | 4trl | A | | - | Human | 2090 | |
| EPHA3 (EphA3) | Eph | TK | 2qod | A | C | - | Human | 2866 | |
| EPHA2 (EphA2) | Eph | TK | 5i9z | A | B | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 7181 | |
| EPHA2 (EphA2) | Eph | TK | 5i9y | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7194 | |
| EPHA2 (EphA2) | Eph | TK | 5ia2 | A | B | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 7172 | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | B | A | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10340 | |
| EPHB4 (EphB4) | Eph | TK | 2vwy | A | A | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-methylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 353 | |
| EPHA2 (EphA2) | Eph | TK | 6hes | A | B | 4-methyl-3-[(2-pyridin-3-ylquinazolin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11566 | |
| EPHB4 (EphB4) | Eph | TK | 2yn8 | B | | staurosporine | Human | 349 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | C | A | alisertib | Human | 7186 | |
| EPHB4 (EphB4) | Eph | TK | 2vwy | A | B | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-methylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 355 | |
| EPHA3 (EphA3) | Eph | TK | 4twn | A | B | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 2865 | |
| EPHA2 (EphA2) | Eph | TK | 6hew | A | C | - | Human | 11553 | |
| EPHA7 (EphA7) | Eph | TK | 2rei | A | A | - | Human | 4 | |
| EPHA7 (EphA7) | Eph | TK | 7eec | A | B | - | Human | 13790 | |
| EPHA7 (EphA7) | Eph | TK | 7eed | A | | - | Human | 13791 | |
| EPHA7 (EphA7) | Eph | TK | 7eec | A | A | - | Human | 13792 | |
| EPHA7 (EphA7) | Eph | TK | 3dko | A | A | 5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamide | Human | 1 | |
| EPHA7 (EphA7) | Eph | TK | 2rei | A | B | - | Human | 2 | |
| EPHA7 (EphA7) | Eph | TK | 7eef | A | | - | Human | 13793 | |
| EPHA7 (EphA7) | Eph | TK | 3dko | A | B | 5-[(2-methyl-5-{[3-(trifluoromethyl)phenyl]carbamoyl}phenyl)amino]pyridine-3-carboxamide | Human | 3 | |
| EPHA2 (EphA2) | Eph | TK | 5nk9 | A | A | (2~{z})-~{n}-(2-chloranyl-6-methyl-phenyl)-2-[3-[(4-methyl-4-oxidanyl-cyclohexyl)carbamoyl]phenyl]imino-1,3-thiazolidine-5-carboxamide | Human | 8073 | |
| EPHA2 (EphA2) | Eph | TK | 5nk6 | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(4-oxidanylcyclohexyl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8061 | |
| EPHA2 (EphA2) | Eph | TK | 6q7e | A | B | 3-[[4-imidazol-1-yl-6-[(3~{r})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11932 | |
| EPHA2 (EphA2) | Eph | TK | 5nka | A | A | 4-[[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylamino]cyclohexane-1-carboxylic acid | Human | 8075 | |
| EPHA2 (EphA2) | Eph | TK | 6hex | A | C | - | Human | 11551 | |
| EPHA2 (EphA2) | Eph | TK | 6q7b | A | B | 3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11935 | |
| EPHB4 (EphB4) | Eph | TK | 6fni | A | B | 4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10333 | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | B | B | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10341 | |
| EPHB4 (EphB4) | Eph | TK | 6fnk | A | A | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10344 | |
| EPHB4 (EphB4) | Eph | TK | 2vwz | A | A | n-[3-[[4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl]amino]phenyl]methanesulfonamide | Human | 360 | |
| EPHA2 (EphA2) | Eph | TK | 8bof | A | B | 4-methyl-~{n}-(3-methylphenyl)-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14652 | |
| EPHA8 (EphA8) | Eph | TK | 3kul | B | A | - | Human | 1249 | |
| EPHA8 (EphA8) | Eph | TK | 3kul | B | B | - | Human | 1250 | |
| EPHA8 (EphA8) | Eph | TK | 3kul | A | B | - | Human | 1252 | |
| EPHA8 (EphA8) | Eph | TK | 3kul | A | A | - | Human | 1251 | |
| EPHA2 (EphA2) | Eph | TK | 8bog | A | A | ~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamide | Human | 14650 | |
| EPHB1 (EphB1) | Eph | TK | 6umw | A | A | 7-chlorotetracycline | Human | 12924 | |
| EPHB4 (EphB4) | Eph | TK | 2xvd | A | A | {4-methyl-3-[(1-methylethyl)(2-{[3-(methylsulfonyl)-5-morpholin-4-ylphenyl]amino}pyrimidin-4-yl)amino]phenyl}methanol | Human | 363 | |
