Search results (17 entries covering 12 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
MLKLTKL-UniqueTKL7jxuA-Human13394
MLKLTKL-UniqueTKL5ko1AA[(1~{r})-2-[(4-fluorophenyl)amino]-2-oxidanylidene-1-phenyl-ethyl] 3-azanylpyrazine-2-carboxylateHuman7269
MLKLTKL-UniqueTKL5knjA1-[4-[methyl-[2-[(3-sulfamoylphenyl)amino]pyrimidin-4-yl]amino]phenyl]-3-[4-(trifluoromethyloxy)phenyl]ureaHuman7270
MLKLTKL-UniqueTKL6bwkA-Human10038
MLKLTKL-UniqueTKL7jw7A-Human13395
MLKLTKL-UniqueTKL4mwiAB-Human3049
MLKLTKL-UniqueTKL7jxuB-Human13396
MLKLTKL-UniqueTKL6lk5A-Human13094
MLKLTKL-UniqueTKL5knjB1-[4-[methyl-[2-[(3-sulfamoylphenyl)amino]pyrimidin-4-yl]amino]phenyl]-3-[4-(trifluoromethyloxy)phenyl]ureaHuman7268
MLKLTKL-UniqueTKL6o5zA-Human12782
MLKLTKL-UniqueTKL4mwiAA-Human3047
MLKLTKL-UniqueTKL5ko1AB[(1~{r})-2-[(4-fluorophenyl)amino]-2-oxidanylidene-1-phenyl-ethyl] 3-azanylpyrazine-2-carboxylateHuman7271
MLKLTKL-UniqueTKL7monAn-[4-({2-[(cyclopropanecarbonyl)amino]pyridin-4-yl}oxy)-3-fluorophenyl]-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamideHuman13980
MLKLTKL-UniqueTKL8slzA-Human14988
MLKLTKL-UniqueTKL4m67A-Human3048
MLKLTKL-UniqueTKL6lk6A-Human13095
MLKLTKL-UniqueTKL6o5zB1-[2-fluoranyl-5-(trifluoromethyl)phenyl]-3-[4-[methyl-[2-[(3-sulfamoylphenyl)amino]pyrimidin-4-yl]amino]phenyl]ureaHuman12783