| STK11 (LKB1) | CAMKL | CAMK | 8vsu | B | | adenosine-5'-diphosphate | Human | 15343 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7uir | A | | adenosine-5'-triphosphate | Human | 14173 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl1 | B | | adenosine-5'-triphosphate | Human | 13062 | |
| DAPK1 | DAPK | CAMK | 5aux | A | | 3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 6136 | |
| DAPK1 | DAPK | CAMK | 5auz | A | | genistein | Human | 6140 | |
| DAPK1 | DAPK | CAMK | 3gu7 | A | A | adenosine-5'-diphosphate | Human | 5624 | |
| DAPK1 | DAPK | CAMK | 3f5g | A | A | adenosine-5'-diphosphate | Human | 5635 | |
| DAPK1 | DAPK | CAMK | 1p4f | A | B | 5,6-dihydro-benzo[h]cinnolin-3-ylamine | Human | 5664 | |
| DAPK1 | DAPK | CAMK | 6qmo | A | A | - | Human | 11587 | |
| DAPK1 | DAPK | CAMK | 4yo4 | A | B | phthalazine | Human | 5649 | |
| DAPK1 | DAPK | CAMK | 3eha | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5687 | |
| DAPK1 | DAPK | CAMK | 2w4j | A | B | adenosine-5'-diphosphate | Human | 5682 | |
| DAPK1 | DAPK | CAMK | 7ccv | A | A | piceatannol | Human | 13232 | |
| DAPK1 | DAPK | CAMK | 3f5u | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5632 | |
| DAPK1 | DAPK | CAMK | 3f5g | A | B | adenosine-5'-diphosphate | Human | 5675 | |
| DAPK1 | DAPK | CAMK | 4pf4 | A | B | - | Human | 5648 | |
| DAPK1 | DAPK | CAMK | 3gub | A | A | 9-alpha-l-lyxofuranosyl-n-(2-phenylethyl)-9h-purin-6-amine | Human | 5674 | |
| DAPK1 | DAPK | CAMK | 3gu7 | A | B | adenosine-5'-diphosphate | Human | 5665 | |
| DAPK1 | DAPK | CAMK | 3eh9 | A | A | adenosine-5'-diphosphate | Human | 5621 | |
| DAPK1 | DAPK | CAMK | 1jkt | A | | - | Human | 5650 | |
| DAPK1 | DAPK | CAMK | 3eha | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5636 | |
| DAPK1 | DAPK | CAMK | 4b4l | A | B | - | Human | 5684 | |
| DAPK1 | DAPK | CAMK | 4uv0 | A | | - | Human | 5639 | |
| DAPK1 | DAPK | CAMK | 2x0g | A | B | - | Human | 5676 | |
| DAPK1 | DAPK | CAMK | 8ie5 | A | | trans-oxyresveratrol | Human | 14749 | |
| DAPK1 | DAPK | CAMK | 2y4p | C | | - | Human | 5688 | |
| DAPK1 | DAPK | CAMK | 5auy | A | | 2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-one | Human | 6134 | |
| DAPK1 | DAPK | CAMK | 1jkl | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5619 | |
| DAPK1 | DAPK | CAMK | 1wvw | A | | - | Human | 5652 | |
| DAPK1 | DAPK | CAMK | 7ccv | A | B | piceatannol | Human | 13233 | |
| DAPK1 | DAPK | CAMK | 7ccu | A | A | resveratrol | Human | 13234 | |
| MARK3 | CAMKL | CAMK | 7p1l | A | | 5-bromo-4-n-[2-(1h-imidazol-5-yl)ethyl]-2-n-[3-(morpholin-4-ylmethyl)phenyl]pyrimidine-2,4-diamine | Human | 13799 | |
| DAPK1 | DAPK | CAMK | 2w4k | A | B | adenosine-5'-diphosphate | Human | 5660 | |
| DAPK1 | DAPK | CAMK | 6qmo | A | B | - | Human | 11588 | |
| DAPK1 | DAPK | CAMK | 5av2 | A | | 3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 6133 | |
| DAPK1 | DAPK | CAMK | 1jkt | B | | - | Human | 5663 | |
| DAPK1 | DAPK | CAMK | 5auu | A | | 2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4h-chromen-4-one | Human | 6145 | |
| DAPK1 | DAPK | CAMK | 2w4k | A | A | adenosine-5'-diphosphate | Human | 5653 | |
| DAPK1 | DAPK | CAMK | 3f5u | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 5630 | |
| DAPK1 | DAPK | CAMK | 5av4 | A | A | genistein | Human | 6135 | |
| DAPK1 | DAPK | CAMK | 5av4 | A | B | genistein | Human | 6141 | |
| DAPK1 | DAPK | CAMK | 2xzs | B | A | - | Human | 5658 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | B | A | - | Human | 5573 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | A | A | - | Human | 6862 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | A | B | - | Human | 5569 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | B | B | - | Human | 5574 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | A | A | - | Human | 5572 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | A | B | - | Human | 5570 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | B | B | - | Human | 6861 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | D | A | - | Human | 5571 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | A | B | - | Human | 6859 | |
| TRIB2 (Trb2) | Trbl | CAMK | 7upm | A | | - | Human | 14365 | |
| DAPK3 | DAPK | CAMK | 5vja | C | A | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10345 | |
| DAPK3 | DAPK | CAMK | 2j90 | A | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 382 | |
| DAPK3 | DAPK | CAMK | 3bqr | A | B | 4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acid | Human | 386 | |
| DAPK3 | DAPK | CAMK | 5a6n | B | B | - | Human | 6161 | |
| MKNK1 (MNK1) | MAPKAPK | CAMK | 2hw6 | B | | - | Human | 2085 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7e | A | A | adenosine-5'-triphosphate | Human | 14520 | |
| DAPK1 | DAPK | CAMK | 3gu6 | A | B | adenosine-5'-diphosphate | Human | 5638 | |
| DAPK1 | DAPK | CAMK | 3gu6 | A | A | adenosine-5'-diphosphate | Human | 5631 | |
| DAPK1 | DAPK | CAMK | 6aar | A | | - | Human | 11468 | |
| DAPK1 | DAPK | CAMK | 1jks | A | B | - | Human | 5633 | |
| DAPK1 | DAPK | CAMK | 1jks | A | A | - | Human | 5657 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | B | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1633 | |
| PIM1 | PIM | CAMK | 4lmu | A | B | 3,5,7,3',4'-pentahydroxyflavone | Human | 2404 | |
| DAPK1 | DAPK | CAMK | 7ccw | A | B | resveratrol | Human | 13236 | |
| DAPK1 | DAPK | CAMK | 4b4l | A | A | - | Human | 5683 | |
| DAPK1 | DAPK | CAMK | 2y4p | D | | - | Human | 5640 | |
| DAPK1 | DAPK | CAMK | 3gub | A | B | 9-alpha-l-lyxofuranosyl-n-(2-phenylethyl)-9h-purin-6-amine | Human | 5673 | |
| DAPK1 | DAPK | CAMK | 6in4 | A | | - | Human | 11795 | |
| DAPK1 | DAPK | CAMK | 2xuu | A | | adenosine-5'-diphosphate | Human | 5627 | |
| DAPK1 | DAPK | CAMK | 3f5u | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5677 | |
| DAPK1 | DAPK | CAMK | 4yo4 | A | A | phthalazine | Human | 5686 | |
| DAPK1 | DAPK | CAMK | 2y4p | A | | - | Human | 5659 | |
| DAPK1 | DAPK | CAMK | 3eh9 | A | C | adenosine-5'-diphosphate | Human | 5655 | |
| DAPK1 | DAPK | CAMK | 4ypd | A | A | 4-methylpyridazine | Human | 5654 | |
| DAPK1 | DAPK | CAMK | 3zxt | B | | phosphomethylphosphonic acid adenylate ester | Human | 5666 | |
| DAPK1 | DAPK | CAMK | 3gu8 | A | A | n6-cyclopentyladenosine | Human | 5679 | |
| DAPK1 | DAPK | CAMK | 6fhb | A | B | - | Human | 11291 | |
| DAPK1 | DAPK | CAMK | 7ccw | A | A | resveratrol | Human | 13235 | |
| DAPK1 | DAPK | CAMK | 8ie8 | A | | 5-[(~{e})-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]benzene-1,3-diol | Human | 14750 | |
| DAPK1 | DAPK | CAMK | 8ie6 | A | | 3-[(e)-2-(4-hydroxyphenyl)ethenyl]-5-methoxy-phenol | Human | 14751 | |
| DAPK1 | DAPK | CAMK | 3gu5 | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 5662 | |
| DAPK1 | DAPK | CAMK | 2yak | A | A | ruthenium octasporine 4 | Human | 7259 | |
| DAPK2 | DAPK | CAMK | 1wmk | G | | - | Human | 1142 | |
| DAPK1 | DAPK | CAMK | 1ig1 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5615 | |
| DAPK1 | DAPK | CAMK | 4txc | A | | 4-(3-{3-[(r)-{[2-(dimethylamino)ethyl]amino}(hydroxy)methyl]phenyl}imidazo[1,2-b]pyridazin-6-yl)-2-methoxyphenol | Human | 5668 | |
| DAPK1 | DAPK | CAMK | 1wvy | A | | staurosporine | Human | 5661 | |
| DAPK1 | DAPK | CAMK | 5auw | A | | 3,5,7,3',4'-pentahydroxyflavone | Human | 6144 | |
| DAPK1 | DAPK | CAMK | 2w4j | A | A | adenosine-5'-diphosphate | Human | 5678 | |
| DAPK1 | DAPK | CAMK | 1jkl | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5685 | |
| DAPK1 | DAPK | CAMK | 4pf4 | A | A | - | Human | 5643 | |
| DAPK1 | DAPK | CAMK | 5aut | A | | 8-anilino-1-naphthalene sulfonate | Human | 6137 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | A | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | 1576 | |
| DAPK1 | DAPK | CAMK | 3gu5 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5669 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ywp | A | | 1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)urea | Human | 1658 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | B | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1623 | |
| DAPK1 | DAPK | CAMK | 3zxt | C | | phosphomethylphosphonic acid adenylate ester | Human | 5646 | |
| DAPK1 | DAPK | CAMK | 4tl0 | A | | - | Human | 5641 | |
| DAPK1 | DAPK | CAMK | 3gu5 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5680 | |
| DAPK1 | DAPK | CAMK | 2y4p | B | | - | Human | 5626 | |
| DAPK1 | DAPK | CAMK | 3zxt | D | | phosphomethylphosphonic acid adenylate ester | Human | 5617 | |
| DAPK1 | DAPK | CAMK | 3eh9 | A | B | adenosine-5'-diphosphate | Human | 5622 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | A | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | 1563 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | A | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | 9503 | |
| DAPK1 | DAPK | CAMK | 2x0g | A | A | - | Human | 5672 | |
| DAPK1 | DAPK | CAMK | 5auv | A | | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 6139 | |
| DAPK1 | DAPK | CAMK | 6fhb | A | A | - | Human | 11290 | |
| DAPK1 | DAPK | CAMK | 4ypd | A | B | 4-methylpyridazine | Human | 5623 | |
| DAPK1 | DAPK | CAMK | 3zxt | A | | phosphomethylphosphonic acid adenylate ester | Human | 5634 | |
| DCLK1 | DCAMKL | CAMK | 6kyr | B | B | - | Human | 12804 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hxl | A | | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrile | Human | 1552 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgx | A | | 2-[(6-amino-7h-purin-8-yl)thio]acetamide | Human | 1595 | |
| DAPK1 | DAPK | CAMK | 5av3 | A | | 3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 6143 | |
| DAPK1 | DAPK | CAMK | 7ccu | A | B | resveratrol | Human | 13237 | |
| DAPK1 | DAPK | CAMK | 3gu4 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5670 | |
| DAPK1 | DAPK | CAMK | 5av0 | A | | 3-(3,4-dihydroxyphenyl)-7-hydroxy-4h-chromen-4-one | Human | 6142 | |
| DAPK1 | DAPK | CAMK | 5av1 | A | | - | Human | 6138 | |
| DAPK1 | DAPK | CAMK | 3eha | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 5647 | |
| DAPK1 | DAPK | CAMK | 8ie7 | A | | pterostilbene | Human | 14752 | |
| DAPK1 | DAPK | CAMK | 2y0a | A | | - | Human | 5651 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | C | A | staurosporine | Human | 9847 | |
| PIM1 | PIM | CAMK | 3vby | A | | furan-2-yl(1h-indol-3-yl)methanone | Human | 2466 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | B | - | Human | 1666 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | B | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | 1583 | |
| CASK | CASK | CAMK | 3c0g | A | B | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3827 | |
| PIM1 | PIM | CAMK | 3vbw | A | | 1,3-dioxo-2,3-dihydro-1h-indene-2-carbonitrile | Human | 2390 | |
| PIM1 | PIM | CAMK | 5v80 | A | | 1-methyl-4-{3-[6-(piperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[3,4-c]pyridin-5-yl}piperazin-2-one | Human | 9828 | |
| PIM1 | PIM | CAMK | 2xix | A | B | 3,5-diamino-1h-[1,2,4]triazole | Human | 2433 | |
| PIM1 | PIM | CAMK | 5n4r | A | A | 2-(azepan-1-yl)-1-(1~{h}-indol-3-yl)propan-1-one | Human | 9584 | |
| PIM1 | PIM | CAMK | 1xws | A | A | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2343 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op4 | A | | [4-[[4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-fluoranyl-5-methoxy-phenyl]-morpholin-4-yl-methanone | Human | 8613 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmv | A | | 1-[(2s)-4-(7h-purin-6-yl)morpholin-2-yl]methanamine | Human | 1562 | |
| DAPK1 | DAPK | CAMK | 1jkk | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5644 | |
| DAPK1 | DAPK | CAMK | 1p4f | A | A | 5,6-dihydro-benzo[h]cinnolin-3-ylamine | Human | 5625 | |
| DAPK1 | DAPK | CAMK | 2xzs | A | B | - | Human | 5642 | |
| DAPK1 | DAPK | CAMK | 3dgk | A | A | - | Human | 5656 | |
| DAPK1 | DAPK | CAMK | 3dfc | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 5645 | |
| DAPK1 | DAPK | CAMK | 2yak | A | B | ruthenium octasporine 4 | Human | 7260 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6bx6 | A | A | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 9878 | |
| CAMK2B (CaMK2b) | CAMK2 | CAMK | 3bhh | D | | - | Human | 1504 | |
| CAMK2B (CaMK2b) | CAMK2 | CAMK | 3bhh | B | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 1506 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | A | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | 1608 | |
| CAMK2B (CaMK2b) | CAMK2 | CAMK | 3bhh | C | | - | Human | 1505 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | B | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | 1535 | |
| CAMK2B (CaMK2b) | CAMK2 | CAMK | 3bhh | A | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 1507 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | B | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 1681 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | B | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | 1659 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8601 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsw | A | A | 8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1541 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmw | A | | 1-[(2s)-4-(5-bromo-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | 1594 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1zlt | A | | (4z)-4-(2-amino-5-oxo-3,5-dihydro-4h-imidazol-4-ylidene)-2,3-dichloro-4,5,6,7-tetrahydropyrrolo[2,3-c]azepin-8(1h)-one | Human | 1596 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq6 | A | | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 8610 | |
| PIM1 | PIM | CAMK | 5vub | B | B | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9076 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydk | A | | 2-(carbamoylamino)-5-phenyl-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | 1646 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | A | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | 8602 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brn | A | | (2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-ol | Human | 1631 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | A | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | 1695 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opv | A | | 4-(3-methylphenyl)-6-[(1-methylpyrazol-3-yl)amino]-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | 8608 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | B | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | 1615 | |
| PIM1 | PIM | CAMK | 3jxw | A | | 8-[(e)-2-cyclopropylethenyl]-2-[(dimethylamino)methyl][1]benzothieno[3,2-d]pyrimidin-4(3h)-one | Human | 2393 | |
| DCLK1 | DCAMKL | CAMK | 6kyq | A | B | - | Human | 12798 | |
| DCLK1 | DCAMKL | CAMK | 6kyq | A | A | - | Human | 12799 | |
| DCLK1 | DCAMKL | CAMK | 6kyr | A | B | - | Human | 12800 | |
| DCLK1 | DCAMKL | CAMK | 6kyq | B | B | - | Human | 12801 | |
| MARK2 | CAMKL | CAMK | 3iec | A | | - | Human | 3045 | |
| MARK2 | CAMKL | CAMK | 5kz7 | A | | 7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-one | Human | 7967 | |
| MARK2 | CAMKL | CAMK | 5kz8 | A | | 5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-one | Human | 7965 | |
| MARK2 | CAMKL | CAMK | 5eak | A | | n-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide | Human | 6410 | |
| DCLK1 | DCAMKL | CAMK | 7kx6 | A | | 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 13907 | |
| DCLK1 | DCAMKL | CAMK | 6kyq | B | A | - | Human | 12802 | |
| PIM1 | PIM | CAMK | 3we8 | A | B | cyclopentadienyl(carbon monoxide)(7-oxo-7,10-dihydro-1,8-phenanthrolin-10-yl-kappa~2~c~10~,n~1~)ruthenium | Human | 7232 | |
| PIM1 | PIM | CAMK | 2o65 | A | | 5,7-dihydroxy-2-(3,4,5-trihydroxyphenyl)-4h-chromen-4-one | Human | 2324 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | B | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 1687 | |
| PIM1 | PIM | CAMK | 2xj0 | A | B | (e)-3-(2-amino-pyridine-5yl)-acrylic acid | Human | 2395 | |
| PIM1 | PIM | CAMK | 6l16 | A | | 2-[4-[2-(7-chloranylpyrido[3,4-b][1,4]benzoxazin-5-yl)ethyl]piperidin-1-yl]ethanamine | Human | 12335 | |
| PIM1 | PIM | CAMK | 4n70 | A | B | n-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | Human | 2357 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 2wnt | B | A | - | Human | 6860 | |
| MKNK1 (MNK1) | MAPKAPK | CAMK | 2hw6 | A | | - | Human | 2084 | |
| MKNK1 (MNK1) | MAPKAPK | CAMK | 5wvd | B | | 1-methyl-n-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamide | Human | 9465 | |
| MKNK1 (MNK1) | MAPKAPK | CAMK | 5wvd | A | | 1-methyl-n-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamide | Human | 9464 | |
| PIM1 | PIM | CAMK | 4jx7 | A | | 2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6h)-one | Human | 2340 | |
| MYLK4 (SgK085) | MLCK | CAMK | 2x4f | B | A | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | 4866 | |
| DAPK1 | DAPK | CAMK | 6fha | A | A | - | Human | 11289 | |
| MYLK4 (SgK085) | MLCK | CAMK | 2x4f | A | B | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | 4867 | |
| PIM1 | PIM | CAMK | 5ndt | A | A | 3-(2-thiophen-2-ylethenyl)-1~{h}-quinoxalin-2-one | Human | 9907 | |
| PIM1 | PIM | CAMK | 2o3p | A | B | 3,5,7,3',4'-pentahydroxyflavone | Human | 2409 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | B | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 13779 | |
| PIM1 | PIM | CAMK | 3vbv | A | | 8-hydroxyquinoline-2-carboxamide | Human | 2399 | |
| PIM1 | PIM | CAMK | 5vuc | B | B | (2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-one | Human | 9075 | |