| EPHB4 (EphB4) | Eph | TK | 2x9f | A | A | n^4^-1h-indazol-4-yl-n^2^-[3-(methylsulfonyl)phenyl]pyrimidine-2,4-diamine | Human | 354 | |
| EPHB4 (EphB4) | Eph | TK | 2vwv | A | B | n'-(3-chloro-4-methoxy-phenyl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazine-2,4-diamine | Human | 369 | |
| EPHA3 (EphA3) | Eph | TK | 2qoq | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2890 | |
| EPHB4 (EphB4) | Eph | TK | 4aw5 | A | B | (3z)-5-[(1-ethylpiperidin-4-yl)amino]-3-[(5-methoxy-1h-benzimidazol-2-yl)(phenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 376 | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | A | A | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10336 | |
| EPHA3 (EphA3) | Eph | TK | 4gk2 | A | A | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2841 | |
| EPHB4 (EphB4) | Eph | TK | 6fni | A | A | 4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10338 | |
| EPHA2 (EphA2) | Eph | TK | 7kja | B | A | phosphomethylphosphonic acid adenylate ester | Human | 13249 | |
| EPHA2 (EphA2) | Eph | TK | 6hes | A | A | 4-methyl-3-[(2-pyridin-3-ylquinazolin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11550 | |
| EPHA3 (EphA3) | Eph | TK | 4gk4 | A | A | 8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2854 | |
| EPHA3 (EphA3) | Eph | TK | 2qof | A | C | - | Human | 2870 | |
| EPHA3 (EphA3) | Eph | TK | 2qol | A | B | - | Human | 2836 | |
| EPHA3 (EphA3) | Eph | TK | 4gk2 | A | B | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2858 | |
| EPHA3 (EphA3) | Eph | TK | 2qo7 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2874 | |
| EPHA3 (EphA3) | Eph | TK | 2qoq | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 2879 | |
| EPHA3 (EphA3) | Eph | TK | 4p5z | A | | 2-amino-1-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenyl]-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 2887 | |
| EPHA3 (EphA3) | Eph | TK | 4p4c | A | | 2-amino-1-(3-methoxyphenyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 2875 | |
| EPHA3 (EphA3) | Eph | TK | 2qo9 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2862 | |
| EPHA3 (EphA3) | Eph | TK | 2qob | A | A | - | Human | 2889 | |
| EPHA3 (EphA3) | Eph | TK | 2qo7 | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 2839 | |
| EPHA3 (EphA3) | Eph | TK | 4two | A | B | 5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acid | Human | 2848 | |
| EPHA3 (EphA3) | Eph | TK | 2qod | A | A | - | Human | 2869 | |
| EPHA3 (EphA3) | Eph | TK | 3dzq | A | A | n-[2-methyl-5-({[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamide | Human | 2852 | |
| EPHA3 (EphA3) | Eph | TK | 6in0 | A | A | 1,4,7,10,13,16-hexaoxacyclooctadecane | Human | 11792 | |
| EPHA3 (EphA3) | Eph | TK | 2qob | A | C | - | Human | 2850 | |
| EPHA3 (EphA3) | Eph | TK | 6in0 | A | B | 1,4,7,10,13,16-hexaoxacyclooctadecane | Human | 11793 | |
| EPHA3 (EphA3) | Eph | TK | 2qoc | A | B | - | Human | 2856 | |
| EPHA3 (EphA3) | Eph | TK | 2qon | A | A | - | Human | 2867 | |
| EPHA3 (EphA3) | Eph | TK | 2qo7 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2857 | |
| EPHA3 (EphA3) | Eph | TK | 3fxx | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2860 | |
| EPHA3 (EphA3) | Eph | TK | 4gk3 | A | B | 8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2885 | |
| EPHA3 (EphA3) | Eph | TK | 2qoo | A | B | - | Human | 2881 | |
| EPHA3 (EphA3) | Eph | TK | 2qon | A | B | - | Human | 2853 | |
| EPHA3 (EphA3) | Eph | TK | 4g2f | A | B | 1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-one | Human | 2838 | |
| EPHA2 (EphA2) | Eph | TK | 5ek7 | B | | - | Human | 6321 | |
| EPHA2 (EphA2) | Eph | TK | 5nk6 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(4-oxidanylcyclohexyl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8094 | |
| EPHA2 (EphA2) | Eph | TK | 5nka | A | B | 4-[[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylamino]cyclohexane-1-carboxylic acid | Human | 8086 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | A | A | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10422 | |
| EPHA2 (EphA2) | Eph | TK | 7kja | B | B | phosphomethylphosphonic acid adenylate ester | Human | 13251 | |
