| CSNK2A1 (CK2a1) | CK2 | CMGC | 8p07 | A | | 7-(cyclopropylamino)-5-[[3-(1,2,4-triazol-4-yl)phenyl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 14743 | |
| CDK2 | CDK | CMGC | 9esp | A | B | 4-bromo-1-(2-methoxyethyl)-1h-pyrazole | Human | 15901 | |
| CDK2 | CDK | CMGC | 2wxv | C | | n,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4504 | |
| CDK2 | CDK | CMGC | 5ano | A | | - | Human | 6537 | |
| CDK2 | CDK | CMGC | 4eop | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4258 | |
| CDK2 | CDK | CMGC | 3rak | A | B | 4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 4331 | |
| CDK2 | CDK | CMGC | 9et2 | A | B | ~{n}-(4-bromophenyl)ethanamide | Human | 15902 | |
| CDK2 | CDK | CMGC | 8ru8 | A | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 15329 | |
| CDK2 | CDK | CMGC | 3unk | A | | 4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acid | Human | 4374 | |
| CDK2 | CDK | CMGC | 2vu3 | A | B | 4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamide | Human | 3884 | |
| SRPK1 | SRPK | CMGC | 1wbp | A | | adenosine-5'-diphosphate | Human | 119 | |
| CDK2 | CDK | CMGC | 1r78 | A | A | 4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one | Human | 4253 | |
| MAPK3 (Erk1) | MAPK | CMGC | 2zoq | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 1716 | |
| CLK3 | CLK | CMGC | 2wu6 | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1823 | |
| GSK3B | GSK | CMGC | 8qji | A | | n-[4-[5-(1,2,4-oxadiazol-3-yl)thiophen-2-yl]pyridin-2-yl]cyclopropanecarboxamide | Human | 15386 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt5 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15306 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pst | A | A | amp phosphoramidate | Human | 15311 | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | A | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | 5212 | |
| CDK2 | CDK | CMGC | 1h00 | A | B | (2r)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | 4428 | |
| DYRK1A | DYRK | CMGC | 6eis | C | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10548 | |
| CDK2 | CDK | CMGC | 2ds1 | A | | (13r,15s)-13-methyl-16-oxa-8,9,12,22,24-pentaazahexacyclo[15.6.2.16,9.1,12,15.0,2,7.0,21,25]heptacosa-1(24),2,4,6,17(25),18,20-heptaene-23,26-dione | Human | 4513 | |
| CDK2 | CDK | CMGC | 4ek5 | A | B | n-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamide | Human | 4145 | |
| CDK2 | CDK | CMGC | 9esz | A | D | 5-iodanylpyrimidine | Human | 15903 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu6 | A | | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 10774 | |
| CDK2 | CDK | CMGC | 2wev | C | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4503 | |
| CDK2 | CDK | CMGC | 6q4f | A | B | pyridine-2,6-diamine | Human | 11211 | |
| CDK2 | CDK | CMGC | 2uzo | A | | 4-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamide | Human | 3862 | |
| DYRK1A | DYRK | CMGC | 2vx3 | C | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3740 | |
| DYRK1A | DYRK | CMGC | 6eiv | B | | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10536 | |
| DYRK1A | DYRK | CMGC | 7a52 | A | B | 3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-one | Human | 13750 | |
| DYRK1A | DYRK | CMGC | 4mq1 | A | B | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3736 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | E | A | - | Human | 4612 | |
| DYRK1A | DYRK | CMGC | 2vx3 | C | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3735 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt0 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15297 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu4 | A | | ~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamine | Human | 10777 | |
| CDK2 | CDK | CMGC | 3s0o | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanone | Human | 4123 | |
| CDK2 | CDK | CMGC | 3qhw | C | B | adenosine-5'-diphosphate | Human | 4143 | |
| CLK2 | CLK | CMGC | 6fyl | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10403 | |
| CLK2 | CLK | CMGC | 6khe | A | | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11651 | |
| CLK2 | CLK | CMGC | 3nr9 | C | | (5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 1929 | |
| CLK2 | CLK | CMGC | 3nr9 | B | | (5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 1928 | |
| CDK2 | CDK | CMGC | 4fx3 | A | B | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 3931 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ooi | A | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9447 | |
| CDK2 | CDK | CMGC | 3qhw | A | B | adenosine-5'-diphosphate | Human | 4156 | |
| CDK2 | CDK | CMGC | 4cfx | A | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4086 | |
| CDK2 | CDK | CMGC | 3qqh | A | A | 2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenol | Human | 4393 | |
| CDK2 | CDK | CMGC | 3rai | A | A | 4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4441 | |
| CDK2 | CDK | CMGC | 3sqq | A | B | 4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 3925 | |
| CDK2 | CDK | CMGC | 6gue | C | | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10772 | |
| CDK2 | CDK | CMGC | 1fvv | A | | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 4065 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ijp | B | B | 4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 5534 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4iir | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5545 | |
| CDK2 | CDK | CMGC | 1pxo | A | B | - | Human | 3860 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ian | A | | - | Human | 5543 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ijp | B | A | 4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 5541 | |
| CDK2 | CDK | CMGC | 3r9h | A | B | 4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4336 | |
| CDK2 | CDK | CMGC | 1e1v | A | | 6-o-cyclohexylmethyl guanine | Human | 3886 | |
| CDK2 | CDK | CMGC | 4bcn | C | A | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4436 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | A | B | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11577 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ifc | A | A | adenosine-5'-diphosphate | Human | 5538 | |
| CLK1 | CLK | CMGC | 6qty | A | A | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 12083 | |
| CDK2 | CDK | CMGC | 4eol | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4089 | |
| CDK2 | CDK | CMGC | 4kd1 | A | A | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 4585 | |
| CDK2 | CDK | CMGC | 4bcp | C | A | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 3872 | |
| CDK2 | CDK | CMGC | 4bcn | A | B | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4298 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4iir | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5539 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | A | A | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11585 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | B | A | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11583 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4iir | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 5537 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ifc | B | B | adenosine-5'-diphosphate | Human | 5540 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | C | B | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11586 | |
| CDK2 | CDK | CMGC | 1h1s | C | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4572 | |
| CDK2 | CDK | CMGC | 3ti1 | A | A | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 4201 | |
| CDK1 (CDC2) | CDK | CMGC | 5hq0 | A | B | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 6421 | |
| CDK2 | CDK | CMGC | 4cfm | A | A | 6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amine | Human | 4207 | |
| CDK2 | CDK | CMGC | 5iev | A | B | roniciclib | Human | 6570 | |
| CDK2 | CDK | CMGC | 4eos | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4008 | |
| CDK2 | CDK | CMGC | 1pxk | A | B | - | Human | 3980 | |
| CDK2 | CDK | CMGC | 3tnw | C | B | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 4493 | |
| CDK2 | CDK | CMGC | 4fks | A | A | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4412 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8bgc | A | | 5-[(phenylmethyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 14545 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmq | A | B | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 10998 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5clp | A | B | 2-(3,4-dichlorophenyl)ethanamine | Human | 6920 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8h | A | B | nicotinic acid | Human | 13259 | |
| CDK8 | CDK | CMGC | 6qtj | A | | ~{n},~{n}-dimethyl-2-[4-[4-(2,6-naphthyridin-4-yl)phenyl]pyrazol-1-yl]ethanamide | Human | 12093 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owl | B | B | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10592 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7x4h | A | A | 5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrile | Human | 14595 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehu | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamine | Human | 9684 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4uba | A | | 4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acid | Human | 5432 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | D | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12116 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8ae7 | A | A | adenosine-5'-diphosphate | Human | 14682 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo6 | A | B | 3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoic acid | Human | 7665 | |
| CDK8 | CDK | CMGC | 5hvy | A | B | n-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}urea | Human | 6552 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | L | | - | Human | 5414 | |
| GSK3B | GSK | CMGC | 3zrl | B | B | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 691 | |
| CDK2 | CDK | CMGC | 1urc | C | A | - | Human | 4006 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moe | B | A | adenosine-5'-diphosphate | Human | 7693 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypk | A | A | - | Human | 12430 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os7 | B | A | adenosine-5'-triphosphate | Human | 9626 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md7 | H | | - | Human | 5481 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehk | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[3,5-bis(chloranyl)-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9641 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu3 | B | A | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6921 | |
| DYRK1A | DYRK | CMGC | 4yu2 | B | A | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3737 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3juh | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5456 | |
| CDK2 | CDK | CMGC | 1pxo | A | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4512 | |
| CDK2 | CDK | CMGC | 6guh | A | B | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10769 | |
| CDK2 | CDK | CMGC | 2c5x | C | B | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 4418 | |
| CDK2 | CDK | CMGC | 2cch | C | C | - | Human | 4431 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oti | A | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9672 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3at2 | A | A | - | Human | 5428 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6eii | A | A | (3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azanium | Human | 9687 | |
| DYRK1A | DYRK | CMGC | 5a4q | A | | n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6717 | |
| DYRK1A | DYRK | CMGC | 4ylj | C | A | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3777 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oni | A | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9459 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6fvf | A | B | - | Human | 11341 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hbn | B | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11270 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9l | A | A | (4~{z})-6,7-bis(chloranyl)-4-[[(4-methylphenyl)amino]methylidene]-8-oxidanyl-1,2-dihydrodibenzofuran-3-one | Human | 9652 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osl | A | B | adenosine-5'-diphosphate | Human | 9629 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moh | A | A | 2-(3-methoxy-4-oxidanyl-phenyl)ethanoic acid | Human | 7658 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4gub | A | | n-[5-({3-cyano-7-[(1-methyl-1h-imidazol-4-yl)amino]pyrazolo[1,5-a]pyrimidin-5-yl}amino)-2-methylphenyl]acetamide | Human | 5491 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osu | A | B | - | Human | 10598 | |
