| NTRK1 (TRKA) | Trk | TK | 6j5l | A | C | n-{2-[({3-[6-(piperazin-1-yl)pyridin-3-yl]-1h-indazol-5-yl}amino)methyl]phenyl}methanesulfonamide | Human | 11437 | |
| NTRK1 (TRKA) | Trk | TK | 6d20 | A | | 5-{[2,4-dichloro-5-(pyridin-2-yl)benzene-1-carbonyl]amino}-n-(2-hydroxy-2-methylpropyl)-1-phenyl-1h-pyrazole-3-carboxamide | Human | 9875 | |
| NTRK1 (TRKA) | Trk | TK | 6dkb | A | | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-5-(1-methyl-1h-imidazol-4-yl)pyridine-3-carboxamide | Human | 10057 | |
| NTRK1 (TRKA) | Trk | TK | 7vkm | A | A | - | Human | 13946 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | C | A | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 11999 | |
| NTRK1 (TRKA) | Trk | TK | 5kmi | A | | 1-(9~{h}-fluoren-9-yl)-3-(2-methyl-4-phenyl-pyrimidin-5-yl)urea | Human | 7330 | |
| NTRK1 (TRKA) | Trk | TK | 6dki | A | B | 6-amino-5-{[(3s)-4,4-difluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}pyrrolidin-3-yl]oxy}-n-methylpyridine-3-carboxamide | Human | 10061 | |
| NTRK1 (TRKA) | Trk | TK | 6iqn | B | | 4-[[4-azanyl-3-(4-cyclohexylpiperazin-1-yl)-9,10-bis(oxidanylidene)anthracen-1-yl]amino]benzoic acid | Human | 11950 | |
| NTRK1 (TRKA) | Trk | TK | 7xbi | A | B | 4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]-~{n}-[3-(1-methylpyrazol-4-yl)-1~{h}-indazol-5-yl]-2-(trifluoromethyl)benzamide | Human | 14686 | |
| NTRK1 (TRKA) | Trk | TK | 7xbi | A | A | 4-[[2-fluoranyl-5-(trifluoromethyl)phenyl]carbamoylamino]-~{n}-[3-(1-methylpyrazol-4-yl)-1~{h}-indazol-5-yl]-2-(trifluoromethyl)benzamide | Human | 14687 | |
| NTRK1 (TRKA) | Trk | TK | 7xaf | A | | 4^6,14-dimethyl-n-(3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-10-oxo-5-oxa-11,14-diaza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclo-tetradecaphan-2-yne-45-carboxamide | Human | 14232 | |
| NTRK2 (TRKB) | Trk | TK | 4asz | A | | - | Human | 3599 | |
| NTRK1 (TRKA) | Trk | TK | 7vko | A | | repotrectinib | Human | 13943 | |
| NTRK1 (TRKA) | Trk | TK | 7vkn | A | B | repotrectinib | Human | 13944 | |
| NTRK1 (TRKA) | Trk | TK | 7vkn | A | A | repotrectinib | Human | 13945 | |
| NTRK1 (TRKA) | Trk | TK | 6dkg | A | A | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-4-(2-hydroxy-2-methylpropoxy)benzamide | Human | 10059 | |
| NTRK1 (TRKA) | Trk | TK | 6dki | A | A | 6-amino-5-{[(3s)-4,4-difluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}pyrrolidin-3-yl]oxy}-n-methylpyridine-3-carboxamide | Human | 10060 | |
| NTRK1 (TRKA) | Trk | TK | 9dai | A | | staurosporine | Human | 16134 | |
| NTRK2 (TRKB) | Trk | TK | 4at3 | A | | (5z)-5-(carbamoylimino)-3-[(5r)-6,7,8,9-tetrahydro-5h-benzo[7]annulen-5-ylsulfanyl]-2,5-dihydroisothiazole-4-carboxamide | Human | 3600 | |
| NTRK1 (TRKA) | Trk | TK | 8j63 | A | | 4^6-methyl-n-(3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-11-oxo-5-oxa-10,14-diaza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamide | Human | 14984 | |
| NTRK1 (TRKA) | Trk | TK | 8j5w | A | | n-(3-cyclopropyl-5-((4-methylpiperazin-1-yl)methyl)phenyl)-4^6-methyl-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamide | Human | 14985 | |
