| LCK | Src | TK | 6pdj | A | B | n-{4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]-3-methylphenyl}-1-methyl-1h-indazole-3-carboxamide | Human | 11699 | |
| LCK | Src | TK | 3kmm | A | | 3-(2,6-dichlorophenyl)-7-({4-[2-(diethylamino)ethoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 2265 | |
| HCK | Src | TK | 3vs3 | B | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2665 | |
| HCK | Src | TK | 3vrz | A | | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-benzylurea | Human | 2658 | |
| SRC | Src | TK | 6e6e | E | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11479 | |
| SRC | Src | TK | 6e6e | G | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11493 | |
| SRC | Src | TK | 2bdf | B | | {[(4-{[2-(4-aminocyclohexyl)-9-ethyl-9h-purin-6-yl]amino}phenyl)(hydroxy)phosphoryl]methyl}phosphonic acid | Human | 975 | |
| LYN | Src | TK | 5xy1 | A | | n-(1h-indazol-6-yl)-8-piperidin-4-yloxy-6-propyl-quinazolin-2-amine | Human | 8271 | |
| SRC | Src | TK | 7ng7 | A | | tert-butyl (4-(4-amino-1-(2-(4-(dimethylamino)piperidin-1-yl)ethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)carbamate | Human | 13900 | |
| HCK | Src | TK | 9byj | A | A | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 15592 | |
| HCK | Src | TK | 9byj | A | B | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 15593 | |
| SRC | Src | TK | 9ns1 | A | 17 | - | Human | 15594 | |
| SRC | Src | TK | 9ns0 | A | 15 | - | Human | 15598 | |
| SRC | Src | TK | 9ns1 | A | 12 | - | Human | 15595 | |
| SRC | Src | TK | 9ns1 | A | 1 | - | Human | 15599 | |
| SRC | Src | TK | 9ns1 | A | 10 | - | Human | 15600 | |
| SRC | Src | TK | 9ns0 | A | 2 | - | Human | 15601 | |
| SRC | Src | TK | 9ns1 | A | 13 | - | Human | 15602 | |
| SRC | Src | TK | 9ns1 | A | 11 | - | Human | 15596 | |
| SRC | Src | TK | 9ns0 | A | 20 | - | Human | 15597 | |
| SRC | Src | TK | 9ns0 | A | 1 | - | Human | 15603 | |
| SRC | Src | TK | 9ns1 | A | 15 | - | Human | 15604 | |
| SRC | Src | TK | 9ns1 | A | 6 | - | Human | 15605 | |
| SRC | Src | TK | 9ns0 | A | 8 | - | Human | 15606 | |
| SRC | Src | TK | 9ns1 | A | 2 | - | Human | 15607 | |
| SRC | Src | TK | 9ns0 | A | 3 | - | Human | 15608 | |
| SRC | Src | TK | 9ns0 | A | 18 | - | Human | 15609 | |
| SRC | Src | TK | 9ns0 | A | 5 | - | Human | 15610 | |
| SRC | Src | TK | 9ns0 | A | 13 | - | Human | 15611 | |
| SRC | Src | TK | 9ns0 | A | 16 | - | Human | 15624 | |
| HCK | Src | TK | 2hck | B | | 3,5,7,3',4'-pentahydroxyflavone | Human | 9482 | |
| SRC | Src | TK | 4mxo | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 978 | |
| FGR | Src | TK | 7uy0 | B | A | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14566 | |
| HCK | Src | TK | 5zj6 | A | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9987 | |
| FGR | Src | TK | 7uy0 | B | C | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14562 | |
| FGR | Src | TK | 7uy0 | A | C | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14564 | |
| FGR | Src | TK | 7uy3 | A | | 3-[(6,7-dimethoxyquinazolin-4-yl)oxy]-n-{4-[(4-ethylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}-4-methylbenzamide | Human | 14567 | |
| FGR | Src | TK | 7uy0 | A | A | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14568 | |
| SRC | Src | TK | 6ate | A | | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10920 | |