| MAPK14 (p38a) | MAPK | CMGC | 1bl7 | A | | 4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazole | Human | 5193 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mpj | A | A | adenosine-5'-diphosphate | Human | 7677 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | K | | - | Human | 5477 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oth | B | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9625 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3war | A | A | nicotinic acid | Human | 5429 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo8 | B | B | 3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acid | Human | 7688 | |
| CDK2 | CDK | CMGC | 1ke9 | A | | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4250 | |
| CDK2 | CDK | CMGC | 2b54 | A | | 6-(3,4-dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4(5h)-one | Human | 4292 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4q | A | A | 2-methoxyimino-5-(quinolin-6-ylmethyl)-1,3-thiazol-4-one | Human | 14238 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gmd | B | B | adenosine-5'-triphosphate | Human | 9992 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u4u | A | | 3-{5-(acetylamino)-3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1h-indol-1-yl}propanoic acid | Human | 5527 | |
| CDK2 | CDK | CMGC | 2iw8 | A | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4377 | |
| CDK2 | CDK | CMGC | 2bhh | A | | (2e,3s)-3-hydroxy-5'-[(4-hydroxypiperidin-1-yl)sulfonyl]-3-methyl-1,3-dihydro-2,3'-biindol-2'(1'h)-one | Human | 4417 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n1v | A | B | pyrazolo-pyrimidine macrocycle | Human | 7589 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwg | A | A | (5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dione | Human | 14772 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu3 | A | B | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6903 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osu | A | A | - | Human | 10595 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4fbx | A | | - | Human | 5415 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyk | A | A | adenosine-5'-diphosphate | Human | 14547 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwg | A | C | (5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dione | Human | 14773 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ctp | B | B | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7291 | |
| CDK2 | CDK | CMGC | 3r8v | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | 3938 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hoq | A | A | 3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acid | Human | 11669 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3qa0 | A | A | - | Human | 5425 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cx9 | A | B | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7290 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mpj | B | B | - | Human | 7683 | |
| CDK2 | CDK | CMGC | 3bhu | A | B | 4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4446 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7at5 | A | A | ~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamide | Human | 13840 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5nqc | A | A | (3e)-6,7-dichloro-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-one | Human | 8112 | |
| CDK2 | CDK | CMGC | 4fko | A | B | 2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamine | Human | 4534 | |
| CDK2 | CDK | CMGC | 4eoi | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4011 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otz | A | B | trifluoroacetic acid | Human | 9618 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlp | A | A | 5,6-dibromobenzotriazole | Human | 13080 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | B | B | - | Human | 5438 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owh | A | | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10597 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9y | A | B | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5526 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otq | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methoxy-phenyl]methyl]ethanamine | Human | 9651 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rfe | A | B | (~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12147 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3wow | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5445 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rb1 | A | A | (~{e})-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)-~{n}-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]prop-2-enamide | Human | 12145 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tll | A | B | 4,5,6,7-tetrabromobenzotriazole | Human | 13081 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n1v | B | B | pyrazolo-pyrimidine macrocycle | Human | 7586 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qge | A | A | 4,5,6,7-tetrabromobenzotriazole | Human | 14469 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mow | B | A | - | Human | 7671 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c5q | A | B | 2-methylpropyl 5-fluoranyl-3-[1-[[1-[2-[[4-(2-methylpropyl)phenyl]sulfonylamino]ethyl]piperidin-4-yl]methyl]-1,2,3-triazol-4-yl]-1~{h}-indole-2-carboxylate | Human | 15175 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7psu | A | B | - | Human | 14164 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owj | A | B | 9-hydroxy-5,11-dimethyl-4,6-dihydro-1h-pyrido[4,3-b]carbazol-1-one | Human | 5470 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n1v | A | A | pyrazolo-pyrimidine macrocycle | Human | 7588 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otp | B | B | - | Human | 10591 | |
| CDK2 | CDK | CMGC | 2c5v | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4012 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mod | A | B | - | Human | 7667 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn5 | A | A | - | Human | 10705 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a49 | A | | 6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13169 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe1 | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5487 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9z | A | B | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5437 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ku8 | B | | ~{n}-[2-[(1~{s},2~{s})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 8663 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tls | A | B | 5,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13082 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oto | B | A | 2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9688 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn0 | A | A | - | Human | 10697 | |
| CDK2 | CDK | CMGC | 4fx3 | C | A | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 4349 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao6 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14396 | |
| CDK2 | CDK | CMGC | 3qqk | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 4568 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3c13 | A | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5530 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlv | A | B | 6-bromanyl-1~{h}-benzotriazole | Human | 13084 | |
| CDK2 | CDK | CMGC | 1oiu | C | B | 3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamide | Human | 4049 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ouu | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 9610 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oto | A | A | 2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9648 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nga | B | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5441 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mov | A | B | 4'-hydroxycinnamic acid | Human | 7674 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4dgl | D | | - | Human | 5521 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | C | B | - | Human | 5476 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6jwa | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 11467 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os7 | A | B | adenosine-5'-triphosphate | Human | 9609 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md7 | G | | - | Human | 5409 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mod | B | B | - | Human | 7694 | |
| CDK2 | CDK | CMGC | 1h1q | C | | 2-anilino-6-cyclohexylmethoxypurine | Human | 4053 | |
| CDK2 | CDK | CMGC | 1e9h | A | | 2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acid | Human | 4302 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4grb | A | | 5-(2-{[4-(dimethylcarbamoyl)phenyl]amino}-4-methoxypyrimidin-5-yl)thiophene-3-carboxylic acid | Human | 5443 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hou | A | A | 4-hydroxy-3-methoxybenzaldehyde | Human | 11671 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cx9 | A | A | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7287 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rcb | A | | (~{e})-2-cyano-~{n}-(2-hydroxyphenyl)-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12144 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owj | A | A | 9-hydroxy-5,11-dimethyl-4,6-dihydro-1h-pyrido[4,3-b]carbazol-1-one | Human | 5452 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo6 | B | A | - | Human | 7664 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | A | B | - | Human | 5522 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9x | B | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5417 | |
| CDK4 | CDK | CMGC | 7sj3 | A | | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 14485 | |
| CLK3 | CLK | CMGC | 6z53 | A | B | 6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12305 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u87 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5442 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3rps | A | | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 5463 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | E | | - | Human | 5411 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot6 | B | A | - | Human | 9613 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlw | A | C | 7-bromanyl-1~{h}-benzotriazole | Human | 13086 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tei | A | B | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12459 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlw | A | A | 7-bromanyl-1~{h}-benzotriazole | Human | 13088 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5kwh | B | B | ~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 8620 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7n8t | A | B | adenosine monophosphate | Human | 14242 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gc8 | A | | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 2766 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gc9 | B | | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 2767 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gc9 | A | | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 2765 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gc8 | B | | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 2769 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gp0 | A | B | nilotinib | Human | 2764 | |
| MAPK11 (p38b) | MAPK | CMGC | 3gp0 | A | A | nilotinib | Human | 2768 | |
| CDKL1 | CDKL | CMGC | 4agu | C | | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 762 | |
| PRPF4B (PRP4) | DYRK | CMGC | 8h6j | H | A | - | Human | 15281 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | C | A | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11578 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pk6 | A | B | 4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11584 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ijp | A | A | 4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 5547 | |
