| VRK1 | VRK | CK1 | 8v42 | A | B | - | Human | 15394 | |
| VRK1 | VRK | CK1 | 8v42 | A | A | - | Human | 15395 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4twc | A | B | 2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamide | Human | 2157 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | D | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4617 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | C | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4619 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | B | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4622 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4621 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4618 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | D | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4623 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | C | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4624 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | B | A | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2174 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 2c47 | B | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 4620 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izu | A | B | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 2225 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izt | A | A | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 2216 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 4hgs | A | | 2-{2-[(3,4-difluorophenoxy)methyl]-5-methoxypyridin-4-yl}-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 2224 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 4g16 | A | | 2-[(4-{[3-(trifluoromethyl)pyridin-2-yl]oxy}phenyl)amino]-1h-benzimidazole-6-carbonitrile | Human | 2219 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izs | A | B | {[4-amino-2-(3-chloroanilino)-1,3-thiazol-5-yl](4-fluorophenyl)methanone | Human | 2223 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izu | A | A | 2-({6-[(3-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 2218 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2chl | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 2220 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izs | A | A | {[4-amino-2-(3-chloroanilino)-1,3-thiazol-5-yl](4-fluorophenyl)methanone | Human | 2228 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izr | A | B | {(2z)-4-amino-2-[(4-methoxyphenyl)imino]-2,3-dihydro-1,3-thiazol-5-yl}(4-methoxyphenyl)methanone | Human | 2221 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 4hgl | A | | 2-[5-methoxy-2-(quinolin-3-yl)pyrimidin-4-yl]-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 2227 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2chl | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 2217 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | C | B | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2184 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 6gro | A | B | 4-[5-(2-azanylpyrimidin-4-yl)-4-(4-fluorophenyl)imidazol-1-yl]cyclohexan-1-ol | Human | 10003 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 4g17 | A | | 2-[(4-tert-butylphenyl)amino]-1h-benzimidazole-6-carbonitrile | Human | 2226 | |
| VRK1 | VRK | CK1 | 6dd4 | A | B | - | Human | 9939 | |
| VRK1 | VRK | CK1 | 2kul | A | 19 | - | Human | 4906 | |
| VRK1 | VRK | CK1 | 6btw | B | B | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9411 | |
| VRK1 | VRK | CK1 | 5uvf | A | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7521 | |
| VRK1 | VRK | CK1 | 6cnx | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9810 | |
| VRK1 | VRK | CK1 | 6cmm | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9759 | |
| VRK1 | VRK | CK1 | 3op5 | A | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4870 | |
| VRK1 | VRK | CK1 | 2lav | A | 13 | - | Human | 4872 | |
| VRK1 | VRK | CK1 | 2kty | A | 1 | - | Human | 4877 | |
| VRK1 | VRK | CK1 | 6bp0 | C | B | - | Human | 8742 | |
| VRK1 | VRK | CK1 | 2kul | A | 10 | - | Human | 4901 | |
| VRK1 | VRK | CK1 | 6dd4 | A | A | - | Human | 9935 | |
| VRK1 | VRK | CK1 | 6cfm | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9722 | |
| VRK1 | VRK | CK1 | 6bp0 | A | A | - | Human | 8744 | |
| VRK1 | VRK | CK1 | 6btw | A | B | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9425 | |
| VRK1 | VRK | CK1 | 5ukf | B | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8029 | |
| VRK1 | VRK | CK1 | 6csw | D | B | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9809 | |
| VRK1 | VRK | CK1 | 2kul | A | 7 | - | Human | 4908 | |
| VRK1 | VRK | CK1 | 6cmm | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9764 | |
| VRK1 | VRK | CK1 | 6csw | B | B | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9808 | |
| VRK1 | VRK | CK1 | 6cqh | C | A | - | Human | 9772 | |
| VRK1 | VRK | CK1 | 2kul | A | 9 | - | Human | 4869 | |
| VRK1 | VRK | CK1 | 2kul | A | 3 | - | Human | 4895 | |
| VRK1 | VRK | CK1 | 2kul | A | 11 | - | Human | 4923 | |
| VRK1 | VRK | CK1 | 2lav | A | 9 | - | Human | 4945 | |
| TTBK2 | TTBK | CK1 | 6vrf | B | A | adenosine-5'-diphosphate | Human | 12345 | |
| VRK1 | VRK | CK1 | 2lav | A | 7 | - | Human | 4936 | |
| VRK1 | VRK | CK1 | 2lav | A | 16 | - | Human | 4888 | |
| VRK1 | VRK | CK1 | 6dd4 | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9938 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | A | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | 6527 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | D | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7539 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4hnf | B | | 3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 2193 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izt | A | B | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 2215 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | B | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7542 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih6 | A | A | 6-(3-bromophenyl)pteridine-2,4,7-triamine | Human | 6535 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4twc | B | A | 2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamide | Human | 2170 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | B | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9860 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6gzm | B | A | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10423 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbc | B | A | {4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanol | Human | 2153 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | C | A | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2169 | |
