| ACVR1 (ALK2) | STKR | TKL | 8c7z | A | A | 9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1]benzoxepino[5,4-c]pyridine | Human | 14605 | |
| ACVR1 (ALK2) | STKR | TKL | 6acr | B | | n-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amine | Human | 10968 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7m | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13666 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7q | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13670 | |
| ACVR1 (ALK2) | STKR | TKL | 6t8n | A | B | cyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanone | Human | 11830 | |
| BMPR1B | STKR | TKL | 3mdy | C | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1500 | |
| BMPR1B | STKR | TKL | 3mdy | C | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1503 | |
| BMPR1B | STKR | TKL | 3mdy | A | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1502 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | C | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1269 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | S | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1259 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | R | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1256 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | L | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1265 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | T | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1264 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | A | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1266 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | O | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1262 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | M | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1268 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | V | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1271 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | E | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1263 | |
| ACVR1 (ALK2) | STKR | TKL | 5s84 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13734 | |
| ACVR1 (ALK2) | STKR | TKL | 5s84 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13656 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7l | A | C | - | Human | 13665 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7l | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13676 | |
| ACVR1 (ALK2) | STKR | TKL | 5s78 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13716 | |
| ACVR1 (ALK2) | STKR | TKL | 5s84 | A | C | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13722 | |
| ACVR1 (ALK2) | STKR | TKL | 5s8b | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13726 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7l | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13736 | |
| ACVR1 (ALK2) | STKR | TKL | 5s8b | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13721 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7d | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13668 | |
| ACVR1 (ALK2) | STKR | TKL | 5s89 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13688 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | D | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1258 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | H | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1260 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2j | A | B | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2115 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | E | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2097 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | C | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2104 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3tzm | A | A | 4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamide | Human | 2095 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2j | A | A | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2124 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | B | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1273 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3tzm | A | B | 4-[5-(1,3-benzodioxol-5-yl)-4-(pyridin-2-yl)-1h-imidazol-2-yl]benzamide | Human | 2110 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2g | A | B | 4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2114 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8u | A | | - | Human | 6616 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7r | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13731 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8s | A | B | - | Human | 6609 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8t | A | A | - | Human | 6608 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qu0 | A | A | 6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrile | Human | 11967 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | E | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2098 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | B | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2106 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | D | | - | Human | 2126 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8w | A | A | staurosporine | Human | 6611 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e90 | A | B | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6607 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | X | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1275 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e90 | A | A | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6610 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1rw8 | A | | 3-(4-fluorophenyl)-2-(6-methylpyridin-2-yl)-5,6-dihydro-4h-pyrrolo[1,2-b]pyrazole | Human | 2100 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | C | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2093 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 6b8y | A | A | n-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9553 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5fri | A | B | n-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamide | Human | 6893 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8z | A | A | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6618 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qu0 | A | B | 6-[4-(3-chloro-4-fluorophenyl)-1-(2-hydroxyethyl)-1h-imidazol-5-yl]imidazo[1,2-b]pyridazine-3-carbonitrile | Human | 11964 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | C | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2130 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | A | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2127 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qik | A | A | n-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10657 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2k | A | A | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2135 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qim | A | A | n-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10658 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | D | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2119 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | D | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2132 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2g | A | A | 4-[(4-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2123 | |
| ACVR1 (ALK2) | STKR | TKL | 9l04 | A | | 4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-[4-[4-(oxetan-3-yl)piperazin-1-yl]phenyl]pyrimidin-2-amine | Human | 15732 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 8ygz | A | A | - | Human | 15262 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 8ygz | A | B | - | Human | 15263 | |
| ACVR2A (ACTR2) | STKR | TKL | 3soc | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2676 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | P | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1270 | |
| ACVR1 (ALK2) | STKR | TKL | 6t8n | B | A | cyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanone | Human | 11828 | |
| ACVR1 (ALK2) | STKR | TKL | 8r7g | A | B | 2-fluoranyl-6-methoxy-4-[4-methyl-5-[4-(4-propan-2-ylpiperazin-1-yl)phenyl]pyridin-3-yl]benzamide | Human | 15266 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | F | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1276 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | G | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1272 | |
| ACVR1 (ALK2) | STKR | TKL | 5s79 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13708 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7t | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13709 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7i | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13699 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7c | A | C | - | Human | 13702 | |
| BMPR1B | STKR | TKL | 3mdy | A | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1501 | |
| ACVR2B (ACTR2B) | STKR | TKL | 2qlu | A | | adenine | Human | 2940 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e8v | A | B | - | Human | 6622 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7c | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13690 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8x | A | B | staurosporine | Human | 6617 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qil | A | A | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10659 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | D | | - | Human | 2131 | |
| ACVR1 (ALK2) | STKR | TKL | 7a21 | A | B | 4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12779 | |
| ACVR1 (ALK2) | STKR | TKL | 5s88 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13657 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7e | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13643 | |
| ACVR1 (ALK2) | STKR | TKL | 3mtf | B | B | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 1530 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7a | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13644 | |
| ACVR1 (ALK2) | STKR | TKL | 6t8n | A | A | cyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanone | Human | 11831 | |
| ACVR1 (ALK2) | STKR | TKL | 5s9k | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13645 | |
| ACVR1 (ALK2) | STKR | TKL | 7a21 | B | A | 4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12776 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7s | A | C | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13651 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7z | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13652 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | B | B | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8519 | |
| ACVR1 (ALK2) | STKR | TKL | 5s80 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13669 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | A | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1528 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7x | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13692 | |
| ACVR1 (ALK2) | STKR | TKL | 5s8a | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13693 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | D | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11785 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | C | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1522 | |
| ACVR1 (ALK2) | STKR | TKL | 6i1s | A | A | (4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione | Human | 11603 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7m | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13739 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | F | | - | Human | 2103 | |
| BMPR2 | STKR | TKL | 3g2f | B | A | adenosine-5'-diphosphate | Human | 6867 | |
| BMPR2 | STKR | TKL | 3g2f | A | B | adenosine-5'-diphosphate | Human | 6868 | |
| BMPR2 | STKR | TKL | 3g2f | B | B | adenosine-5'-diphosphate | Human | 6869 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wou | A | | 4-({4-[(2,6-dimethylpyridin-3-yl)oxy]pyridin-2-yl}amino)benzenesulfonamide | Human | 2125 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | E | | - | Human | 2134 | |
| BMPR2 | STKR | TKL | 6unp | A | B | adenosine-5'-diphosphate | Human | 13794 | |
| BMPR2 | STKR | TKL | 6unp | A | A | adenosine-5'-diphosphate | Human | 13795 | |
| BMPR2 | STKR | TKL | 3g2f | A | A | adenosine-5'-diphosphate | Human | 6870 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | I | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1261 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | Q | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1274 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | N | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1257 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | J | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1277 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | U | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1278 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | W | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1255 | |
