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Search results (436 entries covering 174 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
FGFR4FGFRTK7ybpA~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14500
FGFR4FGFRTK6jpjAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman11051
FGFR4FGFRTK6nvhAAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11388
FGFR4FGFRTK6nviABn-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamideHuman11389
FGFR1FGFRTK7wclAB11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-oneHuman14363
FGFR4FGFRTK4tygAB-Human933
FGFR4FGFRTK4tyiA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman926
FGFR2FGFRTK2pvyCphosphomethylphosphonic acid adenylate esterHuman501
FGFR2FGFRTK8e1xA(5m)-n-methyl-5-{(6m,8s)-5-{[(3s)-oxolan-3-yl]amino}-6-[1-(propan-2-yl)-1h-pyrazol-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl}pyridine-3-carboxamideHuman14511
FGFR4FGFRTK6v9cAAn-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamideHuman12096
FGFR2FGFRTK7kieBAn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13282
FGFR2FGFRTK6agxCBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11537
FGFR2FGFRTK6agxABethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11542
FGFR2FGFRTK4j95DAphosphomethylphosphonic acid adenylate esterHuman490
FGFR2FGFRTK4j97DBphosphomethylphosphonic acid adenylate esterHuman532
FGFR2FGFRTK4j95BBphosphomethylphosphonic acid adenylate esterHuman519
FGFR2FGFRTK4j96AB-Human470
FGFR2FGFRTK6agxCAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11538
FGFR1FGFRTK6itjBB4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11772
FGFR2FGFRTK4j95ABphosphomethylphosphonic acid adenylate esterHuman477
FGFR2FGFRTK5ugxABphosphomethylphosphonic acid adenylate esterHuman7448
FGFR2FGFRTK7kiaAB1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13285
FGFR1FGFRTK5flfBA-Human6465
FGFR1FGFRTK5vndAAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7646
FGFR2FGFRTK6v6qCphosphomethylphosphonic acid adenylate esterHuman12969
FGFR2FGFRTK6lvlAn-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12132
FGFR2FGFRTK6lvlBn-ethyl-2-[[4-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12130
FGFR1FGFRTK5ew8BB~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6471
FGFR1FGFRTK5a46BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3578
FGFR1FGFRTK3c4fBB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3562
FGFR2FGFRTK4j97BAphosphomethylphosphonic acid adenylate esterHuman476
FGFR2FGFRTK6agxBAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11540
FGFR4FGFRTK5nwzA~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamideHuman9789
FGFR2FGFRTK4j95BAphosphomethylphosphonic acid adenylate esterHuman498
FGFR2FGFRTK4j95CAphosphomethylphosphonic acid adenylate esterHuman531
FGFR2FGFRTK2pwlAphosphomethylphosphonic acid adenylate esterHuman523
FGFR2FGFRTK4j98BBphosphomethylphosphonic acid adenylate esterHuman472
FGFR4FGFRTK4qqcABn-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamideHuman932
FGFR2FGFRTK8w38AB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15403
FGFR2FGFRTK6agxBBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11536
FGFR2FGFRTK4j97CAphosphomethylphosphonic acid adenylate esterHuman488
FGFR2FGFRTK6lvkBn-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12129
FGFR2FGFRTK5uglBAphosphoaminophosphonic acid-adenylate esterHuman7450
FGFR1FGFRTK4uwcAB3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6017
FGFR4FGFRTK4qqtA-Human922
FGFR4FGFRTK4qqjA-Human935
FGFR4FGFRTK6jpeAn-[2-[[6-[2-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]amino]pyridin-3-yl]pyrimidin-4-yl]amino]-3-methyl-phenyl]prop-2-enamideHuman12230
FGFR4FGFRTK5nudB3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amineHuman9790
FGFR4FGFRTK7yc3A6-bromanyl-~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14501
FGFR4FGFRTK4tygAA-Human929
FGFR4FGFRTK6yi8ABn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12811
FGFR4FGFRTK6yi8BAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12813
FGFR4FGFRTK6yi8BBn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12814
FGFR4FGFRTK6nvjAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-fluorophenyl]propanamideHuman11391
FGFR4FGFRTK5nudA3-chloranyl-~{n}-(3-nitropyridin-2-yl)-5-(trifluoromethyl)pyridin-2-amineHuman9787
FGFR4FGFRTK7vjlAn-[5-(aminomethyl)-4-(2-methoxyethylamino)pyridin-2-yl]-7-[2,2,2-tris(fluoranyl)ethanoyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman14109
FGFR4FGFRTK6nviAAn-[3-chloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-5-fluorophenyl]propanamideHuman11392
FGFR4FGFRTK4r6vAn-[4-({[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](6-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino}methyl)phenyl]propanamideHuman931