| VRK1 | VRK | CK1 | 2kul | A | 4 | - | Human | 4948 | |
| VRK1 | VRK | CK1 | 6csw | A | B | - | Human | 9813 | |
| VRK1 | VRK | CK1 | 5ukf | A | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8030 | |
| VRK1 | VRK | CK1 | 6dd4 | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9937 | |
| VRK1 | VRK | CK1 | 2lav | A | 11 | - | Human | 4916 | |
| VRK1 | VRK | CK1 | 5uvf | C | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7520 | |
| VRK1 | VRK | CK1 | 6cfm | C | B | - | Human | 9720 | |
| VRK1 | VRK | CK1 | 6bu6 | A | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9423 | |
| VRK1 | VRK | CK1 | 5uvf | B | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7523 | |
| VRK1 | VRK | CK1 | 6ac9 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 10818 | |
| VRK1 | VRK | CK1 | 6cnx | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9806 | |
| VRK1 | VRK | CK1 | 2kul | A | 5 | - | Human | 4954 | |
| VRK1 | VRK | CK1 | 2lav | A | 8 | - | Human | 4881 | |
| VRK1 | VRK | CK1 | 6bru | D | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9083 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | A | A | adenosine-5'-diphosphate | Human | 12258 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru7 | B | A | adenosine-5'-diphosphate | Human | 12252 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | A | A | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2151 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uys | A | | - | Human | 2183 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | C | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8175 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbc | B | B | {4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanol | Human | 2150 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | C | A | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2172 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru7 | B | B | adenosine-5'-diphosphate | Human | 12263 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | A | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7534 | |
| VRK2 | VRK | CK1 | 2v62 | B | B | - | Human | 2631 | |
| VRK1 | VRK | CK1 | 2lav | A | 5 | - | Human | 4891 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qr9 | A | A | 4-[5-(4-fluorophenyl)-3-(pyridin-4-ylmethyl)imidazol-4-yl]-1~{h}-pyrrolo[2,3-b]pyridine | Human | 14579 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qrb | A | B | 3-(dimethylamino)-~{n}-[4-[4-(4-fluorophenyl)-5-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)imidazol-1-yl]cyclohexyl]propane-1-sulfonamide | Human | 14576 | |
| TTBK1 | TTBK | CK1 | 7zhn | A | A | 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol | Human | 14721 | |
| TTBK1 | TTBK | CK1 | 7zhn | A | B | 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol | Human | 14717 | |
| VRK1 | VRK | CK1 | 6cnx | C | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9805 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qra | A | | 4-[3-cyclohexyl-5-(4-fluorophenyl)imidazol-4-yl]-1~{h}-pyrrolo[2,3-b]pyridine | Human | 14578 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qrb | A | A | 3-(dimethylamino)-~{n}-[4-[4-(4-fluorophenyl)-5-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)imidazol-1-yl]cyclohexyl]propane-1-sulfonamide | Human | 14580 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7qr9 | A | B | 4-[5-(4-fluorophenyl)-3-(pyridin-4-ylmethyl)imidazol-4-yl]-1~{h}-pyrrolo[2,3-b]pyridine | Human | 14577 | |
| VRK1 | VRK | CK1 | 3op5 | D | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4878 | |
| VRK1 | VRK | CK1 | 3op5 | B | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4944 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4hnf | A | | 3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 2194 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | B | B | n-benzyl-4-(pyridin-3-yl)pyrimidin-2-amine | Human | 2147 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | B | A | - | Human | 12106 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxo | B | B | - | Human | 11975 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7h | A | | adenosine monophosphate | Human | 14184 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | D | A | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2160 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | C | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7535 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | B | A | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10958 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | A | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8177 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7f | A | B | adenosine monophosphate | Human | 14185 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmp | B | A | - | Human | 11607 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7g | A | A | adenosine monophosphate | Human | 14187 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxp | B | | - | Human | 11973 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | A | A | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10955 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | C | B | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2165 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | A | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9862 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | A | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8174 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmp | A | A | - | Human | 