Browse
Search
Drugs
Favorites
 

Search results (601 entries covering 458 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
PI4KBPIKAtypical4d0mgn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9146
PI4K2APIKAtypical5eutA-Human9264
PIK3CG (p110g)PIKAtypical3nzsA6-(1,1-dioxidothiomorpholin-4-yl)-n-(3-methoxyphenyl)-1-methyl-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9179
TRRAPPIKKAtypical8xvgABadenosine-5'-diphosphateHuman15323
PIK3CA (p110a)PIKAtypical8twyA1-(4-{[2-(4-{(4p)-4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-[(3s)-3-methylmorpholin-4-yl]-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethoxy]methyl}piperidin-1-yl)prop-2-en-1-oneHuman15392
PI4KBPIKAtypical8vofAmethyl 2-chloro-5-(methyl{(8r)-3-[4-(methylcarbamoyl)phenyl]pyrazolo[1,5-a]pyridine-5-carbonyl}amino)benzoateHuman15377
ANTXR1 (DNAPK)PIKKAtypical7k11A-Human13208
PIK3CA (p110a)PIKAtypical8exoAB1-{(4s,11am)-2-[(4r)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-prolinamideHuman14534
ANTXR1 (DNAPK)PIKKAtypical5luqB-Human9319
ANTXR1 (DNAPK)PIKKAtypical7sglABadenosine-5'-triphosphateHuman14062
MTOR (FRAP)PIKKAtypical4jspAphosphothiophosphoric acid-adenylate esterHuman9106
PIK3CA (p110a)PIKAtypical8exlAA2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamideHuman14537
PIK3CA (p110a)PIKAtypical8exoAA1-{(4s,11am)-2-[(4r)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-prolinamideHuman14541
PIK3CA (p110a)PIKAtypical8exvAAn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14542
PIK3CD (p110d)PIKAtypical5m6uA4-azanyl-6-[[(1~{s})-1-(4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]pyrimidine-5-carbonitrileHuman9094
PIK3CA (p110a)PIKAtypical8gudAA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14535
ANTXR1 (DNAPK)PIKKAtypical7sudAAadenosine-5'-triphosphateHuman14055
PIK3CG (p110g)PIKAtypical7mezA-Human13798
PIK3CG (p110g)PIKAtypical4kzcAn-{6-[6-amino-5-(trifluoromethyl)pyridin-3-yl]imidazo[1,2-a]pyridin-2-yl}acetamideHuman9224
PIK3CG (p110g)PIKAtypical5g2nA2-azanyl-~{n}-[7-methoxy-8-(3-morpholin-4-ylpropoxy)-2,3-dihydroimidazo[1,2-c]quinazolin-5-yl]pyrimidine-5-carboxamideHuman9206
PIK3CG (p110g)PIKAtypical5kaeA4-azanyl-6-[[(1~{s})-1-(6-fluoranyl-3-phenyl-4-piperazin-1-ylcarbonyl-quinolin-2-yl)ethyl]amino]pyrimidine-5-carbonitrileHuman9241
PIK3CG (p110g)PIKAtypical4ezkA2-(1-{[2-(2h-indazol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-olHuman9176
PIK3CG (p110g)PIKAtypical5g55A6-cyano-4-[[(1r)-1-(4-methylphenyl)ethyl]amino]quinoline-3-carboxamideHuman9199
PIK3CG (p110g)PIKAtypical4urkA2-[[(1r)-1-(7-methyl-2-morpholin-4-yl-4-oxidanylidene-pyrido[1,2-a]pyrimidin-9-yl)ethyl]amino]benzoic acidHuman9196
PIK3CG (p110g)PIKAtypical4fjzA1'-[7-fluoro-3-methyl-2-(pyridin-2-yl)quinolin-4-yl]-6'-(morpholin-4-yl)-1',2,2',3,5,6-hexahydrospiro[pyran-4,3'-pyrrolo[3,2-b]pyridine]Human9173
PIK3CG (p110g)PIKAtypical6c1sA{4-[2-(5,6-dimethoxypyridin-3-yl)-5-oxo-5,7-dihydro-6h-pyrrolo[3,4-b]pyridin-6-yl]-1h-pyrazol-1-yl}acetonitrileHuman10037
PIK3CG (p110g)PIKAtypical4dk5A4-(2-[(6-methoxypyridin-3-yl)amino]-5-{[4-(methylsulfonyl)piperazin-1-yl]methyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amineHuman9232
PIK3CG (p110g)PIKAtypical1e8zAstaurosporineHuman9228
PIK3CG (p110g)PIKAtypical3qk0An-[6-(6-chloro-5-{[(4-fluorophenyl)sulfonyl]amino}pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamideHuman9213
PIK3CG (p110g)PIKAtypical3l08AA2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamideHuman9217
PIK3CG (p110g)PIKAtypical3apcA5-(7-methanesulfonyl-2-morpholin-4-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamineHuman9231
PIK3CA (p110a)PIKAtypical7pg6AA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14348
PIK3CG (p110g)PIKAtypical6xrlA2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman12774
PIK3CG (p110g)PIKAtypical5jhaA[1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)pyrimidin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanolHuman9246
PIK3CG (p110g)PIKAtypical6t3cA7-methyl-2-[(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(oxan-4-yl)purin-8-oneHuman11907
PIK3CG (p110g)PIKAtypical3zw3An-{6-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]imidazo[1,2-a]pyridin-2-yl}acetamideHuman9207
PIK3C3PIKAtypical4oysA(8s)-9-[(5-chloranylpyridin-3-yl)methyl]-2-[(3r)-3-methylmorpholin-4-yl]-8-(trifluoromethyl)-6,7,8,9a-tetrahydro-3h-pyrimido[1,2-a]pyrimidin-4-oneHuman9327
ANTXR1 (DNAPK)PIKKAtypical7z87AA(~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanolHuman14592
PIK3C3PIKAtypical7rsjABn-{4-[(7r,8r)-4-oxo-7-(propan-2-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]pyridin-2-yl}cyclopropanecarboxamideHuman13982
PIK3C3PIKAtypical3ls8AA-Human9340
PIK3C3PIKAtypical6i3uA2-morpholin-4-yl-6-[7-[(2~{r})-1-morpholin-4-ylpropan-2-yl]oxy-9~{h}-thioxanthen-4-yl]pyran-4-oneHuman11292
PIK3C3PIKAtypical7rsvAA(5as,8ar,9s)-2-[(3r)-3-methylmorpholin-4-yl]-5,5a,6,7,8,8a-hexahydro-4h-cyclopenta[e]pyrazolo[1,5-a]pyrazin-4-oneHuman13985
PIK3C3PIKAtypical3ihyA-Human9341
PIK3C3PIKAtypical3ihyC-Human9331
PIK3C3PIKAtypical5anlA(8s)-2-(morpholin-4-yl)-9-[2-(propan-2-yloxy)ethyl]-8-(trifluoromethyl)-6,7,8,9-tetrahydro-4h-pyrimido[1,2-a]pyrimidin-4-oneHuman9349
PIK3C3PIKAtypical3ls8AB-Human9348
PIK3C3PIKAtypical3ihyD-Human9337
PIK3C3PIKAtypical4ph4BB-Human9330
PIK3C3PIKAtypical7rspAB(7r,8r)-2-[(3r)-3-methylmorpholin-4-yl]-7-(propan-2-yl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5h)-oneHuman13986
SMG1PIKKAtypical6l53A-Human12156
PIK3CG (p110g)PIKAtypical6xrnA2-amino-5-{2-[(1s)-1-cyclopropylethyl]-7-methyl-1-oxo-2,3-dihydro-1h-isoindol-5-yl}-n-(trans-3-hydroxycyclobutyl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman13954
PIK3CA (p110a)PIKAtypical7mlkAA4-[6-(3,4,5-trimethoxyanilino)pyrazin-2-yl]benzamideHuman14216
PI4KBPIKAtypical8q6gAB3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15012
PI4KBPIKAtypical8q6gAA3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15014
PI4KBPIKAtypical8q6gAC3-(3,4-dimethoxyphenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15016
PIK3CA (p110a)PIKAtypical7tz7AA(4s,5r)-3-[2'-amino-2-(morpholin-4-yl)-4'-(trifluoromethyl)[4,5'-bipyrimidin]-6-yl]-4-(hydroxymethyl)-5-methyl-1,3-oxazolidin-2-oneHuman14223
PIK3CG (p110g)PIKAtypical3preA2-amino-8-(trans-4-methoxycyclohexyl)-4-methyl-6-(1h-pyrazol-3-yl)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman9198
PIK3CA (p110a)PIKAtypical8tsdA-Human15090
PI4KBPIKAtypical8q6hAB3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15017