| PRPF4B (PRP4) | DYRK | CMGC | 8h6e | H | | - | Human | 15282 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ifc | A | B | adenosine-5'-diphosphate | Human | 5544 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ijp | A | B | 4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 5535 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6cnh | A | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 9775 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | D | B | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11579 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6cnh | A | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 9776 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | B | B | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11581 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pk6 | A | A | 4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11582 | |
| PRPF4B (PRP4) | DYRK | CMGC | 8h6j | H | B | - | Human | 15283 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ian | B | | - | Human | 5546 | |
| PRPF4B (PRP4) | DYRK | CMGC | 6pjj | D | A | 4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamide | Human | 11580 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4iir | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 5536 | |
| PRPF4B (PRP4) | DYRK | CMGC | 4ifc | B | A | adenosine-5'-diphosphate | Human | 5542 | |
| SRPK2 | SRPK | CMGC | 5myv | B | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7573 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byy | A | A | 2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 6591 | |
| CDK2 | CDK | CMGC | 2r3q | A | A | 3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxide | Human | 4038 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7aya | A | B | ~{n}-[2-[(1~{r},2~{r})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 13992 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ork | A | B | adenosine-5'-diphosphate | Human | 9655 | |
| CDK5 | CDK | CMGC | 4au8 | A | B | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | 2786 | |
| CLK3 | CLK | CMGC | 6yu1 | a | A | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12403 | |
| CLK3 | CLK | CMGC | 6z2v | A | B | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12636 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8i | B | A | - | Human | 13264 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5o7i | A | A | 4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamide | Human | 9995 | |
| MAPK7 (Erk5) | MAPK | CMGC | 7pus | A | B | 4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamide | Human | 14219 | |
| CDK2 | CDK | CMGC | 2c5n | C | B | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 3903 | |
| CDK2 | CDK | CMGC | 7ack | C | A | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | 13450 | |
| CDK2 | CDK | CMGC | 2xnb | A | A | 3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-one | Human | 4217 | |
| CDK2 | CDK | CMGC | 6q49 | A | C | - | Human | 11193 | |
| CDK2 | CDK | CMGC | 2wfy | A | A | - | Human | 4324 | |
| CDK2 | CDK | CMGC | 4bcp | A | B | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4304 | |
| CDK2 | CDK | CMGC | 4i3z | C | | adenosine-5'-diphosphate | Human | 3961 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | A | B | - | Human | 2577 | |
| CDK2 | CDK | CMGC | 2r3n | A | B | 3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4046 | |
| CDK2 | CDK | CMGC | 3qtq | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4103 | |
| CDK2 | CDK | CMGC | 9esu | A | C | - | Human | 15904 | |
| CDK2 | CDK | CMGC | 6q4a | A | B | 5-iodanylpyrimidine | Human | 11200 | |
| CDK2 | CDK | CMGC | 2fvd | A | | (4-amino-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrimidin-5-yl)(2,3-difluoro-6-methoxyphenyl)methanone | Human | 4408 | |
| CDK2 | CDK | CMGC | 6ylk | A | B | methyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | 12494 | |
| CDK2 | CDK | CMGC | 3qx4 | A | A | 4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4409 | |
| CDK2 | CDK | CMGC | 1e1x | A | | 6-cyclohexylmethyloxy-5-nitroso-pyrimidine-2,4-diamine | Human | 4114 | |
| CDK2 | CDK | CMGC | 4cfv | A | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenol | Human | 4328 | |
| CDK2 | CDK | CMGC | 2bpm | C | | (2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamide | Human | 4128 | |
| CDK5 | CDK | CMGC | 1h4l | A | | - | Human | 2788 | |
| CDK5 | CDK | CMGC | 7vdr | A | | (1r)-1-[7-[(2-fluoranyl-4-pyrazol-1-yl-phenyl)amino]-1,6-naphthyridin-2-yl]-1-(1-methylpiperidin-4-yl)ethanol | Human | 14146 | |
| CDK2 | CDK | CMGC | 3eid | C | A | - | Human | 4072 | |
| CDK2 | CDK | CMGC | 2r3k | A | A | 3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amine | Human | 3953 | |
| CDK2 | CDK | CMGC | 3s1h | A | A | 4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4068 | |
| CDK2 | CDK | CMGC | 3ddq | C | A | r-roscovitine | Human | 4364 | |
| CDK2 | CDK | CMGC | 3ral | A | B | 4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 3984 | |
| CDK2 | CDK | CMGC | 2vtt | A | | 4-{[(2,6-difluorophenyl)carbonyl]amino}-n-[(3s)-piperidin-3-yl]-1h-pyrazole-3-carboxamide | Human | 4100 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yum | A | | 4-[5-[2-(2-hydroxyethyloxy)ethyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]pyrazolo[1,5-a]pyrimidin-3-yl]-2-oxidanyl-benzoic acid | Human | 12462 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | G | A | - | Human | 4613 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr5 | A | B | (2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13934 | |
| MAPK1 (Erk2) | MAPK | CMGC | 1wzy | A | | 1-allyl-5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 2618 | |
| CDK2 | CDK | CMGC | 1gii | A | | 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-urea | Human | 4448 | |
| CDK2 | CDK | CMGC | 6q4b | A | B | 5-bromanylpyrimidine | Human | 11210 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu2 | A | B | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | 10776 | |
| CDK2 | CDK | CMGC | 2r3h | A | B | 3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amine | Human | 3970 | |
| GSK3B | GSK | CMGC | 6y9s | B | A | ~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamide | Human | 12285 | |
| CDK2 | CDK | CMGC | 5nev | A | | 4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamide | Human | 8020 | |
| CDK2 | CDK | CMGC | 5mhq | A | B | (2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-ol | Human | 9408 | |
| CDK2 | CDK | CMGC | 2c5v | C | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4384 | |
| GSK3B | GSK | CMGC | 4j1r | D | | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 736 | |
| CDK2 | CDK | CMGC | 3rpr | A | B | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanone | Human | 4241 | |
| CDK8 | CDK | CMGC | 4f7j | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)urea | Human | 3842 | |
| CDK2 | CDK | CMGC | 7rwf | A | | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acid | Human | 14344 | |
| GSK3B | GSK | CMGC | 4j71 | B | B | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 739 | |
| CDK2 | CDK | CMGC | 4ek4 | A | C | 4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamide | Human | 4369 | |
| CDK2 | CDK | CMGC | 2c5y | A | B | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 6777 | |
| CDK2 | CDK | CMGC | 2wmb | C | | - | Human | 4474 | |
| CDK2 | CDK | CMGC | 3qtu | A | A | 4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4009 | |
| CDK2 | CDK | CMGC | 3dog | C | A | (2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol | Human | 4382 | |
| DYRK2 | DYRK | CMGC | 5lxd | B | A | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7123 | |
| GSK3B | GSK | CMGC | 4iq6 | B | | 6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amine | Human | 750 | |
| CDK2 | CDK | CMGC | 2cjm | A | | adenosine-5'-triphosphate | Human | 4406 | |
| CDK2 | CDK | CMGC | 4eok | A | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 3913 | |
| CDK2 | CDK | CMGC | 2vtr | A | A | 5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 4391 | |
| CDK2 | CDK | CMGC | 3eid | C | B | - | Human | 4467 | |
| CDK2 | CDK | CMGC | 3pj8 | A | B | (2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-ol | Human | 4454 | |
| CDK2 | CDK | CMGC | 2c5v | A | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4338 | |
| CDK2 | CDK | CMGC | 4bcm | A | A | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 4290 | |
| CDK2 | CDK | CMGC | 2r3r | A | B | 3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4215 | |
| CDK2 | CDK | CMGC | 7m2f | A | B | [(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acid | Human | 13796 | |
| CDK2 | CDK | CMGC | 3tnw | C | A | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 3940 | |
| CDK2 | CDK | CMGC | 3qhw | C | A | adenosine-5'-diphosphate | Human | 4129 | |
| CDK2 | CDK | CMGC | 2wfy | C | B | - | Human | 4096 | |
| CDK2 | CDK | CMGC | 2wev | C | C | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4288 | |
| CDK2 | CDK | CMGC | 3ddp | C | B | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 6778 | |
| CDK2 | CDK | CMGC | 1jsv | A | | 4-[(6-amino-4-pyrimidinyl)amino]benzenesulfonamide | Human | 4171 | |
| CDK2 | CDK | CMGC | 3qtz | A | A | 4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4109 | |
| CDK2 | CDK | CMGC | 1pxn | A | A | 4-[4-(4-methyl-2-methylamino-thiazol-5-yl)-pyrimidin-2-ylamino]-phenol | Human | 4383 | |
| CDK2 | CDK | CMGC | 1h0w | A | B | 1-amino-6-cyclohex-3-enylmethyloxypurine | Human | 4016 | |
| CDK2 | CDK | CMGC | 3r9d | A | A | 4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4562 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu7 | G | | - | Human | 10779 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4g6n | A | B | 3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazole | Human | 2593 | |
| CDK2 | CDK | CMGC | 2cch | A | A | adenosine-5'-triphosphate | Human | 4303 | |
| CDK2 | CDK | CMGC | 2cch | C | A | adenosine-5'-triphosphate | Human | 3932 | |
| CDK2 | CDK | CMGC | 1fvv | C | | 4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamide | Human | 4461 | |
| CDK2 | CDK | CMGC | 6q4d | A | B | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid | Human | 11215 | |
| CDK2 | CDK | CMGC | 4eoq | C | B | adenosine-5'-triphosphate | Human | 3912 | |
| CDK2 | CDK | CMGC | 1ol1 | C | | - | Human | 3951 | |
| CDK2 | CDK | CMGC | 3rzb | A | B | 4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamide | Human | 4395 | |
| CDK16 (PCTAIRE1) | CDK | CMGC | 3mtl | A | B | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 1702 | |
| CDK2 | CDK | CMGC | 6q4k | A | A | - | Human | 11179 | |
| CDK2 | CDK | CMGC | 1h27 | C | | - | Human | 4030 | |
| CDK2 | CDK | CMGC | 1oiu | A | B | 3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamide | Human | 4556 | |
| CDK2 | CDK | CMGC | 4eor | A | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 3934 | |
| CDK2 | CDK | CMGC | 4bcm | C | B | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 4124 | |
| CDK2 | CDK | CMGC | 3pxq | A | | 8-anilino-1-naphthalene sulfonate | Human | 3947 | |
| CDK2 | CDK | CMGC | 1h0v | A | B | 5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinone | Human | 3933 | |
| CDK2 | CDK | CMGC | 1w8c | A | A | 6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amine | Human | 4332 | |
| CDK2 | CDK | CMGC | 4eok | C | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4385 | |
| CDK2 | CDK | CMGC | 3qtw | A | B | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 3890 | |
| CDK2 | CDK | CMGC | 4bck | A | B | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 3960 | |
| CDK2 | CDK | CMGC | 4eoo | A | A | adenosine-5'-triphosphate | Human | 4403 | |
| CDK2 | CDK | CMGC | 2c6m | A | | 4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 6782 | |
| CDK2 | CDK | CMGC | 3qwj | A | B | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamide | Human | 4182 | |
| DYRK2 | DYRK | CMGC | 6hdr | A | A | curcumin | Human | 11570 | |
| DYRK2 | DYRK | CMGC | 5lxc | B | A | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7125 | |
| DYRK2 | DYRK | CMGC | 3kvw | A | B | (2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acid | Human | 3149 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3o2m | B | | - | Human | 4649 | |
