| AKT1 | Akt | AGC | 8uw2 | A | A | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15379 | |
| AKT1 | Akt | AGC | 8uw2 | A | B | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15380 | |
| AKT1 | Akt | AGC | 8uw9 | A | A | n-({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)-2-(2-fluoro-4-formyl-3-hydroxyphenyl)acetamide | Human | 15383 | |
| PRKCB (PKCb) | PKC | AGC | 2i0e | A | | 3-{1-[3-(dimethylamino)propyl]-2-methyl-1h-indol-3-yl}-4-(2-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2550 | |
| PRKCB (PKCb) | PKC | AGC | 2i0e | B | | 3-{1-[3-(dimethylamino)propyl]-2-methyl-1h-indol-3-yl}-4-(2-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2549 | |
| AKT1 | Akt | AGC | 6buu | B | C | - | Human | 10428 | |
| ROCK2 | DMPK | AGC | 6p5m | A | B | 6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11915 | |
| ROCK2 | DMPK | AGC | 4l6q | A | | 6-[4-(aminomethyl)-2-fluorophenoxy]-2,1-benzoxaborol-1(3h)-ol | Human | 1811 | |
| ROCK2 | DMPK | AGC | 6p5m | D | A | - | Human | 11925 | |
| ROCK2 | DMPK | AGC | 7jov | B | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12765 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | A | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3181 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1oky | A | A | staurosporine | Human | 3164 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvn | A | A | adenosine | Human | 7105 | |
| ROCK2 | DMPK | AGC | 6p5p | C | | 2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11919 | |
| ROCK2 | DMPK | AGC | 7jnt | A | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12754 | |
| ROCK2 | DMPK | AGC | 5u7q | B | | - | Human | 7990 | |
| GRK6 (GPRK6) | GRK | AGC | 2acx | A | | phosphoaminophosphonic acid-adenylate ester | Human | 420 | |
| AKT1 | Akt | AGC | 8uw9 | A | B | n-({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)-2-(2-fluoro-4-formyl-3-hydroxyphenyl)acetamide | Human | 15384 | |
| PRKCI (PKCi) | PKC | AGC | 5li9 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 7074 | |
| GRK5 (GPRK5) | GRK | AGC | 6pjx | A | A | sangivamycin | Human | 13042 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4v | A | A | - | Human | 14790 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 10671 | |
| PRKG1 (PKG1) | PKG | AGC | 6c0t | A | | n-[(3r,4r)-4-{[4-(2-fluoro-3-methoxy-6-propoxybenzene-1-carbonyl)benzene-1-carbonyl]amino}pyrrolidin-3-yl]-1h-indazole-5-carboxamide | Human | 9975 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 10668 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 10665 | |
| PRKG1 (PKG1) | PKG | AGC | 6bdl | A | A | - | Human | 10641 | |
| PRKCA (PKCa) | PKC | AGC | 8u37 | A | A | (6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamide | Human | 15159 | |
| PRKCA (PKCa) | PKC | AGC | 4ra4 | A | | (1r)-9-[(3s,4s)-1,3-dimethylpiperidin-4-yl]-8-(2-fluorophenyl)-1-methyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 3040 | |
| PRKCA (PKCa) | PKC | AGC | 3iw4 | C | | 3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dione | Human | 3042 | |
| PRKCA (PKCa) | PKC | AGC | 8uak | A | A | (6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamide | Human | 15161 | |
| PRKCA (PKCa) | PKC | AGC | 3iw4 | A | | 3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dione | Human | 3041 | |
| PRKCA (PKCa) | PKC | AGC | 3iw4 | B | | 3-(1h-indol-3-yl)-4-[2-(4-methylpiperazin-1-yl)quinazolin-4-yl]-1h-pyrrole-2,5-dione | Human | 3039 | |
| ROCK1 | DMPK | AGC | 5uzj | A | | n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide | Human | 9706 | |
| PRKACA (PKACa) | PKA | AGC | 4uja | A | A | 7-{(3s,4r)-4-[(5-bromothiophen-2-yl)carbonyl]pyrrolidin-3-yl}quinazolin-4(3h)-one | Human | 6549 | |
| STK38 (NDR1) | NDR | AGC | 6bxi | A | | phosphoaminophosphonic acid-adenylate ester | Human | 10326 | |
| STK38 (NDR1) | NDR | AGC | 6bxi | B | | phosphoaminophosphonic acid-adenylate ester | Human | 10325 | |
| AKT1 | Akt | AGC | 6hhi | A | | ~{n}-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]-3-(propanoylamino)benzamide | Human | 10913 | |
| PRKCB (PKCb) | PKC | AGC | 8se4 | A | | - | Human | 16137 | |
| PRKCB (PKCb) | PKC | AGC | 8se3 | A | | - | Human | 16138 | |
| GRK5 (GPRK5) | GRK | AGC | 9brm | A | | (3z)-3-[(4-{[(2s)-2-hydroxy-2-(oxan-4-yl)ethyl]carbamoyl}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16142 | |
| GRK5 (GPRK5) | GRK | AGC | 9ckq | A | | - | Human | 16143 | |
| GRK5 (GPRK5) | GRK | AGC | 6pjx | A | B | sangivamycin | Human | 13041 | |
| GRK5 (GPRK5) | GRK | AGC | 4tnb | A | | sangivamycin | Human | 3276 | |
| GRK5 (GPRK5) | GRK | AGC | 9brh | A | | (3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-({4-[(furan-3-carbonyl)amino]-3,5-dimethyl-1h-pyrrol-2-yl}methylidene)-2-oxo-3,7-dihydro-2h-indole-5-carboxamide | Human | 16144 | |
| GRK5 (GPRK5) | GRK | AGC | 9bre | A | | (3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-[(4-{[(2s)-2-(furan-2-yl)-2-hydroxyacetyl]amino}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 16145 | |
| GRK5 (GPRK5) | GRK | AGC | 9cks | A | | adenosine-5'-triphosphate | Human | 16146 | |
| PRKCB (PKCb) | PKC | AGC | 8se1 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 16139 | |
| GRK5 (GPRK5) | GRK | AGC | 9bri | A | | (3z)-3-[(3,5-dimethyl-4-{[(2s)-5-oxooxolane-2-carbonyl]amino}-1h-pyrrol-2-yl)methylidene]-n-[(1r)-1-(4-fluorophenyl)ethyl]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 16147 | |
| GRK5 (GPRK5) | GRK | AGC | 9brg | A | | (3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-({4-[(furan-2-carbonyl)amino]-3,5-dimethyl-1h-pyrrol-2-yl}methylidene)-2-oxo-3,7-dihydro-2h-indole-5-carboxamide | Human | 16148 | |
| GRK5 (GPRK5) | GRK | AGC | 9brl | A | | (3z)-3-({3,5-dimethyl-4-[(4-methylpiperidin-4-yl)carbamoyl]-1h-pyrrol-2-yl}methylidene)-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16149 | |
| GRK5 (GPRK5) | GRK | AGC | 9cko | A | A | sangivamycin | Human | 16150 | |
| GRK5 (GPRK5) | GRK | AGC | 9brj | A | | (4s)-n-{5-[(z)-(5-{[(1r)-1-(4-fluorophenyl)ethyl]carbamoyl}-2-oxo-2,7-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrol-3-yl}-2-methylimidazo[1,2-a]pyridine-3-carboxamide | Human | 16151 | |
| GRK5 (GPRK5) | GRK | AGC | 9cko | A | B | sangivamycin | Human | 16152 | |
| GRK5 (GPRK5) | GRK | AGC | 9mx2 | A | | sangivamycin | Human | 16153 | |
| GRK5 (GPRK5) | GRK | AGC | 9bro | A | | (3z)-3-[(4-{[(2s)-1-methoxypropan-2-yl]carbamoyl}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16154 | |
| GRK5 (GPRK5) | GRK | AGC | 9brf | A | | (3z)-3-{[3,5-dimethyl-4-(2-oxo-2-phenylacetamido)-1h-pyrrol-2-yl]methylidene}-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16155 | |
| GRK5 (GPRK5) | GRK | AGC | 9brn | A | | (3z)-3-[(4-{[2-(dimethylamino)ethyl]carbamoyl}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16156 | |
| GRK5 (GPRK5) | GRK | AGC | 9brk | A | | tert-butyl (3r)-3-({5-[(z)-(5-{[(1r)-1-(4-fluorophenyl)ethyl]carbamoyl}-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrol-3-yl}carbamoyl)piperazine-1-carboxylate | Human | 16157 | |
| GRK5 (GPRK5) | GRK | AGC | 9brp | A | | (3z)-3-[(4-{[(2r)-2-methoxypropyl]carbamoyl}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-n-[(1r)-1-phenylethyl]-3,7-dihydro-2h-indole-5-carboxamide | Human | 16158 | |
| AKT2 | Akt | AGC | 3e87 | B | B | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | 1903 | |
| AKT2 | Akt | AGC | 3e87 | B | A | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | 1909 | |
| AKT2 | Akt | AGC | 1o6k | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1923 | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9k | B | | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 5987 | |
| PRKG1 (PKG1) | PKG | AGC | 7lv3 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14343 | |
| PRKCH (PKCh) | PKC | AGC | 8fp3 | A | B | (3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | Human | 14695 | |
| PRKCH (PKCh) | PKC | AGC | 8fp3 | A | A | (3p)-3-{4-[(3r,5s)-3-amino-5-methylpiperidin-1-yl]-6-chloro-7h-pyrrolo[2,3-d]pyrimidin-5-yl}benzonitrile | Human | 14696 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5hng | A | | 6-methoxy-2-(1h-pyrazol-5-yl)-1h-benzimidazole | Human | 6675 | |
| AKT2 | Akt | AGC | 2x39 | A | | 4-amino-n-(4-chlorobenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | 1913 | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9l | A | B | 4,4'-(1h-pyrazole-3,4-diyl)diphenol | Human | 5989 | |
| GRK4 (GPRK4) | GRK | AGC | 4yhj | A | | amp phosphoramidate | Human | 422 | |
| GRK4 (GPRK4) | GRK | AGC | 4yhj | B | | amp phosphoramidate | Human | 423 | |
| PRKCA (PKCa) | PKC | AGC | 8u37 | A | B | (6m)-3-amino-n-{4-[(3r,4s)-4-amino-3-methoxypiperidin-1-yl]pyridin-3-yl}-6-[3-(trifluoromethoxy)pyridin-2-yl]pyrazine-2-carboxamide | Human | 15162 | |
| AKT2 | Akt | AGC | 9c1w | A | | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15393 | |
| AKT1 | Akt | AGC | 7nh4 | A | A | ~{n}-[3-[1-[[4-[5-(hydroxymethyl)-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 13865 | |
| AKT1 | Akt | AGC | 8uvy | A | A | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15378 | |
| AKT1 | Akt | AGC | 8uvy | A | B | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15381 | |
| AKT1 | Akt | AGC | 7nh5 | A | B | ~{n}-methyl-6-[4-[[4-[2-oxidanylidene-6-(propanoylamino)-3~{h}-benzimidazol-1-yl]piperidin-1-yl]methyl]phenyl]-5-phenyl-pyridine-3-carboxamide | Human | 13868 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu3 | A | A | (9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dione | Human | 3180 | |
| RPS6KA5 (MSK1) | RSK | AGC | 1vzo | A | A | - | Human | 108 | |
| PRKACA (PKACa) | PKA | AGC | 5n23 | A | A | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 9747 | |
| PRKACA (PKACa) | PKA | AGC | 7y1g | A | B | 1-chloranyl-~{n}-[(~{s})-(3-chloranyl-4-cyano-phenyl)-[(2~{r},4~{s})-4-oxidanylpyrrolidin-2-yl]methyl]-7-methoxy-isoquinoline-6-carboxamide | Human | 14423 | |
| AKT1 | Akt | AGC | 8uw7 | A | B | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15382 | |
| AKT1 | Akt | AGC | 8uw7 | A | A | 4-{2-[({4-[(2p)-2-(2-aminopyridin-3-yl)-5-phenyl-3h-imidazo[4,5-b]pyridin-3-yl]phenyl}methyl)amino]ethyl}-2-hydroxybenzaldehyde | Human | 15385 | |
| PRKCA (PKCa) | PKC | AGC | 8uak | A | B | (6m)-3-amino-n-[3-(4-amino-4-methylpiperidin-1-yl)pyridin-2-yl]-6-[3-(trifluoromethyl)pyridin-2-yl]pyrazine-2-carboxamide | Human | 15160 | |
| PRKCI (PKCi) | PKC | AGC | 9ejk | B | | - | Human | 15444 | |
| PRKCI (PKCi) | PKC | AGC | 8r3x | A | B | - | Human | 15445 | |
| PRKACA (PKACa) | PKA | AGC | 3poo | A | B | n'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5285 | |