| DAPK1 | DAPK | CAMK | 2xzs | B | B | - | Human | 5671 | |
| PIM1 | PIM | CAMK | 4n70 | A | A | n-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | Human | 2388 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xk9 | A | | n-{4-[(1e)-n-(n-hydroxycarbamimidoyl)ethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamide | Human | 4771 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yiq | A | A | (e)-5-(1-(2-carbamimidoylhydrazono)ethyl)-n-(1h-indol-6-yl)-1h-indole-2-carboxamide | Human | 4791 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yir | A | | (e)-n-(5-(2-carbamimidoylhydrazono)-5,6,7,8-tetrahydronaphthalen-2-yl)-7-nitro-1h-indole-2-carboxamide | Human | 4768 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycf | A | B | (2e)-n-hydroxy-2-[1-(4-{[(4-{(1e)-1-[2-(n'-hydroxycarbamimidoyl)hydrazinylidene]ethyl}phenyl)carbamoyl]amino}phenyl)ethylidene]hydrazinecarboximidamide | Human | 4774 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6u | B | | - | Human | 4787 | |
| PIM1 | PIM | CAMK | 2oi4 | X | A | - | Human | 7236 | |
| PIM1 | PIM | CAMK | 3a99 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2322 | |
| PIM1 | PIM | CAMK | 5kge | A | | 5-(3,4-dichlorophenyl)-1~{h}-pyrazol-3-amine | Human | 8310 | |
| PIM1 | PIM | CAMK | 3qf9 | A | A | 6-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}naphthalene-1-carboxamide | Human | 2329 | |
| PIM1 | PIM | CAMK | 5n51 | A | B | 3,4-bis(bromanyl)thiophene-2-carboxylic acid | Human | 9591 | |
| PIM1 | PIM | CAMK | 3c4e | A | | n-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amine | Human | 2413 | |
| PIM1 | PIM | CAMK | 5dgz | A | | (2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amine | Human | 6209 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | B | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1560 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmq | A | | n-(4-oxo-5,6,7,8-tetrahydro-4h-[1,3]thiazolo[5,4-c]azepin-2-yl)acetamide | Human | 1647 | |
| PIM1 | PIM | CAMK | 5kgi | A | | 2-[3,4-bis(chloranyl)phenoxy]ethanamine | Human | 8306 | |
| MYLK4 (SgK085) | MLCK | CAMK | 2x4f | A | A | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | 4865 | |
| DAPK1 | DAPK | CAMK | 3gu4 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5681 | |
| PIM1 | PIM | CAMK | 5n52 | A | A | (~{e})-3-(2,3-dimethoxyphenyl)prop-2-enoic acid | Human | 9581 | |
| PIM1 | PIM | CAMK | 5n50 | A | B | 2-(4-chlorophenyl)sulfanylethanehydrazide | Human | 9598 | |
| PIM1 | PIM | CAMK | 7qfm | A | A | 4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | 14561 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4rer | A | | staurosporine | Human | 121 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4red | A | | - | Human | 122 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4rew | A | | staurosporine | Human | 124 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jhg | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 13816 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9h | A | | staurosporine | Human | 10714 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jhh | A | | - | Human | 13817 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7m74 | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 14017 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 7jij | B | | - | Human | 13819 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9j | A | | staurosporine | Human | 10717 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opb | A | B | (2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholine | Human | 8604 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | A | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13772 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | A | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | 13775 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjx | A | B | 4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13768 | |
| CASK | CASK | CAMK | 7oai | A | B | 4-(cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-n-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | Human | 13583 | |
| CASK | CASK | CAMK | 7oai | A | A | 4-(cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-n-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | Human | 13584 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk1 | A | | 4-amino-2-[(1,3-dimethyl-1h-pyrazol-4-yl)amino]-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13763 | |
| CASK | CASK | CAMK | 7oaj | A | B | 4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-n-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | Human | 13581 | |
| PIM1 | PIM | CAMK | 3cxw | A | B | (4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 2392 | |
| PIM1 | PIM | CAMK | 2bzj | A | B | ruthenium-pyridocarbazole-3 | Human | 7228 | |
| PIM1 | PIM | CAMK | 6l14 | A | | 2-chloranyl-10-[3-[(3~{s})-piperidin-3-yl]propyl]phenoxazine | Human | 12338 | |
| PIM1 | PIM | CAMK | 5v82 | A | | 1-{6-[(3r)-4,4-difluoropiperidin-3-yl]pyridin-2-yl}-6-(6-methylpyrazin-2-yl)-1h-pyrazolo[4,3-c]pyridine | Human | 7581 | |
| PIM1 | PIM | CAMK | 1yxv | A | A | 3,4-dihydroxy-1-methylquinolin-2(1h)-one | Human | 2367 | |
| TRIB1 (Trb1) | Trbl | CAMK | 5cek | A | | - | Human | 6241 | |
| PIM1 | PIM | CAMK | 5vua | B | A | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9074 | |
| PIM1 | PIM | CAMK | 2j2i | B | A | (9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dione | Human | 2318 | |
| PIM1 | PIM | CAMK | 5tel | A | B | 4-chloro-2-{5,6-dimethoxy-1-[2-(4-methylpiperazin-1-yl)ethyl]-1h-indol-3-yl}-1h-pyrrolo[2,3-b]pyridine | Human | 8562 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjo | A | | 4-amino-6-(2,3-difluorophenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13780 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sui | A | | (3r,4r)-4-{(3s,4s)-4-[6-chloro-2-({5-chloro-1-[(1r)-2,2-difluorocyclopropyl]-1h-pyrazol-4-yl}amino)quinazolin-7-yl]-3-fluoropiperidin-1-yl}oxolan-3-ol | Human | 14045 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6vzk | A | | 4'-hydroxycinnamic acid | Human | 12165 | |
| DCLK1 | DCAMKL | CAMK | 5jzj | B | A | amp phosphoramidate | Human | 6985 | |
| DCLK1 | DCAMKL | CAMK | 5jzj | B | B | amp phosphoramidate | Human | 6983 | |
| MARK2 | CAMKL | CAMK | 5kz8 | B | | 5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-one | Human | 7968 | |
| MARK2 | CAMKL | CAMK | 5kz7 | B | | 7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-one | Human | 7966 | |
| PIM1 | PIM | CAMK | 4gw8 | A | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 2428 | |
| MARK2 | CAMKL | CAMK | 3iec | C | | - | Human | 3046 | |
| MARK2 | CAMKL | CAMK | 5eak | B | | n-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide | Human | 6411 | |
| MARK2 | CAMKL | CAMK | 3iec | B | | - | Human | 3044 | |
| MARK2 | CAMKL | CAMK | 3iec | D | | - | Human | 3043 | |
| PIM1 | PIM | CAMK | 5iis | A | | 3-amino-n-(2'-amino-6'-methyl[4,4'-bipyridin]-3-yl)-6-(2-fluorophenyl)pyridine-2-carboxamide | Human | 6504 | |
| MARK1 | CAMKL | CAMK | 2hak | D | | - | Human | 257 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4q | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 15241 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4o | A | | 2-[bis(fluoranyl)methoxy]-4-[6-(2-cyanopropan-2-yl)pyrazolo[1,5-a]pyridin-3-yl]-~{n}-[(1~{r},2~{s})-2-fluoranylcyclopropyl]-6-methoxy-benzamide | Human | 15242 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4u | A | | 8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-one | Human | 15240 | |
| SIK3 (QSK) | CAMKL | CAMK | 8r4v | A | | 1-(2,4-dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]urea | Human | 15243 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 8uso | A | | - | Human | 15247 | |
| PHKG1 (PHKg1) | PHK | CAMK | 8z5t | C | A | adenosine-5'-triphosphate | Human | 15642 | |
| PHKG1 (PHKg1) | PHK | CAMK | 8z5p | C | | - | Human | 15643 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 10ia | A | | (10as,13as)-3-cyclopropyl-1-methyl-8-(trifluoromethyl)-3,4,10a,11,13a,14-hexahydro-10h,13h-9,5-(azeno)furo[3,4-k]pyrazolo[4,3-b][1,4,6,10]oxatriazacyclotridecine | Human | 15693 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 10hz | A | | (10as,13as)-3-cyclobutyl-1-methyl-8-(trifluoromethyl)-3,4,10a,11,13a,14-hexahydro-10h,13h-9,5-(azeno)furo[3,4-k]pyrazolo[4,3-b][1,4,6,10]oxatriazacyclotridecine | Human | 15694 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 10hy | A | | (11r)-8-chloro-3,11-dimethyl-2-(oxan-4-yl)-2,4,10,11,12,13-hexahydro-9,5-(azeno)pyrazolo[3,4-b][1,4,6,10]oxatriazacyclotridecine | Human | 15695 | |
| MAPKAPK2 | MAPKAPK | CAMK | 8xx1 | A | A | - | Human | 15257 | |
| MARK3 | CAMKL | CAMK | 8uoh | A | B | - | Human | 15733 | |
| MARK3 | CAMKL | CAMK | 9vir | A | | ~{n}-[5-[[4-[[(3~{r},3~{a}~{r},6~{a}~{s})-3-methoxy-2,3,3~{a},6~{a}-tetrahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[[(2~{r},8~{r})-2-fluoranyl-1,2,3,5,6,7-hexahydropyrrolizin-8-yl]methoxy]phenyl]-1-methyl-pyrazole-4-carboxamide | Human | 15734 | |
| MARK3 | CAMKL | CAMK | 8uoh | A | A | - | Human | 15735 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up4 | A | A | (5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | 14277 | |
| MAPKAPK2 | MAPKAPK | CAMK | 8xx1 | A | B | - | Human | 15256 | |
| PIM1 | PIM | CAMK | 4rc2 | A | | 1-amino-5,8-dihydroxy-4-({2-[(2-hydroxyethyl)amino]ethyl}amino)anthracene-9,10-dione | Human | 2346 | |
| PIM1 | PIM | CAMK | 1xr1 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2406 | |
| PIM1 | PIM | CAMK | 5n4n | A | B | 3,4-dimethyl-5-(1~{h}-1,2,4-triazol-3-yl)thiophene-2-carbonitrile | Human | 9595 | |
| PIM1 | PIM | CAMK | 7oov | A | | - | Human | 13824 | |
| PIM1 | PIM | CAMK | 4i41 | A | | 1,4-dihydroxy-5,8-bis({2-[(2-hydroxyethyl)amino]ethyl}amino)-9,10-anthracenedione | Human | 2326 | |
| PIM1 | PIM | CAMK | 4gw8 | A | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 2391 | |
| PIM1 | PIM | CAMK | 6bsk | A | | 4-{6-[6-(propan-2-ylamino)-1h-indazol-1-yl]pyrazin-2-yl}benzoic acid | Human | 9758 | |
| PIM1 | PIM | CAMK | 4rc3 | A | | 1,4-dihydroxy-5,8-bis{[2-(2-hydroxyethoxy)ethyl]amino}anthracene-9,10-dione | Human | 2412 | |
| MELK | CAMKL | CAMK | 9f31 | A | | n-[4-(1h-indazol-5-yl)phenyl]propanamide | Human | 15787 | |
| PIM1 | PIM | CAMK | 4lmu | A | A | 3,5,7,3',4'-pentahydroxyflavone | Human | 2376 | |
| PIM1 | PIM | CAMK | 5n4u | A | B | 5-(2-azanyl-1,3-thiazol-4-yl)-1,3-dihydrobenzimidazol-2-one | Human | 9590 | |
| PIM1 | PIM | CAMK | 6ayd | A | A | n-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamide | Human | 9442 | |
| DAPK1 | DAPK | CAMK | 9inw | A | | (~{e})-1-[2,4-bis(oxidanyl)phenyl]-3-(3-chloranyl-4-oxidanyl-phenyl)prop-2-en-1-one | Human | 15839 | |
| DAPK1 | DAPK | CAMK | 9inx | A | | (~{e})-1-[2,4-bis(oxidanyl)phenyl]-3-(3-bromanyl-4-oxidanyl-phenyl)prop-2-en-1-one | Human | 15840 | |
| DAPK1 | DAPK | CAMK | 9dub | A | B | 4-(pyridin-4-yl)pyridazine | Human | 15841 | |
| DAPK1 | DAPK | CAMK | 9dub | A | A | 4-(pyridin-4-yl)pyridazine | Human | 15842 | |
| DAPK1 | DAPK | CAMK | 9inv | A | | 2',4,4'-trihydroxychalcone | Human | 15843 | |
| PIM1 | PIM | CAMK | 5n4y | A | B | 2,5-dihydro-1~{h}-isothiochromeno[4,3-c]pyrazol-3-one | Human | 9597 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 9blh | A | B | 7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 16000 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 9blh | A | A | 7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 16001 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | B | staurosporine | Human | 13495 | |
| CASK | CASK | CAMK | 9m6g | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 16104 | |
| CASK | CASK | CAMK | 8y68 | A | A | - | Human | 16105 | |
| CASK | CASK | CAMK | 9m5y | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 16106 | |
| CASK | CASK | CAMK | 9m5y | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 16107 | |
| CASK | CASK | CAMK | 8y68 | A | B | - | Human | 16108 | |
| PIM1 | PIM | CAMK | 5o11 | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 8657 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | B | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1652 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hog | A | | (5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanol | Human | 1653 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | B | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | 1598 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8595 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyf | A | | 4-[3-amino-6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | 1622 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brg | A | | (5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-acetic | Human | 1589 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 2ac5 | A | B | - | Human | 766 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl0 | A | | methyl 6-o-(heptylcarbamoyl)-beta-l-altropyranoside | Human | 13111 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7uis | A | | - | Human | 14174 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujr | A | | - | Human | 14191 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl2 | A | | - | Human | 13064 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 7myj | A | | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 14273 | |
| TTN | MLCK | CAMK | 6ygn | A | | - | Human | 13488 | |
| TTN | MLCK | CAMK | 6ygn | B | | - | Human | 13487 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjd | A | B | 2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrile | Human | 13774 | |
| PIM1 | PIM | CAMK | 4rbl | A | | 1,4,5,8-tetrahydroxyanthracene-9,10-dione | Human | 2385 | |
| PIM1 | PIM | CAMK | 3bwf | A | B | - | Human | 7235 | |
| PIM1 | PIM | CAMK | 3r02 | A | A | 7-[(cis-4-aminocyclohexyl)amino]-5-bromo-1-benzofuran-2-carboxylic acid | Human | 2420 | |
| PIM2 | PIM | CAMK | 2iwi | B | | ruthenium-pyridocarbazole-1 | Human | 7216 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 8bfs | A | A | 3~{h}-pyrrolo[2,3-c]isoquinolin-5-amine | Human | 14506 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | K | | - | Human | 1293 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | A | | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | 1287 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | D | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1288 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | H | | - | Human | 1348 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | C | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1350 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | E | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1323 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2onl | D | | - | Human | 1345 | |
| MARK1 | CAMKL | CAMK | 2hak | G | | - | Human | 256 | |
| MARK1 | CAMKL | CAMK | 2hak | F | | - | Human | 254 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | C | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1328 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | G | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1339 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2pzy | B | | (4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamide | Human | 1307 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | G | | - | Human | 1369 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | C | | - | Human | 1368 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | E | | - | Human | 1286 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | B | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1320 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | B | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1332 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 2yza | A | | - | Human | 189 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | B | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1897 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | C | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1896 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | A | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1894 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym6 | A | B | 1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamine | Human | 1559 | |
| PIM1 | PIM | CAMK | 2c3i | B | A | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 2348 | |
| PIM1 | PIM | CAMK | 4n6z | A | | 3-amino-n-{4-[(3s)-3-aminopiperidin-1-yl]pyridin-3-yl}pyrazine-2-carboxamide | Human | 2442 | |
| PIM1 | PIM | CAMK | 2xj0 | A | A | (e)-3-(2-amino-pyridine-5yl)-acrylic acid | Human | 2435 | |
| PIM1 | PIM | CAMK | 5toe | A | | 2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrile | Human | 8563 | |
| PIM1 | PIM | CAMK | 2o64 | A | | 3,5,6,7-tetrahydroxy-2-(3,4-dihydroxyphenyl)-4h-chromen-4-one | Human | 2421 | |
| PIM1 | PIM | CAMK | 8r18 | A | B | (e)-4-(4-hydroxystyryl)benzoic acid | Human | 15208 | |
| PIM1 | PIM | CAMK | 4ll5 | A | B | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | 2382 | |
| PIM1 | PIM | CAMK | 2j2i | B | B | (9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dione | Human | 2434 | |
| PIM1 | PIM | CAMK | 4alv | A | B | 8-bromo-2-{2-chloro-4-[(piperidin-4-ylmethyl)amino]phenyl}[1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 2396 | |
| PIM1 | PIM | CAMK | 7qfm | A | B | 4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | 14560 | |
| PIM1 | PIM | CAMK | 3vbx | A | B | 6-bromo-4-hydroxy-2h-chromen-2-one | Human | 2448 | |
