| TRRAP | PIKK | Atypical | 8xvg | A | B | adenosine-5'-diphosphate | Human | 15323 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k11 | A | | - | Human | 13208 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 5luq | B | | - | Human | 9319 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7sgl | A | B | adenosine-5'-triphosphate | Human | 14062 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsp | A | | phosphothiophosphoric acid-adenylate ester | Human | 9106 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7sud | A | A | adenosine-5'-triphosphate | Human | 14055 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7z87 | A | A | (~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanol | Human | 14592 | |
| SMG1 | PIKK | Atypical | 6l53 | A | | - | Human | 12156 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7su3 | A | B | adenosine-5'-triphosphate | Human | 14053 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k17 | B | | - | Human | 13212 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7oty | A | | (~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanol | Human | 14057 | |
| ATM | PIKK | Atypical | 7ni4 | A | | 8-(1,3-dimethylpyrazol-4-yl)-1-(3-fluoranyl-5-methoxy-pyridin-4-yl)-7-methoxy-3-methyl-imidazo[4,5-c]quinolin-2-one | Human | 13864 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7otm | A | | 8-(dibenzo[b,d]thiophen-4-yl)-2-(morpholin-4-yl)-4h-chromen-4-one | Human | 14061 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 8ezb | C | | adenosine-5'-triphosphate | Human | 14798 | |
| ATR | PIKK | Atypical | 9zd1 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15662 | |
| ATR | PIKK | Atypical | 23fd | A | | phosphothiophosphoric acid-adenylate ester | Human | 15663 | |
| MTOR (FRAP) | PIKK | Atypical | 9tds | A | | - | Human | 15768 | |
| MTOR (FRAP) | PIKK | Atypical | 9t92 | A | | - | Human | 15765 | |
| MTOR (FRAP) | PIKK | Atypical | 9ed7 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15766 | |
| MTOR (FRAP) | PIKK | Atypical | 9t93 | A | | - | Human | 15767 | |
| MTOR (FRAP) | PIKK | Atypical | 9zbj | A | | - | Human | 15769 | |
| MTOR (FRAP) | PIKK | Atypical | 9zbk | A | | - | Human | 15770 | |
| MTOR (FRAP) | PIKK | Atypical | 9t7j | A | | adenosine-5'-triphosphate | Human | 15771 | |
| MTOR (FRAP) | PIKK | Atypical | 9tdt | A | | - | Human | 15772 | |
| MTOR (FRAP) | PIKK | Atypical | 8rch | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15773 | |
| MTOR (FRAP) | PIKK | Atypical | 9tpw | A | | - | Human | 15774 | |
| TRRAP | PIKK | Atypical | 9rdk | E | | - | Human | 15849 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 9iax | A | | - | Human | 16042 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 9zob | A | | - | Human | 16043 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7tyr | A | B | - | Human | 14321 | |
| ATM | PIKK | Atypical | 8oxq | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14990 | |
| ATM | PIKK | Atypical | 8oxp | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14991 | |
| ATM | PIKK | Atypical | 6k9l | A | | - | Human | 11896 | |
| ATM | PIKK | Atypical | 8oxm | B | | phosphoaminophosphonic acid-adenylate ester | Human | 14992 | |
| ATM | PIKK | Atypical | 8oxo | B | | phosphoaminophosphonic acid-adenylate ester | Human | 14993 | |
| SMG1 | PIKK | Atypical | 7pw9 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14000 | |
| SMG1 | PIKK | Atypical | 7pw7 | A | | 1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-urea | Human | 14005 | |
| SMG1 | PIKK | Atypical | 7pw6 | A | | 1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-urea | Human | 14001 | |
| SMG1 | PIKK | Atypical | 6syt | A | | - | Human | 11866 | |
| ATM | PIKK | Atypical | 6k9l | B | | - | Human | 11895 | |
| SMG1 | PIKK | Atypical | 7pw5 | A | | 1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-urea | Human | 14002 | |
| SMG1 | PIKK | Atypical | 6l54 | A | | - | Human | 12155 | |
| SMG1 | PIKK | Atypical | 7pw4 | A | | 1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-urea | Human | 14003 | |
| SMG1 | PIKK | Atypical | 7pw8 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14004 | |
| SMG1 | PIKK | Atypical | 6z3r | A | | phosphoaminophosphonic acid-adenylate ester | Human | 12630 | |
