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Search results (128 entries covering 65 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PDPK1 (PDK1)PDK1AGC3orzAB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3181
PDPK1 (PDK1)PDK1AGC1okyAAstaurosporineHuman3164
PDPK1 (PDK1)PDK1AGC5lvnAAadenosineHuman7105
PDPK1 (PDK1)PDK1AGC5hngA6-methoxy-2-(1h-pyrazol-5-yl)-1h-benzimidazoleHuman6675
PDPK1 (PDK1)PDK1AGC1uu3AA(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHuman3180
PDPK1 (PDK1)PDK1AGC8dqtA-Human14812
PDPK1 (PDK1)PDK1AGC3orxC-Human3245
PDPK1 (PDK1)PDK1AGC3qcyAA(2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamideHuman3151
PDPK1 (PDK1)PDK1AGC3qcxAA6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amineHuman3187
PDPK1 (PDK1)PDK1AGC4rqkAAadenosine-5'-triphosphateHuman3175
PDPK1 (PDK1)PDK1AGC4a06ABadenosine-5'-triphosphateHuman3227
PDPK1 (PDK1)PDK1AGC3orzDB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3184
PDPK1 (PDK1)PDK1AGC3rcjA3-(1-benzyl-1h-1,2,3-triazol-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman3154
PDPK1 (PDK1)PDK1AGC3ionA2-(5-{[(2s)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amineHuman3218
PDPK1 (PDK1)PDK1AGC5ho7AA5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamideHuman6673
PDPK1 (PDK1)PDK1AGC2pe0A5-hydroxy-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-2-oneHuman3206
PDPK1 (PDK1)PDK1AGC5lvpBadenosine-5'-triphosphateHuman7113
PDPK1 (PDK1)PDK1AGC3nuuAA3,4-dihydroisoquinolin-1(2h)-oneHuman3214
PDPK1 (PDK1)PDK1AGC3qcqAA6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamineHuman3205
PDPK1 (PDK1)PDK1AGC1uu8AB3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3237
PDPK1 (PDK1)PDK1AGC5ho7AB5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamideHuman6671
PDPK1 (PDK1)PDK1AGC3qcyAB(2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamideHuman3161
PDPK1 (PDK1)PDK1AGC3nunAB6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amineHuman3216
PDPK1 (PDK1)PDK1AGC5lvlAA2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHuman7106
PDPK1 (PDK1)PDK1AGC3nuyABquinazolin-4(1h)-oneHuman3242
PDPK1 (PDK1)PDK1AGC3qcsAB6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amineHuman3157
PDPK1 (PDK1)PDK1AGC5lvpAadenosine-5'-triphosphateHuman7102
PDPK1 (PDK1)PDK1AGC3qd3AAtert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamateHuman3188
PDPK1 (PDK1)PDK1AGC1uvrA3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3193
PDPK1 (PDK1)PDK1AGC3rwpAA[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanoneHuman3208
PDPK1 (PDK1)PDK1AGC2biyAAadenosine-5'-triphosphateHuman3232
PDPK1 (PDK1)PDK1AGC4ct2AAadenosine-5'-triphosphateHuman3153
PDPK1 (PDK1)PDK1AGC3orxD-Human3210
PDPK1 (PDK1)PDK1AGC4rqvABadenosine-5'-triphosphateHuman3182
PDPK1 (PDK1)PDK1AGC4xx9ABadenosine-5'-triphosphateHuman6192
PDPK1 (PDK1)PDK1AGC5lvmACadenineHuman7138
PDPK1 (PDK1)PDK1AGC1uu7A3-(1h-indol-3-yl)-4-(1-{2-[(2s)-1-methylpyrrolidinyl]ethyl}-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3224
PDPK1 (PDK1)PDK1AGC3orxE-Human3202
PDPK1 (PDK1)PDK1AGC3qc4BB1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman9256
PDPK1 (PDK1)PDK1AGC4aw1AAadenosine-5'-triphosphateHuman3229
PDPK1 (PDK1)PDK1AGC3qd3ABtert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamateHuman3171
PDPK1 (PDK1)PDK1AGC4aw1ABadenosine-5'-triphosphateHuman3221