| EPHA2 (EphA2) | Eph | TK | 5nka | A | C | - | Human | 8083 | |
| EPHA2 (EphA2) | Eph | TK | 6hes | A | C | - | Human | 11554 | |
| EPHA2 (EphA2) | Eph | TK | 5nkf | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)-5-(trifluoromethyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8087 | |
| EPHA2 (EphA2) | Eph | TK | 6q7c | A | B | 3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpiperidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11930 | |
| EPHA2 (EphA2) | Eph | TK | 5nkg | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-ethyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8079 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | C | B | alisertib | Human | 7175 | |
| EPHA2 (EphA2) | Eph | TK | 6fnf | A | A | 4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10417 | |
| EPHA2 (EphA2) | Eph | TK | 6q7d | A | A | 3-[[4-imidazol-1-yl-6-(4-oxidanylpiperidin-1-yl)-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11937 | |
| EPHA2 (EphA2) | Eph | TK | 5i9z | A | A | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 7180 | |
| EPHA2 (EphA2) | Eph | TK | 1mqb | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2088 | |
| EPHA2 (EphA2) | Eph | TK | 5ia4 | A | A | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 7189 | |
| EPHA2 (EphA2) | Eph | TK | 8bok | A | A | ~{n}-(3,5-dimethoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14648 | |
| EPHA2 (EphA2) | Eph | TK | 6heu | A | B | 3-[(4,6-dipyridin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11552 | |
| EPHA2 (EphA2) | Eph | TK | 5i9x | A | A | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 7182 | |
| EPHA2 (EphA2) | Eph | TK | 6q7e | A | A | 3-[[4-imidazol-1-yl-6-[(3~{r})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11926 | |
| EPHB3 (EphB3) | Eph | TK | 3zfy | A | B | - | Human | 538 | |
| EPHA2 (EphA2) | Eph | TK | 5nke | A | B | 2-[[3-bromanyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8063 | |
| EPHA2 (EphA2) | Eph | TK | 6hey | A | B | 3-[(4,6-dipyridin-3-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11558 | |
| EPHA2 (EphA2) | Eph | TK | 8bio | A | B | 8-(4-azanylbutyl)-6-[2-chloranyl-5-(trifluoromethyl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14513 | |
| EPHA2 (EphA2) | Eph | TK | 6fng | A | B | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10416 | |
| EPHA2 (EphA2) | Eph | TK | 8bog | A | B | ~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamide | Human | 14649 | |
| EPHA2 (EphA2) | Eph | TK | 6fnf | A | B | 4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10420 | |
| EPHA2 (EphA2) | Eph | TK | 5nke | A | A | 2-[[3-bromanyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8078 | |
| EPHA2 (EphA2) | Eph | TK | 6hev | A | B | 4-methyl-3-[(2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11565 | |
| EPHA2 (EphA2) | Eph | TK | 5nk5 | A | C | - | Human | 8091 | |
| EPHA2 (EphA2) | Eph | TK | 6q7b | A | A | 3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpyrrolidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11927 | |
| EPHA2 (EphA2) | Eph | TK | 5nk4 | A | A | 2-[[3-[[(4~{r})-3,3-bis(fluoranyl)piperidin-4-yl]carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8070 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | B | B | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10413 | |
| EPHA2 (EphA2) | Eph | TK | 8boc | A | B | ~{n}-[3,5-bis(trifluoromethyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 15002 | |
| EPHA2 (EphA2) | Eph | TK | 5nk7 | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8081 | |
| EPHA2 (EphA2) | Eph | TK | 5i9w | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 7178 | |
| EPHA2 (EphA2) | Eph | TK | 5nk0 | A | B | 2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8096 | |
| EPHA2 (EphA2) | Eph | TK | 5nkd | A | B | 2-[(3~{r})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidin-3-yl]ethanoic acid | Human | 8082 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | C | B | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10419 | |
| EPHA2 (EphA2) | Eph | TK | 5nkh | A | B | 2-[[3-(2-aminophenyl)-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8077 | |