| PIM1 | PIM | CAMK | 31ru | A | | 6-chloranyl-3-[4-(1~{h}-indol-3-yl)-1~{h}-pyrazol-5-yl]quinazolin-4-one | Human | 15474 | |
| PIM1 | PIM | CAMK | 1xws | A | B | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2441 | |
| PIM1 | PIM | CAMK | 8r10 | A | B | (z)-4-(4-hydroxystyryl)benzoic acid | Human | 15209 | |
| PIM1 | PIM | CAMK | 8afr | A | B | 4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acid | Human | 14601 | |
| PIM1 | PIM | CAMK | 8r1p | A | | 4-(4-aminostyryl)benzoic acid | Human | 15210 | |
| PIM1 | PIM | CAMK | 8r1t | A | B | 4-(4-aminophenethyl)benzoic acid | Human | 15211 | |
| PIM1 | PIM | CAMK | 8r25 | A | | 4-(5-(4-aminophenyl)-1h-pyrazol-1-yl)benzoic acid | Human | 15475 | |
| PIM1 | PIM | CAMK | 5n5l | A | B | 5-bromanyl-1~{h}-indole-3-carboxylic acid | Human | 9704 | |
| PIM1 | PIM | CAMK | 7z6u | A | A | 4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | 14602 | |
| PIM1 | PIM | CAMK | 5dwr | A | | n-{4-[(1r,3s,5s)-3-amino-5-methylcyclohexyl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamide | Human | 6238 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6bx6 | A | B | 2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acid | Human | 9877 | |
| PIM1 | PIM | CAMK | 3r04 | A | B | 5-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}-1-benzofuran-2-carboxylic acid | Human | 2335 | |
| PIM1 | PIM | CAMK | 3dcv | A | | 4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-one | Human | 2372 | |
| PIM1 | PIM | CAMK | 3umx | A | B | (2z)-7-(azepan-1-ylmethyl)-6-hydroxy-2-(1h-indol-3-ylmethylidene)-1-benzofuran-3(2h)-one | Human | 2375 | |
| PIM1 | PIM | CAMK | 4xh6 | A | | 5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4h-chromen-4-one | Human | 5975 | |
| PIM1 | PIM | CAMK | 8r10 | A | A | (z)-4-(4-hydroxystyryl)benzoic acid | Human | 15214 | |
| PIM1 | PIM | CAMK | 1ywv | A | B | - | Human | 2397 | |
| PIM1 | PIM | CAMK | 8r1n | A | | 4-(4-hydroxyphenethyl)benzoic acid | Human | 15215 | |
| PIM1 | PIM | CAMK | 5n50 | A | A | 2-(4-chlorophenyl)sulfanylethanehydrazide | Human | 9585 | |
| PIM1 | PIM | CAMK | 2xiy | A | B | 2-hydroxymethyl-benzoimidazole | Human | 2363 | |
| PIM1 | PIM | CAMK | 4bzn | A | | n-(2,2-dimethylpropyl)-2-[1-oxo-7-(thiophen-3-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamide | Human | 2402 | |
| PIM1 | PIM | CAMK | 5n4x | A | B | 4,5-bis(bromanyl)thiophene-2-carbohydrazide | Human | 9593 | |
| PIM1 | PIM | CAMK | 6pdo | A | A | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamide | Human | 11461 | |
| PIM1 | PIM | CAMK | 2xj2 | A | B | (2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acid | Human | 2418 | |
| PIM1 | PIM | CAMK | 5n4v | A | A | 2-cyclopropyl-4,5-dimethyl-thieno[2,3-d]pyrimidine-6-carboxylic acid | Human | 9592 | |
| PIM1 | PIM | CAMK | 4eny | A | B | (2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-one | Human | 2424 | |
| PIM1 | PIM | CAMK | 2o3p | A | A | 3,5,7,3',4'-pentahydroxyflavone | Human | 2320 | |
| PIM1 | PIM | CAMK | 7zun | A | | (4~{s})-4-(2-azanylethyl)-6-phenyl-7-[3-(trifluoromethyloxy)phenyl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1-ol | Human | 14383 | |
| PIM1 | PIM | CAMK | 5vub | B | A | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9073 | |
| PIM1 | PIM | CAMK | 8r0y | A | | 3-[(3-hydroxyphenyl)amino]quinoxaline-2-carboxylic acid | Human | 15477 | |
| PIM1 | PIM | CAMK | 5dhj | A | B | 3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridine | Human | 6211 | |
| PIM1 | PIM | CAMK | 5kcx | A | B | 4-chloranyl-1-methyl-2-[4-(4-methylpiperazin-1-yl)phenyl]pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 8248 | |
| PIM1 | PIM | CAMK | 4n6y | A | | 2-(acetylamino)-n-[2-(piperidin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 2383 | |
| PIM1 | PIM | CAMK | 4as0 | A | B | phtalimide-ruthenium complex | Human | 7229 | |
| PIM1 | PIM | CAMK | 7oow | A | | - | Human | 13826 | |
| PIM1 | PIM | CAMK | 5vub | B | C | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9072 | |
| PIM1 | PIM | CAMK | 6pdp | A | A | 5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamide | Human | 11454 | |
| PIM1 | PIM | CAMK | 6pdo | A | B | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamide | Human | 11460 | |
| PIM1 | PIM | CAMK | 5n4o | A | B | (~{e})-3-(4-methylphenyl)prop-2-enoic acid | Human | 9582 | |
| PIM1 | PIM | CAMK | 4alw | A | B | 8-bromanyl-2-[(4-methylpiperazin-1-yl)methyl]-3h-[1]benzofuro[3,2-d]pyrimidin-4-one | Human | 2350 | |
| PIM1 | PIM | CAMK | 5c1q | B | | 3-methoxy[1]benzothieno[2,3-c]quinolin-6(5h)-one | Human | 6288 | |
| PIM1 | PIM | CAMK | 4mbl | A | | (1r,2r)-n-[3-(naphthalen-2-yl)pyrazolo[1,5-a]pyrimidin-5-yl]cyclohexane-1,2-diamine | Human | 2381 | |
| PIM1 | PIM | CAMK | 3r01 | A | | 5-bromo-7-methoxy-1-benzofuran-2-carboxylic acid | Human | 2407 | |
| PIM1 | PIM | CAMK | 3cy2 | A | A | (4r)-7-chloro-9-methyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 2333 | |
| PIM1 | PIM | CAMK | 5n4x | A | A | 4,5-bis(bromanyl)thiophene-2-carbohydrazide | Human | 9600 | |
| PIM1 | PIM | CAMK | 5kzi | A | | ~{n}-[4-[(3~{s})-3-azanylpiperidin-1-yl]pyridin-3-yl]-2-[2,6-bis(fluoranyl)phenyl]imidazo[1,5-b]pyridazin-7-amine | Human | 7195 | |
| PIM1 | PIM | CAMK | 2o63 | A | | 3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)-4h-chromen-4-one | Human | 2453 | |
| PIM1 | PIM | CAMK | 4dtk | A | B | (5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dione | Human | 2451 | |
| PIM1 | PIM | CAMK | 3bwf | A | A | - | Human | 7231 | |
| PIM1 | PIM | CAMK | 6l12 | A | | 4-[(2-chloranylphenoxazin-10-yl)methyl]cyclohexan-1-amine | Human | 12340 | |
| PIM1 | PIM | CAMK | 5n4n | A | A | 3,4-dimethyl-5-(1~{h}-1,2,4-triazol-3-yl)thiophene-2-carbonitrile | Human | 9579 | |
| PIM1 | PIM | CAMK | 6l17 | A | | 7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazin-8-amine | Human | 12740 | |
| PIM1 | PIM | CAMK | 8afr | A | A | 4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acid | Human | 14603 | |
| PIM1 | PIM | CAMK | 5vuc | B | A | (2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-one | Human | 9071 | |
| PIM1 | PIM | CAMK | 5tel | A | A | 4-chloro-2-{5,6-dimethoxy-1-[2-(4-methylpiperazin-1-yl)ethyl]-1h-indol-3-yl}-1h-pyrrolo[2,3-b]pyridine | Human | 8564 | |
| PIM1 | PIM | CAMK | 6kzi | A | | 4-(2-chloro-10h-phenoxazin-10-yl)-n,n-diethylbutan-1-amine | Human | 12019 | |
| CAMK2G (CaMK2g) | CAMK2 | CAMK | 2v7o | A | B | - | Human | 7238 | |
| CAMK2G (CaMK2g) | CAMK2 | CAMK | 2v7o | A | A | - | Human | 7239 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6ck6 | A | | 6'-[(6-aminopyrimidin-4-yl)amino]-8'-methyl-2'h-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dione | Human | 9880 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6jlr | A | | 4-[5-(1-methylpyrazol-4-yl)pyridin-3-yl]benzamide | Human | 11968 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | B | A | - | Human | 8011 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5iso | A | | staurosporine | Human | 7981 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | C | B | staurosporine | Human | 9850 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5iso | C | | staurosporine | Human | 7980 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | C | B | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6423 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4d9u | A | | tert-butyl (2s)-3-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl]-2-cyanopropanoate | Human | 1499 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg8 | A | B | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | 1498 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg8 | A | A | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | 1497 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg7 | A | A | (2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamide | Human | 1496 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg7 | A | B | (2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamide | Human | 1494 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4jg6 | A | | (2s)-2-cyano-3-(1h-indazol-5-yl)propanamide | Human | 1495 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 4d9t | A | | methyl (2s)-3-{4-amino-7-[(1e)-3-hydroxyprop-1-en-1-yl]-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl}-2-cyanopropanoate | Human | 1493 | |
| PIM1 | PIM | CAMK | 2xj1 | A | B | (2e)-3-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}phenyl)prop-2-enoic acid | Human | 2422 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | F | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1362 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 5vlo | A | | n-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Human | 8348 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2pzy | A | | (4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamide | Human | 1314 | |
| PIM1 | PIM | CAMK | 2bik | B | B | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2463 | |
| PIM1 | PIM | CAMK | 4wrs | A | | 3-{6-[(4r)-6-azaspiro[2.5]oct-4-yloxy]pyrazin-2-yl}-5-(2,6-difluorophenyl)-1h-indazole | Human | 2439 | |
| PIM1 | PIM | CAMK | 2xiz | A | B | (e)-pyridin-4-yl-acrylic acid | Human | 2373 | |
| PIM1 | PIM | CAMK | 5n4y | A | A | 2,5-dihydro-1~{h}-isothiochromeno[4,3-c]pyrazol-3-one | Human | 9589 | |
| PIM1 | PIM | CAMK | 3c4e | C | | n-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amine | Human | 2440 | |
| PIM1 | PIM | CAMK | 4rpv | A | | (3s)-1-{6-[5-(2,6-difluorophenyl)-2h-indazol-3-yl]pyrazin-2-yl}piperidin-3-amine | Human | 2364 | |
| PIM1 | PIM | CAMK | 5vua | B | B | (2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-one | Human | 9077 | |
| PIM1 | PIM | CAMK | 3vbq | A | B | 5-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}benzyl)-2h-1lambda~4~,3-thiazole-2,4(3h)-dione | Human | 2454 | |
| PIM1 | PIM | CAMK | 2bil | B | | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2449 | |
| PIM1 | PIM | CAMK | 3ma3 | A | B | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 2347 | |
| PIM1 | PIM | CAMK | 1yxu | D | | adenosine monophosphate | Human | 2332 | |
| PIM1 | PIM | CAMK | 5eol | A | | macrocyclic quinoxaline-pyrrolodihydropiperidinone | Human | 6601 | |
| PIM1 | PIM | CAMK | 5tex | A | | (4-{4-chloro-1-methyl-2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)methanol | Human | 8566 | |
| PIM1 | PIM | CAMK | 4bzo | A | | n-[(1s)-2-amino-1-phenylethyl]-2-[(4s)-7-(2-fluoro-4-pyridinyl)-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamide | Human | 2339 | |
| PIM1 | PIM | CAMK | 6qxk | B | B | 2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-one | Human | 11036 | |
| PIM1 | PIM | CAMK | 2bzi | B | B | - | Human | 7233 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | B | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1895 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | A | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1893 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | C | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1900 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | D | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1899 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 3soa | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 2473 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6x5g | A | A | - | Human | 13061 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6w4o | O | | - | Human | 12485 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujt | A | | adenosine-5'-triphosphate | Human | 14192 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 2vz6 | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 2472 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg7 | A | | adenosine-5'-triphosphate | Human | 4848 | |
| SNRK | CAMKL | CAMK | 5yks | A | | - | Human | 8660 | |
| PIM1 | PIM | CAMK | 1yxt | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2319 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up7 | A | A | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | 14318 | |
| PIM1 | PIM | CAMK | 2xj1 | A | A | (2e)-3-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}phenyl)prop-2-enoic acid | Human | 2469 | |
| PIM1 | PIM | CAMK | 3cy3 | A | | (2s)-1,3-benzothiazol-2-yl{2-[(2-pyridin-3-ylethyl)amino]pyrimidin-4-yl}ethanenitrile | Human | 2443 | |
| PIM1 | PIM | CAMK | 6pdn | A | B | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acid | Human | 11458 | |
| PIM1 | PIM | CAMK | 4alu | A | A | 8-bromo-2-(2-chlorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 2452 | |
| PIM1 | PIM | CAMK | 3vbt | A | | 4-chloro-2-(1h-pyrazol-3-yl)phenol | Human | 2349 | |
| PIM1 | PIM | CAMK | 3qf9 | A | B | 6-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}naphthalene-1-carboxamide | Human | 2331 | |
| PIM1 | PIM | CAMK | 3bgp | A | | 4-[3-(4-chlorophenyl)-2,1-benzisoxazol-5-yl]pyrimidin-2-amine | Human | 2359 | |
| PIM1 | PIM | CAMK | 4k18 | A | | 5-(4-cyanobenzyl)-n-(4-fluorophenyl)-7-hydroxypyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2377 | |
| PIM1 | PIM | CAMK | 6vru | A | A | 3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 13127 | |
| PIM1 | PIM | CAMK | 6qxk | B | A | 2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-one | Human | 11035 | |
| PIM1 | PIM | CAMK | 4jx3 | A | | - | Human | 2380 | |
| PIM1 | PIM | CAMK | 5ndt | A | B | 3-(2-thiophen-2-ylethenyl)-1~{h}-quinoxalin-2-one | Human | 9906 | |
| PIM1 | PIM | CAMK | 5n4z | A | B | (~{e})-4-(4-hydroxyphenyl)but-3-en-2-one | Human | 9599 | |
| PIM1 | PIM | CAMK | 4xhk | B | A | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | 2446 | |
| PIM1 | PIM | CAMK | 5o12 | A | | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 8654 | |
| PIM1 | PIM | CAMK | 3cxw | A | A | (4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 2464 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 2vz6 | B | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 2474 | |
| PIM1 | PIM | CAMK | 6no8 | A | | 5-amino-n-{5-[(4s)-4-aminoazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide | Human | 11832 | |
| PIM1 | PIM | CAMK | 1yxx | A | B | (3e)-3-[(4-hydroxyphenyl)imino]-1h-indol-2(3h)-one | Human | 2437 | |
| PIM1 | PIM | CAMK | 2oi4 | X | B | - | Human | 7226 | |
| PIM1 | PIM | CAMK | 7oox | A | B | - | Human | 13823 | |
| PIM1 | PIM | CAMK | 1yi3 | A | | 2-morpholin-4-yl-7-phenyl-4h-chromen-4-one | Human | 2398 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujp | A | | adenosine-5'-diphosphate | Human | 14193 | |
| PIM1 | PIM | CAMK | 5n5m | A | A | ~{n}-(isoquinolin-5-ylmethyl)-~{n}-methyl-2-[(3~{r})-pyrrolidin-3-yl]benzamide | Human | 9702 | |
| PIM1 | PIM | CAMK | 6pdi | A | | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11459 | |
| PIM1 | PIM | CAMK | 1yxu | A | | adenosine monophosphate | Human | 2438 | |
| PIM1 | PIM | CAMK | 1yxt | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2425 | |
| PIM1 | PIM | CAMK | 4wt6 | A | | 6-[5-(5-amino-1,3,4-thiadiazol-2-yl)-1h-indol-3-yl]-n-cyclopentylpyridin-2-amine | Human | 2386 | |
| PIM1 | PIM | CAMK | 1ywv | A | A | - | Human | 2430 | |
| PIM1 | PIM | CAMK | 5n4z | A | A | (~{e})-4-(4-hydroxyphenyl)but-3-en-2-one | Human | 9587 | |
| PIM1 | PIM | CAMK | 6pcw | A | | 4-[5-(cyclopropylcarbamoyl)thiophen-2-yl]-1-benzothiophene-2-carboxamide | Human | 11455 | |
| PIM1 | PIM | CAMK | 1yxu | C | | adenosine monophosphate | Human | 2408 | |
| PIM1 | PIM | CAMK | 1yxx | A | A | (3e)-3-[(4-hydroxyphenyl)imino]-1h-indol-2(3h)-one | Human | 2351 | |
| PIM1 | PIM | CAMK | 4as0 | A | A | phtalimide-ruthenium complex | Human | 7227 | |
| PIM1 | PIM | CAMK | 6mt0 | A | | 3-(1-methylcyclopropyl)-2-[(1-methylcyclopropyl)amino]-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-one | Human | 10850 | |
| PIM1 | PIM | CAMK | 3jya | A | A | 6,9-dichloro[1]benzothieno[3,2-d]pyrimidin-4(3h)-one | Human | 2371 | |
| PIM1 | PIM | CAMK | 4eny | A | A | (2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-one | Human | 2342 | |
| PIM1 | PIM | CAMK | 3c4e | B | | n-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amine | Human | 2423 | |
| PIM1 | PIM | CAMK | 3bgz | A | | 2,3-diphenyl-1h-indole-7-carboxylic acid | Human | 2462 | |
| PIM1 | PIM | CAMK | 4a7c | A | | n-(piperidin-4-ylmethyl)-3-[3-(trifluoromethyloxy)phenyl]-[1,2,3]triazolo[4,5-b]pyridin-5-amine | Human | 2321 | |
| PIM1 | PIM | CAMK | 5n4r | A | B | 2-(azepan-1-yl)-1-(1~{h}-indol-3-yl)propan-1-one | Human | 9583 | |
| PIM1 | PIM | CAMK | 4mta | A | | 2-methyl-5-phenylfuran-3-carboxylic acid | Human | 2370 | |
| PIM1 | PIM | CAMK | 5n4v | A | B | 2-cyclopropyl-4,5-dimethyl-thieno[2,3-d]pyrimidine-6-carboxylic acid | Human | 9594 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 9hrc | A | | 1-[5-chloranyl-4-[(3~{r})-pyrrolidin-3-yl]oxy-pyrimidin-2-yl]benzimidazole | Human | 15550 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cjy | A | | 5-[(7h-purin-6-yl)amino]-1h-isoindol-1-one | Human | 9881 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cj5 | A | | 3-(pyridin-3-yl)imidazo[1,2-a]pyridine-8-carboxamide | Human | 9886 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6ck3 | A | | (3r)-3-methyl-5-[(pyrimidin-4-yl)amino]-2,3-dihydro-1h-isoindol-1-one | Human | 9883 | |
| PIM1 | PIM | CAMK | 6vru | A | B | 3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 13128 | |
| PIM1 | PIM | CAMK | 2bik | B | A | 3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dione | Human | 2341 | |
| PIM1 | PIM | CAMK | 3r02 | A | B | 7-[(cis-4-aminocyclohexyl)amino]-5-bromo-1-benzofuran-2-carboxylic acid | Human | 2338 | |
| PIM1 | PIM | CAMK | 3f2a | A | | (2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acid | Human | 2460 | |
