Search results (1292 entries covering 704 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
STK11 (LKB1)CAMKLCAMK8vsuBadenosine-5'-diphosphateHuman15343
CAMK2A (CaMK2a)CAMK2CAMK7uirAadenosine-5'-triphosphateHuman14173
CAMK2A (CaMK2a)CAMK2CAMK7kl1Badenosine-5'-triphosphateHuman13062
DAPK1DAPKCAMK5auxA3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman6136
DAPK1DAPKCAMK5auzAgenisteinHuman6140
DAPK1DAPKCAMK3gu7AAadenosine-5'-diphosphateHuman5624
DAPK1DAPKCAMK3f5gAAadenosine-5'-diphosphateHuman5635
DAPK1DAPKCAMK1p4fAB5,6-dihydro-benzo[h]cinnolin-3-ylamineHuman5664
DAPK1DAPKCAMK6qmoAA-Human11587
DAPK1DAPKCAMK4yo4ABphthalazineHuman5649
DAPK1DAPKCAMK3ehaABphosphoaminophosphonic acid-adenylate esterHuman5687
DAPK1DAPKCAMK2w4jABadenosine-5'-diphosphateHuman5682
DAPK1DAPKCAMK7ccvAApiceatannolHuman13232
DAPK1DAPKCAMK3f5uABphosphoaminophosphonic acid-adenylate esterHuman5632
DAPK1DAPKCAMK3f5gABadenosine-5'-diphosphateHuman5675
DAPK1DAPKCAMK4pf4AB-Human5648
DAPK1DAPKCAMK3gubAA9-alpha-l-lyxofuranosyl-n-(2-phenylethyl)-9h-purin-6-amineHuman5674
DAPK1DAPKCAMK3gu7ABadenosine-5'-diphosphateHuman5665
DAPK1DAPKCAMK3eh9AAadenosine-5'-diphosphateHuman5621
DAPK1DAPKCAMK1jktA-Human5650
DAPK1DAPKCAMK3ehaAAphosphoaminophosphonic acid-adenylate esterHuman5636
DAPK1DAPKCAMK4b4lAB-Human5684
DAPK1DAPKCAMK4uv0A-Human5639
DAPK1DAPKCAMK2x0gAB-Human5676
DAPK1DAPKCAMK8ie5Atrans-oxyresveratrolHuman14749
DAPK1DAPKCAMK2y4pC-Human5688
DAPK1DAPKCAMK5auyA2-[2,4-bis(oxidanyl)phenyl]-3,5,7-tris(oxidanyl)chromen-4-oneHuman6134
DAPK1DAPKCAMK1jklABphosphoaminophosphonic acid-adenylate esterHuman5619
DAPK1DAPKCAMK1wvwA-Human5652
DAPK1DAPKCAMK7ccvABpiceatannolHuman13233
DAPK1DAPKCAMK7ccuAAresveratrolHuman13234
MARK3CAMKLCAMK7p1lA5-bromo-4-n-[2-(1h-imidazol-5-yl)ethyl]-2-n-[3-(morpholin-4-ylmethyl)phenyl]pyrimidine-2,4-diamineHuman13799
DAPK1DAPKCAMK2w4kABadenosine-5'-diphosphateHuman5660
DAPK1DAPKCAMK6qmoAB-Human11588
DAPK1DAPKCAMK5av2A3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman6133
DAPK1DAPKCAMK1jktB-Human5663
DAPK1DAPKCAMK5auuA2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4h-chromen-4-oneHuman6145
DAPK1DAPKCAMK2w4kAAadenosine-5'-diphosphateHuman5653
DAPK1DAPKCAMK3f5uACphosphoaminophosphonic acid-adenylate esterHuman5630
DAPK1DAPKCAMK5av4AAgenisteinHuman6135
DAPK1DAPKCAMK5av4ABgenisteinHuman6141
DAPK1DAPKCAMK2xzsBA-Human5658
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyBA-Human5573
RPS6KA1-b (RSK3-b)RSKbCAMK2wntAA-Human6862
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyAB-Human5569
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyBB-Human5574
RPS6KA1-b (RSK3-b)RSKbCAMK4nifAA-Human5572
RPS6KA1-b (RSK3-b)RSKbCAMK4nifAB-Human5570
RPS6KA1-b (RSK3-b)RSKbCAMK2wntBB-Human6861
RPS6KA1-b (RSK3-b)RSKbCAMK4nifDA-Human5571
RPS6KA1-b (RSK3-b)RSKbCAMK2wntAB-Human6859
TRIB2 (Trb2)TrblCAMK7upmA-Human14365
DAPK3DAPKCAMK5vjaCA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10345
DAPK3DAPKCAMK2j90AB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman382
DAPK3DAPKCAMK3bqrAB4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acidHuman386
DAPK3DAPKCAMK5a6nBB-Human6161
MKNK1 (MNK1)MAPKAPKCAMK2hw6B-Human2085
STK17B (DRAK2)DAPKCAMK7q7eAAadenosine-5'-triphosphateHuman14520
DAPK1DAPKCAMK3gu6ABadenosine-5'-diphosphateHuman5638
DAPK1DAPKCAMK3gu6AAadenosine-5'-diphosphateHuman5631
DAPK1DAPKCAMK6aarA-Human11468
DAPK1DAPKCAMK1jksAB-Human5633
DAPK1DAPKCAMK1jksAA-Human5657
CHEK1 (CHK1)CAMKLCAMK4ft5AB1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1633
PIM1PIMCAMK4lmuAB3,5,7,3',4'-pentahydroxyflavoneHuman2404
DAPK1DAPKCAMK7ccwABresveratrolHuman13236
DAPK1DAPKCAMK4b4lAA-Human5683
DAPK1DAPKCAMK2y4pD-Human5640
DAPK1DAPKCAMK3gubAB9-alpha-l-lyxofuranosyl-n-(2-phenylethyl)-9h-purin-6-amineHuman5673
DAPK1DAPKCAMK6in4A-Human11795
DAPK1DAPKCAMK2xuuAadenosine-5'-diphosphateHuman5627
DAPK1DAPKCAMK3f5uAAphosphoaminophosphonic acid-adenylate esterHuman5677
DAPK1DAPKCAMK4yo4AAphthalazineHuman5686
DAPK1DAPKCAMK2y4pA-Human5659
DAPK1DAPKCAMK3eh9ACadenosine-5'-diphosphateHuman5655
DAPK1DAPKCAMK4ypdAA4-methylpyridazineHuman5654
DAPK1DAPKCAMK3zxtBphosphomethylphosphonic acid adenylate esterHuman5666
DAPK1DAPKCAMK3gu8AAn6-cyclopentyladenosineHuman5679
DAPK1DAPKCAMK6fhbAB-Human11291
DAPK1DAPKCAMK7ccwAAresveratrolHuman13235
DAPK1DAPKCAMK8ie8A5-[(~{e})-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]benzene-1,3-diolHuman14750
DAPK1DAPKCAMK8ie6A3-[(e)-2-(4-hydroxyphenyl)ethenyl]-5-methoxy-phenolHuman14751
DAPK1DAPKCAMK3gu5ACphosphoaminophosphonic acid-adenylate esterHuman5662
DAPK1DAPKCAMK2yakAAruthenium octasporine 4Human7259
DAPK2DAPKCAMK1wmkG-Human1142
DAPK1DAPKCAMK1ig1Aphosphoaminophosphonic acid-adenylate esterHuman5615
DAPK1DAPKCAMK4txcA4-(3-{3-[(r)-{[2-(dimethylamino)ethyl]amino}(hydroxy)methyl]phenyl}imidazo[1,2-b]pyridazin-6-yl)-2-methoxyphenolHuman5668
DAPK1DAPKCAMK1wvyAstaurosporineHuman5661
DAPK1DAPKCAMK5auwA3,5,7,3',4'-pentahydroxyflavoneHuman6144
DAPK1DAPKCAMK2w4jAAadenosine-5'-diphosphateHuman5678
DAPK1DAPKCAMK1jklAAphosphoaminophosphonic acid-adenylate esterHuman5685
DAPK1DAPKCAMK4pf4AA-Human5643
DAPK1DAPKCAMK5autA8-anilino-1-naphthalene sulfonateHuman6137
CHEK1 (CHK1)CAMKLCAMK2wmtAA2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-olHuman1576
DAPK1DAPKCAMK3gu5ABphosphoaminophosphonic acid-adenylate esterHuman5669
CHEK1 (CHK1)CAMKLCAMK2ywpA1-(5-chloro-2,4-dimethoxyphenyl)-3-(5-cyanopyrazin-2-yl)ureaHuman1658
CHEK1 (CHK1)CAMKLCAMK4fswAB8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1623
DAPK1DAPKCAMK3zxtCphosphomethylphosphonic acid adenylate esterHuman5646
DAPK1DAPKCAMK4tl0A-Human5641
DAPK1DAPKCAMK3gu5AAphosphoaminophosphonic acid-adenylate esterHuman5680
DAPK1DAPKCAMK2y4pB-Human5626
DAPK1DAPKCAMK3zxtDphosphomethylphosphonic acid adenylate esterHuman5617
DAPK1DAPKCAMK3eh9ABadenosine-5'-diphosphateHuman5622
CHEK1 (CHK1)CAMKLCAMK2ym6AA1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamineHuman1563
CHEK1 (CHK1)CAMKLCAMK6fcfAA4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamideHuman9503
DAPK1DAPKCAMK2x0gAA-Human5672
DAPK1DAPKCAMK5auvA5,7-dihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman6139
DAPK1DAPKCAMK6fhbAA-Human11290
DAPK1DAPKCAMK4ypdAB4-methylpyridazineHuman5623
DAPK1DAPKCAMK3zxtAphosphomethylphosphonic acid adenylate esterHuman5634
DCLK1DCAMKLCAMK6kyrBB-Human12804
CHEK1 (CHK1)CAMKLCAMK2hxlA3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)-1h-indazole-6-carbonitrileHuman1552
CHEK1 (CHK1)CAMKLCAMK2cgxA2-[(6-amino-7h-purin-8-yl)thio]acetamideHuman1595
DAPK1DAPKCAMK5av3A3,5,7-trihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman6143
DAPK1DAPKCAMK7ccuABresveratrolHuman13237
DAPK1DAPKCAMK3gu4AAphosphoaminophosphonic acid-adenylate esterHuman5670
DAPK1DAPKCAMK5av0A3-(3,4-dihydroxyphenyl)-7-hydroxy-4h-chromen-4-oneHuman6142
DAPK1DAPKCAMK5av1A-Human6138
DAPK1DAPKCAMK3ehaACphosphoaminophosphonic acid-adenylate esterHuman5647
DAPK1DAPKCAMK8ie7ApterostilbeneHuman14752
DAPK1DAPKCAMK2y0aA-Human5651
PRKAA2 (AMPKa2)CAMKLCAMK6b1uCAstaurosporineHuman9847
PIM1PIMCAMK3vbyAfuran-2-yl(1h-indol-3-yl)methanoneHuman2466
CHEK1 (CHK1)CAMKLCAMK3f9nAB-Human1666
CHEK1 (CHK1)CAMKLCAMK2yerAB5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-oneHuman1583
CASKCASKCAMK3c0gAB[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3827
PIM1PIMCAMK3vbwA1,3-dioxo-2,3-dihydro-1h-indene-2-carbonitrileHuman2390
PIM1PIMCAMK5v80A1-methyl-4-{3-[6-(piperazin-1-yl)pyridin-2-yl]-1h-pyrazolo[3,4-c]pyridin-5-yl}piperazin-2-oneHuman9828
PIM1PIMCAMK2xixAB3,5-diamino-1h-[1,2,4]triazoleHuman2433
PIM1PIMCAMK5n4rAA2-(azepan-1-yl)-1-(1~{h}-indol-3-yl)propan-1-oneHuman9584
PIM1PIMCAMK1xwsAA3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2343
CHEK1 (CHK1)CAMKLCAMK5op4A[4-[[4-(ethylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino]-2-fluoranyl-5-methoxy-phenyl]-morpholin-4-yl-methanoneHuman8613
CHEK1 (CHK1)CAMKLCAMK2wmvA1-[(2s)-4-(7h-purin-6-yl)morpholin-2-yl]methanamineHuman1562
DAPK1DAPKCAMK1jkkAphosphoaminophosphonic acid-adenylate esterHuman5644
DAPK1DAPKCAMK1p4fAA5,6-dihydro-benzo[h]cinnolin-3-ylamineHuman5625
DAPK1DAPKCAMK2xzsAB-Human5642
DAPK1DAPKCAMK3dgkAA-Human5656
DAPK1DAPKCAMK3dfcBAphosphoaminophosphonic acid-adenylate esterHuman5645
DAPK1DAPKCAMK2yakABruthenium octasporine 4Human7260
PRKAA2 (AMPKa2)CAMKLCAMK6bx6AA2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman9878
CAMK2B (CaMK2b)CAMK2CAMK3bhhD-Human1504
CAMK2B (CaMK2b)CAMK2CAMK3bhhB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1506
CHEK1 (CHK1)CAMKLCAMK4ftkAA3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-olHuman1608
CAMK2B (CaMK2b)CAMK2CAMK3bhhC-Human1505
CHEK1 (CHK1)CAMKLCAMK4ftrAB2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamideHuman1535
CAMK2B (CaMK2b)CAMK2CAMK3bhhA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-6-(methylamino)pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1507
CHEK1 (CHK1)CAMKLCAMK4hyiAB2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman1681
CHEK1 (CHK1)CAMKLCAMK4ftiABmethyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylateHuman1659
CHEK1 (CHK1)CAMKLCAMK5oq7AA5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8601
CHEK1 (CHK1)CAMKLCAMK4fswAA8-chloro-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1541
CHEK1 (CHK1)CAMKLCAMK2wmwA1-[(2s)-4-(5-bromo-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamineHuman1594
CHEK1 (CHK1)CAMKLCAMK1zltA(4z)-4-(2-amino-5-oxo-3,5-dihydro-4h-imidazol-4-ylidene)-2,3-dichloro-4,5,6,7-tetrahydropyrrolo[2,3-c]azepin-8(1h)-oneHuman1596
CHEK1 (CHK1)CAMKLCAMK5oq6A2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman8610
PIM1PIMCAMK5vubBB(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9076
CHEK1 (CHK1)CAMKLCAMK2ydkA2-(carbamoylamino)-5-phenyl-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamideHuman1646
CHEK1 (CHK1)CAMKLCAMK5opbAA(2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholineHuman8602
CHEK1 (CHK1)CAMKLCAMK2brnA(2r)-1-[(5,6-diphenyl-7h-pyrrolo[2,3-d]pyrimidin-4-yl)amino]propan-2-olHuman1631
CHEK1 (CHK1)CAMKLCAMK4ftnAA4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-olHuman1695
CHEK1 (CHK1)CAMKLCAMK5opvA4-(3-methylphenyl)-6-[(1-methylpyrazol-3-yl)amino]-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrileHuman8608
CHEK1 (CHK1)CAMKLCAMK4fsuAB4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrileHuman1615
PIM1PIMCAMK3jxwA8-[(e)-2-cyclopropylethenyl]-2-[(dimethylamino)methyl][1]benzothieno[3,2-d]pyrimidin-4(3h)-oneHuman2393
DCLK1DCAMKLCAMK6kyqAB-Human12798
DCLK1DCAMKLCAMK6kyqAA-Human12799
DCLK1DCAMKLCAMK6kyrAB-Human12800
DCLK1DCAMKLCAMK6kyqBB-Human12801
MARK2CAMKLCAMK3iecA-Human3045
MARK2CAMKLCAMK5kz7A7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-oneHuman7967
MARK2CAMKLCAMK5kz8A5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-oneHuman7965
MARK2CAMKLCAMK5eakAn-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHuman6410
DCLK1DCAMKLCAMK7kx6A2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman13907
DCLK1DCAMKLCAMK6kyqBA-Human12802
PIM1PIMCAMK3we8ABcyclopentadienyl(carbon monoxide)(7-oxo-7,10-dihydro-1,8-phenanthrolin-10-yl-kappa~2~c~10~,n~1~)rutheniumHuman7232
PIM1PIMCAMK2o65A5,7-dihydroxy-2-(3,4,5-trihydroxyphenyl)-4h-chromen-4-oneHuman2324
CHEK1 (CHK1)CAMKLCAMK2ydjB5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman1687
PIM1PIMCAMK2xj0AB(e)-3-(2-amino-pyridine-5yl)-acrylic acidHuman2395
PIM1PIMCAMK6l16A2-[4-[2-(7-chloranylpyrido[3,4-b][1,4]benzoxazin-5-yl)ethyl]piperidin-1-yl]ethanamineHuman12335
PIM1PIMCAMK4n70ABn-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamideHuman2357
RPS6KA1-b (RSK3-b)RSKbCAMK2wntBA-Human6860
MKNK1 (MNK1)MAPKAPKCAMK2hw6A-Human2084
MKNK1 (MNK1)MAPKAPKCAMK5wvdB1-methyl-n-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamideHuman9465
MKNK1 (MNK1)MAPKAPKCAMK5wvdA1-methyl-n-(5-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxamideHuman9464
PIM1PIMCAMK4jx7A2-[(trans-4-aminocyclohexyl)amino]-4-{[3-(trifluoromethyl)phenyl]amino}pyrido[4,3-d]pyrimidin-5(6h)-oneHuman2340
MYLK4 (SgK085)MLCKCAMK2x4fBA4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amineHuman4866
DAPK1DAPKCAMK6fhaAA-Human11289
MYLK4 (SgK085)MLCKCAMK2x4fAB4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amineHuman4867
PIM1PIMCAMK5ndtAA3-(2-thiophen-2-ylethenyl)-1~{h}-quinoxalin-2-oneHuman9907
PIM1PIMCAMK2o3pAB3,5,7,3',4'-pentahydroxyflavoneHuman2409
CHEK1 (CHK1)CAMKLCAMK7bjjAB1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman13779
PIM1PIMCAMK3vbvA8-hydroxyquinoline-2-carboxamideHuman2399
PIM1PIMCAMK5vucBB(2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-oneHuman9075
DAPK1DAPKCAMK2xzsBB-Human5671
PIM1PIMCAMK4n70AAn-{4-[(3r,4r,5s)-3-amino-4-hydroxy-5-methylpiperidin-1-yl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamideHuman2388
CHEK2 (CHK2)RAD53CAMK2xk9An-{4-[(1e)-n-(n-hydroxycarbamimidoyl)ethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamideHuman4771
CHEK2 (CHK2)RAD53CAMK2yiqAA(e)-5-(1-(2-carbamimidoylhydrazono)ethyl)-n-(1h-indol-6-yl)-1h-indole-2-carboxamideHuman4791
CHEK2 (CHK2)RAD53CAMK2yirA(e)-n-(5-(2-carbamimidoylhydrazono)-5,6,7,8-tetrahydronaphthalen-2-yl)-7-nitro-1h-indole-2-carboxamideHuman4768