| NTRK1 (TRKA) | Trk | TK | 8j5x | A | | n-(3-cyclopropyl-5-((4-methylpiperazin-1-yl)methyl)phenyl)-4^6-methyl-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamide | Human | 14987 | |
| NTRK3 (TRKC) | Trk | TK | 6kzc | A | | 3-(2-imidazo[1,2-a]pyrazin-3-ylethynyl)-2-methyl-~{n}-[3-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]benzamide | Human | 11696 | |
| NTRK3 (TRKC) | Trk | TK | 3v5q | A | | 1-(3-{[(3z)-2-oxo-3-(1h-pyrrol-2-ylmethylidene)-2,3-dihydro-1h-indol-6-yl]amino}phenyl)-3-[3-(trifluoromethyl)phenyl]urea | Human | 102 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | B | A | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 100 | |
| NTRK1 (TRKA) | Trk | TK | 5kmj | A | A | ~{n}-(pyridin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)ethanamide | Human | 7334 | |
| NTRK1 (TRKA) | Trk | TK | 6pl1 | A | A | n-(5-{[(7-methyl-4-oxo-4h-pyrido[1,2-a]pyrimidin-2-yl)methyl]sulfanyl}-1,3,4-thiadiazol-2-yl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | 11722 | |
| NTRK1 (TRKA) | Trk | TK | 6dkw | B | A | 5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamide | Human | 10062 | |
| NTRK1 (TRKA) | Trk | TK | 4yps | A | | 4-{6-[(3r)-3-(3-fluorophenyl)morpholin-4-yl]imidazo[1,2-b]pyridazin-3-yl}benzonitrile | Human | 3615 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | B | B | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3604 | |
| NTRK1 (TRKA) | Trk | TK | 6j5l | A | A | n-{2-[({3-[6-(piperazin-1-yl)pyridin-3-yl]-1h-indazol-5-yl}amino)methyl]phenyl}methanesulfonamide | Human | 11436 | |
| NTRK1 (TRKA) | Trk | TK | 5kmm | A | | 1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-naphthalen-1-yl-urea | Human | 7331 | |
| NTRK1 (TRKA) | Trk | TK | 6nsp | A | B | n-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)-2-(3-oxo-2,3-dihydro-4h-1,4-benzothiazin-4-yl)acetamide | Human | 11175 | |
| NTRK1 (TRKA) | Trk | TK | 5h3q | A | A | 1-[(3s,4r)-4-[3,4-bis(fluoranyl)phenyl]-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(5-ethoxy-4-methyl-2-phenyl-pyrazol-3-yl)urea | Human | 7461 | |
| NTRK1 (TRKA) | Trk | TK | 6pl1 | A | B | n-(5-{[(7-methyl-4-oxo-4h-pyrido[1,2-a]pyrimidin-2-yl)methyl]sulfanyl}-1,3,4-thiadiazol-2-yl)-n'-[3-(trifluoromethyl)phenyl]urea | Human | 11723 | |
| NTRK1 (TRKA) | Trk | TK | 4pmt | A | B | n~4~-[4-(morpholin-4-yl)phenyl]-n~6~-(pyridin-3-ylmethyl)pyrido[3,2-d]pyrimidine-4,6-diamine | Human | 3612 | |
| NTRK1 (TRKA) | Trk | TK | 6nsp | A | A | n-(8-methyl-2-phenylimidazo[1,2-a]pyridin-3-yl)-2-(3-oxo-2,3-dihydro-4h-1,4-benzothiazin-4-yl)acetamide | Human | 11173 | |
| NTRK1 (TRKA) | Trk | TK | 4gt5 | A | A | - | Human | 3616 | |
| NTRK1 (TRKA) | Trk | TK | 6dkg | A | B | 2-{[(3r,4s)-3-fluoro-1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl]oxy}-4-(2-hydroxy-2-methylpropoxy)benzamide | Human | 10063 | |
| NTRK1 (TRKA) | Trk | TK | 6pl3 | A | A | 2-[(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)amino]-2-oxoethyl 4-(1h-tetrazol-1-yl)benzoate | Human | 11599 | |
| NTRK1 (TRKA) | Trk | TK | 6d1y | A | B | 2,4-dichloro-n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)benzamide | Human | 9871 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | B | B | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12000 | |