| PRKCI (PKCi) | PKC | AGC | 9ejm | B | | adenosine-5'-diphosphate | Human | 15446 | |
| PRKCI (PKCi) | PKC | AGC | 9ejl | B | | - | Human | 15447 | |
| PRKCI (PKCi) | PKC | AGC | 8r3x | A | A | - | Human | 15448 | |
| AKT2 | Akt | AGC | 1mry | A | | - | Human | 1907 | |
| PRKCI (PKCi) | PKC | AGC | 5li9 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 7068 | |
| RPS6KA2 (RSK1) | RSK | AGC | 8xov | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15216 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4u | A | A | - | Human | 14788 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4u | A | B | - | Human | 14789 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4v | A | B | - | Human | 14792 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4w | A | B | - | Human | 14793 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4t | A | A | adenosine-5'-triphosphate | Human | 14791 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4w | A | A | - | Human | 14794 | |
| PRKG1 (PKG1) | PKG | AGC | 7t4t | A | B | adenosine-5'-triphosphate | Human | 14795 | |
| ROCK1 | DMPK | AGC | 5wnf | A | B | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10444 | |
| ROCK1 | DMPK | AGC | 2etr | B | | (r)-trans-4-(1-aminoethyl)-n-(4-pyridyl) cyclohexanecarboxamide | Human | 2704 | |
| ROCK1 | DMPK | AGC | 3d9v | A | | (s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazine | Human | 2696 | |
| ROCK1 | DMPK | AGC | 5wnh | B | | (2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide | Human | 10449 | |
| ROCK1 | DMPK | AGC | 3ncz | D | | cis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamide | Human | 2724 | |
| AKT1 | Akt | AGC | 9tmz | A | B | ~{n}-[2-oxidanylidene-3-[1-[[4-[3-phenyl-5-[(2-propan-2-ylpyrazol-3-yl)methyl]pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-1~{h}-benzimidazol-5-yl]propanamide | Human | 15711 | |
| AKT1 | Akt | AGC | 9tmv | A | A | ~{n}-[3-[1-[[4-[5-[(3-ethyl-1-methyl-pyrazol-4-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15728 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 7n91 | A | | 4-{[(1s)-1-(3-fluorophenyl)-2-(methylamino)ethyl]amino}quinazoline-8-carboxamide | Human | 14284 | |
| GRK2 (BARK1) | GRK | AGC | 5uvc | A | | n-benzyl-3-({[5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)benzamide | Human | 8256 | |
| GRK2 (BARK1) | GRK | AGC | 5he1 | A | B | (4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamide | Human | 6606 | |
| GRK2 (BARK1) | GRK | AGC | 5ukk | A | B | 5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamide | Human | 7530 | |
| GRK2 (BARK1) | GRK | AGC | 7pwd | A | A | 4-chloranyl-n-[2-(4-chlorophenyl)ethyl]thieno[2,3-c]pyridine-2-carboxamide | Human | 13949 | |
| GRK2 (BARK1) | GRK | AGC | 7pwd | A | B | 4-chloranyl-n-[2-(4-chlorophenyl)ethyl]thieno[2,3-c]pyridine-2-carboxamide | Human | 13950 | |
| GRK2 (BARK1) | GRK | AGC | 7k7l | A | A | 3-benzyl-6-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | 12960 | |
| GRK2 (BARK1) | GRK | AGC | 5wg3 | A | | 2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(1h-pyrazol-3-yl)methyl]benzamide | Human | 9439 | |
| GRK2 (BARK1) | GRK | AGC | 3krw | A | | balanol | Human | 1707 | |
| GRK2 (BARK1) | GRK | AGC | 4mk0 | A | B | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-one | Human | 1704 | |
| GRK2 (BARK1) | GRK | AGC | 4pnk | A | A | (4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide | Human | 1703 | |
| GRK2 (BARK1) | GRK | AGC | 6c2y | A | | (4r,5r,6s)-4-[4-fluoro-3-({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}carbamoyl)phenyl]-n-(2h-indazol-5-yl)-6-methyl-2-oxohexahydropyrimidine-5-carboxamide | Human | 9854 | |
| PKN1 | PKN | AGC | 4oth | A | B | - | Human | 7204 | |
| PKN1 | PKN | AGC | 4otd | A | A | - | Human | 545 | |
| GRK2 (BARK1) | GRK | AGC | 5uuu | A | B | 3-({[4-methyl-5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)-n-[2-(trifluoromethyl)benzyl]benzamide | Human | 8254 | |
| GRK2 (BARK1) | GRK | AGC | 4pnk | A | B | (4s)-4-(4-fluorophenyl)-n-(2h-indazol-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide | Human | 1708 | |
| GRK2 (BARK1) | GRK | AGC | 5wg5 | A | A | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazole | Human | 9437 | |
| PKN1 | PKN | AGC | 4oth | A | A | - | Human | 7203 | |
| PKN1 | PKN | AGC | 4otg | A | A | lestaurtinib | Human | 548 | |
| ROCK2 | DMPK | AGC | 7p6p | A | | ~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-yl-cyclohexane-1-carboxamide | Human | 15972 | |
| ROCK1 | DMPK | AGC | 7s25 | A | A | 2-[3-(methoxymethyl)phenyl]-n-[4-(1h-pyrazol-4-yl)phenyl]acetamide | Human | 14435 | |
| ROCK1 | DMPK | AGC | 7s26 | A | | 2-[methyl(phenyl)amino]-1-[4-(1h-pyrrolo[2,3-b]pyridin-3-yl)-3,6-dihydropyridin-1(2h)-yl]ethan-1-one | Human | 14437 | |
| ROCK1 | DMPK | AGC | 5wnf | D | A | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10451 | |
| PRKCB (PKCb) | PKC | AGC | 9s9t | A | | (9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dione | Human | 16135 | |
| PRKCB (PKCb) | PKC | AGC | 8se2 | A | | - | Human | 16136 | |
| ROCK1 | DMPK | AGC | 9q8r | A | | (7~{s})-7-(2,3-dihydro-1~{h}-inden-2-yl)-2-(hydroxymethyl)-~{n}-isoquinolin-6-yl-5-methyl-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxamide | Human | 16202 | |
| ROCK2 | DMPK | AGC | 6p5p | A | | 2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11914 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 10666 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw5 | A | A | 7-(2-fluoro-6-methoxyphenyl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | 134 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 10667 | |
| PRKACA (PKACa) | PKA | AGC | 5uzk | A | A | 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(1h-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide | Human | 9726 | |
| GRK6 (GPRK6) | GRK | AGC | 3nyo | A | | adenosine monophosphate | Human | 418 | |
| GRK6 (GPRK6) | GRK | AGC | 3nyo | B | | adenosine monophosphate | Human | 421 | |
| GRK6 (GPRK6) | GRK | AGC | 3nyn | A | | sangivamycin | Human | 419 | |
| GRK6 (GPRK6) | GRK | AGC | 2acx | B | | phosphoaminophosphonic acid-adenylate ester | Human | 417 | |
| GRK6 (GPRK6) | GRK | AGC | 3nyn | B | | sangivamycin | Human | 416 | |
| ROCK1 | DMPK | AGC | 5wne | C | | 3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamide | Human | 10462 | |
| ROCK1 | DMPK | AGC | 4w7p | C | | n~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamine | Human | 2688 | |
| ROCK1 | DMPK | AGC | 5bml | A | | n-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-{3-[(methylsulfonyl)amino]phenyl}acetamide | Human | 2713 | |
| ROCK1 | DMPK | AGC | 4yvc | A | | 2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamide | Human | 2715 | |
| ROCK1 | DMPK | AGC | 5wne | D | | 3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamide | Human | 10445 | |
| ROCK1 | DMPK | AGC | 3ndm | B | | (3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamide | Human | 2698 | |
| ROCK1 | DMPK | AGC | 5hvu | B | | 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 7415 | |
| ROCK2 | DMPK | AGC | 7p6n | A | | ~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]-4-pyridin-4-yl-piperidine-1-carboxamide | Human | 14314 | |
| ROCK1 | DMPK | AGC | 3ncz | A | | cis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamide | Human | 2699 | |
| PRKCI (PKCi) | PKC | AGC | 5lih | B | B | adenosine-5'-diphosphate | Human | 7073 | |
| PRKCI (PKCi) | PKC | AGC | 3a8x | B | | - | Human | 3348 | |
| PRKCI (PKCi) | PKC | AGC | 5li1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 7067 | |
| MASTL | MAST | AGC | 5loh | A | B | staurosporine | Human | 7085 | |
| MASTL | MAST | AGC | 5loh | A | A | staurosporine | Human | 7086 | |
| ROCK1 | DMPK | AGC | 5kks | B | | 2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8181 | |
| ROCK1 | DMPK | AGC | 5kkt | A | | 2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8182 | |
| AKT2 | Akt | AGC | 8q61 | A | A | 6-[4-(1-azanyl-3-methyl-3-oxidanyl-cyclobutyl)phenyl]-7-phenyl-1-propyl-pyrido[2,3-b][1,4]oxazin-2-one | Human | 14978 | |
| ROCK1 | DMPK | AGC | 3tv7 | B | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2703 | |
| ROCK1 | DMPK | AGC | 6e9w | A | | n-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamide | Human | 10691 | |
| PRKACA (PKACa) | PKA | AGC | 4wb7 | A | B | adenosine-5'-triphosphate | Human | 6878 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 10670 | |
| PRKG1 (PKG1) | PKG | AGC | 6bdl | B | A | - | Human | 10643 | |
| PRKACA (PKACa) | PKA | AGC | 6c0u | A | | n-[(3r,4r)-4-{[4-(2-fluoro-3-methoxy-6-propoxybenzene-1-carbonyl)benzene-1-carbonyl]amino}pyrrolidin-3-yl]-1h-indazole-5-carboxamide | Human | 9974 | |
| ROCK1 | DMPK | AGC | 7s25 | A | B | 2-[3-(methoxymethyl)phenyl]-n-[4-(1h-pyrazol-4-yl)phenyl]acetamide | Human | 14436 | |
| PRKACA (PKACa) | PKA | AGC | 5izf | A | | - | Human | 6854 | |
| ROCK1 | DMPK | AGC | 2etr | A | | (r)-trans-4-(1-aminoethyl)-n-(4-pyridyl) cyclohexanecarboxamide | Human | 2700 | |
| PRKACA (PKACa) | PKA | AGC | 3l9l | B | | 5-[2-({(2s)-2-amino-3-[4-(trifluoromethyl)phenyl]propyl}amino)-1,3-thiazol-5-yl]-1,3-dihydro-2h-indol-2-one | Human | 5302 | |
| ROCK1 | DMPK | AGC | 2v55 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2694 | |
| PDPK1 (PDK1) | PDK1 | AGC | 8dqt | A | | - | Human | 14812 | |
| PRKACA (PKACa) | PKA | AGC | 5j5x | A | C | - | Human | 6852 | |
| PRKG1 (PKG1) | PKG | AGC | 6bdl | B | B | - | Human | 10642 | |
| PRKCH (PKCh) | PKC | AGC | 3txo | A | | 2-methyl-n~1~-[3-(pyridin-4-yl)-2,6-naphthyridin-1-yl]propane-1,2-diamine | Human | 2316 | |
| ROCK1 | DMPK | AGC | 4yve | A | | 2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 2693 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | C | | - | Human | 3245 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcy | A | A | (2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamide | Human | 3151 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcx | A | A | 6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amine | Human | 3187 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqk | A | A | adenosine-5'-triphosphate | Human | 3175 | |