| ACVRL1 (ALK1) | STKR | TKL | 3my0 | K | | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1267 | |
| ACVR1 (ALK2) | STKR | TKL | 7c3g | A | A | ~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amine | Human | 13389 | |
| ACVR1 (ALK2) | STKR | TKL | 6zgc | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 12638 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7x | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13646 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | B | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1510 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7o | A | C | - | Human | 13647 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7j | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13648 | |
| ACVR1 (ALK2) | STKR | TKL | 7c3g | A | B | ~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amine | Human | 13390 | |
| ACVR1 (ALK2) | STKR | TKL | 6srh | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 11630 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7k | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13649 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | C | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1533 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | A | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1508 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7b | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13650 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | B | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1514 | |
| ACVR1 (ALK2) | STKR | TKL | 6zgc | D | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 12639 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7i | A | C | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13653 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7r | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13654 | |
| ACVR1 (ALK2) | STKR | TKL | 6uns | A | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 13781 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7n | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13655 | |
| ACVR1 (ALK2) | STKR | TKL | 6jux | A | B | 4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amine | Human | 12160 | |
| ACVR1 (ALK2) | STKR | TKL | 3h9r | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 1531 | |
| ACVR1 (ALK2) | STKR | TKL | 6uns | A | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 13782 | |
| ACVR1 (ALK2) | STKR | TKL | 5oy6 | D | | cyclical inhibitor od36 | Human | 8534 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | C | A | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8517 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | C | B | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8513 | |
| ACVR1 (ALK2) | STKR | TKL | 7a21 | A | A | 4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12777 | |
| ACVR1 (ALK2) | STKR | TKL | 6tn8 | A | A | 4-[4-[(dimethylamino)methyl]-2,5-dimethoxy-phenyl]-2-methyl-2,7-naphthyridin-1-one | Human | 11888 | |
| ACVR1 (ALK2) | STKR | TKL | 6zgc | C | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 12640 | |
| ACVR1 (ALK2) | STKR | TKL | 6i1s | A | B | (4~{s},5~{r},6~{z},9~{s},10~{s},12~{e})-16-(ethylamino)-4,5-dimethyl-9,10,18-tris(oxidanyl)-3-oxabicyclo[12.4.0]octadeca-1(14),6,12,15,17-pentaene-2,8-dione | Human | 11604 | |
| ACVR1 (ALK2) | STKR | TKL | 6gin | B | B | 3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-one | Human | 9916 | |
| ACVR1 (ALK2) | STKR | TKL | 5s9k | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13658 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7n | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13659 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | D | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1529 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7h | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13660 | |
| ACVR1 (ALK2) | STKR | TKL | 5s81 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13661 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7w | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13662 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7i | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13663 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7o | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13664 | |
| ACVR1 (ALK2) | STKR | TKL | 6srh | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 11632 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | A | A | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11735 | |
| ACVR1 (ALK2) | STKR | TKL | 3mtf | A | B | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 1521 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | B | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1523 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7s | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13667 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | B | B | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12275 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7w | A | A | 6-methyl-9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,7-dihydropyrido[4,3-d][2]benzazepine | Human | 14608 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | A | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1527 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | D | A | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8520 | |
| ACVR1 (ALK2) | STKR | TKL | 6zgc | B | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 12641 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7z | A | B | 9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,6-dihydro-[1]benzoxepino[5,4-c]pyridine | Human | 14604 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7f | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13671 | |
| ACVR1 (ALK2) | STKR | TKL | 5s76 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13672 | |
| ACVR1 (ALK2) | STKR | TKL | 5s89 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13673 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7z | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13674 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7u | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13675 | |