| NTRK1 (TRKA) | Trk | TK | 5kmo | A | | 1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-pyridin-2-yl-urea | Human | 7329 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | A | B | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12005 | |
| NTRK1 (TRKA) | Trk | TK | 4pmm | A | A | n-(3-cyclopropyl-1-phenyl-1h-pyrazol-5-yl)-2-{4-[3-methoxy-4-(4-methyl-1h-imidazol-1-yl)phenyl]-1h-1,2,3-triazol-1-yl}acetamide | Human | 3618 | |
| NTRK1 (TRKA) | Trk | TK | 5jfv | A | A | n-{5-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}-2-(4-chlorophenyl)acetamide | Human | 7504 | |
| NTRK2 (TRKB) | Trk | TK | 4at4 | A | | 1-[4-(4-aminothieno[2,3-d]pyrimidin-5-yl)phenyl]-3-[2-fluoro-5-(trifluoromethyl)phenyl]urea | Human | 3598 | |
| NTRK2 (TRKB) | Trk | TK | 4at5 | A | | 5-{3-methoxy-4-[(4-methoxybenzyl)oxy]benzyl}pyrimidine-2,4-diamine | Human | 3597 | |
| NTRK1 (TRKA) | Trk | TK | 5kvt | A | B | entrectinib | Human | 9451 | |
| NTRK1 (TRKA) | Trk | TK | 7vkm | A | B | - | Human | 13942 | |
| NTRK1 (TRKA) | Trk | TK | 5jfv | A | B | n-{5-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}-2-(4-chlorophenyl)acetamide | Human | 7503 | |
| NTRK1 (TRKA) | Trk | TK | 4yne | A | B | 6-[(2r)-2-(3-fluorophenyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)imidazo[1,2-b]pyridazine | Human | 3611 | |
| NTRK1 (TRKA) | Trk | TK | 5i8a | A | B | (6r)-3-(methylsulfanyl)-6-phenyl-1-(1h-pyrazol-3-yl)-6,7-dihydrothieno[3,4-c]pyridin-4(5h)-one | Human | 8312 | |
| NTRK1 (TRKA) | Trk | TK | 6d1y | A | A | 2,4-dichloro-n-(3-methyl-1-phenyl-1h-pyrazol-5-yl)benzamide | Human | 9873 | |
| NTRK1 (TRKA) | Trk | TK | 6d1z | A | A | 5-{[5-(6-aminopyridin-2-yl)-2-chlorobenzene-1-carbonyl]amino}-1-phenyl-1h-pyrazole-3-carboxamide | Human | 9874 | |
| NTRK1 (TRKA) | Trk | TK | 5kmk | A | | 2-fluoranyl-~{n}-[2-(4-fluorophenyl)-6-methyl-pyridin-3-yl]-4-(trifluoromethyl)benzamide | Human | 7336 | |
| NTRK1 (TRKA) | Trk | TK | 4pms | A | B | 4-(naphthalen-1-yl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1h-pyrrolo[3,2-c]pyridine-2-carboxylic acid | Human | 3601 | |
| NTRK1 (TRKA) | Trk | TK | 6dkw | A | A | 5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamide | Human | 10056 | |
| NTRK1 (TRKA) | Trk | TK | 6dkw | A | B | 5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamide | Human | 10058 | |
| NTRK1 (TRKA) | Trk | TK | 6pl4 | A | A | n-{[5-(methoxymethyl)-2-(trifluoromethoxy)phenyl]methyl}-n'-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)urea | Human | 12463 | |
| NTRK1 (TRKA) | Trk | TK | 4pmp | A | B | 1-cyclopropyl-1-[3-(1,3-thiazol-2-yl)benzyl]-3-[4-(trifluoromethoxy)phenyl]urea | Human | 3608 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | C | A | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3617 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | A | B | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3610 | |
| NTRK1 (TRKA) | Trk | TK | 5kml | A | | 1-(5-methyl-3-phenyl-1,2-oxazol-4-yl)-3-[[2-(trifluoromethyl)phenyl]methyl]urea | Human | 7333 | |
| NTRK1 (TRKA) | Trk | TK | 5jfw | A | B | 2-(4-cyanophenyl)-n-{5-[7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}acetamide | Human | 7505 | |
| NTRK1 (TRKA) | Trk | TK | 4gt5 | A | B | - | Human | 3609 | |