| FGR | Src | TK | 7uy0 | B | B | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14565 | |
| FGR | Src | TK | 7uy0 | A | B | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14563 | |
| LYN | Src | TK | 3a4o | X | | staurosporine | Human | 1812 | |
| SRC | Src | TK | 2bdf | A | | {[(4-{[2-(4-aminocyclohexyl)-9-ethyl-9h-purin-6-yl]amino}phenyl)(hydroxy)phosphoryl]methyl}phosphonic acid | Human | 980 | |
| SRC | Src | TK | 6e6e | E | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11478 | |
| SRC | Src | TK | 6e6e | H | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11475 | |
| HCK | Src | TK | 2c0t | A | A | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2653 | |
| HCK | Src | TK | 2c0t | B | A | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2642 | |
| HCK | Src | TK | 2c0o | A | A | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2666 | |
| HCK | Src | TK | 4lue | B | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2668 | |
| HCK | Src | TK | 5h09 | A | | ethyl (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-4-methyl-pentanoate | Human | 8537 | |
| HCK | Src | TK | 5h0h | A | | (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-~{n},~{n},4-trimethyl-pentanamide | Human | 8539 | |
| HCK | Src | TK | 2c0t | B | B | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2634 | |
| HCK | Src | TK | 2c0o | A | B | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2652 | |
| HCK | Src | TK | 2hk5 | A | | 3-{[2-(1h-benzimidazol-1-yl)-6-{[2-(diethylamino)ethyl]amino}pyrimidin-4-yl]amino}-4-methylphenol | Human | 2639 | |
| HCK | Src | TK | 3vs3 | A | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2643 | |
| HCK | Src | TK | 3vs6 | A | | tert-butyl {4-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl}carbamate | Human | 2664 | |
| HCK | Src | TK | 4lud | A | | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | 2660 | |
| HCK | Src | TK | 2c0i | A | B | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2649 | |
| SRC | Src | TK | 8jf3 | A | | 2-[4-[4-[bis(oxidanylidene)-$l^5-sulfanyl]oxyphenyl]carbonylpiperazin-1-yl]-6-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-n-prop-2-ynyl-pyrimidine-4-carboxamide | Human | 15226 | |
| SRC | Src | TK | 9ns0 | A | 6 | - | Human | 15613 | |
| SRC | Src | TK | 1yom | A | | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 973 | |
| SRC | Src | TK | 9irl | A | | (2~{r})-2-[3,5-bis(fluoranyl)phenyl]-2-[2-chloranylethanoyl(cyclopropyl)amino]-~{n}-cyclopentyl-ethanamide | Human | 15614 | |
| SRC | Src | TK | 6e6e | E | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11490 | |
| SRC | Src | TK | 9ns0 | A | 14 | - | Human | 15622 | |
| SRC | Src | TK | 9ns1 | A | 16 | - | Human | 15623 | |
| SRC | Src | TK | 8jn9 | A | | n-[(1r)-1-[3,5-bis(fluoranyl)phenyl]-2-(cyclopentylamino)-2-oxidanylidene-ethyl]-n-cyclopropyl-prop-2-enamide | Human | 15313 | |
| SRC | Src | TK | 9ns0 | A | 9 | - | Human | 15625 | |
| PTK6 (BRK) | Src | TK | 5h2u | C | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7342 | |
| PTK6 (BRK) | Src | TK | 5da3 | A | B | (2-chloro-4-{[6-cyclopropyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanone | Human | 6988 | |
| PTK6 (BRK) | Src | TK | 6cz2 | A | B | - | Human | 10031 | |
| PTK6 (BRK) | Src | TK | 5d7v | B | B | - | Human | 6951 | |
