| MAP3K7 (TAK1) | MLK | TKL | 5gjf | A | | n-(2-isopropoxy-4-(4-methylpiperazine-1-carbonyl)phenyl)-2-(3-(3-phenylureido)phenyl)thiazole-4-carboxamide | Human | 7264 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | B | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6063 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | D | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6072 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | A | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9798 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | C | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6070 | |
| MAP3K7 (TAK1) | MLK | TKL | 5gjg | A | | n-(2-isopropoxy-4-(4-methylpiperazine-1-carbonyl)phenyl)-2-(3-(phenylcarbamoyl)phenyl)thiazole-4-carboxamide | Human | 7265 | |
| MAP3K12 (DLK) | MLK | TKL | 8deg | A | | methyl (1s,4s)-5-{(4p)-4-[5-amino-6-(difluoromethoxy)pyrazin-2-yl]-6-[(1r,4r)-2-azabicyclo[2.1.1]hexan-2-yl]pyridin-2-yl}-2,5-diazabicyclo[2.2.1]heptane-2-carboxylate | Human | 14557 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | C | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6067 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | A | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9791 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | A | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6068 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | B | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9794 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | D | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9801 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | C | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6069 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | C | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6073 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | A | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6059 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | C | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9799 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | C | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9793 | |
| TNNI3K (HH498) | MLK | TKL | 7mgk | A | B | n-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | 13970 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | D | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6066 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | A | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6071 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | D | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6074 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | B | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9797 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | B | A | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6065 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | C | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9796 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | D | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6064 | |
| TNNI3K (HH498) | MLK | TKL | 7mgk | A | A | n-(3,5-dichloro-4-{[6-(methylamino)pyrimidin-4-yl]oxy}phenyl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | 13968 | |
| MAP3K9 (MLK1) | MLK | TKL | 3dtc | A | | 12-(2-hydroxyethyl)-2-(1-methylethoxy)-13,14-dihydronaphtho[2,1-a]pyrrolo[3,4-c]carbazol-5(12h)-one | Human | 3839 | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | A | B | - | Human | 6128 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | B | B | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6060 | |
| TNNI3K (HH498) | MLK | TKL | 7mgj | A | | n-methyl-4-[4-({[3-(trifluoromethyl)phenyl]carbamoyl}amino)phenoxy]pyridine-2-carboxamide | Human | 13969 | |