PIK3CA (p110a)PIKAtypical8v8hA(2s)-n~1~-[(4p)-2-tert-butyl-4'-methyl[4,5'-bi-1,3-thiazol]-2'-yl]pyrrolidine-1,2-dicarboxamideHuman15249
ANTXR1 (DNAPK)PIKKAtypical7su3ABadenosine-5'-triphosphateHuman14053
ANTXR1 (DNAPK)PIKKAtypical7k17B-Human13212
ANTXR1 (DNAPK)PIKKAtypical7otyA(~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanolHuman14057
ATMPIKKAtypical7ni4A8-(1,3-dimethylpyrazol-4-yl)-1-(3-fluoranyl-5-methoxy-pyridin-4-yl)-7-methoxy-3-methyl-imidazo[4,5-c]quinolin-2-oneHuman13864
ANTXR1 (DNAPK)PIKKAtypical7otmA8-(dibenzo[b,d]thiophen-4-yl)-2-(morpholin-4-yl)-4h-chromen-4-oneHuman14061
PIK3CA (p110a)PIKAtypical7mynAB-Human13964
PIK3C3PIKAtypical7rspAA(7r,8r)-2-[(3r)-3-methylmorpholin-4-yl]-7-(propan-2-yl)-6,7-dihydropyrazolo[1,5-a]pyrazin-4(5h)-oneHuman13981
ANTXR1 (DNAPK)PIKKAtypical8ezbCadenosine-5'-triphosphateHuman14798
PIK3CA (p110a)PIKAtypical8v8iA(2s)-n~1~-[(4p)-2-tert-butyl-4'-methyl[4,5'-bi-1,3-thiazol]-2'-yl]pyrrolidine-1,2-dicarboxamideHuman15248
ATRPIKKAtypical9zd1Aphosphoaminophosphonic acid-adenylate esterHuman15662
ATRPIKKAtypical23fdAphosphothiophosphoric acid-adenylate esterHuman15663
PIK3CA (p110a)PIKAtypical8v8uA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman15250
PIK3CA (p110a)PIKAtypical8v8vA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman15252
PIK3CA (p110a)PIKAtypical8v8jA(2s)-n~1~-[(4p)-2-tert-butyl-4'-methyl[4,5'-bi-1,3-thiazol]-2'-yl]pyrrolidine-1,2-dicarboxamideHuman15251
MTOR (FRAP)PIKKAtypical9tdsA-Human15768
MTOR (FRAP)PIKKAtypical9t92A-Human15765
MTOR (FRAP)PIKKAtypical9ed7Aphosphoaminophosphonic acid-adenylate esterHuman15766
MTOR (FRAP)PIKKAtypical9t93A-Human15767
MTOR (FRAP)PIKKAtypical9zbjA-Human15769
MTOR (FRAP)PIKKAtypical9zbkA-Human15770
MTOR (FRAP)PIKKAtypical9t7jAadenosine-5'-triphosphateHuman15771
MTOR (FRAP)PIKKAtypical9tdtA-Human15772
MTOR (FRAP)PIKKAtypical8rchAphosphoaminophosphonic acid-adenylate esterHuman15773
MTOR (FRAP)PIKKAtypical9tpwA-Human15774
TRRAPPIKKAtypical9rdkE-Human15849
ANTXR1 (DNAPK)PIKKAtypical9iaxA-Human16042
ANTXR1 (DNAPK)PIKKAtypical9zobA-Human16043
RIOK3RIOAtypical8zddI-Human16169
PIK3CD (p110d)PIKAtypical5ubtA1-[4-(3-{4-amino-5-[1-(oxan-4-yl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)piperazin-1-yl]ethan-1-oneHuman9092
PIK3CD (p110d)PIKAtypical6pyrAB(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11546
PI4KAP2PIKAtypical9b9gAA-Human16198
PI4KAP2PIKAtypical9baxB-Human16199
PI4KAP2PIKAtypical9b9gAB-Human16200
PI4KAP2PIKAtypical9ot6A-Human16201
PIK3CD (p110d)PIKAtypical6ocuA5-{(3r)-3-methyl-4-[(1r,2r)-2-methylcyclopropane-1-carbonyl]piperazin-1-yl}-3-(1-methyl-1h-pyrazol-4-yl)pyrazine-2-carbonitrileHuman11864
PIK3CA (p110a)PIKAtypical4ovuAB-Human9271
PIK3CA (p110a)PIKAtypical6pysAB(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11576
PIK3CA (p110a)PIKAtypical4ovvA-Human9307
PIK3CA (p110a)PIKAtypical7mlkAB4-[6-(3,4,5-trimethoxyanilino)pyrazin-2-yl]benzamideHuman14217
PIK3CA (p110a)PIKAtypical4ovuAA-Human9291
PIK3CA (p110a)PIKAtypical5sxbA-Human9282
PIK3CA (p110a)PIKAtypical5swoA-Human9303
PIK3CD (p110d)PIKAtypical6pyrAA(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11547
ANTXR1 (DNAPK)PIKKAtypical7tyrAB-Human14321
PIK3CG (p110g)PIKAtypical3t8mAn~2~-{2-chloro-4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-n~2~,n~8~-dimethyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2,8-dicarboxamideHuman9186
PIK3CG (p110g)PIKAtypical3ps6A4-amino-n-(6-methoxypyridin-3-yl)-2-methylquinazoline-8-carboxamideHuman9170
PIK3CG (p110g)PIKAtypical2chwA2-((9h-purin-6-ylthio)methyl)-5-chloro-3-(2-methoxyphenyl)quinazolin-4(3h)-oneHuman9182
PIK3CG (p110g)PIKAtypical3zvvA5,7-dimethylpyrazolo[1,5-a]pyrimidin-2-amineHuman9172
PIK3CG (p110g)PIKAtypical3eneA1-methyl-3-naphthalen-2-yl-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9188
PIK3CG (p110g)PIKAtypical3lj3A(2z)-4,6-dihydroxy-2-{[1-methyl-4-(4-methylpiperazin-1-yl)-1h-pyrrolo[2,3-b]pyridin-3-yl]methylidene}-1-benzofuran-3(2h)-oneHuman9214
PIK3CG (p110g)PIKAtypical6fh5A3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-oneHuman10883
PIK3CG (p110g)PIKAtypical2chzAn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9251
PIK3CG (p110g)PIKAtypical6audAB10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepineHuman9216
PIK3CG (p110g)PIKAtypical4wwpAn-{(1s)-1-[8-chloro-2-(2-methylpyridin-3-yl)quinolin-3-yl]ethyl}-9h-purin-6-amineHuman9200
PIK3CG (p110g)PIKAtypical3apdA5-(2-morpholin-4-yl-7-pyridin-3-yl-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl)-pyrimidin-2-ylamineHuman9205
PIK3CG (p110g)PIKAtypical7jweAgedatolisibHuman13412
PIK3CG (p110g)PIKAtypical3tl5A(2s)-1-(4-{[2-(2-aminopyrimidin-5-yl)-7-methyl-4-(morpholin-4-yl)thieno[3,2-d]pyrimidin-6-yl]methyl}piperazin-1-yl)-2-hydroxypropan-1-oneHuman9160
PIK3CG (p110g)PIKAtypical4ps8An-[6-(5,6-dimethoxypyridin-3-yl)-1,3-benzothiazol-2-yl]acetamideHuman9184
PIK3CG (p110g)PIKAtypical3przA4-amino-2-methyl-n-(1h-pyrazol-3-yl)quinazoline-8-carboxamideHuman9210
PIK3CG (p110g)PIKAtypical3ibeA1-(4-{4-morpholin-4-yl-1-[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]-1h-pyrazolo[3,4-d]pyrimidin-6-yl}phenyl)-3-pyridin-4-ylureaHuman9171
PIK3CG (p110g)PIKAtypical4fhjA3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-5-yl)imidazo[1,2-a]pyridin-2-amineHuman9209
PIK3CG (p110g)PIKAtypical5t23A3-(benzotriazol-1-yl)-5-[1-methyl-5-[(1~{s})-1-morpholin-4-ylethyl]-1,2,4-triazol-3-yl]pyrazin-2-amineHuman9157
PIK3CG (p110g)PIKAtypical3oawA2-amino-4-methyl-8-(1-methylethyl)-6-(1h-pyrazol-4-yl)pteridin-7(8h)-oneHuman9240
PIK3CG (p110g)PIKAtypical3dpdA5,5-dimethyl-2-morpholin-4-yl-5,6-dihydro-1,3-benzothiazol-7(4h)-oneHuman9159
PIK3CG (p110g)PIKAtypical4xz4An-[5-(6-methoxypyrazin-2-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamideHuman9194
PIK3CG (p110g)PIKAtypical3cstAmethylated ruthenium pyridocarbazoleHuman9220
PIK3CG (p110g)PIKAtypical2v4lA3-[4-amino-1-(1-methylethyl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]phenolHuman9237
PIK3CG (p110g)PIKAtypical4anuA3-amino-n-methyl-6-[3-(1h-tetrazol-5-yl)phenyl]pyrazine-2-carboxamideHuman9162
PIK3CG (p110g)PIKAtypical3sd5A5-[2,6-di(morpholin-4-yl)pyrimidin-4-yl]-4-(trifluoromethyl)pyridin-2-amineHuman9243
PIK3CG (p110g)PIKAtypical9gg9A3-[(1~{s})-1-[4-azanyl-3-(3-fluoranyl-5-oxidanyl-phenyl)pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-4-phenyl-isochromen-1-oneHuman15415
PIK3CG (p110g)PIKAtypical4anxA5-{3-[(4-{3-[4-(1-methylethyl)phenyl]pyrazin-2-yl}piperazin-1-yl)sulfonyl]phenyl}pyrimidin-2-amineHuman9252
PIK3CG (p110g)PIKAtypical3r7qAn-(2-chlorophenyl)-n-methyl-4h-thieno[3,2-c]chromene-2-carboxamideHuman9227
