| Btk (BTK) | Tec | TK | 8s93 | A | A | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | 14997 | |
| Btk (BTK) | Tec | TK | 8s93 | A | B | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | 14996 | |
| Btk (BTK) | Tec | TK | 8s9f | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 14998 | |
| Btk (BTK) | Tec | TK | 8gmb | A | | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | 14999 | |
| Btk (BTK) | Tec | TK | 8ff0 | A | | 6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-one | Mouse | 14834 | |
| Btk (BTK) | Tec | TK | 8fd9 | A | A | acalabrutinib | Mouse | 14836 | |
| Btk (BTK) | Tec | TK | 8fd9 | A | B | acalabrutinib | Mouse | 14835 | |
| Btk (BTK) | Tec | TK | 9xyv | A | A | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Mouse | 16246 | |
| Btk (BTK) | Tec | TK | 9xz2 | A | B | 6-amino-7-(4-phenoxyphenyl)-9-[(3r)-1-propanoylpyrrolidin-3-yl]-7,9-dihydro-8h-purin-8-one | Mouse | 16247 | |
| Btk (BTK) | Tec | TK | 6mny | B | A | - | Mouse | 11306 | |
| Btk (BTK) | Tec | TK | 9xyv | A | C | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Mouse | 16248 | |
| Btk (BTK) | Tec | TK | 9xz2 | A | A | 6-amino-7-(4-phenoxyphenyl)-9-[(3r)-1-propanoylpyrrolidin-3-yl]-7,9-dihydro-8h-purin-8-one | Mouse | 16249 | |
| Btk (BTK) | Tec | TK | 4xi2 | A | | - | Mouse | 5815 | |
| Btk (BTK) | Tec | TK | 9xyy | A | | (2e)-1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}but-2-en-1-one | Mouse | 16250 | |
| Btk (BTK) | Tec | TK | 6mny | B | B | - | Mouse | 11309 | |
| Btk (BTK) | Tec | TK | 9xyv | A | B | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Mouse | 16251 | |
| Btk (BTK) | Tec | TK | 6mny | A | B | 5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamide | Mouse | 11308 | |
| Btk (BTK) | Tec | TK | 6mny | A | A | 5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamide | Mouse | 11307 | |
| Btk (BTK) | Tec | TK | 9ejx | A | | {(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}(cyclopropyl)methanone | Mouse | 16252 | |