CHEK2 (CHK2)RAD53CAMK2ycfAB(2e)-n-hydroxy-2-[1-(4-{[(4-{(1e)-1-[2-(n'-hydroxycarbamimidoyl)hydrazinylidene]ethyl}phenyl)carbamoyl]amino}phenyl)ethylidene]hydrazinecarboximidamideHuman4774
CHEK2 (CHK2)RAD53CAMK3i6uB-Human4787
PIM1PIMCAMK2oi4XA-Human7236
PIM1PIMCAMK3a99Aphosphoaminophosphonic acid-adenylate esterHuman2322
PIM1PIMCAMK5kgeA5-(3,4-dichlorophenyl)-1~{h}-pyrazol-3-amineHuman8310
PIM1PIMCAMK3qf9AA6-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}naphthalene-1-carboxamideHuman2329
PIM1PIMCAMK5n51AB3,4-bis(bromanyl)thiophene-2-carboxylic acidHuman9591
PIM1PIMCAMK3c4eAn-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amineHuman2413
PIM1PIMCAMK5dgzA(2s)-1-(1h-indol-3-yl)-3-{[5-(3-methyl-1h-indazol-5-yl)pyridin-3-yl]oxy}propan-2-amineHuman6209
CHEK1 (CHK1)CAMKLCAMK2ym4ABethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1560
CHEK1 (CHK1)CAMKLCAMK2wmqAn-(4-oxo-5,6,7,8-tetrahydro-4h-[1,3]thiazolo[5,4-c]azepin-2-yl)acetamideHuman1647
PIM1PIMCAMK5kgiA2-[3,4-bis(chloranyl)phenoxy]ethanamineHuman8306
MYLK4 (SgK085)MLCKCAMK2x4fAA4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amineHuman4865
DAPK1DAPKCAMK3gu4ABphosphoaminophosphonic acid-adenylate esterHuman5681
PIM1PIMCAMK5n52AA(~{e})-3-(2,3-dimethoxyphenyl)prop-2-enoic acidHuman9581
PIM1PIMCAMK5n50AB2-(4-chlorophenyl)sulfanylethanehydrazideHuman9598
PIM1PIMCAMK7qfmAA4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHuman14561
PRKAA1 (AMPKa1)CAMKLCAMK4rerAstaurosporineHuman121
PRKAA1 (AMPKa1)CAMKLCAMK4redA-Human122
PRKAA1 (AMPKa1)CAMKLCAMK4rewAstaurosporineHuman124
PRKAA1 (AMPKa1)CAMKLCAMK7jhgA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman13816
PRKAA1 (AMPKa1)CAMKLCAMK6c9hAstaurosporineHuman10714
PRKAA1 (AMPKa1)CAMKLCAMK7jhhA-Human13817
PRKAA1 (AMPKa1)CAMKLCAMK7m74A6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman14017
PRKAA1 (AMPKa1)CAMKLCAMK7jijB-Human13819
PRKAA1 (AMPKa1)CAMKLCAMK6c9jAstaurosporineHuman10717
CHEK1 (CHK1)CAMKLCAMK5opbAB(2~{r},6~{s})-2,6-dimethyl-4-[6-[5-(1-methylcyclopropyl)oxy-1~{h}-indazol-3-yl]pyrimidin-4-yl]morpholineHuman8604
CHEK1 (CHK1)CAMKLCAMK7bjxAA4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13772
CHEK1 (CHK1)CAMKLCAMK7bjdAA2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrileHuman13775
CHEK1 (CHK1)CAMKLCAMK7bjxAB4-amino-7-methyl-2-[(1-methyl-1h-pyrazol-4-yl)amino]-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13768
CASKCASKCAMK7oaiAB4-(cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-n-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideHuman13583
CASKCASKCAMK7oaiAA4-(cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-n-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideHuman13584
CHEK1 (CHK1)CAMKLCAMK7bk1A4-amino-2-[(1,3-dimethyl-1h-pyrazol-4-yl)amino]-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13763
CASKCASKCAMK7oajAB4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-n-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamideHuman13581
PIM1PIMCAMK3cxwAB(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman2392
PIM1PIMCAMK2bzjABruthenium-pyridocarbazole-3Human7228
PIM1PIMCAMK6l14A2-chloranyl-10-[3-[(3~{s})-piperidin-3-yl]propyl]phenoxazineHuman12338
PIM1PIMCAMK5v82A1-{6-[(3r)-4,4-difluoropiperidin-3-yl]pyridin-2-yl}-6-(6-methylpyrazin-2-yl)-1h-pyrazolo[4,3-c]pyridineHuman7581
PIM1PIMCAMK1yxvAA3,4-dihydroxy-1-methylquinolin-2(1h)-oneHuman2367
TRIB1 (Trb1)TrblCAMK5cekA-Human6241
PIM1PIMCAMK5vuaBA(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9074
PIM1PIMCAMK2j2iBA(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHuman2318
PIM1PIMCAMK5telAB4-chloro-2-{5,6-dimethoxy-1-[2-(4-methylpiperazin-1-yl)ethyl]-1h-indol-3-yl}-1h-pyrrolo[2,3-b]pyridineHuman8562
CHEK1 (CHK1)CAMKLCAMK7bjoA4-amino-6-(2,3-difluorophenyl)-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13780
CHEK1 (CHK1)CAMKLCAMK7suiA(3r,4r)-4-{(3s,4s)-4-[6-chloro-2-({5-chloro-1-[(1r)-2,2-difluorocyclopropyl]-1h-pyrazol-4-yl}amino)quinazolin-7-yl]-3-fluoropiperidin-1-yl}oxolan-3-olHuman14045
CAMK2A (CaMK2a)CAMK2CAMK6vzkA4'-hydroxycinnamic acidHuman12165
DCLK1DCAMKLCAMK5jzjBAamp phosphoramidateHuman6985
DCLK1DCAMKLCAMK5jzjBBamp phosphoramidateHuman6983
MARK2CAMKLCAMK5kz8B5,5-dimethyl-7-[(1~{s})-4-oxidanyl-1~{h}-inden-1-yl]-2-phenylazanyl-pyrrolo[2,3-d]pyrimidin-6-oneHuman7968
MARK2CAMKLCAMK5kz7B7-[(1~{s})-1-(4-fluorophenyl)ethyl]-5,5-dimethyl-2-(pyridin-3-ylamino)pyrrolo[2,3-d]pyrimidin-6-oneHuman7966
PIM1PIMCAMK4gw8AA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman2428
MARK2CAMKLCAMK3iecC-Human3046
MARK2CAMKLCAMK5eakBn-[(1s,2r)-2-aminocyclohexyl]-4-[6-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHuman6411
MARK2CAMKLCAMK3iecB-Human3044
MARK2CAMKLCAMK3iecD-Human3043
PIM1PIMCAMK5iisA3-amino-n-(2'-amino-6'-methyl[4,4'-bipyridin]-3-yl)-6-(2-fluorophenyl)pyridine-2-carboxamideHuman6504
MARK1CAMKLCAMK2hakD-Human257
SIK3 (QSK)CAMKLCAMK8r4qA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman15241
SIK3 (QSK)CAMKLCAMK8r4oA2-[bis(fluoranyl)methoxy]-4-[6-(2-cyanopropan-2-yl)pyrazolo[1,5-a]pyridin-3-yl]-~{n}-[(1~{r},2~{s})-2-fluoranylcyclopropyl]-6-methoxy-benzamideHuman15242
SIK3 (QSK)CAMKLCAMK8r4uA8-[(5-azanyl-1,3-dioxan-2-yl)methyl]-6-[2-chloranyl-4-(3-fluoranylpyridin-2-yl)phenyl]-2-(methylamino)pyrido[2,3-d]pyrimidin-7-oneHuman15240
SIK3 (QSK)CAMKLCAMK8r4vA1-(2,4-dimethoxyphenyl)-3-(2,6-dimethylphenyl)-1-[6-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]ureaHuman15243
CAMK2D (CaMK2d)CAMK2CAMK8usoA-Human15247
PHKG1 (PHKg1)PHKCAMK8z5tCAadenosine-5'-triphosphateHuman15642
PHKG1 (PHKg1)PHKCAMK8z5pC-Human15643
CHEK1 (CHK1)CAMKLCAMK10iaA(10as,13as)-3-cyclopropyl-1-methyl-8-(trifluoromethyl)-3,4,10a,11,13a,14-hexahydro-10h,13h-9,5-(azeno)furo[3,4-k]pyrazolo[4,3-b][1,4,6,10]oxatriazacyclotridecineHuman15693
CHEK1 (CHK1)CAMKLCAMK10hzA(10as,13as)-3-cyclobutyl-1-methyl-8-(trifluoromethyl)-3,4,10a,11,13a,14-hexahydro-10h,13h-9,5-(azeno)furo[3,4-k]pyrazolo[4,3-b][1,4,6,10]oxatriazacyclotridecineHuman15694
CHEK1 (CHK1)CAMKLCAMK10hyA(11r)-8-chloro-3,11-dimethyl-2-(oxan-4-yl)-2,4,10,11,12,13-hexahydro-9,5-(azeno)pyrazolo[3,4-b][1,4,6,10]oxatriazacyclotridecineHuman15695
MAPKAPK2MAPKAPKCAMK8xx1AA-Human15257
MARK3CAMKLCAMK8uohAB-Human15733
MARK3CAMKLCAMK9virA~{n}-[5-[[4-[[(3~{r},3~{a}~{r},6~{a}~{s})-3-methoxy-2,3,3~{a},6~{a}-tetrahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[[(2~{r},8~{r})-2-fluoranyl-1,2,3,5,6,7-hexahydropyrrolizin-8-yl]methoxy]phenyl]-1-methyl-pyrazole-4-carboxamideHuman15734
MARK3CAMKLCAMK8uohAA-Human15735
RPS6KA5-b (MSK1-b)RSKbCAMK7up4AA(5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14277
MAPKAPK2MAPKAPKCAMK8xx1AB-Human15256
PIM1PIMCAMK4rc2A1-amino-5,8-dihydroxy-4-({2-[(2-hydroxyethyl)amino]ethyl}amino)anthracene-9,10-dioneHuman2346
PIM1PIMCAMK1xr1Aphosphoaminophosphonic acid-adenylate esterHuman2406
PIM1PIMCAMK5n4nAB3,4-dimethyl-5-(1~{h}-1,2,4-triazol-3-yl)thiophene-2-carbonitrileHuman9595
PIM1PIMCAMK7oovA-Human13824
PIM1PIMCAMK4i41A1,4-dihydroxy-5,8-bis({2-[(2-hydroxyethyl)amino]ethyl}amino)-9,10-anthracenedioneHuman2326
PIM1PIMCAMK4gw8AB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman2391
PIM1PIMCAMK6bskA4-{6-[6-(propan-2-ylamino)-1h-indazol-1-yl]pyrazin-2-yl}benzoic acidHuman9758
PIM1PIMCAMK4rc3A1,4-dihydroxy-5,8-bis{[2-(2-hydroxyethoxy)ethyl]amino}anthracene-9,10-dioneHuman2412
MELKCAMKLCAMK9f31An-[4-(1h-indazol-5-yl)phenyl]propanamideHuman15787
PIM1PIMCAMK4lmuAA3,5,7,3',4'-pentahydroxyflavoneHuman2376
PIM1PIMCAMK5n4uAB5-(2-azanyl-1,3-thiazol-4-yl)-1,3-dihydrobenzimidazol-2-oneHuman9590
PIM1PIMCAMK6aydAAn-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamideHuman9442
DAPK1DAPKCAMK9inwA(~{e})-1-[2,4-bis(oxidanyl)phenyl]-3-(3-chloranyl-4-oxidanyl-phenyl)prop-2-en-1-oneHuman15839
DAPK1DAPKCAMK9inxA(~{e})-1-[2,4-bis(oxidanyl)phenyl]-3-(3-bromanyl-4-oxidanyl-phenyl)prop-2-en-1-oneHuman15840
DAPK1DAPKCAMK9dubAB4-(pyridin-4-yl)pyridazineHuman15841
DAPK1DAPKCAMK9dubAA4-(pyridin-4-yl)pyridazineHuman15842
DAPK1DAPKCAMK9invA2',4,4'-trihydroxychalconeHuman15843
PIM1PIMCAMK5n4yAB2,5-dihydro-1~{h}-isothiochromeno[4,3-c]pyrazol-3-oneHuman9597
CAMK2D (CaMK2d)CAMK2CAMK9blhAB7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman16000
CAMK2D (CaMK2d)CAMK2CAMK9blhAA7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman16001
CHEK1 (CHK1)CAMKLCAMK7akoABstaurosporineHuman13495
CASKCASKCAMK9m6gABphosphoaminophosphonic acid-adenylate esterHuman16104
CASKCASKCAMK8y68AA-Human16105
CASKCASKCAMK9m5yABphosphoaminophosphonic acid-adenylate esterHuman16106
CASKCASKCAMK9m5yAAphosphoaminophosphonic acid-adenylate esterHuman16107
CASKCASKCAMK8y68AB-Human16108
PIM1PIMCAMK5o11AB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman8657
CHEK1 (CHK1)CAMKLCAMK4gh2AB3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1652
CHEK1 (CHK1)CAMKLCAMK2hogA(5-{3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-1h-indazol-6-yl}-2h-1,2,3-triazol-4-yl)methanolHuman1653
CHEK1 (CHK1)CAMKLCAMK4fsqAB4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-olHuman1598
CHEK1 (CHK1)CAMKLCAMK5op2AA5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8595
CHEK1 (CHK1)CAMKLCAMK4qyfA4-[3-amino-6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acidHuman1622
CHEK1 (CHK1)CAMKLCAMK2brgA(5,6-diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-aceticHuman1589
MKNK2 (MNK2)MAPKAPKCAMK2ac5AB-Human766
CAMK2A (CaMK2a)CAMK2CAMK7kl0Amethyl 6-o-(heptylcarbamoyl)-beta-l-altropyranosideHuman13111
CAMK2A (CaMK2a)CAMK2CAMK7uisA-Human14174
CAMK2A (CaMK2a)CAMK2CAMK7ujrA-Human14191
CAMK2A (CaMK2a)CAMK2CAMK7kl2A-Human13064
PRKAA2 (AMPKa2)CAMKLCAMK7myjA(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman14273
TTNMLCKCAMK6ygnA-Human13488
TTNMLCKCAMK6ygnB-Human13487
CHEK1 (CHK1)CAMKLCAMK7bjdAB2-methyl-2-(3-methyl-4-{[4-(methylamino)-5-(trifluoromethyl)pyrimidin-2-yl]amino}-1h-pyrazol-1-yl)propanenitrileHuman13774
PIM1PIMCAMK4rblA1,4,5,8-tetrahydroxyanthracene-9,10-dioneHuman2385
PIM1PIMCAMK3bwfAB-Human7235
PIM1PIMCAMK3r02AA7-[(cis-4-aminocyclohexyl)amino]-5-bromo-1-benzofuran-2-carboxylic acidHuman2420
PIM2PIMCAMK2iwiBruthenium-pyridocarbazole-1Human7216
CAMK1D (CaMK1d)CAMK1CAMK8bfsAA3~{h}-pyrrolo[2,3-c]isoquinolin-5-amineHuman14506
MAPKAPK2MAPKAPKCAMK3r2bK-Human1293
MAPKAPK2MAPKAPKCAMK3r2bA2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-oneHuman1287
MAPKAPK2MAPKAPKCAMK3kc3Dn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1288
MAPKAPK2MAPKAPKCAMK3r2bH-Human1348
MAPKAPK2MAPKAPKCAMK3gokC2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1350
MAPKAPK2MAPKAPKCAMK3wi6En-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1323
MAPKAPK2MAPKAPKCAMK2onlD-Human1345
MARK1CAMKLCAMK2hakG-Human256
MARK1CAMKLCAMK2hakF-Human254
MAPKAPK2MAPKAPKCAMK3a2cCn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1328
MAPKAPK2MAPKAPKCAMK2jbpG2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1339
MAPKAPK2MAPKAPKCAMK2pzyB(4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamideHuman1307
MAPKAPK2MAPKAPKCAMK3r2bG-Human1369
MAPKAPK2MAPKAPKCAMK3r2bC-Human1368
MAPKAPK2MAPKAPKCAMK3r2bE-Human1286
MAPKAPK2MAPKAPKCAMK2jbpB2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1320
MAPKAPK2MAPKAPKCAMK3a2cBn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1332
PRKAA2 (AMPKa2)CAMKLCAMK2yzaA-Human189
PHKG2 (PHKg2)PHKCAMK2y7jBAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1897
PHKG2 (PHKg2)PHKCAMK2y7jCAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1896
PHKG2 (PHKg2)PHKCAMK2y7jAAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1894
CHEK1 (CHK1)CAMKLCAMK2ym6AB1-[(2r)-4-(9h-pyrido[4',3':4,5]pyrrolo[2,3-d]pyrimidin-4-yl)morpholin-2-yl]methanamineHuman1559
PIM1PIMCAMK2c3iBA1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman2348
PIM1PIMCAMK4n6zA3-amino-n-{4-[(3s)-3-aminopiperidin-1-yl]pyridin-3-yl}pyrazine-2-carboxamideHuman2442
PIM1PIMCAMK2xj0AA(e)-3-(2-amino-pyridine-5yl)-acrylic acidHuman2435
PIM1PIMCAMK5toeA2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrileHuman8563
PIM1PIMCAMK2o64A3,5,6,7-tetrahydroxy-2-(3,4-dihydroxyphenyl)-4h-chromen-4-oneHuman2421
PIM1PIMCAMK8r18AB(e)-4-(4-hydroxystyryl)benzoic acidHuman15208
PIM1PIMCAMK4ll5AB6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazoleHuman2382
PIM1PIMCAMK2j2iBB(9r)-9-[(dimethylamino)methyl]-6,7,10,11-tetrahydro-9h,18h-5,21:12,17-dimethenodibenzo[e,k]pyrrolo[3,4-h][1,4,13]oxadiazacyclohexadecine-18,20-dioneHuman2434
PIM1PIMCAMK4alvAB8-bromo-2-{2-chloro-4-[(piperidin-4-ylmethyl)amino]phenyl}[1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman2396
PIM1PIMCAMK7qfmAB4-[(~{e})-(2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHuman14560
PIM1PIMCAMK3vbxAB6-bromo-4-hydroxy-2h-chromen-2-oneHuman2448
PIM1PIMCAMK31ruA6-chloranyl-3-[4-(1~{h}-indol-3-yl)-1~{h}-pyrazol-5-yl]quinazolin-4-oneHuman15474
PIM1PIMCAMK1xwsAB3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2441
PIM1PIMCAMK8r10AB(z)-4-(4-hydroxystyryl)benzoic acidHuman15209
PIM1PIMCAMK8afrAB4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acidHuman14601
PIM1PIMCAMK8r1pA4-(4-aminostyryl)benzoic acidHuman15210
PIM1PIMCAMK8r1tAB4-(4-aminophenethyl)benzoic acidHuman15211
PIM1PIMCAMK8r25A4-(5-(4-aminophenyl)-1h-pyrazol-1-yl)benzoic acidHuman15475
PIM1PIMCAMK5n5lAB5-bromanyl-1~{h}-indole-3-carboxylic acidHuman9704
PIM1PIMCAMK7z6uAA4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHuman14602