| EPHA2 (EphA2) | Eph | TK | 7kja | A | B | phosphomethylphosphonic acid adenylate ester | Human | 13255 | |
| EPHA2 (EphA2) | Eph | TK | 6hew | A | A | 4-methyl-3-[(1-methyl-6-pyrimidin-5-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11549 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | B | A | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10421 | |
| EPHA2 (EphA2) | Eph | TK | 5nkh | A | A | 2-[[3-(2-aminophenyl)-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8074 | |
| EPHA2 (EphA2) | Eph | TK | 5nk1 | A | A | 2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8064 | |
| EPHA2 (EphA2) | Eph | TK | 6q7g | A | A | 3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11933 | |
| EPHA2 (EphA2) | Eph | TK | 5ia4 | A | B | n-(3-fluoro-4-{[6-methoxy-7-(3-morpholin-4-ylpropoxy)quinolin-4-yl]oxy}phenyl)-n'-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide | Human | 7168 | |
| EPHA2 (EphA2) | Eph | TK | 8bk0 | A | B | ~{n}-(2-chlorophenyl)-6-piperidin-4-yl-imidazo[1,2-a]pyridine-3-carboxamide | Human | 14503 | |
| EPHA2 (EphA2) | Eph | TK | 8bk0 | A | A | ~{n}-(2-chlorophenyl)-6-piperidin-4-yl-imidazo[1,2-a]pyridine-3-carboxamide | Human | 14504 | |
| EPHB4 (EphB4) | Eph | TK | 6fnj | A | B | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10334 | |
| EPHB4 (EphB4) | Eph | TK | 6fnl | A | A | - | Human | 10343 | |
| EPHB4 (EphB4) | Eph | TK | 2vx0 | A | A | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-morpholin-4-ylphenyl)pyrimidine-2,4-diamine | Human | 375 | |
| EPHB4 (EphB4) | Eph | TK | 4bb4 | A | A | n-(2-methoxyethyl)-4-[(6-pyridin-4-ylquinazolin-2-yl)amino]benzamide | Human | 364 | |
| EPHB4 (EphB4) | Eph | TK | 2yn8 | A | | staurosporine | Human | 352 | |
| EPHA3 (EphA3) | Eph | TK | 3fy2 | A | B | - | Human | 2837 | |
| EPHA2 (EphA2) | Eph | TK | 5i9y | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7176 | |
| EPHB3 (EphB3) | Eph | TK | 5l6p | A | | ~{n}-(4-phenylazanylquinazolin-7-yl)ethanamide | Human | 6937 | |
| EPHB3 (EphB3) | Eph | TK | 3zfy | B | B | - | Human | 536 | |
| EPHB3 (EphB3) | Eph | TK | 3zfy | A | A | - | Human | 537 | |
| EPHB3 (EphB3) | Eph | TK | 3zfy | B | A | - | Human | 539 | |
| EPHB3 (EphB3) | Eph | TK | 5l6o | A | | 1-(4-phenylazanylquinazolin-7-yl)ethanone | Human | 6938 | |
| EPHB1 (EphB1) | Eph | TK | 5mjb | A | | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | 7584 | |
| EPHB1 (EphB1) | Eph | TK | 7kpl | A | A | - | Human | 13384 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | G | | - | Human | 554 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | A | | - | Human | 560 | |
| EPHB1 (EphB1) | Eph | TK | 5mja | B | | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | 7583 | |
| EPHB1 (EphB1) | Eph | TK | 7kpl | A | B | - | Human | 13383 | |
| EPHB4 (EphB4) | Eph | TK | 2vww | A | B | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3,4,5- trimethoxyphenyl)pyrimidine-2,4-diamine | Human | 358 | |
| EPHB4 (EphB4) | Eph | TK | 2vwx | A | A | 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 361 | |
| EPHB4 (EphB4) | Eph | TK | 6fnm | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 10339 | |
| EPHB4 (EphB4) | Eph | TK | 2vwz | A | B | n-[3-[[4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl]amino]phenyl]methanesulfonamide | Human | 362 | |
| EPHB4 (EphB4) | Eph | TK | 6fnm | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 10342 | |
| EPHB4 (EphB4) | Eph | TK | 2xvd | A | B | {4-methyl-3-[(1-methylethyl)(2-{[3-(methylsulfonyl)-5-morpholin-4-ylphenyl]amino}pyrimidin-4-yl)amino]phenyl}methanol | Human | 372 | |
| EPHB4 (EphB4) | Eph | TK | 2vx1 | A | B | 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzamide | Human | 374 | |
| EPHB4 (EphB4) | Eph | TK | 4aw5 | A | A | (3z)-5-[(1-ethylpiperidin-4-yl)amino]-3-[(5-methoxy-1h-benzimidazol-2-yl)(phenyl)methylidene]-1,3-dihydro-2h-indol-2-one | Human | 367 | |
| EPHA2 (EphA2) | Eph | TK | 8qqy | A | B | 6-(4-fluoranyl-3-methoxy-phenyl)-13$l^{6}-thia-2,4,8,12,19-pentazatricyclo[12.3.1.1^{3,7}]nonadeca-1(18),3,5,7(19),14,16-hexaene 13,13-dioxide | Human | 15000 | |