PDPK1 (PDK1)PDK1AGC3rwqA[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[2-(pyridin-3-yl)ethyl]amino}pyrazin-2-yl)methanoneHuman3213
PDPK1 (PDK1)PDK1AGC3qd0AA(3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamideHuman3196
PDPK1 (PDK1)PDK1AGC3sc1A6-[2-(hydroxymethyl)phenyl]isoquinolin-1(2h)-oneHuman3173
PDPK1 (PDK1)PDK1AGC5lvlAB2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHuman7110
PDPK1 (PDK1)PDK1AGC3qc4AA1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman9254
PDPK1 (PDK1)PDK1AGC5lvpCadenosine-5'-triphosphateHuman7111
PDPK1 (PDK1)PDK1AGC3orzBA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3160
PDPK1 (PDK1)PDK1AGC4ct1ABadenosine-5'-triphosphateHuman3168
PDPK1 (PDK1)PDK1AGC3hrfABadenosine-5'-triphosphateHuman3247
PDPK1 (PDK1)PDK1AGC4rqkABadenosine-5'-triphosphateHuman3156
PDPK1 (PDK1)PDK1AGC5mrdABadenosine-5'-triphosphateHuman7394
PDPK1 (PDK1)PDK1AGC1uu3AB(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHuman3248
PDPK1 (PDK1)PDK1AGC1z5mAn-(3-{[5-bromo-2-({3-[(pyrrolidin-1-ylcarbonyl)amino]phenyl}amino)pyrimidin-4-yl]amino}propyl)-2,2-dimethylmalonamideHuman3152
PDPK1 (PDK1)PDK1AGC5ho8AB4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman6672
PDPK1 (PDK1)PDK1AGC3orxB-Human3178
PDPK1 (PDK1)PDK1AGC4rrvAAadenosine-5'-triphosphateHuman3244
PDPK1 (PDK1)PDK1AGC5mrdAAadenosine-5'-triphosphateHuman7395
PDPK1 (PDK1)PDK1AGC1uu9AB3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman6799
PDPK1 (PDK1)PDK1AGC4aw0AAadenosine-5'-triphosphateHuman3176
PDPK1 (PDK1)PDK1AGC3pwyAn-[2-({6-[(2-sulfanylethyl)amino]pyrimidin-4-yl}amino)ethyl]propanamideHuman3155
PDPK1 (PDK1)PDK1AGC3nunAA6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amineHuman3183
PDPK1 (PDK1)PDK1AGC3iopA2-(5-{[(2r)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amineHuman3204
PDPK1 (PDK1)PDK1AGC2r7bA10,11-dimethoxy-4-methyldibenzo[c,f]-2,7-naphthyridine-3,6-diamineHuman3215
PDPK1 (PDK1)PDK1AGC3qd4ABtert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamateHuman3190
PDPK1 (PDK1)PDK1AGC4a07ABadenosine-5'-triphosphateHuman3238
PDPK1 (PDK1)PDK1AGC4ct2ABadenosine-5'-triphosphateHuman3230
PDPK1 (PDK1)PDK1AGC3orzCA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3150
PDPK1 (PDK1)PDK1AGC3qcxAB6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amineHuman3249
PDPK1 (PDK1)PDK1AGC3orxA-Human3235
PDPK1 (PDK1)PDK1AGC3orzCB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3243
PDPK1 (PDK1)PDK1AGC2biyABadenosine-5'-triphosphateHuman3169
PDPK1 (PDK1)PDK1AGC4a07AAadenosine-5'-triphosphateHuman3234
PDPK1 (PDK1)PDK1AGC5lvnABadenosineHuman7109
PDPK1 (PDK1)PDK1AGC3nuuAB3,4-dihydroisoquinolin-1(2h)-oneHuman3159
PDPK1 (PDK1)PDK1AGC1okzA7-hydroxystaurosporineHuman3209
PDPK1 (PDK1)PDK1AGC5ackAAadenosine-5'-triphosphateHuman6191
PDPK1 (PDK1)PDK1AGC3orzAA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3197
PDPK1 (PDK1)PDK1AGC3qd0AB(3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamideHuman3162
PDPK1 (PDK1)PDK1AGC3nuyAAquinazolin-4(1h)-oneHuman3236
PDPK1 (PDK1)PDK1AGC5lvoAAadenosine-5'-triphosphateHuman7104
PDPK1 (PDK1)PDK1AGC3qc4AB1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman9253
PDPK1 (PDK1)PDK1AGC4aw0ABadenosine-5'-triphosphateHuman3241
PDPK1 (PDK1)PDK1AGC3qcsAA6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amineHuman3179