| DYRK2 | DYRK | CMGC | 7dh3 | A | | 2,7-dimethoxy-9-piperidin-4-ylsulfanyl-acridine | Human | 13978 | |
| DYRK2 | DYRK | CMGC | 5ztn | B | | (1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | Human | 10483 | |
| DYRK2 | DYRK | CMGC | 7ejv | B | B | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | 14182 | |
| DYRK2 | DYRK | CMGC | 7ejv | B | A | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | 14183 | |
| DYRK2 | DYRK | CMGC | 7dhk | A | | 2-methoxy-7-phenylmethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine | Human | 13977 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu7 | A | | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10781 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2xrw | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 4675 | |
| CDK16 (PCTAIRE1) | CDK | CMGC | 5g6v | B | | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 7274 | |
| CDK2 | CDK | CMGC | 7ack | A | A | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | 13451 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vul | A | | - | Human | 4633 | |
| CLK1 | CLK | CMGC | 6khd | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11645 | |
| CDK2 | CDK | CMGC | 7s4t | A | A | 2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acid | Human | 14374 | |
| DYRK1A | DYRK | CMGC | 7aj2 | A | B | 4-(4-methoxyphenyl)pyridin-2-amine | Human | 13592 | |
| DYRK1A | DYRK | CMGC | 7aja | A | B | 1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazine | Human | 13597 | |
| DYRK1A | DYRK | CMGC | 7aj2 | A | A | 4-(4-methoxyphenyl)pyridin-2-amine | Human | 13609 | |
| CLK1 | CLK | CMGC | 6khd | C | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11648 | |
| CDK2 | CDK | CMGC | 2r3l | A | C | 3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amine | Human | 4496 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5wp1 | A | A | 5,7-dihydroxy-4h-1-benzopyran-4-one | Human | 10441 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7atv | A | B | ~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamide | Human | 13828 | |
| CDK2 | CDK | CMGC | 7s4t | A | B | 2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acid | Human | 14373 | |
| CDK2 | CDK | CMGC | 8h6p | A | | (7s,10r)-11-oxa-2,4,5,13,17,23-hexaazatetracyclo[17.3.1.1~3,6~.1~7,10~]pentacosa-1(23),3(25),5,19,21-pentaene-12,18-dione | Human | 14625 | |
| CDK2 | CDK | CMGC | 5nev | C | | 4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamide | Human | 8019 | |
| CDK2 | CDK | CMGC | 3rm6 | A | B | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamide | Human | 4357 | |
| CDK2 | CDK | CMGC | 8h6t | A | | (1r,3s)-3-{3-[(pyridin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl propan-2-ylcarbamate | Human | 14626 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | A | B | benzoic acid | Human | 11276 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | B | B | benzoic acid | Human | 11278 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | B | A | benzoic acid | Human | 11274 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | D | B | phosphoaminophosphonic acid-adenylate ester | Human | 4666 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | C | B | - | Human | 6447 | |
| CLK1 | CLK | CMGC | 6i5l | C | B | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10841 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqq | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamide | Human | 13926 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr9 | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamide | Human | 13932 | |
| CDK2 | CDK | CMGC | 4fkt | A | B | n-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamide | Human | 4322 | |
| CDK2 | CDK | CMGC | 6p3w | A | A | - | Human | 11515 | |
| CDK2 | CDK | CMGC | 2c5n | A | A | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 4063 | |
| CDK2 | CDK | CMGC | 7m2f | A | A | [(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acid | Human | 13797 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6m | A | A | (5~{z})-5-[(3-methoxy-4-oxidanyl-phenyl)methylidene]-1,3-thiazolidine-2,4-dione | Human | 15277 | |
| CDK2 | CDK | CMGC | 1urc | A | A | - | Human | 4334 | |
| CDK2 | CDK | CMGC | 6p3w | C | A | - | Human | 11514 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao3 | A | A | 2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14386 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoi | A | A | 1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-one | Human | 14387 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aod | A | A | 1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-one | Human | 14417 | |
| CDK2 | CDK | CMGC | 7ra5 | A | B | 4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amine | Human | 13959 | |
| CDK2 | CDK | CMGC | 3qtz | A | B | 4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4337 | |
| CDK2 | CDK | CMGC | 6rij | A | A | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | 12623 | |
| CDK2 | CDK | CMGC | 4ez7 | A | | staurosporine | Human | 4240 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | C | B | phosphoaminophosphonic acid-adenylate ester | Human | 4647 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4l7f | A | B | n-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamide | Human | 4637 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6m | A | B | (5~{z})-5-[(3-methoxy-4-oxidanyl-phenyl)methylidene]-1,3-thiazolidine-2,4-dione | Human | 15278 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt5 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15301 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2g01 | A | | 6-chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4h-pyrazolo[3,4-b]quinolin-4-one | Human | 4662 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3o17 | A | | - | Human | 4670 | |
| CDK2 | CDK | CMGC | 1di8 | A | | 4-[3-hydroxyanilino]-6,7-dimethoxyquinazoline | Human | 4577 | |
| CDK2 | CDK | CMGC | 3rah | A | A | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | 4438 | |
| CDK2 | CDK | CMGC | 2uzl | A | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamide | Human | 3917 | |
| CDK2 | CDK | CMGC | 3lfs | A | | n-(6-chloro-5-phenyl-1h-indazol-3-yl)butanamide | Human | 4069 | |
| CDK2 | CDK | CMGC | 4fkl | A | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4134 | |
| CLK1 | CLK | CMGC | 6q8k | A | A | ~{n}2-(3-morpholin-4-ylpropyl)pyrido[3,4-g]quinazoline-2,10-diamine | Human | 10902 | |
| CDK2 | CDK | CMGC | 1oiq | A | | n-[4-(2-methylimidazo[1,2-a]pyridin-3-yl)-2-pyrimidinyl]acetamide | Human | 4379 | |
| CDK2 | CDK | CMGC | 4eom | A | A | adenosine-5'-triphosphate | Human | 4528 | |
| CDK2 | CDK | CMGC | 2w05 | A | B | n-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 4256 | |
| CDK2 | CDK | CMGC | 2vu3 | A | A | 4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamide | Human | 4582 | |
| CDK2 | CDK | CMGC | 6q4e | A | B | 6-iodanyl-7~{h}-purin-2-amine | Human | 11205 | |
| CDK2 | CDK | CMGC | 1h00 | A | A | (2s)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | 4484 | |
| CDK9 | CDK | CMGC | 7nwk | A | | n-((1r,3r)-3-(7-(4-fluoro-2-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-2-yl)cyclopentyl)acetamide | Human | 13951 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6tgu | A | B | 4-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxidanyl-benzoic acid | Human | 12445 | |
| DYRK2 | DYRK | CMGC | 7akh | A | | 4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13615 | |
| DYRK2 | DYRK | CMGC | 6hdp | A | B | scorzodihydrostilbene a | Human | 11573 | |
| DYRK1A | DYRK | CMGC | 7aj4 | A | B | 4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amine | Human | 13588 | |
| CDK2 | CDK | CMGC | 2c5x | A | B | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 3892 | |
| CDK2 | CDK | CMGC | 3ddq | A | A | r-roscovitine | Human | 4477 | |
| CDK2 | CDK | CMGC | 1vyw | C | | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamide | Human | 4133 | |
| CDK2 | CDK | CMGC | 2c5o | C | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4414 | |
| CDK2 | CDK | CMGC | 7zpc | A | A | ~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamide | Human | 14606 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | C | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | 14401 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6n | A | B | (2~{z},5~{z})-5-[(4-methoxy-3-oxidanyl-phenyl)methylidene]-2-phenylimino-1,3-thiazolidin-4-one | Human | 15279 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2no3 | B | | 2-({2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}amino)benzamide | Human | 4657 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | B | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | 14390 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoj | A | A | 1-[(2~{s})-2-(5-methyl-3-pyridin-4-yl-1~{h}-pyrazol-4-yl)pyrrolidin-1-yl]propan-1-one | Human | 14412 | |
| SRPK2 | SRPK | CMGC | 7zkx | A | B | n-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamide | Human | 14616 | |
| CDK2 | CDK | CMGC | 7s85 | A | | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethoxy)benzoic acid | Human | 14425 | |
| CDK2 | CDK | CMGC | 4i3z | A | | adenosine-5'-diphosphate | Human | 4148 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoj | A | B | - | Human | 14418 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao9 | A | A | 1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-one | Human | 14420 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psy | A | | amp phosphoramidate | Human | 15308 | |
| CDK2 | CDK | CMGC | 7ug1 | A | A | 8-(4-chloroanilino)naphthalene-1-sulfonic acid | Human | 14700 | |
| CDK2 | CDK | CMGC | 7ug1 | A | B | 8-(4-chloroanilino)naphthalene-1-sulfonic acid | Human | 14701 | |
| CDK2 | CDK | CMGC | 4fkr | A | A | (8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 4149 | |
| CDK2 | CDK | CMGC | 1h26 | A | | - | Human | 4122 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8qwy | A | | 4-[6-[(2-methoxy-5-propan-2-yloxy-phenyl)amino]pyrazin-2-yl]benzoic acid | Human | 15174 | |
| CDK2 | CDK | CMGC | 5iey | A | A | 4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamide | Human | 6566 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3v3v | A | | 3,5,6,7-tetrahydroxy-2-(3,4-dihydroxyphenyl)-4h-chromen-4-one | Human | 4653 | |
| CDK2 | CDK | CMGC | 6gub | A | | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | 10764 | |
| CDK2 | CDK | CMGC | 3qzh | A | | 4-methoxy-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 3954 | |
| CDK2 | CDK | CMGC | 2wmb | A | | - | Human | 4060 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | F | B | - | Human | 6453 | |
| CDK2 | CDK | CMGC | 3rmf | A | A | 4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 3873 | |
| CDK2 | CDK | CMGC | 6q4i | A | A | 2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acid | Human | 11183 | |
| CDK2 | CDK | CMGC | 6rij | C | A | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | 12625 | |
| MAPK14 (p38a) | MAPK | CMGC | 3heg | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5112 | |
| CDK2 | CDK | CMGC | 3r6x | A | B | 4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4107 | |
| DYRK1A | DYRK | CMGC | 7ajs | A | A | 4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13599 | |
| DYRK1A | DYRK | CMGC | 7aj5 | A | A | 4-(1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13602 | |
| CDK2 | CDK | CMGC | 1e9h | C | | 2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acid | Human | 4570 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vug | A | | - | Human | 4665 | |
| DYRK1A | DYRK | CMGC | 7akl | A | | 4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13589 | |
| CDK2 | CDK | CMGC | 1b39 | A | | adenosine-5'-triphosphate | Human | 4407 | |
| CDK2 | CDK | CMGC | 5oo3 | A | A | 1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-one | Human | 10569 | |
| CDK2 | CDK | CMGC | 2v22 | C | | - | Human | 4255 | |
| DYRK1A | DYRK | CMGC | 7aka | A | B | 4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13595 | |
| CDK2 | CDK | CMGC | 3py1 | A | B | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 4444 | |
| CDK2 | CDK | CMGC | 2bpm | A | | (2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamide | Human | 4042 | |
| CDK12 (CRK7) | CDK | CMGC | 7nxk | A | | (e)-n-[4-[(1r,3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]cyclohexyl]oxyphenyl]-4-(dimethylamino)but-2-enamide | Human | 13547 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoa | A | A | ~{n}-pyridin-3-ylprop-2-enamide | Human | 14391 | |
