Search results (86 entries covering 42 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
NEK7NEKOther8sxnA-Human15246
NEK7NEKOther8ws0AB-Human15995
NEK7NEKOther9nfqCadenosine-5'-diphosphateHuman15996
NEK7NEKOther8ws1AB-Human15997
NEK7NEKOther8ws1AA-Human15998
NEK7NEKOther8ws0AA-Human15999
NEK2NEKOther2w5bABphosphothiophosphoric acid-adenylate esterHuman305
NEK2NEKOther6sghAA2-[4-[(6-ethenyl-9~{h}-purin-2-yl)amino]phenyl]ethanamideHuman12374
NEK2NEKOther6sk9AA3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12376
NEK7NEKOther2wqnAAadenosine-5'-diphosphateHuman3855
NEK7NEKOther6s76D-Human12361
NEK2NEKOther2w5bAAphosphothiophosphoric acid-adenylate esterHuman320
NEK2NEKOther6sgdAB4-[(6-ethenyl-7~{h}-purin-2-yl)amino]benzenesulfonamideHuman12375
NEK2NEKOther2xnpAB4-{5-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamideHuman322
NEK2NEKOther2xkfAB1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acidHuman311
NEK2NEKOther2xkfAA1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acidHuman315
NEK2NEKOther5m53AA3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n},~{n}-dimethyl-benzamideHuman7159
NEK7NEKOther6s76A-Human12351
NEK7NEKOther6s76C-Human12352
NEK1NEKOther4apcAA-Human1215
NEK1NEKOther4apcAB-Human1208
NEK1NEKOther4b9dBB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman1209
NEK1NEKOther4b9dAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman1211
NEK1NEKOther4b9dAB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman1213
NEK1NEKOther4apcBB-Human1210
NEK1NEKOther4apcBA-Human1212
NEK1NEKOther4b9dBA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman1214
NEK2NEKOther2w5hAA-Human327
NEK2NEKOther2xk7AA(3r,4r)-1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-3-ethylpiperidine-4-carboxylic acidHuman326
NEK2NEKOther2xk3AA4-[3-amino-6-(3-ethylthiophen-2-yl)pyrazin-2-yl]cyclohexane-1-carboxylic acidHuman309
NEK2NEKOther2w5aAAadenosine-5'-diphosphateHuman302
NEK2NEKOther2xkcAB4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methylbenzoic acidHuman307
NEK2NEKOther2xkeA1-[3-amino-6-(3-methoxyphenyl)pyrazin-2-yl]piperidine-4-carboxylic acidHuman299
NEK2NEKOther2xkcAA4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methylbenzoic acidHuman321
NEK2NEKOther2xk8A4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-methoxybenzoic acidHuman300
NEK2NEKOther6sghAB2-[4-[(6-ethenyl-9~{h}-purin-2-yl)amino]phenyl]ethanamideHuman12372
NEK2NEKOther2javAB5-[(z)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman323
NEK2NEKOther2javAA5-[(z)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman332
NEK2NEKOther2xnoAA5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{[2-(trifluoromethyl)benzyl]oxy}thiophene-2-carboxamideHuman319
NEK2NEKOther5m55AA6-[(~{z})-2-(diethylamino)ethenyl]-~{n}-phenyl-7~{h}-purin-2-amineHuman7140
NEK2NEKOther4afeA4-(2-amino-5-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridin-3-yl)-2-{[(1r,2z)-4,4,4-trifluoro-1-methylbut-2-en-1-yl]oxy}benzamideHuman312
NEK2NEKOther4a4xA4-(2-amino-5-{4-[(dimethylamino)methyl]thiophen-2-yl}pyridin-3-yl)-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamideHuman325
NEK2NEKOther6sgdAA4-[(6-ethenyl-7~{h}-purin-2-yl)amino]benzenesulfonamideHuman12373
NEK2NEKOther2w5hAB-Human310
NEK2NEKOther2xkdAA4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]benzoic acidHuman330
NEK2NEKOther2xnmAB5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamideHuman324
NEK2NEKOther2xnnAB5-(1h-benzimidazol-1-yl)-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamideHuman308
NEK2NEKOther2xk4AC4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acidHuman304
NEK2NEKOther2xk3AB4-[3-amino-6-(3-ethylthiophen-2-yl)pyrazin-2-yl]cyclohexane-1-carboxylic acidHuman329
NEK2NEKOther5m55AB6-[(~{z})-2-(diethylamino)ethenyl]-~{n}-phenyl-7~{h}-purin-2-amineHuman7139
NEK2NEKOther5m57Ao6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7272
NEK2NEKOther2xk4AB4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acidHuman316
NEK2NEKOther2w5aABadenosine-5'-diphosphateHuman317
NEK2NEKOther2xk7AB(3r,4r)-1-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-3-ethylpiperidine-4-carboxylic acidHuman318
NEK2NEKOther2xk4AA4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]-2-ethoxybenzoic acidHuman314
NEK2NEKOther2xnnAA5-(1h-benzimidazol-1-yl)-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamideHuman303
NEK2NEKOther6sgkA2-phenylazanyl-9~{h}-purine-6-carbonitrileHuman12377
NEK2NEKOther2wqoA4-[2-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]benzoic acidHuman331
NEK2NEKOther6sgiAA4-[(6-ethyl-7~{h}-purin-2-yl)amino]benzenesulfonamideHuman12378
NEK2NEKOther6sk9AB3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12379
NEK2NEKOther5m51A3-[[6-(cyclohexylmethoxy)-9~{h}-purin-2-yl]amino]benzamideHuman7157
NEK2NEKOther2xnoAB5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{[2-(trifluoromethyl)benzyl]oxy}thiophene-2-carboxamideHuman313
NEK2NEKOther5m53AB3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n},~{n}-dimethyl-benzamideHuman7161
NEK2NEKOther6sgiAB4-[(6-ethyl-7~{h}-purin-2-yl)amino]benzenesulfonamideHuman12380
NEK2NEKOther2xnpAA4-{5-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-2-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}benzamideHuman328
NEK2NEKOther2xkdAB4-[3-amino-6-(3,4,5-trimethoxyphenyl)pyrazin-2-yl]benzoic acidHuman298
NEK2NEKOther2xnmAA5-{6-[(1-methylpiperidin-4-yl)oxy]-1h-benzimidazol-1-yl}-3-{(1r)-1-[2-(trifluoromethyl)phenyl]ethoxy}thiophene-2-carboxamideHuman306
NEK2NEKOther2xk6Acis-4-[3-amino-6-(3-cyclopropylthiophen-2-yl)pyrazin-2-yl]cyclohexanecarboxylic acidHuman301
NEK7NEKOther5de2AA-Human6246
NEK7NEKOther6s73B3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12353
NEK7NEKOther6s76B-Human12354
NEK7NEKOther5de2BA-Human6245
NEK7NEKOther6s73D-Human12355
NEK7NEKOther6npyBA-Human11338
NEK7NEKOther6s75A3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12356
NEK7NEKOther6s73A3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12357
NEK7NEKOther6s75B3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12358
NEK7NEKOther2wqnABadenosine-5'-diphosphateHuman3856
NEK7NEKOther6npyBB-Human11337
NEK7NEKOther6s75D-Human12359
NEK7NEKOther6s75C3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12360
NEK7NEKOther2wqmAA-Human3854
NEK7NEKOther5de2BB-Human6247
NEK7NEKOther5de2AB-Human6244
NEK7NEKOther6s73C3-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]-~{n}-[3-(dimethylamino)propyl]benzenesulfonamideHuman12362
NEK7NEKOther2wqmAB-Human3857