| PTK6 (BRK) | Src | TK | 5d7v | C | B | - | Human | 6954 | |
| PTK6 (BRK) | Src | TK | 6cz3 | A | A | (3-fluoro-4-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanone | Human | 10001 | |
| PTK6 (BRK) | Src | TK | 5da3 | A | A | (2-chloro-4-{[6-cyclopropyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanone | Human | 6989 | |
| PTK6 (BRK) | Src | TK | 6cz2 | A | A | - | Human | 10030 | |
| PTK6 (BRK) | Src | TK | 6cz4 | A | A | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamide | Human | 9998 | |
| PTK6 (BRK) | Src | TK | 5h2u | C | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7341 | |
| HCK | Src | TK | 5h0g | A | | (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-~{n},4-dimethyl-pentanamide | Human | 8536 | |
| LCK | Src | TK | 2pl0 | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 2290 | |
| HCK | Src | TK | 3vrz | B | | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-benzylurea | Human | 2661 | |
| SRC | Src | TK | 1yi6 | B | | - | Human | 991 | |
| PTK6 (BRK) | Src | TK | 5d7v | C | A | - | Human | 6949 | |
| PTK6 (BRK) | Src | TK | 5h2u | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7343 | |
| LCK | Src | TK | 3lck | A | B | - | Human | 2301 | |
| HCK | Src | TK | 2c0i | A | A | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2662 | |
| HCK | Src | TK | 3vs0 | A | | n-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]benzamide | Human | 2633 | |
| HCK | Src | TK | 3vs1 | B | | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-phenylurea | Human | 2636 | |
| HCK | Src | TK | 2c0o | B | A | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2663 | |
| HCK | Src | TK | 2hck | A | | 3,5,7,3',4'-pentahydroxyflavone | Human | 9481 | |
| HCK | Src | TK | 2c0i | B | A | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2650 | |
| HCK | Src | TK | 3vs4 | A | | 5-(4-phenoxyphenyl)-7-(tetrahydro-2h-pyran-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2654 | |
| HCK | Src | TK | 3vs0 | B | | n-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]benzamide | Human | 2644 | |
| HCK | Src | TK | 2c0i | B | B | n-(4-{4-amino-1-[4-(4-methylpiperazin-1-yl)-trans-cyclohexyl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2640 | |
| HCK | Src | TK | 3vs2 | B | | 7-[cis-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2632 | |
| HCK | Src | TK | 3vs5 | B | | 7-(1-methylpiperidin-4-yl)-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2669 | |
| HCK | Src | TK | 3vs2 | A | | 7-[cis-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2651 | |
| HCK | Src | TK | 2c0t | A | B | n-(4-{4-amino-1-[1-(tetrahydro-2h-pyran-4-yl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2667 | |
| HCK | Src | TK | 3vs6 | B | | tert-butyl {4-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-2-methoxyphenyl}carbamate | Human | 2656 | |
| HCK | Src | TK | 3vs7 | A | | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 2659 | |
| HCK | Src | TK | 3vs5 | A | | 7-(1-methylpiperidin-4-yl)-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2645 | |
| HCK | Src | TK | 1qcf | A | | 1-ter-butyl-3-p-tolyl-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 2641 | |
| HCK | Src | TK | 3vs7 | B | | 1-cyclopentyl-3-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 2648 | |