FGFR4FGFRTK6nvkAAn-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamideHuman11395
FGFR4FGFRTK4tyeA-Human927
FGFR4FGFRTK4uxqA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman930
FGFR2FGFRTK6v6qBphosphomethylphosphonic acid adenylate esterHuman12966
FGFR4FGFRTK5nwzB~{n}-[3-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-5-yl]-2-(propanoylamino)benzamideHuman9788
FGFR2FGFRTK4j99DBphosphomethylphosphonic acid adenylate esterHuman481
FGFR4FGFRTK4xcuABn-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamideHuman924
FGFR4FGFRTK7dtzAn-[2-[[5-[[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]methoxy]pyrimidin-2-yl]amino]-3-methyl-phenyl]-2-fluoranyl-prop-2-enamideHuman13506
FGFR2FGFRTK4j95AAphosphomethylphosphonic acid adenylate esterHuman529
FGFR2FGFRTK4j97BCphosphomethylphosphonic acid adenylate esterHuman510
FGFR2FGFRTK4j97CCphosphomethylphosphonic acid adenylate esterHuman483
FGFR2FGFRTK5uhnBAphosphomethylphosphonic acid adenylate esterHuman7451
FGFR2FGFRTK5ugxBBphosphomethylphosphonic acid adenylate esterHuman7445
FGFR1FGFRTK8jmzAAn-(2-(dimethylamino)ethyl)-1-(3-((4-((2-methyl-1h-indol-5-yl)oxy)pyrimidin-2-yl)amino)phenyl)methanesulfonamideHuman15228
FGFR2FGFRTK6v6qAphosphomethylphosphonic acid adenylate esterHuman12968
FGFR1FGFRTK8jmzABn-(2-(dimethylamino)ethyl)-1-(3-((4-((2-methyl-1h-indol-5-yl)oxy)pyrimidin-2-yl)amino)phenyl)methanesulfonamideHuman15227
FGFR4FGFRTK7v29An-[2-[[3-(3,5-dimethoxyphenyl)-2-oxidanylidene-1-[3-(4-propanoylpiperazin-1-yl)propyl]-4h-pyrimido[4,5-d]pyrimidin-7-yl]amino]phenyl]propanamideHuman14165
FGFR4FGFRTK6iuoAn-({4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}methyl)prop-2-enamideHuman11757
FGFR2FGFRTK2psqB-Human530
FGFR2FGFRTK2q0bBphosphomethylphosphonic acid adenylate esterHuman499
FGFR2FGFRTK2py3Bphosphomethylphosphonic acid adenylate esterHuman484
FGFR2FGFRTK4j95DBphosphomethylphosphonic acid adenylate esterHuman492
FGFR2FGFRTK6agxDAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11543
FGFR2FGFRTK2pwlBphosphomethylphosphonic acid adenylate esterHuman534
FGFR4FGFRTK4qrcA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman923
FGFR2FGFRTK5uglAAphosphoaminophosphonic acid-adenylate esterHuman7442
FGFR2FGFRTK8u1fAn-[4-(4-amino-7-methyl-5-{4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7h-pyrrolo[2,3-d]pyrimidin-6-yl)phenyl]-2-methylpropanamideHuman15202
FGFR2FGFRTK5uglBBphosphoaminophosphonic acid-adenylate esterHuman7449
FGFR1FGFRTK5uq0AB2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7458
FGFR3FGFRTK8udvA3-[(6-chloro-1-cyclopropyl-1h-benzimidazol-5-yl)ethynyl]-1-[(3s,5s)-5-(methoxymethyl)-1-(prop-2-enoyl)pyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamideHuman15203
FGFR3FGFRTK9cd7A(3p)-5-[(1r)-1-(3,5-dichloropyridin-4-yl)ethoxy]-3-{6-[6-(methanesulfonyl)-2,6-diazaspiro[3.3]heptan-2-yl]pyridin-3-yl}-1h-indazoleHuman15469
FGFR3FGFRTK12wwA(2s)-2-{[(6p,8s)-3-chloro-6-(1-{1-[(z)-iminomethyl]piperidin-4-yl}-5-methyl-1h-1,2,3-triazol-4-yl)pyrazolo[1,5-a]pyridin-4-yl]oxy}-2-(5-fluoropyridin-2-yl)ethan-1-olHuman15470
FGFR1FGFRTK43xkAB~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)thiolan-2-yl]methyl]prop-2-enamideHuman15684
FGFR1FGFRTK44acA~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methyl]-2-fluoranyl-prop-2-enamideHuman15685
FGFR1FGFRTK9wfkAB(2~{r},3~{r},4~{s},5~{r})-2-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolHuman15686
FGFR1FGFRTK9wfkAA(2~{r},3~{r},4~{s},5~{r})-2-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-5-(hydroxymethyl)oxolane-3,4-diolHuman15687
FGFR1FGFRTK43zyAA~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-[2-(3,5-dimethoxyphenyl)ethynyl]pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methyl]prop-2-enamideHuman15688
FGFR1FGFRTK9w1aAxs8148Human15679
FGFR1FGFRTK43zyAB~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-[2-(3,5-dimethoxyphenyl)ethynyl]pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methyl]prop-2-enamideHuman15680
FGFR1FGFRTK44ahAAderazantinibHuman15681
FGFR1FGFRTK44adAA2-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-3-yl]-6-(4-methylpiperazin-1-yl)-1~{h}-benzimidazoleHuman15682
FGFR1FGFRTK44aaAA(2~{r},3~{s},4~{r},5~{r})-2-[[(azanylidene-$l^{4}-azanylidene)amino]methyl]-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]oxolane-3,4-diolHuman15683
FGFR1FGFRTK43zvA~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methyl]prop-2-enamideHuman15689
FGFR1FGFRTK9wgtAA(2~{r},3~{s},4~{r},5~{r})-2-(aminomethyl)-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]oxolane-3,4-diolHuman15690
FGFR1FGFRTK9uhiA~{n}-[1-methyl-3-[3-[1-(2-morpholin-4-ylethyl)pyrazol-4-yl]quinoxalin-5-yl]indol-6-yl]propanamideHuman15691