PIM1PIMCAMK5dwrAn-{4-[(1r,3s,5s)-3-amino-5-methylcyclohexyl]pyridin-3-yl}-6-(2,6-difluorophenyl)-5-fluoropyridine-2-carboxamideHuman6238
PRKAA2 (AMPKa2)CAMKLCAMK6bx6AB2-({5-bromo-2-[(3,4,5-trimethoxyphenyl)amino]pyrimidin-4-yl}oxy)-n-methylbenzene-1-carboximidic acidHuman9877
PIM1PIMCAMK3r04AB5-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}-1-benzofuran-2-carboxylic acidHuman2335
PIM1PIMCAMK3dcvA4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHuman2372
PIM1PIMCAMK3umxAB(2z)-7-(azepan-1-ylmethyl)-6-hydroxy-2-(1h-indol-3-ylmethylidene)-1-benzofuran-3(2h)-oneHuman2375
PIM1PIMCAMK4xh6A5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4h-chromen-4-oneHuman5975
PIM1PIMCAMK8r10AA(z)-4-(4-hydroxystyryl)benzoic acidHuman15214
PIM1PIMCAMK1ywvAB-Human2397
PIM1PIMCAMK8r1nA4-(4-hydroxyphenethyl)benzoic acidHuman15215
PIM1PIMCAMK5n50AA2-(4-chlorophenyl)sulfanylethanehydrazideHuman9585
PIM1PIMCAMK2xiyAB2-hydroxymethyl-benzoimidazoleHuman2363
PIM1PIMCAMK4bznAn-(2,2-dimethylpropyl)-2-[1-oxo-7-(thiophen-3-yl)-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamideHuman2402
PIM1PIMCAMK5n4xAB4,5-bis(bromanyl)thiophene-2-carbohydrazideHuman9593
PIM1PIMCAMK6pdoAA4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamideHuman11461
PIM1PIMCAMK2xj2AB(2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acidHuman2418
PIM1PIMCAMK5n4vAA2-cyclopropyl-4,5-dimethyl-thieno[2,3-d]pyrimidine-6-carboxylic acidHuman9592
PIM1PIMCAMK4enyAB(2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-oneHuman2424
PIM1PIMCAMK2o3pAA3,5,7,3',4'-pentahydroxyflavoneHuman2320
PIM1PIMCAMK7zunA(4~{s})-4-(2-azanylethyl)-6-phenyl-7-[3-(trifluoromethyloxy)phenyl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1-olHuman14383
PIM1PIMCAMK5vubBA(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9073
PIM1PIMCAMK8r0yA3-[(3-hydroxyphenyl)amino]quinoxaline-2-carboxylic acidHuman15477
PIM1PIMCAMK5dhjAB3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridineHuman6211
PIM1PIMCAMK5kcxAB4-chloranyl-1-methyl-2-[4-(4-methylpiperazin-1-yl)phenyl]pyrrolo[2,3-b]pyridine-6-carboxamideHuman8248
PIM1PIMCAMK4n6yA2-(acetylamino)-n-[2-(piperidin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman2383
PIM1PIMCAMK4as0ABphtalimide-ruthenium complexHuman7229
PIM1PIMCAMK7oowA-Human13826
PIM1PIMCAMK5vubBC(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[3,2-b]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9072
PIM1PIMCAMK6pdpAA5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamideHuman11454
PIM1PIMCAMK6pdoAB4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxamideHuman11460
PIM1PIMCAMK5n4oAB(~{e})-3-(4-methylphenyl)prop-2-enoic acidHuman9582
PIM1PIMCAMK4alwAB8-bromanyl-2-[(4-methylpiperazin-1-yl)methyl]-3h-[1]benzofuro[3,2-d]pyrimidin-4-oneHuman2350
PIM1PIMCAMK5c1qB3-methoxy[1]benzothieno[2,3-c]quinolin-6(5h)-oneHuman6288
PIM1PIMCAMK4mblA(1r,2r)-n-[3-(naphthalen-2-yl)pyrazolo[1,5-a]pyrimidin-5-yl]cyclohexane-1,2-diamineHuman2381
PIM1PIMCAMK3r01A5-bromo-7-methoxy-1-benzofuran-2-carboxylic acidHuman2407
PIM1PIMCAMK3cy2AA(4r)-7-chloro-9-methyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman2333
PIM1PIMCAMK5n4xAA4,5-bis(bromanyl)thiophene-2-carbohydrazideHuman9600
PIM1PIMCAMK5kziA~{n}-[4-[(3~{s})-3-azanylpiperidin-1-yl]pyridin-3-yl]-2-[2,6-bis(fluoranyl)phenyl]imidazo[1,5-b]pyridazin-7-amineHuman7195
PIM1PIMCAMK2o63A3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)-4h-chromen-4-oneHuman2453
PIM1PIMCAMK4dtkAB(5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dioneHuman2451
PIM1PIMCAMK3bwfAA-Human7231
PIM1PIMCAMK6l12A4-[(2-chloranylphenoxazin-10-yl)methyl]cyclohexan-1-amineHuman12340
PIM1PIMCAMK5n4nAA3,4-dimethyl-5-(1~{h}-1,2,4-triazol-3-yl)thiophene-2-carbonitrileHuman9579
PIM1PIMCAMK6l17A7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazin-8-amineHuman12740
PIM1PIMCAMK8afrAA4-((6-hydroxybenzofuran-3-yl)methyl)benzoic acidHuman14603
PIM1PIMCAMK5vucBA(2z)-2-(1h-indol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3-oneHuman9071
PIM1PIMCAMK5telAA4-chloro-2-{5,6-dimethoxy-1-[2-(4-methylpiperazin-1-yl)ethyl]-1h-indol-3-yl}-1h-pyrrolo[2,3-b]pyridineHuman8564
PIM1PIMCAMK6kziA4-(2-chloro-10h-phenoxazin-10-yl)-n,n-diethylbutan-1-amineHuman12019
CAMK2G (CaMK2g)CAMK2CAMK2v7oAB-Human7238
CAMK2G (CaMK2g)CAMK2CAMK2v7oAA-Human7239
MKNK2 (MNK2)MAPKAPKCAMK6ck6A6'-[(6-aminopyrimidin-4-yl)amino]-8'-methyl-2'h-spiro[cyclohexane-1,3'-imidazo[1,5-a]pyridine]-1',5'-dioneHuman9880
MKNK2 (MNK2)MAPKAPKCAMK6jlrA4-[5-(1-methylpyrazol-4-yl)pyridin-3-yl]benzamideHuman11968
STK40 (SgK495)SgK495CAMK5l2qBA-Human8011
PRKAA2 (AMPKa2)CAMKLCAMK5isoAstaurosporineHuman7981
PRKAA2 (AMPKa2)CAMKLCAMK6b1uCBstaurosporineHuman9850
PRKAA2 (AMPKa2)CAMKLCAMK5isoCstaurosporineHuman7980
PRKAA2 (AMPKa2)CAMKLCAMK4zhxCB(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6423
RPS6KA3-b (RSK2-b)RSKbCAMK4d9uAtert-butyl (2s)-3-[4-amino-7-(3-hydroxypropyl)-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl]-2-cyanopropanoateHuman1499
RPS6KA3-b (RSK2-b)RSKbCAMK4jg8AB(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman1498
RPS6KA3-b (RSK2-b)RSKbCAMK4jg8AA(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman1497
RPS6KA3-b (RSK2-b)RSKbCAMK4jg7AA(2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamideHuman1496
RPS6KA3-b (RSK2-b)RSKbCAMK4jg7AB(2r)-2-cyano-3-[3-(1h-pyrrolo[2,3-b]pyridin-3-ylcarbonyl)phenyl]propanamideHuman1494
RPS6KA3-b (RSK2-b)RSKbCAMK4jg6A(2s)-2-cyano-3-(1h-indazol-5-yl)propanamideHuman1495
RPS6KA3-b (RSK2-b)RSKbCAMK4d9tAmethyl (2s)-3-{4-amino-7-[(1e)-3-hydroxyprop-1-en-1-yl]-5-(4-methylphenyl)-7h-pyrrolo[2,3-d]pyrimidin-6-yl}-2-cyanopropanoateHuman1493
PIM1PIMCAMK2xj1AB(2e)-3-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}phenyl)prop-2-enoic acidHuman2422
MAPKAPK2MAPKAPKCAMK3gokF2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1362
CAMK2D (CaMK2d)CAMK2CAMK5vloAn-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideHuman8348
MAPKAPK2MAPKAPKCAMK2pzyA(4r)-n-[4-({[2-(dimethylamino)ethyl]amino}carbonyl)-1,3-thiazol-2-yl]-4-methyl-1-oxo-2,3,4,9-tetrahydro-1h-beta-carboline-6-carboxamideHuman1314
PIM1PIMCAMK2bikBB3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2463
PIM1PIMCAMK4wrsA3-{6-[(4r)-6-azaspiro[2.5]oct-4-yloxy]pyrazin-2-yl}-5-(2,6-difluorophenyl)-1h-indazoleHuman2439
PIM1PIMCAMK2xizAB(e)-pyridin-4-yl-acrylic acidHuman2373
PIM1PIMCAMK5n4yAA2,5-dihydro-1~{h}-isothiochromeno[4,3-c]pyrazol-3-oneHuman9589
PIM1PIMCAMK3c4eCn-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amineHuman2440
PIM1PIMCAMK4rpvA(3s)-1-{6-[5-(2,6-difluorophenyl)-2h-indazol-3-yl]pyrazin-2-yl}piperidin-3-amineHuman2364
PIM1PIMCAMK5vuaBB(2z)-6-methoxy-7-(piperazin-1-ylmethyl)-2-(1h-pyrrolo[2,3-c]pyridin-3-ylmethylidene)-1-benzofuran-3-oneHuman9077
PIM1PIMCAMK3vbqAB5-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}benzyl)-2h-1lambda~4~,3-thiazole-2,4(3h)-dioneHuman2454
PIM1PIMCAMK2bilB3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2449
PIM1PIMCAMK3ma3ABnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman2347
PIM1PIMCAMK1yxuDadenosine monophosphateHuman2332
PIM1PIMCAMK5eolA macrocyclic quinoxaline-pyrrolodihydropiperidinoneHuman6601
PIM1PIMCAMK5texA(4-{4-chloro-1-methyl-2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}phenyl)methanolHuman8566
PIM1PIMCAMK4bzoAn-[(1s)-2-amino-1-phenylethyl]-2-[(4s)-7-(2-fluoro-4-pyridinyl)-1-oxo-1,2,3,4-tetrahydropyrrolo[1,2-a]pyrazin-4-yl]acetamideHuman2339
PIM1PIMCAMK6qxkBB2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-oneHuman11036
PIM1PIMCAMK2bziBB-Human7233
PHKG2 (PHKg2)PHKCAMK2y7jBBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1895
PHKG2 (PHKg2)PHKCAMK2y7jABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1893
PHKG2 (PHKg2)PHKCAMK2y7jCBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1900
PHKG2 (PHKg2)PHKCAMK2y7jDBn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1899
CAMK2A (CaMK2a)CAMK2CAMK3soaA4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrileHuman2473
CAMK2A (CaMK2a)CAMK2CAMK6x5gAA-Human13061
CAMK2A (CaMK2a)CAMK2CAMK6w4oO-Human12485
CAMK2A (CaMK2a)CAMK2CAMK7ujtAadenosine-5'-triphosphateHuman14192
CAMK2A (CaMK2a)CAMK2CAMK2vz6AA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2472
CAMK1 (CaMK1a)CAMK1CAMK4fg7Aadenosine-5'-triphosphateHuman4848
SNRKCAMKLCAMK5yksA-Human8660
PIM1PIMCAMK1yxtABphosphoaminophosphonic acid-adenylate esterHuman2319
RPS6KA5-b (MSK1-b)RSKbCAMK7up7AA(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman14318
PIM1PIMCAMK2xj1AA(2e)-3-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}phenyl)prop-2-enoic acidHuman2469
PIM1PIMCAMK3cy3A(2s)-1,3-benzothiazol-2-yl{2-[(2-pyridin-3-ylethyl)amino]pyrimidin-4-yl}ethanenitrileHuman2443
PIM1PIMCAMK6pdnAB4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acidHuman11458
PIM1PIMCAMK4aluAA8-bromo-2-(2-chlorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman2452
PIM1PIMCAMK3vbtA4-chloro-2-(1h-pyrazol-3-yl)phenolHuman2349
PIM1PIMCAMK3qf9AB6-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-n-{3-[(4-ethylpiperazin-1-yl)methyl]-5-(trifluoromethyl)phenyl}naphthalene-1-carboxamideHuman2331
PIM1PIMCAMK3bgpA4-[3-(4-chlorophenyl)-2,1-benzisoxazol-5-yl]pyrimidin-2-amineHuman2359
PIM1PIMCAMK4k18A5-(4-cyanobenzyl)-n-(4-fluorophenyl)-7-hydroxypyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2377
PIM1PIMCAMK6vruAA3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamideHuman13127
PIM1PIMCAMK6qxkBA2-[(1-methylpiperidin-4-yl)methylamino]-5-[[2-[4-(trifluoromethyloxy)phenyl]-1,3-thiazol-4-yl]methyl]-1,3-thiazol-4-oneHuman11035
PIM1PIMCAMK4jx3A-Human2380
PIM1PIMCAMK5ndtAB3-(2-thiophen-2-ylethenyl)-1~{h}-quinoxalin-2-oneHuman9906
PIM1PIMCAMK5n4zAB(~{e})-4-(4-hydroxyphenyl)but-3-en-2-oneHuman9599
PIM1PIMCAMK4xhkBA2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHuman2446
PIM1PIMCAMK5o12A(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman8654
PIM1PIMCAMK3cxwAA(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman2464
CAMK2A (CaMK2a)CAMK2CAMK2vz6BA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2474
PIM1PIMCAMK6no8A5-amino-n-{5-[(4s)-4-aminoazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamideHuman11832
PIM1PIMCAMK1yxxAB(3e)-3-[(4-hydroxyphenyl)imino]-1h-indol-2(3h)-oneHuman2437
PIM1PIMCAMK2oi4XB-Human7226
PIM1PIMCAMK7ooxAB-Human13823
PIM1PIMCAMK1yi3A2-morpholin-4-yl-7-phenyl-4h-chromen-4-oneHuman2398
CAMK2A (CaMK2a)CAMK2CAMK7ujpAadenosine-5'-diphosphateHuman14193
PIM1PIMCAMK5n5mAA~{n}-(isoquinolin-5-ylmethyl)-~{n}-methyl-2-[(3~{r})-pyrrolidin-3-yl]benzamideHuman9702
PIM1PIMCAMK6pdiA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11459
PIM1PIMCAMK1yxuAadenosine monophosphateHuman2438
PIM1PIMCAMK1yxtAAphosphoaminophosphonic acid-adenylate esterHuman2425
PIM1PIMCAMK4wt6A6-[5-(5-amino-1,3,4-thiadiazol-2-yl)-1h-indol-3-yl]-n-cyclopentylpyridin-2-amineHuman2386
PIM1PIMCAMK1ywvAA-Human2430
PIM1PIMCAMK5n4zAA(~{e})-4-(4-hydroxyphenyl)but-3-en-2-oneHuman9587
PIM1PIMCAMK6pcwA4-[5-(cyclopropylcarbamoyl)thiophen-2-yl]-1-benzothiophene-2-carboxamideHuman11455
PIM1PIMCAMK1yxuCadenosine monophosphateHuman2408
PIM1PIMCAMK1yxxAA(3e)-3-[(4-hydroxyphenyl)imino]-1h-indol-2(3h)-oneHuman2351
PIM1PIMCAMK4as0AAphtalimide-ruthenium complexHuman7227
PIM1PIMCAMK6mt0A3-(1-methylcyclopropyl)-2-[(1-methylcyclopropyl)amino]-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-oneHuman10850
PIM1PIMCAMK3jyaAA6,9-dichloro[1]benzothieno[3,2-d]pyrimidin-4(3h)-oneHuman2371
PIM1PIMCAMK4enyAA(2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-methoxybenzylidene)-1,3-thiazolidin-4-oneHuman2342
PIM1PIMCAMK3c4eBn-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amineHuman2423
PIM1PIMCAMK3bgzA2,3-diphenyl-1h-indole-7-carboxylic acidHuman2462
PIM1PIMCAMK4a7cAn-(piperidin-4-ylmethyl)-3-[3-(trifluoromethyloxy)phenyl]-[1,2,3]triazolo[4,5-b]pyridin-5-amineHuman2321
PIM1PIMCAMK5n4rAB2-(azepan-1-yl)-1-(1~{h}-indol-3-yl)propan-1-oneHuman9583
PIM1PIMCAMK4mtaA2-methyl-5-phenylfuran-3-carboxylic acidHuman2370
PIM1PIMCAMK5n4vAB2-cyclopropyl-4,5-dimethyl-thieno[2,3-d]pyrimidine-6-carboxylic acidHuman9594
MKNK2 (MNK2)MAPKAPKCAMK9hrcA1-[5-chloranyl-4-[(3~{r})-pyrrolidin-3-yl]oxy-pyrimidin-2-yl]benzimidazoleHuman15550
MKNK2 (MNK2)MAPKAPKCAMK6cjyA5-[(7h-purin-6-yl)amino]-1h-isoindol-1-oneHuman9881
MKNK2 (MNK2)MAPKAPKCAMK6cj5A3-(pyridin-3-yl)imidazo[1,2-a]pyridine-8-carboxamideHuman9886
MKNK2 (MNK2)MAPKAPKCAMK6ck3A(3r)-3-methyl-5-[(pyrimidin-4-yl)amino]-2,3-dihydro-1h-isoindol-1-oneHuman9883
PIM1PIMCAMK6vruAB3,4-dichloro-2-cyclopropyl-1-[(piperidin-4-yl)methyl]-1h-pyrrolo[2,3-b]pyridine-6-carboxamideHuman13128
PIM1PIMCAMK2bikBA3-{1-[3-(dimethylamino)propyl]-1h-indol-3-yl}-4-(1h-indol-3-yl)-1h-pyrrole-2,5-dioneHuman2341
PIM1PIMCAMK3r02AB7-[(cis-4-aminocyclohexyl)amino]-5-bromo-1-benzofuran-2-carboxylic acidHuman2338
PIM1PIMCAMK3f2aA(2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acidHuman2460
PIM1PIMCAMK7xsvAB8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaeneHuman14288
DCLK1DCAMKLCAMK5jznA5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHuman6986
PIM1PIMCAMK6aydABn-[6-(4-hydroxyphenyl)-2h-indazol-3-yl]cyclopropanecarboxamideHuman9443
DCLK1DCAMKLCAMK5jzjABamp phosphoramidateHuman6987
MARK1CAMKLCAMK6c9dBB-Human10050