| PIM1 | PIM | CAMK | 7xsv | A | B | 8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaene | Human | 14288 | |
| DCLK1 | DCAMKL | CAMK | 5jzn | A | | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 6986 | |
| PIM1 | PIM | CAMK | 6ayd | A | B | n-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamide | Human | 9443 | |
| DCLK1 | DCAMKL | CAMK | 5jzj | A | B | amp phosphoramidate | Human | 6987 | |
| MARK1 | CAMKL | CAMK | 6c9d | B | B | - | Human | 10050 | |
| MARK1 | CAMKL | CAMK | 6c9d | B | A | - | Human | 10049 | |
| MARK1 | CAMKL | CAMK | 2hak | H | | - | Human | 261 | |
| MARK1 | CAMKL | CAMK | 6c9d | A | A | - | Human | 10052 | |
| PIM1 | PIM | CAMK | 5n5l | A | A | 5-bromanyl-1~{h}-indole-3-carboxylic acid | Human | 9703 | |
| DCLK1 | DCAMKL | CAMK | 5jzn | B | | 5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamine | Human | 6982 | |
| DCLK1 | DCAMKL | CAMK | 7f3g | A | | (3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrile | Human | 13853 | |
| PIM1 | PIM | CAMK | 5kgk | A | | 3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amine | Human | 8307 | |
| DCLK1 | DCAMKL | CAMK | 6kyr | A | A | - | Human | 12803 | |
| DCLK1 | DCAMKL | CAMK | 6kyr | B | A | - | Human | 12805 | |
| PIM1 | PIM | CAMK | 6vrv | A | | 4-chloro-1-{(1s)-1-[(3s)-3-fluoropyrrolidin-3-yl]ethyl}-3-methyl-1h-pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 13129 | |
| PIM1 | PIM | CAMK | 2bzj | A | A | ruthenium-pyridocarbazole-3 | Human | 7224 | |
| PIM1 | PIM | CAMK | 3r04 | A | A | 5-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}-1-benzofuran-2-carboxylic acid | Human | 2353 | |
| PIM1 | PIM | CAMK | 5kcx | A | A | 4-chloranyl-1-methyl-2-[4-(4-methylpiperazin-1-yl)phenyl]pyrrolo[2,3-b]pyridine-6-carboxamide | Human | 8247 | |
| PIM1 | PIM | CAMK | 6ykd | A | A | ~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamide | Human | 12402 | |
| PIM1 | PIM | CAMK | 4alv | A | A | 8-bromo-2-{2-chloro-4-[(piperidin-4-ylmethyl)amino]phenyl}[1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 2323 | |
| PIM1 | PIM | CAMK | 7oox | A | A | - | Human | 13825 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cfe | C | | staurosporine | Human | 192 | |
| PIM1 | PIM | CAMK | 2xix | A | A | 3,5-diamino-1h-[1,2,4]triazole | Human | 2468 | |
| PIM1 | PIM | CAMK | 3ma3 | A | A | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 2368 | |
| PIM1 | PIM | CAMK | 3cy2 | A | B | (4r)-7-chloro-9-methyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 2459 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cff | A | | staurosporine | Human | 191 | |
| DAPK2 | DAPK | CAMK | 2a27 | D | | - | Human | 1118 | |
| PIM1 | PIM | CAMK | 4mbi | A | | n,n-dimethyl-n'-[3-(1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]ethane-1,2-diamine | Human | 2447 | |
| PIM1 | PIM | CAMK | 3uix | A | A | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | 2456 | |
| PIM1 | PIM | CAMK | 2bzh | B | B | ruthenium-pyridocarbazole-1 | Human | 7234 | |
| DAPK2 | DAPK | CAMK | 2cke | B | | n-(2-aminoethyl)isoquinoline-5-sulfonamide | Human | 1132 | |
| DAPK2 | DAPK | CAMK | 1wmk | H | | - | Human | 1151 | |
| DAPK2 | DAPK | CAMK | 1zws | E | | - | Human | 1130 | |
| DAPK2 | DAPK | CAMK | 2a2a | D | B | - | Human | 1149 | |
| DAPK2 | DAPK | CAMK | 1zws | B | | - | Human | 1128 | |
| DAPK2 | DAPK | CAMK | 2a2a | B | B | - | Human | 1119 | |
| DAPK2 | DAPK | CAMK | 2a27 | H | | - | Human | 1137 | |
| DAPK2 | DAPK | CAMK | 1z9x | B | | - | Human | 1136 | |
| DAPK2 | DAPK | CAMK | 2cke | C | | n-(2-aminoethyl)isoquinoline-5-sulfonamide | Human | 1135 | |
| DAPK2 | DAPK | CAMK | 2a27 | G | | - | Human | 1146 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3she | A | B | n-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamide | Human | 4599 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3fhr | A | A | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4590 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3r1n | A | B | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | 4588 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 8bfm | A | | pyrazolo[5,1-a]phthalazin-6-amine | Human | 14516 | |
| PIM1 | PIM | CAMK | 1yxu | B | | adenosine monophosphate | Human | 2410 | |
| PIM1 | PIM | CAMK | 6pdp | A | B | 5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamide | Human | 11457 | |
| PIM1 | PIM | CAMK | 5dhj | A | A | 3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridine | Human | 6212 | |
| PIM1 | PIM | CAMK | 7qb2 | A | | 4-[(e)-(6-azanyl-1-methyl-2-oxidanylidene-indol-3-ylidene)methyl]benzoic acid | Human | 14518 | |
| PIM1 | PIM | CAMK | 3r00 | A | | 5-bromo-1-benzofuran-2-carboxylic acid | Human | 2467 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6qp5 | A | A | - | Human | 12028 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl1 | A | | adenosine-5'-triphosphate | Human | 13059 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6w4p | H | | - | Human | 12484 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7kl0 | B | | methyl 6-o-(heptylcarbamoyl)-beta-l-altropyranoside | Human | 13114 | |
| PIM1 | PIM | CAMK | 5o11 | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 8656 | |
| DCLK1 | DCAMKL | CAMK | 7kxw | A | | 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 13910 | |
| RPS6KA2-b (RSK1-b) | RSKb | CAMK | 8wf4 | A | | - | Human | 15082 | |
| DAPK2 | DAPK | CAMK | 1wmk | F | | - | Human | 1126 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6x5q | A | | - | Human | 13056 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujs | A | | adenosine-5'-diphosphate | Human | 14190 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 6x5g | A | B | - | Human | 13068 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 2vz6 | B | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 2470 | |
| TRIB1 (Trb1) | Trbl | CAMK | 5cem | A | A | - | Human | 6242 | |
| TRIB1 (Trb1) | Trbl | CAMK | 6dc0 | A | B | - | Human | 10623 | |
| TRIB1 (Trb1) | Trbl | CAMK | 6dc0 | A | A | - | Human | 10622 | |
| TRIB1 (Trb1) | Trbl | CAMK | 6dc0 | B | A | - | Human | 10620 | |
| TRIB1 (Trb1) | Trbl | CAMK | 5cem | A | B | - | Human | 6243 | |
| TRIB1 (Trb1) | Trbl | CAMK | 6dc0 | B | B | - | Human | 10621 | |
| PHKG1 (PHKg1) | PHK | CAMK | 8z5q | C | | - | Human | 15641 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t6f | B | A | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamide | Human | 11941 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t29 | A | B | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamide | Human | 13203 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t6f | A | B | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamide | Human | 11940 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t6f | B | B | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamide | Human | 11942 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | A | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | 1664 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | B | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1543 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | B | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1602 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftq | A | B | 5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrile | Human | 1550 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk3 | A | | 4-amino-7-methyl-2-({5-methyl-1-[(3s)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13764 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | B | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1590 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgv | A | | (2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-ol | Human | 1545 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | B | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | 6652 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4jik | A | | 2-(4-chlorophenyl)-8-[(3s)-piperidin-3-ylamino]imidazo[1,2-c]pyrimidine-5-carboxamide | Human | 1698 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | A | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | 1564 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | A | staurosporine | Human | 13492 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | B | - | Human | 13493 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | A | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1651 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft9 | A | B | 1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylurea | Human | 1648 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4gh2 | A | A | 3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-one | Human | 1600 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8594 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3l | A | | 3-(1h-benzimidazol-2-yl)-1h-indazole | Human | 1612 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siv | A | | n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)cyclopropanecarboxamide | Human | 14886 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | B | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | 1607 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op2 | A | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8611 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | A | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | 1547 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | A | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | 9500 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bkn | A | | adenine | Human | 13769 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tki | A | | n-(2-aminoethyl)-5-(2-{[4-(morpholin-4-yl)pyridin-2-yl]amino}-1,3-thiazol-5-yl)pyridine-3-carboxamide | Human | 1599 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgu | A | | 2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acid | Human | 1697 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq5 | A | | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 8597 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | B | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8596 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjm | A | | 4-amino-6-{[(2-fluorophenyl)methyl]amino}-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13770 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | B | A | - | Human | 13494 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | B | n,n-dimethyl-7h-purin-6-amine | Human | 13771 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e80 | A | | 2-[(1r,4r)-2-{(6p)-6-[(6m)-6-(1h-pyrazol-5-yl)-1h-indazol-1-yl]pyrimidin-4-yl}-2-azabicyclo[2.1.1]hexan-4-yl]propan-2-ol | Human | 14621 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3j | A | | debromohymenialdisine | Human | 1551 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyi | A | A | 2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 1538 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yex | A | B | 5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1567 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvk | A | | n-[3-(6-cyano-9h-pyrrolo[2,3-b:5,4-c']dipyridin-3-yl)phenyl]acetamide | Human | 1549 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | H | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1326 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | A | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | 1603 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | A | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1689 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsy | A | B | 2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamide | Human | 1537 | |
| TTN | MLCK | CAMK | 1tki | B | | - | Human | 126 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3tkh | A | | 1-(morpholin-4-yl)-2-[4-(2-{[5-(pyridin-3-yl)-1,3-thiazol-2-yl]amino}pyridin-4-yl)piperazin-1-yl]ethanone | Human | 1665 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvl | A | | 3-(2-hydroxyphenyl)-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1634 | |
| PIM1 | PIM | CAMK | 7vsy | A | | - | Human | 15098 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | B | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1640 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | B | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | 14044 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | A | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | 1540 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | A | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1673 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftj | A | B | trans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanol | Human | 1613 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | 1566 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wms | A | | [4-amino-2-(tert-butylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 1657 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | B | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | 1575 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | A | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | 1593 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9u | A | | 18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-one | Human | 1584 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2yer | A | A | 5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-one | Human | 1611 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | B | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | 1693 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | E | B | - | Human | 12503 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | B | | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | 1329 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2y | A | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1361 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1ny3 | A | | adenosine-5'-diphosphate | Human | 1318 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1kwp | A | | - | Human | 1280 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3ka0 | A | | 6-{5-[(2-aminopyrimidin-4-yl)amino]-2-hydroxyphenyl}-n-methylidene-1-benzothiophene-2-carboxamide | Human | 1290 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2p3g | X | | 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1349 | |
| DAPK1 | DAPK | CAMK | 1wvx | A | | 6-(3-aminopropyl)-4,9-dimethylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dione | Human | 5616 | |
| MARK2 | CAMKL | CAMK | 8txy | A | | n-[(5p,8r)-5-(2-cyano-5-{[(3r)-1-methylpyrrolidin-3-yl]methoxy}pyridin-4-yl)pyrazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamide | Human | 15136 | |
| SIK3 (QSK) | CAMKL | CAMK | 8oku | A | | ~{n}-ethyl-4-[5-[1-(2-hydroxyethyl)pyrazol-4-yl]benzimidazol-1-yl]-2,6-dimethoxy-benzamide | Human | 15169 | |
| MARK1 | CAMKL | CAMK | 2hak | C | | - | Human | 260 | |
| DAPK2 | DAPK | CAMK | 1zws | H | | - | Human | 1133 | |
| STK17B (DRAK2) | DAPK | CAMK | 7akg | A | B | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 13004 | |
| STK17B (DRAK2) | DAPK | CAMK | 6y6h | A | B | 2-[6-(1-benzothiophen-2-yl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12044 | |
| DAPK2 | DAPK | CAMK | 1zws | F | | - | Human | 1114 | |
| DAPK2 | DAPK | CAMK | 2cke | D | | n-(2-aminoethyl)isoquinoline-5-sulfonamide | Human | 1141 | |
| DAPK3 | DAPK | CAMK | 1yrp | A | | - | Human | 384 | |
| DAPK3 | DAPK | CAMK | 5a6o | B | B | - | Human | 6166 | |
| DAPK3 | DAPK | CAMK | 5a6n | A | A | 5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ide | Human | 6164 | |
| DAPK3 | DAPK | CAMK | 5vja | C | B | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10352 | |
| DAPK3 | DAPK | CAMK | 2j90 | A | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 387 | |
| DAPK3 | DAPK | CAMK | 5a6n | B | A | - | Human | 6162 | |
| DAPK3 | DAPK | CAMK | 5vja | B | A | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10346 | |
| DAPK3 | DAPK | CAMK | 5vja | A | A | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10351 | |
| DAPK3 | DAPK | CAMK | 5vja | D | B | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10347 | |
| DAPK3 | DAPK | CAMK | 3bqr | A | A | 4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acid | Human | 380 | |
| DAPK3 | DAPK | CAMK | 2j90 | B | A | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 378 | |
| MELK | CAMKL | CAMK | 5m5a | A | A | k-252a | Human | 8735 | |
| MELK | CAMKL | CAMK | 5mai | A | A | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 8728 | |
| MELK | CAMKL | CAMK | 5twy | B | | 2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 8669 | |
| MELK | CAMKL | CAMK | 4d2p | D | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2486 | |
| MELK | CAMKL | CAMK | 6vxr | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 12644 | |
| MELK | CAMKL | CAMK | 5k00 | A | A | 4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamide | Human | 7497 | |
| MELK | CAMKL | CAMK | 4d2w | A | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2515 | |
| MELK | CAMKL | CAMK | 4ump | C | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2479 | |
| PIM1 | PIM | CAMK | 5mzl | A | B | ~{n}-quinolin-5-ylpyridine-3-carboxamide | Human | 9563 | |
| MELK | CAMKL | CAMK | 4d2v | D | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2502 | |
| MYLK4 (SgK085) | MLCK | CAMK | 2x4f | B | B | 4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amine | Human | 4868 | |
| MELK | CAMKL | CAMK | 6vxr | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 12645 | |