| CDK2 | CDK | CMGC | 2cci | A | | adenosine-5'-triphosphate | Human | 4373 | |
| CDK2 | CDK | CMGC | 1ke6 | A | | n-methyl-{4-[2-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)hydrazino]phenyl}methanesulfonamide | Human | 4219 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao5 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamide | Human | 14392 | |
| CDK2 | CDK | CMGC | 1ogu | A | B | 4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamide | Human | 3935 | |
| CDK2 | CDK | CMGC | 7b7s | A | A | 7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxide | Human | 13833 | |
| CDK2 | CDK | CMGC | 2r3l | A | A | 3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amine | Human | 4200 | |
| CDK9 | CDK | CMGC | 8i0l | A | | 2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 15170 | |
| CDK2 | CDK | CMGC | 6guk | A | A | ~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamine | Human | 10773 | |
| CDK2 | CDK | CMGC | 2w1h | A | | n-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamide | Human | 4228 | |
| CDK2 | CDK | CMGC | 4cfw | A | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4557 | |
| CDK2 | CDK | CMGC | 3my5 | C | C | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 3929 | |
| CDK2 | CDK | CMGC | 2uzn | A | | 4-{5-[(1z)-1-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)ethyl]-2-furyl}benzenesulfonamide | Human | 4064 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8qwz | A | | 4-[6-(6-propan-2-yloxyindol-1-yl)pyrazin-2-yl]benzoic acid | Human | 15176 | |
| DYRK1A | DYRK | CMGC | 7akb | A | B | 4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13604 | |
| CDK2 | CDK | CMGC | 3sw7 | A | A | n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamine | Human | 4198 | |
| CDK2 | CDK | CMGC | 4bco | A | B | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4051 | |
| CDK2 | CDK | CMGC | 3lfn | A | | n-[6-(4-hydroxyphenyl)-5-phenyl-1h-indazol-3-yl]butanamide | Human | 4330 | |
| CDK2 | CDK | CMGC | 5ank | A | | 2,4,6-trioxo-1-phenyl-hexahydropyrimidine-5-carboxamide | Human | 6538 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q38 | A | B | benzoic acid | Human | 11285 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7s1n | A | A | 4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13958 | |
| CDK2 | CDK | CMGC | 3rmf | A | B | 4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4014 | |
| CDK2 | CDK | CMGC | 3qtx | A | A | 4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4339 | |
| CDK2 | CDK | CMGC | 1h1r | A | A | 6-cyclohexylmethoxy-2-(3'-chloroanilino) purine | Human | 3906 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt1 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15302 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aog | A | B | ~{n}-(5-methyl-1,2-oxazol-3-yl)propanamide | Human | 14421 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7s1n | A | B | 4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13957 | |
| DYRK2 | DYRK | CMGC | 7dhv | A | | 2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine-4-carboxylic acid | Human | 13974 | |
| CDK2 | CDK | CMGC | 4cfn | A | B | 6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amine | Human | 4437 | |
| CDK2 | CDK | CMGC | 4eom | C | A | adenosine-5'-triphosphate | Human | 4481 | |
| CDK2 | CDK | CMGC | 2wev | A | B | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4580 | |
| DYRK1A | DYRK | CMGC | 7aj8 | A | A | 4-(1-benzofuran-5-yl)pyridin-2-amine | Human | 13587 | |
| DYRK1A | DYRK | CMGC | 7ake | A | | 4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13601 | |
| GSK3B | GSK | CMGC | 7oy5 | A | B | ~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamine | Human | 14119 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr8 | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamide | Human | 13933 | |
| GSK3B | GSK | CMGC | 7oy5 | A | A | ~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamine | Human | 14118 | |
| CDK2 | CDK | CMGC | 7kjs | A | | 6-(difluoromethyl)-8-[(1r,2r)-2-hydroxy-2-methylcyclopentyl]-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 13740 | |
| DYRK2 | DYRK | CMGC | 7dhh | A | | [9-(azetidin-3-ylmethylsulfanyl)-2,7-dimethoxy-acridin-4-yl]methanol | Human | 13975 | |
| CDK2 | CDK | CMGC | 7b7s | A | B | 7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxide | Human | 13834 | |
| CDK2 | CDK | CMGC | 1pxl | A | B | - | Human | 4074 | |
| CDK2 | CDK | CMGC | 3eoc | A | | 5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine | Human | 4390 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6l | A | B | 5-azanyl-3-[(~{z})-1-cyano-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]-3~{h}-pyrazole-4-carbonitrile | Human | 15280 | |
| GSK3B | GSK | CMGC | 5t31 | B | | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9564 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoh | A | B | ~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamide | Human | 14404 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt3 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15305 | |
| SRPK1 | SRPK | CMGC | 3beg | A | | phosphoaminophosphonic acid-adenylate ester | Human | 9472 | |
| CDK2 | CDK | CMGC | 4bck | C | D | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4080 | |
| CDK2 | CDK | CMGC | 7mkx | A | | 2-[(5-bromo-2-{4-[(cyanomethyl)sulfamoyl]anilino}pyrimidin-4-yl)amino]-6-fluorobenzamide | Human | 14490 | |
| CDK2 | CDK | CMGC | 1jvp | P | 1 | 3-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazole | Human | 3919 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4awi | A | B | n-(1,1-dioxidotetrahydro-2h-thiopyran-4-yl)-4-[2-(1-methylethyl)-1h-pyrrolo[2,3-b]pyridin-4-yl]benzenesulfonamide | Human | 4634 | |
| CDK2 | CDK | CMGC | 2vto | A | B | n-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamide | Human | 3946 | |
| CDK2 | CDK | CMGC | 3rni | A | A | 3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 3993 | |
| CDK2 | CDK | CMGC | 3ral | A | A | 4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4017 | |
| CDK2 | CDK | CMGC | 4eoj | A | B | adenosine-5'-triphosphate | Human | 4015 | |
| CDK2 | CDK | CMGC | 3py1 | A | A | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 4361 | |
| CDK1 (CDC2) | CDK | CMGC | 4y72 | A | A | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4610 | |
| MAPK8 (JNK1) | MAPK | CMGC | 6zr5 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 12984 | |
| CDK2 | CDK | CMGC | 6q4i | A | B | 2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acid | Human | 11197 | |
| CDK2 | CDK | CMGC | 1oiu | C | A | 3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamide | Human | 4524 | |
| DYRK1A | DYRK | CMGC | 6s17 | A | A | ~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11369 | |
| MAPK7 (Erk5) | MAPK | CMGC | 9lta | A | | 4-[5-chloranyl-2-[[3-[(dimethylamino)methyl]phenyl]amino]pyrimidin-4-yl]-~{n}-morpholin-4-yl-thiophene-2-carboxamide | Human | 15439 | |
| CDKL5 | CDKL | CMGC | 9epu | A | | ~{n}-[5-[(5-propan-2-yl-1,3-oxazol-2-yl)methylsulfanyl]-1,3-thiazol-2-yl]piperidine-4-carboxamide | Human | 15440 | |
| CLK3 | CLK | CMGC | 29mo | A | | 3^{3}-methoxy-1^{7}-(2-(2-(4-methylpiperazin-1-yl)ethoxy)ethoxy)-4,7,10-trioxa-2-aza-1(4,6)-quinolina-3(1,2)-benzenacyclodecaphane-1^{3}-carbonitrile | Human | 15441 | |
| CLK3 | CLK | CMGC | 29mp | A | | 1^{7}-methoxy-4,7,10-trioxa-2-aza-1(4,6)-quinolina-3(1,2)-benzenacyclodecaphane-1^{3}-carbonitrile | Human | 15442 | |
| CLK3 | CLK | CMGC | 9ez3 | A | | 1-(5-~{tert}-butyl-2-quinolin-6-yl-pyrazol-3-yl)-3-[3-(4-morpholin-4-yl-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]urea | Human | 15443 | |
| CDK16 (PCTAIRE1) | CDK | CMGC | 9r2i | C | | phosphothiophosphoric acid-adenylate ester | Human | 15481 | |
| CDK2 | CDK | CMGC | 3r7y | A | A | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamide | Human | 4476 | |
| CDK2 | CDK | CMGC | 4ii5 | C | A | adenosine-5'-diphosphate | Human | 4530 | |
| CDK2 | CDK | CMGC | 1oiy | C | A | 4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamide | Human | 4465 | |
| CDK2 | CDK | CMGC | 1pxi | A | B | - | Human | 3924 | |
| CDK2 | CDK | CMGC | 5and | A | | 2-imidazol-1-yl-1h-benzimidazole | Human | 6543 | |
| CDK2 | CDK | CMGC | 4bco | C | B | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4018 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8u8j | A | | (4m)-4-{(4r)-3-[(2s)-2-methylbutyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(1-methyl-1h-pyrazol-5-yl)pyrimidin-2-amine | Human | 15224 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8u8k | A | | (4m)-4-{(4s)-3-[(2-chloropyridin-3-yl)methyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(oxan-4-yl)pyrimidin-2-amine | Human | 15225 | |
| MAPK1 (Erk2) | MAPK | CMGC | 9tyh | A | | adenosine-5'-diphosphate | Human | 15552 | |
| MAPK1 (Erk2) | MAPK | CMGC | 9tyg | B | | adenosine-5'-diphosphate | Human | 15553 | |
| MAPK1 (Erk2) | MAPK | CMGC | 9tyi | A | | - | Human | 15554 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 9ihi | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 15555 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 9fbi | A | B | nicotinic acid | Human | 15556 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 9r57 | A | A | 5,6-dibromobenzotriazole | Human | 15557 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 9r5c | A | B | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 15558 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 9hk5 | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 15559 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 9hk5 | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 15560 | |
| DYRK1A | DYRK | CMGC | 9ft2 | A | | 3-[[[4-[(3-cyclobutyl-1~{h}-pyrazol-5-yl)amino]furo[3,2-d]pyrimidin-2-yl]amino]methyl]benzamide | Human | 15583 | |
| MAPK11 (p38b) | MAPK | CMGC | 8ygw | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 15234 | |
| CDK7 | CDK | CMGC | 8p4z | A | A | 2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine | Human | 14796 | |
| DYRK1A | DYRK | CMGC | 9ft6 | A | | ~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)furo[3,2-d]pyrimidine-2,4-diamine | Human | 15584 | |
| DYRK1A | DYRK | CMGC | 9ft4 | A | | ~{n}4-(5-cyclopropyl-1~{h}-pyrazol-3-yl)-~{n}2-(phenylmethyl)furo[3,2-d]pyrimidine-2,4-diamine | Human | 15585 | |
| DYRK1A | DYRK | CMGC | 8yev | A | | coumestrol | Human | 15586 | |
| DYRK1A | DYRK | CMGC | 9fpx | A | | curcumin | Human | 15587 | |
| DYRK1A | DYRK | CMGC | 7fht | A | C | (5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | 15588 | |
| DYRK1A | DYRK | CMGC | 9fuf | A | | 3-[[[4-[(3-cyclopropyl-1~{h}-pyrazol-5-yl)amino]thieno[3,2-d]pyrimidin-2-yl]amino]methyl]benzamide | Human | 15589 | |
| DYRK1A | DYRK | CMGC | 9ft3 | A | | ~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)thieno[3,2-d]pyrimidine-2,4-diamine | Human | 15590 | |
| DYRK1A | DYRK | CMGC | 9yko | A | | (5,6-dihydroxy-1,3-benzothiazol-2-yl)(3,4-dihydroxyphenyl)methanone | Human | 15591 | |
| CDK7 | CDK | CMGC | 8p4z | A | B | 2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine | Human | 14797 | |
| CDK2 | CDK | CMGC | 8uv0 | A | A | 1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-ol | Human | 15238 | |
| CLK2 | CLK | CMGC | 3nr9 | A | | (5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 1927 | |
| CDK2 | CDK | CMGC | 3r9n | A | A | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | 3885 | |
| CDK2 | CDK | CMGC | 8uv0 | A | B | 1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-ol | Human | 15239 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | A | A | - | Human | 4607 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v61 | A | A | - | Human | 8265 | |
| CDK2 | CDK | CMGC | 4fkv | A | B | (3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamide | Human | 3939 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oto | B | B | 2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9611 | |
| CDK2 | CDK | CMGC | 3qx2 | A | B | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamide | Human | 4297 | |
| CDK2 | CDK | CMGC | 1gy3 | C | | adenosine-5'-triphosphate | Human | 4445 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4b | A | B | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13165 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7l1x | A | A | (2~{z})-6-[[2,6-bis(chloranyl)phenyl]methylsulfonyl]-2-[[4-oxidanyl-3-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methylidene]-4~{h}-1,4-benzothiazin-3-one | Human | 13847 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6nbs | A | A | - | Human | 11510 | |