PIK3CG (p110g)PIKAtypical6xrmA5-[2-amino-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]-2-[(1s)-1-cyclopropylethyl]-7-(trifluoromethyl)-2,3-dihydro-1h-isoindol-1-oneHuman12775
PIK3CG (p110g)PIKAtypical4anvAA2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazineHuman9195
PI4K2BPIKAtypical4wtvBBadenosine-5'-triphosphateHuman9096
PIK3CG (p110g)PIKAtypical7jx0An~3~-{[5-(4-acetylphenyl)-4-methyl-1,3-thiazol-2-yl]carbamoyl}-n-tert-butyl-beta-alaninamideHuman13411
PIK3CG (p110g)PIKAtypical4anwAB3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamideHuman9175
PIK3CG (p110g)PIKAtypical3qaqA[(4-{2-[(3-hydroxyphenyl)amino]-1h-benzimidazol-1-yl}-1,3,5-triazin-2-yl)amino]acetonitrileHuman9211
PIK3CG (p110g)PIKAtypical4flhA4-(2-[(5-fluoro-6-methoxypyridin-3-yl)amino]-5-{(1r)-1-[4-(methylsulfonyl)piperazin-1-yl]ethyl}pyridin-3-yl)-6-methyl-1,3,5-triazin-2-amineHuman9212
PIK3CG (p110g)PIKAtypical1he8A-Human9201
PIK3CG (p110g)PIKAtypical3l16A5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyridin-2-amineHuman9233
PIK3CA (p110a)PIKAtypical8tgdABn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14970
PIK3CA (p110a)PIKAtypical8tu6A-Human14971
PIK3CA (p110a)PIKAtypical8ilsABn-[(2r)-1-(ethylamino)-1-oxidanylidene-3-[4-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamideHuman14968
PIK3CA (p110a)PIKAtypical8ilvAn-[(2r)-1-(ethylamino)-1-oxidanylidene-3-[3-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamideHuman14974
ATMPIKKAtypical8oxqAphosphoaminophosphonic acid-adenylate esterHuman14990
ATMPIKKAtypical8oxpAphosphoaminophosphonic acid-adenylate esterHuman14991
ATMPIKKAtypical6k9lA-Human11896
ATMPIKKAtypical8oxmBphosphoaminophosphonic acid-adenylate esterHuman14992
ATMPIKKAtypical8oxoBphosphoaminophosphonic acid-adenylate esterHuman14993
RIOK1RIOAtypical6g5iz-Human10004
PIK3CG (p110g)PIKAtypical4ezlA2-(1-{[2-(2-aminopyrimidin-5-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-olHuman9235
PIK3CG (p110g)PIKAtypical4xx5An-[5-(5-methoxypyridin-3-yl)-4,5,6,7-tetrahydro[1,3]thiazolo[5,4-c]pyridin-2-yl]acetamideHuman9236
PIK3CG (p110g)PIKAtypical4ps7An-[6-(pyridin-3-yl)-1,3-benzothiazol-2-yl]acetamideHuman9163
PIK3CG (p110g)PIKAtypical3l54A6-(1h-pyrazolo[3,4-b]pyridin-5-yl)-4-pyridin-4-ylquinolineHuman9197
PIK3CG (p110g)PIKAtypical3qarA1-(4-amino-6-methyl-1,3,5-triazin-2-yl)-n-(1h-pyrazol-3-yl)-1h-benzimidazol-2-amineHuman9178
PIK3CG (p110g)PIKAtypical4g11A2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyrimidin-2-yl]-n-phenylacetamideHuman9223
PIK3C3PIKAtypical5ennBA1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-olHuman9345
PIK3CD (p110d)PIKAtypical5dxuA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHuman9091
PI4KBPIKAtypical4d0mCn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9153
PIK3CA (p110a)PIKAtypical8w9bA-Human15273
PIK3CA (p110a)PIKAtypical8w9aA-Human15274
PI4KBPIKAtypical4d0mIn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9151
PI4KBPIKAtypical5fbwA~{n}-[2-[[6-chloranyl-3-[4-methoxy-3-[[(2~{r})-1-oxidanylbutan-2-yl]sulfamoyl]phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9149
SMG1PIKKAtypical7pw9Aphosphoaminophosphonic acid-adenylate esterHuman14000
SMG1PIKKAtypical7pw7A1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-ureaHuman14005
SMG1PIKKAtypical7pw6A1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-ureaHuman14001
SMG1PIKKAtypical6sytA-Human11866
PIK3CD (p110d)PIKAtypical8bcyAB9-[2-(3,4-dichlorophenyl)ethyl]-2-(3-hydroxyphenyl)-8-oxidanylidene-7~{h}-purine-6-carboxamideHuman14734
PIK3C3PIKAtypical13bvA-Human15507
COQ8A (ADCK3)ABC1Atypical4pedAB-Human9120
PIK3C3PIKAtypical4uwkAB-Human9335
PIK3C3PIKAtypical9mhgB-Human15508
PIK3C3PIKAtypical7bl1B-Human13361
PIK3C3PIKAtypical9rx6A-Human15509
PIK3C3PIKAtypical9tw3A-Human15510
PIK3C3PIKAtypical4uwkAA-Human9342
PIK3C3PIKAtypical9mhhB-Human15511
PIK3C3PIKAtypical4uwhAA-Human9346
PIK3C3PIKAtypical9rx8A-Human15512
COQ8A (ADCK3)ABC1Atypical5i35Aphosphoaminophosphonic acid-adenylate esterHuman9122
COQ8A (ADCK3)ABC1Atypical4pedAA-Human9121
PIK3C3PIKAtypical4uwgAA-Human9347
PIK3C3PIKAtypical4uwfA-Human9328
PIK3C3PIKAtypical9s47A-Human15513
PIK3C3PIKAtypical5ennAA1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-olHuman9343
PIK3C3PIKAtypical9tz3Aadenosine-5'-diphosphateHuman15514
PIK3C3PIKAtypical5ennBB1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-olHuman9329
PIK3C3PIKAtypical3ls8BB-Human9339
PIK3C3PIKAtypical4uwlA-Human9332
PIK3C3PIKAtypical9rx7A-Human15517
PIK3C3PIKAtypical3ls8BA-Human9333
ATMPIKKAtypical6k9lB-Human11895
PIK3C3PIKAtypical9rxbA-Human15519
PIK3C3PIKAtypical4uwhAB-Human9334
PIK3C3PIKAtypical9rxaA-Human15518
PIK3C3PIKAtypical4ph4BA-Human9326
PIK3C3PIKAtypical9rx9A-Human15520
PIK3C3PIKAtypical9rx5A-Human15521
PIK3C3PIKAtypical5ennAB1-[[4-(cyclopropylmethyl)-5-[2-(pyridin-4-ylamino)pyrimidin-4-yl]pyrimidin-2-yl]amino]-2-methyl-propan-2-olHuman9338
SMG1PIKKAtypical7pw5A1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-ureaHuman14002
SMG1PIKKAtypical6l54A-Human12155
SMG1PIKKAtypical7pw4A1-[4-[4-[2-[[4-chloranyl-3-(diethylsulfamoyl)phenyl]amino]pyrimidin-4-yl]pyridin-2-yl]phenyl]-3-methyl-ureaHuman14003
SMG1PIKKAtypical7pw8Aphosphoaminophosphonic acid-adenylate esterHuman14004
SMG1PIKKAtypical6z3rAphosphoaminophosphonic acid-adenylate esterHuman12630
PI4K2BPIKAtypical4wtvABadenosine-5'-triphosphateHuman9098
PI4K2BPIKAtypical8a5xA4-azanyl-7-[3-(hydroxymethyl)phenyl]quinazoline-6-carboxamideHuman14384
PI4K2BPIKAtypical4wtvBAadenosine-5'-triphosphateHuman9097
MTOR (FRAP)PIKKAtypical5zcsB-Human9749
PI4K2APIKAtypical5i0nAAadenosine-5'-triphosphateHuman9260
PIK3CA (p110a)PIKAtypical5fi4AB~{n}-[6-[5-azanyl-6-[(2~{s})-1,1,1-tris(fluoranyl)propan-2-yl]oxy-pyrazin-2-yl]imidazo[1,2-a]pyridin-2-yl]ethanamideHuman9309
PI4KBPIKAtypical4d0mMn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9138
PIK3CA (p110a)PIKAtypical8ow2AA-Human14765
PIK3CG (p110g)PIKAtypical5oq4AA5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amineHuman9244
PI4KBPIKAtypical4d0mSn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9142
PI4KBPIKAtypical4d0mYn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9133
PI4KBPIKAtypical6gl3A(3~{s})-4-(6-azanyl-1-methyl-pyrazolo[3,4-d]pyrimidin-4-yl)-~{n}-(4-methoxy-2-methyl-phenyl)-3-methyl-piperazine-1-carboxamideHuman10442
PI4KBPIKAtypical4d0lAn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9152
PI4KBPIKAtypical5euqE~{n}-[5-[3-[[(4-hydroxyphenyl)amino]-bis(oxidanyl)-$l^{4}-sulfanyl]-4-methoxy-phenyl]-4-methyl-1,3-thiazol-2-yl]cyclopentanecarboxamideHuman9132
