Search results (29 entries covering 14 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
LIMK1LISKTKL8aauLB~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamideHuman14554
LIMK1LISKTKL8aauLA~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamideHuman14555
LIMK2LISKTKL5nxdAB4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamideHuman7621
LIMK2LISKTKL5nxdBB4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamideHuman7622
LIMK1LISKTKL7b8wA2-(2-methylpropanoylamino)-~{n}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamideHuman14126
LIMK1LISKTKL9z6eAB-Human16002
LIMK1LISKTKL9z6eAA-Human16003
LIMK1LISKTKL3s95BAstaurosporineHuman1245
LIMK2LISKTKL5nxdBA4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamideHuman7624
LIMK2LISKTKL8wswAB~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamideHuman14861
LIMK2LISKTKL5nxdAA4-[(3-chlorophenyl)sulfamoyl]-~{n}-(phenylmethyl)-~{n}-propyl-benzamideHuman7623
LIMK2LISKTKL8wswAA~{n}-[5-[2-[2,6-bis(chloranyl)phenyl]-5-[bis(fluoranyl)methyl]pyrazol-3-yl]-1,3-thiazol-2-yl]-2-methyl-propanamideHuman14862
LIMK2LISKTKL7qhgAB2-(2-methylpropanoylamino)-~{n}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamideHuman14020
LIMK2LISKTKL4tptBn-{4-[(1s)-1,2-dihydroxyethyl]benzyl}-n-methyl-4-(phenylsulfamoyl)benzamideHuman2475
LIMK2LISKTKL7qhgAA2-(2-methylpropanoylamino)-~{n}-[2-[(phenylmethyl)-[4-(phenylsulfamoyl)phenyl]carbonyl-amino]ethyl]-1,3-thiazole-5-carboxamideHuman14021
LIMK2LISKTKL4tptAn-{4-[(1s)-1,2-dihydroxyethyl]benzyl}-n-methyl-4-(phenylsulfamoyl)benzamideHuman2476
LIMK1LISKTKL5nxcL(2~{r})-2-azanyl-2-cyclohexyl-~{n}-[2-(1-methylpyrazol-4-yl)-9-oxidanylidene-3,10,11-triazatricyclo[6.4.1.0^{4,13}]trideca-1,4,6,8(13),11-pentaen-6-yl]ethanamideHuman7592
LIMK1LISKTKL3s95AAstaurosporineHuman1246
LIMK1LISKTKL3s95ABstaurosporineHuman1248
LIMK1LISKTKL5hvjAAphosphoaminophosphonic acid-adenylate esterHuman6599
LIMK1LISKTKL5l6wLphosphothiophosphoric acid-adenylate esterHuman6668
LIMK1LISKTKL5hvkCphosphoaminophosphonic acid-adenylate esterHuman6596
LIMK1LISKTKL5hvjBB-Human6595
LIMK1LISKTKL7atsAn-[3-[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridine-3-carbonyl]-2,4-difluorophenyl]benzenesulfonamideHuman13164
LIMK1LISKTKL5hvjABphosphoaminophosphonic acid-adenylate esterHuman6598
LIMK1LISKTKL3s95BBstaurosporineHuman1247
LIMK1LISKTKL5hvkAphosphoaminophosphonic acid-adenylate esterHuman6600
LIMK1LISKTKL5hvjBA-Human6597
LIMK1LISKTKL7atuA(s)-2-benzyl-6-(8-chloro-5-methyl-4-oxo-2,3,4,5-tetrahydrobenzo[b][1,4]oxazepin-3-yl)-7-oxo-4,5,6,7-tetrahydro-2h-pyrazolo[3,4-c]pyridine-3-carboxamideHuman14019