| CDK2 | CDK | CMGC | 5jq8 | A | | (3s,4s)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 7417 | |
| CDK2 | CDK | CMGC | 3rm6 | A | A | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamide | Human | 4262 | |
| CDK2 | CDK | CMGC | 7qhl | A | A | 5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidine | Human | 14275 | |
| CDK2 | CDK | CMGC | 3qqj | A | B | 2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 4204 | |
| CDK2 | CDK | CMGC | 3qqg | A | B | 4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 4310 | |
| CDK2 | CDK | CMGC | 3qqf | A | A | 5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4211 | |
| CDK2 | CDK | CMGC | 2iw8 | C | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4350 | |
| CDK7 | CDK | CMGC | 8pyr | A | B | - | Human | 15253 | |
| CDK2 | CDK | CMGC | 2c4g | C | | (3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-ium | Human | 4453 | |
| CDK2 | CDK | CMGC | 1okw | A | | - | Human | 4314 | |
| CDK2 | CDK | CMGC | 1w0x | C | A | olomoucine | Human | 4537 | |
| CLK3 | CLK | CMGC | 6ft7 | A | B | 3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9903 | |
| CLK3 | CLK | CMGC | 6z52 | B | B | 11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12626 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7bu4 | A | A | 4-(6-aminocarbonyl-8-oxidanylidene-9-phenyl-7h-purin-2-yl)benzoic acid | Human | 13486 | |
| CLK3 | CLK | CMGC | 6z53 | A | A | 6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12300 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao8 | A | B | 1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-one | Human | 14405 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mp8 | B | A | adenosine-5'-diphosphate | Human | 7695 | |
| CDK2 | CDK | CMGC | 6guk | A | B | ~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamine | Human | 10768 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1jwh | B | | - | Human | 5524 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oti | A | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9667 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moe | B | B | adenosine-5'-diphosphate | Human | 7687 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao8 | A | A | 1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-one | Human | 14410 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owk | A | A | 7-chloro-10-methyl-11h-benzo[g]pyrido[4,3-b]indol-3-ol | Human | 5467 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9y | A | A | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5493 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oni | B | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9458 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvh | A | A | adenosine-5'-diphosphate | Human | 6896 | |
| CLK3 | CLK | CMGC | 3raw | B | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 1824 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao2 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)propanamide | Human | 14415 | |
| GSK3B | GSK | CMGC | 9hv3 | A | | 2-oxidanylidene-~{n}-[3-(4-phenylpiperazin-1-yl)propyl]-6-pyridin-3-yl-3~{h}-benzimidazole-1-carboxamide | Human | 15794 | |
| GSK3B | GSK | CMGC | 9x2y | A | A | - | Human | 15795 | |
| GSK3B | GSK | CMGC | 9hul | A | | ~{n}-[3-[4-[2,3-bis(chloranyl)phenyl]piperazin-1-yl]propyl]-2-oxidanylidene-6-pyridin-3-yl-3~{h}-benzimidazole-1-carboxamide | Human | 15796 | |
| GSK3B | GSK | CMGC | 9fr6 | A | | 3-[[[4-[(3-cyclopropyl-1~{h}-pyrazol-5-yl)amino]thieno[3,2-d]pyrimidin-2-yl]amino]methyl]benzamide | Human | 15797 | |
| CLK3 | CLK | CMGC | 6yty | A | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12409 | |
| GSK3B | GSK | CMGC | 9huk | A | | ~{n}-[4-[4-[2,3-bis(chloranyl)phenyl]piperazin-1-yl]butyl]-2-oxidanylidene-6-pyridin-3-yl-3~{h}-benzimidazole-1-carboxamide | Human | 15800 | |
| GSK3B | GSK | CMGC | 9fr7 | A | | ~{n}4-(5-cyclopropyl-1~{h}-pyrazol-3-yl)-~{n}2-(phenylmethyl)furo[3,2-d]pyrimidine-2,4-diamine | Human | 15801 | |
| GSK3B | GSK | CMGC | 9x2y | A | B | - | Human | 15802 | |
| CDK2 | CDK | CMGC | 2vtn | A | | 4-(acetylamino)-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4027 | |
| MAPK7 (Erk5) | MAPK | CMGC | 7pus | A | A | 4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamide | Human | 14218 | |
| MAPK7 (Erk5) | MAPK | CMGC | 6hkn | A | A | [2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanone | Human | 10918 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic7 | D | | phosphoaminophosphonic acid-adenylate ester | Human | 391 | |
| CLK3 | CLK | CMGC | 2wu7 | A | A | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 1828 | |
| GSK3B | GSK | CMGC | 9fr9 | A | | 3-[[[4-[(3-cyclobutyl-1~{h}-pyrazol-5-yl)amino]furo[3,2-d]pyrimidin-2-yl]amino]methyl]benzamide | Human | 15798 | |
| GSK3B | GSK | CMGC | 9x2q | A | A | - | Human | 15799 | |
| CDK2 | CDK | CMGC | 2c6t | C | | 4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 3994 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4g6n | A | A | 3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazole | Human | 2609 | |
| GSK3B | GSK | CMGC | 9x2x | A | A | - | Human | 15803 | |
| GSK3B | GSK | CMGC | 9x2v | A | A | - | Human | 15804 | |
| GSK3B | GSK | CMGC | 9x2u | A | B | - | Human | 15805 | |
| GSK3B | GSK | CMGC | 9x2v | A | B | - | Human | 15806 | |
| GSK3B | GSK | CMGC | 9x2w | A | | - | Human | 15807 | |
| GSK3B | GSK | CMGC | 9x2x | A | B | - | Human | 15808 | |
| CDK2 | CDK | CMGC | 2xmy | A | B | 4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamide | Human | 3985 | |
| CLK1 | CLK | CMGC | 6i5h | A | A | 5-(1-methylpyrazol-4-yl)-3-(3-phenoxyphenyl)furo[3,2-b]pyridine | Human | 10848 | |
| DYRK1A | DYRK | CMGC | 7aj4 | A | A | 4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amine | Human | 13605 | |
| CDK2 | CDK | CMGC | 9qjj | B | | ots964 | Human | 15914 | |
| CDK2 | CDK | CMGC | 13gk | A | C | - | Human | 15915 | |
| CDK2 | CDK | CMGC | 9nyr | A | B | - | Human | 15916 | |
| CDK2 | CDK | CMGC | 9et1 | A | A | 4-iodanylbenzamide | Human | 15917 | |
| CDK2 | CDK | CMGC | 9gla | A | A | 7-dimethylphosphoryl-3-[2-[[(3~{s})-6,6-dimethylpiperidin-3-yl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]-1~{h}-indole-6-carbonitrile | Human | 15918 | |
| CDK2 | CDK | CMGC | 9fr2 | A | | 4-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]benzenesulfonyl fluoride | Human | 15919 | |
| CDK2 | CDK | CMGC | 9esw | A | D | - | Human | 15920 | |
| CDK2 | CDK | CMGC | 9esk | A | B | (4-bromo-2-oxopyridin-1(2h)-yl)acetic acid | Human | 15913 | |
| CDK2 | CDK | CMGC | 9esj | A | A | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid | Human | 15953 | |
| CDK2 | CDK | CMGC | 9esw | A | B | (4-bromanylpyridin-2-yl)methanol | Human | 15954 | |
| CDK2 | CDK | CMGC | 9esu | A | B | 4-bromanyl-2-(methoxymethyl)pyridine | Human | 15955 | |
| CDK2 | CDK | CMGC | 9eso | A | B | - | Human | 15956 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bve | A | A | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6029 | |
| CDK2 | CDK | CMGC | 7s7a | A | A | 2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14427 | |
| CDK2 | CDK | CMGC | 9esy | A | A | 4-bromanyl-1,8-naphthyridine | Human | 15930 | |
| CDK2 | CDK | CMGC | 9et1 | A | B | 4-iodanylbenzamide | Human | 15951 | |
| CDK2 | CDK | CMGC | 9etp | A | A | 4-bromo-1h-pyrazole | Human | 15952 | |
| CDK2 | CDK | CMGC | 2r3k | A | B | 3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amine | Human | 3876 | |
| CDK2 | CDK | CMGC | 7sa0 | A | A | 2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14428 | |
| CDK2 | CDK | CMGC | 7sa0 | A | B | 2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14429 | |
| CDK2 | CDK | CMGC | 7s84 | A | B | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14432 | |
| CDK2 | CDK | CMGC | 9nyq | A | | 4-({4-[(1s,4s)-4-hydroxy-4-methylcyclohexyl]-5-(trifluoromethyl)pyrimidin-2-yl}amino)-n,3-dimethylbenzene-1-sulfonamide | Human | 15957 | |
| CDK2 | CDK | CMGC | 9gp3 | A | | (3~{s})-~{n}-ethyl-3-[[9-ethyl-2-[[(2~{r},3~{s})-2-oxidanylpentan-3-yl]amino]purin-6-yl]amino]pyrrolidine-1-sulfonamide | Human | 15958 | |
| CDK2 | CDK | CMGC | 9esq | A | A | 4-bromanyl-2-oxidanyl-benzoic acid | Human | 15959 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgc | A | A | 5,6-dibromobenzotriazole | Human | 14433 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvd | A | B | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-one | Human | 6028 | |
| CDK2 | CDK | CMGC | 7s9x | A | A | 2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acid | Human | 14430 | |
| CDK9 | CDK | CMGC | 32aw | A | | 4-[[[6-[5-chloranyl-2-[[4-[[(2~{r})-1-methoxypropan-2-yl]amino]phenyl]amino]pyridin-4-yl]pyridin-2-yl]amino]methyl]oxane-4-carbonitrile | Human | 15994 | |
| CDK13 (CHED) | CDK | CMGC | 7nxj | A | | n-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamide | Human | 13544 | |
| MAPK7 (Erk5) | MAPK | CMGC | 6hkn | A | B | [2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanone | Human | 10919 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9qsr | A | | 5-[7-[(3-chloranyl-4-phenyl-phenyl)methylamino]heptylamino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 16063 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s6g | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 16064 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9qss | A | | 5-[8-[(3-chloranyl-4-phenyl-phenyl)methylamino]octylamino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 16065 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9fbl | A | B | nicotinic acid | Human | 16066 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9rcy | A | B | - | Human | 16067 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9fbm | A | A | nicotinic acid | Human | 16068 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s77 | A | A | nicotinic acid | Human | 16069 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s7i | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 16070 | |
| MAPK3 (Erk1) | MAPK | CMGC | 9uux | B | | phosphoaminophosphonic acid-adenylate ester | Human | 16039 | |
| MAPK3 (Erk1) | MAPK | CMGC | 9uur | B | | phosphoaminophosphonic acid-adenylate ester | Human | 16040 | |
| MAPK3 (Erk1) | MAPK | CMGC | 9tu0 | A | | - | Human | 16041 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9qrh | A | | 5-[[(3~{e})-3-[4-[2-(3,4-dichlorophenyl)ethylamino]-4-oxidanylidene-butanoyl]iminopropyl]amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 16061 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7i85 | A | A | 5-(ethylamino)benzo[c][2,6]naphthyridine-8-carboxamide | Human | 16062 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | C | A | - | Human | 6449 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9rfn | A | A | - | Human | 16071 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9rcx | A | B | - | Human | 16072 | |
| DYRK2 | DYRK | CMGC | 9kqy | A | | - | Human | 16123 | |
| DYRK2 | DYRK | CMGC | 9mc0 | A | | [2-[[4-(1,3-benzothiazol-5-yl)-5-fluoranyl-pyrimidin-2-yl]amino]-1,3-thiazol-5-yl]-piperazin-1-yl-methanone | Human | 16124 | |
| CDK2 | CDK | CMGC | 3pxr | A | A | - | Human | 3941 | |
| CDK2 | CDK | CMGC | 7s7a | A | B | 2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14426 | |
| CDK2 | CDK | CMGC | 2clx | A | A | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 3909 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8e | A | | ~{n}-[2-[2-azanylethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 6409 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otr | A | B | adenosine-5'-triphosphate | Human | 9634 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4x21 | A | | n-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamide | Human | 6240 | |
| CDK2 | CDK | CMGC | 4eoj | A | A | adenosine-5'-triphosphate | Human | 4271 | |
| CDK2 | CDK | CMGC | 4eom | C | B | adenosine-5'-triphosphate | Human | 4423 | |
| CDK2 | CDK | CMGC | 3r71 | A | A | 4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 3962 | |