PI4KBPIKAtypical4waeAadenosine-5'-triphosphateHuman9144
PI4KBPIKAtypical4d0mAn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9136
PI4KBPIKAtypical5fbvA~{n}-[2-[[6-chloranyl-3-[3-(2-hydroxyethylsulfamoyl)-4-methoxy-phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9147
PI4KBPIKAtypical4d0lCn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9143
PI4KBPIKAtypical5fblA~{n}-[2-[[6-chloranyl-3-(4-methoxy-3-morpholin-4-ylsulfonyl-phenyl)-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9150
PI4KBPIKAtypical8q6hAA3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-7-[(4-fluorosulfonyloxyphenyl)methylamino]-2,5-dimethyl-pyrazolo[1,5-a]pyrimidineHuman15015
PI4KBPIKAtypical4d0mQn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9145
PI4KBPIKAtypical5fbrA~{n}-[2-[[3-[3-[(4-azanylcyclohexyl)sulfamoyl]-4-methoxy-phenyl]-6-chloranyl-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9140
PI4KBPIKAtypical8q6fAC3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidineHuman15011
PIK3C3PIKAtypical3ihyB-Human9336
PIK3C3PIKAtypical3ihyE-Human9344
ANTXR1 (DNAPK)PIKKAtypical6zh2A-Human12927
ANTXR1 (DNAPK)PIKKAtypical7su3AAadenosine-5'-triphosphateHuman14058
ANTXR1 (DNAPK)PIKKAtypical6zheA-Human12928
ANTXR1 (DNAPK)PIKKAtypical7sglAAadenosine-5'-triphosphateHuman14059
ANTXR1 (DNAPK)PIKKAtypical6zh6A-Human12929
ANTXR1 (DNAPK)PIKKAtypical7sudABadenosine-5'-triphosphateHuman14060
ANTXR1 (DNAPK)PIKKAtypical7z87AB(~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanolHuman14593
ANTXR1 (DNAPK)PIKKAtypical7otvA(1s,6br,9as,11r,11br)-9a,11b-dimethyl-1-[(methyloxy)methyl]-3,6,9-trioxo-1,6,6b,7,8,9,9a,10,11,11b-decahydro-3h-furo[4,3,2-de]indeno[4,5-h][2]benzopyran-11-yl acetateHuman14063
ANTXR1 (DNAPK)PIKKAtypical7nfcA-Human13852
ANTXR1 (DNAPK)PIKKAtypical6zhaA-Human12931
ANTXR1 (DNAPK)PIKKAtypical7z88A(~{s})-[2-chloranyl-4-fluoranyl-5-(7-morpholin-4-ylquinazolin-4-yl)phenyl]-(6-methoxypyridazin-3-yl)methanolHuman14594
ATMPIKKAtypical7ni6Aphosphothiophosphoric acid-adenylate esterHuman13862
ATMPIKKAtypical5np0B-Human9266
ATMPIKKAtypical7sicAphosphoaminophosphonic acid-adenylate esterHuman14101
ATMPIKKAtypical5np0A-Human9267
PIK3CG (p110g)PIKAtypical8dp0A-Human14838
PIK3CA (p110a)PIKAtypical8tscA-Human15084
PIK3CA (p110a)PIKAtypical8tsbA-Human15085
PIK3CA (p110a)PIKAtypical8tsaA-Human15087
PIK3CA (p110a)PIKAtypical8ts7A-Human15088
PIK3CA (p110a)PIKAtypical8ts9A-Human15089
ATMPIKKAtypical7ni5A2-morpholin-4-yl-6-thianthren-1-yl-pyran-4-oneHuman13863
ATMPIKKAtypical6k9kA-Human11897
ATRPIKKAtypical9l4dAcamonsertibHuman15644
ATRPIKKAtypical23fcAphosphothiophosphoric acid-adenylate esterHuman15653
ATRPIKKAtypical9zcyAphosphoaminophosphonic acid-adenylate esterHuman15654
ATRPIKKAtypical9zd3Aphosphoaminophosphonic acid-adenylate esterHuman15655
ATRPIKKAtypical26znAphosphothiophosphoric acid-adenylate esterHuman15656
ATRPIKKAtypical23feAphosphothiophosphoric acid-adenylate esterHuman15657
ATRPIKKAtypical5yz0B-Human9524
ATRPIKKAtypical9l4bAcamonsertibHuman15658
PIK3CA (p110a)PIKAtypical7myoBA-Human13962
PIK3CA (p110a)PIKAtypical5fi4AA~{n}-[6-[5-azanyl-6-[(2~{s})-1,1,1-tris(fluoranyl)propan-2-yl]oxy-pyrazin-2-yl]imidazo[1,2-a]pyridin-2-yl]ethanamideHuman9302
PIK3CA (p110a)PIKAtypical6oacA4-(difluoromethyl)-5-{4-[(3s)-3-methylmorpholin-4-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}pyridin-2-amineHuman11381
PIK3CA (p110a)PIKAtypical4tuuA-Human9281
PIK3CA (p110a)PIKAtypical5ul1AB3-amino-6-(4-{[(2s)-1-(dimethylamino)propan-2-yl]sulfonyl}phenyl)-n-phenylpyrazine-2-carboxamideHuman9308
PIK3CA (p110a)PIKAtypical5sxfA-Human9284
PIK3CA (p110a)PIKAtypical8tduABn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14969
PIK3CA (p110a)PIKAtypical8ts8A-Human15086
PI4K2APIKAtypical4hneAadenosine-5'-diphosphateHuman9262
PI4KBPIKAtypical5fbqA~{n}-[2-[[6-chloranyl-3-[3-[4-(hydroxymethyl)piperidin-1-yl]sulfonyl-4-methoxy-phenyl]-2-methyl-imidazo[1,2-b]pyridazin-8-yl]amino]ethyl]ethanamideHuman9131
PIK3CA (p110a)PIKAtypical7jiuAB(3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-oneHuman13761
PIK3CA (p110a)PIKAtypical5sxeA-Human9280
PIK3CA (p110a)PIKAtypical5xghA3-[(4-fluorophenyl)methylamino]-5-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenolHuman9864
PIK3CA (p110a)PIKAtypical4wafAAn,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamideHuman9288
PIK3CA (p110a)PIKAtypical5sxkA-Human9296
PIK3CA (p110a)PIKAtypical7k6mAB2,2-difluoroethyl (3s)-3-{[2'-amino-5-fluoro-2-(morpholin-4-yl)[4,5'-bipyrimidin]-6-yl]amino}-3-(hydroxymethyl)pyrrolidine-1-carboxylateHuman13227
PIK3CA (p110a)PIKAtypical7r9yAn-[2-(4-{4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethyl]-n-methyl-1-(prop-2-enoyl)piperidine-4-carboxamideHuman14179
PIK3CA (p110a)PIKAtypical3hhmA(1s,6br,9as,11r,11br)-9a,11b-dimethyl-1-[(methyloxy)methyl]-3,6,9-trioxo-1,6,6b,7,8,9,9a,10,11,11b-decahydro-3h-furo[4,3,2-de]indeno[4,5-h][2]benzopyran-11-yl acetateHuman9275
MTOR (FRAP)PIKKAtypical7uxcA-Human14525
MTOR (FRAP)PIKKAtypical4jsvAadenosine-5'-diphosphateHuman9109
MTOR (FRAP)PIKKAtypical6sb2B-Human11726
MTOR (FRAP)PIKKAtypical7pebA-Human13869
MTOR (FRAP)PIKKAtypical4jsxB9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-oneHuman9111
MTOR (FRAP)PIKKAtypical9f45A-Human15315
MTOR (FRAP)PIKKAtypical5h64a-Human9110
PIK3CD (p110d)PIKAtypical7lq1An-(5-(6-(2-((2s,6r)-2,6-dimethylmorpholino)pyridin-4-yl)-1-oxoisoindolin-4-yl)-2-methoxypyridin-3-yl)methanesulfonamideHuman14106
RIOK2RIOAtypical6fdmABphosphoaminophosphonic acid-adenylate esterHuman10877
RIOK2RIOAtypical6fdmDB-Human10872
RIOK2RIOAtypical6hk6G2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10640
RIOK2RIOAtypical6g51v-Human9985
RIOK2RIOAtypical6hk6H2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10632
RIOK2RIOAtypical6fdoB-Human10870
PIK3CG (p110g)PIKAtypical8sc8AAn-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamideHuman15289
PIK3CG (p110g)PIKAtypical8sc8ACn-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamideHuman15290
PIK3CG (p110g)PIKAtypical8sc8ABn-[(5p)-2-chloro-5-(4-{[(1r)-1-phenylethyl]amino}quinazolin-6-yl)pyridin-3-yl]methanesulfonamideHuman15291
PIK3CG (p110g)PIKAtypical4fhkA3-[2-methyl-6-(pyrazin-2-ylamino)pyrimidin-4-yl]-n-(1h-pyrazol-3-yl)imidazo[1,2-b]pyridazin-2-amineHuman9204
PIK3CG (p110g)PIKAtypical1e8yA-Human9248
PIK3CG (p110g)PIKAtypical3ml8A8-cyclopentyl-6-[3-(hydroxymethyl)phenyl]-4-methyl-2-(methylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman9192
PIK3CA (p110a)PIKAtypical5sxjA-Human9301
PIK3CA (p110a)PIKAtypical5dxtA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHuman9299