| MTOR (FRAP) | PIKK | Atypical | 5zcs | B | | - | Human | 9749 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zh2 | A | | - | Human | 12927 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7su3 | A | A | adenosine-5'-triphosphate | Human | 14058 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zhe | A | | - | Human | 12928 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7sgl | A | A | adenosine-5'-triphosphate | Human | 14059 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zh6 | A | | - | Human | 12929 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7sud | A | B | adenosine-5'-triphosphate | Human | 14060 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7z87 | A | B | (~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanol | Human | 14593 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7otv | A | | (1s,6br,9as,11r,11br)-9a,11b-dimethyl-1-[(methyloxy)methyl]-3,6,9-trioxo-1,6,6b,7,8,9,9a,10,11,11b-decahydro-3h-furo[4,3,2-de]indeno[4,5-h][2]benzopyran-11-yl acetate | Human | 14063 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7nfc | A | | - | Human | 13852 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zha | A | | - | Human | 12931 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7z88 | A | | (~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanol | Human | 14594 | |
| ATM | PIKK | Atypical | 7ni6 | A | | phosphothiophosphoric acid-adenylate ester | Human | 13862 | |
| ATM | PIKK | Atypical | 5np0 | B | | - | Human | 9266 | |
| ATM | PIKK | Atypical | 7sic | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14101 | |
| ATM | PIKK | Atypical | 5np0 | A | | - | Human | 9267 | |
| ATM | PIKK | Atypical | 7ni5 | A | | 2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-one | Human | 13863 | |
| ATM | PIKK | Atypical | 6k9k | A | | - | Human | 11897 | |
| ATR | PIKK | Atypical | 9l4d | A | | camonsertib | Human | 15644 | |
| ATR | PIKK | Atypical | 23fc | A | | phosphothiophosphoric acid-adenylate ester | Human | 15653 | |
| ATR | PIKK | Atypical | 9zcy | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15654 | |
| ATR | PIKK | Atypical | 9zd3 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15655 | |
| ATR | PIKK | Atypical | 26zn | A | | phosphothiophosphoric acid-adenylate ester | Human | 15656 | |
| ATR | PIKK | Atypical | 23fe | A | | phosphothiophosphoric acid-adenylate ester | Human | 15657 | |
| ATR | PIKK | Atypical | 5yz0 | B | | - | Human | 9524 | |
| ATR | PIKK | Atypical | 9l4b | A | | camonsertib | Human | 15658 | |
| MTOR (FRAP) | PIKK | Atypical | 7uxc | A | | - | Human | 14525 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsv | A | | adenosine-5'-diphosphate | Human | 9109 | |
| MTOR (FRAP) | PIKK | Atypical | 6sb2 | B | | - | Human | 11726 | |
| MTOR (FRAP) | PIKK | Atypical | 7peb | A | | - | Human | 13869 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsx | B | | 9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-one | Human | 9111 | |
| MTOR (FRAP) | PIKK | Atypical | 9f45 | A | | - | Human | 15315 | |
| MTOR (FRAP) | PIKK | Atypical | 5h64 | a | | - | Human | 9110 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k1n | A | | - | Human | 13210 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 5luq | A | | - | Human | 9321 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k1k | A | | - | Human | 13211 | |
| TRRAP | PIKK | Atypical | 8h7g | A | | - | Human | 14556 | |
| TRRAP | PIKK | Atypical | 8xvg | A | A | adenosine-5'-diphosphate | Human | 15321 | |
| TRRAP | PIKK | Atypical | 8qri | A | | - | Human | 15322 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7nfe | A | | - | Human | 13851 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7otw | A | | 7-methyl-2-[(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(oxan-4-yl)purin-8-one | Human | 14056 | |
| ATR | PIKK | Atypical | 23ey | A | | elimusertib | Human | 15645 | |
| ATR | PIKK | Atypical | 9l40 | A | | ve-822 | Human | 15646 | |
| ATR | PIKK | Atypical | 23fa | A | | gartisertib | Human | 15647 | |
| ATR | PIKK | Atypical | 23ex | A | | ceralasertib | Human | 15648 | |
| ATR | PIKK | Atypical | 5yz0 | A | | - | Human | 9523 | |
| ATR | PIKK | Atypical | 9l45 | A | | ve-822 | Human | 15649 | |
| ATR | PIKK | Atypical | 23ew | A | | ve-822 | Human | 15650 | |
| ATR | PIKK | Atypical | 13de | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15651 | |
| ATR | PIKK | Atypical | 9zd4 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15652 | |
| ATR | PIKK | Atypical | 23fb | A | | phosphothiophosphoric acid-adenylate ester | Human | 15659 | |
| ATR | PIKK | Atypical | 9l4f | A | | phosphothiophosphoric acid-adenylate ester | Human | 15660 | |
| ATR | PIKK | Atypical | 9l46 | A | | phosphothiophosphoric acid-adenylate ester | Human | 15661 | |
| MTOR (FRAP) | PIKK | Atypical | 9t94 | A | | adenosine-5'-triphosphate | Human | 15763 | |
| MTOR (FRAP) | PIKK | Atypical | 9ed8 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15764 | |
| MTOR (FRAP) | PIKK | Atypical | 7pe8 | A | | - | Human | 13870 | |
| MTOR (FRAP) | PIKK | Atypical | 9f44 | A | | - | Human | 15316 | |
| MTOR (FRAP) | PIKK | Atypical | 6sb0 | A | | - | Human | 11727 | |
| MTOR (FRAP) | PIKK | Atypical | 3jbz | A | | adenosine-5'-diphosphate | Human | 9113 | |
| MTOR (FRAP) | PIKK | Atypical | 7pe9 | A | | - | Human | 13871 | |
| MTOR (FRAP) | PIKK | Atypical | 4jt5 | A | | 2-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-1h-indol-5-ol | Human | 9116 | |