FGFR1FGFRTK9wgtAB(2~{r},3~{s},4~{r},5~{r})-2-(aminomethyl)-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]oxolane-3,4-diolHuman15692
FGFR2FGFRTK2pvyAphosphomethylphosphonic acid adenylate esterHuman489
FGFR2FGFRTK4j99BBphosphomethylphosphonic acid adenylate esterHuman495
FGFR2FGFRTK8sweAAn-{4-[4-amino-5-(4-methoxyphenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}prop-2-enamideHuman15200
FGFR2FGFRTK5ugxAAphosphomethylphosphonic acid adenylate esterHuman7443
FGFR4FGFRTK7wcwA~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamideHuman14168
FGFR1FGFRTK2fgiB1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHuman3541
FGFR1FGFRTK3gqlB(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHuman3506
FGFR1FGFRTK5ur1BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7969
FGFR1FGFRTK1fgkBB-Human3557
FGFR1FGFRTK5am7AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3488
FGFR2FGFRTK4j97BBphosphomethylphosphonic acid adenylate esterHuman493
FGFR2FGFRTK5ui0AB-Human7447
FGFR4FGFRTK6yi8AAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-7-methanoyl-6-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3,4-dihydro-2h-1,8-naphthyridine-1-carboxamideHuman12812
FGFR4FGFRTK9k0jA~{n}-[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]-2-fluoranyl-6-(propanoylamino)benzamideHuman15404
FGFR4FGFRTK7yboA~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14499
FGFR4FGFRTK5jkgA2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanolHuman7089
FGFR4FGFRTK6nvkABn-[(3s,4s)-3-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}oxan-4-yl]propanamideHuman11390
FGFR4FGFRTK4qqcAAn-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamideHuman934
FGFR4FGFRTK6iupABn-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamideHuman11796
FGFR4FGFRTK6nvgAn-[3,5-dichloro-2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)phenyl]propanamideHuman11394
FGFR2FGFRTK6v6qDphosphomethylphosphonic acid adenylate esterHuman12967
FGFR2FGFRTK4j99AAphosphomethylphosphonic acid adenylate esterHuman474
FGFR2FGFRTK8w2xA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]propan-1-oneHuman15406
FGFR2FGFRTK5ui0BBphosphomethylphosphonic acid adenylate esterHuman7440
FGFR2FGFRTK2pz5Aphosphomethylphosphonic acid adenylate esterHuman511
FGFR2FGFRTK4j97AAphosphomethylphosphonic acid adenylate esterHuman496
FGFR2FGFRTK2pz5Bphosphomethylphosphonic acid adenylate esterHuman513
FGFR2FGFRTK4j99ACphosphomethylphosphonic acid adenylate esterHuman469
FGFR2FGFRTK4j99CBphosphomethylphosphonic acid adenylate esterHuman506
FGFR2FGFRTK5eg3Aphosphomethylphosphonic acid adenylate esterHuman6368
FGFR2FGFRTK2pvfAphosphomethylphosphonic acid adenylate esterHuman525
FGFR2FGFRTK5uhnABphosphomethylphosphonic acid adenylate esterHuman7441
FGFR2FGFRTK9u3nA~{n}-[4-[4-azanyl-7-methyl-5-[2-(3-methylimidazo[4,5-b]pyridin-6-yl)ethynyl]pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]prop-2-enamideHuman15407
FGFR2FGFRTK4j99BAphosphomethylphosphonic acid adenylate esterHuman518
FGFR2FGFRTK6lvkAn-ethyl-2-[[4-[[4-(4-methylpiperazin-1-yl)-3-(2-morpholin-4-ylethoxy)phenyl]amino]-1,3,5-triazin-2-yl]amino]benzenesulfonamideHuman12131
FGFR2FGFRTK2pzpBphosphomethylphosphonic acid adenylate esterHuman524
FGFR2FGFRTK4j98AB-Human475
FGFR2FGFRTK4j98BAphosphomethylphosphonic acid adenylate esterHuman516
FGFR2FGFRTK2pvyDphosphomethylphosphonic acid adenylate esterHuman482
FGFR2FGFRTK5uhnBBphosphomethylphosphonic acid adenylate esterHuman7444
FGFR2FGFRTK4j96BBphosphomethylphosphonic acid adenylate esterHuman486
FGFR2FGFRTK8w3bAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15408
FGFR2FGFRTK7ozyAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman13999
FGFR2FGFRTK5uglABphosphoaminophosphonic acid-adenylate esterHuman7452
FGFR2FGFRTK6agxDBethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11539
FGFR2FGFRTK2pzrAphosphomethylphosphonic acid adenylate esterHuman526
FGFR2FGFRTK8w3dAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15409
FGFR2FGFRTK4j99DAphosphomethylphosphonic acid adenylate esterHuman533
FGFR2FGFRTK1gjoA-Human478
FGFR2FGFRTK5ugxBAphosphomethylphosphonic acid adenylate esterHuman7454
FGFR2FGFRTK4j99CCphosphomethylphosphonic acid adenylate esterHuman471
FGFR2FGFRTK7kiaAA1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13283
FGFR2FGFRTK2pzpAphosphomethylphosphonic acid adenylate esterHuman497
FGFR2FGFRTK7kieBBn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13284
FGFR2FGFRTK2q0bAphosphomethylphosphonic acid adenylate esterHuman512
FGFR2FGFRTK5uhnAAphosphomethylphosphonic acid adenylate esterHuman7455
FGFR2FGFRTK4j97DAphosphomethylphosphonic acid adenylate esterHuman507
FGFR2FGFRTK8w3dAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15410
FGFR2FGFRTK4j97ACphosphomethylphosphonic acid adenylate esterHuman521