| ILK | MLK | TKL | 9d5e | A | | gefitinib | Human | 15992 | |
| ILK | MLK | TKL | 9d5h | A | | gefitinib | Human | 15989 | |
| ILK | MLK | TKL | 9d5f | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 15990 | |
| ILK | MLK | TKL | 9d5i | A | | adenosine-5'-triphosphate | Human | 15991 | |
| ILK | MLK | TKL | 9d5p | A | | [6,7-bis(2-methoxy-ethoxy)quinazoline-4-yl]-(3-ethynylphenyl)amine | Human | 15993 | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | B | A | - | Human | 6129 | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | B | B | - | Human | 6130 | |
| MAP3K9 (MLK1) | MLK | TKL | 4uy9 | A | A | - | Human | 6127 | |
| MAP3K7 (TAK1) | MLK | TKL | 5v5n | A | A | n~1~-(1-propyl-1,3-dihydro-2h-benzimidazol-2-ylidene)benzene-1,3-dicarboxamide | Human | 8350 | |
| MAP3K7 (TAK1) | MLK | TKL | 7nti | A | B | ~{n}-[[2-[bis(fluoranyl)methoxy]phenyl]methyl]-~{n}-[2-(methylamino)-2-oxidanylidene-ethyl]-2-pyrrolidin-1-ylcarbonyl-1~{h}-imidazole-4-carboxamide | Human | 13457 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l53 | A | B | trans-4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}cyclohexanol | Human | 1892 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l3p | A | | 2-(1-benzothiophen-7-yl)-4-[1-(piperidin-4-yl)-1h-pyrazol-4-yl]furo[2,3-c]pyridin-7-amine | Human | 1891 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jgb | A | | n-(2-methoxy-4-{[3-(4-methylpiperazin-1-yl)propyl]carbamoyl}phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamide | Human | 6885 | |
| MAP3K7 (TAK1) | MLK | TKL | 4gs6 | A | B | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 1886 | |
| MAP3K7 (TAK1) | MLK | TKL | 5gjd | A | | 1-(4-((1h-pyrrolo[2,3-b]pyridin-4-yl)oxy)phenyl)-3-(5-(4-methylpiperazin-1-yl)naphthalen-2-yl)urea | Human | 7263 | |
| MAP3K7 (TAK1) | MLK | TKL | 5v5n | A | B | n~1~-(1-propyl-1,3-dihydro-2h-benzimidazol-2-ylidene)benzene-1,3-dicarboxamide | Human | 8351 | |
| ILK | MLK | TKL | 3kmu | A | | - | Human | 4606 | |
| ILK | MLK | TKL | 3rep | A | | adenosine-5'-triphosphate | Human | 4604 | |
| MAP3K12 (DLK) | MLK | TKL | 8out | A | B | (1r)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-fluoranyl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2,2,2-tris(fluoranyl)ethanol | Human | 14855 | |
| MAP3K12 (DLK) | MLK | TKL | 8our | A | A | 5-[1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)-2-propan-2-yl-imidazol-4-yl]-3-(trifluoromethyloxy)pyridin-2-amine | Human | 14856 | |
| MAP3K7 (TAK1) | MLK | TKL | 5j7s | A | | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 7429 | |
| MAP3K7 (TAK1) | MLK | TKL | 2eva | A | B | adenosine | Human | 1882 | |
| MAP3K7 (TAK1) | MLK | TKL | 5e7r | A | | 2-chloro-n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}acetamide | Human | 7412 | |
| MAP3K12 (DLK) | MLK | TKL | 8our | A | B | 5-[1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)-2-propan-2-yl-imidazol-4-yl]-3-(trifluoromethyloxy)pyridin-2-amine | Human | 14852 | |
| MAP3K12 (DLK) | MLK | TKL | 8out | A | A | (1r)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-fluoranyl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2,2,2-tris(fluoranyl)ethanol | Human | 14853 | |
| MAP3K12 (DLK) | MLK | TKL | 8ous | A | B | (1s)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2-methyl-propan-1-ol | Human | 14854 | |
| MAP3K12 (DLK) | MLK | TKL | 5vo2 | A | A | 5-{5-[1-(oxetan-3-yl)piperidin-4-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | 8543 | |
| TNNI3K (HH498) | MLK | TKL | 4yfi | B | A | n-methyl-3-(9h-purin-6-ylamino)benzenesulfonamide | Human | 6061 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | B | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9802 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | D | A | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9792 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | A | B | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9800 | |