| ACVR1 (ALK2) | STKR | TKL | 4c02 | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 1532 | |
| ACVR1 (ALK2) | STKR | TKL | 8c7w | A | B | 6-methyl-9-piperazin-1-yl-4-(3,4,5-trimethoxyphenyl)-5,7-dihydropyrido[4,3-d][2]benzazepine | Human | 14609 | |
| ACVR1 (ALK2) | STKR | TKL | 5oy6 | A | | cyclical inhibitor od36 | Human | 8532 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7s | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13677 | |
| ACVR1 (ALK2) | STKR | TKL | 6t8n | B | B | cyclopropyl-[4-[6-[5-(4-ethoxy-1-propan-2-yl-piperidin-4-yl)pyridin-2-yl]pyrrolo[1,2-b]pyridazin-4-yl]piperazin-1-yl]methanone | Human | 11829 | |
| ACVR1 (ALK2) | STKR | TKL | 6gin | B | A | 3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-one | Human | 9920 | |
| ACVR1 (ALK2) | STKR | TKL | 6eix | A | A | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 8530 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7q | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13678 | |
| ACVR1 (ALK2) | STKR | TKL | 6tn8 | A | B | 4-[4-[(dimethylamino)methyl]-2,5-dimethoxy-phenyl]-2-methyl-2,7-naphthyridin-1-one | Human | 11887 | |
| ACVR1 (ALK2) | STKR | TKL | 5s85 | A | C | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13679 | |
| ACVR1 (ALK2) | STKR | TKL | 7a21 | B | B | 4-methyl-3-[4-(pyrrolidin-1-ylmethyl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12778 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7c | A | D | - | Human | 13680 | |
| ACVR1 (ALK2) | STKR | TKL | 5s82 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13681 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7h | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13682 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7a | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13683 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7y | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13684 | |
| ACVR1 (ALK2) | STKR | TKL | 3mtf | B | A | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 1515 | |
| ACVR1 (ALK2) | STKR | TKL | 4c02 | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 1525 | |
| ACVR1 (ALK2) | STKR | TKL | 5s83 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13685 | |
| ACVR1 (ALK2) | STKR | TKL | 5s78 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13686 | |
| ACVR1 (ALK2) | STKR | TKL | 7nns | B | B | momelotinib | Human | 13464 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7p | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13687 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | B | A | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11734 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7c | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13689 | |
| ACVR1 (ALK2) | STKR | TKL | 6gip | A | A | 2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-one | Human | 9915 | |
| ACVR1 (ALK2) | STKR | TKL | 4dym | A | | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 1509 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | A | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11779 | |
| ACVR1 (ALK2) | STKR | TKL | 6acr | A | | n-(4-methoxyphenyl)-4-[3-(pyridin-3-yl)-1h-pyrazol-4-yl]pyrimidin-2-amine | Human | 10969 | |
| ACVR1 (ALK2) | STKR | TKL | 5s76 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13691 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | D | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11783 | |
| ACVR1 (ALK2) | STKR | TKL | 6gin | A | B | 3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-one | Human | 9918 | |
| ACVR1 (ALK2) | STKR | TKL | 6gip | A | B | 2,5-dimethyl-6-quinolin-4-yl-3~{h}-quinazolin-4-one | Human | 9917 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | B | A | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12276 | |
| ACVR1 (ALK2) | STKR | TKL | 5s77 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13694 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7p | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13695 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7u | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13696 | |
| ACVR1 (ALK2) | STKR | TKL | 5s81 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13697 | |
| ACVR1 (ALK2) | STKR | TKL | 7nns | B | A | momelotinib | Human | 13465 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | B | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1526 | |
| ACVR1 (ALK2) | STKR | TKL | 6srh | B | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 11631 | |
| ACVR1 (ALK2) | STKR | TKL | 5s77 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13698 | |
| ACVR1 (ALK2) | STKR | TKL | 6eix | A | B | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 8533 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7w | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13700 | |
| ACVR1 (ALK2) | STKR | TKL | 5s82 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13701 | |
| ACVR1 (ALK2) | STKR | TKL | 7c3g | B | B | ~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amine | Human | 13391 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | B | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11782 | |
| ACVR1 (ALK2) | STKR | TKL | 8pod | A | | 6-(4-piperazin-1-ylphenyl)-3-quinolin-4-yl-furo[3,2-b]pyridine | Human | 15314 | |
| ACVR1 (ALK2) | STKR | TKL | 7c3g | B | A | ~{n}-[4-(4-methylpiperazin-1-yl)phenyl]-4-(2-pyridin-3-yl-6,7-dihydro-4~{h}-pyrazolo[5,1-c][1,4]oxazin-3-yl)pyrimidin-2-amine | Human | 13392 | |
| ACVR1 (ALK2) | STKR | TKL | 5s88 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13703 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | B | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11781 | |
| ACVR1 (ALK2) | STKR | TKL | 5s79 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13704 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7m | A | C | - | Human | 13705 | |
| ACVR1 (ALK2) | STKR | TKL | 5s83 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13706 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | B | A | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8516 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7v | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13707 | |
| ACVR1 (ALK2) | STKR | TKL | 6unq | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 13783 | |
| ACVR1 (ALK2) | STKR | TKL | 5s85 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13710 | |
| ACVR1 (ALK2) | STKR | TKL | 5oy6 | C | | cyclical inhibitor od36 | Human | 8529 | |
