Search results (7 entries covering 4 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
| Jak2 (JAK2) | JakA | TK | 4gl9 | D | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6935 | |||
| Jak2 (JAK2) | JakA | TK | 4gl9 | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6936 | |||
| Jak2 (JAK2) | JakA | TK | 4gl9 | C | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6934 | |||
| Jak2 (JAK2) | JakA | TK | 4gl9 | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6933 | |||
| Tyk2 (TYK2) | JakA | TK | 4e1z | A | n-[5-(4-{[(3-chlorophenyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]furan-2-carboxamide | Mouse | 5828 | |||
| Tyk2 (TYK2) | JakA | TK | 4e20 | A | n-[4-(3-amino-1h-indazol-5-yl)phenyl]-3-chlorobenzenesulfonamide | Mouse | 5827 | |||
| Jak1 (JAK1) | JakA | TK | 8ewy | A | - | Mouse | 14664 |