Search results (62 entries covering 30 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PRKCB (PKCb)PKCAGC2i0eA3-{1-[3-(dimethylamino)propyl]-2-methyl-1h-indol-3-yl}-4-(2-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2550
PRKCB (PKCb)PKCAGC2i0eB3-{1-[3-(dimethylamino)propyl]-2-methyl-1h-indol-3-yl}-4-(2-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2549
PRKCI (PKCi)PKCAGC5li9ABphosphomethylphosphonic acid adenylate esterHuman7074
PRKCA (PKCa)PKCAGC8u37AA(6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamideHuman15159
PRKCA (PKCa)PKCAGC4ra4A(1r)-9-[(3s,4s)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman3040
PRKCA (PKCa)PKCAGC3iw4C3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dioneHuman3042
PRKCA (PKCa)PKCAGC8uakAA(6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamideHuman15161
PRKCA (PKCa)PKCAGC3iw4A3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dioneHuman3041
PRKCA (PKCa)PKCAGC3iw4B3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dioneHuman3039
PRKCB (PKCb)PKCAGC8se4A-Human16137
PRKCB (PKCb)PKCAGC8se3A-Human16138
PRKCB (PKCb)PKCAGC8se1Aphosphoaminophosphonic acid-adenylate esterHuman16139
PRKCH (PKCh)PKCAGC8fp3AB(3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrileHuman14695
PRKCH (PKCh)PKCAGC8fp3AA(3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrileHuman14696
PRKCA (PKCa)PKCAGC8u37AB(6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamideHuman15162
PRKCA (PKCa)PKCAGC8uakAB(6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamideHuman15160
PRKCI (PKCi)PKCAGC9ejkB-Human15444
PRKCI (PKCi)PKCAGC8r3xAB-Human15445
PRKCI (PKCi)PKCAGC9ejmBadenosine-5'-diphosphateHuman15446
PRKCI (PKCi)PKCAGC9ejlB-Human15447
PRKCI (PKCi)PKCAGC8r3xAA-Human15448
PRKCI (PKCi)PKCAGC5li9AAphosphomethylphosphonic acid adenylate esterHuman7068
PRKCB (PKCb)PKCAGC9s9tA(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHuman16135
PRKCB (PKCb)PKCAGC8se2A-Human16136
PRKCI (PKCi)PKCAGC5lihBBadenosine-5'-diphosphateHuman7073
PRKCI (PKCi)PKCAGC3a8xB-Human3348
PRKCI (PKCi)PKCAGC5li1ABphosphoaminophosphonic acid-adenylate esterHuman7067
PRKCH (PKCh)PKCAGC3txoA2-methyl-n~1~-[3-(pyridin-4-yl)-2,6-naphthyridin-1-yl]propane-1,2-diamineHuman2316
PRKCI (PKCi)PKCAGC3zh8BA(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3356
PRKCI (PKCi)PKCAGC3a8xA-Human3351
PRKCI (PKCi)PKCAGC3zh8AB(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3350
PRKCI (PKCi)PKCAGC3a8wAadenosine-5'-triphosphateHuman3353
PRKCI (PKCi)PKCAGC6ilzE2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamideHuman11356
PRKCQ (PKCt)PKCAGC2jedB3-(8-dimethylaminomethyl-6,7,8,9-tetrahydro-pyrido[1,2-a]indol-10-yl)-4-(1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman5358
PRKCQ (PKCt)PKCAGC5f9eBA2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHuman6631
PRKCQ (PKCt)PKCAGC5f9eBB2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHuman6628
PRKCQ (PKCt)PKCAGC5f9eAB2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHuman6629
PRKCQ (PKCt)PKCAGC4ra5BB(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5360
PRKCQ (PKCt)PKCAGC5f9eAA2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-oneHuman6630
PRKCI (PKCi)PKCAGC3zh8AA(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3349
PRKCI (PKCi)PKCAGC3zh8BB(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3347
PRKCI (PKCi)PKCAGC3zh8CB(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3352
PRKCI (PKCi)PKCAGC1zrzA3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman3354
PRKCI (PKCi)PKCAGC3a8wBadenosine-5'-triphosphateHuman3346
PRKCI (PKCi)PKCAGC5lihABadenosine-5'-diphosphateHuman7070
PRKCI (PKCi)PKCAGC6ilzA2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamideHuman11358
PRKCI (PKCi)PKCAGC5lihAAadenosine-5'-diphosphateHuman7071
PRKCI (PKCi)PKCAGC3zh8CA(2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamineHuman3355
PRKCI (PKCi)PKCAGC6ilzG2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamideHuman11355
PRKCI (PKCi)PKCAGC6ilzC2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamideHuman11357
PRKCI (PKCi)PKCAGC5li1AAphosphoaminophosphonic acid-adenylate esterHuman7072
PRKCI (PKCi)PKCAGC5lihBAadenosine-5'-diphosphateHuman7069
PRKCH (PKCh)PKCAGC8fp1A(3p)-3-[6-chloro-4-(9-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrileHuman14694
PRKCQ (PKCt)PKCAGC1xjdAstaurosporineHuman5357
PRKCQ (PKCt)PKCAGC4q9zBB(1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5362
PRKCQ (PKCt)PKCAGC4ra5AB(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5359
PRKCQ (PKCt)PKCAGC4ra5BA(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5361
PRKCQ (PKCt)PKCAGC4q9zAA(1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5356
PRKCQ (PKCt)PKCAGC2jedA3-(8-dimethylaminomethyl-6,7,8,9-tetrahydro-pyrido[1,2-a]indol-10-yl)-4-(1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman5352
PRKCQ (PKCt)PKCAGC4ra5AA(1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5354
PRKCQ (PKCt)PKCAGC4q9zBA(1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5355
PRKCQ (PKCt)PKCAGC4q9zAB(1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-oneHuman5353