PIK3CA (p110a)PIKAtypical9xw5AB-Human16019
PIK3CA (p110a)PIKAtypical5xgjA3-(4-morpholin-4-ylfuro[3,2-d]pyrimidin-2-yl)-5-[(phenylmethyl)amino]phenolHuman9863
PIK3CA (p110a)PIKAtypical8ow2AB-Human14764
PIK3CA (p110a)PIKAtypical9b4sA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHuman16024
PIK3CA (p110a)PIKAtypical8dcpAA-Human14380
PIK3CA (p110a)PIKAtypical5swtA-Human9273
PIK3CA (p110a)PIKAtypical4zopAA(2s,3r)-n~1~-(8-tert-butyl-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-2-yl)-3-methylpyrrolidine-1,2-dicarboxamideHuman9298
PIK3CA (p110a)PIKAtypical5xgiA3-azanyl-5-(4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenolHuman9865
PIK3CA (p110a)PIKAtypical5swpA-Human9293
PIK3CA (p110a)PIKAtypical5sxdA-Human9304
PIK3CA (p110a)PIKAtypical9xw7AB-Human16025
PIK3CA (p110a)PIKAtypical5dxhAmethyl {2-[4-(2-chlorophenyl)-4h-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl}carbamateHuman9310
PIK3CA (p110a)PIKAtypical4zopAB(2s,3r)-n~1~-(8-tert-butyl-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-2-yl)-3-methylpyrrolidine-1,2-dicarboxamideHuman9312
PIK3CA (p110a)PIKAtypical8sbcAB(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(pyridin-2-yl)-1h-imidazo[4,5-b]pyridineHuman14842
PIK3CA (p110a)PIKAtypical7myoBB-Human13965
PIK3CA (p110a)PIKAtypical7pg6AB(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14349
PIK3CA (p110a)PIKAtypical4yknAA3-(6-methoxypyridin-3-yl)-5-[({4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl}amino)methyl]benzoic acidHuman9283
PIK3CA (p110a)PIKAtypical6nctA-Human11221
PIK3CA (p110a)PIKAtypical8ilrABn-[(2s)-1-(ethylamino)-1-oxidanylidene-3-[4-(2-quinoxalin-6-ylethynyl)phenyl]propan-2-yl]-2,3-dimethyl-quinoxaline-6-carboxamideHuman14973
PIK3CA (p110a)PIKAtypical9nidA-Human16026
PIK3CA (p110a)PIKAtypical9nlcA-Human16027
PIK3CA (p110a)PIKAtypical9xw8AA-Human16028
PIK3CA (p110a)PIKAtypical9xw5AA-Human16029
ANTXR1 (DNAPK)PIKKAtypical7k1nA-Human13210
ANTXR1 (DNAPK)PIKKAtypical5luqA-Human9321
ANTXR1 (DNAPK)PIKKAtypical7k1kA-Human13211
TRRAPPIKKAtypical8h7gA-Human14556
TRRAPPIKKAtypical8xvgAAadenosine-5'-diphosphateHuman15321
TRRAPPIKKAtypical8qriA-Human15322
RIOK1RIOAtypical6zv6IA-Human13546
RIOK1RIOAtypical6zv6IB-Human13545
RIOK1RIOAtypical6zxfzadenosine-5'-triphosphateHuman13010
RIOK1RIOAtypical6zxez-Human13011
RIOK1RIOAtypical4otpAadenosine-5'-diphosphateHuman9156
RIOK1RIOAtypical6zxgzadenosine-5'-triphosphateHuman13012
RIOK1RIOAtypical6zxdz-Human13013
PIK3CG (p110g)PIKAtypical4aofAn-[6-(5-methylsulfonylpyridin-3-yl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]ethanamideHuman9245
PIK3CG (p110g)PIKAtypical4wwoAn-{(1s)-1-[8-chloro-2-(3-fluorophenyl)quinolin-3-yl]ethyl}-9h-purin-6-amineHuman9190
PIK3CG (p110g)PIKAtypical4kz0Amethyl 2-(acetylamino)-1,3-benzothiazole-6-carboxylateHuman9161
PIK3CG (p110g)PIKAtypical5jhbA[1-{4-[6-amino-4-(trifluoromethyl)pyridin-3-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}-3-(chloromethyl)azetidin-3-yl]methanolHuman9238
PIK3CG (p110g)PIKAtypical3l13A[3-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)phenyl]methanolHuman9167
PIK3CG (p110g)PIKAtypical7z61A9-[(3~{r},4~{r})-4-fluoranylpyrrolidin-3-yl]-7-methyl-2-[(7-methylquinolin-6-yl)amino]purin-8-oneHuman14286
PIK3CG (p110g)PIKAtypical4anwAA3-amino-6-{4-chloro-3-[(2,3-difluorophenyl)sulfamoyl]phenyl}-n-methylpyrazine-2-carboxamideHuman9174
PIK3CG (p110g)PIKAtypical7kkeAn-[2-(3,3-dimethylbutoxy)ethyl]-n'-{4-methyl-5-[(pyridin-4-yl)ethynyl]-1,3-thiazol-2-yl}ureaHuman13433
PIK3CG (p110g)PIKAtypical3ml9A2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman9187
PIK3CG (p110g)PIKAtypical3l08AB2,4-difluoro-n-[2-methoxy-5-(4-pyridazin-4-ylquinolin-6-yl)pyridin-3-yl]benzenesulfonamideHuman9164
PIK3CG (p110g)PIKAtypical3p2bAB3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenolHuman9165
PIK3CG (p110g)PIKAtypical3p2bAA3-[2-morpholin-4-yl-6-(pyridin-3-ylamino)pyrimidin-4-yl]phenolHuman9169
PIK3CG (p110g)PIKAtypical4fa6A2-amino-8-cyclopentyl-4-methyl-6-(1h-pyrazol-4-yl)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman9191
PIK3CG (p110g)PIKAtypical4ezjA2-(1-{[2-(5-fluoro-1h-indol-4-yl)-4-(morpholin-4-yl)pyrido[3,2-d]pyrimidin-6-yl]methyl}piperidin-4-yl)propan-2-olHuman9222
PIK3CG (p110g)PIKAtypical4fadA2-amino-6-(5-fluoro-6-methoxypyridin-3-yl)-4-methyl-8-(pyrrolidin-1-yl)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman9202
PIK3CG (p110g)PIKAtypical2chxAn-(2,3-dihydro-7,8-dimethoxyimidazo[1,2-c] quinazolin-5-yl)nicotinamideHuman9247
PIK3CG (p110g)PIKAtypical4f1sAn-(5-{[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-5-(tetrahydro-2h-pyran-4-yl)pyridin-2-yl]amino}-2-chloropyridin-3-yl)methanesulfonamideHuman9221
PIK3CG (p110g)PIKAtypical5edsA4-azanyl-6-[[(1~{s})-1-[6-fluoranyl-1-(3-methylsulfonylphenyl)benzimidazol-2-yl]ethyl]amino]pyrimidine-5-carbonitrileHuman9208
PIK3CG (p110g)PIKAtypical3csfA-Human9215
PIK3CG (p110g)PIKAtypical3l17A4-methyl-5-(6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-ylthieno[3,2-d]pyrimidin-2-yl)pyrimidin-2-amineHuman9185
PIK3CG (p110g)PIKAtypical2a4zA(5e)-5-[(2,2-difluoro-1,3-benzodioxol-5-yl)methylene]-1,3-thiazolidine-2,4-dioneHuman9180
PIK3CG (p110g)PIKAtypical7jwzA2-amino-n-[(1s)-1-{8-[(1-methyl-1h-pyrazol-4-yl)ethynyl]-1-oxo-2-phenyl-1,2-dihydroisoquinolin-3-yl}ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman13410
PIK3CG (p110g)PIKAtypical3tjpAn~6~-(3,4-dimethoxyphenyl)-2-(morpholin-4-yl)-4,5'-bipyrimidine-2',6-diamineHuman9234
PIK3CG (p110g)PIKAtypical3nzuA6-(2h-indazol-4-yl)-1-methyl-n-[3-(methylsulfonyl)propyl]-1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman9177
PIK3CG (p110g)PIKAtypical4j6iA2-methyl-1-(4-{2-[1-(2,2,2-trifluoroethyl)-1h-1,2,4-triazol-5-yl]-4,5-dihydro[1]benzoxepino[5,4-d][1,3]thiazol-8-yl}-1h-pyrazol-1-yl)propan-2-olHuman9189
PIK3CG (p110g)PIKAtypical4hvbA1-{1-[(2s)-2-hydroxypropanoyl]piperidin-4-yl}-3-methyl-8-(6-methylpyridin-3-yl)-1,3-dihydro-2h-imidazo[4,5-c][1,5]naphthyridin-2-oneHuman9225
PIK3CG (p110g)PIKAtypical3s2aAn-{2-chloro-5-[4-(morpholin-4-yl)quinolin-6-yl]pyridin-3-yl}-4-fluorobenzenesulfonamideHuman9158
PIK3CG (p110g)PIKAtypical4fulA4-({4-[3-(piperidin-1-ylcarbonyl)phenyl]pyrimidin-2-yl}amino)benzenesulfonamideHuman9242
PIK3CG (p110g)PIKAtypical4wwnAn-{(1s)-1-[7-fluoro-2-(pyridin-2-yl)quinolin-3-yl]ethyl}-9h-purin-6-amineHuman9226
PIK3CG (p110g)PIKAtypical5oq4AB5-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-4-(trifluoromethyl)pyridin-2-amineHuman9203
PIK3CG (p110g)PIKAtypical3dbsA2-(1h-indazol-4-yl)-6-{[4-(methylsulfonyl)piperazin-1-yl]methyl}-4-morpholin-4-yl-thieno[3,2-d]pyrimidineHuman9230