| MTOR (FRAP) | PIKK | Atypical | 8era | A | | 1-[6-{[(3m)-4-amino-3-(2-amino-1,3-benzoxazol-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-3,4-dihydroisoquinolin-2(1h)-yl]-3-hydroxypropan-1-one | Human | 14569 | |
| MTOR (FRAP) | PIKK | Atypical | 6zwo | B | | phosphothiophosphoric acid-adenylate ester | Human | 12987 | |
| MTOR (FRAP) | PIKK | Atypical | 7pe7 | A | | - | Human | 13901 | |
| MTOR (FRAP) | PIKK | Atypical | 4jt6 | B | | 3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenol | Human | 9102 | |
| MTOR (FRAP) | PIKK | Atypical | 5h64 | A | | - | Human | 9099 | |
| MTOR (FRAP) | PIKK | Atypical | 6sb2 | A | | - | Human | 11724 | |
| MTOR (FRAP) | PIKK | Atypical | 5flc | B | B | - | Human | 9108 | |
| MTOR (FRAP) | PIKK | Atypical | 6sb0 | B | | - | Human | 11725 | |
| MTOR (FRAP) | PIKK | Atypical | 5wbu | A | | - | Human | 9407 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsv | B | | adenosine-5'-diphosphate | Human | 9100 | |
| MTOR (FRAP) | PIKK | Atypical | 4jt6 | A | | 3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenol | Human | 9103 | |
| MTOR (FRAP) | PIKK | Atypical | 5zcs | A | | - | Human | 9748 | |
| MTOR (FRAP) | PIKK | Atypical | 6zwm | B | | phosphothiophosphoric acid-adenylate ester | Human | 12988 | |
| MTOR (FRAP) | PIKK | Atypical | 5wby | B | | - | Human | 9406 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsp | B | | phosphothiophosphoric acid-adenylate ester | Human | 9107 | |
| MTOR (FRAP) | PIKK | Atypical | 4jt5 | B | | 2-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-1h-indol-5-ol | Human | 9104 | |
| MTOR (FRAP) | PIKK | Atypical | 6zwm | A | | phosphothiophosphoric acid-adenylate ester | Human | 12989 | |
| MTOR (FRAP) | PIKK | Atypical | 5flc | F | B | - | Human | 9117 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsx | A | | 9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-one | Human | 9112 | |
| MTOR (FRAP) | PIKK | Atypical | 5wby | A | | - | Human | 9404 | |
| MTOR (FRAP) | PIKK | Atypical | 7pec | A | | - | Human | 13872 | |
| MTOR (FRAP) | PIKK | Atypical | 5flc | B | A | - | Human | 9105 | |
| MTOR (FRAP) | PIKK | Atypical | 7pea | A | | - | Human | 13873 | |
| MTOR (FRAP) | PIKK | Atypical | 5wbu | B | | - | Human | 9405 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsn | B | | - | Human | 9115 | |
| MTOR (FRAP) | PIKK | Atypical | 4jsn | A | | - | Human | 9114 | |
| MTOR (FRAP) | PIKK | Atypical | 7tzo | A | | - | Human | 14575 | |
| MTOR (FRAP) | PIKK | Atypical | 5flc | F | A | - | Human | 9101 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 5w1r | A | | - | Human | 9320 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7otp | A | | phosphothiophosphoric acid-adenylate ester | Human | 14054 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zh8 | A | | - | Human | 12925 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 8bh3 | A | | - | Human | 14768 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k1j | A | | - | Human | 13209 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zfp | A | | - | Human | 12926 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k0y | A | A | - | Human | 13213 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 8bhv | A | | - | Human | 14769 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 9qcs | A | | - | Human | 16044 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k0y | A | B | - | Human | 13214 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k17 | A | | - | Human | 13215 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7lt3 | C | | adenosine-5'-diphosphate | Human | 13500 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7lt3 | L | | adenosine-5'-diphosphate | Human | 13501 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 9zp0 | K | | - | Human | 16045 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 8rd4 | A | | - | Human | 16046 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zh4 | A | | - | Human | 12930 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k19 | A | | - | Human | 13216 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 9g9l | A | | - | Human | 16047 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k10 | A | | - | Human | 13217 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 9q9f | E | | - | Human | 16048 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 8bhy | A | | - | Human | 14770 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7k1b | A | | - | Human | 13218 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 7tyr | A | A | - | Human | 14322 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 6zhe | F | | - | Human | 12932 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 5y3r | C | | - | Human | 9318 | |
| ANTXR1 (DNAPK) | PIKK | Atypical | 9zp9 | M | | - | Human | 16049 | |
| ATM | PIKK | Atypical | 5np1 | A | | - | Human | 9268 | |
| ATM | PIKK | Atypical | 7sid | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14102 | |