| ACVR1 (ALK2) | STKR | TKL | 3oom | A | A | 1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanone | Human | 1517 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | A | B | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8518 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7v | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13711 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7j | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13712 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7g | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13713 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | D | B | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1512 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | C | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1516 | |
| ACVR1 (ALK2) | STKR | TKL | 6unq | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 13784 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | C | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11780 | |
| ACVR1 (ALK2) | STKR | TKL | 6unr | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13785 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7e | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13715 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7g | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13717 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | A | A | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12277 | |
| ACVR1 (ALK2) | STKR | TKL | 5s75 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13718 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7b | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13719 | |
| ACVR1 (ALK2) | STKR | TKL | 3mtf | A | A | 3-[6-amino-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenol | Human | 1513 | |
| ACVR1 (ALK2) | STKR | TKL | 8r7g | A | A | 2-fluoranyl-6-methoxy-4-[4-methyl-5-[4-(4-propan-2-ylpiperazin-1-yl)phenyl]pyridin-3-yl]benzamide | Human | 15267 | |
| ACVR1 (ALK2) | STKR | TKL | 5s85 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13720 | |
| ACVR1 (ALK2) | STKR | TKL | 6gi6 | A | | 5-methyl-6-quinolin-5-yl-3~{h}-quinazolin-4-one | Human | 9919 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | D | B | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8515 | |
| ACVR1 (ALK2) | STKR | TKL | 3oom | A | B | 1-{3-[6-(tetrahydro-2h-pyran-4-ylamino)imidazo[1,2-b]pyridazin-3-yl]phenyl}ethanone | Human | 1518 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7t | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13723 | |
| ACVR1 (ALK2) | STKR | TKL | 5s86 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13724 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | A | B | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1524 | |
| ACVR1 (ALK2) | STKR | TKL | 5s8a | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13725 | |
| ACVR1 (ALK2) | STKR | TKL | 5oxg | A | A | 5-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 8514 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7y | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13727 | |
| ACVR1 (ALK2) | STKR | TKL | 5s80 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13728 | |
| ACVR1 (ALK2) | STKR | TKL | 3q4u | D | A | 4-[6-(4-piperazin-1-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinoline | Human | 1520 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | A | B | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11784 | |
| ACVR1 (ALK2) | STKR | TKL | 5s86 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13729 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7d | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13730 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | A | B | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11737 | |
| ACVR1 (ALK2) | STKR | TKL | 6szm | B | B | 1-[4-[4-methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl]piperazine | Human | 11736 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7k | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13732 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7o | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13733 | |
| ACVR1 (ALK2) | STKR | TKL | 6srh | B | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 11633 | |
| ACVR1 (ALK2) | STKR | TKL | 6gin | A | A | 3-(4-morpholin-4-ylphenyl)-6-quinolin-4-yl-quinazolin-4-one | Human | 9914 | |
| ACVR1 (ALK2) | STKR | TKL | 5s7f | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13737 | |
| ACVR1 (ALK2) | STKR | TKL | 6z36 | A | B | 4-methyl-3-(4-piperidin-4-ylphenyl)-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 12278 | |
| ACVR1 (ALK2) | STKR | TKL | 5s87 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13738 | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | A | B | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | 2681 | |
| ACVR2A (ACTR2) | STKR | TKL | 3q4t | B | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 2680 | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | A | A | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | 2678 | |
| ACVR2A (ACTR2) | STKR | TKL | 3soc | B | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2677 | |
| ACVR2A (ACTR2) | STKR | TKL | 3soc | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2675 | |
| ACVR2A (ACTR2) | STKR | TKL | 3q4t | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 2686 | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | B | A | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | 2683 | |
| ACVR2A (ACTR2) | STKR | TKL | 3q4t | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 2682 | |
| ACVR2A (ACTR2) | STKR | TKL | 3q4t | B | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 2684 | |
| ACVR2A (ACTR2) | STKR | TKL | 3soc | B | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2685 | |
| ACVR2A (ACTR2) | STKR | TKL | 4asx | B | B | 7,8-bis(chloranyl)-9-methyl-3,4-dihydro-2h-pyrido[3,4-b]indol-1-one | Human | 2679 | |
| ACVR1 (ALK2) | STKR | TKL | 6t6d | C | A | 2-methoxy-4-[4-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]benzamide | Human | 11778 | |
| ACVR1 (ALK2) | STKR | TKL | 5s75 | A | A | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13714 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | C | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1511 | |
| ACVR1 (ALK2) | STKR | TKL | 5oy6 | B | | cyclical inhibitor od36 | Human | 8531 | |
| ACVR1 (ALK2) | STKR | TKL | 4bgg | D | A | 1-{4-[5-(3,4,5-trimethoxyphenyl)pyridin-3-yl]phenyl}piperazine | Human | 1519 | |