| EPHB4 (EphB4) | Eph | TK | 3zew | B | A | staurosporine | Human | 351 | |
| EPHA2 (EphA2) | Eph | TK | 8boc | A | A | ~{n}-[3,5-bis(trifluoromethyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 15003 | |
| EPHA2 (EphA2) | Eph | TK | 5ia1 | A | | 4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acid | Human | 7191 | |
| EPHB4 (EphB4) | Eph | TK | 2vx0 | A | B | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3-morpholin-4-ylphenyl)pyrimidine-2,4-diamine | Human | 368 | |
| EPHA2 (EphA2) | Eph | TK | 8bog | A | C | ~{n}-[4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]phenyl]-3-(trifluoromethyl)benzamide | Human | 14654 | |
| EPHA2 (EphA2) | Eph | TK | 8bof | A | A | 4-methyl-~{n}-(3-methylphenyl)-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14656 | |
| EPHA2 (EphA2) | Eph | TK | 8boh | A | A | 4-methyl-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14647 | |
| EPHA2 (EphA2) | Eph | TK | 8boi | A | B | 4-methyl-~{n}-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14655 | |
| EPHA2 (EphA2) | Eph | TK | 8boh | A | B | 4-methyl-~{n}-[3-(4-methylimidazol-1-yl)-5-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14651 | |
| EPHB4 (EphB4) | Eph | TK | 6fnl | A | B | - | Human | 10335 | |
| EPHB4 (EphB4) | Eph | TK | 6fnk | A | B | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10337 | |
| EPHB4 (EphB4) | Eph | TK | 4bb4 | A | B | n-(2-methoxyethyl)-4-[(6-pyridin-4-ylquinazolin-2-yl)amino]benzamide | Human | 366 | |
| EPHB4 (EphB4) | Eph | TK | 3zew | A | A | staurosporine | Human | 373 | |
| EPHA2 (EphA2) | Eph | TK | 8xpv | A | B | 1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}urea | Human | 15135 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | D | | - | Human | 552 | |
| EPHB1 (EphB1) | Eph | TK | 7kpm | A | B | adenosine-5'-diphosphate | Human | 13382 | |
| EPHA3 (EphA3) | Eph | TK | 4p5q | A | A | 2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 2892 | |
| EPHA2 (EphA2) | Eph | TK | 8boi | A | A | 4-methyl-~{n}-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14645 | |
| EPHA2 (EphA2) | Eph | TK | 5nkc | A | B | (3~{s})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidine-3-carboxylic acid | Human | 8072 | |
| EPHA2 (EphA2) | Eph | TK | 8bod | A | B | ~{n}-[3,5-bis(chloranyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14646 | |
| EPHA2 (EphA2) | Eph | TK | 8bin | A | C | 8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14512 | |
| EPHA2 (EphA2) | Eph | TK | 7kja | A | A | phosphomethylphosphonic acid adenylate ester | Human | 13250 | |
| EPHA2 (EphA2) | Eph | TK | 5nki | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]-1,3-thiazole-5-carboxamide | Human | 8084 | |
| EPHA2 (EphA2) | Eph | TK | 6het | A | C | - | Human | 11562 | |
| EPHA2 (EphA2) | Eph | TK | 8xpv | A | A | 1-(3,3-dimethylbutyl)-3-{2-fluoro-4-methyl-5-[7-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-6-yl]phenyl}urea | Human | 15134 | |
| EPHA2 (EphA2) | Eph | TK | 5i9x | A | B | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 7177 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | A | B | alisertib | Human | 7171 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | C | A | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10415 | |
| EPHA2 (EphA2) | Eph | TK | 5nkf | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)-5-(trifluoromethyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8071 | |
| EPHA2 (EphA2) | Eph | TK | 5nk4 | A | B | 2-[[3-[[(4~{r})-3,3-bis(fluoranyl)piperidin-4-yl]carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8076 | |
| EPHA2 (EphA2) | Eph | TK | 6q7c | A | A | 3-[[4-imidazol-1-yl-6-[(3~{s})-3-oxidanylpiperidin-1-yl]-1,3,5-triazin-2-yl]amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11931 | |
| EPHA2 (EphA2) | Eph | TK | 5nkg | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-ethyl-5-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8090 | |
| EPHA2 (EphA2) | Eph | TK | 6q7f | A | A | 3-[(4-imidazol-1-yl-6-piperazin-1-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11929 | |