| MELK | CAMKL | CAMK | 4d2p | A | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2513 | |
| MELK | CAMKL | CAMK | 4d2p | C | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2501 | |
| MELK | CAMKL | CAMK | 4ump | D | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2525 | |
| MELK | CAMKL | CAMK | 5twz | A | | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 8675 | |
| MELK | CAMKL | CAMK | 5m5a | A | B | k-252a | Human | 8733 | |
| MELK | CAMKL | CAMK | 4ump | B | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2504 | |
| MELK | CAMKL | CAMK | 5tx3 | B | | 7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-one | Human | 8674 | |
| MELK | CAMKL | CAMK | 4d2v | D | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2506 | |
| MELK | CAMKL | CAMK | 4d2v | A | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2522 | |
| MELK | CAMKL | CAMK | 4umq | A | B | 3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminium | Human | 2523 | |
| MELK | CAMKL | CAMK | 5tvt | A | | 9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3-methyl-3,4-dihydropyrimido[5,4-c][1,5]naphthyridin-2(1h)-one | Human | 8667 | |
| MELK | CAMKL | CAMK | 4d2w | C | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2503 | |
| MELK | CAMKL | CAMK | 6gvx | A | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11139 | |
| MELK | CAMKL | CAMK | 5iha | A | A | 1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazine | Human | 6663 | |
| MELK | CAMKL | CAMK | 5twl | A | | 9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3,4-dihydropyrimido[5,4-c]quinolin-2(1h)-one | Human | 8668 | |
| MELK | CAMKL | CAMK | 4d2t | A | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2489 | |
| MELK | CAMKL | CAMK | 5mag | A | A | pf-3758309 | Human | 8736 | |
| MELK | CAMKL | CAMK | 4bky | A | B | 3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamide | Human | 2490 | |
| MELK | CAMKL | CAMK | 4d2v | B | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2507 | |
| MELK | CAMKL | CAMK | 4bkz | A | B | n-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 2484 | |
| MELK | CAMKL | CAMK | 4ump | A | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2497 | |
| MELK | CAMKL | CAMK | 5maf | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 8732 | |
| MELK | CAMKL | CAMK | 5ihc | A | A | 4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridine | Human | 6660 | |
| MELK | CAMKL | CAMK | 4ixp | A | | - | Human | 2528 | |
| MELK | CAMKL | CAMK | 4d2w | D | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2495 | |
| MELK | CAMKL | CAMK | 5ih8 | A | | n-[(pyridin-2-yl)methyl]-4-[4-(pyridin-4-yl)-1h-pyrazol-1-yl]benzamide | Human | 6661 | |
| DAPK1 | DAPK | CAMK | 6fha | A | B | - | Human | 11288 | |
| DAPK1 | DAPK | CAMK | 3dgk | A | B | - | Human | 5629 | |
| DAPK1 | DAPK | CAMK | 2xzs | A | A | - | Human | 5618 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 8p9b | A | | 4-[6-(4-morpholin-4-ylcarbonylphenyl)imidazo[1,2-a]pyridin-3-yl]benzenecarbonitrile | Human | 15296 | |
| DAPK1 | DAPK | CAMK | 3gu8 | A | B | n6-cyclopentyladenosine | Human | 5628 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 2vz6 | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 2471 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | B | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | 1573 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7ujq | A | | methyl 6-o-(heptylcarbamoyl)-beta-l-altropyranoside | Human | 14189 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9n | A | | 3-(4'-hydroxybiphenyl-4-yl)-n-(4-hydroxycyclohexyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamide | Human | 1690 | |
| PIM1 | PIM | CAMK | 6l15 | A | | 7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazine | Human | 12339 | |
| PIM1 | PIM | CAMK | 1yxv | A | B | 3,4-dihydroxy-1-methylquinolin-2(1h)-one | Human | 2366 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cjh | A | | 3-phenyl-5-(pyridin-4-yl)-1h-indazole | Human | 9885 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up8 | A | A | (5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | 14282 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up6 | A | B | (e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound form | Human | 14354 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3fxw | A | A | 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4596 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3fxw | A | B | 2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4593 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 6ayw | B | | n-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 8665 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | A | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1366 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | I | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1364 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | C | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1303 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1nxk | A | | staurosporine | Human | 1342 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | K | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1363 | |
| PASK | CAMKL | CAMK | 3dls | B | | adenosine-5'-diphosphate | Human | 3381 | |
| PASK | CAMKL | CAMK | 3dls | A | | adenosine-5'-diphosphate | Human | 3382 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xm8 | A | | 2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenol | Human | 4773 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bde | A | | 6-methylquinazolin-4-amine | Human | 4781 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycr | A | A | 1,3-bis{4-[(1e)-n-(4,5-dihydro-1h-imidazol-2-yl)ethanehydrazonoyl]phenyl}urea | Human | 4760 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycf | A | A | (2e)-n-hydroxy-2-[1-(4-{[(4-{(1e)-1-[2-(n'-hydroxycarbamimidoyl)hydrazinylidene]ethyl}phenyl)carbamoyl]amino}phenyl)ethylidene]hydrazinecarboximidamide | Human | 4810 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot8 | A | A | n-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1569 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fcf | A | B | 4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamide | Human | 9498 | |
| CASK | CASK | CAMK | 3mfr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 3822 | |
| CASK | CASK | CAMK | 3c0g | B | B | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3826 | |
| DCLK1 | DCAMKL | CAMK | 5jzj | A | A | amp phosphoramidate | Human | 6984 | |
| DCLK1 | DCAMKL | CAMK | 7kxw | B | | 2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 13908 | |
| DCLK1 | DCAMKL | CAMK | 7kx8 | A | | 5-ethyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 13909 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | A | A | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6425 | |
| DAPK1 | DAPK | CAMK | 3dfc | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 5620 | |
| DAPK1 | DAPK | CAMK | 6qn4 | A | | - | Human | 11589 | |
| MARK1 | CAMKL | CAMK | 6c9d | A | B | - | Human | 10051 | |
| MARK1 | CAMKL | CAMK | 2hak | E | | - | Human | 255 | |
| MARK1 | CAMKL | CAMK | 2hak | A | | - | Human | 258 | |
| MARK1 | CAMKL | CAMK | 2hak | B | | - | Human | 259 | |
| RPS6KA3-b (RSK2-b) | RSKb | CAMK | 8xey | A | | - | Human | 15207 | |
| PIM1 | PIM | CAMK | 4k0y | A | A | n-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2455 | |
| PIM1 | PIM | CAMK | 4dtk | A | A | (5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dione | Human | 2344 | |
| PIM1 | PIM | CAMK | 5n4u | A | A | 5-(2-azanyl-1,3-thiazol-4-yl)-1,3-dihydrobenzimidazol-2-one | Human | 9588 | |
| PIM1 | PIM | CAMK | 2bzh | B | A | ruthenium-pyridocarbazole-1 | Human | 7230 | |
| PIM1 | PIM | CAMK | 3umw | A | A | (2z)-2-(1h-indazol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3(2h)-one | Human | 2411 | |
| PIM1 | PIM | CAMK | 5tur | A | | 1-methyl-2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrile | Human | 8565 | |
| PIM1 | PIM | CAMK | 4rc4 | A | | 1,4-bis[(2-aminoethyl)amino]-5,8-dihydroxyanthracene-9,10-dione | Human | 2369 | |
| PIM1 | PIM | CAMK | 4lm5 | A | A | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | 2400 | |
| PIM1 | PIM | CAMK | 3umx | A | A | (2z)-7-(azepan-1-ylmethyl)-6-hydroxy-2-(1h-indol-3-ylmethylidene)-1-benzofuran-3(2h)-one | Human | 2432 | |
| PIM1 | PIM | CAMK | 5o13 | A | B | (3~{e})-5-chloranyl-3-[[5-[3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl]furan-2-yl]methylidene]-1~{h}-indol-2-one | Human | 8655 | |
| PIM1 | PIM | CAMK | 7z6u | A | B | 4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acid | Human | 14600 | |
| PIM1 | PIM | CAMK | 8r1k | A | | 6-bromanyl-1,3-benzoxazol-2-amine | Human | 15473 | |
| PIM1 | PIM | CAMK | 1xqz | A | | - | Human | 2361 | |
| PIM1 | PIM | CAMK | 5o13 | A | A | (3~{e})-5-chloranyl-3-[[5-[3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl]furan-2-yl]methylidene]-1~{h}-indol-2-one | Human | 8653 | |
| PIM1 | PIM | CAMK | 5kgg | A | | 2-(5-chloranyl-1~{h}-indol-3-yl)ethanamine | Human | 8308 | |
| PIM1 | PIM | CAMK | 2obj | A | | 6-(5-bromo-2-hydroxyphenyl)-2-oxo-4-phenyl-1,2-dihydropyridine-3-carbonitrile | Human | 2336 | |
| PIM1 | PIM | CAMK | 4wsy | A | | 5-[3-(quinolin-3-yl)-2h-indazol-5-yl]-1,3-thiazol-2-amine | Human | 2429 | |
| PIM1 | PIM | CAMK | 3we8 | A | A | cyclopentadienyl(carbon monoxide)(7-oxo-7,10-dihydro-1,8-phenanthrolin-10-yl-kappa~2~c~10~,n~1~)ruthenium | Human | 7237 | |
| PIM1 | PIM | CAMK | 4alw | A | A | 8-bromanyl-2-[(4-methylpiperazin-1-yl)methyl]-3h-[1]benzofuro[3,2-d]pyrimidin-4-one | Human | 2419 | |
| PIM1 | PIM | CAMK | 6ykd | A | B | ~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamide | Human | 12401 | |
| PIM1 | PIM | CAMK | 3c4e | D | | n-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amine | Human | 2378 | |
| PIM1 | PIM | CAMK | 3vc4 | A | | (5z)-5-[3-(trifluoromethyl)benzylidene]-1,3-thiazolidine-2,4-dione | Human | 2356 | |
| PIM1 | PIM | CAMK | 3uix | A | B | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | 2387 | |
| PIM1 | PIM | CAMK | 1yi4 | A | | adenosine | Human | 2403 | |
| PIM1 | PIM | CAMK | 5n4o | A | A | (~{e})-3-(4-methylphenyl)prop-2-enoic acid | Human | 9580 | |
| PIM1 | PIM | CAMK | 4ll5 | A | A | 6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazole | Human | 2365 | |
| PIM1 | PIM | CAMK | 4ty1 | A | | n-tert-butyl-5-[3-(4-cyclopropylpyrimidin-2-yl)-1h-indol-5-yl]-1,3,4-oxadiazol-2-amine | Human | 2394 | |
| PIM1 | PIM | CAMK | 6l11 | A | | 5-(2-chloranylphenoxazin-10-yl)-~{n},~{n}-diethyl-pentan-1-amine | Human | 12336 | |
| PIM1 | PIM | CAMK | 6no9 | A | | 5-amino-n-{5-[(4r,5r)-4-amino-5-fluoroazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamide | Human | 10936 | |
| PIM1 | PIM | CAMK | 5ipj | A | | 2-(tert-butylamino)-3-methyl-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-one | Human | 6703 | |
| PIM1 | PIM | CAMK | 4k1b | A | | n-[5-(2-fluorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-5-({[(3r,4r)-3-fluoropiperidin-4-yl]methyl}amino)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2362 | |
| PIM1 | PIM | CAMK | 5n5m | A | B | ~{n}-(isoquinolin-5-ylmethyl)-~{n}-methyl-2-[(3~{r})-pyrrolidin-3-yl]benzamide | Human | 9705 | |
| PIM1 | PIM | CAMK | 1yhs | A | | staurosporine | Human | 2444 | |
| PIM1 | PIM | CAMK | 3jpv | A | | 1,10-dihydropyrrolo[2,3-a]carbazole-3-carbaldehyde | Human | 2431 | |
| PIM1 | PIM | CAMK | 3vbq | A | A | 5-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}benzyl)-2h-1lambda~4~,3-thiazole-2,4(3h)-dione | Human | 2354 | |
| PIM1 | PIM | CAMK | 3umw | A | B | (2z)-2-(1h-indazol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3(2h)-one | Human | 2414 | |
| PIM1 | PIM | CAMK | 4xhk | B | B | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | 2355 | |
| PIM1 | PIM | CAMK | 5n52 | A | B | (~{e})-3-(2,3-dimethoxyphenyl)prop-2-enoic acid | Human | 9586 | |
| PIM1 | PIM | CAMK | 2bzk | B | | phosphoaminophosphonic acid-adenylate ester | Human | 2330 | |
| PIM1 | PIM | CAMK | 7xsv | A | A | 8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaene | Human | 14287 | |
| PIM1 | PIM | CAMK | 6pdn | A | A | 4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acid | Human | 11456 | |
| PIM1 | PIM | CAMK | 1yxs | A | A | - | Human | 2417 | |
| PIM1 | PIM | CAMK | 1yxs | A | B | - | Human | 2461 | |
| PIM1 | PIM | CAMK | 2c3i | B | B | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 2374 | |
| PIM1 | PIM | CAMK | 5dia | A | | (1s,3s)-n-{6-[5-(pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridin-3-yl]pyridin-2-yl}cyclohexane-1,3-diamine | Human | 6210 | |
| PIM1 | PIM | CAMK | 2xiz | A | A | (e)-pyridin-4-yl-acrylic acid | Human | 2436 | |
| PIM1 | PIM | CAMK | 3jy0 | A | A | 8-chloro-2-{[(3s)-3-hydroxypyrrolidin-1-yl]methyl}[1]benzothieno[3,2-d]pyrimidin-4(3h)-one | Human | 2405 | |
| PIM1 | PIM | CAMK | 4iaa | A | | 10-{2-[(2r)-1-methylpiperidin-2-yl]ethyl}-2-(methylsulfanyl)-10h-phenothiazine | Human | 2325 | |
| PIM1 | PIM | CAMK | 4k0y | A | B | n-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide | Human | 2445 | |
| PIM1 | PIM | CAMK | 5mzl | A | A | ~{n}-quinolin-5-ylpyridine-3-carboxamide | Human | 9562 | |
| PIM1 | PIM | CAMK | 6l13 | A | | 2-chloranyl-10-(2-piperidin-4-ylethyl)phenoxazine | Human | 12337 | |
| PIM1 | PIM | CAMK | 8r1t | A | A | 4-(4-aminophenethyl)benzoic acid | Human | 15212 | |
| PIM1 | PIM | CAMK | 3vbx | A | A | 6-bromo-4-hydroxy-2h-chromen-2-one | Human | 2427 | |
| PIM1 | PIM | CAMK | 2xj2 | A | A | (2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acid | Human | 2334 | |
| PIM1 | PIM | CAMK | 3bgq | A | | n-cyclohexyl-3-[3-(trifluoromethyl)phenyl][1,2,4]triazolo[4,3-b]pyridazin-6-amine | Human | 2465 | |
| PIM1 | PIM | CAMK | 4alu | A | B | 8-bromo-2-(2-chlorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3h)-one | Human | 2384 | |
| PIM1 | PIM | CAMK | 5kgd | A | | 2-pyridin-3-yl-1~{h}-benzimidazole | Human | 8309 | |
| PIM1 | PIM | CAMK | 8r18 | A | A | (e)-4-(4-hydroxystyryl)benzoic acid | Human | 15213 | |
| PIM1 | PIM | CAMK | 2bzi | B | A | - | Human | 7225 | |
| PIM1 | PIM | CAMK | 8r1w | A | | 4-(5-(4-aminophenyl)-2h-1,2,3-triazol-4-yl)benzoic acid | Human | 15476 | |
| PIM1 | PIM | CAMK | 4lm5 | A | B | 2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenol | Human | 2327 | |
| PIM1 | PIM | CAMK | 3t9i | A | | 2-methoxy-4-(3-phenyl-2h-pyrazolo[3,4-b]pyridin-6-yl)phenol | Human | 2450 | |
| PIM1 | PIM | CAMK | 2xiy | A | A | 2-hydroxymethyl-benzoimidazole | Human | 2415 | |
| PIM1 | PIM | CAMK | 5n51 | A | A | 3,4-bis(bromanyl)thiophene-2-carboxylic acid | Human | 9596 | |
| PIM1 | PIM | CAMK | 4enx | A | | (2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-nitrobenzylidene)-1,3-thiazolidin-4-one | Human | 2352 | |
| PIM2 | PIM | CAMK | 2iwi | A | | ruthenium-pyridocarbazole-1 | Human | 7217 | |
| PIM2 | PIM | CAMK | 4x7q | B | | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | 1416 | |
| PIM2 | PIM | CAMK | 4x7q | A | | 2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamide | Human | 1415 | |
| PHKG2 (PHKg2) | PHK | CAMK | 2y7j | D | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1898 | |
| CAMK2A (CaMK2a) | CAMK2 | CAMK | 7uiq | A | | - | Human | 14175 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg9 | A | | adenosine-5'-triphosphate | Human | 4846 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg9 | B | | adenosine-5'-triphosphate | Human | 4845 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fgb | A | | - | Human | 4847 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg8 | B | | adenosine-5'-triphosphate | Human | 4849 | |
| CAMK1 (CaMK1a) | CAMK1 | CAMK | 4fg8 | A | | adenosine-5'-triphosphate | Human | 4850 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 2hw7 | A | | staurosporine | Human | 764 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cjw | A | | 3-(pyridin-4-yl)imidazo[1,2-b]pyridazine | Human | 9879 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 2ac5 | A | A | - | Human | 763 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cki | A | | 3,3-dimethyl-6-[(pyrimidin-4-yl)amino]-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dione | Human | 9882 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 6cje | A | | 4-[(9h-purin-6-yl)amino]benzamide | Human | 9884 | |
| MKNK2 (MNK2) | MAPKAPK | CAMK | 2ac3 | A | | - | Human | 765 | |
| MARK4 | CAMKL | CAMK | 5es1 | A | | ~{n}-[(1~{r},6~{r})-6-azanyl-2,2-bis(fluoranyl)cyclohexyl]-5-ethyl-4-[6-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamide | Human | 6260 | |
| MARK4 | CAMKL | CAMK | 8xfl | A | | - | Human | 15101 | |
| DAPK2 | DAPK | CAMK | 2a2a | B | A | - | Human | 1115 | |
| DAPK2 | DAPK | CAMK | 2a27 | F | | - | Human | 1127 | |
| DAPK2 | DAPK | CAMK | 1z9x | A | | - | Human | 1144 | |
| DAPK2 | DAPK | CAMK | 2a27 | A | | - | Human | 1113 | |
| DAPK2 | DAPK | CAMK | 1zws | G | | - | Human | 1150 | |
| DAPK2 | DAPK | CAMK | 2a2a | C | B | - | Human | 1148 | |
| DAPK2 | DAPK | CAMK | 1wmk | E | | - | Human | 1117 | |
| DAPK2 | DAPK | CAMK | 6paw | E | | - | Human | 12439 | |
| DAPK2 | DAPK | CAMK | 1zws | D | | - | Human | 1131 | |
| DAPK2 | DAPK | CAMK | 1zws | A | | - | Human | 1121 | |
| DAPK2 | DAPK | CAMK | 2a2a | D | A | - | Human | 1120 | |
| DAPK2 | DAPK | CAMK | 1wmk | D | | - | Human | 1139 | |
| DAPK2 | DAPK | CAMK | 1zws | C | | - | Human | 1134 | |
| DAPK2 | DAPK | CAMK | 2a2a | A | B | - | Human | 1123 | |
| DAPK2 | DAPK | CAMK | 2cke | A | | n-(2-aminoethyl)isoquinoline-5-sulfonamide | Human | 1143 | |
| DAPK2 | DAPK | CAMK | 2a27 | C | | - | Human | 1125 | |