| AKT1 | Akt | AGC | 7apj | A | | - | Human | 13854 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4a06 | A | B | adenosine-5'-triphosphate | Human | 3227 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | D | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3184 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3rcj | A | | 3-(1-benzyl-1h-1,2,3-triazol-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 3154 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3ion | A | | 2-(5-{[(2s)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amine | Human | 3218 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ho7 | A | A | 5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamide | Human | 6673 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2pe0 | A | | 5-hydroxy-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-2-one | Human | 3206 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvp | B | | adenosine-5'-triphosphate | Human | 7113 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nuu | A | A | 3,4-dihydroisoquinolin-1(2h)-one | Human | 3214 | |
| ROCK2 | DMPK | AGC | 7jnt | G | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12767 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcq | A | A | 6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamine | Human | 3205 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu8 | A | B | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3237 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ho7 | A | B | 5-amino-3-(methylsulfanyl)-1h-pyrazole-1,4-dicarboxamide | Human | 6671 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 10672 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 7n93 | A | A | 4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamide | Human | 14285 | |
| DMPK (DMPK1) | DMPK | AGC | 2vd5 | A | | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 1901 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | B | A | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3356 | |
| PRKG1 (PKG1) | PKG | AGC | 6bg2 | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 10669 | |
| PRKCI (PKCi) | PKC | AGC | 3a8x | A | | - | Human | 3351 | |
| MASTL | MAST | AGC | 5loh | B | A | staurosporine | Human | 7088 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcy | A | B | (2s)-4-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-n-phenylmorpholine-2-carboxamide | Human | 3161 | |
| ROCK1 | DMPK | AGC | 4w7p | B | | n~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamine | Human | 2708 | |
| GRK5 (GPRK5) | GRK | AGC | 8uaq | A | | (3z)-n-[(1r)-1-(4-fluorophenyl)ethyl]-3-[(4-{[(2s)-2-(furan-2-yl)-2-hydroxyacetyl]amino}-3,5-dimethyl-1h-pyrrol-2-yl)methylidene]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 15092 | |
| GRK5 (GPRK5) | GRK | AGC | 8uap | A | | (3z)-3-{[4-(2-chloroacetamido)-3,5-dimethyl-1h-pyrrol-2-yl]methylidene}-n-[(1r)-1-(4-fluorophenyl)ethyl]-2-oxo-2,3-dihydro-1h-indole-5-carboxamide | Human | 15093 | |
| ROCK2 | DMPK | AGC | 7jnt | C | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12745 | |
| ROCK2 | DMPK | AGC | 5u7r | C | | (1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-one | Human | 7983 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nun | A | B | 6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amine | Human | 3216 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvl | A | A | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | 7106 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nuy | A | B | quinazolin-4(1h)-one | Human | 3242 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcs | A | B | 6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amine | Human | 3157 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvp | A | | adenosine-5'-triphosphate | Human | 7102 | |
| ROCK2 | DMPK | AGC | 4wot | A | | methyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoate | Human | 6827 | |
| ROCK2 | DMPK | AGC | 7jnt | F | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12758 | |
| ROCK2 | DMPK | AGC | 6p5p | D | | 2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11918 | |
| ROCK2 | DMPK | AGC | 5u7q | A | | - | Human | 7988 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd3 | A | A | tert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamate | Human | 3188 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uvr | A | | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3193 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3rwp | A | A | [4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanone | Human | 3208 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2biy | A | A | adenosine-5'-triphosphate | Human | 3232 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4ct2 | A | A | adenosine-5'-triphosphate | Human | 3153 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | D | | - | Human | 3210 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqv | A | B | adenosine-5'-triphosphate | Human | 3182 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4xx9 | A | B | adenosine-5'-triphosphate | Human | 6192 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvm | A | C | adenine | Human | 7138 | |
| ROCK1 | DMPK | AGC | 5wnh | C | | (2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide | Human | 10456 | |
| ROCK2 | DMPK | AGC | 7jov | E | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12762 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu7 | A | | 3-(1h-indol-3-yl)-4-(1-{2-[(2s)-1-methylpyrrolidinyl]ethyl}-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3224 | |
| ROCK2 | DMPK | AGC | 7jov | G | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12763 | |
| ROCK2 | DMPK | AGC | 5u7q | C | | - | Human | 7987 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | E | | - | Human | 3202 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | B | B | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 9256 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4aw1 | A | A | adenosine-5'-triphosphate | Human | 3229 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd3 | A | B | tert-butyl {(3r,6s)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methylpiperidin-3-yl}carbamate | Human | 3171 | |
| ROCK2 | DMPK | AGC | 5u7q | D | | - | Human | 7986 | |
| ROCK2 | DMPK | AGC | 7jov | D | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12764 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4aw1 | A | B | adenosine-5'-triphosphate | Human | 3221 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3rwq | A | | [4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[2-(pyridin-3-yl)ethyl]amino}pyrazin-2-yl)methanone | Human | 3213 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd0 | A | A | (3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamide | Human | 3196 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3sc1 | A | | 6-[2-(hydroxymethyl)phenyl]isoquinolin-1(2h)-one | Human | 3173 | |
| ROCK2 | DMPK | AGC | 4wot | B | | methyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoate | Human | 6829 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | D | B | staurosporine | Human | 4687 | |
| PKN1 | PKN | AGC | 4oti | A | A | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 551 | |
| PKN1 | PKN | AGC | 4oti | A | B | 3-{(3r,4r)-4-methyl-3-[methyl(7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]piperidin-1-yl}-3-oxopropanenitrile | Human | 547 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvl | A | B | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | 7110 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 3tku | B | | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 4859 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | C | B | staurosporine | Human | 4694 | |
| ROCK2 | DMPK | AGC | 5u7r | B | | (1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-one | Human | 7984 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | D | A | staurosporine | Human | 4688 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | F | A | staurosporine | Human | 4691 | |
| ROCK1 | DMPK | AGC | 5wng | A | | (2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamide | Human | 10459 | |
| ROCK1 | DMPK | AGC | 5wnf | B | B | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10450 | |
| ROCK1 | DMPK | AGC | 3twj | D | | - | Human | 2690 | |
| ROCK1 | DMPK | AGC | 4w7p | A | | n~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamine | Human | 2721 | |
| AKT1 | Akt | AGC | 9tn2 | A | A | ~{n}-[3-[1-[[4-[5-[(2-cyclobutylpyrazol-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15707 | |
| AKT1 | Akt | AGC | 3qkk | A | | n-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(2r)-6-hydroxy-4-oxo-3,4-dihydro-1'h-spiro[chromene-2,3'-piperidin]-1'-yl]propyl}-2,6-dimethylbenzenesulfonamide | Human | 2535 | |
| AKT1 | Akt | AGC | 3qkl | A | | n-{(2s)-3-[(3s)-8',9'-dihydro-1h,3'h-spiro[piperidine-3,7'-pyrano[3,2-e]indazol]-1-yl]-2-hydroxypropyl}-n-(2-ethoxyethyl)-2,6-dimethylbenzenesulfonamide | Human | 2544 | |
| AKT1 | Akt | AGC | 3ow4 | B | | (2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amine | Human | 2533 | |
| AKT1 | Akt | AGC | 6ccy | A | B | (5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-one | Human | 9869 | |
| AKT1 | Akt | AGC | 9tmw | A | A | ~{n}-[3-[1-[[4-[5-[(3-ethyl-1-methyl-pyrazol-4-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15708 | |
| AKT1 | Akt | AGC | 9tmy | A | A | ~{n}-[3-[1-[[4-[5-[(2-ethylpyrazol-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15709 | |
| AKT1 | Akt | AGC | 3qkm | A | | n-(2-ethoxyethyl)-n-{(2s)-2-hydroxy-3-[(5r)-2-(quinazolin-4-yl)-2,7-diazaspiro[4.5]dec-7-yl]propyl}-2,6-dimethylbenzenesulfonamide | Human | 2546 | |
| AKT1 | Akt | AGC | 9tn1 | A | B | ~{n}-[3-[1-[[4-[5-[(2-methylpyridin-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15710 | |
| AKT1 | Akt | AGC | 3cqw | A | A | 5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine | Human | 6763 | |
| AKT1 | Akt | AGC | 4gv1 | A | B | 4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | 2536 | |
| AKT1 | Akt | AGC | 6npz | A | B | - | Human | 10882 | |
| AKT1 | Akt | AGC | 9tmz | A | A | ~{n}-[2-oxidanylidene-3-[1-[[4-[3-phenyl-5-[(2-propan-2-ylpyrazol-3-yl)methyl]pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-1~{h}-benzimidazol-5-yl]propanamide | Human | 15713 | |
| AKT1 | Akt | AGC | 3ocb | B | | (2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amine | Human | 2534 | |
| AKT1 | Akt | AGC | 9zbk | E | | - | Human | 15714 | |
| AKT1 | Akt | AGC | 9tn4 | A | A | ~{n}-[3-[1-[[4-[5-[(6-azanyl-2-methyl-pyridin-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15715 | |
| AKT1 | Akt | AGC | 9tn1 | A | A | ~{n}-[3-[1-[[4-[5-[(2-methylpyridin-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15716 | |
| AKT1 | Akt | AGC | 3ocb | A | | (2s)-2-(4-chlorobenzyl)-3-oxo-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperazin-1-yl]propan-1-amine | Human | 2548 | |
| AKT1 | Akt | AGC | 6buu | A | B | - | Human | 10433 | |
