Search results (61 entries covering 28 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
IKBKB (IKKb)IKKOther4e3cE-Human289
TBK1IKKOther4im0ABn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman607
TBK1IKKOther4euuAAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman615
TBK1IKKOther4eutABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman621
TBK1IKKOther6cq5A2-amino-7-(1,1-dioxo-1lambda~6~-thian-4-yl)-5-oxo-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acidHuman10758
TBK1IKKOther4iwqAn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman605
TBK1IKKOther6cq0A2-amino-7-[3-(dimethylamino)propyl]-5-oxo-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acidHuman10756
TBK1IKKOther4eutAAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman609
TBK1IKKOther4euuBAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman606
CHUK (IKKa)IKKOther5ebzD2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7144
CHUK (IKKa)IKKOther5ebzK2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7150
CHUK (IKKa)IKKOther5tqwB-Human7248
CHUK (IKKa)IKKOther5ebzG2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7154
CHUK (IKKa)IKKOther5tqxB-Human7262
CHUK (IKKa)IKKOther5ebzI2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7152
CHUK (IKKa)IKKOther5ebzC2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7146
CHUK (IKKa)IKKOther5tqyA-Human7196
CHUK (IKKa)IKKOther5ebzE2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7151
TBK1IKKOther4im3ABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman622
TBK1IKKOther4eutBBn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman617
TBK1IKKOther4im0AAn-{3-[(5-cyclopropyl-2-{[3-(morpholin-4-ylmethyl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman610
IKBKB (IKKb)IKKOther8omvA-Human15271
TBK1IKKOther4im3AAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman619
TBK1IKKOther6boeA2-amino-5-oxo-7-(propan-2-yl)-n-(1h-tetrazol-5-yl)-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxamideHuman10371
CHUK (IKKa)IKKOther5tqxA-Human7261
CHUK (IKKa)IKKOther5tqwA-Human7249
CHUK (IKKa)IKKOther5ebzL2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7147
CHUK (IKKa)IKKOther5ebzA2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7153
CHUK (IKKa)IKKOther5ebzB2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7145
CHUK (IKKa)IKKOther5ebzF2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7149
TBK1IKKOther4iw0An-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman608
TBK1IKKOther5w5vA2-amino-7-(1-methylethyl)-5-oxo-5h-chromeno[2,3-b]pyridine-3-carboxylic acidHuman10024
TBK1IKKOther6cq4A2-amino-7-(4,4-difluorocyclohexyl)-5-oxo-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylic acidHuman10757
TBK1IKKOther6o8bBn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman11054
TBK1IKKOther6bnyA2-amino-7-(propan-2-yl)-3-(1h-tetrazol-5-yl)-5h-[1]benzopyrano[2,3-b]pyridin-5-oneHuman10369
TBK1IKKOther6nt9A-Human10940
TBK1IKKOther4iwoAn-{3-[(5-cyclopropyl-2-{[3-(2-oxopyrrolidin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]propyl}cyclobutanecarboxamideHuman614
IKBKB (IKKb)IKKOther4kikBBk-252aHuman293
IKBKB (IKKb)IKKOther4e3cB-Human294
IKBKB (IKKb)IKKOther4kikABk-252aHuman288
TBK1IKKOther6rstA1-[4-[(1~{r})-1-[2-[[5-[1-(cyclopropylmethyl)pyrazol-4-yl]-1~{h}-benzimidazol-2-yl]amino]pyridin-4-yl]ethyl]piperazin-1-yl]-3,3,3-tris(fluoranyl)propan-1-oneHuman11902
TBK1IKKOther4eutBAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman618
TBK1IKKOther4iwpAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman612
TBK1IKKOther6o8bAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman11053
TBK1IKKOther6bodAethyl 2-amino-5-oxo-7-(propan-2-yl)-5h-[1]benzopyrano[2,3-b]pyridine-3-carboxylateHuman10370
CHUK (IKKa)IKKOther5ebzJ2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7148
CHUK (IKKa)IKKOther5ebzH2-azanyl-5-phenyl-3-(4-sulfamoylphenyl)benzamideHuman7155
CHUK (IKKa)IKKOther5tqyB-Human7197
TBK1IKKOther4euuABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman611
TBK1IKKOther6nt9B-Human10941
TBK1IKKOther4im2AAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman620
TBK1IKKOther4euuBBn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman616
TBK1IKKOther6rsuA3,3,3-tris(fluoranyl)-1-[4-[(1~{r})-1-[2-[[(2~{s})-5-(5-propan-2-yloxypyrimidin-4-yl)-2,3-dihydro-1~{h}-benzimidazol-2-yl]amino]pyridin-4-yl]ethyl]piperazin-1-yl]propan-1-oneHuman12126
TBK1IKKOther4im2ABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideHuman613
TBK1IKKOther6rsrA~{n}-(cyclopropen-1-ylmethyl)-2-[[4-[[4-[3,3,3-tris(fluoranyl)propanoyl]piperazin-1-yl]methyl]pyridin-2-yl]amino]-1~{h}-benzimidazole-5-carboxamideHuman11903
IKBKB (IKKb)IKKOther4e3cA-Human297
IKBKB (IKKb)IKKOther4e3cC-Human296
IKBKB (IKKb)IKKOther4e3cF-Human292
IKBKB (IKKb)IKKOther4kikAAk-252aHuman290
IKBKB (IKKb)IKKOther4kikBAk-252aHuman295
IKBKB (IKKb)IKKOther4e3cD-Human291