PIK3CG (p110g)PIKAtypical6audAA10-[(s)-(1-tert-butylpiperidin-4-yl)sulfinyl]-2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepineHuman9239
PIK3CG (p110g)PIKAtypical6t3bA2-[(4-methoxy-2-methyl-phenyl)amino]-7-methyl-9-(4-oxidanylcyclohexyl)purin-8-oneHuman11906
PIK3CG (p110g)PIKAtypical3r7rA8-(acetylamino)-n-(2-chlorophenyl)-n-methyl-4,5-dihydrothieno[3,2-d][1]benzoxepine-2-carboxamideHuman9168
PIK3CG (p110g)PIKAtypical4anvAB2-{4-[(4'-methoxybiphenyl-3-yl)sulfonyl]piperazin-1-yl}-3-(4-methoxyphenyl)pyrazineHuman9166
PIK3CG (p110g)PIKAtypical4fjyA4-[3,3-dimethyl-6-(morpholin-4-yl)-2,3-dihydro-1h-indol-1-yl]-7-fluoro-3-methyl-2-(pyridin-3-yl)quinolineHuman9249
PIK3CG (p110g)PIKAtypical3apfA3-[7-(1h-benzimidazol-5-yl)-2-(morpholin-4-yl)-6,7-dihydro-5h-pyrrolo[2,3-d]pyrimidin-4-yl]phenolHuman9250
PIK3CG (p110g)PIKAtypical2a5uA(5e)-5-(quinoxalin-6-ylmethylene)-1,3-thiazolidine-2,4-dioneHuman9183
PIK3CG (p110g)PIKAtypical4ps3A1-[6-(5-methoxypyridin-3-yl)-1,3-benzothiazol-2-yl]-3-[2-(1-propyl-1h-imidazol-4-yl)ethyl]ureaHuman9193
PIK3CG (p110g)PIKAtypical6gq7A3-methyl-1-(oxan-4-yl)-8-pyridin-3-yl-imidazo[4,5-c]quinolin-2-oneHuman10009
PIK3CG (p110g)PIKAtypical3mjwA(2z)-4,6-dihydroxy-2-[(8-methoxy-1,2,3,4-tetrahydropyrazino[1,2-a]indol-10-yl)methylidene]-1-benzofuran-3(2h)-oneHuman9229
PIK3CG (p110g)PIKAtypical3qjzAn-{6-[2-(methylsulfanyl)pyrimidin-4-yl]-1,3-benzothiazol-2-yl}acetamideHuman9181
PIK3CG (p110g)PIKAtypical4gb9A2-[1-({2-[2-(dimethylamino)-1h-benzimidazol-1-yl]-9-methyl-6-(morpholin-4-yl)-9h-purin-8-yl}methyl)piperidin-4-yl]propan-2-olHuman9218
PIK3CG (p110g)PIKAtypical4hleA2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepine-8-carboxamideHuman9219
PIK3CD (p110d)PIKAtypical6g6wAB~{n}-[3-[4-[[(1~{s})-1-(5-methyl-4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-5-oxidanyl-phenyl]methanesulfonamideHuman10674
PIK3CD (p110d)PIKAtypical7jisA(3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-oneHuman13201
PIK3CD (p110d)PIKAtypical6g6wAA~{n}-[3-[4-[[(1~{s})-1-(5-methyl-4-oxidanylidene-3-phenyl-pyrrolo[2,1-f][1,2,4]triazin-2-yl)ethyl]amino]-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]-5-oxidanyl-phenyl]methanesulfonamideHuman10673
PIK3CD (p110d)PIKAtypical9gdiA3-[(1s)-1-[4-azanyl-3-(3-fluoranyl-5-oxidanyl-phenyl)pyrazolo[3,4-d]pyrimidin-1-yl]ethyl]-4-(1-methyl-3,6-dihydro-2h-pyridin-4-yl)isochromen-1-oneHuman15480
PIK3CD (p110d)PIKAtypical7lm2Acyclopropyl[(3s)-3-{[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]amino}pyrrolidin-1-yl]methanoneHuman13532
PIK3CD (p110d)PIKAtypical5vlrA4-acetyl-1-(3-{4-amino-5-[1-(2,2,2-trifluoroethyl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)-3,3-dimethylpiperazin-2-oneHuman9090
PIK3CD (p110d)PIKAtypical5t8fA2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamideHuman9093
PIK3CD (p110d)PIKAtypical6pyuA(3s)-1'-(cyclopropanecarbonyl)-5-(quinoxalin-6-yl)spiro[indole-3,2'-pyrrolidin]-2(1h)-oneHuman11548
PIK3CD (p110d)PIKAtypical6ocoA4-[(1s,4s)-5-(3-chlorophenyl)-2,5-diazabicyclo[2.2.1]heptan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carbonitrileHuman11865
PIK3CD (p110d)PIKAtypical8bcyAA9-[2-(3,4-dichlorophenyl)ethyl]-2-(3-hydroxyphenyl)-8-oxidanylidene-7~{h}-purine-6-carboxamideHuman14735
PIK3C3PIKAtypical6ykgA4-morpholin-4-yl-6-[(2~{r})-2-(phenylmethyl)pyrrolidin-1-yl]-1~{h}-pyridin-2-oneHuman13509
PIK3C3PIKAtypical4uwgAB-Human9350
PIK3C3PIKAtypical7rsjAAn-{4-[(7r,8r)-4-oxo-7-(propan-2-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-2-yl]pyridin-2-yl}cyclopropanecarboxamideHuman13983
PIK3C3PIKAtypical9tw2A-Human15515
PIK3C3PIKAtypical9rx4A-Human15516
PIK3C3PIKAtypical7rsvAB(5as,8ar,9s)-2-[(3r)-3-methylmorpholin-4-yl]-5,5a,6,7,8,8a-hexahydro-4h-cyclopenta[e]pyrazolo[1,5-a]pyrazin-4-oneHuman13984
PI4KBPIKAtypical4d0lEn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9139
PI4KBPIKAtypical4d0mWn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9155
PI4KBPIKAtypical8q6fAB3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidineHuman15013
PI4KBPIKAtypical5c46E-Human9141
PI4KBPIKAtypical4d0mcn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9148
PI4KBPIKAtypical4d0mOn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9154
PI4KBPIKAtypical5c4gEn~2~-[7-(3,4-dimethoxyphenyl)quinoxalin-2-yl]-n-methylglycinamideHuman9135
PI4KBPIKAtypical4wagA6-chloro-3-(3,4-dimethoxyphenyl)-2-methylimidazo[1,2-b]pyridazin-8-amineHuman9137
PI4KBPIKAtypical8q6fAA3-(3-fluorosulfonyloxy-4-methoxy-phenyl)-2,5-dimethyl-7-(pyridin-4-ylmethylamino)pyrazolo[1,5-a]pyrimidineHuman15018
PI4KBPIKAtypical4d0mGn-(5-(4-chloro-3-(2-hydroxy-ethylsulfamoyl)- phenylthiazole-2-yl)-acetamideHuman9134
PI4KBPIKAtypical6gl3B-Human10443
ANTXR1 (DNAPK)PIKKAtypical7nfeA-Human13851
ANTXR1 (DNAPK)PIKKAtypical7otwA7-methyl-2-[(7-methyl-[1,2,4]triazolo[1,5-a]pyridin-6-yl)amino]-9-(oxan-4-yl)purin-8-oneHuman14056
ATRPIKKAtypical23eyAelimusertibHuman15645
ATRPIKKAtypical9l40Ave-822Human15646
ATRPIKKAtypical23faAgartisertibHuman15647
ATRPIKKAtypical23exAceralasertibHuman15648
ATRPIKKAtypical5yz0A-Human9523
ATRPIKKAtypical9l45Ave-822Human15649
ATRPIKKAtypical23ewAve-822Human15650
ATRPIKKAtypical13deAphosphoaminophosphonic acid-adenylate esterHuman15651
ATRPIKKAtypical9zd4Aphosphoaminophosphonic acid-adenylate esterHuman15652
ATRPIKKAtypical23fbAphosphothiophosphoric acid-adenylate esterHuman15659
ATRPIKKAtypical9l4fAphosphothiophosphoric acid-adenylate esterHuman15660
ATRPIKKAtypical9l46Aphosphothiophosphoric acid-adenylate esterHuman15661
MTOR (FRAP)PIKKAtypical9t94Aadenosine-5'-triphosphateHuman15763
MTOR (FRAP)PIKKAtypical9ed8Aphosphoaminophosphonic acid-adenylate esterHuman15764
MTOR (FRAP)PIKKAtypical7pe8A-Human13870
MTOR (FRAP)PIKKAtypical9f44A-Human15316
MTOR (FRAP)PIKKAtypical6sb0A-Human11727
MTOR (FRAP)PIKKAtypical3jbzAadenosine-5'-diphosphateHuman9113
MTOR (FRAP)PIKKAtypical7pe9A-Human13871
MTOR (FRAP)PIKKAtypical4jt5A2-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-1h-indol-5-olHuman9116
MTOR (FRAP)PIKKAtypical8eraA1-[6-{[(3m)-4-amino-3-(2-amino-1,3-benzoxazol-5-yl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]methyl}-3,4-dihydroisoquinolin-2(1h)-yl]-3-hydroxypropan-1-oneHuman14569
MTOR (FRAP)PIKKAtypical6zwoBphosphothiophosphoric acid-adenylate esterHuman12987
MTOR (FRAP)PIKKAtypical7pe7A-Human13901
MTOR (FRAP)PIKKAtypical4jt6B3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenolHuman9102
MTOR (FRAP)PIKKAtypical5h64A-Human9099
MTOR (FRAP)PIKKAtypical6sb2A-Human11724
MTOR (FRAP)PIKKAtypical5flcBB-Human9108