| EPHA2 (EphA2) | Eph | TK | 6hex | A | B | 4-methyl-3-[(1-methyl-6-pyrazin-2-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11555 | |
| EPHA2 (EphA2) | Eph | TK | 5i9w | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 7187 | |
| EPHB4 (EphB4) | Eph | TK | 2x9f | A | B | n^4^-1h-indazol-4-yl-n^2^-[3-(methylsulfonyl)phenyl]pyrimidine-2,4-diamine | Human | 359 | |
| EPHB4 (EphB4) | Eph | TK | 2vwu | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-6-methoxy-7-(3-piperidin-1-ylpropoxy)quinazolin-4-amine | Human | 370 | |
| EPHA2 (EphA2) | Eph | TK | 8bod | A | A | ~{n}-[3,5-bis(chloranyl)phenyl]-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14657 | |
| EPHA2 (EphA2) | Eph | TK | 8bom | A | A | ~{n}-(3-methoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14658 | |
| EPHA2 (EphA2) | Eph | TK | 5ia3 | A | B | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Human | 7184 | |
| EPHA2 (EphA2) | Eph | TK | 5nk9 | A | B | (2~{z})-~{n}-(2-chloranyl-6-methyl-phenyl)-2-[3-[(4-methyl-4-oxidanyl-cyclohexyl)carbamoyl]phenyl]imino-1,3-thiazolidine-5-carboxamide | Human | 8067 | |
| EPHA2 (EphA2) | Eph | TK | 8bok | A | B | ~{n}-(3,5-dimethoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14659 | |
| EPHA2 (EphA2) | Eph | TK | 5nk5 | A | A | 2-[[3-[(3-aminophenyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8068 | |
| EPHA2 (EphA2) | Eph | TK | 7kjc | B | A | phosphomethylphosphonic acid adenylate ester | Human | 13252 | |
| EPHA2 (EphA2) | Eph | TK | 5i9u | A | A | - | Human | 7190 | |
| EPHA2 (EphA2) | Eph | TK | 7kjb | A | | - | Human | 13253 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | B | B | alisertib | Human | 7179 | |
| EPHA2 (EphA2) | Eph | TK | 5nk3 | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8080 | |
| EPHB1 (EphB1) | Eph | TK | 7kpm | A | A | adenosine-5'-diphosphate | Human | 13385 | |
| EPHA3 (EphA3) | Eph | TK | 2qof | A | A | - | Human | 2888 | |
| EPHA3 (EphA3) | Eph | TK | 2qo2 | A | A | - | Human | 2880 | |
| EPHA3 (EphA3) | Eph | TK | 3fy2 | A | A | - | Human | 2851 | |
| EPHA3 (EphA3) | Eph | TK | 4p5q | A | B | 2-amino-1-(2-chlorophenyl)-n-(3-ethoxypropyl)-1h-pyrrolo[2,3-b]quinoxaline-3-carboxamide | Human | 2878 | |
| EPHA3 (EphA3) | Eph | TK | 4g2f | A | A | 1-amino-5-(5-hydroxy-2-methylphenyl)-7,8,9,10-tetrahydropyrimido[4,5-c]isoquinolin-6(5h)-one | Human | 2843 | |
| EPHA3 (EphA3) | Eph | TK | 4two | A | A | 5-{[3-carbamoyl-4-(3,4-dimethylphenyl)-5-methylthiophen-2-yl]amino}-5-oxopentanoic acid | Human | 2893 | |
| EPHA3 (EphA3) | Eph | TK | 2qol | A | D | - | Human | 2877 | |
| EPHA3 (EphA3) | Eph | TK | 2qo2 | A | B | - | Human | 2886 | |
| EPHA3 (EphA3) | Eph | TK | 2qo9 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2864 | |
| EPHA3 (EphA3) | Eph | TK | 2qok | A | A | - | Human | 2873 | |
| EPHA3 (EphA3) | Eph | TK | 2qoc | A | C | - | Human | 2871 | |
| EPHA3 (EphA3) | Eph | TK | 2qoi | A | B | - | Human | 2891 | |
| EPHA3 (EphA3) | Eph | TK | 2qoc | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2882 | |
| EPHA3 (EphA3) | Eph | TK | 2qok | A | C | - | Human | 2884 | |
| EPHA3 (EphA3) | Eph | TK | 2qoo | A | A | - | Human | 2847 | |
| EPHA3 (EphA3) | Eph | TK | 2qok | A | B | - | Human | 2876 | |
| EPHA3 (EphA3) | Eph | TK | 3dzq | A | B | n-[2-methyl-5-({[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]carbonyl}amino)phenyl]isoxazole-5-carboxamide | Human | 2868 | |
| EPHA3 (EphA3) | Eph | TK | 2qof | A | B | - | Human | 2859 | |
| EPHA3 (EphA3) | Eph | TK | 4twn | A | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 2846 | |
| EPHA3 (EphA3) | Eph | TK | 4gk4 | A | B | 8-butyl-1-methyl-7-(5-methyl-1h-indazol-4-yl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2840 | |
| EPHA3 (EphA3) | Eph | TK | 2qoq | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2849 | |
| EPHA3 (EphA3) | Eph | TK | 2qoi | A | A | - | Human | 2855 | |
| EPHA3 (EphA3) | Eph | TK | 2qob | A | B | - | Human | 2872 | |
| EPHA3 (EphA3) | Eph | TK | 4gk3 | A | A | 8-butyl-1-methyl-7-(2-methylphenyl)-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 2844 | |
| EPHA3 (EphA3) | Eph | TK | 2gsf | A | | - | Human | 2861 | |
