| STK16 (MPSK1) | NAK | Other | 2buj | B | | staurosporine | Human | 2230 | |
| GAK | NAK | Other | 4y8d | B | B | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | 342 | |
| GAK | NAK | Other | 4c57 | B | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 348 | |
| GAK | NAK | Other | 4c57 | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 340 | |
| GAK | NAK | Other | 4c57 | B | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 334 | |
| GAK | NAK | Other | 4c59 | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 346 | |
| GAK | NAK | Other | 5y80 | A | A | gefitinib | Human | 10329 | |
| GAK | NAK | Other | 4y8d | A | A | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | 344 | |
| GAK | NAK | Other | 4c59 | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 337 | |
| GAK | NAK | Other | 5y7z | A | | gefitinib | Human | 10332 | |
| GAK | NAK | Other | 4c57 | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 341 | |
| AAK1 | NAK | Other | 5te0 | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 7156 | |
| GAK | NAK | Other | 4o38 | B | A | - | Human | 338 | |
| GAK | NAK | Other | 5y7z | B | | gefitinib | Human | 10331 | |
| AAK1 | NAK | Other | 9qb5 | A | | ~{n}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide | Human | 16225 | |
| AAK1 | NAK | Other | 5l4q | B | A | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6680 | |
| AAK1 | NAK | Other | 5l4q | A | B | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6677 | |
| AAK1 | NAK | Other | 8gmd | A | | (5p)-3-({(8r)-5-[(4-aminopiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-[2-(propan-2-yl)-2h-tetrazol-5-yl]phenol | Human | 14844 | |
| AAK1 | NAK | Other | 8gmc | A | | 5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 14843 | |
| GAK | NAK | Other | 4o38 | A | B | - | Human | 335 | |
| GAK | NAK | Other | 4c58 | A | B | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 333 | |
| BMP2K (BIKE) | NAK | Other | 5i3o | B | | n-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamide | Human | 6434 | |
| BMP2K (BIKE) | NAK | Other | 5ikw | A | | n-(6-{3-[(cyclopropylsulfonyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamide | Human | 6709 | |
| BMP2K (BIKE) | NAK | Other | 5i3o | A | | n-(6-{3-[(dimethylsulfamoyl)amino]phenyl}-1h-indazol-3-yl)cyclopropanecarboxamide | Human | 6437 | |
| BMP2K (BIKE) | NAK | Other | 4w9x | A | | baricitinib | Human | 3273 | |
| GAK | NAK | Other | 4y8d | B | A | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | 347 | |
| GAK | NAK | Other | 4o38 | A | A | - | Human | 345 | |
| GAK | NAK | Other | 5y80 | A | B | gefitinib | Human | 10330 | |
| GAK | NAK | Other | 4c58 | A | A | 9-hydroxy-4-phenylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 336 | |
| GAK | NAK | Other | 4o38 | B | B | - | Human | 343 | |
| GAK | NAK | Other | 4y8d | A | B | 2-methoxy-4-[3-(morpholin-4-yl)[1,2]thiazolo[4,3-b]pyridin-6-yl]aniline | Human | 339 | |
| STK16 (MPSK1) | NAK | Other | 2buj | A | | staurosporine | Human | 2229 | |
| BMP2K (BIKE) | NAK | Other | 5i3r | B | | n-[6-(3-{[(cyclopropylmethyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]cyclopropanecarboxamide | Human | 6436 | |
| BMP2K (BIKE) | NAK | Other | 5i3r | A | | n-[6-(3-{[(cyclopropylmethyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]cyclopropanecarboxamide | Human | 6435 | |
| BMP2K (BIKE) | NAK | Other | 4w9w | A | A | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 3274 | |
| BMP2K (BIKE) | NAK | Other | 4w9w | A | B | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 3272 | |
| AAK1 | NAK | Other | 5l4q | A | A | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6679 | |
| AAK1 | NAK | Other | 4wsq | B | B | k-252a | Human | 3835 | |
| AAK1 | NAK | Other | 4wsq | A | A | k-252a | Human | 3834 | |
| AAK1 | NAK | Other | 5l4q | B | B | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6678 | |
| AAK1 | NAK | Other | 4wsq | B | A | k-252a | Human | 3833 | |
| AAK1 | NAK | Other | 4wsq | A | B | k-252a | Human | 3836 | |