| HCK | Src | TK | 4lue | A | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2655 | |
| HCK | Src | TK | 3vry | A | | 4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentane | Human | 2647 | |
| HCK | Src | TK | 3vs1 | A | | 1-[4-(4-amino-7-cyclopentyl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]-3-phenylurea | Human | 2635 | |
| HCK | Src | TK | 1ad5 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 9483 | |
| HCK | Src | TK | 5h0e | A | | (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]amino]-4-methyl-pentanamide | Human | 8538 | |
| HCK | Src | TK | 4lud | B | | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | 2637 | |
| HCK | Src | TK | 3vry | B | | 4-amino-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl-cyclopentane | Human | 2646 | |
| HCK | Src | TK | 2c0o | B | B | n-(4-{1-[4-(4-acetylpiperazin-1-yl)-trans-cyclohexyl]-4-amino-1h-pyrazolo[3,4-d]pyrimidin-3-yl}-2-methoxyphenyl)-1-methyl-1h-indole-2-carboxamide | Human | 2657 | |
| HCK | Src | TK | 5h0b | A | | (2~{s})-2-[[4-[4-azanyl-5-(4-phenoxyphenyl)pyrrolo[2,3-d]pyrimidin-7-yl]cyclohexyl]azaniumyl]-4-methyl-pentanoate | Human | 8567 | |
| HCK | Src | TK | 5zj6 | B | | 7-[trans-4-(4-methylpiperazin-1-yl)cyclohexyl]-5-(4-phenoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 9988 | |
| HCK | Src | TK | 3vs4 | B | | 5-(4-phenoxyphenyl)-7-(tetrahydro-2h-pyran-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 2638 | |
| HCK | Src | TK | 1ad5 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 9480 | |
| SRC | Src | TK | 6e6e | D | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11494 | |
| SRC | Src | TK | 8haq | A | | 4-[(~{e})-(7-oxidanyl-6~{h}-pyrrolo[2,3-g][1,3]benzothiazol-8-yl)methylideneamino]-~{n}-pyridin-2-yl-benzenesulfonamide | Human | 14883 | |
| SRC | Src | TK | 1fmk | A | | - | Human | 981 | |
| SRC | Src | TK | 4mxy | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 982 | |
| SRC | Src | TK | 6e6e | F | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11487 | |
| SRC | Src | TK | 1yol | B | | 1-{4-[4-amino-5-(3-methoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl]benzyl}piperidin-4-ol | Human | 966 | |
| SRC | Src | TK | 6e6e | A | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11485 | |
| SRC | Src | TK | 6e6e | H | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11481 | |
| SRC | Src | TK | 6e6e | C | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11488 | |
| SRC | Src | TK | 1y57 | A | | 4-[(4-methylpiperazin-1-yl)methyl]-n-{3-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl}benzamide | Human | 986 | |
| SRC | Src | TK | 6e6e | G | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11477 | |
| SRC | Src | TK | 1yoj | B | | - | Human | 974 | |
| SRC | Src | TK | 6e6e | F | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11472 | |
| SRC | Src | TK | 8jn8 | A | | (2r)-n-cyclopentyl-2-[cyclopropyl(ethanoyl)amino]-2-(4-fluorophenyl)ethanamide | Human | 15312 | |
| SRC | Src | TK | 4k11 | A | A | 1-tert-butyl-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 983 | |
| SRC | Src | TK | 6e6e | D | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11489 | |
| SRC | Src | TK | 6e6e | B | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11480 | |
| SRC | Src | TK | 4mxy | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 972 | |
