Search results (39 entries covering 17 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b55 | A | A | - | Mouse | 14244 | ||
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b57 | A | A | - | Mouse | 14246 | ||
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b55 | A | B | - | Mouse | 14247 | ||
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b56 | A | B | - | Mouse | 14249 | ||
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b57 | A | B | - | Mouse | 14248 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2yaa | A | B | adenosine-5'-triphosphate | Mouse | 5747 | ||
| Prkaa1 (AMPKa1) | CAMKL | CAMK | 5ufu | A | staurosporine | Mouse | 7590 | |||
| Dapk2 (DAPK2) | DAPK | CAMK | 2yab | A | A | adenosine monophosphate | Mouse | 5750 | ||
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | D | A | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8695 | ||
| Brsk2 (BRSK2) | CAMKL | CAMK | 4yom | B | - | Mouse | 6292 | |||
| Brsk2 (BRSK2) | CAMKL | CAMK | 4ynz | B | - | Mouse | 6291 | |||
| Brsk2 (BRSK2) | CAMKL | CAMK | 4ynz | A | - | Mouse | 6293 | |||
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr7 | A | B | - | Mouse | 5757 | ||
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr8 | A | B | - | Mouse | 5755 | ||
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr7 | A | A | - | Mouse | 5759 | ||
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 4m8t | A | (2e)-2-cyano-3-[3-(1h-pyrazol-4-yl)phenyl]prop-2-enamide | Mouse | 5756 | |||
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 5o1s | A | dimethyl fumarate | Mouse | 9976 | |||
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 4mao | A | (2z)-2-(1h-1,2,4-triazol-1-yl)-3-[3-(3,4,5-trimethoxyphenyl)-1h-indazol-5-yl]prop-2-enenitrile | Mouse | 5758 | |||
| Rps6ka3-b (RSK2-b) | RSKb | CAMK | 2qr8 | A | A | - | Mouse | 5760 | ||
| Camk2a (CaMK2a) | CAMK2 | CAMK | 7b56 | A | A | - | Mouse | 14245 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2ya9 | B | B | - | Mouse | 5744 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2yab | B | B | adenosine monophosphate | Mouse | 5745 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2ya9 | B | A | - | Mouse | 5743 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2yaa | B | B | adenosine-5'-triphosphate | Mouse | 5754 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2yaa | B | A | adenosine-5'-triphosphate | Mouse | 5751 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2yaa | A | A | adenosine-5'-triphosphate | Mouse | 5746 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2yab | A | B | adenosine monophosphate | Mouse | 5753 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2ya9 | A | A | - | Mouse | 5749 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2yab | B | A | adenosine monophosphate | Mouse | 5748 | ||
| Dapk2 (DAPK2) | DAPK | CAMK | 2ya9 | A | B | - | Mouse | 5752 | ||
| Melk (MELK) | CAMKL | CAMK | 4cqg | A | 1-[6-(3,5-dichloro-4-hydroxyphenyl)-4-({trans-4-[(dimethylamino)methyl]cyclohexyl}amino)-1,5-naphthyridin-3-yl]ethanone | Mouse | 6865 | |||
| Melk (MELK) | CAMKL | CAMK | 4bfm | A | phosphoaminophosphonic acid-adenylate ester | Mouse | 5798 | |||
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | A | A | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8694 | ||
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | B | B | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8693 | ||
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | D | B | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8696 | ||
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | A | B | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8691 | ||
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | C | A | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8697 | ||
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | C | B | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8692 | ||
| Camk2d (CaMK2d) | CAMK2 | CAMK | 6bab | B | A | n-[(2s)-2-(diethylamino)propyl]-2-(3-hydroxyazetidin-1-yl)-6-[5-(thiophen-2-yl)pyrazolo[1,5-a]pyrimidin-3-yl]pyridine-4-carboxamide | Mouse | 8690 |