| AKT1 | Akt | AGC | 6hhg | A | | ~{n}-[2-chloranyl-5-[[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]carbamoylamino]phenyl]propanamide | Human | 10916 | |
| AKT1 | Akt | AGC | 6s9w | A | B | ~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 11747 | |
| AKT1 | Akt | AGC | 4ekl | A | | (2s)-2-(4-chlorophenyl)-1-{4-[(5r,7r)-7-hydroxy-5-methyl-6,7-dihydro-5h-cyclopenta[d]pyrimidin-4-yl]piperazin-1-yl}-3-(propan-2-ylamino)propan-1-one | Human | 2540 | |
| AKT1 | Akt | AGC | 9tmy | A | B | ~{n}-[3-[1-[[4-[5-[(2-ethylpyrazol-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15725 | |
| AKT1 | Akt | AGC | 3mv5 | A | B | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 2532 | |
| AKT1 | Akt | AGC | 3mvh | A | B | n-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamide | Human | 2531 | |
| AKT1 | Akt | AGC | 9tmt | A | B | ~{n}-[3-[1-[[4-[5-[(3,5-dimethyl-1~{h}-pyrazol-4-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]prop-2-enamide | Human | 15726 | |
| AKT1 | Akt | AGC | 3mvh | A | A | n-{[(3s)-3-amino-1-(5-ethyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-yl]methyl}-2,4-difluorobenzamide | Human | 2538 | |
| AKT1 | Akt | AGC | 9tn4 | A | B | ~{n}-[3-[1-[[4-[5-[(6-azanyl-2-methyl-pyridin-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15727 | |
| AKT1 | Akt | AGC | 9tmv | A | B | ~{n}-[3-[1-[[4-[5-[(3-ethyl-1-methyl-pyrazol-4-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15729 | |
| AKT1 | Akt | AGC | 6hhj | A | | ~{n}-[1-methyl-2-oxidanylidene-3-[1-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperidin-4-yl]benzimidazol-5-yl]propanamide | Human | 10914 | |
| PRKACA (PKACa) | PKA | AGC | 4wb8 | A | A | adenosine-5'-triphosphate | Human | 5304 | |
| PRKACA (PKACa) | PKA | AGC | 3vqh | A | A | n-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamide | Human | 5271 | |
| PRKACA (PKACa) | PKA | AGC | 3amb | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 5276 | |
| PRKACA (PKACa) | PKA | AGC | 6qj7 | A | B | ~{n}'-[(2~{s})-2-[3,5-bis(fluoranyl)phenyl]-2-oxidanyl-ethanoyl]-2-ethyl-3-methyl-4-oxidanyl-benzohydrazide | Human | 11991 | |
| PRKACA (PKACa) | PKA | AGC | 4uja | A | B | 7-{(3s,4r)-4-[(5-bromothiophen-2-yl)carbonyl]pyrrolidin-3-yl}quinazolin-4(3h)-one | Human | 6547 | |
| PRKACA (PKACa) | PKA | AGC | 9edc | A | A | adenosine-5'-triphosphate | Human | 15739 | |
| PRKACA (PKACa) | PKA | AGC | 6qj7 | A | A | ~{n}'-[(2~{s})-2-[3,5-bis(fluoranyl)phenyl]-2-oxidanyl-ethanoyl]-2-ethyl-3-methyl-4-oxidanyl-benzohydrazide | Human | 11990 | |
| PRKACA (PKACa) | PKA | AGC | 3mvj | B | | - | Human | 5288 | |
| PRKACA (PKACa) | PKA | AGC | 3oog | A | A | 1-(4-hydroxy-3-methylphenyl)ethanone | Human | 5281 | |
| PRKACA (PKACa) | PKA | AGC | 5izj | A | A | - | Human | 6857 | |
| PRKACA (PKACa) | PKA | AGC | 6no7 | A | | - | Human | 11465 | |
| PRKACA (PKACa) | PKA | AGC | 2gu8 | A | | n-[(1s)-2-amino-1-(2,4-dichlorobenzyl)ethyl]-5-[2-(methylamino)pyrimidin-4-yl]thiophene-2-carboxamide | Human | 5295 | |
| PRKACA (PKACa) | PKA | AGC | 6wjg | A | | - | Human | 13006 | |
| PRKACA (PKACa) | PKA | AGC | 9edc | A | B | adenosine-5'-triphosphate | Human | 15740 | |
| PRKACA (PKACa) | PKA | AGC | 4uj1 | A | | 7-[(3s,4r)-4-(3-chlorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6548 | |
| PRKACA (PKACa) | PKA | AGC | 3oxt | A | | (2s)-2-amino-n'-[(1e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-phenylethanehydrazide | Human | 5268 | |
| PRKACA (PKACa) | PKA | AGC | 3agm | A | | - | Human | 5282 | |
| PRKACA (PKACa) | PKA | AGC | 3ovv | A | B | n'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5269 | |
| PRKACA (PKACa) | PKA | AGC | 3agl | A | | (10r,20r,23r)-1-[(2s,3s,4r,5r)-5-(6-amino-9h-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]-20,23-bis(3-carbamimidamidopropyl)-10-methyl-1,8,11,18,21-pentaoxo-2,9,12,19,22-pentaazatetracosan-24-amide | Human | 5267 | |
| PRKACA (PKACa) | PKA | AGC | 4wb7 | B | B | adenosine-5'-triphosphate | Human | 6877 | |
| PRKACA (PKACa) | PKA | AGC | 8fec | A | | 6-[(6p)-6-(4-bromo-1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-7h-purine | Human | 14890 | |
| PRKACA (PKACa) | PKA | AGC | 4ae9 | B | B | - | Human | 5286 | |
| PRKACA (PKACa) | PKA | AGC | 3nx8 | A | B | - | Human | 5294 | |
| PRKACA (PKACa) | PKA | AGC | 5j5x | A | B | - | Human | 6856 | |
| PRKACA (PKACa) | PKA | AGC | 3ama | A | | 4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamide | Human | 5284 | |
| PRKACA (PKACa) | PKA | AGC | 4uj2 | A | B | 7-[(3s,4r)-4-(3-iodanylphenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6551 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | A | B | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3350 | |
| PRKCI (PKCi) | PKC | AGC | 3a8w | A | | adenosine-5'-triphosphate | Human | 3353 | |
| PRKG1 (PKG1) | PKG | AGC | 6bdl | A | B | - | Human | 10644 | |
| PRKCI (PKCi) | PKC | AGC | 6ilz | E | | 2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamide | Human | 11356 | |
| ROCK2 | DMPK | AGC | 7jnt | B | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12766 | |
| PKN2 | PKN | AGC | 4crs | A | | phosphothiophosphoric acid-adenylate ester | Human | 535 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | A | A | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 9254 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvp | C | | adenosine-5'-triphosphate | Human | 7111 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | B | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3160 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4ct1 | A | B | adenosine-5'-triphosphate | Human | 3168 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3hrf | A | B | adenosine-5'-triphosphate | Human | 3247 | |
| PRKCQ (PKCt) | PKC | AGC | 2jed | B | | 3-(8-dimethylaminomethyl-6,7,8,9-tetrahydro-pyrido[1,2-a]indol-10-yl)-4-(1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 5358 | |
| PRKCQ (PKCt) | PKC | AGC | 5f9e | B | A | 2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-one | Human | 6631 | |
| PRKCQ (PKCt) | PKC | AGC | 5f9e | B | B | 2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-one | Human | 6628 | |
| PRKCQ (PKCt) | PKC | AGC | 5f9e | A | B | 2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-one | Human | 6629 | |
| PRKCQ (PKCt) | PKC | AGC | 4ra5 | B | B | (1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5360 | |
| PRKCQ (PKCt) | PKC | AGC | 5f9e | A | A | 2,2-dimethyl-7-(2-oxidanylidene-3~{h}-imidazo[4,5-b]pyridin-1-yl)-1-(phenylmethyl)-3~{h}-quinazolin-4-one | Human | 6630 | |
| AKT2 | Akt | AGC | 2xh5 | A | | 4-(4-tert-butylbenzyl)-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-aminium | Human | 1924 | |
| AKT2 | Akt | AGC | 3e88 | A | | 4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1908 | |
| AKT2 | Akt | AGC | 2jdo | A | | isoquinoline-5-sulfonic acid (2-(2-(4-chlorobenzyloxy)ethylamino)ethyl)amide | Human | 1922 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a61 | A | | staurosporine | Human | 1846 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l45 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1850 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf5 | A | B | 4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | 1845 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf6 | A | B | 4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | 1859 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf7 | A | A | 1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamide | Human | 1854 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf8 | A | | 2-oxo-2-[(4-sulfamoylphenyl)amino]ethyl 7,8,9,10-tetrahydro-6h-cyclohepta[b]quinoline-11-carboxylate | Human | 1848 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a62 | A | | staurosporine | Human | 1867 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l46 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1847 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l3l | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1863 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l43 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1861 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3we4 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1860 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf5 | A | A | 4-[4-(1h-benzimidazol-2-yl)piperidin-1-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | 1857 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4rlp | A | | [(amino-kappan)methanethiolato](3-fluoro-9-methoxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(n-methyl-1,4,7-trithiecan-9-amine-kappa~3~s~1~,s~4~,s~7~)ruthenium | Human | 7219 | |
| GRK5 (GPRK5) | GRK | AGC | 9ckp | A | | sangivamycin | Human | 16141 | |
| GRK5 (GPRK5) | GRK | AGC | 9ckr | A | | adenosine-5'-triphosphate | Human | 16159 | |
| GRK2 (BARK1) | GRK | AGC | 7k7z | A | B | 3-benzyl-7-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | 12961 | |
| ROCK1 | DMPK | AGC | 5hvu | A | | 2-{3-[3-(piperidin-4-yl)propoxy]phenyl}-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 7414 | |
| ROCK1 | DMPK | AGC | 5wnf | D | B | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10452 | |
| ROCK1 | DMPK | AGC | 5wnf | B | A | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10463 | |
| ROCK1 | DMPK | AGC | 3twj | B | | - | Human | 2718 | |
| ROCK1 | DMPK | AGC | 5wne | A | | 3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamide | Human | 10446 | |
| ROCK1 | DMPK | AGC | 2etk | A | | 1-(1-hydroxy-5-isoquinolinesulfonyl)homopiperazine | Human | 2707 | |
| ROCK1 | DMPK | AGC | 2esm | A | | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 2726 | |
| ROCK1 | DMPK | AGC | 5wnf | C | B | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10460 | |
| ROCK1 | DMPK | AGC | 3ndm | D | | (3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamide | Human | 2705 | |
| ROCK1 | DMPK | AGC | 3tv7 | C | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2717 | |
| ROCK1 | DMPK | AGC | 7jou | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12768 | |
| ROCK1 | DMPK | AGC | 4yvc | B | | 2-fluoro-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]benzamide | Human | 2727 | |
| ROCK1 | DMPK | AGC | 3v8s | C | | 1-(1h-indazol-5-yl)-3-(2-phenylethyl)urea | Human | 2702 | |
| ROCK1 | DMPK | AGC | 3ncz | B | | cis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamide | Human | 2720 | |
| ROCK1 | DMPK | AGC | 5bml | B | | n-[4-(2-fluoropyridin-4-yl)thiophen-2-yl]-2-{3-[(methylsulfonyl)amino]phenyl}acetamide | Human | 2691 | |
| ROCK1 | DMPK | AGC | 5kkt | B | | 2-[3-[3-(4-methylpiperazin-1-yl)propoxy]phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8184 | |