| NTRK1 (TRKA) | Trk | TK | 5kmn | A | | 1-(2-methyl-4-phenyl-pyrimidin-5-yl)-3-[[2-(trifluoromethyl)phenyl]methyl]urea | Human | 7332 | |
| NTRK1 (TRKA) | Trk | TK | 6pmb | A | | 2-[5,7-dimethyl-2-(pyridin-3-yl)[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-n-[3-(trifluoromethyl)phenyl]acetamide | Human | 12001 | |
| NTRK1 (TRKA) | Trk | TK | 6pl4 | A | B | n-{[5-(methoxymethyl)-2-(trifluoromethoxy)phenyl]methyl}-n'-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)urea | Human | 12464 | |
| NTRK1 (TRKA) | Trk | TK | 8j61 | A | | 4^6-methyl-n-(3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl)-14-oxo-5-oxa-13-aza-1(3,6)-imidazo[1,2-b]pyridazina-4(1,3)-benzenacyclotetradecaphan-2-yne-4^5-carboxamide | Human | 14986 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | A | A | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3602 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | A | A | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12004 | |
| NTRK1 (TRKA) | Trk | TK | 5jfw | A | A | 2-(4-cyanophenyl)-n-{5-[7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}acetamide | Human | 7500 | |
| NTRK1 (TRKA) | Trk | TK | 6pma | A | | n-[2-chloro-5-(trifluoromethyl)phenyl]-2-[1-(4-methoxyphenyl)-4-oxo-1,4-dihydro-5h-pyrazolo[3,4-d]pyrimidin-5-yl]acetamide | Human | 12006 | |
| NTRK1 (TRKA) | Trk | TK | 6j5l | A | B | n-{2-[({3-[6-(piperazin-1-yl)pyridin-3-yl]-1h-indazol-5-yl}amino)methyl]phenyl}methanesulfonamide | Human | 11435 | |
| NTRK1 (TRKA) | Trk | TK | 5h3q | A | B | 1-[(3s,4r)-4-[3,4-bis(fluoranyl)phenyl]-1-(2-methoxyethyl)pyrrolidin-3-yl]-3-(5-ethoxy-4-methyl-2-phenyl-pyrazol-3-yl)urea | Human | 7460 | |
| NTRK1 (TRKA) | Trk | TK | 6iqn | A | | 4-[[4-azanyl-3-(4-cyclohexylpiperazin-1-yl)-9,10-bis(oxidanylidene)anthracen-1-yl]amino]benzoic acid | Human | 11951 | |
| NTRK1 (TRKA) | Trk | TK | 5i8a | A | A | (6r)-3-(methylsulfanyl)-6-phenyl-1-(1h-pyrazol-3-yl)-6,7-dihydrothieno[3,4-c]pyridin-4(5h)-one | Human | 8311 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | C | B | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3621 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | B | A | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12007 | |
| NTRK1 (TRKA) | Trk | TK | 6dkw | B | B | 5-(1-methyl-1h-imidazol-4-yl)-2-[(1-{[4-(trifluoromethoxy)phenyl]acetyl}piperidin-4-yl)oxy]benzamide | Human | 10064 | |
| NTRK1 (TRKA) | Trk | TK | 4pmt | A | A | n~4~-[4-(morpholin-4-yl)phenyl]-n~6~-(pyridin-3-ylmethyl)pyrido[3,2-d]pyrimidine-4,6-diamine | Human | 3614 | |
| NTRK1 (TRKA) | Trk | TK | 6nss | A | B | n-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)-2-(10h-phenoxazin-10-yl)acetamide | Human | 11176 | |
| NTRK1 (TRKA) | Trk | TK | 6npt | A | | 4-tert-butyl-n-(1,3-diphenyl-1h-pyrazol-5-yl)benzamide | Human | 11172 | |
| NTRK1 (TRKA) | Trk | TK | 5jfs | A | B | n-{4-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-2-yl}-n'-(2,4-difluorophenyl)urea | Human | 7502 | |
| NTRK1 (TRKA) | Trk | TK | 4pmp | A | A | 1-cyclopropyl-1-[3-(1,3-thiazol-2-yl)benzyl]-3-[4-(trifluoromethoxy)phenyl]urea | Human | 3613 | |
| NTRK1 (TRKA) | Trk | TK | 4f0i | B | | - | Human | 3605 | |