FGFR2FGFRTK3b2tA5'-o-[(s)-hydroxy{[(s)-hydroxy(methyl)phosphoryl]oxy}phosphoryl]adenosineHuman520
FGFR2FGFRTK8w38AA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15411
FGFR2FGFRTK9vlmA~{n}-[3-[2-[[3-[2-(dimethylamino)ethylsulfamoylmethyl]phenyl]amino]pyrimidin-4-yl]-1-methyl-indol-6-yl]propanamideHuman15413
FGFR2FGFRTK7kieABn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13286
FGFR2FGFRTK2pvyBphosphomethylphosphonic acid adenylate esterHuman504
FGFR2FGFRTK7kieAAn-{4-[(e)-2-{4-(4-methylpiperazin-1-yl)-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}ethenyl]phenyl}prop-2-enamideHuman13287
FGFR2FGFRTK7kiaBB1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13288
FGFR2FGFRTK6agxAAethyl [4-({3-[2-(3,5-dimethoxyphenyl)ethyl]-5h-pyrrolo[2,3-b]pyrazin-5-yl}sulfonyl)-1h-imidazol-1-yl]acetateHuman11541
FGFR2FGFRTK4j96AA-Human473
FGFR1FGFRTK5flfDA-Human6468
FGFR3FGFRTK6pnxAAphosphomethylphosphonic acid adenylate esterHuman11948
FGFR3FGFRTK6lvmA2-[[5-[2-(3,5-dimethoxyphenyl)ethyl]-2-[[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]amino]pyrimidin-4-yl]amino]-n-ethyl-benzenesulfonamideHuman12134
FGFR3FGFRTK6pnxABphosphomethylphosphonic acid adenylate esterHuman11946
FGFR2FGFRTK8h75A4-[9-(2-chlorophenyl)-6-methyl-2,4,5,8,12-pentazatricyclo[8.4.0.0^{3,7}]tetradeca-1(10),3,6,8,11,13-hexaen-13-yl]morpholineHuman14860
FGFR4FGFRTK7f3mA6-[2,6-bis(chloranyl)-3,5-dimethoxy-phenyl]-2-(methylamino)-8-[3-(4-prop-2-enoylpiperazin-1-yl)propyl]pyrido[2,3-d]pyrimidin-7-oneHuman14034
FGFR3FGFRTK7dhlA5-[2-(3,5-dimethoxyphenyl)ethyl]-n-[3-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]pyrimidin-2-amineHuman13258
FGFR4FGFRTK7wcxA~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamideHuman14166
FGFR2FGFRTK4j96BAphosphomethylphosphonic acid adenylate esterHuman485
FGFR3FGFRTK4k33ABphosphomethylphosphonic acid adenylate esterHuman1870
FGFR3FGFRTK6pnxBBphosphomethylphosphonic acid adenylate esterHuman11949
FGFR3FGFRTK4k33AAphosphomethylphosphonic acid adenylate esterHuman1871
FGFR3FGFRTK6pnxBAphosphomethylphosphonic acid adenylate esterHuman11947
FGFR3FGFRTK8uduAB3-[(6-chloro-1-cyclopropyl-1h-benzimidazol-5-yl)ethynyl]-1-[(3s,5s)-5-(methoxymethyl)-1-(prop-2-enoyl)pyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamideHuman15204
FGFR2FGFRTK3ri1B(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman528
FGFR4FGFRTK6iupAAn-{4-[4-amino-3-(3,5-dimethyl-1-benzofuran-2-yl)-7-oxo-6,7-dihydro-2h-pyrazolo[3,4-d]pyridazin-2-yl]phenyl}prop-2-enamideHuman11797
FGFR4FGFRTK4qq5An-(4-{[3-(3,5-dimethoxyphenyl)-7-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)propanamideHuman921
FGFR1FGFRTK5uq0AA2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7456
FGFR1FGFRTK4rwlB6-({7-[(1-aminocyclopropyl)methoxy]-6-methoxyquinolin-4-yl}oxy)-n-methylnaphthalene-1-carboxamideHuman3596
FGFR1FGFRTK6mzwBA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11165
FGFR1FGFRTK3rhxB(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman3522
FGFR1FGFRTK4zsaAA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3491
FGFR1FGFRTK6c1bBB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11167
FGFR1FGFRTK4rwjBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3559
FGFR1FGFRTK4v05ABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3593
FGFR1FGFRTK5z0sBB1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10814
FGFR1FGFRTK44adAB2-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1~{h}-pyrazol-3-yl]-6-(4-methylpiperazin-1-yl)-1~{h}-benzimidazoleHuman15672
FGFR1FGFRTK3tt0BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3547
FGFR1FGFRTK1agwBB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3510
FGFR1FGFRTK8jqiB-Human15678
FGFR1FGFRTK5vndBAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7647
FGFR1FGFRTK7ozdAAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHuman14007
FGFR1FGFRTK5am7AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3533
FGFR1FGFRTK6mzqBB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11171
FGFR1FGFRTK6nvlDBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11398
FGFR1FGFRTK6p69BAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11331
FGFR1FGFRTK5zv2B4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHuman10054
FGFR1FGFRTK4v04AA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3542
FGFR1FGFRTK4uwyAB-Human3582
FGFR1FGFRTK5a46BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3526
FGFR1FGFRTK4f65BA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3545
FGFR1FGFRTK1fgkBA-Human3513
FGFR1FGFRTK6c18AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11168
FGFR1FGFRTK1agwAA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3520
FGFR1FGFRTK5a4cAA1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3543