| ROCK1 | DMPK | AGC | 3v8s | B | | 1-(1h-indazol-5-yl)-3-(2-phenylethyl)urea | Human | 2709 | |
| ROCK1 | DMPK | AGC | 3tv7 | D | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2725 | |
| ROCK1 | DMPK | AGC | 5wne | B | | 3,4-dimethoxy-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)benzamide | Human | 10453 | |
| ROCK1 | DMPK | AGC | 5wnh | D | | (2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide | Human | 10454 | |
| ROCK1 | DMPK | AGC | 5wnf | A | A | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10447 | |
| ROCK1 | DMPK | AGC | 3twj | C | | 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2689 | |
| ROCK1 | DMPK | AGC | 3ndm | C | | (3s,4r)-n-(7-chloro-1-oxo-1,4-dihydroisoquinolin-6-yl)-4-(4-chlorophenyl)pyrrolidine-3-carboxamide | Human | 2722 | |
| ROCK1 | DMPK | AGC | 3ndm | A | | - | Human | 2695 | |
| ROCK1 | DMPK | AGC | 2etk | B | | 1-(1-hydroxy-5-isoquinolinesulfonyl)homopiperazine | Human | 2723 | |
| DMPK (DMPK1) | DMPK | AGC | 2vd5 | B | | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1-methyl-1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 1902 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | A | A | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3349 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | B | B | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3347 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | C | B | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3352 | |
| PRKCI (PKCi) | PKC | AGC | 1zrz | A | | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3354 | |
| PRKCI (PKCi) | PKC | AGC | 3a8w | B | | adenosine-5'-triphosphate | Human | 3346 | |
| PRKCI (PKCi) | PKC | AGC | 5lih | A | B | adenosine-5'-diphosphate | Human | 7070 | |
| PRKCI (PKCi) | PKC | AGC | 6ilz | A | | 2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamide | Human | 11358 | |
| PRKCI (PKCi) | PKC | AGC | 5lih | A | A | adenosine-5'-diphosphate | Human | 7071 | |
| PRKCI (PKCi) | PKC | AGC | 3zh8 | C | A | (2s)-3-phenyl-n~1~-[2-(pyridin-4-yl)-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4-yl]propane-1,2-diamine | Human | 3355 | |
| PRKCI (PKCi) | PKC | AGC | 6ilz | G | | 2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamide | Human | 11355 | |
| PRKCI (PKCi) | PKC | AGC | 6ilz | C | | 2-amino-5-[3-(piperazin-1-yl)phenyl]-n-(pyridin-4-yl)pyridine-3-carboxamide | Human | 11357 | |
| PRKCI (PKCi) | PKC | AGC | 5li1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 7072 | |
| PRKCI (PKCi) | PKC | AGC | 5lih | B | A | adenosine-5'-diphosphate | Human | 7069 | |
| MASTL | MAST | AGC | 5loh | B | B | staurosporine | Human | 7087 | |
| RPS6KA3 (RSK2) | RSK | AGC | 8eq5 | A | A | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Human | 14713 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw6 | A | B | 7-(1h-benzimidazol-7-yl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | 136 | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9l | A | A | 4,4'-(1h-pyrazole-3,4-diyl)diphenol | Human | 5986 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw6 | A | A | 7-(1h-benzimidazol-7-yl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | 132 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nw5 | A | B | 7-(2-fluoro-6-methoxyphenyl)-n-(3,4,5-trimethoxyphenyl)-1,3-benzoxazol-2-amine | Human | 135 | |
| RPS6KA3 (RSK2) | RSK | AGC | 8r58 | A | A | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Human | 15478 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nus | A | B | 2,6-difluoro-4-{4-[4-(4-methylpiperazin-1-yl)phenyl]pyridin-3-yl}phenol | Human | 131 | |
| RPS6KA3 (RSK2) | RSK | AGC | 7opo | A | | phosphoaminophosphonic acid-adenylate ester | Human | 14079 | |
| RPS6KA3 (RSK2) | RSK | AGC | 8r58 | A | B | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Human | 15479 | |
| RPS6KA3 (RSK2) | RSK | AGC | 8eq5 | A | B | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4-oxo-4h-chromen-3-yl 6-deoxy-alpha-l-mannopyranoside | Human | 14714 | |
| RPS6KA3 (RSK2) | RSK | AGC | 5d9k | A | | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 5988 | |
| RPS6KA3 (RSK2) | RSK | AGC | 4nus | A | A | 2,6-difluoro-4-{4-[4-(4-methylpiperazin-1-yl)phenyl]pyridin-3-yl}phenol | Human | 133 | |
| RPS6KA1 (RSK3) | RSK | AGC | 2z7q | A | | phosphomethylphosphonic acid adenylate ester | Human | 2778 | |
| RPS6KA1 (RSK3) | RSK | AGC | 2z7s | A | | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 2776 | |
| RPS6KA1 (RSK3) | RSK | AGC | 2z7r | A | | staurosporine | Human | 2777 | |
| RPS6KA5 (MSK1) | RSK | AGC | 1vzo | A | B | - | Human | 107 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g77 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11005 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g78 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11010 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g76 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11006 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g78 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 11007 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g76 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 11008 | |
| RPS6KA6 (RSK4) | RSK | AGC | 6g77 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 11009 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | B | A | staurosporine | Human | 4692 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | A | A | staurosporine | Human | 4693 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | E | A | staurosporine | Human | 4689 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | E | B | staurosporine | Human | 4685 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | B | B | staurosporine | Human | 4695 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | F | B | staurosporine | Human | 4686 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | A | B | staurosporine | Human | 4690 | |
| STK32A (YANK1) | YANK | AGC | 4fr4 | C | A | staurosporine | Human | 4684 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 4ual | A | A | 4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamide | Human | 4861 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 3qfv | A | | 2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide | Human | 4860 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 5ote | A | | 2-[4-[(6~{s})-1,8-diazaspiro[5.5]undecan-8-yl]-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]-1,3-thiazole | Human | 9578 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 5otf | A | | (6~{s})-8-(3-pyrimidin-4-yl-1~{h}-pyrrolo[2,3-b]pyridin-4-yl)-1,8-diazaspiro[5.5]undecane | Human | 9577 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 3tku | A | | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 4862 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 4uak | A | A | adenosine-5'-diphosphate | Human | 4864 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 4ual | A | B | 4-chloro-1-(piperidin-4-yl)-n-[3-(pyridin-2-yl)-1h-pyrazol-4-yl]-1h-pyrazole-3-carboxamide | Human | 4858 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 3qfv | B | | 2-(carbamoylamino)-5-(4-fluorophenyl)thiophene-3-carboxamide | Human | 4857 | |
| CDC42BPB (MRCKb) | DMPK | AGC | 4uak | A | B | adenosine-5'-diphosphate | Human | 4863 | |
| AKT1 | Akt | AGC | 6npz | B | B | - | Human | 10879 | |
| AKT1 | Akt | AGC | 3mv5 | A | A | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 2537 | |
| AKT1 | Akt | AGC | 4ejn | A | | - | Human | 2542 | |
| AKT1 | Akt | AGC | 6buu | B | B | - | Human | 10439 | |
| AKT1 | Akt | AGC | 6hhf | A | | borussertib | Human | 10970 | |
| AKT1 | Akt | AGC | 9tn0 | A | A | ~{n}-[2-oxidanylidene-3-[1-[[4-[3-phenyl-5-[(2-propylpyrazol-3-yl)methyl]pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-1~{h}-benzimidazol-5-yl]propanamide | Human | 15717 | |
| AKT1 | Akt | AGC | 4gv1 | A | A | 4-amino-n-[(1s)-1-(4-chlorophenyl)-3-hydroxypropyl]-1-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)piperidine-4-carboxamide | Human | 2543 | |
| AKT1 | Akt | AGC | 3o96 | A | | - | Human | 2545 | |
| AKT1 | Akt | AGC | 3ow4 | A | | (2r)-3-(1h-indol-3-yl)-1-{4-[(5s)-5-methyl-5,7-dihydrothieno[3,4-d]pyrimidin-4-yl]piperazin-1-yl}-1-oxopropan-2-amine | Human | 2547 | |
| AKT1 | Akt | AGC | 7nh4 | A | B | ~{n}-[3-[1-[[4-[5-(hydroxymethyl)-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 13866 | |
| AKT1 | Akt | AGC | 6npz | A | A | - | Human | 10880 | |
| AKT1 | Akt | AGC | 6buu | A | C | - | Human | 10438 | |
| AKT1 | Akt | AGC | 3cqu | A | A | n-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6764 | |
| AKT1 | Akt | AGC | 6hhh | A | | ~{n}-[4-[4-[[4-(5-oxidanylidene-3-phenyl-6~{h}-1,6-naphthyridin-2-yl)phenyl]methyl]piperazin-1-yl]phenyl]propanamide | Human | 10915 | |
| AKT1 | Akt | AGC | 6npz | B | A | - | Human | 10881 | |
| AKT1 | Akt | AGC | 9tmt | A | A | ~{n}-[3-[1-[[4-[5-[(3,5-dimethyl-1~{h}-pyrazol-4-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]prop-2-enamide | Human | 15712 | |
| AKT1 | Akt | AGC | 6s9x | A | | ~{n}-[3-[1-[[4-[5-[(4-hydroxyphenyl)methyl]-6-oxidanylidene-2-phenyl-1~{h}-pyrazin-3-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 11746 | |
| AKT1 | Akt | AGC | 5kcv | A | | 3-[3-[4-(1-azanylcyclobutyl)phenyl]-5-phenyl-imidazo[4,5-b]pyridin-2-yl]pyridin-2-amine | Human | 6708 | |
| AKT1 | Akt | AGC | 7nh5 | A | A | ~{n}-methyl-6-[4-[[4-[2-oxidanylidene-6-(propanoylamino)-3~{h}-benzimidazol-1-yl]piperidin-1-yl]methyl]phenyl]-5-phenyl-pyridine-3-carboxamide | Human | 13867 | |
| AKT1 | Akt | AGC | 9tmu | A | B | ~{n}-[2-oxidanylidene-3-[1-[[4-[3-phenyl-5-[(1,3,5-trimethylpyrazol-4-yl)methyl]pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-1~{h}-benzimidazol-5-yl]propanamide | Human | 15718 | |
| AKT1 | Akt | AGC | 9tmu | A | A | ~{n}-[2-oxidanylidene-3-[1-[[4-[3-phenyl-5-[(1,3,5-trimethylpyrazol-4-yl)methyl]pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-1~{h}-benzimidazol-5-yl]propanamide | Human | 15719 | |
| AKT1 | Akt | AGC | 6buu | B | A | - | Human | 10430 | |
| AKT1 | Akt | AGC | 9tmw | A | B | ~{n}-[3-[1-[[4-[5-[(3-ethyl-1-methyl-pyrazol-4-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15720 | |
| AKT1 | Akt | AGC | 6buu | A | A | - | Human | 10432 | |
| AKT1 | Akt | AGC | 6s9w | A | A | ~{n}-[3-[1-[[4-(5-methyl-6-oxidanylidene-3-phenyl-1~{h}-pyrazin-2-yl)phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 11748 | |
| AKT1 | Akt | AGC | 9tn2 | A | B | ~{n}-[3-[1-[[4-[5-[(2-cyclobutylpyrazol-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15721 | |
