Search results (9 entries covering 5 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
Aak1 (AAK1)NAKOther7rj6AB5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineMouse14131
Aak1 (AAK1)NAKOther7rj7AA2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrileMouse14128
Aak1 (AAK1)NAKOther7lviAB(2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamideMouse13821
Aak1 (AAK1)NAKOther7lviAA(2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamideMouse13822
Aak1 (AAK1)NAKOther7lvhAn-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse13820
Aak1 (AAK1)NAKOther7rj8ABn-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse14127
Aak1 (AAK1)NAKOther7rj7AB2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrileMouse14129
Aak1 (AAK1)NAKOther7rj8AAn-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse14130
Aak1 (AAK1)NAKOther7rj6AA5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineMouse14132