| ACVR1 (ALK2) | STKR | TKL | 6jux | A | A | 4-(1-ethyl-3-pyridin-3-yl-pyrazol-4-yl)-~{n}-(4-piperazin-1-ylphenyl)pyrimidin-2-amine | Human | 12161 | |
| ACVR1 (ALK2) | STKR | TKL | 5s87 | A | B | 4-methyl-3-[4-(1-methylpiperidin-4-yl)phenyl]-5-(3,4,5-trimethoxyphenyl)pyridine | Human | 13735 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qik | A | B | n-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1h-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10662 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qim | A | B | n-{4-[3-(5-methoxypyridin-2-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10661 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | A | | - | Human | 2113 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5fri | A | A | n-[4-[(6-chloro-[1,3]dioxolo[4,5-b]pyridin-7-yl)amino]-2-pyridyl]cyclopropanecarboxamide | Human | 6894 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | D | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2107 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qtz | A | A | 6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridine | Human | 11965 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2f | A | B | 4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 6208 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1vjy | A | | 2-[5-(6-methylpyridin-2-yl)-2,3-dihydro-1h-pyrazol-4-yl]-1,5-naphthyridine | Human | 2096 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8s | A | A | - | Human | 6619 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5usq | A | A | n-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amine | Human | 7558 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qil | A | B | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10660 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x0m | A | B | 4-aminopyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2121 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2n | A | B | - | Human | 2109 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8z | A | B | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6612 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1py5 | A | | 4-(3-pyridin-2-yl-1h-pyrazol-4-yl)quinoline | Human | 2094 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3hmm | A | | 2-(6-methylpyridin-2-yl)-n-pyridin-4-ylquinazolin-4-amine | Human | 2111 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | C | | - | Human | 2117 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8t | A | B | - | Human | 6613 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wot | A | B | 4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amine | Human | 2092 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | B | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2108 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5usq | A | B | n-[2-(5-chloro-2-fluorophenyl)pyridin-4-yl]-2-[(piperidin-4-yl)methyl]-2h-pyrazolo[4,3-b]pyridin-7-amine | Human | 7557 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1ias | B | | - | Human | 2102 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3gxl | A | | n-1h-indazol-5-yl-2-(6-methylpyridin-2-yl)quinazolin-4-amine | Human | 2116 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2f | A | A | 4-amino-8-(4-aminophenyl)pyrido[2,3-d]pyrimidin-5(8h)-one | Human | 6207 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 6b8y | A | B | n-(3-fluoropyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-2-yl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9552 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | E | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2105 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2n | A | A | - | Human | 2129 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8w | A | B | staurosporine | Human | 6614 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3kcf | A | | 4-[3-(methoxymethyl)phenyl]-1,2-dimethyl-5-quinoxalin-6-yl-1,2-dihydro-3h-pyrazol-3-one | Human | 2112 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5qtz | A | B | 6-[1-(2,2-difluoroethyl)-4-(6-methylpyridin-2-yl)-1h-imidazol-5-yl]imidazo[1,2-a]pyridine | Human | 11966 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | B | | - | Human | 2133 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x0m | A | A | 4-aminopyrido[2,3-d]pyrimidin-5(8h)-one | Human | 2122 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 3faa | A | | n-[4-(5-fluoro-6-methylpyridin-2-yl)-5-quinoxalin-6-yl-1h-imidazol-2-yl]acetamide | Human | 2118 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2x7o | B | | (3z)-n-ethyl-n-methyl-2-oxo-3-(phenyl{[4-(piperidin-1-ylmethyl)phenyl]amino}methylidene)-2,3-dihydro-1h-indole-6-carboxamide | Human | 2128 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 4x2k | A | B | 4-[(3-aminophenyl)amino]pyrido[2,3-d]pyrimidin-5(6h)-one | Human | 2101 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 2wot | A | A | 4-[(5,6-dimethyl-2,2'-bipyridin-3-yl)oxy]-n-(3,4,5-trimethoxyphenyl)pyridin-2-amine | Human | 2120 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 9f6x | A | | 2-[5-(1,3-benzodioxol-5-yl)-2-~{tert}-butyl-1~{h}-imidazol-4-yl]-6-methyl-pyridine | Human | 16116 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 5e8x | A | A | staurosporine | Human | 6615 | |
| TGFBR1 (TGFbR1) | STKR | TKL | 1b6c | H | | - | Human | 2099 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e92 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 6623 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5qin | A | B | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10663 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e8v | A | A | - | Human | 6626 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e92 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 6624 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e8y | A | | staurosporine | Human | 6627 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5qin | A | A | n-{4-[3-(6-methoxypyridin-3-yl)-1h-pyrrolo[3,2-b]pyridin-2-yl]pyridin-2-yl}acetamide | Human | 10664 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 5e91 | A | | 3-amino-6-[4-(2-hydroxyethyl)phenyl]-n-[4-(morpholin-4-yl)pyridin-3-yl]pyrazine-2-carboxamide | Human | 6625 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 7dv6 | A | B | 5-[(3s)-5,5-dimethyloxolan-3-yl]-6-methoxy-3-(2-methoxypyridin-4-yl)pyrazolo[1,5-a]pyrimidine | Human | 13628 | |
| TGFBR2 (TGFbR2) | STKR | TKL | 7dv6 | A | A | 5-[(3s)-5,5-dimethyloxolan-3-yl]-6-methoxy-3-(2-methoxypyridin-4-yl)pyrazolo[1,5-a]pyrimidine | Human | 13629 | |