| EPHA3 (EphA3) | Eph | TK | 3fxx | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2883 | |
| EPHA3 (EphA3) | Eph | TK | 2qol | A | A | - | Human | 2863 | |
| EPHA3 (EphA3) | Eph | TK | 2qol | A | C | - | Human | 2845 | |
| EPHA3 (EphA3) | Eph | TK | 2qod | A | B | - | Human | 2842 | |
| EPHA2 (EphA2) | Eph | TK | 6het | A | A | ~{n}-(3-chlorophenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 11564 | |
| EPHA2 (EphA2) | Eph | TK | 6q7g | A | C | 3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11934 | |
| EPHA2 (EphA2) | Eph | TK | 6q7g | A | B | 3-[(4-imidazol-1-yl-6-morpholin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11938 | |
| EPHA2 (EphA2) | Eph | TK | 6hex | A | A | 4-methyl-3-[(1-methyl-6-pyrazin-2-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11559 | |
| EPHA2 (EphA2) | Eph | TK | 5nk2 | A | B | - | Human | 8060 | |
| EPHA2 (EphA2) | Eph | TK | 5nk8 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(2,2,6,6-tetramethyl-1-oxidanyl-piperidin-4-yl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8062 | |
| EPHA2 (EphA2) | Eph | TK | 4pdo | B | | - | Human | 2087 | |
| EPHA2 (EphA2) | Eph | TK | 5ia5 | A | A | golvatinib | Human | 7192 | |
| EPHA2 (EphA2) | Eph | TK | 6fng | A | A | 4-methyl-3-[(2-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 10414 | |
| EPHA2 (EphA2) | Eph | TK | 5njz | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8093 | |
| EPHA2 (EphA2) | Eph | TK | 5nk3 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{s})-pyrrolidin-3-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8092 | |
| EPHA2 (EphA2) | Eph | TK | 8qqy | A | A | 6-(4-fluoranyl-3-methoxy-phenyl)-13$l^{6}-thia-2,4,8,12,19-pentazatricyclo[12.3.1.1^{3,7}]nonadeca-1(18),3,5,7(19),14,16-hexaene 13,13-dioxide | Human | 15001 | |
| EPHA2 (EphA2) | Eph | TK | 5nk2 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8100 | |
| EPHA2 (EphA2) | Eph | TK | 5nk2 | A | C | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8065 | |
| EPHA2 (EphA2) | Eph | TK | 1mqb | B | | phosphoaminophosphonic acid-adenylate ester | Human | 2089 | |
| EPHA2 (EphA2) | Eph | TK | 8bom | A | B | ~{n}-(3-methoxyphenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 14653 | |
| EPHA2 (EphA2) | Eph | TK | 5i9v | A | A | phosphothiophosphoric acid-adenylate ester | Human | 7188 | |
| EPHA2 (EphA2) | Eph | TK | 5i9u | A | B | - | Human | 7185 | |
| EPHA2 (EphA2) | Eph | TK | 5ia2 | A | A | 7-(5-hydroxy-2-methylphenyl)-8-(2-methoxyphenyl)-1-methyl-1h-imidazo[2,1-f]purine-2,4(3h,8h)-dione | Human | 7170 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | B | A | alisertib | Human | 7174 | |
| EPHA2 (EphA2) | Eph | TK | 6heu | A | A | 3-[(4,6-dipyridin-4-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11563 | |
| EPHA2 (EphA2) | Eph | TK | 6hev | A | A | 4-methyl-3-[(2-pyridin-3-ylpyrido[2,3-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11561 | |
| EPHA2 (EphA2) | Eph | TK | 6hey | A | A | 3-[(4,6-dipyridin-3-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11557 | |
| EPHA2 (EphA2) | Eph | TK | 7kjc | B | B | phosphomethylphosphonic acid adenylate ester | Human | 13254 | |
| EPHA2 (EphA2) | Eph | TK | 5ia3 | A | A | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Human | 7193 | |
| EPHA2 (EphA2) | Eph | TK | 5njz | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-(piperidin-4-ylcarbamoyl)phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8085 | |
| EPHA2 (EphA2) | Eph | TK | 8bin | A | A | 8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14514 | |
| EPHA2 (EphA2) | Eph | TK | 6fnh | A | B | 1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 10418 | |
| EPHA2 (EphA2) | Eph | TK | 5ia5 | A | B | golvatinib | Human | 7183 | |
| EPHA2 (EphA2) | Eph | TK | 8bin | A | B | 8-(4-azanylbutyl)-6-(2-chlorophenyl)-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 14515 | |
| EPHA2 (EphA2) | Eph | TK | 6hew | A | B | 4-methyl-3-[(1-methyl-6-pyrimidin-5-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11556 | |
| EPHA2 (EphA2) | Eph | TK | 5ia0 | A | A | alisertib | Human | 7169 | |