| SRC | Src | TK | 4mxz | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 969 | |
| SRC | Src | TK | 6e6e | B | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11484 | |
| SRC | Src | TK | 9ns0 | A | 7 | - | Human | 15612 | |
| SRC | Src | TK | 2bdj | A | | 3-[2-(2-cyclopentyl-6-{[4-(dimethylphosphoryl)phenyl]amino}-9h-purin-9-yl)ethyl]phenol | Human | 971 | |
| SRC | Src | TK | 4mxz | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 988 | |
| SRC | Src | TK | 9ns1 | A | 8 | - | Human | 15615 | |
| SRC | Src | TK | 2h8h | A | A | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 970 | |
| SRC | Src | TK | 9ns1 | A | 14 | - | Human | 15616 | |
| SRC | Src | TK | 6e6e | C | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11492 | |
| SRC | Src | TK | 9ns0 | A | 10 | - | Human | 15617 | |
| SRC | Src | TK | 6e6e | H | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11483 | |
| SRC | Src | TK | 9ns1 | A | 4 | - | Human | 15618 | |
| SRC | Src | TK | 4mxx | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 976 | |
| SRC | Src | TK | 4mxo | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 990 | |
| SRC | Src | TK | 6e6e | C | A | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11471 | |
| SRC | Src | TK | 6e6e | D | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11473 | |
| SRC | Src | TK | 1yol | A | | 1-{4-[4-amino-5-(3-methoxyphenyl)-7h-pyrrolo[2,3-d]pyrimidin-7-yl]benzyl}piperidin-4-ol | Human | 968 | |
| SRC | Src | TK | 6e6e | F | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11486 | |
| SRC | Src | TK | 9ns0 | A | 11 | - | Human | 15619 | |
| SRC | Src | TK | 9ns1 | A | 5 | - | Human | 15620 | |
| SRC | Src | TK | 6e6e | G | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11474 | |
| SRC | Src | TK | 2h8h | A | B | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 992 | |
| SRC | Src | TK | 9ns0 | A | 19 | - | Human | 15621 | |
| SRC | Src | TK | 6e6e | A | C | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11491 | |
| SRC | Src | TK | 6e6e | A | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11482 | |
| SRC | Src | TK | 1yi6 | A | | - | Human | 967 | |
| SRC | Src | TK | 9ns0 | A | 17 | - | Human | 15626 | |
| SRC | Src | TK | 9ns1 | A | 3 | - | Human | 15627 | |
| SRC | Src | TK | 9ns1 | A | 19 | - | Human | 15628 | |
| SRC | Src | TK | 6e6e | B | B | n-(2-chloro-6-methylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4-{[2-(propanoylamino)phenyl]amino}pyrimidine-5-carboxamide | Human | 11476 | |
| SRC | Src | TK | 1yoj | A | | - | Human | 984 | |
| SRC | Src | TK | 1ksw | A | | n6-benzyl adenosine-5'-diphosphate | Human | 985 | |
| SRC | Src | TK | 9ns1 | A | 7 | - | Human | 15629 | |
| SRC | Src | TK | 9ns1 | A | 9 | - | Human | 15630 | |
| SRC | Src | TK | 7ote | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Human | 14240 | |
| SRC | Src | TK | 4k11 | A | B | 1-tert-butyl-3-(naphthalen-1-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 977 | |
| SRC | Src | TK | 9ns1 | A | 18 | - | Human | 15631 | |
| SRC | Src | TK | 4mxx | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 989 | |
| SRC | Src | TK | 1yom | B | | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 987 | |
| SRC | Src | TK | 9ns1 | A | 20 | - | Human | 15632 | |
| SRC | Src | TK | 9ns0 | A | 12 | - | Human | 15633 | |