FGFR1FGFRTK4nk9Bn~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3535
FGFR1FGFRTK7ozbAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman14008
FGFR1FGFRTK5ur1BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7971
FGFR1FGFRTK4uwyBA-Human3537
FGFR1FGFRTK4f64BA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3576
FGFR1FGFRTK4rwkABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3517
FGFR1FGFRTK1fgiAA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3555
FGFR1FGFRTK3c4fAA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3515
FGFR1FGFRTK5uq0BA2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7459
FGFR1FGFRTK6c19AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11163
FGFR1FGFRTK3ky2A-Human3534
FGFR1FGFRTK5am6BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3521
FGFR1FGFRTK5o4aAA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9554
FGFR1FGFRTK4rwiBB-Human3527
FGFR1FGFRTK5flfCB-Human6466
FGFR1FGFRTK5a4cBB1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3540
FGFR1FGFRTK5o4aAB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9558
FGFR1FGFRTK6c1oAAn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11159
FGFR1FGFRTK5b7vA[5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanoneHuman6705
FGFR1FGFRTK4nkaAn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3501
FGFR1FGFRTK4zsaBB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3512
FGFR1FGFRTK6mzwAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11157
FGFR1FGFRTK6mzqAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11156
FGFR1FGFRTK6itjBA4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11775
FGFR1FGFRTK4f64AB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3589
FGFR1FGFRTK4uwcAA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6019
FGFR1FGFRTK3tt0BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3581
FGFR1FGFRTK4rwlA-Human3516
FGFR1FGFRTK3c4fAB3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3564
FGFR1FGFRTK5am6AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3494
FGFR1FGFRTK6mzwBB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman10857
FGFR1FGFRTK5am7BB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3531
FGFR1FGFRTK6itjAA4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11773
FGFR1FGFRTK6c19AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10859
FGFR1FGFRTK5flfCA-Human6469
FGFR1FGFRTK6nvlBAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11403
FGFR1FGFRTK7ozbAA4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman14010
FGFR1FGFRTK5ur1AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7970
FGFR1FGFRTK6c1bAA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11169
FGFR1FGFRTK3gqiAphosphomethylphosphonic acid adenylate esterHuman3566
FGFR1FGFRTK4v05BAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3518
FGFR1FGFRTK7ozfAAn-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamideHuman14011
FGFR1FGFRTK4rwiAB-Human3551
FGFR1FGFRTK6nvlABn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11401
FGFR1FGFRTK3gqlA(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHuman3509
FGFR1FGFRTK6c19BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10855
FGFR1FGFRTK6c1bAB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10861
FGFR1FGFRTK6p69ABn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11330
FGFR4FGFRTK8kh9A1-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-3-[6-methanoyl-5-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3-(2-morpholin-4-ylethoxy)pyridin-2-yl]ureaHuman15284
FGFR4FGFRTK8kh7A1-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-3-[6-methanoyl-5-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3-(2-morpholin-4-ylethoxy)pyridin-2-yl]ureaHuman15286
FGFR4FGFRTK8kh6A1-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-3-[5-bromanyl-6-(hydroxymethyl)-3-methoxy-pyridin-2-yl]ureaHuman15287
FGFR4FGFRTK8w5cAn-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-6-[(4-methylpiperazin-1-yl)methyl]-1-propan-2-yl-pyrrolo[3,2-b]pyridine-3-carboxamideHuman15288
FGFR4FGFRTK4tyjA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman925
FGFR4FGFRTK5xfjA2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanolHuman10376
FGFR4FGFRTK6nvhABn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11393
FGFR2FGFRTK3ri1A(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman503
FGFR2FGFRTK8stgAn-{4-[(5p)-4-amino-5-{3-fluoro-4-[(4-methylpyrimidin-2-yl)oxy]phenyl}-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}-2-methylprop-2-enamideHuman14762
FGFR2FGFRTK4j98AA-Human500
FGFR1FGFRTK4v01AB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3590
FGFR4FGFRTK7yc1A~{n}-[5-cyano-4-(2-methoxyethylamino)pyridin-2-yl]-5-methanoyl-1-propyl-pyrrolo[3,2-b]pyridine-3-carboxamideHuman14498