MARK1CAMKLCAMK6c9dBA-Human10049
MARK1CAMKLCAMK2hakH-Human261
MARK1CAMKLCAMK6c9dAA-Human10052
PIM1PIMCAMK5n5lAA5-bromanyl-1~{h}-indole-3-carboxylic acidHuman9703
DCLK1DCAMKLCAMK5jznB5-chloro-n-[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]phenyl]-n'-(2-propan-2-ylsulfonylphenyl)pyrimidine-2,4-diamineHuman6982
DCLK1DCAMKLCAMK7f3gA(3r)-3-cyclopentyl-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]propanenitrileHuman13853
PIM1PIMCAMK5kgkA3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amineHuman8307
DCLK1DCAMKLCAMK6kyrAA-Human12803
DCLK1DCAMKLCAMK6kyrBA-Human12805
PIM1PIMCAMK6vrvA4-chloro-1-{(1s)-1-[(3s)-3-fluoropyrrolidin-3-yl]ethyl}-3-methyl-1h-pyrrolo[2,3-b]pyridine-6-carboxamideHuman13129
PIM1PIMCAMK2bzjAAruthenium-pyridocarbazole-3Human7224
PIM1PIMCAMK3r04AA5-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}-1-benzofuran-2-carboxylic acidHuman2353
PIM1PIMCAMK5kcxAA4-chloranyl-1-methyl-2-[4-(4-methylpiperazin-1-yl)phenyl]pyrrolo[2,3-b]pyridine-6-carboxamideHuman8247
PIM1PIMCAMK6ykdAA~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamideHuman12402
PIM1PIMCAMK4alvAA8-bromo-2-{2-chloro-4-[(piperidin-4-ylmethyl)amino]phenyl}[1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman2323
PIM1PIMCAMK7ooxAA-Human13825
PRKAA2 (AMPKa2)CAMKLCAMK4cfeCstaurosporineHuman192
PIM1PIMCAMK2xixAA3,5-diamino-1h-[1,2,4]triazoleHuman2468
PIM1PIMCAMK3ma3AAnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman2368
PIM1PIMCAMK3cy2AB(4r)-7-chloro-9-methyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman2459
PRKAA2 (AMPKa2)CAMKLCAMK4cffAstaurosporineHuman191
DAPK2DAPKCAMK2a27D-Human1118
PIM1PIMCAMK4mbiAn,n-dimethyl-n'-[3-(1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-5-yl]ethane-1,2-diamineHuman2447
PIM1PIMCAMK3uixAA2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHuman2456
PIM1PIMCAMK2bzhBBruthenium-pyridocarbazole-1Human7234
DAPK2DAPKCAMK2ckeBn-(2-aminoethyl)isoquinoline-5-sulfonamideHuman1132
DAPK2DAPKCAMK1wmkH-Human1151
DAPK2DAPKCAMK1zwsE-Human1130
DAPK2DAPKCAMK2a2aDB-Human1149
DAPK2DAPKCAMK1zwsB-Human1128
DAPK2DAPKCAMK2a2aBB-Human1119
DAPK2DAPKCAMK2a27H-Human1137
DAPK2DAPKCAMK1z9xB-Human1136
DAPK2DAPKCAMK2ckeCn-(2-aminoethyl)isoquinoline-5-sulfonamideHuman1135
DAPK2DAPKCAMK2a27G-Human1146
MAPKAPK3MAPKAPKCAMK3sheABn-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamideHuman4599
MAPKAPK3MAPKAPKCAMK3fhrAA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4590
MAPKAPK3MAPKAPKCAMK3r1nAB2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-oneHuman4588
CAMK1D (CaMK1d)CAMK1CAMK8bfmApyrazolo[5,1-a]phthalazin-6-amineHuman14516
PIM1PIMCAMK1yxuBadenosine monophosphateHuman2410
PIM1PIMCAMK6pdpAB5-[2-(acetylamino)-1-benzothiophen-4-yl]-n-cyclopropylthiophene-2-carboxamideHuman11457
PIM1PIMCAMK5dhjAA3-methyl-5-(pyridin-3-yl)-2h-pyrazolo[3,4-c]pyridineHuman6212
PIM1PIMCAMK7qb2A4-[(e)-(6-azanyl-1-methyl-2-oxidanylidene-indol-3-ylidene)methyl]benzoic acidHuman14518
PIM1PIMCAMK3r00A5-bromo-1-benzofuran-2-carboxylic acidHuman2467
CAMK1D (CaMK1d)CAMK1CAMK6qp5AA-Human12028
CAMK2A (CaMK2a)CAMK2CAMK7kl1Aadenosine-5'-triphosphateHuman13059
CAMK2A (CaMK2a)CAMK2CAMK6w4pH-Human12484
CAMK2A (CaMK2a)CAMK2CAMK7kl0Bmethyl 6-o-(heptylcarbamoyl)-beta-l-altropyranosideHuman13114
PIM1PIMCAMK5o11AA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman8656
DCLK1DCAMKLCAMK7kxwA2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman13910
RPS6KA2-b (RSK1-b)RSKbCAMK8wf4A-Human15082
DAPK2DAPKCAMK1wmkF-Human1126
CAMK2A (CaMK2a)CAMK2CAMK6x5qA-Human13056
CAMK2A (CaMK2a)CAMK2CAMK7ujsAadenosine-5'-diphosphateHuman14190
CAMK2A (CaMK2a)CAMK2CAMK6x5gAB-Human13068
CAMK2A (CaMK2a)CAMK2CAMK2vz6BB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2470
TRIB1 (Trb1)TrblCAMK5cemAA-Human6242
TRIB1 (Trb1)TrblCAMK6dc0AB-Human10623
TRIB1 (Trb1)TrblCAMK6dc0AA-Human10622
TRIB1 (Trb1)TrblCAMK6dc0BA-Human10620
TRIB1 (Trb1)TrblCAMK5cemAB-Human6243
TRIB1 (Trb1)TrblCAMK6dc0BB-Human10621
PHKG1 (PHKg1)PHKCAMK8z5qC-Human15641
CAMK1D (CaMK1d)CAMK1CAMK6t6fBA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11941
CAMK1D (CaMK1d)CAMK1CAMK6t29AB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamideHuman13203
CAMK1D (CaMK1d)CAMK1CAMK6t6fAB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11940
CAMK1D (CaMK1d)CAMK1CAMK6t6fBB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11942
CHEK1 (CHK1)CAMKLCAMK4ftqAA5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrileHuman1664
CHEK1 (CHK1)CAMKLCAMK2ym3ABethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1543
CHEK1 (CHK1)CAMKLCAMK3ot3AB5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amineHuman1602
CHEK1 (CHK1)CAMKLCAMK4ftqAB5-{7-ethyl-6-[(3s)-tetrahydrofuran-3-yloxy]-2,4-dihydroindeno[1,2-c]pyrazol-3-yl}pyridine-2-carbonitrileHuman1550
CHEK1 (CHK1)CAMKLCAMK7bk3A4-amino-7-methyl-2-({5-methyl-1-[(3s)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13764
CHEK1 (CHK1)CAMKLCAMK3ot8ABn-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amineHuman1590
CHEK1 (CHK1)CAMKLCAMK2cgvA(2s)-1-amino-3-[(5-nitroquinolin-8-yl)amino]propan-2-olHuman1545
CHEK1 (CHK1)CAMKLCAMK5f4nABmethyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylateHuman6652
CHEK1 (CHK1)CAMKLCAMK4jikA2-(4-chlorophenyl)-8-[(3s)-piperidin-3-ylamino]imidazo[1,2-c]pyrimidine-5-carboxamideHuman1698
CHEK1 (CHK1)CAMKLCAMK4ft9AA1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylureaHuman1564
CHEK1 (CHK1)CAMKLCAMK7akoBAstaurosporineHuman13492
CHEK1 (CHK1)CAMKLCAMK7akmBB-Human13493
CHEK1 (CHK1)CAMKLCAMK2yexAA5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1651
CHEK1 (CHK1)CAMKLCAMK4ft9AB1-(5-cyanopyrazin-2-yl)-3-isoquinolin-3-ylureaHuman1648
CHEK1 (CHK1)CAMKLCAMK4gh2AA3-(3-methoxy-4-nitrophenyl)-6-[2-(morpholin-4-yl)ethoxy]-5,10-dihydro-11h-dibenzo[b,e][1,4]diazepin-11-oneHuman1600
CHEK1 (CHK1)CAMKLCAMK5oq7AB5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8594
CHEK1 (CHK1)CAMKLCAMK2c3lA3-(1h-benzimidazol-2-yl)-1h-indazoleHuman1612
CHEK1 (CHK1)CAMKLCAMK8sivAn-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)cyclopropanecarboxamideHuman14886
CHEK1 (CHK1)CAMKLCAMK4qygB3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acidHuman1607
CHEK1 (CHK1)CAMKLCAMK5op2AB5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8611
CHEK1 (CHK1)CAMKLCAMK4fsyAA2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamideHuman1547
CHEK1 (CHK1)CAMKLCAMK6fc8AA2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamideHuman9500
CHEK1 (CHK1)CAMKLCAMK7bknAadenineHuman13769
CHEK1 (CHK1)CAMKLCAMK3tkiAn-(2-aminoethyl)-5-(2-{[4-(morpholin-4-yl)pyridin-2-yl]amino}-1,3-thiazol-5-yl)pyridine-3-carboxamideHuman1599
CHEK1 (CHK1)CAMKLCAMK2cguA2,2'-{[9-(hydroxyimino)-9h-fluorene-2,7-diyl]bis(oxy)}diacetic acidHuman1697
CHEK1 (CHK1)CAMKLCAMK5oq5A2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman8597
CHEK1 (CHK1)CAMKLCAMK5oq7BB5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8596
CHEK1 (CHK1)CAMKLCAMK7bjmA4-amino-6-{[(2-fluorophenyl)methyl]amino}-7-methyl-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13770
CHEK1 (CHK1)CAMKLCAMK7akmBA-Human13494
CHEK1 (CHK1)CAMKLCAMK7bjhABn,n-dimethyl-7h-purin-6-amineHuman13771
CHEK1 (CHK1)CAMKLCAMK8e80A2-[(1r,4r)-2-{(6p)-6-[(6m)-6-(1h-pyrazol-5-yl)-1h-indazol-1-yl]pyrimidin-4-yl}-2-azabicyclo[2.1.1]hexan-4-yl]propan-2-olHuman14621
CHEK1 (CHK1)CAMKLCAMK2c3jAdebromohymenialdisineHuman1551
CHEK1 (CHK1)CAMKLCAMK4hyiAA2-(1h-indazol-1-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman1538
CHEK1 (CHK1)CAMKLCAMK2yexAB5-methyl-8-(1h-pyrrol-2-yl)[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1567
CHEK1 (CHK1)CAMKLCAMK4rvkAn-[3-(6-cyano-9h-pyrrolo[2,3-b:5,4-c']dipyridin-3-yl)phenyl]acetamideHuman1549
MAPKAPK2MAPKAPKCAMK2jbpH2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1326
CHEK1 (CHK1)CAMKLCAMK4ftjAAtrans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanolHuman1603
CHEK1 (CHK1)CAMKLCAMK4qyhA3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1689
CHEK1 (CHK1)CAMKLCAMK4fsyAB2-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzamideHuman1537
TTNMLCKCAMK1tkiB-Human126
CHEK1 (CHK1)CAMKLCAMK3tkhA1-(morpholin-4-yl)-2-[4-(2-{[5-(pyridin-3-yl)-1,3-thiazol-2-yl]amino}pyridin-4-yl)piperazin-1-yl]ethanoneHuman1665
CHEK1 (CHK1)CAMKLCAMK4rvlA3-(2-hydroxyphenyl)-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1634
PIM1PIMCAMK7vsyA-Human15098
CHEK1 (CHK1)CAMKLCAMK4ftuABmethyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1640
CHEK1 (CHK1)CAMKLCAMK7sufAB8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amineHuman14044
CHEK1 (CHK1)CAMKLCAMK4ftaAA6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acidHuman1540
CHEK1 (CHK1)CAMKLCAMK2x8dAA5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1673
CHEK1 (CHK1)CAMKLCAMK4ftjABtrans-4-({[3-(furan-3-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-yl]methyl}amino)cyclohexanolHuman1613
CHEK1 (CHK1)CAMKLCAMK3pa4AB2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamideHuman1566
CHEK1 (CHK1)CAMKLCAMK2wmsA[4-amino-2-(tert-butylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman1657
CHEK1 (CHK1)CAMKLCAMK4fsrAB6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazoleHuman1575
CHEK1 (CHK1)CAMKLCAMK4ftcAA1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)ureaHuman1593
CHEK1 (CHK1)CAMKLCAMK2e9uA18-chloro-11,12,13,14-tetrahydro-1h,10h-8,4-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecin-2-oneHuman1584
CHEK1 (CHK1)CAMKLCAMK2yerAA5-(hydroxymethyl)-8-(1h-pyrrol-2-yl)-2h-[1,2,4]triazolo[4,3-a]quinolin-1-oneHuman1611
CHEK1 (CHK1)CAMKLCAMK4ft0AB2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acidHuman1693
MAPKAPK2MAPKAPKCAMK6tcaEB-Human12503
MAPKAPK2MAPKAPKCAMK3r2bB2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-oneHuman1329
MAPKAPK2MAPKAPKCAMK3r2yA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1361
MAPKAPK2MAPKAPKCAMK1ny3Aadenosine-5'-diphosphateHuman1318
MAPKAPK2MAPKAPKCAMK1kwpA-Human1280
MAPKAPK2MAPKAPKCAMK3ka0A6-{5-[(2-aminopyrimidin-4-yl)amino]-2-hydroxyphenyl}-n-methylidene-1-benzothiophene-2-carboxamideHuman1290
MAPKAPK2MAPKAPKCAMK2p3gX2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1349
DAPK1DAPKCAMK1wvxA6-(3-aminopropyl)-4,9-dimethylpyrrolo[3,4-c]carbazole-1,3(2h,6h)-dioneHuman5616
MARK2CAMKLCAMK8txyAn-[(5p,8r)-5-(2-cyano-5-{[(3r)-1-methylpyrrolidin-3-yl]methoxy}pyridin-4-yl)pyrazolo[1,5-a]pyridin-2-yl]cyclopropanecarboxamideHuman15136
SIK3 (QSK)CAMKLCAMK8okuA~{n}-ethyl-4-[5-[1-(2-hydroxyethyl)pyrazol-4-yl]benzimidazol-1-yl]-2,6-dimethoxy-benzamideHuman15169
MARK1CAMKLCAMK2hakC-Human260
DAPK2DAPKCAMK1zwsH-Human1133
STK17B (DRAK2)DAPKCAMK7akgAB4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman13004
STK17B (DRAK2)DAPKCAMK6y6hAB2-[6-(1-benzothiophen-2-yl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12044
DAPK2DAPKCAMK1zwsF-Human1114
DAPK2DAPKCAMK2ckeDn-(2-aminoethyl)isoquinoline-5-sulfonamideHuman1141
DAPK3DAPKCAMK1yrpA-Human384
DAPK3DAPKCAMK5a6oBB-Human6166
DAPK3DAPKCAMK5a6nAA5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ideHuman6164
DAPK3DAPKCAMK5vjaCB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10352
DAPK3DAPKCAMK2j90AA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman387
DAPK3DAPKCAMK5a6nBA-Human6162
DAPK3DAPKCAMK5vjaBA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10346
DAPK3DAPKCAMK5vjaAA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10351
DAPK3DAPKCAMK5vjaDB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10347
DAPK3DAPKCAMK3bqrAA4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acidHuman380
DAPK3DAPKCAMK2j90BA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman378
MELKCAMKLCAMK5m5aAAk-252aHuman8735
MELKCAMKLCAMK5maiAA3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman8728
MELKCAMKLCAMK5twyB2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman8669
MELKCAMKLCAMK4d2pDA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2486
MELKCAMKLCAMK6vxrAB(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman12644
MELKCAMKLCAMK5k00AA4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamideHuman7497
MELKCAMKLCAMK4d2wAA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2515
MELKCAMKLCAMK4umpCA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2479
PIM1PIMCAMK5mzlAB~{n}-quinolin-5-ylpyridine-3-carboxamideHuman9563
MELKCAMKLCAMK4d2vDA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2502
MYLK4 (SgK085)MLCKCAMK2x4fBB4-(2-amino-4-methyl-1,3-thiazol-5-yl)-n-(3-dioxaziridin-3-ylphenyl)pyrimidin-2-amineHuman4868
MELKCAMKLCAMK6vxrAA(7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-oneHuman12645
MELKCAMKLCAMK4d2pAA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2513
MELKCAMKLCAMK4d2pCB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2501
MELKCAMKLCAMK4umpDB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2525
MELKCAMKLCAMK5twzA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman8675
MELKCAMKLCAMK5m5aABk-252aHuman8733
MELKCAMKLCAMK4umpBB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2504
MELKCAMKLCAMK5tx3B7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-oneHuman8674
MELKCAMKLCAMK4d2vDB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2506
MELKCAMKLCAMK4d2vAB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2522