MTOR (FRAP)PIKKAtypical6sb0B-Human11725
MTOR (FRAP)PIKKAtypical5wbuA-Human9407
MTOR (FRAP)PIKKAtypical4jsvBadenosine-5'-diphosphateHuman9100
MTOR (FRAP)PIKKAtypical4jt6A3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenolHuman9103
MTOR (FRAP)PIKKAtypical5zcsA-Human9748
MTOR (FRAP)PIKKAtypical6zwmBphosphothiophosphoric acid-adenylate esterHuman12988
MTOR (FRAP)PIKKAtypical5wbyB-Human9406
MTOR (FRAP)PIKKAtypical4jspBphosphothiophosphoric acid-adenylate esterHuman9107
MTOR (FRAP)PIKKAtypical4jt5B2-[4-amino-1-(propan-2-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-yl]-1h-indol-5-olHuman9104
MTOR (FRAP)PIKKAtypical6zwmAphosphothiophosphoric acid-adenylate esterHuman12989
MTOR (FRAP)PIKKAtypical5flcFB-Human9117
MTOR (FRAP)PIKKAtypical4jsxA9-(6-aminopyridin-3-yl)-1-[3-(trifluoromethyl)phenyl]benzo[h][1,6]naphthyridin-2(1h)-oneHuman9112
MTOR (FRAP)PIKKAtypical5wbyA-Human9404
MTOR (FRAP)PIKKAtypical7pecA-Human13872
MTOR (FRAP)PIKKAtypical5flcBA-Human9105
MTOR (FRAP)PIKKAtypical7peaA-Human13873
MTOR (FRAP)PIKKAtypical5wbuB-Human9405
MTOR (FRAP)PIKKAtypical4jsnB-Human9115
MTOR (FRAP)PIKKAtypical4jsnA-Human9114
MTOR (FRAP)PIKKAtypical7tzoA-Human14575
MTOR (FRAP)PIKKAtypical5flcFA-Human9101
RIOK2RIOAtypical6hk6C2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10639
RIOK2RIOAtypical6hk6F2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10637
RIOK2RIOAtypical6fdnA-Human10873
PI4K2BPIKAtypical4wtvAAadenosine-5'-triphosphateHuman9095
RIOK2RIOAtypical6fdnB-Human10867
RIOK2RIOAtypical6fdmAAphosphoaminophosphonic acid-adenylate esterHuman10875
RIOK2RIOAtypical6fdmDA-Human10868
RIOK2RIOAtypical6hk6E2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10633
RIOK2RIOAtypical6hk6B2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10636
RIOK2RIOAtypical6fdmBA-Human10869
RIOK2RIOAtypical7vbtA8-(6-methoxypyridin-3-yl)-1-[4-piperazin-1-yl-3-(trifluoromethyl)phenyl]-5h-[1,2,3]triazolo[4,5-c]quinolin-4-oneHuman14274
RIOK2RIOAtypical6fdoA-Human10878
RIOK2RIOAtypical6fdmBB-Human10871
RIOK2RIOAtypical6g18v-Human9986
RIOK2RIOAtypical6hk6A2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10638
RIOK2RIOAtypical6hk6I2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10631
RIOK2RIOAtypical6fdmCAphosphoaminophosphonic acid-adenylate esterHuman10874
RIOK2RIOAtypical6fdmCBphosphoaminophosphonic acid-adenylate esterHuman10876
RIOK2RIOAtypical6hk6D2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10634
RIOK2RIOAtypical6hk6J2-naphthalen-2-yl-~{n}-pyridin-2-yl-ethanamideHuman10635
RIOK2RIOAtypical9f81An-(4-quinazolin-4-ylphenyl)propanamideHuman15836
RIOK1RIOAtypical6zxhzadenosine-5'-triphosphateHuman13073
COQ8A (ADCK3)ABC1Atypical7udqA4-[(3,4,5-trimethoxyphenyl)amino]quinoline-7-carbonitrileHuman14588
COQ8A (ADCK3)ABC1Atypical7udpA4-[(3,4,5-trimethoxyphenyl)amino]quinoline-7-carbonitrileHuman14589
PIK3CA (p110a)PIKAtypical9lwsA-Human16011
PIK3CA (p110a)PIKAtypical6gviAA3-(2-azanyl-1,3-benzoxazol-5-yl)-1-propan-2-yl-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman11656
PIK3CA (p110a)PIKAtypical9ni8A-Human16007
PIK3CA (p110a)PIKAtypical5itdA5-{4-[3-(4-acetylpiperazine-1-carbonyl)phenyl]quinazolin-6-yl}-2-methoxypyridine-3-carbonitrileHuman9313
PIK3CA (p110a)PIKAtypical8tduAAn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14967
PIK3CA (p110a)PIKAtypical5sx9A-Human9305
PIK3CA (p110a)PIKAtypical8sbjAA(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(1h-pyrazol-3-yl)-3h-imidazo[4,5-b]pyridineHuman14839
PIK3CA (p110a)PIKAtypical9cmvA-Human16008
PIK3CA (p110a)PIKAtypical6gviAB3-(2-azanyl-1,3-benzoxazol-5-yl)-1-propan-2-yl-pyrazolo[3,4-d]pyrimidine-4,6-diamineHuman11654
PIK3CA (p110a)PIKAtypical4l1bA-Human9292
PIK3CA (p110a)PIKAtypical8bfuA-Human14613
PIK3CA (p110a)PIKAtypical8dd8A-Human14375
PIK3CA (p110a)PIKAtypical9lwrAA-Human16009
PIK3CA (p110a)PIKAtypical7k6nABtert-butyl (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-3-methylpyrrolidine-1-carboxylateHuman13224
PIK3CA (p110a)PIKAtypical6gvfAB5-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11658
PIK3CA (p110a)PIKAtypical6gvfAA5-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11659
PIK3CA (p110a)PIKAtypical7mynAA-Human13963
PIK3CA (p110a)PIKAtypical8am0A(2r)-2-[[2-[(4s)-4-[bis(fluoranyl)methyl]-2-oxidanylidene-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl]amino]propanamideHuman15083
PIK3CA (p110a)PIKAtypical5swgA-Human9306
PIK3CA (p110a)PIKAtypical7r9vAn-[2-(4-{4-[2-amino-4-(difluoromethyl)pyrimidin-5-yl]-6-(morpholin-4-yl)-1,3,5-triazin-2-yl}piperazin-1-yl)-2-oxoethyl]-1-(prop-2-enoyl)piperidine-4-carboxamideHuman14178
PIK3CA (p110a)PIKAtypical5swrA-Human9279
PIK3CA (p110a)PIKAtypical9ni7A-Human16010
PIK3CA (p110a)PIKAtypical7k71A2-(morpholin-4-yl)[4,5'-bipyrimidin]-2'-amineHuman13219
PIK3CA (p110a)PIKAtypical7pg5AA-Human14346
PIK3CA (p110a)PIKAtypical8dcpAB-Human14376
PIK3CA (p110a)PIKAtypical5ul1AA3-amino-6-(4-{[(2s)-1-(dimethylamino)propan-2-yl]sulfonyl}phenyl)-n-phenylpyrazine-2-carboxamideHuman9316
PIK3CA (p110a)PIKAtypical7k6oAB(3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-n-methylpyrrolidine-1-sulfonamideHuman13206
PIK3CA (p110a)PIKAtypical7pg5AB-Human14347
PIK3CA (p110a)PIKAtypical8sbjAB(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(1h-pyrazol-3-yl)-3h-imidazo[4,5-b]pyridineHuman14840
PIK3CA (p110a)PIKAtypical5sxaA-Human9285
PIK3CA (p110a)PIKAtypical9b4tA(2s)-2-({2-[1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}oxy)propanamideHuman16012
PIK3CA (p110a)PIKAtypical7jiuAA(3s)-3-benzyl-5-[9-ethyl-8-(2-methylpyrimidin-5-yl)-9h-purin-6-yl]-3-methyl-1,3-dihydro-2h-indol-2-oneHuman13760
PIK3CA (p110a)PIKAtypical4wafABn,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamideHuman9272
PIK3CA (p110a)PIKAtypical6gvhAA5-(6-azanyl-4-chloranyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11657
PIK3CA (p110a)PIKAtypical8exlAB2-methyl-2-(4-{2-[3-methyl-1-(propan-2-yl)-1h-1,2,4-triazol-5-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-1h-pyrazol-1-yl)propanamideHuman14536
PIK3CA (p110a)PIKAtypical5ubrA1-[4-(3-{4-amino-5-[1-(oxan-4-yl)-1h-pyrazol-5-yl]pyrrolo[2,1-f][1,2,4]triazin-7-yl}phenyl)piperazin-1-yl]ethan-1-oneHuman9289
PIK3CA (p110a)PIKAtypical7k6mAA2,2-difluoroethyl (3s)-3-{[2'-amino-5-fluoro-2-(morpholin-4-yl)[4,5'-bipyrimidin]-6-yl]amino}-3-(hydroxymethyl)pyrrolidine-1-carboxylateHuman13225
PIK3CA (p110a)PIKAtypical4jpsAA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman9317
PIK3CA (p110a)PIKAtypical8dcxA-Human14377
PIK3CA (p110a)PIKAtypical9ni5A-Human16013