| NTRK1 (TRKA) | Trk | TK | 5jfx | A | | n-{5-[2-amino-7-(1-hydroxy-2-methylpropan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-3-yl}-2-(5-chloropyridin-2-yl)acetamide | Human | 7501 | |
| NTRK1 (TRKA) | Trk | TK | 6d1z | A | B | 5-{[5-(6-aminopyridin-2-yl)-2-chlorobenzene-1-carbonyl]amino}-1-phenyl-1h-pyrazole-3-carboxamide | Human | 9870 | |
| NTRK1 (TRKA) | Trk | TK | 4aoj | B | A | 5-chloranyl-n2-[(1s)-1-(5-fluoranylpyridin-2-yl)ethyl]-n4-(3-propan-2-yloxy-1h-pyrazol-5-yl)pyrimidine-2,4-diamine | Human | 3607 | |
| NTRK1 (TRKA) | Trk | TK | 6d22 | A | | - | Human | 9872 | |
| NTRK1 (TRKA) | Trk | TK | 6pl3 | A | B | 2-[(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)amino]-2-oxoethyl 4-(1h-tetrazol-1-yl)benzoate | Human | 11600 | |
| NTRK1 (TRKA) | Trk | TK | 6pmc | A | | n-(6-{[(5-chloro-2-methoxyphenyl)carbamoyl]amino}-1,3-benzothiazol-2-yl)benzamide | Human | 12002 | |
| NTRK1 (TRKA) | Trk | TK | 4yne | A | A | 6-[(2r)-2-(3-fluorophenyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)imidazo[1,2-b]pyridazine | Human | 3620 | |
| NTRK1 (TRKA) | Trk | TK | 4pms | A | A | 4-(naphthalen-1-yl)-1-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1h-pyrrolo[3,2-c]pyridine-2-carboxylic acid | Human | 3606 | |
| NTRK1 (TRKA) | Trk | TK | 6nss | A | A | n-(8-methyl-2-phenylimidazo[1,2-a]pyrazin-3-yl)-2-(10h-phenoxazin-10-yl)acetamide | Human | 11174 | |
| NTRK1 (TRKA) | Trk | TK | 6pl2 | A | | n-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-2-{[1-(4-hydroxyphenyl)-1h-tetrazol-5-yl]sulfanyl}acetamide | Human | 11598 | |
| NTRK1 (TRKA) | Trk | TK | 6pme | C | B | n-[2,4-bis(morpholin-4-yl)phenyl]-3-phenoxybenzamide | Human | 12003 | |
| NTRK1 (TRKA) | Trk | TK | 5kvt | A | A | entrectinib | Human | 9450 | |
| NTRK1 (TRKA) | Trk | TK | 4f0i | A | | - | Human | 3603 | |
| NTRK1 (TRKA) | Trk | TK | 4pmm | A | B | n-(3-cyclopropyl-1-phenyl-1h-pyrazol-5-yl)-2-{4-[3-methoxy-4-(4-methyl-1h-imidazol-1-yl)phenyl]-1h-1,2,3-triazol-1-yl}acetamide | Human | 3619 | |
| NTRK1 (TRKA) | Trk | TK | 5kmj | A | B | ~{n}-(pyridin-2-ylmethyl)-2-(2-thiophen-2-ylindol-1-yl)ethanamide | Human | 7335 | |
| NTRK1 (TRKA) | Trk | TK | 5wr7 | A | | n-tert-butyl-2-[2-[6,6-dimethyl-8-(methylsulfonylamino)-11-oxidanylidene-naphtho[2,3-b][1]benzofuran-3-yl]ethynyl]-6-methyl-pyridine-4-carboxamide | Human | 8737 | |
| NTRK1 (TRKA) | Trk | TK | 5jfs | A | A | n-{4-[4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidine-5-carbonyl]pyridin-2-yl}-n'-(2,4-difluorophenyl)urea | Human | 7506 | |
| NTRK3 (TRKC) | Trk | TK | 3v5q | B | | 1-(3-{[(3z)-2-oxo-3-(1h-pyrrol-2-ylmethylidene)-2,3-dihydro-1h-indol-6-yl]amino}phenyl)-3-[3-(trifluoromethyl)phenyl]urea | Human | 97 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | A | A | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 101 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | A | B | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 98 | |
| NTRK3 (TRKC) | Trk | TK | 6kzd | A | | 3-[2-[6-(4-aminophenyl)imidazo[1,2-a]pyrazin-3-yl]ethynyl]-2-methyl-~{n}-[3-(4-methylpiperazin-1-yl)-5-propan-2-yl-phenyl]benzamide | Human | 11697 | |
| NTRK3 (TRKC) | Trk | TK | 4ymj | B | B | 4-[6-(benzylamino)imidazo[1,2-b]pyridazin-3-yl]benzonitrile | Human | 99 | |