| DAPK2 | DAPK | CAMK | 1z9x | C | | - | Human | 1116 | |
| DAPK2 | DAPK | CAMK | 1wmk | A | | - | Human | 1124 | |
| DAPK2 | DAPK | CAMK | 2a2a | A | A | - | Human | 1145 | |
| DAPK2 | DAPK | CAMK | 2a27 | E | | - | Human | 1147 | |
| DAPK2 | DAPK | CAMK | 6paw | B | | - | Human | 12440 | |
| DAPK2 | DAPK | CAMK | 1wmk | C | | - | Human | 1138 | |
| DAPK2 | DAPK | CAMK | 2a2a | C | A | - | Human | 1122 | |
| DAPK2 | DAPK | CAMK | 2a27 | B | | - | Human | 1129 | |
| DAPK2 | DAPK | CAMK | 6paw | F | | - | Human | 12441 | |
| DAPK2 | DAPK | CAMK | 6paw | A | | - | Human | 12442 | |
| DAPK2 | DAPK | CAMK | 1wmk | B | | - | Human | 1140 | |
| CAMK1G (CaMK1g) | CAMK1 | CAMK | 2jam | A | B | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1221 | |
| CAMK1G (CaMK1g) | CAMK1 | CAMK | 2jam | A | A | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1218 | |
| CAMK1G (CaMK1g) | CAMK1 | CAMK | 2jam | B | A | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1220 | |
| CAMK1G (CaMK1g) | CAMK1 | CAMK | 2jam | B | B | 5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 1219 | |
| PHKG1 (PHKg1) | PHK | CAMK | 8xyb | C | | - | Human | 15264 | |
| PHKG1 (PHKg1) | PHK | CAMK | 8z5t | C | B | adenosine-5'-triphosphate | Human | 15640 | |
| PHKG1 (PHKg1) | PHK | CAMK | 8jfl | B | | - | Human | 15265 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t28 | A | A | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamide | Human | 13202 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | C | A | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4832 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | C | B | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4831 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t6f | A | A | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamide | Human | 11939 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | A | B | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4830 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 8bfs | A | B | 3~{h}-pyrrolo[2,3-c]isoquinolin-5-amine | Human | 14505 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t29 | A | A | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamide | Human | 13204 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 2jc6 | A | A | n-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amine | Human | 4829 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6qp5 | A | B | - | Human | 12029 | |
| CAMK1D (CaMK1d) | CAMK1 | CAMK | 6t28 | A | B | 2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamide | Human | 13205 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3ot3 | A | A | 5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 1696 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opu | A | | 6-azanyl-4-(3-methylphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | 8615 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym3 | A | A | ethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1644 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8siw | A | | (1s,2s)-n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)-2-(1-methyl-1h-pyrazol-4-yl)cyclopropane-1-carboxamide | Human | 14885 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5dls | A | | 1-benzyl-n-(5-{5-[3-(dimethylamino)-2,2-dimethylpropoxy]-1h-indol-2-yl}-6-oxo-1,6-dihydropyridin-3-yl)-1h-pyrazole-4-carboxamide | Human | 6151 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1zys | A | | n-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamide | Human | 1655 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | B | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1670 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmt | A | B | 2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-ol | Human | 1685 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa4 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamide | Human | 1592 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | A | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | 1684 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | A | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | 9501 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvs | A | | rel-(9r,12s)-9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2h)-dione | Human | 1591 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4rvm | A | | 3-[4-(piperidin-1-ylmethyl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1624 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft0 | A | A | 2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acid | Human | 1637 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | B | | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | 1638 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ghg | A | | 5-{5-[(s)-2-amino-3-(1h-indol-3-yl)-propoxyl]-pyridin-3-yl}-3-[1-(1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one | Human | 1581 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9p | A | | 1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}urea | Human | 1618 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | B | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | 1626 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftt | A | A | methyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1565 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | B | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | 1605 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | A | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | 1619 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bko | A | | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 13765 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftk | A | B | 3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-ol | Human | 1536 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op7 | A | | [4-[[5-chloranyl-4-(methylamino)-7~{h}-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-phenyl]-morpholin-4-yl-methanone | Human | 8609 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | A | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | 1553 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2c3k | A | | 4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenol | Human | 1674 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | B | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | 1556 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftc | A | B | 1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)urea | Human | 1680 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | A | phosphothiophosphoric acid-adenylate ester | Human | 13489 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9v | A | | 18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrile | Human | 1574 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hxq | A | | 3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-one | Human | 1587 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvr | A | | staurosporine | Human | 1585 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | A | 6-morpholin-4-yl-9h-purine | Human | 1662 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftn | A | B | 4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-ol | Human | 1678 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsu | A | A | 4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrile | Human | 1539 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2gdo | A | | 4-[(3s)-1-azabicyclo[2.2.2]oct-3-ylamino]-3-(1h-benzimidazol-2-yl)-6-chloroquinolin-2(1h)-one | Human | 1606 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2bro | A | | (2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diol | Human | 1686 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydj | A | | 5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamide | Human | 1649 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym4 | A | A | ethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylate | Human | 1572 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym8 | A | | (r)-5-(8-chloroisoquinolin-3-ylamino)-3-(1-(dimethylamino)propan-2-yloxy)pyrazine-2-carbonitrile | Human | 1588 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bk2 | A | | 4-amino-7-methyl-2-({5-methyl-1-[(3r)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13766 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3nlb | A | | 3-methyl-5-[5-(1-methylethyl)-1h-benzimidazol-2-yl]-n-(1-methylpiperidin-4-yl)-1h-pyrazole-4-carboxamide | Human | 1641 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qye | A | | 4-[6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acid | Human | 1601 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | A | adenine | Human | 13767 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyh | B | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrile | Human | 1586 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym5 | A | | (3-{4-[(2s)-2-(aminomethyl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}phenyl)methanol | Human | 1627 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8e81 | A | | (1s)-1-[(1p)-1-{6-[(3r)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}-1h-indazol-6-yl]spiro[2.2]pentane-1-carbonitrile | Human | 14620 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmx | A | | 1-[(2s)-4-(5-phenyl-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamine | Human | 1636 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | A | A | staurosporine | Human | 13490 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brb | A | | 2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanol | Human | 1582 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fta | A | B | 6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acid | Human | 1660 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4qyg | A | | 3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acid | Human | 1568 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7akm | A | B | phosphothiophosphoric acid-adenylate ester | Human | 13491 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | A | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | 14039 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | A | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | 1677 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bje | A | B | adenine | Human | 13773 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | A | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | 1691 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | B | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | 1643 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft5 | A | A | 1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1617 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ydi | A | B | 5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamide | Human | 1579 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 8six | A | | (1s)-n-(7-chloro-6-{4-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperazin-1-yl}isoquinolin-3-yl)-6-oxaspiro[2.5]octane-1-carboxamide | Human | 14887 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsq | A | A | 4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-ol | Human | 1688 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | B | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | 1645 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | A | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1699 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5f4n | A | A | methyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylate | Human | 6651 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5op5 | A | | 3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrile | Human | 8600 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ym7 | A | A | 5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrile | Human | 1650 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftl | A | A | 4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-ol | Human | 1614 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsr | A | A | 6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazole | Human | 1629 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | C | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | 1616 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brm | A | A | 3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-one | Human | 1621 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftm | A | A | 4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenol | Human | 1546 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2e9o | A | | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | 1667 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5ops | A | | 4-(3-hydroxyphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrile | Human | 8598 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | A | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | 1542 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2r0u | A | | 6-(3-aminopropyl)-4-(3-hydroxyphenyl)-9-(1h-pyrazol-4-yl)benzo[h]isoquinolin-1(2h)-one | Human | 1632 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xf0 | A | | 3-phenyl-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | 1534 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjh | A | A | n,n-dimethyl-7h-purin-6-amine | Human | 13776 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fti | A | A | methyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylate | Human | 1577 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suf | A | A | 8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amine | Human | 14040 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oor | A | | staurosporine | Human | 8603 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftr | A | A | 2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamide | Human | 1692 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | B | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1557 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2hy0 | A | | 3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-pyrazol-4-yl)quinolin-2(1h)-one | Human | 1555 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fck | A | B | 2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamide | Human | 9499 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2qhn | A | | 5-ethyl-3-methyl-1,5-dihydro-4h-pyrazolo[4,3-c]quinolin-4-one | Human | 1675 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq8 | A | | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8606 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 6fc8 | A | B | 2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamide | Human | 9502 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xez | A | | 6-(1h-pyrazol-3-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | 1580 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8e | A | | 5-methyl-8-pyridin-4-yl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1548 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oq7 | B | A | 5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamide | Human | 8605 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | B | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | 1544 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjj | A | A | 1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 13777 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suj | A | | (3r,4r)-4-{4-[6-chloro-2-({1-[(1r)-2,2-difluorocyclopropyl]-5-methyl-1h-pyrazol-4-yl}amino)quinazolin-7-yl]piperidin-1-yl}-4-methyloxolan-3-ol | Human | 14041 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvs | A | | - | Human | 1630 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | B | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | 1672 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | A | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | 1694 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7sug | A | B | 1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrile | Human | 14042 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7suh | A | | 1-[5-chloro-4-({6-chloro-7-[1-(oxetan-3-yl)piperidin-4-yl]quinazolin-2-yl}amino)-1h-pyrazol-1-yl]-2-methylpropan-2-ol | Human | 14043 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft3 | A | A | 1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylurea | Human | 1554 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3jvr | A | | - | Human | 1625 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa3 | A | B | 2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamide | Human | 1635 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fst | A | B | 4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenol | Human | 1663 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2ayp | A | | (3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-one | Human | 1682 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmu | A | B | 6-morpholin-4-yl-9h-purine | Human | 1578 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8d | A | B | 5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1620 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fto | A | A | 4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrile | Human | 1661 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oot | A | | 2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 8599 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1ia8 | A | | - | Human | 1656 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | B | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | 1671 