Search results (7 entries covering 4 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
Jak2 (JAK2)JakATK4gl9D2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouse6935
Jak2 (JAK2)JakATK4gl9B2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouse6936
Jak2 (JAK2)JakATK4gl9C2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouse6934
Jak2 (JAK2)JakATK4gl9A2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneMouse6933
Tyk2 (TYK2)JakATK4e1zAn-[5-(4-{[(3-chlorophenyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]furan-2-carboxamideMouse5828
Tyk2 (TYK2)JakATK4e20An-[4-(3-amino-1h-indazol-5-yl)phenyl]-3-chlorobenzenesulfonamideMouse5827
Jak1 (JAK1)JakATK8ewyA-Mouse14664