Search results (38 entries covering 12 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
EIF2AK4-b (GCN2-b)STE-UniqueSTE9yakA-Human16226
MAP3K14 (NIK)STE-UniqueSTE6z1qBBdesf-3r/4076Human12449
MAP3K14 (NIK)STE-UniqueSTE6wppAB5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amineHuman12736
MAP3K14 (NIK)STE-UniqueSTE4idtAB11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amineHuman2204
MAP3K14 (NIK)STE-UniqueSTE4dn5Aphosphothiophosphoric acid-adenylate esterHuman2205
MAP3K14 (NIK)STE-UniqueSTE6z1tAA4s/3694Human12450
MAP3K14 (NIK)STE-UniqueSTE6wppAA5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amineHuman12737
MAP3K14 (NIK)STE-UniqueSTE4idtBA11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amineHuman2210
MAP3K14 (NIK)STE-UniqueSTE4idtBB11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amineHuman2207
MAP3K14 (NIK)STE-UniqueSTE8yhwAphosphothiophosphoric acid-adenylate esterHuman15233
MAP3K14 (NIK)STE-UniqueSTE4g3dD-Human2212
MAP3K14 (NIK)STE-UniqueSTE6z1tBB4s/3694Human12452
MAP3K14 (NIK)STE-UniqueSTE6wppBA5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amineHuman12738
MAP3K14 (NIK)STE-UniqueSTE4idvAA4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-olHuman2211
MAP3K14 (NIK)STE-UniqueSTE4idvCA4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-olHuman2201
MAP3K14 (NIK)STE-UniqueSTE4dn5Bphosphothiophosphoric acid-adenylate esterHuman2202
MAP3K14 (NIK)STE-UniqueSTE4g3dA-Human2208
MAP3K14 (NIK)STE-UniqueSTE4g3dE-Human2214
MAP3K14 (NIK)STE-UniqueSTE6z1tBA4s/3694Human12453
MAP3K14 (NIK)STE-UniqueSTE4idvBA4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-olHuman2206
MAP3K14 (NIK)STE-UniqueSTE6z1qABdesf-3r/4076Human12454
MAP3K14 (NIK)STE-UniqueSTE6wppBB5-fluoro-n-methyl-2-(7h-pyrrolo[2,3-d]pyrimidin-5-yl)pyrimidin-4-amineHuman12739
MAP3K14 (NIK)STE-UniqueSTE4idtAA11-bromo-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-2-amineHuman2203
MAP3K14 (NIK)STE-UniqueSTE4g3dB-Human2209
MAP3K14 (NIK)STE-UniqueSTE6z1qBAdesf-3r/4076Human12455
MAP3K14 (NIK)STE-UniqueSTE4idvDA4-{3-[2-amino-5-(2-methoxyethoxy)pyrimidin-4-yl]-1h-indol-5-yl}-2-methylbut-3-yn-2-olHuman2213
MAP3K14 (NIK)STE-UniqueSTE6z1tAB4s/3694Human12456
MAP3K8 (COT)STE-UniqueSTE4y85A5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amineHuman427
MAP3K8 (COT)STE-UniqueSTE4y85C5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amineHuman424
MAP3K8 (COT)STE-UniqueSTE5iu2AAn-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amineHuman6980
MAP3K8 (COT)STE-UniqueSTE4y83A5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman428
MAP3K8 (COT)STE-UniqueSTE4y83B5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman426
MAP3K8 (COT)STE-UniqueSTE5iu2BBn-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amineHuman6978
MAP3K8 (COT)STE-UniqueSTE5iu2ABn-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amineHuman6981
MAP3K8 (COT)STE-UniqueSTE4y85B5-[5-(1h-indol-3-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-1,3,4-oxadiazol-2-amineHuman429
MAP3K8 (COT)STE-UniqueSTE5iu2BAn-[2-(morpholin-4-yl)ethyl]-6-(8-phenyl-1h-imidazo[4,5-c][1,7]naphthyridin-1-yl)-1,3-benzothiazol-2-amineHuman6979
MAP3K8 (COT)STE-UniqueSTE4y83C5-[2-amino-5-(quinolin-3-yl)pyridin-3-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman425
MAP3K14 (NIK)STE-UniqueSTE6z1qAAdesf-3r/4076Human12451