| AKT1 | Akt | AGC | 9tn3 | A | A | ~{n}-[3-[1-[[4-[5-[(2-methylpyridin-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15722 | |
| AKT1 | Akt | AGC | 3cqw | A | B | 5-(5-chloro-7h-pyrrolo[2,3-d]pyrimidin-4-yl)-4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine | Human | 6765 | |
| AKT1 | Akt | AGC | 6ccy | A | A | (5r)-4-(4-{4-[4-fluoro-3-(trifluoromethyl)phenyl]-1-[2-(pyrrolidin-1-yl)ethyl]-1h-imidazol-2-yl}piperidin-1-yl)-5-methyl-5,8-dihydropyrido[2,3-d]pyrimidin-7(6h)-one | Human | 9868 | |
| AKT1 | Akt | AGC | 9tn3 | A | B | ~{n}-[3-[1-[[4-[5-[(2-methylpyridin-3-yl)methyl]-3-phenyl-pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-2-oxidanylidene-1~{h}-benzimidazol-5-yl]propanamide | Human | 15723 | |
| AKT1 | Akt | AGC | 4ekk | B | | phosphoaminophosphonic acid-adenylate ester | Human | 2539 | |
| AKT1 | Akt | AGC | 9tn0 | A | B | ~{n}-[2-oxidanylidene-3-[1-[[4-[3-phenyl-5-[(2-propylpyrazol-3-yl)methyl]pyridin-2-yl]phenyl]methyl]piperidin-4-yl]-1~{h}-benzimidazol-5-yl]propanamide | Human | 15724 | |
| AKT1 | Akt | AGC | 4ekk | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2541 | |
| AKT1 | Akt | AGC | 3cqu | A | B | n-[2-(5-methyl-4h-1,2,4-triazol-3-yl)phenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 6762 | |
| PRKACA (PKACa) | PKA | AGC | 5izj | A | B | - | Human | 6855 | |
| PRKACA (PKACa) | PKA | AGC | 5bx7 | A | A | 1-benzothiophen-3-ylmethanol | Human | 7076 | |
| PRKACA (PKACa) | PKA | AGC | 4wb5 | A | A | adenosine-5'-triphosphate | Human | 5280 | |
| PRKACA (PKACa) | PKA | AGC | 4wb7 | A | A | adenosine-5'-triphosphate | Human | 6876 | |
| PRKACA (PKACa) | PKA | AGC | 4ae9 | A | B | - | Human | 5307 | |
| PRKACA (PKACa) | PKA | AGC | 6no7 | G | | adenosine-5'-triphosphate | Human | 11464 | |
| PRKACA (PKACa) | PKA | AGC | 8fe5 | A | | 6-[(6p)-6-(1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-7,9-dihydro-8h-purin-8-one | Human | 14888 | |
| PRKACA (PKACa) | PKA | AGC | 5bx6 | A | B | 4-chlorophthalazin-1(2h)-one | Human | 7078 | |
| PRKACA (PKACa) | PKA | AGC | 6bys | G | | - | Human | 11260 | |
| PRKACA (PKACa) | PKA | AGC | 4ae9 | A | A | - | Human | 5265 | |
| PRKACA (PKACa) | PKA | AGC | 5n23 | A | B | 1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}urea | Human | 9746 | |
| PRKACA (PKACa) | PKA | AGC | 3agl | B | | (10r,20r,23r)-1-[(2s,3s,4r,5r)-5-(6-amino-9h-purin-9-yl)-3,4-dihydroxytetrahydrofuran-2-yl]-20,23-bis(3-carbamimidamidopropyl)-10-methyl-1,8,11,18,21-pentaoxo-2,9,12,19,22-pentaazatetracosan-24-amide | Human | 5283 | |
| PRKACA (PKACa) | PKA | AGC | 3l9m | B | | (2s)-n~1~-[5-(3-methyl-1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamine | Human | 5278 | |
| PRKACA (PKACa) | PKA | AGC | 4uj9 | A | | 7-[(3s,4r)-4-[4-(trifluoromethyl)phenyl]carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6544 | |
| PRKACA (PKACa) | PKA | AGC | 6bys | E | | - | Human | 11262 | |
| PRKACA (PKACa) | PKA | AGC | 5bx7 | A | B | 1-benzothiophen-3-ylmethanol | Human | 7077 | |
| PRKACA (PKACa) | PKA | AGC | 4uj2 | A | A | 7-[(3s,4r)-4-(3-iodanylphenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6550 | |
| PRKACA (PKACa) | PKA | AGC | 3owp | A | B | (2s)-2-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylethanehydrazide | Human | 5296 | |
| PRKACA (PKACa) | PKA | AGC | 6frx | A | | ~{n}-[3-[(5-chloranyl-2-phenylazanyl-pyrimidin-4-yl)amino]phenyl]prop-2-enamide | Human | 11261 | |
| PRKACA (PKACa) | PKA | AGC | 3nx8 | A | A | - | Human | 5277 | |
| PRKACA (PKACa) | PKA | AGC | 4ae6 | A | B | - | Human | 5301 | |
| PRKACA (PKACa) | PKA | AGC | 3l9n | A | | (2s)-n~1~-[5-(1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamine | Human | 5292 | |
| PRKACA (PKACa) | PKA | AGC | 4wb8 | A | B | adenosine-5'-triphosphate | Human | 5287 | |
| PRKACA (PKACa) | PKA | AGC | 6no7 | E | | adenosine-5'-triphosphate | Human | 11463 | |
| PRKACA (PKACa) | PKA | AGC | 5j5x | A | A | - | Human | 6853 | |
| PRKACA (PKACa) | PKA | AGC | 6bys | C | | - | Human | 11257 | |
| PRKACA (PKACa) | PKA | AGC | 5bx6 | A | A | 4-chlorophthalazin-1(2h)-one | Human | 7075 | |
| PRKACA (PKACa) | PKA | AGC | 3poo | A | A | n'-[(e)-(2,4-dihydroxy-6-methylphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5300 | |
| PRKACA (PKACa) | PKA | AGC | 9edd | A | | adenosine-5'-triphosphate | Human | 15741 | |
| PRKACA (PKACa) | PKA | AGC | 6byr | A | | adenosine-5'-triphosphate | Human | 11256 | |
| PRKACA (PKACa) | PKA | AGC | 5izj | B | A | - | Human | 6851 | |
| PRKACA (PKACa) | PKA | AGC | 7y1g | A | A | 1-chloranyl-~{n}-[(~{s})-(3-chloranyl-4-cyano-phenyl)-[(2~{r},4~{s})-4-oxidanylpyrrolidin-2-yl]methyl]-7-methoxy-isoquinoline-6-carboxamide | Human | 14422 | |
| PRKACA (PKACa) | PKA | AGC | 4wb5 | A | B | adenosine-5'-triphosphate | Human | 5306 | |
| PRKACA (PKACa) | PKA | AGC | 8fe2 | A | | 6-[(6m)-6-(1-methyl-1h-imidazol-5-yl)-2,3-dihydro-4h-1,4-thiazin-4-yl]-9h-purine | Human | 14889 | |
| PRKACA (PKACa) | PKA | AGC | 3oog | A | B | 1-(4-hydroxy-3-methylphenyl)ethanone | Human | 5272 | |
| PRKACA (PKACa) | PKA | AGC | 3l9m | A | | (2s)-n~1~-[5-(3-methyl-1h-indazol-5-yl)-1,3,4-thiadiazol-2-yl]-3-(4-methylphenyl)propane-1,2-diamine | Human | 5270 | |
| PRKACA (PKACa) | PKA | AGC | 4wb6 | B | | adenosine-5'-triphosphate | Human | 5293 | |
| PRKACA (PKACa) | PKA | AGC | 3mvj | E | | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 5291 | |
| PRKACA (PKACa) | PKA | AGC | 9ede | A | | adenosine-5'-triphosphate | Human | 15742 | |
| PRKACA (PKACa) | PKA | AGC | 3owp | A | A | (2s)-2-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylethanehydrazide | Human | 5273 | |
| PRKACA (PKACa) | PKA | AGC | 4ae6 | B | B | - | Human | 5298 | |
| PRKACA (PKACa) | PKA | AGC | 4wb7 | B | A | adenosine-5'-triphosphate | Human | 6875 | |
| PRKACA (PKACa) | PKA | AGC | 5izj | B | B | - | Human | 6858 | |
| PRKACA (PKACa) | PKA | AGC | 9dc6 | A | | n-(2-aminoethyl)-4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-3,4-dihydro-2h-1,4-thiazine-6-carboxamide | Human | 15743 | |
| PRKACA (PKACa) | PKA | AGC | 6bys | A | | - | Human | 11259 | |
| PRKACA (PKACa) | PKA | AGC | 4ae9 | B | A | - | Human | 5299 | |
| PRKACA (PKACa) | PKA | AGC | 4ae6 | A | A | - | Human | 5274 | |
| PRKACA (PKACa) | PKA | AGC | 3mvj | A | | (3r)-1-(5-methyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyrrolidin-3-amine | Human | 5289 | |
| PRKACA (PKACa) | PKA | AGC | 3ovv | A | A | n'-[(1e)-(4-hydroxyphenyl)methylidene]-2-(3-methoxyphenyl)acetohydrazide | Human | 5266 | |
| PRKACA (PKACa) | PKA | AGC | 3p0m | A | A | (2r)-4-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylbutanehydrazide | Human | 5297 | |
| PRKACA (PKACa) | PKA | AGC | 6byr | C | | adenosine-5'-triphosphate | Human | 11258 | |
| PRKACA (PKACa) | PKA | AGC | 4ujb | A | B | 7-[(3s,4r)-4-(3-fluorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6545 | |
| PRKACA (PKACa) | PKA | AGC | 3vqh | A | B | n-[2-(4-bromocinnamylamino)ethyl]-5-isoquinoline sulfonamide | Human | 5275 | |
| PRKACA (PKACa) | PKA | AGC | 6wjf | A | | - | Human | 13008 | |
| PRKACA (PKACa) | PKA | AGC | 6wjf | B | | - | Human | 13009 | |
| PRKACA (PKACa) | PKA | AGC | 3l9l | A | | 5-[2-({(2s)-2-amino-3-[4-(trifluoromethyl)phenyl]propyl}amino)-1,3-thiazol-5-yl]-1,3-dihydro-2h-indol-2-one | Human | 5305 | |
| PRKACA (PKACa) | PKA | AGC | 3p0m | A | B | (2r)-4-amino-n'-[(1e)-(3-bromo-4-hydroxyphenyl)methylidene]-2-phenylbutanehydrazide | Human | 5279 | |
| PRKACA (PKACa) | PKA | AGC | 4ae6 | B | A | - | Human | 5290 | |
| PRKACA (PKACa) | PKA | AGC | 4wb6 | A | | adenosine-5'-triphosphate | Human | 5303 | |
| PRKACA (PKACa) | PKA | AGC | 8x5l | A | | (2s)-2-(4-chlorophenyl)-2-hydroxy-2-[4-(1h-pyrazol-4-yl)phenyl]ethanaminium | Human | 15111 | |
| PRKACA (PKACa) | PKA | AGC | 4ujb | A | A | 7-[(3s,4r)-4-(3-fluorophenyl)carbonylpyrrolidin-3-yl]-3h-quinazolin-4-one | Human | 6546 | |
| ROCK1 | DMPK | AGC | 4yve | B | | 2-(3-methoxyphenyl)-n-[4-(pyridin-4-yl)-1,3-thiazol-2-yl]acetamide | Human | 2706 | |
| PRKACA (PKACa) | PKA | AGC | 6no7 | C | | - | Human | 11466 | |
| PRKACA (PKACa) | PKA | AGC | 6wjg | B | | - | Human | 13007 | |
| ROCK2 | DMPK | AGC | 7jnt | A | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12744 | |
| ROCK2 | DMPK | AGC | 7jnt | E | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12746 | |
| ROCK2 | DMPK | AGC | 7jnt | E | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12747 | |
| ROCK2 | DMPK | AGC | 7jov | C | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12748 | |
| ROCK2 | DMPK | AGC | 8x8z | A | | ~{n}-methyl-3-[[6-(3-methyl-1,2-oxazol-4-yl)-1-oxidanylidene-isoquinolin-2-yl]methyl]benzamide | Human | 15967 | |
| ROCK2 | DMPK | AGC | 7jnt | F | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12749 | |
| ROCK2 | DMPK | AGC | 7jnt | D | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12750 | |
| ROCK2 | DMPK | AGC | 7jov | H | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12751 | |
| ROCK2 | DMPK | AGC | 6ed6 | A | | n-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamide | Human | 10689 | |
| ROCK2 | DMPK | AGC | 6p5m | A | A | 6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11920 | |
| ROCK2 | DMPK | AGC | 7jnt | C | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12752 | |
| ROCK2 | DMPK | AGC | 8x8x | A | | ~{n}-methyl-3-[[1-oxidanylidene-6-[5-(trifluoromethyl)-1~{h}-pyrazol-4-yl]isoquinolin-2-yl]methyl]benzamide | Human | 15968 | |
| ROCK2 | DMPK | AGC | 7jnt | H | B | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12753 | |
| ROCK2 | DMPK | AGC | 9hfp | A | | ~{n}-[4-[(3~{r})-piperidin-3-yl]oxyphenyl]-1~{h}-pyrrolo[2,3-b]pyridin-4-amine | Human | 15969 | |
| ROCK2 | DMPK | AGC | 6p5m | B | A | 6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11921 | |
| ROCK2 | DMPK | AGC | 6p5p | B | | 2-[(2s)-1-azabicyclo[2.2.2]octan-2-yl]-6-(5-methyl-1h-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11923 | |
| ROCK2 | DMPK | AGC | 7jnt | D | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12755 | |
| ROCK2 | DMPK | AGC | 7jnt | B | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12756 | |
| ROCK2 | DMPK | AGC | 6p5m | B | B | 6-(5-methyl-1h-pyrazol-4-yl)-2-[(pyrrolidin-1-yl)methyl]thieno[3,2-d]pyrimidin-4(3h)-one | Human | 11924 | |
| ROCK2 | DMPK | AGC | 7jov | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12757 | |
| ROCK2 | DMPK | AGC | 9hjq | A | | [3,3-bis(fluoranyl)azetidin-1-yl]-[1-methyl-6-[4-[[4-(1~{h}-pyrazol-4-yl)phenyl]amino]pyrimidin-2-yl]indol-2-yl]methanone | Human | 15970 | |
| ROCK2 | DMPK | AGC | 5u7r | A | | (1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-one | Human | 7989 | |