| SRC | Src | TK | 2src | A | | phosphoaminophosphonic acid-adenylate ester | Human | 979 | |
| SRC | Src | TK | 9ns0 | A | 4 | - | Human | 15634 | |
| LCK | Src | TK | 1qpe | A | | 1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Human | 2271 | |
| LCK | Src | TK | 3mpm | A | B | 4-{(6r,7r)-7-amino-3-[3-(4-methylpiperazin-1-yl)phenyl]-6,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl}phenol | Human | 2295 | |
| LCK | Src | TK | 2ofv | A | | 3-(2-aminoquinazolin-6-yl)-4-methyl-n-[3-(trifluoromethyl)phenyl]benzamide | Human | 2280 | |
| LCK | Src | TK | 3b2w | A | | n-[5-({[2-fluoro-3-(trifluoromethyl)phenyl]amino}carbonyl)-2-methylphenyl]-4-methoxy-2-[(4-piperazin-1-ylphenyl)amino]pyrimidine-5-carboxamide | Human | 2299 | |
| LCK | Src | TK | 2ofu | A | | 2,6-dimethylphenyl 2-(3,5-dimethoxy-4-(3-(4-methylpiperazin-1-yl)propoxy)phenylamino)pyrimidin- 4-yl(2,4-dimethoxyphenyl)carbamate | Human | 2259 | |
| LCK | Src | TK | 6pdj | A | A | n-{4-[(6-methoxypyrazolo[1,5-a]pyridine-3-carbonyl)amino]-3-methylphenyl}-1-methyl-1h-indazole-3-carboxamide | Human | 11698 | |
| LCK | Src | TK | 3byo | A | | 6-(2,6-dimethylphenyl)-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimido[5',4':5,6]pyrimido[1,2-a]benzimidazol-5(6h)-one | Human | 2272 | |
| LCK | Src | TK | 3mpm | A | A | 4-{(6r,7r)-7-amino-3-[3-(4-methylpiperazin-1-yl)phenyl]-6,7-dihydropyrazolo[1,5-a]pyrimidin-6-yl}phenol | Human | 2279 | |
| LCK | Src | TK | 2of4 | A | | 5,6-diphenyl-n-(2-piperazin-1-ylethyl)furo[2,3-d]pyrimidin-4-amine | Human | 2296 | |
| LCK | Src | TK | 3ac4 | A | | 5-[(2-amino-1,1-dimethylethyl)amino]-7-[(3,5-dimethoxyphenyl)amino][1,2,4]triazolo[4,3-c]pyrimidine-8-carboxamide | Human | 2278 | |
| LCK | Src | TK | 3ac5 | A | | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-7-[(3,5-dimethoxyphenyl)amino]-2-(3-hydroxyphenyl)[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxamide | Human | 2277 | |
| LCK | Src | TK | 1qpd | A | | staurosporine | Human | 2267 | |
| LCK | Src | TK | 2og8 | B | | n-{2-[(n,n-diethylglycyl)amino]-5-(trifluoromethyl)phenyl}-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamide | Human | 2282 | |
| LCK | Src | TK | 1qpc | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2291 | |
| LCK | Src | TK | 3bym | A | | n-phenyl-1-{4-[(3,4,5-trimethoxyphenyl)amino]-1,3,5-triazin-2-yl}-1h-benzimidazol-2-amine | Human | 2264 | |
| LCK | Src | TK | 2of2 | A | | 2,3-diphenyl-n-(2-piperazin-1-ylethyl)furo[2,3-b]pyridin-4-amine | Human | 2261 | |
| LCK | Src | TK | 4c3f | A | B | n-phenyl-4-(5-phenyl-1h-pyrazol-4-yl)pyrimidin-2-amine | Human | 2297 | |
| LCK | Src | TK | 2zm4 | A | | n-(2-chloro-6-methylphenyl)-8-[(3s)-3-methylpiperazin-1-yl]imidazo[1,5-a]quinoxalin-4-amine | Human | 2262 | |
| LCK | Src | TK | 3ad5 | A | | 4-[4-(benzyloxy)phenyl]-5-{[2-(4-chlorophenyl)-2-oxoethyl]sulfanyl}-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 2270 | |
| LCK | Src | TK | 2og8 | A | | n-{2-[(n,n-diethylglycyl)amino]-5-(trifluoromethyl)phenyl}-4-methyl-3-[2-(methylamino)quinazolin-6-yl]benzamide | Human | 2286 | |
| LCK | Src | TK | 3lck | A | A | - | Human | 2263 | |
| LCK | Src | TK | 2zm1 | A | | n-(2-chlorophenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine | Human | 2273 | |