| CDK2 | CDK | CMGC | 1pxo | A | C | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4546 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rff | A | A | (~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-nitro-4-oxidanyl-phenyl)prop-2-enamide | Human | 12146 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aod | A | B | 1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-one | Human | 14388 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hor | A | B | (~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-one | Human | 11663 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1pjk | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5410 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l23 | A | B | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 13454 | |
| CDK2 | CDK | CMGC | 4eop | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4061 | |
| CDK2 | CDK | CMGC | 3r8l | A | B | (5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4523 | |
| CDK2 | CDK | CMGC | 6ath | A | B | - | Human | 10570 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nga | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5515 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmf | A | B | (3-chloranyl-4-phenyl-phenyl)methyl-propyl-azanium | Human | 7666 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3qa0 | B | A | - | Human | 5495 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5clp | B | A | 2-(3,4-dichlorophenyl)ethanamine | Human | 6909 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9k | A | A | 1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diol | Human | 9682 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u87 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 5513 | |
| MAPK12 (p38g) | MAPK | CMGC | 6una | A | B | - | Human | 11900 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rb1 | A | B | (~{e})-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)-~{n}-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]prop-2-enamide | Human | 12142 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hot | A | B | (2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enal | Human | 11670 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5t1h | A | A | 7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 8685 | |
| MAPK12 (p38g) | MAPK | CMGC | 6una | B | A | - | Human | 11901 | |
| CDK2 | CDK | CMGC | 3qqg | A | A | 4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 4130 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5buj | A | A | 4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-one | Human | 2560 | |
| CDK2 | CDK | CMGC | 4bck | C | C | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4029 | |
| CDK2 | CDK | CMGC | 7qhl | A | B | 5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidine | Human | 14276 | |
| CDK2 | CDK | CMGC | 4eol | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4521 | |
| CDK2 | CDK | CMGC | 6q4k | A | C | - | Human | 11189 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | E | B | - | Human | 4614 | |
| CDK7 | CDK | CMGC | 1ua2 | C | | adenosine-5'-triphosphate | Human | 542 | |
| CDK7 | CDK | CMGC | 7b5o | J | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13278 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoc | A | A | ~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamide | Human | 14409 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2y9q | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2626 | |
| CDK2 | CDK | CMGC | 7zpc | A | B | ~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamide | Human | 14607 | |
| CDK7 | CDK | CMGC | 7nvr | 8 | | - | Human | 13543 | |
| CDK2 | CDK | CMGC | 1fq1 | B | | adenosine-5'-triphosphate | Human | 4266 | |
| CDK2 | CDK | CMGC | 4cfv | A | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenol | Human | 4180 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h36 | A | B | - | Human | 3461 | |
| CDK8 | CDK | CMGC | 5hnb | A | B | [6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanone | Human | 6563 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwu | A | B | - | Human | 11249 | |
| MAPK14 (p38a) | MAPK | CMGC | 4zth | A | B | 6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazine | Human | 6707 | |
| MAPK8 (JNK1) | MAPK | CMGC | 1ukh | A | | - | Human | 4628 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | G | | - | Human | 5483 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hor | A | A | (~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-one | Human | 11668 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypn | B | B | adenosine-5'-diphosphate | Human | 12436 | |
| CDK5 | CDK | CMGC | 7vdq | A | | 2-[[7-[[2-fluoranyl-4-[3-(hydroxymethyl)pyrazol-1-yl]phenyl]amino]-1,6-naphthyridin-2-yl]-(1-methylpiperidin-4-yl)amino]ethanoic acid | Human | 14144 | |
| CDK5 | CDK | CMGC | 7vds | A | A | 5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrile | Human | 14148 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2h96 | A | | 5-cyano-n-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamide | Human | 4655 | |
| CDK5 | CDK | CMGC | 1unh | A | | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | 2780 | |
| CDK5 | CDK | CMGC | 3o0g | A | | - | Human | 2782 | |
| CDK5 | CDK | CMGC | 1unl | B | | - | Human | 2790 | |
| CDK2 | CDK | CMGC | 7rxo | A | B | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acid | Human | 14351 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csh | A | A | adenosine-5'-triphosphate | Human | 6918 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osz | A | A | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azanium | Human | 9669 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5kwh | A | B | ~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 8619 | |
| CDK2 | CDK | CMGC | 7uxk | A | | - | Human | 14570 | |
| CDK2 | CDK | CMGC | 7uxi | A | A | - | Human | 14571 | |
| CDK2 | CDK | CMGC | 7rxo | A | A | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acid | Human | 14352 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4qtd | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 4651 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4g1w | A | | methyl 7-fluoro-3-{4-[(2-hydroxyethyl)sulfonyl]benzyl}-4-oxo-1-phenyl-1,4-dihydroquinoline-2-carboxylate | Human | 4631 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2xs0 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 4629 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2gmx | B | | n-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-bromo-2,5-dimethoxyphenyl)acetamide | Human | 4638 | |
| CDK2 | CDK | CMGC | 7uxi | A | B | - | Human | 14572 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qux | A | B | adenosine-5'-diphosphate | Human | 14573 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo6 | B | B | - | Human | 7652 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qux | A | A | adenosine-5'-diphosphate | Human | 14574 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlr | A | A | 4,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13089 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4c | A | B | 3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acid | Human | 7403 | |
| MAPK8 (JNK1) | MAPK | CMGC | 1uki | A | | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | 4630 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8i | A | A | - | Human | 13263 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | E | A | - | Human | 6451 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aek | A | A | adenosine-5'-triphosphate | Human | 14442 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hnw | A | B | coumestrol | Human | 11521 | |
| MAPK8 (JNK1) | MAPK | CMGC | 6zr5 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 12985 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4hys | A | | trans-4-{[4-(1h-indazol-1-yl)pyrimidin-2-yl]amino}cyclohexanol | Human | 4672 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyd | A | A | adenosine-5'-triphosphate | Human | 14438 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy0 | A | B | adenosine-5'-diphosphate | Human | 14439 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyo | A | B | adenosine-5'-triphosphate | Human | 14440 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyr | A | B | adenosine-5'-triphosphate | Human | 14456 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu0 | A | B | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7293 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csh | B | A | adenosine-5'-triphosphate | Human | 6923 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vui | A | | - | Human | 4652 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy2 | A | A | adenosine-5'-triphosphate | Human | 14443 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyr | A | A | adenosine-5'-triphosphate | Human | 14444 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aec | A | C | adenosine-5'-triphosphate | Human | 14446 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aek | A | B | adenosine-5'-triphosphate | Human | 14447 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy0 | A | A | adenosine-5'-diphosphate | Human | 14452 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aec | A | A | adenosine-5'-triphosphate | Human | 14455 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 4646 | |
| CDK2 | CDK | CMGC | 7vdu | A | B | [1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanol | Human | 14137 | |
| CDK2 | CDK | CMGC | 1gz8 | A | B | 1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanol | Human | 3956 | |
| CDK2 | CDK | CMGC | 4eoj | C | A | adenosine-5'-triphosphate | Human | 4041 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyo | A | A | adenosine-5'-triphosphate | Human | 14448 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2xrw | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 4660 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vud | A | | - | Human | 4664 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmn | A | A | 6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 5196 | |
| CDK2 | CDK | CMGC | 4fkr | A | B | (8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-one | Human | 4535 | |
| CDK2 | CDK | CMGC | 3eid | A | A | (2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-ol | Human | 4386 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7l1x | A | B | (2~{z})-6-[[2,6-bis(chloranyl)phenyl]methylsulfonyl]-2-[[4-oxidanyl-3-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methylidene]-4~{h}-1,4-benzothiazin-3-one | Human | 13848 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6a1c | A | B | 5-bromanyl-2-methoxy-4-[(e)-(3-methylsulfanyl-5-phenyl-1,2,4-triazol-4-yl)iminomethyl]phenol | Human | 11286 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ct0 | B | A | 3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-ol | Human | 7288 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9w | A | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5436 | |
| DYRK1A | DYRK | CMGC | 2wo6 | A | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3758 | |
| CDK2 | CDK | CMGC | 6p3w | A | B | - | Human | 11517 | |
| CDK2 | CDK | CMGC | 4bcm | A | B | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 4203 | |
| CDK2 | CDK | CMGC | 1h24 | A | | - | Human | 4199 | |
| CDK2 | CDK | CMGC | 1ogu | C | B | 4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamide | Human | 4560 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyd | A | B | adenosine-5'-triphosphate | Human | 14450 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsj | A | B | 3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | 6585 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic7 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 392 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 4 | - | Human | 5067 | |
| CDK2 | CDK | CMGC | 4bgh | A | B | 4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamide | Human | 4509 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aec | A | B | adenosine-5'-triphosphate | Human | 14451 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3bqc | A | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5490 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5o7i | A | B | 4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamide | Human | 9994 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byy | A | B | 2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 6587 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsl | A | | 3-amino-5-[(4-chlorophenyl)amino]-n-[(1s)-1-phenylethyl]-1h-1,2,4-triazole-1-carboxamide | Human | 6586 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsg | A | B | 3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | 6584 | |