| TNNI3K (HH498) | MLK | TKL | 6b5j | D | C | n-methyl-3-[(6-{[4-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]benzene-1-sulfonamide | Human | 9795 | |
| MAP3K7 (TAK1) | MLK | TKL | 7nth | A | A | 2-[[5-[[2-[bis(fluoranyl)methoxy]phenyl]methyl-[(2~{r})-1-(methylamino)-1-oxidanylidene-propan-2-yl]carbamoyl]-1~{h}-imidazol-2-yl]carbonyl]isoindole-5-carboxamide | Human | 13456 | |
| MAP3K7 (TAK1) | MLK | TKL | 2yiy | A | | (1e)-1-[5-tert-butyl-2-(3-fluorophenyl)-1h-pyrazol-3-ylidene]-3-(4-pyridin-3-yloxyphenyl)urea | Human | 1890 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l53 | A | A | trans-4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)-3-chlorofuro[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}cyclohexanol | Human | 1887 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jh6 | A | | 2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl prop-2-enoate | Human | 7427 | |
| MAP3K7 (TAK1) | MLK | TKL | 9fpd | A | | 6-[5-[6-(4-oxidanylcyclohexyl)oxy-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-1,2-oxazol-3-yl]pyridine-2-carboxamide | Human | 15551 | |
| MAP3K7 (TAK1) | MLK | TKL | 5j9l | A | | n-(4-((2-((4-(4-methylpiperazin-1-yl)phenyl)amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)phenyl)acrylamide | Human | 7426 | |
| MAP3K7 (TAK1) | MLK | TKL | 4o91 | A | | n-{4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-4-methyl-3-(1h-pyrrolo[2,3-b]pyridin-4-yloxy)benzamide | Human | 1888 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l52 | A | B | 1-(4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}piperidin-1-yl)ethanone | Human | 1889 | |
| MAP3K7 (TAK1) | MLK | TKL | 2eva | A | A | adenosine | Human | 1884 | |
| MAP3K7 (TAK1) | MLK | TKL | 7nth | A | B | 2-[[5-[[2-[bis(fluoranyl)methoxy]phenyl]methyl-[(2~{r})-1-(methylamino)-1-oxidanylidene-propan-2-yl]carbamoyl]-1~{h}-imidazol-2-yl]carbonyl]isoindole-5-carboxamide | Human | 13458 | |
| MAP3K7 (TAK1) | MLK | TKL | 4l52 | A | A | 1-(4-{4-[7-amino-2-(1,2,3-benzothiadiazol-7-yl)furo[2,3-c]pyridin-4-yl]-1h-pyrazol-1-yl}piperidin-1-yl)ethanone | Human | 1883 | |
| MAP3K7 (TAK1) | MLK | TKL | 8gw3 | A | | - | Human | 14877 | |
| MAP3K7 (TAK1) | MLK | TKL | 4gs6 | A | A | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 1885 | |
| MAP3K7 (TAK1) | MLK | TKL | 7nti | A | A | ~{n}-[[2-[bis(fluoranyl)methoxy]phenyl]methyl]-~{n}-[2-(methylamino)-2-oxidanylidene-ethyl]-2-pyrrolidin-1-ylcarbonyl-1~{h}-imidazole-4-carboxamide | Human | 13459 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jgd | A | | n-(2-isopropoxy-3-(4-methylpiperazine-1-carbonyl)phenyl)-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamide | Human | 6884 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jga | A | | n-[5-(4-methylpiperazine-1-carbonyl)[1,1'-biphenyl]-2-yl]-4-oxo-3,4-dihydrothieno[3,2-d]pyrimidine-7-carboxamide | Human | 6886 | |
| MAP3K7 (TAK1) | MLK | TKL | 5j8i | A | | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)oxy]phenyl}prop-2-enamide | Human | 7428 | |
| MAP3K7 (TAK1) | MLK | TKL | 5jk3 | A | | ~{n}-[2-[5-chloranyl-2-[(1-methylpyrazol-4-yl)amino]pyrimidin-4-yl]oxyphenyl]prop-2-enamide | Human | 7430 | |
| MAP3K21 (MLK4) | MLK | TKL | 4uya | A | | phosphothiophosphoric acid-adenylate ester | Human | 6126 | |
| MAP3K20 (ZAK) | MLK | TKL | 5hes | A | B | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6458 | |
| MAP3K20 (ZAK) | MLK | TKL | 5hes | B | A | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6459 | |
| MAP3K20 (ZAK) | MLK | TKL | 5x5o | A | A | n-[2,4-bis(fluoranyl)-3-[2-(3-methoxy-1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-bromanyl-benzenesulfonamide | Human | 9449 | |
