Search results (44 entries covering 27 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
EIF2AK2 (PKR)PEKOther6d3lA-Human11384
EIF2AK2 (PKR)PEKOther6d3kBadenosine-5'-diphosphateHuman11385
EIF2AK2 (PKR)PEKOther6d3kAadenosine-5'-diphosphateHuman11386
EIF2AK2 (PKR)PEKOther8qelB(3~{z})-3-[(4-methyl-1~{h}-imidazol-5-yl)methylidene]-2-oxidanylidene-1~{h}-indole-5-carboxamideHuman14954
EIF2AK2 (PKR)PEKOther2a19Bphosphoaminophosphonic acid-adenylate esterHuman920
EIF2AK2 (PKR)PEKOther3uiuB-Human916
EIF2AK1 (HRI)PEKOther9rhhA-Human15549
EIF2AK4 (GCN2)PEKOther6n3lAAn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHuman11691
EIF2AK4 (GCN2)PEKOther8t7tAA-Human15229
EIF2AK3 (PEK)PEKOther4x7hABn-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1h-pyrazole-4-carboxamideHuman7240
EIF2AK3 (PEK)PEKOther4g34AB1-[5-(4-aminothieno[3,2-c]pyridin-3-yl)-2,3-dihydro-1h-indol-1-yl]-2-phenylethanoneHuman2670
EIF2AK3 (PEK)PEKOther4x7kAB4-{2-amino-3-[5-fluoro-2-(methylamino)quinazolin-6-yl]-4-methylbenzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman7242
EIF2AK3 (PEK)PEKOther4x7oAB1-[5-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanoneHuman7244
EIF2AK3 (PEK)PEKOther8eqeA(2r)-n-[(4m)-4-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-hydroxy-2-[3-(trifluoromethyl)phenyl]acetamideHuman14522
EIF2AK3 (PEK)PEKOther4x7nAB4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman7241
EIF2AK3 (PEK)PEKOther4m7iA1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-4-fluoro-1h-indol-1-yl]-2-(6-methylpyridin-2-yl)ethanoneHuman2673
EIF2AK2 (PKR)PEKOther3uiuA-Human917
EIF2AK2 (PKR)PEKOther9yufAdabrafenibHuman15962
EIF2AK2 (PKR)PEKOther2a1aB-Human919
EIF2AK2 (PKR)PEKOther2a19Cphosphoaminophosphonic acid-adenylate esterHuman918
EIF2AK2 (PKR)PEKOther6d3kCadenosine-5'-diphosphateHuman11387
EIF2AK4 (GCN2)PEKOther6n3nAn-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-2,5-dichloro-3-(hydroxymethyl)benzene-1-sulfonamideHuman11690
EIF2AK4 (GCN2)PEKOther7qwkA(2~{s})-~{n}-[(1~{s})-1-[4-[(6-pyridin-4-ylquinazolin-2-yl)amino]phenyl]ethyl]piperidine-2-carboxamideHuman14209
EIF2AK4 (GCN2)PEKOther6n3lBAn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHuman11693
EIF2AK4 (GCN2)PEKOther6n3lBBn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHuman11692
EIF2AK4 (GCN2)PEKOther6n3lABn-{6-[(1-methyl-2-{[4-(trifluoromethyl)phenyl]amino}-1h-benzimidazol-5-yl)oxy]pyrimidin-4-yl}cyclopropanecarboxamideHuman11694
EIF2AK4 (GCN2)PEKOther7qq6A4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman14116
EIF2AK4 (GCN2)PEKOther8t7tAB-Human15230
EIF2AK3 (PEK)PEKOther4g31AB1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanoneHuman2671
EIF2AK3 (PEK)PEKOther4x7lAB4-{2-amino-4-methyl-3-[2-(methylamino)-1,3-benzothiazol-6-yl]benzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman6843
EIF2AK3 (PEK)PEKOther4x7jAA2-amino-n-[4-methoxy-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamideHuman6848
EIF2AK3 (PEK)PEKOther8eq9AB(2r)-n-[(4m)-4-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamideHuman14521
EIF2AK3 (PEK)PEKOther4x7jAB2-amino-n-[4-methoxy-3-(trifluoromethyl)phenyl]-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamideHuman6841
EIF2AK3 (PEK)PEKOther4x7kAA4-{2-amino-3-[5-fluoro-2-(methylamino)quinazolin-6-yl]-4-methylbenzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman7246
EIF2AK3 (PEK)PEKOther4x7nAA4-[2-amino-4-methyl-3-(2-methylquinolin-6-yl)benzoyl]-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman7245
EIF2AK3 (PEK)PEKOther4g31AA1-[5-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-(trifluoromethyl)phenyl]ethanoneHuman2672
EIF2AK3 (PEK)PEKOther4x7oAA1-[5-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1h-indol-1-yl]-2-[3-fluoro-5-(trifluoromethyl)phenyl]ethanoneHuman7243
EIF2AK3 (PEK)PEKOther7mf0A2-amino-n-cyclopropyl-5-(4-{[(2r)-2-(3,5-difluorophenyl)-2-hydroxyacetyl]amino}-2-methylphenyl)pyridine-3-carboxamideHuman13577
EIF2AK3 (PEK)PEKOther8eqdA(2r)-n-[(4m)-4-(4-amino-2,7-dimethyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamideHuman14523
EIF2AK3 (PEK)PEKOther8eq9AA(2r)-n-[(4m)-4-(4-amino-7-methyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-3-methylphenyl]-2-(3-fluorophenyl)-2-hydroxyacetamideHuman14524
EIF2AK3 (PEK)PEKOther4x7hAAn-{5-[(6,7-dimethoxyquinolin-4-yl)oxy]pyridin-2-yl}-1-methyl-3-oxo-2-phenyl-5-(pyridin-4-yl)-2,3-dihydro-1h-pyrazole-4-carboxamideHuman7247
EIF2AK3 (PEK)PEKOther4x7lAA4-{2-amino-4-methyl-3-[2-(methylamino)-1,3-benzothiazol-6-yl]benzoyl}-1-methyl-2,5-diphenyl-1,2-dihydro-3h-pyrazol-3-oneHuman6844
EIF2AK3 (PEK)PEKOther4g34AA1-[5-(4-aminothieno[3,2-c]pyridin-3-yl)-2,3-dihydro-1h-indol-1-yl]-2-phenylethanoneHuman2674
EIF2AK4 (GCN2)PEKOther6n3oAn-{3-[(2-aminopyrimidin-5-yl)ethynyl]-2,4-difluorophenyl}-5-chloro-2-methoxypyridine-3-sulfonamideHuman11695