| LCK | Src | TK | 3ac8 | A | | 7-[(2-amino-2-methylpropyl)amino]-5-cyclopropyl-2-[(3,5-dimethoxyphenyl)amino]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2300 | |
| LCK | Src | TK | 4c3f | A | A | n-phenyl-4-(5-phenyl-1h-pyrazol-4-yl)pyrimidin-2-amine | Human | 2276 | |
| LCK | Src | TK | 3acj | A | | 7-(3,4-dimethoxyphenyl)-5-(ethylsulfanyl)imidazo[1,2-c]pyrimidine | Human | 2260 | |
| LCK | Src | TK | 3byu | A | | 2-methyl-n-{4-methyl-3-[(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-5-yl)carbamoyl]phenyl}-3-(trifluoromethyl)benzamide | Human | 2288 | |
| LCK | Src | TK | 2zyb | A | | n-(2,6-dimethylphenyl)-5-phenylimidazo[1,5-a]pyrazin-8-amine | Human | 2275 | |
| LCK | Src | TK | 1qpj | A | | staurosporine | Human | 2283 | |
| LCK | Src | TK | 3ac1 | A | | 5-{[(1r,2s)-2-aminocyclohexyl]amino}-3-[(3,5-dimethoxyphenyl)amino]pyrazine-2-carboxamide | Human | 2287 | |
| LCK | Src | TK | 3kxz | A | | 3-[7-[(3-hydroxyphenyl)amino]pyrazolo[1,5-a]pyrimidin-2-yl]-n-(1-hydroxy-2,2,6,6-tetramethyl-piperidin-4-yl)benzamide | Human | 2281 | |
| LCK | Src | TK | 3ad6 | A | | 7-[(cyclopropylmethyl)amino]-2-[(4-methoxyphenyl)amino]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2274 | |
| LCK | Src | TK | 3ac2 | A | | 7-[(2-amino-2-methylpropyl)amino]-2-[(3,5-dimethoxyphenyl)amino]-5-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2266 | |
| LCK | Src | TK | 3ack | A | | 6-(5-methoxy-1-methyl-1h-indol-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 2284 | |
| LCK | Src | TK | 3ac3 | A | | 2-[(3,5-dimethoxyphenyl)amino]-5-ethyl-7-[(2r)-2-(hydroxymethyl)pyrrolidin-1-yl]pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2292 | |
| LCK | Src | TK | 2ofv | B | | 3-(2-aminoquinazolin-6-yl)-4-methyl-n-[3-(trifluoromethyl)phenyl]benzamide | Human | 2294 | |
| LCK | Src | TK | 3ad4 | A | | (4-chlorophenyl)(5-methoxy-1-benzofuran-2-yl)methanone | Human | 2268 | |
| LCK | Src | TK | 3bys | A | | 4-methyl-n~3~-(2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-5-yl)-n~1~-[3-(trifluoromethyl)phenyl]benzene-1,3-dicarboxamide | Human | 2293 | |
| FYN | Src | TK | 2dq7 | X | | staurosporine | Human | 1941 | |
| FYN | Src | TK | 10dj | A | | n-(5-chloro-1,3-benzodioxol-4-yl)-7-[2-(4-methylpiperazin-1-yl)ethoxy]-5-(tetrahydro-2h-pyran-4-yloxy)quinazolin-4-amine | Human | 16102 | |
| PTK6 (BRK) | Src | TK | 5d7v | D | B | - | Human | 6952 | |
| PTK6 (BRK) | Src | TK | 5d7v | D | A | - | Human | 6948 | |
| PTK6 (BRK) | Src | TK | 5h2u | D | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7340 | |
| PTK6 (BRK) | Src | TK | 5h2u | B | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7337 | |
| PTK6 (BRK) | Src | TK | 5d7v | A | A | - | Human | 6953 | |
| PTK6 (BRK) | Src | TK | 5h2u | D | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7344 | |
| PTK6 (BRK) | Src | TK | 6cz3 | A | B | (3-fluoro-4-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}phenyl)(morpholin-4-yl)methanone | Human | 9999 | |
| PTK6 (BRK) | Src | TK | 5d7v | A | B | - | Human | 6950 | |
| PTK6 (BRK) | Src | TK | 5d7v | B | A | - | Human | 6955 | |
| PTK6 (BRK) | Src | TK | 5h2u | B | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7339 | |
| PTK6 (BRK) | Src | TK | 5h2u | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 7338 | |
| PTK6 (BRK) | Src | TK | 6cz4 | A | B | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamide | Human | 10000 | |