| MAP3K20 (ZAK) | MLK | TKL | 7yaw | A | A | ~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamide | Human | 14891 | |
| MAP3K20 (ZAK) | MLK | TKL | 7yaz | A | B | ~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamide | Human | 14892 | |
| MAP3K20 (ZAK) | MLK | TKL | 5hes | A | A | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6460 | |
| MAP3K20 (ZAK) | MLK | TKL | 5x5o | A | B | n-[2,4-bis(fluoranyl)-3-[2-(3-methoxy-1h-pyrazolo[3,4-b]pyridin-5-yl)ethynyl]phenyl]-3-bromanyl-benzenesulfonamide | Human | 9448 | |
| MAP3K20 (ZAK) | MLK | TKL | 6juu | A | B | ~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamide | Human | 12166 | |
| MAP3K20 (ZAK) | MLK | TKL | 7yaw | A | B | ~{n}-[3-[[5-[1-[2,6-bis(fluoranyl)-3-[(3-phenylphenyl)sulfonylamino]phenyl]-1,2,3-triazol-4-yl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]oxy]propyl]propanamide | Human | 14893 | |
| MAP3K20 (ZAK) | MLK | TKL | 5hes | B | B | n-(3-{[5-(4-chlorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]carbonyl}-2,4-difluorophenyl)propane-1-sulfonamide | Human | 6457 | |
| MAP3K20 (ZAK) | MLK | TKL | 7yaz | A | A | ~{n}-[2,4-bis(fluoranyl)-3-[4-[3-[(3~{s})-1-propanoylpyrrolidin-3-yl]oxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl]-1,2,3-triazol-1-yl]phenyl]-3-phenyl-benzenesulfonamide | Human | 14894 | |
| MAP3K20 (ZAK) | MLK | TKL | 6juu | A | A | ~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]naphthalene-1-sulfonamide | Human | 12167 | |
| MAP3K20 (ZAK) | MLK | TKL | 6jut | A | | ~{n}-[2,4-bis(fluoranyl)-3-[4-(3-methoxy-1~{h}-pyrazolo[3,4-b]pyridin-5-yl)-1,2,3-triazol-1-yl]phenyl]-3-bromanyl-benzenesulfonamide | Human | 11462 | |
| ILK | MLK | TKL | 6mib | A | | - | Human | 10687 | |
| ILK | MLK | TKL | 3kmw | A | | adenosine-5'-triphosphate | Human | 4605 | |
| MAP3K12 (DLK) | MLK | TKL | 5cep | A | B | n-(5-piperidin-4-yl-1-propan-2-yl-pyrazol-3-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | 6154 | |
| MAP3K12 (DLK) | MLK | TKL | 5cen | A | A | - | Human | 6157 | |
| MAP3K12 (DLK) | MLK | TKL | 5ceq | A | A | 2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrile | Human | 6159 | |
| MAP3K12 (DLK) | MLK | TKL | 5cep | A | A | n-(5-piperidin-4-yl-1-propan-2-yl-pyrazol-3-yl)-4-(trifluoromethyl)pyridin-2-amine | Human | 6158 | |
| MAP3K12 (DLK) | MLK | TKL | 5ceo | A | A | 2-[[6-[3,3-bis(fluoranyl)pyrrolidin-1-yl]-4-[1-(oxetan-3-yl)piperidin-4-yl]pyridin-2-yl]amino]pyridine-4-carbonitrile | Human | 6156 | |
| MAP3K12 (DLK) | MLK | TKL | 5ceq | A | B | 2-[[1-cyclopentyl-5-[1-(oxetan-3-yl)piperidin-4-yl]pyrazol-3-yl]amino]pyridine-4-carbonitrile | Human | 6153 | |
| MAP3K12 (DLK) | MLK | TKL | 5cen | A | B | - | Human | 6160 | |
| MAP3K12 (DLK) | MLK | TKL | 5vo2 | A | B | 5-{5-[1-(oxetan-3-yl)piperidin-4-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | 8542 | |
| MAP3K12 (DLK) | MLK | TKL | 8ous | A | A | (1s)-1-[4-[6-azanyl-5-(trifluoromethyloxy)pyridin-3-yl]-1-(3-morpholin-4-yl-1-bicyclo[1.1.1]pentanyl)imidazol-2-yl]-2-methyl-propan-1-ol | Human | 14857 | |
| MAP3K12 (DLK) | MLK | TKL | 5vo1 | A | B | 5-{5-[(1r,5s,6r)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | 8541 | |
| MAP3K12 (DLK) | MLK | TKL | 5vo1 | A | A | 5-{5-[(1r,5s,6r)-3-(oxetan-3-yl)-3-azabicyclo[3.1.0]hexan-6-yl]-1-(propan-2-yl)-1h-pyrazol-3-yl}-3-(trifluoromethyl)pyridin-2-amine | Human | 8540 | |
| MAP3K12 (DLK) | MLK | TKL | 5ceo | A | B | 2-[[6-[3,3-bis(fluoranyl)pyrrolidin-1-yl]-4-[1-(oxetan-3-yl)piperidin-4-yl]pyridin-2-yl]amino]pyridine-4-carbonitrile | Human | 6155 | |
| TNNI3K (HH498) | MLK | TKL | 4yff | A | B | 3-[(5-bromo-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]-n-methyl-4-(morpholin-4-yl)benzenesulfonamide | Human | 6062 | |