11608 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | D | A | n-benzyl-4-(pyridin-3-yl)pyrimidin-2-amine | Human | 2146 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmr | B | B | - | Human | 11611 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | A | B | adenosine-5'-diphosphate | Human | 12255 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | E | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7538 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9siw | A | B | 6-(4-fluorophenyl)-3-piperazin-1-yl-5-pyridin-4-yl-pyrazin-2-amine | Human | 15452 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | C | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | 6526 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | A | B | 1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamine | Human | 2161 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9sj0 | A | B | ~{n}2-(2-azanylethyl)-5-(4-fluorophenyl)-6-pyridin-4-yl-pyrazine-2,3-diamine | Human | 15453 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9sj0 | A | A | ~{n}2-(2-azanylethyl)-5-(4-fluorophenyl)-6-pyridin-4-yl-pyrazine-2,3-diamine | Human | 15454 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9six | A | C | 6-(4-fluorophenyl)-3-(4-methylpiperazin-1-yl)-5-pyridin-4-yl-pyrazin-2-amine | Human | 15455 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9six | A | B | 6-(4-fluorophenyl)-3-(4-methylpiperazin-1-yl)-5-pyridin-4-yl-pyrazin-2-amine | Human | 15456 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9siy | A | B | 3-(tetrahydro-1,4-oxazin-4-yl)-6-(4-fluorophenyl)-5-pyridin-4-yl-pyrazin-2-amine | Human | 15457 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9siz | A | B | 5-(4-fluorophenyl)-~{n}2-piperidin-4-yl-6-pyridin-4-yl-pyrazine-2,3-diamine | Human | 15468 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 10ji | B | A | - | Human | 15505 | |
| VRK1 | VRK | CK1 | 6bru | C | B | - | Human | 9086 | |
| VRK1 | VRK | CK1 | 2kty | A | 14 | - | Human | 4926 | |
| VRK1 | VRK | CK1 | 2kty | A | 13 | - | Human | 4922 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 10jk | B | B | - | Human | 15503 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 10ji | B | B | - | Human | 15504 | |
| VRK1 | VRK | CK1 | 2lav | A | 12 | - | Human | 4946 | |
| VRK1 | VRK | CK1 | 6bp0 | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8739 | |
| VRK1 | VRK | CK1 | 6bu6 | D | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9413 | |
| VRK1 | VRK | CK1 | 6npn | B | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11244 | |
| VRK1 | VRK | CK1 | 3op5 | C | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4886 | |
| VRK1 | VRK | CK1 | 6cnx | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9814 | |
| VRK1 | VRK | CK1 | 5ukf | C | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8027 | |
| VRK1 | VRK | CK1 | 2kul | A | 2 | - | Human | 4921 | |
| VRK1 | VRK | CK1 | 6cqh | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9771 | |
| VRK1 | VRK | CK1 | 5ukf | D | | 4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}benzene-1-sulfonamide | Human | 8028 | |
| VRK1 | VRK | CK1 | 6vzh | D | | (7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-one | Human | 12055 | |
| VRK1 | VRK | CK1 | 6dd4 | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9934 | |
| VRK1 | VRK | CK1 | 6csw | C | A | - | Human | 9816 | |
| VRK1 | VRK | CK1 | 2kul | A | 17 | - | Human | 4893 | |
| VRK1 | VRK | CK1 | 2lav | A | 18 | - | Human | 4927 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 5fqd | C | | - | Human | 6415 | |
| VRK1 | VRK | CK1 | 2kty | A | 5 | - | Human | 4900 | |
| VRK1 | VRK | CK1 | 2rsv | A | 12 | - | Human | 4952 | |
| VRK2 | VRK | CK1 | 9fet | A | | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 15788 | |
| VRK1 | VRK | CK1 | 6bu6 | C | B | - | Human | 9414 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 30ix | A | B | - | Human | 16059 | |
| CSNK1G2 (CK1g2) | CK1 | CK1 | 30ix | A | A | - | Human | 16060 | |
| VRK1 | VRK | CK1 | 9zkg | A | A | - | Human | 16122 | |
| VRK1 | VRK | CK1 | 2lav | A | 1 | - | Human | 4930 | |
| VRK1 | VRK | CK1 | 6bru | A | A | - | Human | 9085 | |
| VRK1 | VRK | CK1 | 6bu6 | D | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9410 | |
| VRK1 | VRK | CK1 | 3op5 | D | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4892 | |
| VRK1 | VRK | CK1 | 6csw | C | B | - | Human | 9811 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8izc | A | B | ~{n}5-~{tert}-butyl-2-(3-chloranyl-4-fluoranyl-phenyl)-6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazine-3,5-dicarboxamide | Human | 15269 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8izc | A | A | ~{n}5-~{tert}-butyl-2-(3-chloranyl-4-fluoranyl-phenyl)-6,7-dihydro-4~{h}-pyrazolo[1,5-a]pyrazine-3,5-dicarboxamide | Human | 15270 | |
| VRK3 | VRK | CK1 | 2jii | A | B | - | Human | 2938 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tw9 | A | A | octyl beta-l-talopyranoside | Human | 2143 | |
| VRK1 | VRK | CK1 | 2kty | A | 18 | - | Human | 4904 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | F | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7536 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7g | A | B | adenosine monophosphate | Human | 14186 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | D | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9856 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | D | B | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2145 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | B | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8179 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tw9 | B | A | n-(2,2-difluoro-5h-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-2-{[2-(trifluoromethoxy)benzoyl]amino}-1,3-thiazole-4-carboxamide | Human | 2178 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9six | A | A | 6-(4-fluorophenyl)-3-(4-methylpiperazin-1-yl)-5-pyridin-4-yl-pyrazin-2-amine | Human | 15458 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | A | B | ~{n}-[[4,5-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-naphthalen-2-yl-purin-6-amine | Human | 12107 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru6 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 12256 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | D | B | adenosine-5'-diphosphate | Human | 12257 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | D | B | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2142 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | B | C | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10952 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | A | C | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10954 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | A | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9861 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9b3s | A | A | - | Human | 15460 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uyt | C | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2152 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih6 | A | B | 6-(3-bromophenyl)pteridine-2,4,7-triamine | Human | 6532 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9siy | A | A | 3-(tetrahydro-1,4-oxazin-4-yl)-6-(4-fluorophenyl)-5-pyridin-4-yl-pyrazin-2-amine | Human | 15461 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | C | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9859 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | D | B | n-benzyl-4-(pyridin-3-yl)pyrimidin-2-amine | Human | 2188 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | A | C | ~{n}-[[4,5-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-naphthalen-2-yl-purin-6-amine | Human | 12111 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | A | A | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2192 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | A | B | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2141 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | A | B | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10953 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6gzm | A | B | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10425 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | C | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8178 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | C | B | 1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamine | Human | 2164 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tw9 | A | B | octyl beta-l-talopyranoside | Human | 2155 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih4 | A | B | - | Human | 6534 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rcg | A | A | ~{n}-[[6,7-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(3-fluorophenyl)-2-morpholin-4-yl-purin-6-amine | Human | 12112 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | B | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | 6533 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih4 | A | A | - | Human | 6530 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f1w | A | A | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10959 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tw9 | B | B | n-(2,2-difluoro-5h-[1,3]dioxolo[4,5-f]benzimidazol-6-yl)-2-{[2-(trifluoromethoxy)benzoyl]amino}-1,3-thiazole-4-carboxamide | Human | 2167 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmr | B | A | - | Human | 11605 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxo | A | B | - | Human | 11976 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4hgt | A | | 2-{2-[(3,4-difluorophenoxy)methyl]-5-methoxypyridin-4-yl}-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 2181 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | D | B | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8180 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | B | B | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9857 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f1w | B | B | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10961 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9siw | A | A | 6-(4-fluorophenyl)-3-piperazin-1-yl-5-pyridin-4-yl-pyrazin-2-amine | Human | 15463 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uyt | D | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2163 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9sj1 | A | B | 6-(4-fluorophenyl)-5-pyridin-4-yl-pyrazin-2-amine | Human | 15464 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7p7f | A | A | adenosine monophosphate | Human | 14188 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9siv | A | B | 6-(4-fluorophenyl)-5-pyridin-4-yl-pyrazin-2-amine | Human | 15465 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | B | B | - | Human | 12110 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxn | A | A | - | Human | 11972 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | C | A | adenosine-5'-diphosphate | Human | 12266 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | B | A | adenosine-5'-diphosphate | Human | 12265 | |
| VRK1 | VRK | CK1 | 2rsv | A | 5 | - | Human | 4899 | |
| VRK1 | VRK | CK1 | 6dd4 | C | A | - | Human | 9940 | |
| VRK1 | VRK | CK1 | 6cfm | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9725 | |
| VRK1 | VRK | CK1 | 6bp0 | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8740 | |
| VRK1 | VRK | CK1 | 2kty | A | 4 | - | Human | 4938 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 6gzd | A | B | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10561 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 5fqd | F | | - | Human | 6416 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 6gzd | A | A | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10560 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 9oty | C | | - | Human | 15502 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 10jk | B | A | - | Human | 15506 | |
| VRK1 | VRK | CK1 | 6cqh | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9767 | |
| VRK1 | VRK | CK1 | 6cfm | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9721 | |
| VRK1 | VRK | CK1 | 2lav | A | 14 | - | Human | 4898 | |