| ROCK2 | DMPK | AGC | 6p5m | C | A | - | Human | 11917 | |
| ROCK2 | DMPK | AGC | 8x8y | A | | 3-fluoranyl-~{n}-methyl-5-[[1-oxidanylidene-6-[5-(trifluoromethyl)-1~{h}-pyrazol-4-yl]isoquinolin-2-yl]methyl]benzamide | Human | 15971 | |
| ROCK2 | DMPK | AGC | 7jov | F | | n-[(1s)-2-hydroxy-1-phenylethyl]-3-methoxy-4-(1h-pyrazol-4-yl)benzamide | Human | 12759 | |
| ROCK2 | DMPK | AGC | 7jnt | H | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12760 | |
| ROCK2 | DMPK | AGC | 4l6q | B | | 6-[4-(aminomethyl)-2-fluorophenoxy]-2,1-benzoxaborol-1(3h)-ol | Human | 1810 | |
| ROCK2 | DMPK | AGC | 6p5m | D | B | - | Human | 11922 | |
| ROCK2 | DMPK | AGC | 7jnt | G | A | n-[(3-methoxyphenyl)methyl]-5h-[1]benzopyrano[3,4-c]pyridine-8-carboxamide | Human | 12761 | |
| ROCK2 | DMPK | AGC | 5u7r | D | | (1s,4s)-4-(4-fluorophenyl)-4-hydroxy-6'-(5-methyl-1h-pyrazol-4-yl)-1'h-spiro[cyclohexane-1,2'-thieno[3,2-d]pyrimidin]-4'(3'h)-one | Human | 7985 | |
| ROCK2 | DMPK | AGC | 6p5m | C | B | - | Human | 11916 | |
| ROCK2 | DMPK | AGC | 6ed6 | B | | n-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamide | Human | 10688 | |
| ROCK2 | DMPK | AGC | 4wot | C | | methyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoate | Human | 6828 | |
| ROCK2 | DMPK | AGC | 4wot | D | | methyl 3-[({2'-(aminomethyl)-5'-[(3-fluoropyridin-4-yl)carbamoyl]biphenyl-3-yl}carbonyl)amino]-4-fluorobenzoate | Human | 6830 | |
| ROCK2 | DMPK | AGC | 8gds | A | | 4-{4-[2-(2,3-dihydro-1h-indol-1-yl)-2-oxoethyl]phenyl}phthalazin-1(2h)-one | Human | 14736 | |
| PRKCH (PKCh) | PKC | AGC | 8fp1 | A | | (3p)-3-[6-chloro-4-(9-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | 14694 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqk | A | B | adenosine-5'-triphosphate | Human | 3156 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5mrd | A | B | adenosine-5'-triphosphate | Human | 7394 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu3 | A | B | (9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dione | Human | 3248 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1z5m | A | | n-(3-{[5-bromo-2-({3-[(pyrrolidin-1-ylcarbonyl)amino]phenyl}amino)pyrimidin-4-yl]amino}propyl)-2,2-dimethylmalonamide | Human | 3152 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ho8 | A | B | 4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 6672 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | B | | - | Human | 3178 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rrv | A | A | adenosine-5'-triphosphate | Human | 3244 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5mrd | A | A | adenosine-5'-triphosphate | Human | 7395 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu9 | A | B | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 6799 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4aw0 | A | A | adenosine-5'-triphosphate | Human | 3176 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3pwy | A | | n-[2-({6-[(2-sulfanylethyl)amino]pyrimidin-4-yl}amino)ethyl]propanamide | Human | 3155 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nun | A | A | 6-(2-aminopyrimidin-4-yl)-1h-indazol-3-amine | Human | 3183 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3iop | A | | 2-(5-{[(2r)-2-amino-3-phenylpropyl]oxy}pyridin-3-yl)-8,9-dimethoxybenzo[c][2,7]naphthyridin-4-amine | Human | 3204 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2r7b | A | | 10,11-dimethoxy-4-methyldibenzo[c,f]-2,7-naphthyridine-3,6-diamine | Human | 3215 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd4 | A | B | tert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamate | Human | 3190 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4a07 | A | B | adenosine-5'-triphosphate | Human | 3238 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4ct2 | A | B | adenosine-5'-triphosphate | Human | 3230 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | C | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3150 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcx | A | B | 6-{2-amino-6-[(3r)-3-methylmorpholin-4-yl]pyrimidin-4-yl}-2h-indazol-3-amine | Human | 3249 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | A | | - | Human | 3235 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | C | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3243 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2biy | A | B | adenosine-5'-triphosphate | Human | 3169 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4a07 | A | A | adenosine-5'-triphosphate | Human | 3234 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvn | A | B | adenosine | Human | 7109 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nuu | A | B | 3,4-dihydroisoquinolin-1(2h)-one | Human | 3159 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1okz | A | | 7-hydroxystaurosporine | Human | 3209 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ack | A | A | adenosine-5'-triphosphate | Human | 6191 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | A | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3197 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd0 | A | B | (3s,6r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-6-methyl-n-phenylpiperidine-3-carboxamide | Human | 3162 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nuy | A | A | quinazolin-4(1h)-one | Human | 3236 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvo | A | A | adenosine-5'-triphosphate | Human | 7104 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | A | B | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 9253 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4aw0 | A | B | adenosine-5'-triphosphate | Human | 3241 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcs | A | A | 6-[2-amino-6-(morpholin-4-yl)pyrimidin-4-yl]-2h-indazol-3-amine | Human | 3179 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rrv | A | C | adenosine-5'-triphosphate | Human | 3191 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3h9o | A | | 2-(1h-imidazol-1-yl)-9-methoxy-8-(2-methoxyethoxy)benzo[c][2,7]naphthyridin-4-amine | Human | 3226 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3hrc | A | A | adenosine-5'-triphosphate | Human | 3172 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvm | A | A | adenine | Human | 7112 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqk | A | C | adenosine-5'-triphosphate | Human | 3211 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nus | A | B | 1h-indazol-3-amine | Human | 3185 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu8 | A | A | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 3239 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3rwp | A | B | [4-amino-7-(propan-2-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl](6-{[(3s,4r)-4-(4-fluorophenyl)tetrahydrofuran-3-yl]amino}pyrazin-2-yl)methanone | Human | 3199 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2xch | A | | 8-(cyclohexa-2,5-dien-1-ylideneamino)-1-(piperidin-4-ylmethyl)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 3220 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3hrc | A | B | adenosine-5'-triphosphate | Human | 3223 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvp | D | | adenosine-5'-triphosphate | Human | 7108 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqv | A | C | adenosine-5'-triphosphate | Human | 3222 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvo | A | B | adenosine-5'-triphosphate | Human | 7114 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nay | A | | 4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-one | Human | 3231 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | H | | - | Human | 3177 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | D | A | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3192 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2xck | A | | 1-methyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-n-[(2-methylpyridin-4-yl)methyl]-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 3201 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2pe2 | A | | 3-[5-({5-[(aminocarbonyl)amino]-2-oxo-2h-indol-3-yl}methyl)-1h-pyrrol-3-yl]-n-(2-piperidin-1-ylethyl)benzamide | Human | 3163 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nus | A | A | 1h-indazol-3-amine | Human | 3233 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | F | | - | Human | 3228 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3hrf | A | A | adenosine-5'-triphosphate | Human | 3170 | |
| PDPK1 (PDK1) | PDK1 | AGC | 2pe1 | A | | 1-{2-oxo-3-[(1r)-1-(1h-pyrrol-2-yl)ethyl]-2h-indol-5-yl}urea | Human | 3167 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rrv | A | B | adenosine-5'-triphosphate | Human | 3212 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4ct1 | A | A | adenosine-5'-triphosphate | Human | 3158 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5hkm | A | | 4-ethyl-6-[5-(1h-pyrazol-4-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]pyrimidin-2-amine | Human | 6670 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orz | B | B | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3198 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4rqv | A | A | adenosine-5'-triphosphate | Human | 3219 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1h1w | A | B | adenosine-5'-triphosphate | Human | 3194 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3orx | G | | - | Human | 3189 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qd4 | A | A | tert-butyl {(3r,5r)-1-[2-amino-6-(3-amino-2h-indazol-6-yl)pyrimidin-4-yl]-5-methylpiperidin-3-yl}carbamate | Human | 3225 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qc4 | B | A | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 9255 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3otu | A | | 3-(1h-indol-3-yl)-4-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1h-indol-3-yl}-1h-pyrrole-2,5-dione | Human | 3217 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3qcq | A | B | 6-(3-amino-2h-indazol-6-yl)-n~4~-ethylpyrimidine-2,4-diamine | Human | 3166 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4a06 | A | A | adenosine-5'-triphosphate | Human | 3207 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ho8 | A | A | 4-butyl-6-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 6674 | |