FGFR4FGFRTK7ybxA~{n}-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-6-bromanyl-5-(hydroxymethyl)-1-(2-morpholin-4-ylethyl)pyrrolo[3,2-b]pyridine-3-carboxamideHuman14502
FGFR4FGFRTK6v9cABn-[(3r,4s)-4-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)-8-methyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}oxolan-3-yl]prop-2-enamideHuman12095
FGFR4FGFRTK9k0iA(2~{s})-~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]-2-cyano-3-cyclopropyl-propanamideHuman15405
FGFR4FGFRTK4xcuAAn-(2-{[6-(2,6-dichloro-3,5-dimethoxyphenyl)quinazolin-2-yl]amino}-3-methylphenyl)prop-2-enamideHuman928
FGFR4FGFRTK7wctA~{n}-[2-[[5-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1~{h}-indazol-3-yl]amino]-3-fluoranyl-5-(4-morpholin-4-ylpiperidin-1-yl)phenyl]propanamideHuman14167
FGFR4FGFRTK5xffA2-[4-[e-2-[5-[(1r)-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-1h-indazol-3-yl]ethenyl]pyrazol-1-yl]ethanolHuman10375
FGFR2FGFRTK7kiaBA1-[4-(4-{4-(4-methylpiperazin-1-yl)-6-[(3-methyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}phenyl)piperidin-1-yl]prop-2-en-1-oneHuman13281
FGFR2FGFRTK1oecA4-aryl-2-phenylamino pyrimidineHuman479
FGFR2FGFRTK4j95CBphosphomethylphosphonic acid adenylate esterHuman502
FGFR2FGFRTK2py3Aphosphomethylphosphonic acid adenylate esterHuman509
FGFR2FGFRTK3clyAphosphomethylphosphonic acid adenylate esterHuman522
FGFR2FGFRTK7ozyAB4-[3-(4-piperazin-4-ium-1-ylphenyl)-1h-indazol-6-yl]phenolHuman13998
FGFR2FGFRTK4j99CAphosphomethylphosphonic acid adenylate esterHuman505
FGFR2FGFRTK4j99DCphosphomethylphosphonic acid adenylate esterHuman480
FGFR2FGFRTK4j99BCphosphomethylphosphonic acid adenylate esterHuman491
FGFR2FGFRTK2psqA-Human515
FGFR2FGFRTK2pzrBphosphomethylphosphonic acid adenylate esterHuman508
FGFR2FGFRTK5ui0AA-Human7446
FGFR2FGFRTK4j97ABphosphomethylphosphonic acid adenylate esterHuman527
FGFR2FGFRTK8sweABn-{4-[4-amino-5-(4-methoxyphenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl}prop-2-enamideHuman15201
FGFR2FGFRTK4j99ABphosphomethylphosphonic acid adenylate esterHuman494
FGFR2FGFRTK5ui0BAphosphomethylphosphonic acid adenylate esterHuman7453
FGFR2FGFRTK3b2tB5'-o-[(s)-hydroxy{[(s)-hydroxy(methyl)phosphoryl]oxy}phosphoryl]adenosineHuman517
FGFR2FGFRTK8w3bAB1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman15412
FGFR2FGFRTK4j97CBphosphomethylphosphonic acid adenylate esterHuman487
FGFR2FGFRTK4j97DCphosphomethylphosphonic acid adenylate esterHuman514
FGFR2FGFRTK10ooA(4p)-n-[4-(4-aminopiperidin-1-yl)-2-methoxyphenyl]-5-chloro-4-(1h-indol-3-yl)pyrimidin-2-amineHuman15414
FGFR3FGFRTK8uduAA3-[(6-chloro-1-cyclopropyl-1h-benzimidazol-5-yl)ethynyl]-1-[(3s,5s)-5-(methoxymethyl)-1-(prop-2-enoyl)pyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamideHuman15205
FGFR3FGFRTK8udtA3-[(1-cyclopropyl-4,6-difluoro-1h-benzimidazol-5-yl)ethynyl]-1-[(3r,5r)-5-(methoxymethyl)-1-propanoylpyrrolidin-3-yl]-5-(methylamino)-1h-pyrazole-4-carboxamideHuman15206
FGFR1FGFRTK6nvlCAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11404
FGFR1FGFRTK4wunABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3595
FGFR1FGFRTK4nksBAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3492
FGFR1FGFRTK3kxxD-Human3503
FGFR1FGFRTK44aaAB(2~{r},3~{s},4~{r},5~{r})-2-[[(azanylidene-$l^{4}-azanylidene)amino]methyl]-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]oxolane-3,4-diolHuman15671
FGFR1FGFRTK5o4aBB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9555
FGFR1FGFRTK5z0sBA1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10812
FGFR1FGFRTK6nvlAAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11400
FGFR1FGFRTK5b7vB[5-amino-1-(2-methyl-1h-benzimidazol-6-yl)-1h-pyrazol-4-yl](1h-indol-2-yl)methanoneHuman6704
FGFR1FGFRTK7ozfABn-[6-(3-ethoxyphenyl)-1h-indazol-3-yl]benzamideHuman14006
FGFR1FGFRTK4v05BBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3493
FGFR1FGFRTK4v01AA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3556
FGFR1FGFRTK5am7BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3588
FGFR1FGFRTK5flfBB-Human6467
FGFR1FGFRTK6p68An-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHuman11336
FGFR1FGFRTK5flfEA-Human6473
FGFR1FGFRTK4rwkAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3500
FGFR1FGFRTK5am6BA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3587
FGFR1FGFRTK6mzqAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman10860
FGFR1FGFRTK3js2B5-(2-thienyl)nicotinic acidHuman3504
FGFR1FGFRTK5o49BB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9557
FGFR1FGFRTK6p68Cn-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHuman11332
FGFR1FGFRTK4rwkBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3591
FGFR1FGFRTK5ew8BA~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6474
FGFR1FGFRTK5am6AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3514