| VRK1 | VRK | CK1 | 6ac9 | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 10822 | |
| VRK1 | VRK | CK1 | 2lav | A | 19 | - | Human | 4940 | |
| VRK1 | VRK | CK1 | 2kul | A | 12 | - | Human | 4883 | |
| VRK1 | VRK | CK1 | 6vxu | B | | (7r)-8-(cyclopropylmethyl)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 13362 | |
| VRK1 | VRK | CK1 | 6cfm | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9723 | |
| VRK1 | VRK | CK1 | 2lav | A | 6 | - | Human | 4871 | |
| VRK1 | VRK | CK1 | 6cnx | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9803 | |
| VRK1 | VRK | CK1 | 6cnx | C | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9804 | |
| VRK1 | VRK | CK1 | 5uvf | D | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7522 | |
| VRK1 | VRK | CK1 | 6cmm | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9761 | |
| VRK1 | VRK | CK1 | 6ac9 | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 10819 | |
| VRK1 | VRK | CK1 | 2rsv | A | 3 | - | Human | 4913 | |
| VRK1 | VRK | CK1 | 2kul | A | 14 | - | Human | 4909 | |
| VRK1 | VRK | CK1 | 6dd4 | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-dipropyl-7,8-dihydropteridin-6(5h)-one | Human | 9933 | |
| VRK1 | VRK | CK1 | 6cmm | A | B | - | Human | 9760 | |
| VRK1 | VRK | CK1 | 6ac9 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 10817 | |
| VRK1 | VRK | CK1 | 6bp0 | D | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8745 | |
| VRK1 | VRK | CK1 | 3op5 | C | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4879 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmr | A | B | - | Human | 11606 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rcg | A | B | ~{n}-[[6,7-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(3-fluorophenyl)-2-morpholin-4-yl-purin-6-amine | Human | 12109 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | B | B | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2175 | |
| VRK1 | VRK | CK1 | 2kty | A | 3 | - | Human | 4874 | |
| VRK1 | VRK | CK1 | 6btw | C | A | - | Human | 9419 | |
| VRK1 | VRK | CK1 | 6cmm | C | A | - | Human | 9765 | |
| VRK1 | VRK | CK1 | 6vzh | B | | (7~{r})-2-[[3,5-bis(fluoranyl)-4-oxidanyl-phenyl]amino]-5,7-dimethyl-8-prop-2-ynyl-7~{h}-pteridin-6-one | Human | 12056 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8d7n | A | | - | Human | 14738 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8d7o | A | | - | Human | 14739 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8d7m | A | | - | Human | 14740 | |
| VRK1 | VRK | CK1 | 6bp0 | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 8741 | |
| CSNK1D (CK1d) | CK1 | CK1 | 8d7p | A | | - | Human | 14737 | |
| VRK1 | VRK | CK1 | 2kty | A | 8 | - | Human | 4939 | |
| VRK1 | VRK | CK1 | 6npn | A | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11243 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uyt | B | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2166 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | C | B | adenosine-5'-diphosphate | Human | 12254 | |
| CSNK1A1 (CK1a) | CK1 | CK1 | 8g66 | C | | - | Human | 15006 | |
| VRK1 | VRK | CK1 | 2lav | A | 17 | - | Human | 4950 | |
| VRK1 | VRK | CK1 | 2lav | A | 10 | - | Human | 4882 | |
| VRK1 | VRK | CK1 | 6bu6 | B | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9422 | |
| VRK1 | VRK | CK1 | 2rsv | A | 7 | - | Human | 4889 | |
| VRK1 | VRK | CK1 | 6bu6 | C | A | - | Human | 9412 | |
| VRK1 | VRK | CK1 | 2rsv | A | 17 | - | Human | 4951 | |
| VRK1 | VRK | CK1 | 6bu6 | A | B | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9417 | |
| VRK1 | VRK | CK1 | 6cmm | A | A | - | Human | 9763 | |
| VRK1 | VRK | CK1 | 6cqh | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9768 | |
| VRK1 | VRK | CK1 | 6bru | C | A | - | Human | 9089 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru6 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 12251 | |
| VRK1 | VRK | CK1 | 2rsv | A | 2 | - | Human | 4914 | |
| VRK1 | VRK | CK1 | 2kty | A | 15 | - | Human | 4953 | |
| VRK1 | VRK | CK1 | 2kty | A | 12 | - | Human | 4897 | |
| VRK1 | VRK | CK1 | 2rsv | A | 14 | - | Human | 4925 | |
| VRK1 | VRK | CK1 | 2rsv | A | 18 | - | Human | 4934 | |
| VRK1 | VRK | CK1 | 6csw | B | A | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9812 | |
| VRK1 | VRK | CK1 | 3op5 | B | A | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4894 | |
| VRK1 | VRK | CK1 | 2rsv | A | 6 | - | Human | 4943 | |
| VRK1 | VRK | CK1 | 2lav | A | 2 | - | Human | 4903 | |
| VRK1 | VRK | CK1 | 6npn | C | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11241 | |
| VRK1 | VRK | CK1 | 2kty | A | 10 | - | Human | 4932 | |
| VRK1 | VRK | CK1 | 6csw | A | A | - | Human | 9818 | |
| VRK1 | VRK | CK1 | 6bru | A | B | - | Human | 9082 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hni | A | | 3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 1722 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | I | | - | Human | 1724 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru7 | A | B | adenosine-5'-diphosphate | Human | 12253 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih4 | A | C | - | Human | 6529 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbc | A | B | {4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanol | Human | 2156 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih5 | A | D | 6-(3-chlorophenyl)pteridine-2,4,7-triamine | Human | 6528 | |
| VRK1 | VRK | CK1 | 6cfm | A | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9718 | |
| VRK1 | VRK | CK1 | 6dd4 | C | B | - | Human | 9936 | |
| TTBK1 | TTBK | CK1 | 7jxx | A | A | 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol | Human | 13579 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxn | A | B | - | Human | 11977 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | E | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7543 | |
| VRK3 | VRK | CK1 | 2jii | B | B | - | Human | 2937 | |
| VRK3 | VRK | CK1 | 2jii | B | A | - | Human | 2936 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | D | A | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2190 | |
| VRK1 | VRK | CK1 | 6btw | D | B | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9420 | |