| EPHA2 (EphA2) | Eph | TK | 5nki | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3-methylsulfonyl-5-morpholin-4-yl-phenyl)amino]-1,3-thiazole-5-carboxamide | Human | 8069 | |
| EPHA2 (EphA2) | Eph | TK | 5nkb | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3,5-dimorpholin-4-ylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 8097 | |
| EPHA2 (EphA2) | Eph | TK | 5nkd | A | A | 2-[(3~{r})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidin-3-yl]ethanoic acid | Human | 8058 | |
| EPHA2 (EphA2) | Eph | TK | 5i9v | A | B | phosphothiophosphoric acid-adenylate ester | Human | 7173 | |
| EPHA2 (EphA2) | Eph | TK | 7kjc | A | B | phosphomethylphosphonic acid adenylate ester | Human | 13256 | |
| EPHA2 (EphA2) | Eph | TK | 5nkb | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[(3,5-dimorpholin-4-ylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 8098 | |
| EPHA2 (EphA2) | Eph | TK | 5nk8 | A | B | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[(2,2,6,6-tetramethyl-1-oxidanyl-piperidin-4-yl)carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8088 | |
| EPHA2 (EphA2) | Eph | TK | 5ek7 | A | | - | Human | 6322 | |
| EPHA2 (EphA2) | Eph | TK | 6q7f | A | B | 3-[(4-imidazol-1-yl-6-piperazin-1-yl-1,3,5-triazin-2-yl)amino]-4-methyl-~{n}-[3-(trifluoromethyl)phenyl]benzamide | Human | 11936 | |
| EPHA2 (EphA2) | Eph | TK | 6het | A | B | ~{n}-(3-chlorophenyl)-4-methyl-3-[(1-methyl-6-pyridin-3-yl-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 11560 | |
| EPHA2 (EphA2) | Eph | TK | 5nk5 | A | B | 2-[[3-[(3-aminophenyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8066 | |
| EPHA2 (EphA2) | Eph | TK | 5nkc | A | A | (3~{s})-1-[3-[[5-[(2-chloranyl-6-methyl-phenyl)carbamoyl]-1,3-thiazol-2-yl]amino]phenyl]carbonylpyrrolidine-3-carboxylic acid | Human | 8099 | |
| EPHA2 (EphA2) | Eph | TK | 5nk1 | A | B | 2-[[3-[(4-azanyl-6-methyl-1,3,5-triazin-2-yl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8059 | |
| EPHA2 (EphA2) | Eph | TK | 7kjc | A | A | phosphomethylphosphonic acid adenylate ester | Human | 13257 | |
| EPHA2 (EphA2) | Eph | TK | 5nk7 | A | A | ~{n}-(2-chloranyl-6-methyl-phenyl)-2-[[3-[[(3~{r},4~{r})-3-fluoranylpiperidin-4-yl]carbamoyl]phenyl]amino]-1,3-thiazole-5-carboxamide | Human | 8089 | |
| EPHA2 (EphA2) | Eph | TK | 4pdo | A | | - | Human | 2086 | |
| EPHA2 (EphA2) | Eph | TK | 5nk0 | A | A | 2-[[3-[(3-azanyl-2,2-dimethyl-propyl)carbamoyl]phenyl]amino]-~{n}-(2-chloranyl-6-methyl-phenyl)-1,3-thiazole-5-carboxamide | Human | 8095 | |
| EPHB4 (EphB4) | Eph | TK | 2vwx | A | B | 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 350 | |
| EPHB4 (EphB4) | Eph | TK | 3zew | A | B | staurosporine | Human | 377 | |
| EPHB4 (EphB4) | Eph | TK | 2vwv | A | A | n'-(3-chloro-4-methoxy-phenyl)-n-(3,4,5-trimethoxyphenyl)-1,3,5-triazine-2,4-diamine | Human | 365 | |
| EPHB4 (EphB4) | Eph | TK | 3zew | B | B | staurosporine | Human | 357 | |
| EPHB4 (EphB4) | Eph | TK | 2vx1 | A | A | 3-({4-[(5-chloro-1,3-benzodioxol-4-yl)amino]pyrimidin-2-yl}amino)benzamide | Human | 371 | |
| EPHB4 (EphB4) | Eph | TK | 2vww | A | A | n'-(5-chloro-1,3-benzodioxol-4-yl)-n-(3,4,5- trimethoxyphenyl)pyrimidine-2,4-diamine | Human | 356 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | I | | - | Human | 559 | |
| EPHB1 (EphB1) | Eph | TK | 6umw | A | B | 7-chlorotetracycline | Human | 12923 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | C | | - | Human | 557 | |
| EPHB1 (EphB1) | Eph | TK | 5mjb | B | | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | 7585 | |
| EPHB1 (EphB1) | Eph | TK | 5mja | A | | 2-chloranyl-~{n}-[4-[(2-chloranyl-5-oxidanyl-phenyl)amino]quinazolin-7-yl]ethanamide | Human | 7582 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | H | | - | Human | 556 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | B | | - | Human | 558 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | E | | - | Human | 555 | |
| EPHB1 (EphB1) | Eph | TK | 3zfx | F | | - | Human | 553 | |
| EPHA5 (EphA5) | Eph | TK | 2r2p | A | B | - | Human | 3413 | |
| EPHA5 (EphA5) | Eph | TK | 2r2p | A | A | - | Human | 3412 | |
| EPHB2 (EphB2) | Eph | TK | 3zfm | A | | - | Human | 2731 | |