FGFR1FGFRTK5o49AA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9560
FGFR1FGFRTK4f65AA5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3558
FGFR1FGFRTK4nk9An~4~-{5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3550
FGFR1FGFRTK5flfAA-Human6462
FGFR1FGFRTK9vljA~{n}-[3-[2-[[3-[2-(dimethylamino)ethylsulfamoylmethyl]phenyl]amino]pyrimidin-4-yl]-1-methyl-indol-6-yl]propanamideHuman15673
FGFR1FGFRTK3kxxB-Human3575
FGFR1FGFRTK5o4aBA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 4-ethyl-3-fluorosulfonyl-benzoateHuman9559
FGFR1FGFRTK4uwbABn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6023
FGFR1FGFRTK43xkAA~{n}-[[(2~{r},3~{s},4~{r},5~{r})-5-[4-azanyl-5-(7-methoxy-5-methyl-1-benzothiophen-2-yl)pyrrolo[2,3-d]pyrimidin-7-yl]-3,4-bis(oxidanyl)thiolan-2-yl]methyl]prop-2-enamideHuman15674
FGFR1FGFRTK1fgkAA-Human3592
FGFR1FGFRTK6nvlBBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11399
FGFR1FGFRTK6mzqBA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11161
FGFR1FGFRTK6c19BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(methylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10862
FGFR1FGFRTK9u7gA(e)-4-methyl-17-(1-methyl-1h-pyrazol-4-yl)-7,10-dioxa-4-aza-1(3,6)-imidazo[1,2-b]pyridazina-2(3,5)-pyridinacyclodecaphan-3-oneHuman15675
FGFR1FGFRTK5a4cAB1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3498
FGFR1FGFRTK6c1oBAn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11160
FGFR1FGFRTK1fgiBA3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3586
FGFR1FGFRTK6c1cBB7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11158
FGFR1FGFRTK6c18BA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10854
FGFR1FGFRTK9uhcA~{n}-[1-methyl-3-[2-[1-(2-morpholin-4-ylethyl)pyrazol-4-yl]-5~{h}-pyrrolo[2,3-b]pyrazin-7-yl]indol-6-yl]propanamideHuman15676
FGFR1FGFRTK44ahABderazantinibHuman15677
FGFR1FGFRTK6c1cAA7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11164
FGFR1FGFRTK5ew8AA~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6470
FGFR1FGFRTK4f64BB5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3553
FGFR1FGFRTK5zv2A4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamideHuman10055
FGFR1FGFRTK5o49AB[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9556
FGFR1FGFRTK4f63B5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHuman3574
FGFR1FGFRTK3tt0AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3567
FGFR1FGFRTK5o49BA[(2~{r},3~{s},4~{r},5~{r})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl 3-fluorosulfonylbenzoateHuman9561
FGFR1FGFRTK4wunBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3529
FGFR1FGFRTK1fgiAB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3552
FGFR1FGFRTK4f64AA5-bromo-n~4~-[3-(3-methoxypropyl)-1h-pyrazol-5-yl]-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3548
FGFR1FGFRTK6c1oBBn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11154
FGFR1FGFRTK5vndBBn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7645
FGFR1FGFRTK4uwbBAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6018
FGFR1FGFRTK4f63A5-bromo-n~4~-(3-methyl-1h-pyrazol-5-yl)-n~2~-[2-(pyridin-3-yl)ethyl]pyrimidine-2,4-diamineHuman3563
FGFR1FGFRTK3js2A5-(2-thienyl)nicotinic acidHuman3523
FGFR1FGFRTK1agwAB3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3528
FGFR1FGFRTK6mzwAA1-[(3s)-3-{4-amino-3-[(3,5-dimethoxyphenyl)ethynyl]-1h-pyrazolo[3,4-d]pyrimidin-1-yl}pyrrolidin-1-yl]prop-2-en-1-oneHuman11162
FGFR1FGFRTK1fgkAB-Human3546
FGFR1FGFRTK4v04AB-Human3571
FGFR1FGFRTK4uwyAA-Human3489
FGFR1FGFRTK6nvlCBn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11405
FGFR1FGFRTK3ky2B-Human3525
FGFR1FGFRTK6p68Bn-{3-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-1-(2-hydroxyethyl)-1h-pyrazol-4-yl}prop-2-enamideHuman11334
FGFR1FGFRTK4rwjABn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3519
FGFR1FGFRTK5flfEB-Human6472
FGFR1FGFRTK3c4fBA3-(3-methoxybenzyl)-1h-pyrrolo[2,3-b]pyridineHuman3573
FGFR1FGFRTK4rwjAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3584
FGFR1FGFRTK6c1bBA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10856
FGFR1FGFRTK4rwkBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3530
FGFR1FGFRTK4zsaAB4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3487
FGFR1FGFRTK4v01BA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3497
FGFR1FGFRTK4uwbBBn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6022
FGFR1FGFRTK3tt0AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-(6-{[4-(4-ethylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)-1-methylureaHuman3538
FGFR1FGFRTK4nksAAn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3570
FGFR1FGFRTK4nksBBn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3577