PDPK1 (PDK1)PDK1AGC4rrvACadenosine-5'-triphosphateHuman3191
PDPK1 (PDK1)PDK1AGC3h9oA2-(1h-imidazol-1-yl)-9-methoxy-8-(2-methoxyethoxy)benzo[c][2,7]naphthyridin-4-amineHuman3226
PDPK1 (PDK1)PDK1AGC3hrcAAadenosine-5'-triphosphateHuman3172
PDPK1 (PDK1)PDK1AGC5lvmAAadenineHuman7112
PDPK1 (PDK1)PDK1AGC4rqkACadenosine-5'-triphosphateHuman3211
PDPK1 (PDK1)PDK1AGC3nusAB1h-indazol-3-amineHuman3185
PDPK1 (PDK1)PDK1AGC1uu8AA3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3239
PDPK1 (PDK1)PDK1AGC3rwpAB[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanoneHuman3199
PDPK1 (PDK1)PDK1AGC2xchA8-(cyclohexa-2,5-dien-1-ylideneamino)-1-(piperidin-4-ylmethyl)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman3220
PDPK1 (PDK1)PDK1AGC3hrcABadenosine-5'-triphosphateHuman3223
PDPK1 (PDK1)PDK1AGC5lvpDadenosine-5'-triphosphateHuman7108
PDPK1 (PDK1)PDK1AGC4rqvACadenosine-5'-triphosphateHuman3222
PDPK1 (PDK1)PDK1AGC5lvoABadenosine-5'-triphosphateHuman7114
PDPK1 (PDK1)PDK1AGC3nayA4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-oneHuman3231
PDPK1 (PDK1)PDK1AGC3orxH-Human3177
PDPK1 (PDK1)PDK1AGC3orzDA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3192
PDPK1 (PDK1)PDK1AGC2xckA1-methyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-n-[(2-methylpyridin-4-yl)methyl]-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman3201
PDPK1 (PDK1)PDK1AGC2pe2A3-[5-({5-[(aminocarbonyl)amino]-2-oxo-2h-indol-3-yl}methyl)-1h-pyrrol-3-yl]-n-(2-piperidin-1-ylethyl)benzamideHuman3163
PDPK1 (PDK1)PDK1AGC3nusAA1h-indazol-3-amineHuman3233
PDPK1 (PDK1)PDK1AGC3orxF-Human3228
PDPK1 (PDK1)PDK1AGC3hrfAAadenosine-5'-triphosphateHuman3170
PDPK1 (PDK1)PDK1AGC2pe1A1-{2-oxo-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-5-yl}ureaHuman3167
PDPK1 (PDK1)PDK1AGC4rrvABadenosine-5'-triphosphateHuman3212
PDPK1 (PDK1)PDK1AGC4ct1AAadenosine-5'-triphosphateHuman3158
PDPK1 (PDK1)PDK1AGC5hkmA4-ethyl-6-[5-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-2-amineHuman6670
PDPK1 (PDK1)PDK1AGC3orzBB3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3198
PDPK1 (PDK1)PDK1AGC4rqvAAadenosine-5'-triphosphateHuman3219
PDPK1 (PDK1)PDK1AGC1h1wABadenosine-5'-triphosphateHuman3194
PDPK1 (PDK1)PDK1AGC3orxG-Human3189
PDPK1 (PDK1)PDK1AGC3qd4AAtert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamateHuman3225
PDPK1 (PDK1)PDK1AGC3qc4BA1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman9255
PDPK1 (PDK1)PDK1AGC3otuA3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dioneHuman3217
PDPK1 (PDK1)PDK1AGC3qcqAB6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamineHuman3166
PDPK1 (PDK1)PDK1AGC4a06AAadenosine-5'-triphosphateHuman3207
PDPK1 (PDK1)PDK1AGC5ho8AA4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman6674
PDPK1 (PDK1)PDK1AGC4xx9AAadenosine-5'-triphosphateHuman6193
PDPK1 (PDK1)PDK1AGC1h1wAAadenosine-5'-triphosphateHuman3186
PDPK1 (PDK1)PDK1AGC5ackABadenosine-5'-triphosphateHuman6194
PDPK1 (PDK1)PDK1AGC3naxA1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamideHuman3200
PDPK1 (PDK1)PDK1AGC5lvmABadenineHuman7103
PDPK1 (PDK1)PDK1AGC3nayB4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-oneHuman3203
PDPK1 (PDK1)PDK1AGC1uu9AA3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman6800
PDPK1 (PDK1)PDK1AGC1okyABstaurosporineHuman3195
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