| VRK1 | VRK | CK1 | 3op5 | A | B | [4-({4-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4942 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | A | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7532 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | D | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8176 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 6gro | A | A | 4-[5-(2-azanylpyrimidin-4-yl)-4-(4-fluorophenyl)imidazol-1-yl]cyclohexan-1-ol | Human | 10002 | |
| CSNK1G3 (CK1g3) | CK1 | CK1 | 2izr | A | A | {(2z)-4-amino-2-[(4-methoxyphenyl)imino]-2,3-dihydro-1,3-thiazol-5-yl}(4-methoxyphenyl)methanone | Human | 2222 | |
| VRK1 | VRK | CK1 | 6bru | B | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9088 | |
| VRK1 | VRK | CK1 | 2kul | A | 20 | - | Human | 4915 | |
| VRK1 | VRK | CK1 | 2rsv | A | 8 | - | Human | 4918 | |
| VRK1 | VRK | CK1 | 2lav | A | 3 | - | Human | 4912 | |
| TTBK1 | TTBK | CK1 | 7q8v | A | | ~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14133 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | C | A | 1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamine | Human | 2189 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tn6 | B | B | - | Human | 2162 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9b3s | A | B | - | Human | 15462 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | D | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7537 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | D | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9855 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | C | A | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7541 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxn | B | B | - | Human | 11978 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f1w | B | A | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10960 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uyt | A | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2182 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kba | B | A | 9-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-2,3,4,5-tetrahydropyrido[2,3-f][1,4]oxazepine | Human | 2191 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5w4w | B | A | 4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]-6-methyl-6,7-dihydro-5h-pyrrolo[3,4-b]pyridin-5-one | Human | 8173 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru6 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 12259 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9siv | A | A | 6-(4-fluorophenyl)-5-pyridin-4-yl-pyrazin-2-amine | Human | 15459 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmp | B | B | - | Human | 11610 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | A | B | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2176 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tn6 | A | A | 4-{4-(4-fluorophenyl)-1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1h-imidazol-5-yl}pyrimidin-2-amine | Human | 2168 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru6 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 12260 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmr | A | A | - | Human | 11612 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxp | A | | - | Human | 11970 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4twc | B | B | 2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamide | Human | 2144 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f1w | A | B | (9~{r},10~{r},11~{s})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10957 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxn | B | A | - | Human | 11969 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6gzm | A | A | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10426 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxo | A | A | - | Human | 11971 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7nzy | A | A | 9-chloranyl-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine | Human | 14381 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbc | A | A | {4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-yl}methanol | Human | 2154 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6hmp | A | B | - | Human | 11609 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | B | C | - | Human | 12113 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uzp | B | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2177 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | A | A | 1-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}-n-methylmethanamine | Human | 2171 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4twc | A | A | 2-{[2-(trifluoromethoxy)benzoyl]amino}-n-[6-(trifluoromethyl)-1h-benzimidazol-2-yl]-1,3-thiazole-4-carboxamide | Human | 2185 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5okt | C | A | ~{n}-(6-methyl-1,3-benzothiazol-2-yl)-2-[(4-oxidanylidene-3-phenyl-6,7-dihydrothieno[3,2-d]pyrimidin-2-yl)sulfanyl]ethanamide | Human | 9858 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uys | D | | - | Human | 2180 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6gzm | B | B | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10424 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | B | B | adenosine-5'-diphosphate | Human | 12261 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kbk | B | B | (3s)-3-{4-[3-(4-fluorophenyl)-1-methyl-1h-pyrazol-4-yl]pyridin-2-yl}morpholine | Human | 2187 | |
