Search results (41 entries covering 22 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
TTBK2TTBKCK16vrfBAadenosine-5'-diphosphateHuman12345
TTBK1TTBKCK17zhnAA4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHuman14721
TTBK1TTBKCK17zhnAB4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHuman14717
TTBK1TTBKCK17jxxAA4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHuman13579
TTBK1TTBKCK17q8vA~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14133
TTBK1TTBKCK14nfnAB3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenolHuman770
TTBK1TTBKCK131hoA~{n}-[4-(furan-2-yl)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman15850
TTBK1TTBKCK17jxxAB4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-olHuman13578
TTBK1TTBKCK14nfnAA3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenolHuman773
TTBK1TTBKCK17qhwA~{n}-[4-(4-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14477
TTBK1TTBKCK17zhoAA4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-olHuman14718
TTBK1TTBKCK17zhpAB1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-olHuman14719
TTBK1TTBKCK17zhqAA(3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-olHuman14720
TTBK1TTBKCK14btmBmethyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoateHuman774
TTBK1TTBKCK14btmAmethyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoateHuman772
TTBK1TTBKCK17jxyA(3s)-1-[1-(2-aminopyrimidin-4-yl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-methylpent-1-yn-3-olHuman13580
TTBK1TTBKCK17zhoAB4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-olHuman14722
TTBK1TTBKCK17zhqAB(3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-olHuman14723
TTBK1TTBKCK14btjAadenosine-5'-diphosphateHuman769
TTBK1TTBKCK17zhpAA1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-olHuman14724
TTBK1TTBKCK14btjBadenosine-5'-triphosphateHuman767
TTBK1TTBKCK17q8wAA~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14134
TTBK1TTBKCK14nfmA-Human768
TTBK1TTBKCK17q8wAB~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14135
TTBK1TTBKCK14btkA4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman771
TTBK1TTBKCK18xpzA-Human15163
TTBK2TTBKCK16u0kBA4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman12049
TTBK2TTBKCK16vrfBBadenosine-5'-diphosphateHuman12342
TTBK2TTBKCK16vrfABadenosine-5'-diphosphateHuman12343
TTBK2TTBKCK16u0kAA4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman12046
TTBK2TTBKCK17q8yAB~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14138
TTBK2TTBKCK17q90AA~{n}-[4-(4-methoxyphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14139
TTBK2TTBKCK16vrfAAadenosine-5'-diphosphateHuman12344
TTBK2TTBKCK17q8zAB~{n}-(4-phenoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14140
TTBK2TTBKCK16u0kBB4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman12047
TTBK2TTBKCK17q8yAA~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14141
TTBK2TTBKCK17q8zAA~{n}-(4-phenoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14142
TTBK2TTBKCK16u0kAB4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman12048
TTBK2TTBKCK17q90AB~{n}-[4-(4-methoxyphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman14143
TTBK1TTBKCK19hhwAB~{n}-[2-(1~{h}-pyrrolo[2,3-b]pyridin-5-yl)phenyl]propanamideHuman15851
TTBK1TTBKCK19hhwAA~{n}-[2-(1~{h}-pyrrolo[2,3-b]pyridin-5-yl)phenyl]propanamideHuman15852