Search results (9 entries covering 5 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
| Aak1 (AAK1) | NAK | Other | 7rj6 | A | B | 5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Mouse | 14131 | ||
| Aak1 (AAK1) | NAK | Other | 7rj7 | A | A | 2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrile | Mouse | 14128 | ||
| Aak1 (AAK1) | NAK | Other | 7lvi | A | B | (2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamide | Mouse | 13821 | ||
| Aak1 (AAK1) | NAK | Other | 7lvi | A | A | (2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamide | Mouse | 13822 | ||
| Aak1 (AAK1) | NAK | Other | 7lvh | A | n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamide | Mouse | 13820 | |||
| Aak1 (AAK1) | NAK | Other | 7rj8 | A | B | n-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamide | Mouse | 14127 | ||
| Aak1 (AAK1) | NAK | Other | 7rj7 | A | B | 2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrile | Mouse | 14129 | ||
| Aak1 (AAK1) | NAK | Other | 7rj8 | A | A | n-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamide | Mouse | 14130 | ||
| Aak1 (AAK1) | NAK | Other | 7rj6 | A | A | 5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Mouse | 14132 |