FGFR1FGFRTK4uwcBA3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6021
FGFR1FGFRTK4rwjBAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3579
FGFR1FGFRTK4zsaBA4-(4-ethylpiperazin-1-yl)-n-[6-(3-methoxyphenyl)-2h-indazol-3-yl]benzamideHuman3572
FGFR1FGFRTK3kxxA-Human3495
FGFR1FGFRTK4v04BB-Human3496
FGFR1FGFRTK1agwBA3-[4-(1-formylpiperazin-4-yl)-benzylidenyl]-2-indolinoneHuman3568
FGFR1FGFRTK4nksABn~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[5-(2-phenylethyl)-1h-pyrazol-3-yl]pyrimidine-2,4-diamineHuman3561
FGFR1FGFRTK5a4cBA1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]ureaHuman3585
FGFR1FGFRTK5vndABn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl](methyl)amino}pyrimidin-4-yl)amino]-5-(4-ethylpiperazin-1-yl)phenyl}propanamideHuman7648
FGFR1FGFRTK5z0sAA1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10813
FGFR1FGFRTK6c18BB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11170
FGFR1FGFRTK5flfAB-Human6464
FGFR1FGFRTK5z0sAB1-[(6-chloroimidazo[1,2-b]pyridazin-3-yl)sulfonyl]-6-(1-methyl-1h-pyrazol-4-yl)-1h-pyrazolo[4,3-b]pyridineHuman10815
FGFR1FGFRTK4nkaBn~4~-{3-[2-(3,4-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamineHuman3539
FGFR1FGFRTK4uwbAAn-[4-(4-methylpiperazin-1-yl)phenyl]-1h-indazole-3-carboxamideHuman6020
FGFR1FGFRTK5a46AA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3532
FGFR1FGFRTK6c1oABn-(3-{[3-(2,6-dichloro-3,5-dimethoxyphenyl)-7-{[4-(diethylamino)butyl]amino}-2-oxo-3,4-dihydropyrimido[4,5-d]pyrimidin-1(2h)-yl]methyl}phenyl)prop-2-enamideHuman11166
FGFR1FGFRTK3kxxC-Human3549
FGFR1FGFRTK2fgiA1-tert-butyl-3-[6-(3,5-dimethoxy-phenyl)-2-(4-diethylamino-butylamino)-pyrido[2,3-d]pyrimidin-7-yl]-ureaHuman3490
FGFR1FGFRTK7ozdABn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]benzamideHuman14009
FGFR1FGFRTK3gqlC(e)-[4-(3,5-difluorophenyl)-3h-pyrrolo[2,3-b]pyridin-3-ylidene](3-methoxyphenyl)methanolHuman3536
FGFR1FGFRTK5ur1AB3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{1-[4-(dimethylamino)but-2-enoyl]piperidin-4-yl}-7-(phenylamino)-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman7972
FGFR1FGFRTK1fgiBB3-[(3-(2-carboxyethyl)-4-methylpyrrol-2-yl)methylene]-2-indolinoneHuman3580
FGFR1FGFRTK4rwiAA-Human3499
FGFR1FGFRTK6c1cBA7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10858
FGFR1FGFRTK6p69AAn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11333
FGFR1FGFRTK6p69BBn-{2-[(6-{[(2,6-dichloro-3,5-dimethoxyphenyl)carbamoyl][3-(4-methylpiperazin-1-yl)propyl]amino}pyrimidin-4-yl)amino]phenyl}prop-2-enamideHuman11335
FGFR1FGFRTK4v04BA3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3524
FGFR1FGFRTK4v05AAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3560
FGFR1FGFRTK4uwyBB-Human3583
FGFR1FGFRTK5uq0BB2,2-dimethyl-2,3-dihydro-1-benzofuran-7-carboxamideHuman7457
FGFR1FGFRTK4uwcBB3,4-dimethoxy-n-(5-phenyl-1h-pyrazol-3-yl)benzamideHuman6016
FGFR1FGFRTK6c18AA3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-7-[(propan-2-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman11155
FGFR1FGFRTK4v01BB3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamideHuman3594
FGFR1FGFRTK4f65BB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3502
FGFR1FGFRTK7wclAA11-[2,6-bis(fluoranyl)-3,5-dimethoxy-phenyl]-13-ethyl-4-(morpholin-4-ylmethyl)-5,7,11,13-tetrazatricyclo[7.4.0.0^{2,6}]trideca-1(9),2(6),3,7-tetraen-12-oneHuman14364
FGFR1FGFRTK5a46AB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman3505
FGFR1FGFRTK6c1cAB7-(cyclohexylamino)-3-(2,6-dichloro-3,5-dimethoxyphenyl)-1-{(3s)-1-[(2e)-4-(dimethylamino)but-2-enoyl]pyrrolidin-3-yl}-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman10853
FGFR1FGFRTK4wunAAn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3511
FGFR4FGFRTK8kh8A1-[4-[(1~{r})-1-[3,5-bis(chloranyl)pyridin-4-yl]ethoxy]-5-cyano-pyridin-2-yl]-3-[6-methanoyl-5-[(4-methyl-2-oxidanylidene-piperazin-1-yl)methyl]-3-(2-morpholin-4-ylethoxy)pyridin-2-yl]ureaHuman15285
FGFR1FGFRTK6itjAB4-azanyl-3-(3,5-dimethyl-1-benzofuran-2-yl)-2-phenyl-6~{h}-pyrazolo[3,4-d]pyridazin-7-oneHuman11774
FGFR1FGFRTK6nvlDAn-[2-({5-[(2,6-dichloro-3,5-dimethoxyphenyl)methoxy]pyrimidin-2-yl}amino)-3-methylphenyl]propanamideHuman11402
FGFR1FGFRTK3rhxA(6s)-6-phenyl-5,6-dihydrobenzo[h]quinazolin-2-amineHuman3554
FGFR1FGFRTK5ew8AB~{n}'-(3,5-dimethoxyphenyl)-~{n}'-[3-(1-methylpyrazol-4-yl)quinoxalin-6-yl]-~{n}-propan-2-yl-ethane-1,2-diamineHuman6461
FGFR1FGFRTK4rwiBA-Human3569
FGFR1FGFRTK5flfDB-Human6463
FGFR1FGFRTK4f65AB5-bromo-n~2~-[(3-methyl-1,2-oxazol-5-yl)methyl]-n~4~-[3-(2-phenylethyl)-1h-pyrazol-5-yl]pyrimidine-2,4-diamineHuman3508
FGFR1FGFRTK4wunBBn-{3-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-5-yl}-4-[(3r,5s)-3,5-dimethylpiperazin-1-yl]benzamideHuman3565
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