PIK3CA (p110a)PIKAtypical9xw7AA-Human16014
PIK3CA (p110a)PIKAtypical7k6nAAtert-butyl (3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-3-methylpyrrolidine-1-carboxylateHuman13226
PIK3CA (p110a)PIKAtypical3zimA1-[4-[[2-(1h-indazol-4-yl)-4-morpholin-4-yl-thieno[3,2-d]pyrimidin-6-yl]methyl]piperazin-1-yl]-6-methyl-hept-5-ene-1,4-dioneHuman9294
PIK3CA (p110a)PIKAtypical5sw8A-Human9274
PIK3CA (p110a)PIKAtypical4tv3A2-amino-8-[trans-4-(2-hydroxyethoxy)cyclohexyl]-6-(6-methoxypyridin-3-yl)-4-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman9278
PIK3CA (p110a)PIKAtypical5uk8AA(r)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1h-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholineHuman9295
PIK3CA (p110a)PIKAtypical5ukjAn,n-dimethyl-4-[(6r)-6-methyl-5-(1h-pyrrolo[2,3-b]pyridin-4-yl)-4,5,6,7-tetrahydropyrazolo[1,5-a]pyrazin-3-yl]benzenesulfonamideHuman9277
PIK3CA (p110a)PIKAtypical7k6oAA(3s)-3-[4-(2-aminopyrimidin-5-yl)-2-(morpholin-4-yl)-5,6-dihydro-7h-pyrrolo[2,3-d]pyrimidin-7-yl]-n-methylpyrrolidine-1-sulfonamideHuman13207
PIK3CA (p110a)PIKAtypical2rd0A-Human9287
PIK3CA (p110a)PIKAtypical4l23A3-(4-morpholin-4-ylpyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl)phenolHuman9290
PIK3CA (p110a)PIKAtypical6pysAA(3s)-3-benzyl-3-methyl-5-[5-(2-methylpyrimidin-5-yl)pyrazolo[1,5-a]pyrimidin-3-yl]-1,3-dihydro-2h-indol-2-oneHuman11575
PIK3CA (p110a)PIKAtypical4l2yA3-amino-5-[4-(morpholin-4-yl)pyrido[3',2':4,5]furo[3,2-d]pyrimidin-2-yl]phenolHuman9276
PIK3CA (p110a)PIKAtypical6gvgA5-(6-azanyl-4-methyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11655
PIK3CA (p110a)PIKAtypical7tz7AB(4s,5r)-3-[2'-amino-2-(morpholin-4-yl)-4'-(trifluoromethyl)[4,5'-bipyrimidin]-6-yl]-4-(hydroxymethyl)-5-methyl-1,3-oxazolidin-2-oneHuman14222
PIK3CA (p110a)PIKAtypical3hizA-Human9311
PIK3CA (p110a)PIKAtypical9nieA-Human16015
PIK3CA (p110a)PIKAtypical4jpsAB(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman9314
PIK3CA (p110a)PIKAtypical8exvABn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14538
PIK3CA (p110a)PIKAtypical9lwqA-Human16016
PIK3CA (p110a)PIKAtypical9yf2An~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman16017
PIK3CA (p110a)PIKAtypical9ni3A-Human16018
PIK3CA (p110a)PIKAtypical5sxiA-Human9270
PIK3CA (p110a)PIKAtypical4yknAB3-(6-methoxypyridin-3-yl)-5-[({4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfamoyl]phenyl}amino)methyl]benzoic acidHuman9315
PIK3CA (p110a)PIKAtypical8exuAA(2s)-2-cyclopropyl-2-({(4s,11am)-2-[(4s)-2-oxo-4-(trifluoromethyl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}amino)acetamideHuman14539
PIK3CA (p110a)PIKAtypical8guaA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14540
PIK3CA (p110a)PIKAtypical9lwrAB-Human16020
PIK3CA (p110a)PIKAtypical5dxhDmethyl {2-[4-(2-chlorophenyl)-4h-1,2,4-triazol-3-yl]-4,5-dihydrothieno[3,2-d][1]benzoxepin-8-yl}carbamateHuman9300
PIK3CA (p110a)PIKAtypical5sx8A-Human9269
PIK3CA (p110a)PIKAtypical8sbcAA(2m)-7-[(3r)-3-methylmorpholin-4-yl]-5-[(3s)-3-methylmorpholin-4-yl]-2-(pyridin-2-yl)-1h-imidazo[4,5-b]pyridineHuman14841
PIK3CA (p110a)PIKAtypical9nifA-Human16021
PIK3CA (p110a)PIKAtypical8tgdAAn~2~-{(4s,11ap)-2-[(4s)-4-(difluoromethyl)-2-oxo-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}-l-alaninamideHuman14972
PIK3CA (p110a)PIKAtypical8dd4AA-Human14378
PIK3CA (p110a)PIKAtypical9c15A-Human16022
PIK3CA (p110a)PIKAtypical8dd4AB-Human14379
PIK3CA (p110a)PIKAtypical9xw8AB-Human16023
PIK3CA (p110a)PIKAtypical6gvhAB5-(6-azanyl-4-chloranyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-1,3-benzoxazol-2-amineHuman11653
PIK3CA (p110a)PIKAtypical5sxcA-Human9297
PIK3CA (p110a)PIKAtypical9ni4A-Human16030
PIK3CA (p110a)PIKAtypical8gubA(2s)-n~1~-{4-methyl-5-[2-(1,1,1-trifluoro-2-methylpropan-2-yl)pyridin-4-yl]-1,3-thiazol-2-yl}pyrrolidine-1,2-dicarboxamideHuman14543
PIK3CA (p110a)PIKAtypical8exuAB(2s)-2-cyclopropyl-2-({(4s,11am)-2-[(4s)-2-oxo-4-(trifluoromethyl)-1,3-oxazolidin-3-yl]-5,6-dihydroimidazo[1,2-d][1,4]benzoxazepin-9-yl}amino)acetamideHuman14544
PIK3CA (p110a)PIKAtypical5uk8AB(r)-4-(6-(1-(cyclopropylsulfonyl)cyclopropyl)-2-(1h-indol-4-yl)pyrimidin-4-yl)-3-methylmorpholineHuman9286
PI4K2APIKAtypical4hndAadenosine-5'-diphosphateHuman9265
PI4K2APIKAtypical4hneBadenosine-5'-diphosphateHuman9263
PI4K2APIKAtypical4plaAadenosine-5'-triphosphateHuman9259
PI4K2APIKAtypical4yc4A[(1s,3s,4s)-3-(6-amino-9h-purin-9-yl)bicyclo[2.2.1]hept-1-yl]methanolHuman9258
PI4K2APIKAtypical4hndBadenosine-5'-diphosphateHuman9261
PI4K2APIKAtypical5i0nABadenosine-5'-triphosphateHuman9257
ANTXR1 (DNAPK)PIKKAtypical5w1rA-Human9320
ANTXR1 (DNAPK)PIKKAtypical7otpAphosphothiophosphoric acid-adenylate esterHuman14054
ANTXR1 (DNAPK)PIKKAtypical6zh8A-Human12925
ANTXR1 (DNAPK)PIKKAtypical8bh3A-Human14768
ANTXR1 (DNAPK)PIKKAtypical7k1jA-Human13209
ANTXR1 (DNAPK)PIKKAtypical6zfpA-Human12926
ANTXR1 (DNAPK)PIKKAtypical7k0yAA-Human13213
ANTXR1 (DNAPK)PIKKAtypical8bhvA-Human14769
ANTXR1 (DNAPK)PIKKAtypical9qcsA-Human16044
ANTXR1 (DNAPK)PIKKAtypical7k0yAB-Human13214
ANTXR1 (DNAPK)PIKKAtypical7k17A-Human13215
ANTXR1 (DNAPK)PIKKAtypical7lt3Cadenosine-5'-diphosphateHuman13500
ANTXR1 (DNAPK)PIKKAtypical7lt3Ladenosine-5'-diphosphateHuman13501
ANTXR1 (DNAPK)PIKKAtypical9zp0K-Human16045
ANTXR1 (DNAPK)PIKKAtypical8rd4A-Human16046
ANTXR1 (DNAPK)PIKKAtypical6zh4A-Human12930
ANTXR1 (DNAPK)PIKKAtypical7k19A-Human13216
ANTXR1 (DNAPK)PIKKAtypical9g9lA-Human16047
ANTXR1 (DNAPK)PIKKAtypical7k10A-Human13217
ANTXR1 (DNAPK)PIKKAtypical9q9fE-Human16048
ANTXR1 (DNAPK)PIKKAtypical8bhyA-Human14770
ANTXR1 (DNAPK)PIKKAtypical7k1bA-Human13218
ANTXR1 (DNAPK)PIKKAtypical7tyrAA-Human14322
ANTXR1 (DNAPK)PIKKAtypical6zheF-Human12932
ANTXR1 (DNAPK)PIKKAtypical5y3rC-Human9318
ANTXR1 (DNAPK)PIKKAtypical9zp9M-Human16049
PI4KAPIKAtypical6bq1E5-{2-amino-1-[4-(morpholin-4-yl)phenyl]-1h-benzimidazol-6-yl}-n-(2-fluorophenyl)-2-methoxypyridine-3-sulfonamideHuman9069
PI4KAPIKAtypical6bq1A5-{2-amino-1-[4-(morpholin-4-yl)phenyl]-1h-benzimidazol-6-yl}-n-(2-fluorophenyl)-2-methoxypyridine-3-sulfonamideHuman9070
RIOK3RIOAtypical8zdbJ-Human16170
RIOK3RIOAtypical8zdcJ-Human16171
ATMPIKKAtypical5np1A-Human9268
ATMPIKKAtypical7sidAphosphoaminophosphonic acid-adenylate esterHuman14102
Kinome view
Your browser unfortunately does not support an HTML5 canvas. Your browser unfortunately does not support an HTML5 canvas.
 Download structures
Here are the search results - click on something ;-)
Feedback form

E-mail (optional)

Message

Please type the digits from the image into the input field (robot check):

Verification code:

Settings