MELKCAMKLCAMK4umqAB3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminiumHuman2523
MELKCAMKLCAMK5tvtA9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3-methyl-3,4-dihydropyrimido[5,4-c][1,5]naphthyridin-2(1h)-oneHuman8667
MELKCAMKLCAMK4d2wCB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2503
MELKCAMKLCAMK6gvxAB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11139
MELKCAMKLCAMK5ihaAA1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazineHuman6663
MELKCAMKLCAMK5twlA9-(3,5-dichloro-4-hydroxyphenyl)-1-{trans-4-[(dimethylamino)methyl]cyclohexyl}-3,4-dihydropyrimido[5,4-c]quinolin-2(1h)-oneHuman8668
MELKCAMKLCAMK4d2tAB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2489
MELKCAMKLCAMK5magAApf-3758309Human8736
MELKCAMKLCAMK4bkyAB3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamideHuman2490
MELKCAMKLCAMK4d2vBB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2507
MELKCAMKLCAMK4bkzABn-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamideHuman2484
MELKCAMKLCAMK4umpAA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2497
MELKCAMKLCAMK5mafAmethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman8732
MELKCAMKLCAMK5ihcAA4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridineHuman6660
MELKCAMKLCAMK4ixpA-Human2528
MELKCAMKLCAMK4d2wDB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2495
MELKCAMKLCAMK5ih8An-[(pyridin-2-yl)methyl]-4-[4-(pyridin-4-yl)-1h-pyrazol-1-yl]benzamideHuman6661
DAPK1DAPKCAMK6fhaAB-Human11288
DAPK1DAPKCAMK3dgkAB-Human5629
DAPK1DAPKCAMK2xzsAA-Human5618
MKNK2 (MNK2)MAPKAPKCAMK8p9bA4-[6-(4-morpholin-4-ylcarbonylphenyl)imidazo[1,2-a]pyridin-3-yl]benzenecarbonitrileHuman15296
DAPK1DAPKCAMK3gu8ABn6-cyclopentyladenosineHuman5628
CAMK2A (CaMK2a)CAMK2CAMK2vz6AB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human2471
CHEK1 (CHK1)CAMKLCAMK4ftlAB4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-olHuman1573
CAMK2A (CaMK2a)CAMK2CAMK7ujqAmethyl 6-o-(heptylcarbamoyl)-beta-l-altropyranosideHuman14189
CHEK1 (CHK1)CAMKLCAMK2e9nA3-(4'-hydroxybiphenyl-4-yl)-n-(4-hydroxycyclohexyl)-1,4-dihydroindeno[1,2-c]pyrazole-6-carboxamideHuman1690
PIM1PIMCAMK6l15A7-chloranyl-5-[3-[(3~{s})-piperidin-3-yl]propyl]pyrido[3,4-b][1,4]benzoxazineHuman12339
PIM1PIMCAMK1yxvAB3,4-dihydroxy-1-methylquinolin-2(1h)-oneHuman2366
MKNK2 (MNK2)MAPKAPKCAMK6cjhA3-phenyl-5-(pyridin-4-yl)-1h-indazoleHuman9885
RPS6KA5-b (MSK1-b)RSKbCAMK7up8AA(5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14282
RPS6KA5-b (MSK1-b)RSKbCAMK7up6AB(e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound formHuman14354
MAPKAPK3MAPKAPKCAMK3fxwAA2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4596
MAPKAPK3MAPKAPKCAMK3fxwAB2-[2-(2-fluorophenyl)pyridin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4593
CAMK2D (CaMK2d)CAMK2CAMK6aywBn-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman8665
MAPKAPK2MAPKAPKCAMK2jbpA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1366
MAPKAPK2MAPKAPKCAMK2jbpI2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1364
MAPKAPK2MAPKAPKCAMK3kc3Cn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1303
MAPKAPK2MAPKAPKCAMK1nxkAstaurosporineHuman1342
MAPKAPK2MAPKAPKCAMK2jbpK2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1363
PASKCAMKLCAMK3dlsBadenosine-5'-diphosphateHuman3381
PASKCAMKLCAMK3dlsAadenosine-5'-diphosphateHuman3382
CHEK2 (CHK2)RAD53CAMK2xm8A2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenolHuman4773
CHEK2 (CHK2)RAD53CAMK4bdeA6-methylquinazolin-4-amineHuman4781
CHEK2 (CHK2)RAD53CAMK2ycrAA1,3-bis{4-[(1e)-n-(4,5-dihydro-1h-imidazol-2-yl)ethanehydrazonoyl]phenyl}ureaHuman4760
CHEK2 (CHK2)RAD53CAMK2ycfAA(2e)-n-hydroxy-2-[1-(4-{[(4-{(1e)-1-[2-(n'-hydroxycarbamimidoyl)hydrazinylidene]ethyl}phenyl)carbamoyl]amino}phenyl)ethylidene]hydrazinecarboximidamideHuman4810
CHEK1 (CHK1)CAMKLCAMK3ot8AAn-(3-methylisothiazol-5-yl)-3-(1-methyl-1h-pyrazol-4-yl)-5-[(3r)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidin-7-amineHuman1569
CHEK1 (CHK1)CAMKLCAMK6fcfAB4-[[(2~{r},3~{s})-2-methylpiperidin-3-yl]amino]-2-phenyl-thieno[3,2-c]pyridine-7-carboxamideHuman9498
CASKCASKCAMK3mfrAAphosphoaminophosphonic acid-adenylate esterHuman3822
CASKCASKCAMK3c0gBB[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3826
DCLK1DCAMKLCAMK5jzjAAamp phosphoramidateHuman6984
DCLK1DCAMKLCAMK7kxwB2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5-(2,2,2-trifluoroethyl)-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman13908
DCLK1DCAMKLCAMK7kx8A5-ethyl-2-{[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino}-11-methyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman13909
PRKAA2 (AMPKa2)CAMKLCAMK4zhxAA(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6425
DAPK1DAPKCAMK3dfcBBphosphoaminophosphonic acid-adenylate esterHuman5620
DAPK1DAPKCAMK6qn4A-Human11589
MARK1CAMKLCAMK6c9dAB-Human10051
MARK1CAMKLCAMK2hakE-Human255
MARK1CAMKLCAMK2hakA-Human258
MARK1CAMKLCAMK2hakB-Human259
RPS6KA3-b (RSK2-b)RSKbCAMK8xeyA-Human15207
PIM1PIMCAMK4k0yAAn-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2455
PIM1PIMCAMK4dtkAA(5z)-5-{2-[(3r)-3-aminopiperidin-1-yl]-3-(propan-2-yloxy)benzylidene}-1,3-thiazolidine-2,4-dioneHuman2344
PIM1PIMCAMK5n4uAA5-(2-azanyl-1,3-thiazol-4-yl)-1,3-dihydrobenzimidazol-2-oneHuman9588
PIM1PIMCAMK2bzhBAruthenium-pyridocarbazole-1Human7230
PIM1PIMCAMK3umwAA(2z)-2-(1h-indazol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3(2h)-oneHuman2411
PIM1PIMCAMK5turA1-methyl-2-[4-(piperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridine-4-carbonitrileHuman8565
PIM1PIMCAMK4rc4A1,4-bis[(2-aminoethyl)amino]-5,8-dihydroxyanthracene-9,10-dioneHuman2369
PIM1PIMCAMK4lm5AA2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHuman2400
PIM1PIMCAMK3umxAA(2z)-7-(azepan-1-ylmethyl)-6-hydroxy-2-(1h-indol-3-ylmethylidene)-1-benzofuran-3(2h)-oneHuman2432
PIM1PIMCAMK5o13AB(3~{e})-5-chloranyl-3-[[5-[3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl]furan-2-yl]methylidene]-1~{h}-indol-2-oneHuman8655
PIM1PIMCAMK7z6uAB4-[(~{e})-(6-azanyl-2-oxidanylidene-1~{h}-indol-3-ylidene)methyl]benzoic acidHuman14600
PIM1PIMCAMK8r1kA6-bromanyl-1,3-benzoxazol-2-amineHuman15473
PIM1PIMCAMK1xqzA-Human2361
PIM1PIMCAMK5o13AA(3~{e})-5-chloranyl-3-[[5-[3-[(4-methyl-1,4-diazepan-1-yl)carbonyl]phenyl]furan-2-yl]methylidene]-1~{h}-indol-2-oneHuman8653
PIM1PIMCAMK5kggA2-(5-chloranyl-1~{h}-indol-3-yl)ethanamineHuman8308
PIM1PIMCAMK2objA6-(5-bromo-2-hydroxyphenyl)-2-oxo-4-phenyl-1,2-dihydropyridine-3-carbonitrileHuman2336
PIM1PIMCAMK4wsyA5-[3-(quinolin-3-yl)-2h-indazol-5-yl]-1,3-thiazol-2-amineHuman2429
PIM1PIMCAMK3we8AAcyclopentadienyl(carbon monoxide)(7-oxo-7,10-dihydro-1,8-phenanthrolin-10-yl-kappa~2~c~10~,n~1~)rutheniumHuman7237
PIM1PIMCAMK4alwAA8-bromanyl-2-[(4-methylpiperazin-1-yl)methyl]-3h-[1]benzofuro[3,2-d]pyrimidin-4-oneHuman2419
PIM1PIMCAMK6ykdAB~{n}-[3-[6-[(3~{r})-piperidin-3-yl]-2-pyridin-4-yl-pyrimidin-4-yl]oxyphenyl]ethanamideHuman12401
PIM1PIMCAMK3c4eDn-phenyl-1h-pyrrolo[2,3-b]pyridin-3-amineHuman2378
PIM1PIMCAMK3vc4A(5z)-5-[3-(trifluoromethyl)benzylidene]-1,3-thiazolidine-2,4-dioneHuman2356
PIM1PIMCAMK3uixAB2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHuman2387
PIM1PIMCAMK1yi4AadenosineHuman2403
PIM1PIMCAMK5n4oAA(~{e})-3-(4-methylphenyl)prop-2-enoic acidHuman9580
PIM1PIMCAMK4ll5AA6-(4-fluorophenyl)-5-(pyridin-4-yl)-2,3-dihydroimidazo[2,1-b][1,3]thiazoleHuman2365
PIM1PIMCAMK4ty1An-tert-butyl-5-[3-(4-cyclopropylpyrimidin-2-yl)-1h-indol-5-yl]-1,3,4-oxadiazol-2-amineHuman2394
PIM1PIMCAMK6l11A5-(2-chloranylphenoxazin-10-yl)-~{n},~{n}-diethyl-pentan-1-amineHuman12336
PIM1PIMCAMK6no9A5-amino-n-{5-[(4r,5r)-4-amino-5-fluoroazepan-1-yl]-1-methyl-1h-pyrazol-4-yl}-2-(2,6-difluorophenyl)-1,3-thiazole-4-carboxamideHuman10936
PIM1PIMCAMK5ipjA2-(tert-butylamino)-3-methyl-8-[(6r)-6-methyl-4-oxo-1,4,5,6-tetrahydropyrrolo[3,4-b]pyrrol-2-yl]quinazolin-4(3h)-oneHuman6703
PIM1PIMCAMK4k1bAn-[5-(2-fluorophenyl)-1h-pyrrolo[2,3-b]pyridin-3-yl]-5-({[(3r,4r)-3-fluoropiperidin-4-yl]methyl}amino)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2362
PIM1PIMCAMK5n5mAB~{n}-(isoquinolin-5-ylmethyl)-~{n}-methyl-2-[(3~{r})-pyrrolidin-3-yl]benzamideHuman9705
PIM1PIMCAMK1yhsAstaurosporineHuman2444
PIM1PIMCAMK3jpvA1,10-dihydropyrrolo[2,3-a]carbazole-3-carbaldehydeHuman2431
PIM1PIMCAMK3vbqAA5-(3-{6-[(trans-4-aminocyclohexyl)amino]pyrazin-2-yl}benzyl)-2h-1lambda~4~,3-thiazole-2,4(3h)-dioneHuman2354
PIM1PIMCAMK3umwAB(2z)-2-(1h-indazol-3-ylmethylidene)-6-methoxy-7-(piperazin-1-ylmethyl)-1-benzofuran-3(2h)-oneHuman2414
PIM1PIMCAMK4xhkBB2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHuman2355
PIM1PIMCAMK5n52AB(~{e})-3-(2,3-dimethoxyphenyl)prop-2-enoic acidHuman9586
PIM1PIMCAMK2bzkBphosphoaminophosphonic acid-adenylate esterHuman2330
PIM1PIMCAMK7xsvAA8-methyl-2,5,20-trioxa-8,13,17-triazatetracyclo[11.10.2.014,19.021,25]pentacosa-1(24),14(19),15,17,21(25),22-hexaeneHuman14287
PIM1PIMCAMK6pdnAA4-{5-[(3-aminopropyl)carbamoyl]thiophen-2-yl}-1-benzothiophene-2-carboxylic acidHuman11456
PIM1PIMCAMK1yxsAA-Human2417
PIM1PIMCAMK1yxsAB-Human2461
PIM1PIMCAMK2c3iBB1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman2374
PIM1PIMCAMK5diaA(1s,3s)-n-{6-[5-(pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridin-3-yl]pyridin-2-yl}cyclohexane-1,3-diamineHuman6210
PIM1PIMCAMK2xizAA(e)-pyridin-4-yl-acrylic acidHuman2436
PIM1PIMCAMK3jy0AA8-chloro-2-{[(3s)-3-hydroxypyrrolidin-1-yl]methyl}[1]benzothieno[3,2-d]pyrimidin-4(3h)-oneHuman2405
PIM1PIMCAMK4iaaA10-{2-[(2r)-1-methylpiperidin-2-yl]ethyl}-2-(methylsulfanyl)-10h-phenothiazineHuman2325
PIM1PIMCAMK4k0yABn-(4-fluorophenyl)-7-hydroxy-5-(piperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamideHuman2445
PIM1PIMCAMK5mzlAA~{n}-quinolin-5-ylpyridine-3-carboxamideHuman9562
PIM1PIMCAMK6l13A2-chloranyl-10-(2-piperidin-4-ylethyl)phenoxazineHuman12337
PIM1PIMCAMK8r1tAA4-(4-aminophenethyl)benzoic acidHuman15212
PIM1PIMCAMK3vbxAA6-bromo-4-hydroxy-2h-chromen-2-oneHuman2427
PIM1PIMCAMK2xj2AA(2e)-3-{3-[6-(4-methyl-1,4-diazepan-1-yl)pyrazin-2-yl]phenyl}prop-2-enoic acidHuman2334
PIM1PIMCAMK3bgqAn-cyclohexyl-3-[3-(trifluoromethyl)phenyl][1,2,4]triazolo[4,3-b]pyridazin-6-amineHuman2465
PIM1PIMCAMK4aluAB8-bromo-2-(2-chlorophenyl)[1]benzofuro[3,2-d]pyrimidin-4(3h)-oneHuman2384
PIM1PIMCAMK5kgdA2-pyridin-3-yl-1~{h}-benzimidazoleHuman8309
PIM1PIMCAMK8r18AA(e)-4-(4-hydroxystyryl)benzoic acidHuman15213
PIM1PIMCAMK2bziBA-Human7225
PIM1PIMCAMK8r1wA4-(5-(4-aminophenyl)-2h-1,2,3-triazol-4-yl)benzoic acidHuman15476
PIM1PIMCAMK4lm5AB2-{4-[(3-aminopropyl)amino]quinazolin-2-yl}phenolHuman2327
PIM1PIMCAMK3t9iA2-methoxy-4-(3-phenyl-2h-pyrazolo[3,4-b]pyridin-6-yl)phenolHuman2450
PIM1PIMCAMK2xiyAA2-hydroxymethyl-benzoimidazoleHuman2415
PIM1PIMCAMK5n51AA3,4-bis(bromanyl)thiophene-2-carboxylic acidHuman9596
PIM1PIMCAMK4enxA(2z,5z)-2-[(2-chlorophenyl)imino]-5-(4-hydroxy-3-nitrobenzylidene)-1,3-thiazolidin-4-oneHuman2352
PIM2PIMCAMK2iwiAruthenium-pyridocarbazole-1Human7217
PIM2PIMCAMK4x7qB2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHuman1416
PIM2PIMCAMK4x7qA2-(2,6-difluorophenyl)-n-{4-[(3s)-pyrrolidin-3-yloxy]pyridin-3-yl}-1,3-thiazole-4-carboxamideHuman1415
PHKG2 (PHKg2)PHKCAMK2y7jDAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1898
CAMK2A (CaMK2a)CAMK2CAMK7uiqA-Human14175
CAMK1 (CaMK1a)CAMK1CAMK4fg9Aadenosine-5'-triphosphateHuman4846
CAMK1 (CaMK1a)CAMK1CAMK4fg9Badenosine-5'-triphosphateHuman4845
CAMK1 (CaMK1a)CAMK1CAMK4fgbA-Human4847
CAMK1 (CaMK1a)CAMK1CAMK4fg8Badenosine-5'-triphosphateHuman4849
CAMK1 (CaMK1a)CAMK1CAMK4fg8Aadenosine-5'-triphosphateHuman4850
MKNK2 (MNK2)MAPKAPKCAMK2hw7AstaurosporineHuman764
MKNK2 (MNK2)MAPKAPKCAMK6cjwA3-(pyridin-4-yl)imidazo[1,2-b]pyridazineHuman9879
MKNK2 (MNK2)MAPKAPKCAMK2ac5AA-Human763
MKNK2 (MNK2)MAPKAPKCAMK6ckiA3,3-dimethyl-6-[(pyrimidin-4-yl)amino]-2,3-dihydroimidazo[1,5-a]pyridine-1,5-dioneHuman9882
MKNK2 (MNK2)MAPKAPKCAMK6cjeA4-[(9h-purin-6-yl)amino]benzamideHuman9884
MKNK2 (MNK2)MAPKAPKCAMK2ac3A-Human765
MARK4CAMKLCAMK5es1A~{n}-[(1~{r},6~{r})-6-azanyl-2,2-bis(fluoranyl)cyclohexyl]-5-ethyl-4-[6-(trifluoromethyl)pyrazolo[1,5-a]pyrimidin-3-yl]thiophene-2-carboxamideHuman6260
MARK4CAMKLCAMK8xflA-Human15101
DAPK2DAPKCAMK2a2aBA-Human1115
DAPK2DAPKCAMK2a27F-Human1127
DAPK2DAPKCAMK1z9xA-Human1144
DAPK2DAPKCAMK2a27A-Human1113
DAPK2DAPKCAMK1zwsG-Human1150
DAPK2DAPKCAMK2a2aCB-Human1148
DAPK2DAPKCAMK1wmkE-Human1117
DAPK2DAPKCAMK6pawE-Human12439
DAPK2DAPKCAMK1zwsD-Human1131
DAPK2DAPKCAMK1zwsA-Human1121
DAPK2DAPKCAMK2a2aDA-Human1120
DAPK2DAPKCAMK1wmkD-Human1139
DAPK2DAPKCAMK1zwsC-Human1134
DAPK2DAPKCAMK2a2aAB-Human1123
DAPK2DAPKCAMK2ckeAn-(2-aminoethyl)isoquinoline-5-sulfonamideHuman1143
DAPK2DAPKCAMK2a27C-Human1125
DAPK2DAPKCAMK1z9xC-Human1116
DAPK2DAPKCAMK1wmkA-Human1124
DAPK2DAPKCAMK2a2aAA-Human1145
DAPK2DAPKCAMK2a27E-Human1147
DAPK2DAPKCAMK6pawB-Human12440
DAPK2DAPKCAMK1wmkC-Human1138
DAPK2DAPKCAMK2a2aCA-Human1122
DAPK2DAPKCAMK2a27B-Human1129
DAPK2DAPKCAMK6pawF-Human12441
DAPK2DAPKCAMK6pawA-Human12442
DAPK2DAPKCAMK1wmkB-Human1140
CAMK1G (CaMK1g)CAMK1CAMK2jamAB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1221
CAMK1G (CaMK1g)CAMK1CAMK2jamAA5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1218
CAMK1G (CaMK1g)CAMK1CAMK2jamBA5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1220