| CSNK1D (CK1d) | CK1 | CK1 | 7nzy | A | B | 9-chloranyl-2-(furan-2-yl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine | Human | 14382 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6pxo | B | A | - | Human | 11974 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uys | B | | - | Human | 2159 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uzp | A | | 4-[1-cyclohexyl-4-(4-fluorophenyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 2158 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tn6 | B | A | - | Human | 2173 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6f26 | B | B | (9~{s},10~{s},11~{r})-~{n}-[4-[3-(4-fluorophenyl)-5-propan-2-yl-1,2-oxazol-4-yl]pyridin-2-yl]-4-(4-methoxyphenyl)-10,11-bis(oxidanyl)-1,7-diazatricyclo[7.3.0.0^{3,7}]dodeca-3,5-diene-6-carboxamide | Human | 10956 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4kb8 | B | A | n-benzyl-4-(pyridin-3-yl)pyrimidin-2-amine | Human | 2148 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | B | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7540 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4tn6 | A | B | 4-{4-(4-fluorophenyl)-1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1h-imidazol-5-yl}pyrimidin-2-amine | Human | 2186 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5ih4 | A | D | - | Human | 6531 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9siz | A | A | 5-(4-fluorophenyl)-~{n}2-piperidin-4-yl-6-pyridin-4-yl-pyrazine-2,3-diamine | Human | 15466 | |
| CSNK1D (CK1d) | CK1 | CK1 | 4hgt | B | | 2-{2-[(3,4-difluorophenoxy)methyl]-5-methoxypyridin-4-yl}-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 2179 | |
| CSNK1D (CK1d) | CK1 | CK1 | 9sj1 | A | A | 6-(4-fluorophenyl)-5-pyridin-4-yl-pyrazin-2-amine | Human | 15467 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru8 | D | A | adenosine-5'-diphosphate | Human | 12262 | |
| CSNK1D (CK1d) | CK1 | CK1 | 3uys | C | | - | Human | 2149 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6ru7 | A | A | adenosine-5'-diphosphate | Human | 12264 | |
| CSNK1D (CK1d) | CK1 | CK1 | 6rch | A | A | ~{n}-[[4,5-bis(fluoranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-naphthalen-2-yl-purin-6-amine | Human | 12108 | |
| CSNK1D (CK1d) | CK1 | CK1 | 5mqv | F | B | 4-(2,5-dimethoxyphenyl)-n-(4-(5-(4-fluorphenyl)-2-(methylthio)-1h-imidazol-4-yl)-pyridin-2-yl)-1-methyl-1h-pyrrole-2-carboxamide | Human | 7533 | |
| VRK3 | VRK | CK1 | 2jii | A | A | - | Human | 2939 | |
| VRK1 | VRK | CK1 | 2rsv | A | 13 | - | Human | 4935 | |
| VRK1 | VRK | CK1 | 2kul | A | 6 | - | Human | 4949 | |
| VRK1 | VRK | CK1 | 6bp0 | A | B | - | Human | 8738 | |
| VRK2 | VRK | CK1 | 5uu1 | A | | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(3-methylbutyl)-7,8-dihydropteridin-6(5h)-one | Human | 7499 | |
| VRK2 | VRK | CK1 | 2v62 | A | B | - | Human | 2629 | |
| VRK2 | VRK | CK1 | 6ncg | B | | 4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamide | Human | 10851 | |
| VRK2 | VRK | CK1 | 2v62 | B | A | - | Human | 2630 | |
| VRK2 | VRK | CK1 | 8q1z | A | B | 2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrile | Human | 14898 | |
| VRK2 | VRK | CK1 | 2v62 | A | A | - | Human | 2628 | |
| VRK2 | VRK | CK1 | 8q1z | A | A | 2-[4-[[4-[(3-~{tert}-butyl-1~{h}-pyrazol-5-yl)amino]pyrimidin-2-yl]amino]phenyl]ethanenitrile | Human | 14899 | |
| VRK2 | VRK | CK1 | 6ncg | A | | 4-[6-amino-5-(3,5-difluoro-4-hydroxyphenyl)pyridin-3-yl]benzene-1-sulfonamide | Human | 10852 | |
| TTBK1 | TTBK | CK1 | 4nfn | A | B | 3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenol | Human | 770 | |
| TTBK1 | TTBK | CK1 | 31ho | A | | ~{n}-[4-(furan-2-yl)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 15850 | |
| TTBK1 | TTBK | CK1 | 7jxx | A | B | 4-(2-amino-5,6,7,8-tetrahydropyrimido[4',5':3,4]cyclohepta[1,2-b]indol-11-yl)-2-methylbut-3-yn-2-ol | Human | 13578 | |
| TTBK1 | TTBK | CK1 | 4nfn | A | A | 3-({5-[(4-amino-4-methylpiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-bromophenol | Human | 773 | |
| TTBK1 | TTBK | CK1 | 7qhw | A | | ~{n}-[4-(4-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14477 | |
| TTBK1 | TTBK | CK1 | 7zho | A | A | 4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-ol | Human | 14718 | |
| TTBK1 | TTBK | CK1 | 7zhp | A | B | 1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-ol | Human | 14719 | |
| TTBK1 | TTBK | CK1 | 7zhq | A | A | (3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-ol | Human | 14720 | |
| TTBK1 | TTBK | CK1 | 4btm | B | | methyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoate | Human | 774 | |
| TTBK1 | TTBK | CK1 | 4btm | A | | methyl 2-bromo-5-(7h-pyrrolo[2,3-d]pyrimidin-4-ylamino)benzoate | Human | 772 | |
| TTBK1 | TTBK | CK1 | 7jxy | A | | (3s)-1-[1-(2-aminopyrimidin-4-yl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-methylpent-1-yn-3-ol | Human | 13580 | |
| TTBK1 | TTBK | CK1 | 7zho | A | B | 4-[3-(2-azanylpyrimidin-4-yl)-1~{h}-indol-5-yl]-2-methyl-but-3-yn-2-ol | Human | 14722 | |
| TTBK1 | TTBK | CK1 | 7zhq | A | B | (3~{s})-1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-methyl-pent-1-yn-3-ol | Human | 14723 | |
| TTBK1 | TTBK | CK1 | 4btj | A | | adenosine-5'-diphosphate | Human | 769 | |
| TTBK1 | TTBK | CK1 | 7zhp | A | A | 1-(4-azanyl-3,5,12-triazatetracyclo[9.7.0.0^{2,7}.0^{13,18}]octadeca-1(11),2,4,6,13(18),14,16-heptaen-16-yl)-3-ethyl-pent-1-yn-3-ol | Human | 14724 | |
| TTBK1 | TTBK | CK1 | 4btj | B | | adenosine-5'-triphosphate | Human | 767 | |
| TTBK1 | TTBK | CK1 | 7q8w | A | A | ~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14134 | |
| TTBK1 | TTBK | CK1 | 4nfm | A | | - | Human | 768 | |
| TTBK1 | TTBK | CK1 | 7q8w | A | B | ~{n}-(4-methoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14135 | |
| TTBK1 | TTBK | CK1 | 4btk | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 771 | |
| TTBK1 | TTBK | CK1 | 8xpz | A | | - | Human | 15163 | |
| CSNK1G1 (CK1g1) | CK1 | CK1 | 2cmw | A | B | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 5566 | |
| CSNK1G1 (CK1g1) | CK1 | CK1 | 2cmw | A | A | 2-(2-hydroxyethylamino)-6-(3-chloroanilino)-9-isopropylpurine | Human | 5567 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | W | | - | Human | 1728 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | M | | - | Human | 1727 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | U | | - | Human | 1725 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | E | | - | Human | 1720 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hni | B | | 3-[(3-chlorophenoxy)methyl]-1-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-4-amine | Human | 1731 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | A | | - | Human | 1718 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | Q | | - | Human | 1730 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | C | | - | Human | 1723 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | K | | - | Human | 1729 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | G | | - | Human | 1719 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | S | | - | Human | 1721 | |