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3f9n | A | A | - | Human | 1700 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsn | A | B | 4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acid | Human | 1679 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsm | A | A | 4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenol | Human | 1570 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2qhm | A | | (3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylate | Human | 1669 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7bjr | A | | 4-amino-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13778 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4fsz | A | B | (3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acid | Human | 1628 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7mck | A | | n-{5-[(3s)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl}-6-(1-methyl-1h-pyrazol-4-yl)pyridine-2-carboxamide | Human | 13622 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 8612 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ftu | A | A | methyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetate | Human | 1639 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4hyh | A | A | 2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamide | Human | 1561 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 4ft7 | A | A | 1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)urea | Human | 1610 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2brh | A | B | n-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycine | Human | 1654 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2cgw | A | | 4,4'-(1-propyl-1h-1,2,4-triazole-3,5-diyl)bis(2,5-dihydro-1,2,5-oxadiazol-3-amine) | Human | 1683 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2br1 | A | B | 2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanol | Human | 1571 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2x8i | A | B | 7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-one | Human | 1558 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | B | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | 1604 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3pa5 | A | A | 2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamide | Human | 1676 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5oop | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 8607 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2xey | A | | 3-(1h-indol-3-yl)-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazine | Human | 1668 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 3u9n | A | | 2-(2,3-dihydro-1-benzofuran-5-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamide | Human | 1597 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 7ako | B | B | staurosporine | Human | 13496 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 1nvq | A | | 7-hydroxystaurosporine | Human | 1642 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 5opr | A | | 5-[4-(morpholin-4-ylmethyl)phenyl]-3-(1-propan-2-yl-1,2,3-triazol-4-yl)pyridin-2-amine | Human | 8614 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7e | A | B | adenosine-5'-triphosphate | Human | 14507 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7c | A | B | adenosine-5'-diphosphate | Human | 14508 | |
| STK17B (DRAK2) | DAPK | CAMK | 3lm0 | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-5-methylpyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 6796 | |
| STK17B (DRAK2) | DAPK | CAMK | 6y6h | A | A | 2-[6-(1-benzothiophen-2-yl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12043 | |
| STK17B (DRAK2) | DAPK | CAMK | 3lm0 | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-5-methylpyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 6797 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7d | A | B | adenosine-5'-triphosphate | Human | 14509 | |
| STK17B (DRAK2) | DAPK | CAMK | 6zjf | A | A | 2-[6-(4-cyclopropylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12642 | |
| STK17B (DRAK2) | DAPK | CAMK | 3lm5 | A | A | 3,5,7,3',4'-pentahydroxyflavone | Human | 6795 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7c | A | A | adenosine-5'-diphosphate | Human | 14510 | |
| STK17B (DRAK2) | DAPK | CAMK | 6zjf | A | B | 2-[6-(4-cyclopropylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12643 | |
| STK17B (DRAK2) | DAPK | CAMK | 6y6f | A | A | 2-[6-(4-methylsulfanylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12045 | |
| STK17B (DRAK2) | DAPK | CAMK | 6y6f | A | B | 2-[6-(4-methylsulfanylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acid | Human | 12042 | |
| STK17B (DRAK2) | DAPK | CAMK | 7q7d | A | A | adenosine-5'-triphosphate | Human | 14519 | |
| STK17B (DRAK2) | DAPK | CAMK | 6qf4 | A | B | adenosine-5'-diphosphate | Human | 11396 | |
| STK17B (DRAK2) | DAPK | CAMK | 7akg | A | A | 4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-one | Human | 13005 | |
| STK17B (DRAK2) | DAPK | CAMK | 3lm5 | A | B | 3,5,7,3',4'-pentahydroxyflavone | Human | 6798 | |
| MARK3 | CAMKL | CAMK | 3fe3 | A | A | - | Human | 3267 | |
| MARK3 | CAMKL | CAMK | 2qnj | A | | - | Human | 3269 | |
| MARK3 | CAMKL | CAMK | 3fe3 | B | B | - | Human | 3265 | |
| MARK3 | CAMKL | CAMK | 2qnj | B | | - | Human | 3264 | |
| MARK3 | CAMKL | CAMK | 9vgr | A | | n-[5-[[4-[[(3r,3ar,6r,6ar)-3-methoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]-1-methyl-pyrazole-4-carboxamide | Human | 15736 | |
| MARK3 | CAMKL | CAMK | 9ysq | A | | 3-({5-chloro-2-[2-(difluoromethoxy)-4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl}amino)thiophene-2-carboxamide | Human | 15737 | |
| MARK3 | CAMKL | CAMK | 9vfo | A | | n-[5-[[4-[[(3r,3ar,6r,6ar)-3-methoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]-2-azanyl-ethanamide | Human | 15738 | |
| MARK3 | CAMKL | CAMK | 3fe3 | A | B | - | Human | 3266 | |
| MARK3 | CAMKL | CAMK | 3fe3 | B | A | - | Human | 3268 | |
| STK17A (DRAK1) | DAPK | CAMK | 7quf | A | | ~{n}-~{tert}-butyl-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide | Human | 14093 | |
| STK17A (DRAK1) | DAPK | CAMK | 7que | A | | ~{n}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide | Human | 14094 | |
| DAPK3 | DAPK | CAMK | 2j90 | B | B | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Human | 379 | |
| DAPK3 | DAPK | CAMK | 5vja | B | B | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10350 | |
| DAPK3 | DAPK | CAMK | 5a6o | A | B | - | Human | 6163 | |
| DAPK3 | DAPK | CAMK | 5a6n | A | B | 5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ide | Human | 6165 | |
| DAPK3 | DAPK | CAMK | 3bhy | A | A | (4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 385 | |
| DAPK3 | DAPK | CAMK | 5vja | A | B | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10349 | |
| DAPK3 | DAPK | CAMK | 3bhy | A | B | (4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrile | Human | 381 | |
| DAPK3 | DAPK | CAMK | 5vja | D | A | (2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamide | Human | 10348 | |
| DAPK3 | DAPK | CAMK | 5a6o | B | A | - | Human | 6168 | |
| DAPK3 | DAPK | CAMK | 1yrp | B | | - | Human | 383 | |
| DAPK3 | DAPK | CAMK | 5a6o | A | A | - | Human | 6167 | |
| MELK | CAMKL | CAMK | 4d2t | B | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2512 | |
| MELK | CAMKL | CAMK | 6gvx | B | B | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11138 | |
| MELK | CAMKL | CAMK | 5ih9 | A | B | 1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazine | Human | 6657 | |
| MELK | CAMKL | CAMK | 4bkz | A | A | n-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 2505 | |
| MELK | CAMKL | CAMK | 5mah | A | A | ~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide | Human | 8729 | |
| MELK | CAMKL | CAMK | 4d2w | B | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2482 | |
| MELK | CAMKL | CAMK | 4ump | C | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2508 | |
| MELK | CAMKL | CAMK | 4d2p | C | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2496 | |
| MELK | CAMKL | CAMK | 5iha | A | B | 1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazine | Human | 6658 | |
| MELK | CAMKL | CAMK | 4umr | A | | 4-fluoro-n-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamide | Human | 2521 | |
| MELK | CAMKL | CAMK | 6gvx | A | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11137 | |
| MELK | CAMKL | CAMK | 5twu | B | | - | Human | 8672 | |
| MELK | CAMKL | CAMK | 4d2t | B | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2520 | |
| MELK | CAMKL | CAMK | 4d2t | A | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2487 | |
| MELK | CAMKL | CAMK | 4d2p | D | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2518 | |
| MELK | CAMKL | CAMK | 4ump | D | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2516 | |
| MELK | CAMKL | CAMK | 4d2w | C | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2527 | |
| MELK | CAMKL | CAMK | 5k00 | A | B | 4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamide | Human | 7498 | |
| MELK | CAMKL | CAMK | 4d2w | D | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2481 | |
| MELK | CAMKL | CAMK | 4bl1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2519 | |
| MELK | CAMKL | CAMK | 5ihc | A | B | 4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridine | Human | 6662 | |
| MELK | CAMKL | CAMK | 4d2t | D | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2530 | |
| MELK | CAMKL | CAMK | 4d2v | A | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2493 | |
| MELK | CAMKL | CAMK | 4d2p | B | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2498 | |
| MELK | CAMKL | CAMK | 4d2w | B | A | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2500 | |
| MELK | CAMKL | CAMK | 5ih9 | A | A | 1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazine | Human | 6659 | |
| MELK | CAMKL | CAMK | 4umu | A | | (2-ethoxy-4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}phenyl)methanaminium | Human | 2517 | |
| MELK | CAMKL | CAMK | 4d2p | B | A | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2494 | |
| MELK | CAMKL | CAMK | 5mai | A | B | 3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamide | Human | 8730 | |
| MELK | CAMKL | CAMK | 6gvx | B | A | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 11136 | |
| MELK | CAMKL | CAMK | 5twy | A | | 2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 8671 | |
| MELK | CAMKL | CAMK | 4d2v | B | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2483 | |
| MELK | CAMKL | CAMK | 4umq | A | A | 3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminium | Human | 2488 | |
| MELK | CAMKL | CAMK | 4d2t | C | A | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2491 | |
| MELK | CAMKL | CAMK | 5mah | A | B | ~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamide | Human | 8734 | |
| MELK | CAMKL | CAMK | 4bky | A | A | 3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamide | Human | 2480 | |
| MELK | CAMKL | CAMK | 4d2t | C | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2526 | |
| MELK | CAMKL | CAMK | 4d2w | A | B | 4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamide | Human | 2509 | |
| MELK | CAMKL | CAMK | 4ump | A | B | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2485 | |
| MELK | CAMKL | CAMK | 5twu | A | | - | Human | 8670 | |
| MELK | CAMKL | CAMK | 5tx3 | A | | 7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-one | Human | 8673 | |
| MELK | CAMKL | CAMK | 4bl1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2514 | |
| MELK | CAMKL | CAMK | 4d2v | C | B | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2492 | |
| MELK | CAMKL | CAMK | 4umt | A | | 1-(4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}-2-methoxybenzyl)piperazinediium | Human | 2510 | |
| MELK | CAMKL | CAMK | 5mag | A | B | pf-3758309 | Human | 8731 | |
| MELK | CAMKL | CAMK | 4ump | B | A | 3-(isoquinolin-7-yl)prop-2-yn-1-ol | Human | 2524 | |
| MELK | CAMKL | CAMK | 4d2v | C | A | 7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepinium | Human | 2529 | |
| MELK | CAMKL | CAMK | 4d2p | A | B | 7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinolinium | Human | 2499 | |
| MELK | CAMKL | CAMK | 4d2t | D | B | 3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminium | Human | 2511 | |
| CHEK1 (CHK1) | CAMKL | CAMK | 2wmr | A | A | 5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-one | Human | 1609 | |
| STK17B (DRAK2) | DAPK | CAMK | 6qf4 | A | A | adenosine-5'-diphosphate | Human | 11397 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn6 | A | | - | Human | 4602 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn6 | B | | - | Human | 4601 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up7 | A | B | (2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamide | Human | 14317 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up5 | A | B | (2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrile | Human | 14278 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn5 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 4600 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up4 | A | B | (5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | 14279 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up5 | A | A | (2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrile | Human | 14280 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up6 | A | A | (e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound form | Human | 14353 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 7up8 | A | B | (5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidine | Human | 14281 | |
| RPS6KA5-b (MSK1-b) | RSKb | CAMK | 3kn5 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 4603 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3r1n | A | A | 2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-one | Human | 4589 | |
| MAPKAPK3 | MAPKAPK | CAMK | 7nrb | A | B | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 14051 | |
| MAPKAPK3 | MAPKAPK | CAMK | 7nrb | A | A | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 14052 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3fhr | A | B | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 4598 | |
| MAPKAPK3 | MAPKAPK | CAMK | 3she | A | A | n-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamide | Human | 4594 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2wel | A | B | (3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamide | Human | 2137 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 6ayw | A | | n-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamide | Human | 8666 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2vn9 | A | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2140 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2vn9 | B | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrile | Human | 2139 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 5vlo | B | | n-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Human | 8347 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2wel | A | C | (3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamide | Human | 2136 | |
| CAMK2D (CaMK2d) | CAMK2 | CAMK | 2wel | A | A | (3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamide | Human | 2138 | |
| STK11 (LKB1) | CAMKL | CAMK | 2wtk | F | | phosphoaminophosphonic acid-adenylate ester | Human | 1869 | |