CAMK1G (CaMK1g)CAMK1CAMK2jamBB5-[(e)-(5-chloro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-n-[2-(diethylamino)ethyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman1219
PHKG1 (PHKg1)PHKCAMK8xybC-Human15264
PHKG1 (PHKg1)PHKCAMK8z5tCBadenosine-5'-triphosphateHuman15640
PHKG1 (PHKg1)PHKCAMK8jflB-Human15265
CAMK1D (CaMK1d)CAMK1CAMK6t28AA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamideHuman13202
CAMK1D (CaMK1d)CAMK1CAMK2jc6CAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4832
CAMK1D (CaMK1d)CAMK1CAMK2jc6CBn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4831
CAMK1D (CaMK1d)CAMK1CAMK6t6fAA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3-(trifluoromethyl)phenyl]amino]pyrimidine-5-carboxamideHuman11939
CAMK1D (CaMK1d)CAMK1CAMK2jc6ABn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4830
CAMK1D (CaMK1d)CAMK1CAMK8bfsAB3~{h}-pyrrolo[2,3-c]isoquinolin-5-amineHuman14505
CAMK1D (CaMK1d)CAMK1CAMK6t29AA2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[3,5-bis(2-cyanopropan-2-yl)phenyl]amino]pyrimidine-5-carboxamideHuman13204
CAMK1D (CaMK1d)CAMK1CAMK2jc6AAn-(5-methyl-1h-pyrazol-3-yl)-2-phenylquinazolin-4-amineHuman4829
CAMK1D (CaMK1d)CAMK1CAMK6qp5AB-Human12029
CAMK1D (CaMK1d)CAMK1CAMK6t28AB2-[(3~{s})-3-azanylpiperidin-1-yl]-4-[[2,6-di(propan-2-yl)pyridin-4-yl]amino]pyrimidine-5-carboxamideHuman13205
CHEK1 (CHK1)CAMKLCAMK3ot3AA5-[(1r,3s)-3-aminocyclohexyl]-6-bromo-3-(1-methyl-1h-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-7-amineHuman1696
CHEK1 (CHK1)CAMKLCAMK5opuA6-azanyl-4-(3-methylphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrileHuman8615
CHEK1 (CHK1)CAMKLCAMK2ym3AAethyl 4-(2-(aminomethyl)morpholino)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1644
CHEK1 (CHK1)CAMKLCAMK8siwA(1s,2s)-n-(7-chloro-6-{1-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperidin-4-yl}isoquinolin-3-yl)-2-(1-methyl-1h-pyrazol-4-yl)cyclopropane-1-carboxamideHuman14885
CHEK1 (CHK1)CAMKLCAMK5dlsA1-benzyl-n-(5-{5-[3-(dimethylamino)-2,2-dimethylpropoxy]-1h-indol-2-yl}-6-oxo-1,6-dihydropyridin-3-yl)-1h-pyrazole-4-carboxamideHuman6151
CHEK1 (CHK1)CAMKLCAMK1zysAn-{5-[4-(4-methylpiperazin-1-yl)phenyl]-1h-pyrrolo[2,3-b]pyridin-3-yl}nicotinamideHuman1655
CHEK1 (CHK1)CAMKLCAMK4fttABmethyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1670
CHEK1 (CHK1)CAMKLCAMK2wmtAB2-(methylsulfanyl)-5-(thiophen-2-ylmethyl)-1h-imidazol-4-olHuman1685
CHEK1 (CHK1)CAMKLCAMK3pa4AA2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[3,2-c]pyridine-7-carboxamideHuman1592
CHEK1 (CHK1)CAMKLCAMK2ydiAA5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamideHuman1684
CHEK1 (CHK1)CAMKLCAMK6fckAA2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamideHuman9501
CHEK1 (CHK1)CAMKLCAMK1nvsArel-(9r,12s)-9,10,11,12-tetrahydro-9,12-epoxy-1h-diindolo[1,2,3-fg:3',2',1'-kl]pyrrolo[3,4-i][1,6]benzodiazocine-1,3(2h)-dioneHuman1591
CHEK1 (CHK1)CAMKLCAMK4rvmA3-[4-(piperidin-1-ylmethyl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1624
CHEK1 (CHK1)CAMKLCAMK4ft0AA2-methoxy-4-(11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-3-yl)benzoic acidHuman1637
CHEK1 (CHK1)CAMKLCAMK2e9vB18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrileHuman1638
CHEK1 (CHK1)CAMKLCAMK2ghgA5-{5-[(s)-2-amino-3-(1h-indol-3-yl)-propoxyl]-pyridin-3-yl}-3-[1-(1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman1581
CHEK1 (CHK1)CAMKLCAMK2e9pA1-(5-chloro-2-methoxyphenyl)-3-{6-[2-(dimethylamino)-1-methylethoxy]pyrazin-2-yl}ureaHuman1618
CHEK1 (CHK1)CAMKLCAMK4hyhAB2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamideHuman1626
CHEK1 (CHK1)CAMKLCAMK4fttAAmethyl [3-(1-methyl-1h-imidazol-5-yl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1565
CHEK1 (CHK1)CAMKLCAMK4ftoAB4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrileHuman1605
CHEK1 (CHK1)CAMKLCAMK4fstAA4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenolHuman1619
CHEK1 (CHK1)CAMKLCAMK7bkoA1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman13765
CHEK1 (CHK1)CAMKLCAMK4ftkAB3-(4'-hydroxybiphenyl-4-yl)-2,4-dihydroindeno[1,2-c]pyrazol-6-olHuman1536
CHEK1 (CHK1)CAMKLCAMK5op7A[4-[[5-chloranyl-4-(methylamino)-7~{h}-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-phenyl]-morpholin-4-yl-methanoneHuman8609
CHEK1 (CHK1)CAMKLCAMK4fszAA(3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acidHuman1553
CHEK1 (CHK1)CAMKLCAMK2c3kA4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-2-methoxyphenolHuman1674
CHEK1 (CHK1)CAMKLCAMK4ftmAB4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenolHuman1556
CHEK1 (CHK1)CAMKLCAMK4ftcAB1-(5-cyanopyrazin-2-yl)-3-(5-phenyl-1h-pyrazol-3-yl)ureaHuman1680
CHEK1 (CHK1)CAMKLCAMK7akmAAphosphothiophosphoric acid-adenylate esterHuman13489
CHEK1 (CHK1)CAMKLCAMK2e9vA18-chloro-2-oxo-17-[(pyridin-4-ylmethyl)amino]-2,3,11,12,13,14-hexahydro-1h,10h-4,8-(azeno)-9,15,1,3,6-benzodioxatriazacycloheptadecine-7-carbonitrileHuman1574
CHEK1 (CHK1)CAMKLCAMK2hxqA3-(5-{[4-(aminomethyl)piperidin-1-yl]methyl}-1h-indol-2-yl)quinolin-2(1h)-oneHuman1587
CHEK1 (CHK1)CAMKLCAMK1nvrAstaurosporineHuman1585
CHEK1 (CHK1)CAMKLCAMK2wmuAA6-morpholin-4-yl-9h-purineHuman1662
CHEK1 (CHK1)CAMKLCAMK4ftnAB4'-{6-methoxy-7-[2-(piperidin-1-yl)ethoxy]-1,2-dihydroindeno[1,2-c]pyrazol-3-yl}biphenyl-4-olHuman1678
CHEK1 (CHK1)CAMKLCAMK4fsuAA4-[6-(1h-imidazol-1-ylmethyl)-7-methoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]benzonitrileHuman1539
CHEK1 (CHK1)CAMKLCAMK2gdoA4-[(3s)-1-azabicyclo[2.2.2]oct-3-ylamino]-3-(1h-benzimidazol-2-yl)-6-chloroquinolin-2(1h)-oneHuman1606
CHEK1 (CHK1)CAMKLCAMK2broA(2r)-3-{[(4z)-5,6-diphenyl-6,7-dihydro-4h-pyrrolo[2,3-d]pyrimidin-4-ylidene]amino}propane-1,2-diolHuman1686
CHEK1 (CHK1)CAMKLCAMK2ydjA5-(3-fluorophenyl)-n-[(3s)-3-piperidyl]-3-ureido-thiophene-2-carboxamideHuman1649
CHEK1 (CHK1)CAMKLCAMK2ym4AAethyl 4-[(2r)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1h-pyrazolo[3,4-b]pyridine-5-carboxylateHuman1572
CHEK1 (CHK1)CAMKLCAMK2ym8A(r)-5-(8-chloroisoquinolin-3-ylamino)-3-(1-(dimethylamino)propan-2-yloxy)pyrazine-2-carbonitrileHuman1588
CHEK1 (CHK1)CAMKLCAMK7bk2A4-amino-7-methyl-2-({5-methyl-1-[(3r)-oxolan-3-yl]-1h-pyrazol-4-yl}amino)-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13766
CHEK1 (CHK1)CAMKLCAMK3nlbA3-methyl-5-[5-(1-methylethyl)-1h-benzimidazol-2-yl]-n-(1-methylpiperidin-4-yl)-1h-pyrazole-4-carboxamideHuman1641
CHEK1 (CHK1)CAMKLCAMK4qyeA4-[6-(3-hydroxyphenyl)pyrazin-2-yl]benzoic acidHuman1601
CHEK1 (CHK1)CAMKLCAMK7bjeAAadenineHuman13767
CHEK1 (CHK1)CAMKLCAMK4qyhB3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carbonitrileHuman1586
CHEK1 (CHK1)CAMKLCAMK2ym5A(3-{4-[(2s)-2-(aminomethyl)morpholin-4-yl]-7h-pyrrolo[2,3-d]pyrimidin-5-yl}phenyl)methanolHuman1627
CHEK1 (CHK1)CAMKLCAMK8e81A(1s)-1-[(1p)-1-{6-[(3r)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]pyrimidin-4-yl}-1h-indazol-6-yl]spiro[2.2]pentane-1-carbonitrileHuman14620
CHEK1 (CHK1)CAMKLCAMK2wmxA1-[(2s)-4-(5-phenyl-1h-pyrazolo[3,4-b]pyridin-4-yl)morpholin-2-yl]methanamineHuman1636
CHEK1 (CHK1)CAMKLCAMK7akoAAstaurosporineHuman13490
CHEK1 (CHK1)CAMKLCAMK2brbA2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanolHuman1582
CHEK1 (CHK1)CAMKLCAMK4ftaAB6-{[(5-cyanopyrazin-2-yl)carbamoyl]amino}naphthalene-2-carboxylic acidHuman1660
CHEK1 (CHK1)CAMKLCAMK4qygA3-[4-(4-methylpiperazin-1-yl)phenyl]-9h-pyrrolo[2,3-b:5,4-c']dipyridine-6-carboxylic acidHuman1568
CHEK1 (CHK1)CAMKLCAMK7akmABphosphothiophosphoric acid-adenylate esterHuman13491
CHEK1 (CHK1)CAMKLCAMK7sugAA1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrileHuman14039
CHEK1 (CHK1)CAMKLCAMK2br1AA2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanolHuman1677
CHEK1 (CHK1)CAMKLCAMK7bjeABadenineHuman13773
CHEK1 (CHK1)CAMKLCAMK3pa3AA2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamideHuman1691
CHEK1 (CHK1)CAMKLCAMK2brmAB3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-oneHuman1643
CHEK1 (CHK1)CAMKLCAMK4ft5AA1-{5-chloro-2-[(3r)-pyrrolidin-3-yloxy]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1617
CHEK1 (CHK1)CAMKLCAMK2ydiAB5-[4-(2-dimethylaminoethyloxy)phenyl]-2-ureido-thiophene-3-carboxamideHuman1579
CHEK1 (CHK1)CAMKLCAMK8sixA(1s)-n-(7-chloro-6-{4-[(3r,4r)-4-hydroxy-3-methyloxolan-3-yl]piperazin-1-yl}isoquinolin-3-yl)-6-oxaspiro[2.5]octane-1-carboxamideHuman14887
CHEK1 (CHK1)CAMKLCAMK4fsqAA4'-(6,7-dimethoxyindeno[1,2-c]pyrazol-3-yl)biphenyl-4-olHuman1688
CHEK1 (CHK1)CAMKLCAMK2ym7AB5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrileHuman1645
CHEK1 (CHK1)CAMKLCAMK2x8iAA7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1699
CHEK1 (CHK1)CAMKLCAMK5f4nAAmethyl 6-[(5-cyanopyrazin-2-yl)amino]-4-[[(2~{r})-morpholin-2-yl]methylamino]pyridine-3-carboxylateHuman6651
CHEK1 (CHK1)CAMKLCAMK5op5A3-[4-(morpholin-4-yl)-7h-pyrrolo[2,3-d]pyrimidin-5-yl]benzonitrileHuman8600
CHEK1 (CHK1)CAMKLCAMK2ym7AA5-({6-[(piperidin-4-ylmethyl)amino]pyrimidin-4-yl}amino)pyrazine-2-carbonitrileHuman1650
CHEK1 (CHK1)CAMKLCAMK4ftlAA4'-[7-(hydroxymethyl)-2,4-dihydroindeno[1,2-c]pyrazol-3-yl]biphenyl-4-olHuman1614
CHEK1 (CHK1)CAMKLCAMK4fsrAA6,7-dimethoxy-3-[4-(1h-tetrazol-5-yl)phenyl]-1,4-dihydroindeno[1,2-c]pyrazoleHuman1629
CHEK1 (CHK1)CAMKLCAMK4ftmAC4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenolHuman1616
CHEK1 (CHK1)CAMKLCAMK2brmAA3-amino-3-benzyl-[4.3.0]bicyclo-1,6-diazanonan-2-oneHuman1621
CHEK1 (CHK1)CAMKLCAMK4ftmAA4-[2-(2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethyl]-2-methoxyphenolHuman1546
CHEK1 (CHK1)CAMKLCAMK2e9oA4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHuman1667
CHEK1 (CHK1)CAMKLCAMK5opsA4-(3-hydroxyphenyl)-1~{h}-pyrrolo[2,3-b]pyridine-3-carbonitrileHuman8598
CHEK1 (CHK1)CAMKLCAMK4fsnAA4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHuman1542
CHEK1 (CHK1)CAMKLCAMK2r0uA6-(3-aminopropyl)-4-(3-hydroxyphenyl)-9-(1h-pyrazol-4-yl)benzo[h]isoquinolin-1(2h)-oneHuman1632
CHEK1 (CHK1)CAMKLCAMK2xf0A3-phenyl-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazineHuman1534
CHEK1 (CHK1)CAMKLCAMK7bjhAAn,n-dimethyl-7h-purin-6-amineHuman13776
CHEK1 (CHK1)CAMKLCAMK4ftiAAmethyl 5-(6-{[(cis-4-hydroxycyclohexyl)amino]methyl}-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)furan-2-carboxylateHuman1577
CHEK1 (CHK1)CAMKLCAMK7sufAA8-cyclopropyl-n-[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]quinazolin-2-amineHuman14040
CHEK1 (CHK1)CAMKLCAMK5oorAstaurosporineHuman8603
CHEK1 (CHK1)CAMKLCAMK4ftrAA2-[3-(3-methoxy-4-nitrophenyl)-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]-n,n-dimethylacetamideHuman1692
CHEK1 (CHK1)CAMKLCAMK4ft7AB1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1557
CHEK1 (CHK1)CAMKLCAMK2hy0A3-[5-(piperidin-1-ylmethyl)-1h-indol-2-yl]-6-(1h-pyrazol-4-yl)quinolin-2(1h)-oneHuman1555
CHEK1 (CHK1)CAMKLCAMK6fckAB2-phenyl-4-[[(3~{s})-piperidin-3-yl]amino]-1~{h}-indole-7-carboxamideHuman9499
CHEK1 (CHK1)CAMKLCAMK2qhnA5-ethyl-3-methyl-1,5-dihydro-4h-pyrazolo[4,3-c]quinolin-4-oneHuman1675
CHEK1 (CHK1)CAMKLCAMK5oq8A5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8606
CHEK1 (CHK1)CAMKLCAMK6fc8AB2-(3-fluorophenyl)-4-[[(3~{s})-piperidin-3-yl]amino]thieno[3,2-c]pyridine-7-carboxamideHuman9502
CHEK1 (CHK1)CAMKLCAMK2xezA6-(1h-pyrazol-3-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazineHuman1580
CHEK1 (CHK1)CAMKLCAMK2x8eA5-methyl-8-pyridin-4-yl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1548
CHEK1 (CHK1)CAMKLCAMK5oq7BA5-(4-methylpiperazin-1-yl)-2-phenylmethoxy-~{n}-pyridin-3-yl-benzamideHuman8605
CHEK1 (CHK1)CAMKLCAMK3pa5AB2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamideHuman1544
CHEK1 (CHK1)CAMKLCAMK7bjjAA1h-pyrazolo[3,4-d]pyrimidin-4-amineHuman13777
CHEK1 (CHK1)CAMKLCAMK7sujA(3r,4r)-4-{4-[6-chloro-2-({1-[(1r)-2,2-difluorocyclopropyl]-5-methyl-1h-pyrazol-4-yl}amino)quinazolin-7-yl]piperidin-1-yl}-4-methyloxolan-3-olHuman14041
CHEK1 (CHK1)CAMKLCAMK3jvsA-Human1630
CHEK1 (CHK1)CAMKLCAMK4ft3AB1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylureaHuman1672
CHEK1 (CHK1)CAMKLCAMK2brhAAn-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycineHuman1694
CHEK1 (CHK1)CAMKLCAMK7sugAB1-(2-{[5-methyl-1-(oxan-4-yl)-1h-pyrazol-4-yl]amino}quinazolin-8-yl)cyclopropane-1-carbonitrileHuman14042
CHEK1 (CHK1)CAMKLCAMK7suhA1-[5-chloro-4-({6-chloro-7-[1-(oxetan-3-yl)piperidin-4-yl]quinazolin-2-yl}amino)-1h-pyrazol-1-yl]-2-methylpropan-2-olHuman14043
CHEK1 (CHK1)CAMKLCAMK4ft3AA1-(5-chloro-2,4-dimethoxyphenyl)-3-pyrazin-2-ylureaHuman1554
CHEK1 (CHK1)CAMKLCAMK3jvrA-Human1625
CHEK1 (CHK1)CAMKLCAMK3pa3AB2-(4-chlorophenyl)-4-[(3s)-piperidin-3-ylamino]thieno[2,3-d]pyridazine-7-carboxamideHuman1635
CHEK1 (CHK1)CAMKLCAMK4fstAB4-[(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)ethynyl]-2-methoxyphenolHuman1663
CHEK1 (CHK1)CAMKLCAMK2aypA(3z)-6-(4-hydroxy-3-methoxyphenyl)-3-(1h-pyrrol-2-ylmethylene)-1,3-dihydro-2h-indol-2-oneHuman1682
CHEK1 (CHK1)CAMKLCAMK2wmuAB6-morpholin-4-yl-9h-purineHuman1578
CHEK1 (CHK1)CAMKLCAMK2x8dAB5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1620
CHEK1 (CHK1)CAMKLCAMK4ftoAA4-{7-methoxy-6-[3-(morpholin-4-yl)propoxy]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl}benzonitrileHuman1661
CHEK1 (CHK1)CAMKLCAMK5ootA2-[(2-methoxy-4-{[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl}phenyl)amino]-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman8599