| CSNK1E (CK1e) | CK1 | CK1 | 4hok | O | | - | Human | 1726 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12049 | |
| TTBK2 | TTBK | CK1 | 6vrf | B | B | adenosine-5'-diphosphate | Human | 12342 | |
| TTBK2 | TTBK | CK1 | 6vrf | A | B | adenosine-5'-diphosphate | Human | 12343 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | A | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12046 | |
| TTBK2 | TTBK | CK1 | 7q8y | A | B | ~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14138 | |
| TTBK2 | TTBK | CK1 | 7q90 | A | A | ~{n}-[4-(4-methoxyphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14139 | |
| TTBK2 | TTBK | CK1 | 6vrf | A | A | adenosine-5'-diphosphate | Human | 12344 | |
| TTBK2 | TTBK | CK1 | 7q8z | A | B | ~{n}-(4-phenoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14140 | |
| TTBK2 | TTBK | CK1 | 6u0k | B | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12047 | |
| TTBK2 | TTBK | CK1 | 7q8y | A | A | ~{n}-[4-(2-chloranylphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14141 | |
| TTBK2 | TTBK | CK1 | 7q8z | A | A | ~{n}-(4-phenoxyphenyl)-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14142 | |
| TTBK2 | TTBK | CK1 | 6u0k | A | B | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 12048 | |
| TTBK2 | TTBK | CK1 | 7q90 | A | B | ~{n}-[4-(4-methoxyphenoxy)phenyl]-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 14143 | |
| VRK1 | VRK | CK1 | 2kty | A | 17 | - | Human | 4920 | |
| VRK1 | VRK | CK1 | 2lav | A | 4 | - | Human | 4884 | |
| VRK1 | VRK | CK1 | 6cnx | D | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9807 | |
| VRK1 | VRK | CK1 | 6npn | D | | (7r)-7-methyl-2-[(3-oxo-2,3-dihydro-1h-indazol-6-yl)amino]-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 11242 | |
| VRK1 | VRK | CK1 | 6cqh | C | B | - | Human | 9773 | |
| VRK1 | VRK | CK1 | 2kul | A | 13 | - | Human | 4941 | |
| VRK1 | VRK | CK1 | 2kty | A | 9 | - | Human | 4885 | |
| VRK1 | VRK | CK1 | 2kty | A | 7 | - | Human | 4880 | |
| VRK1 | VRK | CK1 | 2lav | A | 20 | - | Human | 4933 | |
| VRK1 | VRK | CK1 | 2rsv | A | 16 | - | Human | 4905 | |
| VRK1 | VRK | CK1 | 2kul | A | 8 | - | Human | 4887 | |
| VRK1 | VRK | CK1 | 6ac9 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 10823 | |
| VRK1 | VRK | CK1 | 6btw | A | A | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9418 | |
| VRK1 | VRK | CK1 | 9zkg | A | B | - | Human | 16121 | |
| VRK1 | VRK | CK1 | 6cqh | B | B | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9770 | |
| VRK1 | VRK | CK1 | 6cqh | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9769 | |
| VRK1 | VRK | CK1 | 2kul | A | 18 | - | Human | 4896 | |
| VRK1 | VRK | CK1 | 6bru | D | A | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9084 | |
| VRK1 | VRK | CK1 | 6bp0 | C | A | - | Human | 8743 | |
| VRK1 | VRK | CK1 | 2kty | A | 11 | - | Human | 4917 | |
| VRK1 | VRK | CK1 | 6cfm | C | A | - | Human | 9719 | |
| VRK1 | VRK | CK1 | 6csw | D | A | (7r)-5-butyl-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7,8-dimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9817 | |
| VRK1 | VRK | CK1 | 6cmm | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-5,8-di(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9766 | |
| VRK1 | VRK | CK1 | 2kty | A | 16 | - | Human | 4937 | |
| VRK1 | VRK | CK1 | 6cnx | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-7-methyl-8-(3-methylbutyl)-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9815 | |
| VRK1 | VRK | CK1 | 6cfm | B | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimethyl-8-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9724 | |
| VRK1 | VRK | CK1 | 2rsv | A | 10 | - | Human | 4873 | |
| VRK1 | VRK | CK1 | 2rsv | A | 9 | - | Human | 4928 | |
| VRK1 | VRK | CK1 | 2kul | A | 15 | - | Human | 4876 | |
| VRK1 | VRK | CK1 | 2kul | A | 16 | - | Human | 4924 | |
| VRK1 | VRK | CK1 | 6ac9 | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 10821 | |
| VRK1 | VRK | CK1 | 2rsv | A | 11 | - | Human | 4902 | |
| VRK1 | VRK | CK1 | 2kul | A | 1 | - | Human | 4919 | |
| VRK1 | VRK | CK1 | 2kty | A | 6 | - | Human | 4929 | |
| VRK1 | VRK | CK1 | 2rsv | A | 4 | - | Human | 4907 | |
| VRK1 | VRK | CK1 | 6btw | D | A | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9415 | |
| VRK1 | VRK | CK1 | 2rsv | A | 15 | - | Human | 4911 | |
| VRK1 | VRK | CK1 | 6ac9 | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 10820 | |
| VRK1 | VRK | CK1 | 6bru | B | B | (7s)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7,8-trimethyl-7,8-dihydropteridin-6(5h)-one | Human | 9087 | |
| VRK1 | VRK | CK1 | 2kty | A | 2 | - | Human | 4947 | |
| VRK1 | VRK | CK1 | 2kty | A | 19 | - | Human | 4875 | |
| VRK1 | VRK | CK1 | 6btw | C | B | - | Human | 9416 | |
| VRK1 | VRK | CK1 | 2lav | A | 15 | - | Human | 4931 | |
| VRK1 | VRK | CK1 | 2kty | A | 20 | - | Human | 4890 | |
| VRK1 | VRK | CK1 | 6cqh | A | A | (7r)-2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-ethyl-7-methyl-5-(prop-2-yn-1-yl)-7,8-dihydropteridin-6(5h)-one | Human | 9774 | |
| VRK1 | VRK | CK1 | 6vzh | A | | - | Human | 12057 | |
| VRK1 | VRK | CK1 | 6btw | B | A | 2-[(3,5-difluoro-4-hydroxyphenyl)amino]-8-phenyl-7,8-dihydropteridin-6(5h)-one | Human | 9424 | |
| VRK1 | VRK | CK1 | 6cmm | C | B | - | Human | 9762 | |
| VRK1 | VRK | CK1 | 6ac9 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 10816 | |
| VRK1 | VRK | CK1 | 6vzh | C | | - | Human | 12058 | |
| VRK1 | VRK | CK1 | 6bu6 | B | A | 4,4'-(2-aminopyridine-3,5-diyl)bis(2,6-difluorophenol) | Human | 9421 | |
| VRK1 | VRK | CK1 | 2rsv | A | 1 | - | Human | 4910 | |
| TTBK1 | TTBK | CK1 | 9hhw | A | B | ~{n}-[2-(1~{h}-pyrrolo[2,3-b]pyridin-5-yl)phenyl]propanamide | Human | 15851 | |
| TTBK1 | TTBK | CK1 | 9hhw | A | A | ~{n}-[2-(1~{h}-pyrrolo[2,3-b]pyridin-5-yl)phenyl]propanamide | Human | 15852 | |