| STK11 (LKB1) | CAMKL | CAMK | 2wtk | C | | phosphoaminophosphonic acid-adenylate ester | Human | 1868 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2onl | C | | - | Human | 1306 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | D | | - | Human | 1337 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6t8x | A | | (10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one | Human | 13548 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | D | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1340 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | J | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1319 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | I | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1354 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | E | A | - | Human | 12500 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | L | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1283 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kga | A | A | 6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-one | Human | 9476 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | H | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1338 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | H | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1291 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | I | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1305 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | A | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1289 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | A | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1330 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | A | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1308 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | L | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1365 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1nxk | C | | staurosporine | Human | 1312 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1nxk | D | | staurosporine | Human | 1334 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3m2w | A | A | 2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-one | Human | 9474 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | G | B | - | Human | 12501 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3fyk | X | | (3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-one | Human | 1297 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | H | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1325 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbo | A | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1333 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | A | A | - | Human | 12502 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | C | A | - | Human | 12504 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r30 | A | B | 1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acid | Human | 1309 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | A | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1281 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | D | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1284 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | G | A | - | Human | 12505 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | K | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1360 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | G | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1351 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | L | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1301 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3fyj | X | | (10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-one | Human | 1336 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | F | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1313 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | C | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1344 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | D | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1327 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | L | | - | Human | 1295 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2pzy | D | | - | Human | 1357 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3m42 | A | | 2-[5-(2-methoxyethoxy)pyridin-3-yl]-8,9,10,11-tetrahydro-7h-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin-7-one | Human | 9475 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | I | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1311 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | C | B | - | Human | 12506 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | E | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1285 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1kwp | B | | - | Human | 1296 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | L | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1324 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | G | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1343 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kga | A | B | 6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-one | Human | 9477 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | G | | - | Human | 1356 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | J | | - | Human | 1331 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | K | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1299 | |
| MAPKAPK2 | MAPKAPK | CAMK | 6tca | A | B | - | Human | 12507 | |
| MAPKAPK2 | MAPKAPK | CAMK | 9r59 | A | | 5-[3-[bis(oxidanyl)-$l^{3}-sulfanyl]oxy-4-chloranyl-phenyl]-~{n}-(4-piperazin-1-ylphenyl)-~{n}-(pyridin-2-ylmethyl)furan-2-carboxamide | Human | 16033 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r30 | A | A | 1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acid | Human | 1352 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | B | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1282 | |
| MAPKAPK2 | MAPKAPK | CAMK | 4tyh | A | A | - | Human | 1302 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | B | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1304 | |
| MAPKAPK2 | MAPKAPK | CAMK | 8xu4 | A | | - | Human | 15173 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | F | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1355 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2oza | A | | - | Human | 1310 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | B | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1298 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | F | | - | Human | 1321 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3wi6 | C | | n-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amine | Human | 1346 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | E | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1315 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | F | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1335 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3fpm | A | | 3-{[(1r)-1-phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dione | Human | 1367 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | E | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1358 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3m2w | A | B | 2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-one | Human | 9473 | |
| MAPKAPK2 | MAPKAPK | CAMK | 4tyh | A | B | - | Human | 1322 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3gok | E | | 2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 1300 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | D | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1316 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | K | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1317 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | J | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1347 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2jbp | J | | - | Human | 1359 | |
| MAPKAPK2 | MAPKAPK | CAMK | 2pzy | C | | staurosporine | Human | 1279 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3kc3 | F | | n~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamine | Human | 1341 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3a2c | J | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 1353 | |
| MAPKAPK2 | MAPKAPK | CAMK | 1nxk | B | | staurosporine | Human | 1292 | |
| MAPKAPK2 | MAPKAPK | CAMK | 3r2b | I | | - | Human | 1294 | |
| PASK | CAMKL | CAMK | 3dls | F | | adenosine-5'-diphosphate | Human | 3380 | |
| PASK | CAMKL | CAMK | 3dls | C | | adenosine-5'-diphosphate | Human | 3377 | |
| PASK | CAMKL | CAMK | 3dls | E | | adenosine-5'-diphosphate | Human | 3379 | |
| PASK | CAMKL | CAMK | 3dls | D | | adenosine-5'-diphosphate | Human | 3378 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xbj | A | | 4-fluoro-2-(4-{[(3s,4r)-4-(1-hydroxy-1-methylethyl)pyrrolidin-3-yl]amino}-6,7-dimethoxyquinazolin-2-yl)phenol | Human | 4783 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdf | A | | 5-methyl-3-phenyl-1h-pyrazole | Human | 4765 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2cn5 | A | | adenosine-5'-diphosphate | Human | 4789 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycq | A | A | n-{4-[(1e)-n-1h-imidazol-2-ylethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamide | Human | 4766 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | G | | - | Human | 4793 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | C | | - | Human | 4802 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | B | | - | Human | 4792 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wtj | A | B | 2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)-n-[2-(dimethylamino)ethyl]pyridine-3-carboxamide | Human | 4761 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdg | A | | 3-(pyridin-3-yl)-1h-pyrazol-5-amine | Human | 4796 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2cn8 | A | | debromohymenialdisine | Human | 4808 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yit | A | B | n-{4-[(1e)-n-carbamimidoylbutanehydrazonoyl]phenyl}-5-methoxy-1h-indole-2-carboxamide | Human | 4770 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdj | A | | 3-cyclopropyl-4-(furan-2-yl)-1h-pyrazolo[3,4-b]pyridine | Human | 4795 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycs | A | B | n-{4-[(1e)-n-carbamimidoylethanehydrazonoyl]phenyl}-1h-indole-3-carboxamide | Human | 4764 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycr | A | B | 1,3-bis{4-[(1e)-n-(4,5-dihydro-1h-imidazol-2-yl)ethanehydrazonoyl]phenyl}urea | Human | 4775 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2w7x | A | B | n-[4-[(e)-n-carbamimidamido-c-methyl-carbonimidoyl]phenyl]-7-nitro-1h-indole-2-carboxamide | Human | 4780 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9s | A | B | 2-(4-(3-hydroxyphenoxy)phenyl)-1h-benzo[d]imidazole-5-carboxamide | Human | 4801 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9s | A | A | 2-(4-(3-hydroxyphenoxy)phenyl)-1h-benzo[d]imidazole-5-carboxamide | Human | 4772 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdd | A | | 1-(tert-butyl)-3-(quinoxalin-6-yl)urea | Human | 4786 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wtd | A | | 4-[2-amino-5-(1,3-benzodioxol-4-yl)pyridin-3-yl]benzamide | Human | 4769 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycq | A | B | n-{4-[(1e)-n-1h-imidazol-2-ylethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamide | Human | 4790 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xm9 | A | A | 4-(1h-pyrazol-5-yl)-2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenol | Human | 4785 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9u | A | | 2-{4-[(1-benzylpiperidin-4-yl)methoxy]phenyl}-1h-benzimidazole-6-carboxamide | Human | 4778 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yit | A | A | n-{4-[(1e)-n-carbamimidoylbutanehydrazonoyl]phenyl}-5-methoxy-1h-indole-2-carboxamide | Human | 4777 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | F | | - | Human | 4776 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2w0j | A | | 4,4'-diacetyldiphenylurea-bis(guanylhydrazone) | Human | 4811 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9r | A | | 2-[4-(4-chlorophenoxy)phenyl]-1h-benzimidazole-6-carboxamide | Human | 4763 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdb | A | | 4-[(e)-c-methyl-n-oxidanyl-carbonimidoyl]benzene-1,3-diol | Human | 4797 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bda | A | | 3,4-dihydro[1,2,4]triazolo[1,5-a][3,1]benzimidazol-9-ium | Human | 4788 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4a9t | A | | 2-(4-{[1-(4-chlorobenzyl)piperidin-4-yl]methoxy}phenyl)-1h-benzimidazole-5-carboxamide | Human | 4814 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdk | A | | n-[(4-methoxyphenyl)methyl]quinoxaline-6-carboxamide | Human | 4809 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2ycs | A | A | n-{4-[(1e)-n-carbamimidoylethanehydrazonoyl]phenyl}-1h-indole-3-carboxamide | Human | 4804 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wti | A | A | 4-[2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)pyridin-3-yl]benzamide | Human | 4812 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wtj | A | A | 2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)-n-[2-(dimethylamino)ethyl]pyridine-3-carboxamide | Human | 4779 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wtc | A | | 4-[2-amino-5-(4-hydroxy-3-methoxyphenyl)pyridin-3-yl]benzamide | Human | 4767 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | E | | - | Human | 4806 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | D | | - | Human | 4805 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2xm9 | A | B | 4-(1h-pyrazol-5-yl)-2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenol | Human | 4803 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdi | A | | 1-acetyl-n-(5-methylpyridin-2-yl)piperidine-4-carboxamide | Human | 4762 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdc | A | | n-(furan-2-ylmethyl)quinoxaline-6-carboxamide | Human | 4794 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2w7x | A | A | n-[4-[(e)-n-carbamimidamido-c-methyl-carbonimidoyl]phenyl]-7-nitro-1h-indole-2-carboxamide | Human | 4784 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2yiq | A | B | (e)-5-(1-(2-carbamimidoylhydrazono)ethyl)-n-(1h-indol-6-yl)-1h-indole-2-carboxamide | Human | 4800 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | H | | - | Human | 4799 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 2wti | A | B | 4-[2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)pyridin-3-yl]benzamide | Human | 4807 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 4bdh | A | | 3-methyl-4-(thiophen-2-yl)-1h-pyrazol-5-amine | Human | 4782 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6u | A | | - | Human | 4798 | |
| CHEK2 (CHK2) | RAD53 | CAMK | 3i6w | A | | - | Human | 4813 | |
| CASK | CASK | CAMK | 3mfs | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 3829 | |
| CASK | CASK | CAMK | 3c0i | A | B | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3819 | |
| CASK | CASK | CAMK | 7oaj | A | A | 4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-n-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | Human | 13582 | |
| CASK | CASK | CAMK | 3c0h | A | | adenosine monophosphate | Human | 3825 | |
| CASK | CASK | CAMK | 3mft | A | B | - | Human | 3821 | |
| CASK | CASK | CAMK | 9m6g | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 16103 | |
| CASK | CASK | CAMK | 3mfu | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 3832 | |
| CASK | CASK | CAMK | 6kmh | B | | - | Human | 12671 | |
| CASK | CASK | CAMK | 3c0g | B | A | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3824 | |
| CASK | CASK | CAMK | 3mfr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 3831 | |
| CASK | CASK | CAMK | 3mfs | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 3818 | |
| CASK | CASK | CAMK | 3c0h | B | | adenosine monophosphate | Human | 3817 | |
| CASK | CASK | CAMK | 3tac | A | | - | Human | 3820 | |
| CASK | CASK | CAMK | 6kmh | A | | - | Human | 12672 | |
| CASK | CASK | CAMK | 7oak | A | | 2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclopentylamino)-n-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | Human | 13585 | |
| CASK | CASK | CAMK | 3mfu | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 3816 | |
| CASK | CASK | CAMK | 3mft | A | A | - | Human | 3823 | |
| CASK | CASK | CAMK | 3c0i | A | A | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3830 | |
| CASK | CASK | CAMK | 3c0g | A | A | [(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphate | Human | 3828 | |
| CASK | CASK | CAMK | 7oal | A | | 2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclohexylamino)-n-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide | Human | 13586 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9g | A | | staurosporine | Human | 10715 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 4red | B | | - | Human | 123 | |
| PRKAA1 (AMPKa1) | CAMKL | CAMK | 6c9f | A | | staurosporine | Human | 10716 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 3rny | A | A | - | Human | 5568 | |
| RPS6KA1-b (RSK3-b) | RSKb | CAMK | 4nif | D | B | - | Human | 5575 | |
| SNRK | CAMKL | CAMK | 5yks | B | | - | Human | 8661 | |
| TTN | MLCK | CAMK | 4jnw | B | B | - | Human | 128 | |
| TTN | MLCK | CAMK | 1tki | A | | - | Human | 130 | |
| TTN | MLCK | CAMK | 4jnw | B | A | - | Human | 125 | |
| TTN | MLCK | CAMK | 4jnw | A | B | - | Human | 129 | |
| TTN | MLCK | CAMK | 4jnw | A | A | - | Human | 127 | |
| CAMK4 (CaMK4) | CAMK1 | CAMK | 2w4o | A | | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 2687 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | A | B | - | Human | 8014 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | D | B | - | Human | 8013 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | B | B | - | Human | 8017 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | D | A | - | Human | 8012 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | A | A | - | Human | 8015 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | C | A | - | Human | 8018 | |
| STK40 (SgK495) | SgK495 | CAMK | 5l2q | C | B | - | Human | 8016 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 2h6d | A | B | - | Human | 194 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | A | B | staurosporine | Human | 6428 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | A | B | staurosporine | Human | 9849 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 3aqv | A | | 6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidine | Human | 193 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cfe | A | | staurosporine | Human | 195 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | C | A | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6427 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b1u | A | A | staurosporine | Human | 9848 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | C | A | staurosporine | Human | 6430 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4cff | C | | staurosporine | Human | 190 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 2h6d | A | A | - | Human | 196 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | C | B | staurosporine | Human | 6426 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 5ezv | A | A | staurosporine | Human | 6424 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 6b2e | A | | staurosporine | Human | 9851 | |
| PRKAA2 (AMPKa2) | CAMKL | CAMK | 4zhx | A | B | (5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol | Human | 6429 | |