CHEK1 (CHK1)CAMKLCAMK1ia8A-Human1656
CHEK1 (CHK1)CAMKLCAMK4fsmAB4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenolHuman1671
CHEK1 (CHK1)CAMKLCAMK3f9nAA-Human1700
CHEK1 (CHK1)CAMKLCAMK4fsnAB4-(6-{[(4-methylcyclohexyl)amino]methyl}-1,4-dihydroindeno[1,2-c]pyrazol-3-yl)benzoic acidHuman1679
CHEK1 (CHK1)CAMKLCAMK4fsmAA4-(6,7-dimethoxy-2,4-dihydroindeno[1,2-c]pyrazol-3-yl)phenolHuman1570
CHEK1 (CHK1)CAMKLCAMK2qhmA(3-endo)-8-methyl-8-azabicyclo[3.2.1]oct-3-yl 1h-pyrrolo[2,3-b]pyridine-3-carboxylateHuman1669
CHEK1 (CHK1)CAMKLCAMK7bjrA4-amino-7-methyl-6-[(2r)-2-methylpyrrolidin-1-yl]-7h-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13778
CHEK1 (CHK1)CAMKLCAMK4fszAB(3-chloro-11-oxo-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl)acetic acidHuman1628
CHEK1 (CHK1)CAMKLCAMK7mckAn-{5-[(3s)-3-(2-hydroxypropan-2-yl)pyrrolidin-1-yl]-2-(trifluoromethyl)pyridin-3-yl}-6-(1-methyl-1h-pyrazol-4-yl)pyridine-2-carboxamideHuman13622
CHEK1 (CHK1)CAMKLCAMK5oopAAphosphoaminophosphonic acid-adenylate esterHuman8612
CHEK1 (CHK1)CAMKLCAMK4ftuAAmethyl [11-oxo-3-(pyridin-4-ylamino)-10,11-dihydro-5h-dibenzo[b,e][1,4]diazepin-8-yl]acetateHuman1639
CHEK1 (CHK1)CAMKLCAMK4hyhAA2-(6-methoxy-1-oxo-1,3-dihydro-2h-isoindol-2-yl)-n-[4-(piperazin-1-yl)pyridin-3-yl]-1,3-thiazole-4-carboxamideHuman1561
CHEK1 (CHK1)CAMKLCAMK4ft7AA1-{5-bromo-2-[(3r)-3-hydroxypiperidin-1-yl]phenyl}-3-(5-cyanopyrazin-2-yl)ureaHuman1610
CHEK1 (CHK1)CAMKLCAMK2brhABn-(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)glycineHuman1654
CHEK1 (CHK1)CAMKLCAMK2cgwA4,4'-(1-propyl-1h-1,2,4-triazole-3,5-diyl)bis(2,5-dihydro-1,2,5-oxadiazol-3-amine)Human1683
CHEK1 (CHK1)CAMKLCAMK2br1AB2-[5,6-bis-(4-methoxy-phenyl)-furo[2,3-d]pyrimidin-4-ylamino]-ethanolHuman1571
CHEK1 (CHK1)CAMKLCAMK2x8iAB7-(3-hydroxyphenyl)-5-methyl[1,2,4]triazolo[4,3-a]quinolin-1(2h)-oneHuman1558
CHEK1 (CHK1)CAMKLCAMK2wmrAB5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-oneHuman1604
CHEK1 (CHK1)CAMKLCAMK3pa5AA2-(carbamoylamino)-5-(4-chlorophenyl)-n-[(3s)-piperidin-3-yl]thiophene-3-carboxamideHuman1676
CHEK1 (CHK1)CAMKLCAMK5oopABphosphoaminophosphonic acid-adenylate esterHuman8607
CHEK1 (CHK1)CAMKLCAMK2xeyA3-(1h-indol-3-yl)-6-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazineHuman1668
CHEK1 (CHK1)CAMKLCAMK3u9nA2-(2,3-dihydro-1-benzofuran-5-yl)-n-[2-(piperazin-1-yl)phenyl]-1,3-thiazole-4-carboxamideHuman1597
CHEK1 (CHK1)CAMKLCAMK7akoBBstaurosporineHuman13496
CHEK1 (CHK1)CAMKLCAMK1nvqA7-hydroxystaurosporineHuman1642
CHEK1 (CHK1)CAMKLCAMK5oprA5-[4-(morpholin-4-ylmethyl)phenyl]-3-(1-propan-2-yl-1,2,3-triazol-4-yl)pyridin-2-amineHuman8614
STK17B (DRAK2)DAPKCAMK7q7eABadenosine-5'-triphosphateHuman14507
STK17B (DRAK2)DAPKCAMK7q7cABadenosine-5'-diphosphateHuman14508
STK17B (DRAK2)DAPKCAMK3lm0AA[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-5-methylpyrimidin-2-yl}amino)phenyl]acetonitrileHuman6796
STK17B (DRAK2)DAPKCAMK6y6hAA2-[6-(1-benzothiophen-2-yl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12043
STK17B (DRAK2)DAPKCAMK3lm0AB[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-5-methylpyrimidin-2-yl}amino)phenyl]acetonitrileHuman6797
STK17B (DRAK2)DAPKCAMK7q7dABadenosine-5'-triphosphateHuman14509
STK17B (DRAK2)DAPKCAMK6zjfAA2-[6-(4-cyclopropylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12642
STK17B (DRAK2)DAPKCAMK3lm5AA3,5,7,3',4'-pentahydroxyflavoneHuman6795
STK17B (DRAK2)DAPKCAMK7q7cAAadenosine-5'-diphosphateHuman14510
STK17B (DRAK2)DAPKCAMK6zjfAB2-[6-(4-cyclopropylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12643
STK17B (DRAK2)DAPKCAMK6y6fAA2-[6-(4-methylsulfanylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12045
STK17B (DRAK2)DAPKCAMK6y6fAB2-[6-(4-methylsulfanylphenyl)thieno[3,2-d]pyrimidin-4-yl]sulfanylethanoic acidHuman12042
STK17B (DRAK2)DAPKCAMK7q7dAAadenosine-5'-triphosphateHuman14519
STK17B (DRAK2)DAPKCAMK6qf4ABadenosine-5'-diphosphateHuman11396
STK17B (DRAK2)DAPKCAMK7akgAA4-amino-5-fluoro-3-[5-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]quinolin-2(1h)-oneHuman13005
STK17B (DRAK2)DAPKCAMK3lm5AB3,5,7,3',4'-pentahydroxyflavoneHuman6798
MARK3CAMKLCAMK3fe3AA-Human3267
MARK3CAMKLCAMK2qnjA-Human3269
MARK3CAMKLCAMK3fe3BB-Human3265
MARK3CAMKLCAMK2qnjB-Human3264
MARK3CAMKLCAMK9vgrAn-[5-[[4-[[(3r,3ar,6r,6ar)-3-methoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]-1-methyl-pyrazole-4-carboxamideHuman15736
MARK3CAMKLCAMK9ysqA3-({5-chloro-2-[2-(difluoromethoxy)-4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl}amino)thiophene-2-carboxamideHuman15737
MARK3CAMKLCAMK9vfoAn-[5-[[4-[[(3r,3ar,6r,6ar)-3-methoxy-2,3,3a,5,6,6a-hexahydrofuro[3,2-b]furan-6-yl]oxy]-5-chloranyl-pyrimidin-2-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]-2-azanyl-ethanamideHuman15738
MARK3CAMKLCAMK3fe3AB-Human3266
MARK3CAMKLCAMK3fe3BA-Human3268
STK17A (DRAK1)DAPKCAMK7qufA~{n}-~{tert}-butyl-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamideHuman14093
STK17A (DRAK1)DAPKCAMK7queA~{n}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamideHuman14094
DAPK3DAPKCAMK2j90BB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman379
DAPK3DAPKCAMK5vjaBB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10350
DAPK3DAPKCAMK5a6oAB-Human6163
DAPK3DAPKCAMK5a6nAB5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ideHuman6165
DAPK3DAPKCAMK3bhyAA(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman385
DAPK3DAPKCAMK5vjaAB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10349
DAPK3DAPKCAMK3bhyAB(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman381
DAPK3DAPKCAMK5vjaDA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10348
DAPK3DAPKCAMK5a6oBA-Human6168
DAPK3DAPKCAMK1yrpB-Human383
DAPK3DAPKCAMK5a6oAA-Human6167
MELKCAMKLCAMK4d2tBB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2512
MELKCAMKLCAMK6gvxBB6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11138
MELKCAMKLCAMK5ih9AB1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazineHuman6657
MELKCAMKLCAMK4bkzAAn-(3-aminopropyl)-8-[(3-fluorophenyl)amino]-2,4,5,7-tetrahydropyrazolo[3,4-e]indazole-3-carboxamideHuman2505
MELKCAMKLCAMK5mahAA~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamideHuman8729
MELKCAMKLCAMK4d2wBB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2482
MELKCAMKLCAMK4umpCB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2508
MELKCAMKLCAMK4d2pCA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2496
MELKCAMKLCAMK5ihaAB1-methyl-4-(4-{4-[3-(2-methylpropoxy)pyridin-4-yl]-1h-pyrazol-1-yl}phenyl)piperazineHuman6658
MELKCAMKLCAMK4umrA4-fluoro-n-(1,2,3,4-tetrahydroisoquinolin-7-yl)benzamideHuman2521
MELKCAMKLCAMK6gvxAA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11137
MELKCAMKLCAMK5twuB-Human8672
MELKCAMKLCAMK4d2tBA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2520
MELKCAMKLCAMK4d2tAA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2487
MELKCAMKLCAMK4d2pDB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2518
MELKCAMKLCAMK4umpDA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2516
MELKCAMKLCAMK4d2wCA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2527
MELKCAMKLCAMK5k00AB4-{2-[(3-methoxyphenyl)amino]-4-[(piperidin-4-yl)methoxy]pyrimidin-5-yl}-n-[2-oxo-2-(phenylamino)ethyl]benzamideHuman7498
MELKCAMKLCAMK4d2wDA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2481
MELKCAMKLCAMK4bl1ABphosphoaminophosphonic acid-adenylate esterHuman2519
MELKCAMKLCAMK5ihcAB4-[1-(2-fluorophenyl)-1h-pyrazol-4-yl]-3-[(piperidin-4-yl)methoxy]pyridineHuman6662
MELKCAMKLCAMK4d2tDA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2530
MELKCAMKLCAMK4d2vAA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2493
MELKCAMKLCAMK4d2pBB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2498
MELKCAMKLCAMK4d2wBA4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2500
MELKCAMKLCAMK5ih9AA1-methyl-4-[4-(4-{3-[(piperidin-4-yl)methoxy]pyridin-4-yl}-1h-pyrazol-1-yl)phenyl]piperazineHuman6659
MELKCAMKLCAMK4umuA(2-ethoxy-4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}phenyl)methanaminiumHuman2517
MELKCAMKLCAMK4d2pBA7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2494
MELKCAMKLCAMK5maiAB3-[(3~{z})-3-[[[4-[(dimethylamino)methyl]phenyl]amino]-phenyl-methylidene]-2-oxidanylidene-1~{h}-indol-6-yl]-~{n}-ethyl-prop-2-ynamideHuman8730
MELKCAMKLCAMK6gvxBA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman11136
MELKCAMKLCAMK5twyA2-(benzyloxy)-4-(1h-pyrazol-4-yl)-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman8671
MELKCAMKLCAMK4d2vBA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2483
MELKCAMKLCAMK4umqAA3-{5-[(3-hydroxy-5-methoxyphenyl)amino]-2-(phenylcarbamoyl)phenoxy}propan-1-aminiumHuman2488
MELKCAMKLCAMK4d2tCA3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2491
MELKCAMKLCAMK5mahAB~{n}-methyl-4-[[4-[[3-[methyl(methylsulfonyl)amino]pyrazin-2-yl]methylamino]-5-(trifluoromethyl)pyrimidin-2-yl]amino]benzamideHuman8734
MELKCAMKLCAMK4bkyAA3'-{[(4-bromo-1-methyl-1h-pyrrol-2-yl)carbonyl]amino}-n-[(1s)-1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1',4'-dihydro-5'h-spiro[cyclopropane-1,6'-pyrrolo[3,4-c]pyrazole]-5'-carboxamideHuman2480
MELKCAMKLCAMK4d2tCB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2526
MELKCAMKLCAMK4d2wAB4-bromo-n-(2,3,4,5-tetrahydro-1h-3-benzazepin-7-yl)benzamideHuman2509
MELKCAMKLCAMK4umpAB3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2485
MELKCAMKLCAMK5twuA-Human8670
MELKCAMKLCAMK5tx3A7-[(1s)-4-hydroxy-2,3-dihydro-1h-inden-1-yl]-5,5-dimethyl-2-({3-[(pyrrolidin-1-yl)methyl]phenyl}amino)-5,7-dihydro-6h-pyrrolo[2,3-d]pyrimidin-6-oneHuman8673
MELKCAMKLCAMK4bl1AAphosphoaminophosphonic acid-adenylate esterHuman2514
MELKCAMKLCAMK4d2vCB7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2492
MELKCAMKLCAMK4umtA1-(4-{[3-(isoquinolin-7-yl)prop-2-yn-1-yl]oxy}-2-methoxybenzyl)piperazinediiumHuman2510
MELKCAMKLCAMK5magABpf-3758309Human8731
MELKCAMKLCAMK4umpBA3-(isoquinolin-7-yl)prop-2-yn-1-olHuman2524
MELKCAMKLCAMK4d2vCA7-{[2-methoxy-4-(1h-pyrazol-4-yl)benzoyl]amino}-2,3,4,5-tetrahydro-1h-3-benzazepiniumHuman2529
MELKCAMKLCAMK4d2pAB7-({4-[(3-hydroxy-5-methoxyphenyl)amino]benzoyl}amino)-1,2,3,4-tetrahydroisoquinoliniumHuman2499
MELKCAMKLCAMK4d2tDB3-[2-(phenylcarbamoyl)-5-(1h-pyrazol-4-yl)phenoxy]propan-1-aminiumHuman2511
CHEK1 (CHK1)CAMKLCAMK2wmrAA5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3h)-oneHuman1609
STK17B (DRAK2)DAPKCAMK6qf4AAadenosine-5'-diphosphateHuman11397
RPS6KA5-b (MSK1-b)RSKbCAMK3kn6A-Human4602
RPS6KA5-b (MSK1-b)RSKbCAMK3kn6B-Human4601
RPS6KA5-b (MSK1-b)RSKbCAMK7up7AB(2s)-2-cyano-n-(1-hydroxy-2-methylpropan-2-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]propanamideHuman14317
RPS6KA5-b (MSK1-b)RSKbCAMK7up5AB(2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrileHuman14278
RPS6KA5-b (MSK1-b)RSKbCAMK3kn5Bphosphoaminophosphonic acid-adenylate esterHuman4600
RPS6KA5-b (MSK1-b)RSKbCAMK7up4AB(5m)-5-(2,5-dichloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14279
RPS6KA5-b (MSK1-b)RSKbCAMK7up5AA(2m)-6-chloro-2-(5h-pyrrolo[3,2-d]pyrimidin-5-yl)pyridine-3-carbonitrileHuman14280
RPS6KA5-b (MSK1-b)RSKbCAMK7up6AA(e)-3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)phenyl)-2-cyanoacrylamide bound formHuman14353
RPS6KA5-b (MSK1-b)RSKbCAMK7up8AB(5m)-5-(5-bromo-2-chloropyrimidin-4-yl)-5h-pyrrolo[3,2-d]pyrimidineHuman14281
RPS6KA5-b (MSK1-b)RSKbCAMK3kn5Aphosphoaminophosphonic acid-adenylate esterHuman4603
MAPKAPK3MAPKAPKCAMK3r1nAA2'-[2-(1,3-benzodioxol-5-yl)pyrimidin-4-yl]-5',6'-dihydrospiro[piperidine-4,7'-pyrrolo[3,2-c]pyridin]-4'(1'h)-oneHuman4589
MAPKAPK3MAPKAPKCAMK7nrbAB2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman14051
MAPKAPK3MAPKAPKCAMK7nrbAA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman14052
MAPKAPK3MAPKAPKCAMK3fhrAB2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman4598
MAPKAPK3MAPKAPKCAMK3sheAAn-{4-[(3s)-4'-oxo-1',4',5',6'-tetrahydrospiro[piperidine-3,7'-pyrrolo[3,2-c]pyridin]-2'-yl]pyridin-2-yl}-3-(trifluoromethyl)benzamideHuman4594
CAMK2D (CaMK2d)CAMK2CAMK2welAB(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2137
CAMK2D (CaMK2d)CAMK2CAMK6aywAn-[2-(dimethylamino)ethyl]-3-[6-(thiophen-2-yl)imidazo[1,2-b]pyridazin-3-yl]benzamideHuman8666
CAMK2D (CaMK2d)CAMK2CAMK2vn9A[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2140
CAMK2D (CaMK2d)CAMK2CAMK2vn9B[4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]quinazolin-2-yl}imino)cyclohexa-2,5-dien-1-yl]acetonitrileHuman2139
CAMK2D (CaMK2d)CAMK2CAMK5vloBn-[(2s)-2-(diethylamino)propyl]-2-[(2s)-2-(methylcarbamoyl)azetidin-1-yl]-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamideHuman8347
CAMK2D (CaMK2d)CAMK2CAMK2welAC(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2136
CAMK2D (CaMK2d)CAMK2CAMK2welAA(3z)-n,n-dimethyl-2-oxo-3-(4,5,6,7-tetrahydro-1h-indol-2-ylmethylidene)-2,3-dihydro-1h-indole-5-sulfonamideHuman2138
STK11 (LKB1)CAMKLCAMK2wtkFphosphoaminophosphonic acid-adenylate esterHuman1869
STK11 (LKB1)CAMKLCAMK2wtkCphosphoaminophosphonic acid-adenylate esterHuman1868
MAPKAPK2MAPKAPKCAMK2onlC-Human1306
MAPKAPK2MAPKAPKCAMK3r2bD-Human1337
MAPKAPK2MAPKAPKCAMK6t8xA(10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-oneHuman13548