| PDPK1 (PDK1) | PDK1 | AGC | 4xx9 | A | A | adenosine-5'-triphosphate | Human | 6193 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1h1w | A | A | adenosine-5'-triphosphate | Human | 3186 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5ack | A | B | adenosine-5'-triphosphate | Human | 6194 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nax | A | | 1-(3,4-difluorobenzyl)-2-oxo-n-{(1r)-2-[(2-oxo-2,3-dihydro-1h-benzimidazol-5-yl)oxy]-1-phenylethyl}-1,2-dihydropyridine-3-carboxamide | Human | 3200 | |
| PDPK1 (PDK1) | PDK1 | AGC | 5lvm | A | B | adenine | Human | 7103 | |
| PDPK1 (PDK1) | PDK1 | AGC | 3nay | B | | 4-(2-cyclopropylethylidene)-9-(1h-pyrazol-4-yl)-6-{[(1r)-1,2,2-trimethylpropyl]amino}benzo[c][1,6]naphthyridin-1(4h)-one | Human | 3203 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1uu9 | A | A | 3-[1-(3-aminopropyl)-1h-indol-3-yl]-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 6800 | |
| PDPK1 (PDK1) | PDK1 | AGC | 1oky | A | B | staurosporine | Human | 3195 | |
| PRKCQ (PKCt) | PKC | AGC | 1xjd | A | | staurosporine | Human | 5357 | |
| PRKCQ (PKCt) | PKC | AGC | 4q9z | B | B | (1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5362 | |
| PRKCQ (PKCt) | PKC | AGC | 4ra5 | A | B | (1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5359 | |
| PRKCQ (PKCt) | PKC | AGC | 4ra5 | B | A | (1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5361 | |
| PRKCQ (PKCt) | PKC | AGC | 4q9z | A | A | (1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5356 | |
| PRKCQ (PKCt) | PKC | AGC | 2jed | A | | 3-(8-dimethylaminomethyl-6,7,8,9-tetrahydro-pyrido[1,2-a]indol-10-yl)-4-(1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 5352 | |
| PRKCQ (PKCt) | PKC | AGC | 4ra5 | A | A | (1r)-9-[(1,3-dimethylazetidin-3-yl)(methyl)amino]-1-methyl-8-phenyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5354 | |
| PRKCQ (PKCt) | PKC | AGC | 4q9z | B | A | (1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5355 | |
| PRKCQ (PKCt) | PKC | AGC | 4q9z | A | B | (1r)-9-(azetidin-3-ylamino)-1,8-dimethyl-3,5-dihydro[1,2,4]triazino[3,4-c][1,4]benzoxazin-2(1h)-one | Human | 5353 | |
| SGK1 | SGK | AGC | 3hdn | A | | [4-(5-naphthalen-2-yl-1h-pyrrolo[2,3-b]pyridin-3-yl)phenyl]acetic acid | Human | 3270 | |
| SGK1 | SGK | AGC | 3hdm | A | | 4-(5-phenyl-1h-pyrrolo[2,3-b]pyridin-3-yl)benzoic acid | Human | 3271 | |
| SGK1 | SGK | AGC | 7pue | A | | 6-[4-[[2,3-bis(chloranyl)phenyl]sulfonylamino]phenyl]-~{n}-[(3~{r})-pyrrolidin-3-yl]-2~{h}-pyrazolo[3,4-b]pyridine-4-carboxamide | Human | 14012 | |
| SGK1 | SGK | AGC | 2r5t | A | | phosphoaminophosphonic acid-adenylate ester | Human | 6849 | |
| PKN1 | PKN | AGC | 4otg | A | B | lestaurtinib | Human | 549 | |
| PKN1 | PKN | AGC | 4otd | A | B | - | Human | 546 | |
| AKT2 | Akt | AGC | 3e87 | A | A | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | 1910 | |
| AKT2 | Akt | AGC | 2jdr | A | | (2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amine | Human | 1918 | |
| AKT2 | Akt | AGC | 3e8d | A | B | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1926 | |
| AKT2 | Akt | AGC | 1gzo | A | | - | Human | 1914 | |
| AKT2 | Akt | AGC | 8q61 | A | B | 6-[4-(1-azanyl-3-methyl-3-oxidanyl-cyclobutyl)phenyl]-7-phenyl-1-propyl-pyrido[2,3-b][1,4]oxazin-2-one | Human | 14979 | |
| AKT2 | Akt | AGC | 3e8d | A | A | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1921 | |
| AKT2 | Akt | AGC | 3d0e | A | | 4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-ol | Human | 1912 | |
| AKT2 | Akt | AGC | 3e8d | B | B | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1904 | |
| AKT2 | Akt | AGC | 3e88 | B | | 4-[2-(4-amino-1,2,5-oxadiazol-3-yl)-6-{[(2r)-2-amino-3-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1905 | |
| AKT2 | Akt | AGC | 3d0e | B | | 4-{2-(4-amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-[(3s)-piperidin-3-ylmethoxy]-1h-imidazo[4,5-c]pyridin-4-yl}-2-methylbut-3-yn-2-ol | Human | 1920 | |
| AKT2 | Akt | AGC | 3e8d | B | A | 4-[2-(4-amino-2,5-dihydro-1,2,5-oxadiazol-3-yl)-6-{[(1s)-3-amino-1-phenylpropyl]oxy}-1-ethyl-1h-imidazo[4,5-c]pyridin-4-yl]-2-methylbut-3-yn-2-ol | Human | 1925 | |
| AKT2 | Akt | AGC | 3e87 | A | B | n-[(1s)-2-amino-1-phenylethyl]-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)thiophene-2-carboxamide | Human | 1911 | |
| AKT2 | Akt | AGC | 1gzn | A | | - | Human | 1915 | |
| AKT2 | Akt | AGC | 1o6l | A | | phosphoaminophosphonic acid-adenylate ester | Human | 1906 | |
| AKT2 | Akt | AGC | 1mrv | A | | - | Human | 1917 | |
| AKT2 | Akt | AGC | 1gzk | A | | - | Human | 1916 | |
| AKT2 | Akt | AGC | 2uw9 | A | | 4-(4-chlorophenyl)-4-[4-(1h-pyrazol-4-yl)phenyl]piperidine | Human | 1919 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf7 | A | B | 1-(9h-purin-6-yl)-n-[3-(trifluoromethyl)phenyl]piperidine-4-carboxamide | Human | 1851 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l42 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1865 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l3j | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1858 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 7n93 | A | B | 4-({(1s)-2-(azetidin-1-yl)-1-[4-chloro-3-(trifluoromethyl)phenyl]ethyl}amino)quinazoline-8-carboxamide | Human | 14283 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf9 | A | | (2s)-1-oxo-1-[(4-sulfamoylphenyl)amino]propan-2-yl (2s)-2-methyl-1,2,3,4-tetrahydroacridine-9-carboxylate | Human | 1866 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4rlo | A | | [(amino-kappan)methanethiolato](3-fluoro-9-hydroxypyrido[2,3-a]pyrrolo[3,4-c]carbazole-5,7(6h,12h)-dionato-kappa~2~n,n')(1,4,7-trithionane-kappa~3~s~1~,s~4~,s~7~)ruthenium | Human | 7218 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a60 | B | | staurosporine | Human | 1856 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3a60 | A | | staurosporine | Human | 1852 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 3wf6 | A | A | 4-[4-(1h-indol-3-yl)-3,6-dihydropyridin-1(2h)-yl]-1h-pyrazolo[3,4-d]pyrimidine | Human | 1864 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4l44 | A | | 2-{[4-(5-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-5-(trifluoromethyl)-1h-benzimidazole | Human | 1849 | |
| RPS6KB1 (p70S6K) | RSK | AGC | 4rlo | B | | staurosporine | Human | 7220 | |
| GRK5 (GPRK5) | GRK | AGC | 4tnd | A | | phosphoaminophosphonic acid-adenylate ester | Human | 3275 | |
| GRK2 (BARK1) | GRK | AGC | 5wg5 | A | B | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-2h-indazole | Human | 9440 | |
| GRK2 (BARK1) | GRK | AGC | 5wg4 | A | B | 2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamide | Human | 9438 | |
| GRK2 (BARK1) | GRK | AGC | 3v5w | A | A | paroxetine | Human | 1705 | |
| GRK2 (BARK1) | GRK | AGC | 7k7l | A | B | 3-benzyl-6-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | 12958 | |
| GRK2 (BARK1) | GRK | AGC | 7k7z | A | A | 3-benzyl-7-(1h-pyrazol-4-yl)quinazolin-4(3h)-one | Human | 12959 | |
| GRK2 (BARK1) | GRK | AGC | 5ukk | A | A | 5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(pyridin-2-yl)methyl]benzamide | Human | 7529 | |
| GRK2 (BARK1) | GRK | AGC | 5ukl | A | A | 2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamide | Human | 7528 | |
| GRK2 (BARK1) | GRK | AGC | 3v5w | A | B | paroxetine | Human | 1711 | |
| GRK2 (BARK1) | GRK | AGC | 4mk0 | A | A | 5-{[(3s,4r)-4-(4-fluorophenyl)piperidin-3-yl]methoxy}-1h-isoindol-1-one | Human | 1710 | |
| GRK2 (BARK1) | GRK | AGC | 5uuu | A | A | 3-({[4-methyl-5-(pyridin-4-yl)-4h-1,2,4-triazol-3-yl]methyl}amino)-n-[2-(trifluoromethyl)benzyl]benzamide | Human | 8255 | |
| GRK2 (BARK1) | GRK | AGC | 3krx | A | | balanol | Human | 1709 | |
| GRK2 (BARK1) | GRK | AGC | 6u7c | A | | 5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluoro-n-[(2h-indazol-3-yl)methyl]benzamide | Human | 12162 | |
| GRK2 (BARK1) | GRK | AGC | 3cik | A | | - | Human | 1706 | |
| GRK2 (BARK1) | GRK | AGC | 5he1 | A | A | (4~{s})-4-[4-fluoranyl-3-(isoquinolin-1-ylmethylcarbamoyl)phenyl]-~{n}-(1~{h}-indazol-5-yl)-6-methyl-2-oxidanylidene-3,4-dihydro-1~{h}-pyrimidine-5-carboxamide | Human | 6605 | |
| GRK2 (BARK1) | GRK | AGC | 5wg4 | A | A | 2-fluoro-5-[(3s,4r)-3-{[(1h-indazol-5-yl)oxy]methyl}piperidin-4-yl]-n-[(pyridin-2-yl)methyl]benzamide | Human | 9441 | |
| GRK2 (BARK1) | GRK | AGC | 5ukl | A | B | 2-{5-[(3s,4r)-3-{[(2h-1,3-benzodioxol-5-yl)oxy]methyl}piperidin-4-yl]-2-fluorophenyl}-n-[2-(1h-pyrazol-4-yl)ethyl]acetamide | Human | 7531 | |
| ROCK1 | DMPK | AGC | 4w7p | D | | n~1~-[2-(1h-indazol-5-yl)pyrido[3,4-d]pyrimidin-4-yl]-2-methylpropane-1,2-diamine | Human | 2712 | |
| ROCK1 | DMPK | AGC | 5wnf | C | A | 1-(4-amino-1,2,5-oxadiazol-3-yl)-5-methyl-n-({3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}methyl)-1h-1,2,3-triazole-4-carboxamide | Human | 10455 | |
| ROCK1 | DMPK | AGC | 6e9w | B | | n-[(2,3-dihydro-1,4-benzodioxin-5-yl)methyl]-4-(pyridin-4-yl)benzamide | Human | 10690 | |
| ROCK1 | DMPK | AGC | 3d9v | B | | (s)-2-methyl-1-[(4-methyl-5-isoquinoline)sulfonyl]-homopiperazine | Human | 2701 | |
| ROCK1 | DMPK | AGC | 3v8s | A | | 1-(1h-indazol-5-yl)-3-(2-phenylethyl)urea | Human | 2716 | |
| ROCK1 | DMPK | AGC | 5kks | A | | 2-[3-(methylsulfonylamino)phenyl]-~{n}-[4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]ethanamide | Human | 8183 | |
| ROCK1 | DMPK | AGC | 5wnh | A | | (2r)-n-(3-cyanophenyl)-2-{3-[(5-methyl-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl)carbamoyl]phenyl}pyrrolidine-1-carboxamide | Human | 10448 | |
| ROCK1 | DMPK | AGC | 5wng | B | | (2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamide | Human | 10461 | |
| ROCK1 | DMPK | AGC | 5wng | C | | (2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamide | Human | 10458 | |
| ROCK1 | DMPK | AGC | 3v8s | D | | 1-(1h-indazol-5-yl)-3-(2-phenylethyl)urea | Human | 2692 | |
| ROCK1 | DMPK | AGC | 3twj | A | | 1-[(3-hydroxyphenyl)methyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2710 | |
| ROCK1 | DMPK | AGC | 8zh5 | A | | - | Human | 15364 | |
| ROCK1 | DMPK | AGC | 2esm | B | | 5-(1,4-diazepan-1-sulfonyl)isoquinoline | Human | 2714 | |
| ROCK1 | DMPK | AGC | 3ncz | C | | cis-4-amino-n-(7-chloro-1-oxo-1,2-dihydroisoquinolin-6-yl)cyclohexanecarboxamide | Human | 2719 | |
| ROCK1 | DMPK | AGC | 2v55 | C | | phosphoaminophosphonic acid-adenylate ester | Human | 2711 | |
| ROCK1 | DMPK | AGC | 5wng | D | | (2r)-n-(3-cyanophenyl)-2-(3-{[(6s)-6-(dimethylamino)-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]carbamoyl}phenyl)pyrrolidine-1-carboxamide | Human | 10457 | |
| ROCK1 | DMPK | AGC | 5uzj | B | | n-[4-(2-aminopyridin-4-yl)-1,3-thiazol-2-yl]-2-(3-methoxyphenyl)acetamide | Human | 9707 | |
| ROCK1 | DMPK | AGC | 3tv7 | A | | 1-[(1r)-1-(3-methoxyphenyl)ethyl]-3-(4-pyridin-4-yl-1,3-thiazol-2-yl)urea | Human | 2697 | |