MAPKAPK2MAPKAPKCAMK3wi6Dn-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1340
MAPKAPK2MAPKAPKCAMK3gokJ2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1319
MAPKAPK2MAPKAPKCAMK3kc3In~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1354
MAPKAPK2MAPKAPKCAMK6tcaEA-Human12500
MAPKAPK2MAPKAPKCAMK2jbpL2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1283
MAPKAPK2MAPKAPKCAMK3kgaAA6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-oneHuman9476
MAPKAPK2MAPKAPKCAMK3gokH2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1338
MAPKAPK2MAPKAPKCAMK3kc3Hn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1291
MAPKAPK2MAPKAPKCAMK3gokI2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1305
MAPKAPK2MAPKAPKCAMK3kc3An~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1289
MAPKAPK2MAPKAPKCAMK3a2cAn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1330
MAPKAPK2MAPKAPKCAMK3wi6An-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1308
MAPKAPK2MAPKAPKCAMK3gokL2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1365
MAPKAPK2MAPKAPKCAMK1nxkCstaurosporineHuman1312
MAPKAPK2MAPKAPKCAMK1nxkDstaurosporineHuman1334
MAPKAPK2MAPKAPKCAMK3m2wAA2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-oneHuman9474
MAPKAPK2MAPKAPKCAMK6tcaGB-Human12501
MAPKAPK2MAPKAPKCAMK3fykX(3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-oneHuman1297
MAPKAPK2MAPKAPKCAMK3a2cHn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1325
MAPKAPK2MAPKAPKCAMK2jboA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1333
MAPKAPK2MAPKAPKCAMK6tcaAA-Human12502
MAPKAPK2MAPKAPKCAMK6tcaCA-Human12504
MAPKAPK2MAPKAPKCAMK3r30AB1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acidHuman1309
MAPKAPK2MAPKAPKCAMK3gokA2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1281
MAPKAPK2MAPKAPKCAMK3gokD2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1284
MAPKAPK2MAPKAPKCAMK6tcaGA-Human12505
MAPKAPK2MAPKAPKCAMK3a2cKn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1360
MAPKAPK2MAPKAPKCAMK3gokG2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1351
MAPKAPK2MAPKAPKCAMK3a2cLn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1301
MAPKAPK2MAPKAPKCAMK3fyjX(10r)-10-methyl-3-(6-methylpyridin-3-yl)-9,10,11,12-tetrahydro-8h-[1,4]diazepino[5',6':4,5]thieno[3,2-f]quinolin-8-oneHuman1336
MAPKAPK2MAPKAPKCAMK3wi6Fn-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1313
MAPKAPK2MAPKAPKCAMK2jbpC2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1344
MAPKAPK2MAPKAPKCAMK2jbpD2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1327
MAPKAPK2MAPKAPKCAMK3r2bL-Human1295
MAPKAPK2MAPKAPKCAMK2pzyD-Human1357
MAPKAPK2MAPKAPKCAMK3m42A2-[5-(2-methoxyethoxy)pyridin-3-yl]-8,9,10,11-tetrahydro-7h-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin-7-oneHuman9475
MAPKAPK2MAPKAPKCAMK3a2cIn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1311
MAPKAPK2MAPKAPKCAMK6tcaCB-Human12506
MAPKAPK2MAPKAPKCAMK3kc3En~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1285
MAPKAPK2MAPKAPKCAMK1kwpB-Human1296
MAPKAPK2MAPKAPKCAMK3kc3Ln~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1324
MAPKAPK2MAPKAPKCAMK3a2cGn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1343
MAPKAPK2MAPKAPKCAMK3kgaAB6-{3-amino-1-[3-(1h-indol-6-yl)phenyl]-1h-pyrazol-4-yl}-3,4-dihydroisoquinolin-1(2h)-oneHuman9477
MAPKAPK2MAPKAPKCAMK3kc3G-Human1356
MAPKAPK2MAPKAPKCAMK3r2bJ-Human1331
MAPKAPK2MAPKAPKCAMK3gokK2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1299
MAPKAPK2MAPKAPKCAMK6tcaAB-Human12507
MAPKAPK2MAPKAPKCAMK9r59A5-[3-[bis(oxidanyl)-$l^{3}-sulfanyl]oxy-4-chloranyl-phenyl]-~{n}-(4-piperazin-1-ylphenyl)-~{n}-(pyridin-2-ylmethyl)furan-2-carboxamideHuman16033
MAPKAPK2MAPKAPKCAMK3r30AA1-(2-aminoethyl)-3-[2-(quinolin-3-yl)pyridin-4-yl]-1h-pyrazole-5-carboxylic acidHuman1352
MAPKAPK2MAPKAPKCAMK3wi6Bn-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1282
MAPKAPK2MAPKAPKCAMK4tyhAA-Human1302
MAPKAPK2MAPKAPKCAMK3gokB2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1304
MAPKAPK2MAPKAPKCAMK8xu4A-Human15173
MAPKAPK2MAPKAPKCAMK3a2cFn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1355
MAPKAPK2MAPKAPKCAMK2ozaA-Human1310
MAPKAPK2MAPKAPKCAMK3kc3Bn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1298
MAPKAPK2MAPKAPKCAMK3r2bF-Human1321
MAPKAPK2MAPKAPKCAMK3wi6Cn-[(3s)-piperidin-3-yl]-7,8-dihydro-6h-pyrazolo[1,5-a]pyrrolo[3,2-e]pyrimidin-5-amineHuman1346
MAPKAPK2MAPKAPKCAMK3a2cEn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1315
MAPKAPK2MAPKAPKCAMK2jbpF2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1335
MAPKAPK2MAPKAPKCAMK3fpmA3-{[(1r)-1-phenylethyl]amino}-4-(pyridin-4-ylamino)cyclobut-3-ene-1,2-dioneHuman1367
MAPKAPK2MAPKAPKCAMK2jbpE2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1358
MAPKAPK2MAPKAPKCAMK3m2wAB2'-(2-fluorophenyl)-1-methyl-6',8',9',11'-tetrahydrospiro[azetidine-3,10'-pyrido[3',4':4,5]pyrrolo[2,3-f]isoquinolin]-7'(5'h)-oneHuman9473
MAPKAPK2MAPKAPKCAMK4tyhAB-Human1322
MAPKAPK2MAPKAPKCAMK3gokE2-(2-quinolin-3-ylpyridin-4-yl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman1300
MAPKAPK2MAPKAPKCAMK3a2cDn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1316
MAPKAPK2MAPKAPKCAMK3kc3Kn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1317
MAPKAPK2MAPKAPKCAMK3kc3Jn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1347
MAPKAPK2MAPKAPKCAMK2jbpJ-Human1359
MAPKAPK2MAPKAPKCAMK2pzyCstaurosporineHuman1279
MAPKAPK2MAPKAPKCAMK3kc3Fn~4~-[7-(1-benzofuran-2-yl)-1h-indazol-5-yl]pyrimidine-2,4-diamineHuman1341
MAPKAPK2MAPKAPKCAMK3a2cJn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman1353
MAPKAPK2MAPKAPKCAMK1nxkBstaurosporineHuman1292
MAPKAPK2MAPKAPKCAMK3r2bI-Human1294
PASKCAMKLCAMK3dlsFadenosine-5'-diphosphateHuman3380
PASKCAMKLCAMK3dlsCadenosine-5'-diphosphateHuman3377
PASKCAMKLCAMK3dlsEadenosine-5'-diphosphateHuman3379
PASKCAMKLCAMK3dlsDadenosine-5'-diphosphateHuman3378
CHEK2 (CHK2)RAD53CAMK2xbjA4-fluoro-2-(4-{[(3s,4r)-4-(1-hydroxy-1-methylethyl)pyrrolidin-3-yl]amino}-6,7-dimethoxyquinazolin-2-yl)phenolHuman4783
CHEK2 (CHK2)RAD53CAMK4bdfA5-methyl-3-phenyl-1h-pyrazoleHuman4765
CHEK2 (CHK2)RAD53CAMK2cn5Aadenosine-5'-diphosphateHuman4789
CHEK2 (CHK2)RAD53CAMK2ycqAAn-{4-[(1e)-n-1h-imidazol-2-ylethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamideHuman4766
CHEK2 (CHK2)RAD53CAMK3i6wG-Human4793
CHEK2 (CHK2)RAD53CAMK3i6wC-Human4802
CHEK2 (CHK2)RAD53CAMK3i6wB-Human4792
CHEK2 (CHK2)RAD53CAMK2wtjAB2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)-n-[2-(dimethylamino)ethyl]pyridine-3-carboxamideHuman4761
CHEK2 (CHK2)RAD53CAMK4bdgA3-(pyridin-3-yl)-1h-pyrazol-5-amineHuman4796
CHEK2 (CHK2)RAD53CAMK2cn8AdebromohymenialdisineHuman4808
CHEK2 (CHK2)RAD53CAMK2yitABn-{4-[(1e)-n-carbamimidoylbutanehydrazonoyl]phenyl}-5-methoxy-1h-indole-2-carboxamideHuman4770
CHEK2 (CHK2)RAD53CAMK4bdjA3-cyclopropyl-4-(furan-2-yl)-1h-pyrazolo[3,4-b]pyridineHuman4795
CHEK2 (CHK2)RAD53CAMK2ycsABn-{4-[(1e)-n-carbamimidoylethanehydrazonoyl]phenyl}-1h-indole-3-carboxamideHuman4764
CHEK2 (CHK2)RAD53CAMK2ycrAB1,3-bis{4-[(1e)-n-(4,5-dihydro-1h-imidazol-2-yl)ethanehydrazonoyl]phenyl}ureaHuman4775
CHEK2 (CHK2)RAD53CAMK2w7xABn-[4-[(e)-n-carbamimidamido-c-methyl-carbonimidoyl]phenyl]-7-nitro-1h-indole-2-carboxamideHuman4780
CHEK2 (CHK2)RAD53CAMK4a9sAB2-(4-(3-hydroxyphenoxy)phenyl)-1h-benzo[d]imidazole-5-carboxamideHuman4801
CHEK2 (CHK2)RAD53CAMK4a9sAA2-(4-(3-hydroxyphenoxy)phenyl)-1h-benzo[d]imidazole-5-carboxamideHuman4772
CHEK2 (CHK2)RAD53CAMK4bddA1-(tert-butyl)-3-(quinoxalin-6-yl)ureaHuman4786
CHEK2 (CHK2)RAD53CAMK2wtdA4-[2-amino-5-(1,3-benzodioxol-4-yl)pyridin-3-yl]benzamideHuman4769
CHEK2 (CHK2)RAD53CAMK2ycqABn-{4-[(1e)-n-1h-imidazol-2-ylethanehydrazonoyl]phenyl}-7-nitro-1h-indole-2-carboxamideHuman4790
CHEK2 (CHK2)RAD53CAMK2xm9AA4-(1h-pyrazol-5-yl)-2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenolHuman4785
CHEK2 (CHK2)RAD53CAMK4a9uA2-{4-[(1-benzylpiperidin-4-yl)methoxy]phenyl}-1h-benzimidazole-6-carboxamideHuman4778
CHEK2 (CHK2)RAD53CAMK2yitAAn-{4-[(1e)-n-carbamimidoylbutanehydrazonoyl]phenyl}-5-methoxy-1h-indole-2-carboxamideHuman4777
CHEK2 (CHK2)RAD53CAMK3i6wF-Human4776
CHEK2 (CHK2)RAD53CAMK2w0jA4,4'-diacetyldiphenylurea-bis(guanylhydrazone)Human4811
CHEK2 (CHK2)RAD53CAMK4a9rA2-[4-(4-chlorophenoxy)phenyl]-1h-benzimidazole-6-carboxamideHuman4763
CHEK2 (CHK2)RAD53CAMK4bdbA4-[(e)-c-methyl-n-oxidanyl-carbonimidoyl]benzene-1,3-diolHuman4797
CHEK2 (CHK2)RAD53CAMK4bdaA3,4-dihydro[1,2,4]triazolo[1,5-a][3,1]benzimidazol-9-iumHuman4788
CHEK2 (CHK2)RAD53CAMK4a9tA2-(4-{[1-(4-chlorobenzyl)piperidin-4-yl]methoxy}phenyl)-1h-benzimidazole-5-carboxamideHuman4814
CHEK2 (CHK2)RAD53CAMK4bdkAn-[(4-methoxyphenyl)methyl]quinoxaline-6-carboxamideHuman4809
CHEK2 (CHK2)RAD53CAMK2ycsAAn-{4-[(1e)-n-carbamimidoylethanehydrazonoyl]phenyl}-1h-indole-3-carboxamideHuman4804
CHEK2 (CHK2)RAD53CAMK2wtiAA4-[2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)pyridin-3-yl]benzamideHuman4812
CHEK2 (CHK2)RAD53CAMK2wtjAA2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)-n-[2-(dimethylamino)ethyl]pyridine-3-carboxamideHuman4779
CHEK2 (CHK2)RAD53CAMK2wtcA4-[2-amino-5-(4-hydroxy-3-methoxyphenyl)pyridin-3-yl]benzamideHuman4767
CHEK2 (CHK2)RAD53CAMK3i6wE-Human4806
CHEK2 (CHK2)RAD53CAMK3i6wD-Human4805
CHEK2 (CHK2)RAD53CAMK2xm9AB4-(1h-pyrazol-5-yl)-2-{4-[(3s)-pyrrolidin-3-ylamino]quinazolin-2-yl}phenolHuman4803
CHEK2 (CHK2)RAD53CAMK4bdiA1-acetyl-n-(5-methylpyridin-2-yl)piperidine-4-carboxamideHuman4762
CHEK2 (CHK2)RAD53CAMK4bdcAn-(furan-2-ylmethyl)quinoxaline-6-carboxamideHuman4794
CHEK2 (CHK2)RAD53CAMK2w7xAAn-[4-[(e)-n-carbamimidamido-c-methyl-carbonimidoyl]phenyl]-7-nitro-1h-indole-2-carboxamideHuman4784
CHEK2 (CHK2)RAD53CAMK2yiqAB(e)-5-(1-(2-carbamimidoylhydrazono)ethyl)-n-(1h-indol-6-yl)-1h-indole-2-carboxamideHuman4800
CHEK2 (CHK2)RAD53CAMK3i6wH-Human4799
CHEK2 (CHK2)RAD53CAMK2wtiAB4-[2-amino-5-(2,3-dihydrothieno[3,4-b][1,4]dioxin-5-yl)pyridin-3-yl]benzamideHuman4807
CHEK2 (CHK2)RAD53CAMK4bdhA3-methyl-4-(thiophen-2-yl)-1h-pyrazol-5-amineHuman4782
CHEK2 (CHK2)RAD53CAMK3i6uA-Human4798
CHEK2 (CHK2)RAD53CAMK3i6wA-Human4813
CASKCASKCAMK3mfsABphosphoaminophosphonic acid-adenylate esterHuman3829
CASKCASKCAMK3c0iAB[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3819
CASKCASKCAMK7oajAA4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-n-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamideHuman13582
CASKCASKCAMK3c0hAadenosine monophosphateHuman3825
CASKCASKCAMK3mftAB-Human3821
CASKCASKCAMK9m6gAAphosphoaminophosphonic acid-adenylate esterHuman16103
CASKCASKCAMK3mfuABphosphoaminophosphonic acid-adenylate esterHuman3832
CASKCASKCAMK6kmhB-Human12671
CASKCASKCAMK3c0gBA[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3824
CASKCASKCAMK3mfrABphosphoaminophosphonic acid-adenylate esterHuman3831
CASKCASKCAMK3mfsAAphosphoaminophosphonic acid-adenylate esterHuman3818
CASKCASKCAMK3c0hBadenosine monophosphateHuman3817
CASKCASKCAMK3tacA-Human3820
CASKCASKCAMK6kmhA-Human12672
CASKCASKCAMK7oakA2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclopentylamino)-n-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideHuman13585
CASKCASKCAMK3mfuAAphosphoaminophosphonic acid-adenylate esterHuman3816
CASKCASKCAMK3mftAA-Human3823
CASKCASKCAMK3c0iAA[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3830
CASKCASKCAMK3c0gAA[(2r,3s,4r,5r)-5-(6-aminopurin-9-yl)-4-hydroxy-2-(hydroxymethyl)oxolan-3-yl] dihydrogen phosphateHuman3828
CASKCASKCAMK7oalA2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclohexylamino)-n-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamideHuman13586
PRKAA1 (AMPKa1)CAMKLCAMK6c9gAstaurosporineHuman10715
PRKAA1 (AMPKa1)CAMKLCAMK4redB-Human123
PRKAA1 (AMPKa1)CAMKLCAMK6c9fAstaurosporineHuman10716
RPS6KA1-b (RSK3-b)RSKbCAMK3rnyAA-Human5568
RPS6KA1-b (RSK3-b)RSKbCAMK4nifDB-Human5575
SNRKCAMKLCAMK5yksB-Human8661
TTNMLCKCAMK4jnwBB-Human128
TTNMLCKCAMK1tkiA-Human130
TTNMLCKCAMK4jnwBA-Human125
TTNMLCKCAMK4jnwAB-Human129
TTNMLCKCAMK4jnwAA-Human127
CAMK4 (CaMK4)CAMK1CAMK2w4oA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman2687
STK40 (SgK495)SgK495CAMK5l2qAB-Human8014
STK40 (SgK495)SgK495CAMK5l2qDB-Human8013
STK40 (SgK495)SgK495CAMK5l2qBB-Human8017
STK40 (SgK495)SgK495CAMK5l2qDA-Human8012
STK40 (SgK495)SgK495CAMK5l2qAA-Human8015
STK40 (SgK495)SgK495CAMK5l2qCA-Human8018
STK40 (SgK495)SgK495CAMK5l2qCB-Human8016
PRKAA2 (AMPKa2)CAMKLCAMK2h6dAB-Human194
PRKAA2 (AMPKa2)CAMKLCAMK5ezvABstaurosporineHuman6428
PRKAA2 (AMPKa2)CAMKLCAMK6b1uABstaurosporineHuman9849
PRKAA2 (AMPKa2)CAMKLCAMK3aqvA6-[4-(2-piperidin-1-ylethoxy)phenyl]-3-pyridin-4-ylpyrazolo[1,5-a]pyrimidineHuman193
PRKAA2 (AMPKa2)CAMKLCAMK4cfeAstaurosporineHuman195
PRKAA2 (AMPKa2)CAMKLCAMK4zhxCA(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6427
PRKAA2 (AMPKa2)CAMKLCAMK6b1uAAstaurosporineHuman9848
PRKAA2 (AMPKa2)CAMKLCAMK5ezvCAstaurosporineHuman6430
PRKAA2 (AMPKa2)CAMKLCAMK4cffCstaurosporineHuman190
PRKAA2 (AMPKa2)CAMKLCAMK2h6dAA-Human196
PRKAA2 (AMPKa2)CAMKLCAMK5ezvCBstaurosporineHuman6426
PRKAA2 (AMPKa2)CAMKLCAMK5ezvAAstaurosporineHuman6424
PRKAA2 (AMPKa2)CAMKLCAMK6b2eAstaurosporineHuman9851
PRKAA2 (AMPKa2)CAMKLCAMK4zhxAB(5s,6r,7r,9r,13cr,14r,16as)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5h,13ch-5,9-epoxy-4b,9a,15-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-olHuman6429