| CDK16 (PCTAIRE1) | CDK | CMGC | 5g6v | A | | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 7273 | |
| CDK2 | CDK | CMGC | 2c6i | A | | 4-{[5-(cyclohexylmethoxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 6774 | |
| CDK2 | CDK | CMGC | 2wfy | C | A | - | Human | 4329 | |
| CDK2 | CDK | CMGC | 3r8l | A | A | (5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4186 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb7 | A | A | naphtho[2,1-b:7,8-b']difuran-2,9-dicarboxylic acid | Human | 5448 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmr | A | A | ~{n}'-[(3-chloranyl-4-phenyl-phenyl)methyl]butane-1,4-diamine | Human | 7668 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tei | B | A | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12460 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn2 | A | A | - | Human | 10698 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9k | A | B | 1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diol | Human | 9695 | |
| CDK2 | CDK | CMGC | 1gih | A | | 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-urea | Human | 3922 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3rps | B | | - | Human | 5450 | |
| CLK3 | CLK | CMGC | 2exe | A | B | - | Human | 1819 | |
| CLK3 | CLK | CMGC | 6rct | B | A | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11128 | |
| CLK3 | CLK | CMGC | 6z55 | A | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12298 | |
| CLK3 | CLK | CMGC | 6yu1 | c | A | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12405 | |
| CDK2 | CDK | CMGC | 1f5q | C | A | - | Human | 4281 | |
| CLK3 | CLK | CMGC | 6yty | A | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12406 | |
| CLK3 | CLK | CMGC | 6ytw | A | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12407 | |
| CDK2 | CDK | CMGC | 8erd | A | A | (2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanone | Human | 14949 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5kwh | B | A | ~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 8618 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv7 | A | | 1-[1-(3-aminophenyl)-3-tert-butyl-1h-pyrazol-5-yl]-3-naphthalen-1-ylurea | Human | 5223 | |
| CDK2 | CDK | CMGC | 8ern | A | A | n,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamide | Human | 14948 | |
| CDK2 | CDK | CMGC | 8ern | A | B | n,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamide | Human | 14950 | |
| CDK2 | CDK | CMGC | 3pxf | A | A | 8-anilino-1-naphthalene sulfonate | Human | 4047 | |
| CDK2 | CDK | CMGC | 8erd | A | B | (2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanone | Human | 14951 | |
| SRPK2 | SRPK | CMGC | 7zkx | A | A | n-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamide | Human | 14617 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2no3 | A | | 2-({2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}amino)benzamide | Human | 4640 | |
| SRPK2 | SRPK | CMGC | 5myv | C | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7580 | |
| CDK2 | CDK | CMGC | 4eoq | C | A | adenosine-5'-triphosphate | Human | 4004 | |
| CDK2 | CDK | CMGC | 5fp5 | A | | 4-fluorobenzoic acid | Human | 6285 | |
| CDK2 | CDK | CMGC | 2vtj | A | | 4-[(6-chloropyrazin-2-yl)amino]benzenesulfonamide | Human | 3959 | |
| CDK2 | CDK | CMGC | 7s9x | A | B | 2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acid | Human | 14431 | |
| CDK2 | CDK | CMGC | 6guf | C | | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 10762 | |
| CDK2 | CDK | CMGC | 2uzb | A | D | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamide | Human | 3866 | |
| CDK2 | CDK | CMGC | 6gva | A | B | 5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | 11204 | |
| CDK2 | CDK | CMGC | 2c6k | A | | 4-{[5-(cyclohexylamino)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 6773 | |
| CDK2 | CDK | CMGC | 1pkd | A | | 7-hydroxystaurosporine | Human | 4170 | |
| CDK2 | CDK | CMGC | 6q48 | A | C | 4-iodanyl-3~{h}-pyridin-2-one | Human | 11196 | |
| CDK2 | CDK | CMGC | 6q3b | A | A | 4-iodopyrazole | Human | 11177 | |
| CDK2 | CDK | CMGC | 1h25 | C | | - | Human | 4112 | |
| CDK2 | CDK | CMGC | 3pj8 | A | A | (2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-ol | Human | 4375 | |
| CDK2 | CDK | CMGC | 2c5x | A | A | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 4312 | |
| CDK2 | CDK | CMGC | 3sw7 | A | B | n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamine | Human | 4584 | |
| CDK2 | CDK | CMGC | 3rah | A | B | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | 4206 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8pvo | A | | 2-[1-(1,3-benzothiazol-6-ylsulfonyl)piperidin-4-yl]-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 14976 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v62 | A | B | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 8262 | |
| DYRK1A | DYRK | CMGC | 4mq2 | D | A | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3757 | |
| CDK2 | CDK | CMGC | 1pxm | A | A | 3-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-ylamino]-phenol | Human | 3944 | |
| CDK2 | CDK | CMGC | 4bgh | A | A | 4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamide | Human | 4073 | |
| CDK2 | CDK | CMGC | 3bhv | C | A | 9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-ol | Human | 4353 | |
| CDK2 | CDK | CMGC | 2x1n | C | B | 2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amine | Human | 4062 | |
| CDK8 | CDK | CMGC | 5fgk | A | B | 8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-one | Human | 6388 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8pvp | A | | ~{n}-[5-[(3-chloranyl-4-phenyl-phenyl)methylamino]pentyl]isoquinoline-5-sulfonamide | Human | 14977 | |
| CDK2 | CDK | CMGC | 3qrt | A | A | (5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 4586 | |
| CDK2 | CDK | CMGC | 3rak | A | A | 4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 4574 | |
| CDK8 | CDK | CMGC | 4f70 | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[2-(morpholin-4-yl)ethyl]urea | Human | 3852 | |
| CDK6 | CDK | CMGC | 3nux | A | | 4-[5-chloro-3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amine | Human | 2807 | |
| MAPK14 (p38a) | MAPK | CMGC | 2baj | A | | 1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2,3-dichlorophenyl)urea | Human | 5176 | |
| CDK8 | CDK | CMGC | 5xqx | A | | n-methyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamide | Human | 8313 | |
| CDK6 | CDK | CMGC | 5l2t | A | | 7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 6992 | |
| MAPK14 (p38a) | MAPK | CMGC | 3obj | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 4994 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4g6o | A | | 4-{4-[4-(aminomethyl)-3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamide | Human | 2565 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | A | tak-715 | Human | 5033 | |
| DYRK1A | DYRK | CMGC | 5a4l | B | B | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6735 | |
| MAPK14 (p38a) | MAPK | CMGC | 2i0h | A | A | 2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dione | Human | 5062 | |
| CDK2 | CDK | CMGC | 5iev | A | A | roniciclib | Human | 6567 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao7 | A | A | ~{n}-[(1-methylindazol-6-yl)methyl]propanamide | Human | 14389 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoi | A | B | 1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-one | Human | 14393 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aac | A | | n-isoxazol-3-yl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxo-quinazolin-3-yl]benzamide | Human | 5048 | |
| MAPK14 (p38a) | MAPK | CMGC | 1r3c | A | B | - | Human | 4996 | |
| CDK2 | CDK | CMGC | 3qqh | A | B | 2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenol | Human | 4533 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8p06 | A | | 7-(cyclopropylamino)-5-[[2-(1,2,4-triazol-4-yl)pyridin-4-yl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 14813 | |
| MAPK14 (p38a) | MAPK | CMGC | 3c5u | A | | 6-[4-(2-fluorophenyl)-1,3-oxazol-5-yl]-n-(1-methylethyl)-1,3-benzothiazol-2-amine | Human | 5125 | |
| CDK2 | CDK | CMGC | 3rkb | A | B | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4039 | |
| CDK2 | CDK | CMGC | 4ek6 | A | B | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamide | Human | 4056 | |
| CDK2 | CDK | CMGC | 4eor | C | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4221 | |
| CDK2 | CDK | CMGC | 3r83 | A | A | 4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamide | Human | 4234 | |
| CDK2 | CDK | CMGC | 2clx | A | B | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 3880 | |
| MAPK14 (p38a) | MAPK | CMGC | 3oc1 | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5019 | |
| CDK2 | CDK | CMGC | 5uq2 | A | | - | Human | 8221 | |
| CDK2 | CDK | CMGC | 3r1s | A | B | 2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamide | Human | 4358 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv4 | A | A | 9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrile | Human | 2623 | |
| CDK2 | CDK | CMGC | 3pxy | A | B | 2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenol | Human | 3904 | |
| CDK2 | CDK | CMGC | 6q3f | A | A | - | Human | 11181 | |
| CDK2 | CDK | CMGC | 3qx4 | A | B | 4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 3990 | |
| CDK2 | CDK | CMGC | 5cyi | A | A | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | 6052 | |
| CDK2 | CDK | CMGC | 4cfx | A | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4485 | |
| CDK2 | CDK | CMGC | 3r6x | A | A | 4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4398 | |
| CDK2 | CDK | CMGC | 2g9x | A | | 3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-ol | Human | 3883 | |
| CDK2 | CDK | CMGC | 3r8v | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | 4191 | |
| CDK2 | CDK | CMGC | 2a4l | A | | r-roscovitine | Human | 4238 | |
| CDK2 | CDK | CMGC | 3s00 | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanone | Human | 4248 | |
| CDK2 | CDK | CMGC | 1ke5 | A | | n-methyl-4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamide | Human | 4376 | |
| CDK2 | CDK | CMGC | 4nj3 | A | A | 6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | 4075 | |
| CDK2 | CDK | CMGC | 1gy3 | A | | adenosine-5'-triphosphate | Human | 3978 | |
| CDK2 | CDK | CMGC | 1jst | C | | adenosine-5'-triphosphate | Human | 4356 | |
| CDK2 | CDK | CMGC | 1h1p | A | | 6-o-cyclohexylmethyl guanine | Human | 4309 | |
| CDK2 | CDK | CMGC | 9esj | A | B | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid | Human | 15905 | |
| CDK2 | CDK | CMGC | 9esy | A | B | 4-bromanyl-1,8-naphthyridine | Human | 15906 | |
| CDK2 | CDK | CMGC | 6rij | C | B | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | 12622 | |
| CDK2 | CDK | CMGC | 7s84 | A | A | 2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acid | Human | 14424 | |
| CDK2 | CDK | CMGC | 6q4j | A | A | 2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acid | Human | 11209 | |
| CDK2 | CDK | CMGC | 2bhe | A | | (2z)-5'-bromo-2,3'-biindole-2',3(1h,1'h)-dione ammoniate | Human | 4184 | |
| CDK2 | CDK | CMGC | 1ol2 | C | | - | Human | 4497 | |
| CDK2 | CDK | CMGC | 6q4c | A | B | 4-bromanyl-1,8-naphthyridine | Human | 11207 | |
| CDK2 | CDK | CMGC | 4rj3 | A | B | 1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | 4127 | |
| CDK2 | CDK | CMGC | 1pf8 | A | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 3861 | |
| CDK2 | CDK | CMGC | 1hcl | A | A | - | Human | 4545 | |
| CDK2 | CDK | CMGC | 1b38 | A | | adenosine-5'-triphosphate | Human | 4483 | |
| CDK2 | CDK | CMGC | 1g5s | A | | 2-[trans-(4-aminocyclohexyl)amino]-6-(benzyl-amino)-9-cyclopentylpurine | Human | 3888 | |
| CDK2 | CDK | CMGC | 4ek3 | A | A | - | Human | 3971 | |
| CDK2 | CDK | CMGC | 3r8u | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | 3926 | |
| CDK2 | CDK | CMGC | 4eoi | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4307 | |
| CDK2 | CDK | CMGC | 1h1r | A | B | 6-cyclohexylmethoxy-2-(3'-chloroanilino) purine | Human | 4494 | |
| CDK2 | CDK | CMGC | 4eon | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4326 | |
| CDK2 | CDK | CMGC | 3qtx | A | B | 4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4419 | |
| CDK2 | CDK | CMGC | 4cfu | A | B | 3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acid | Human | 4308 | |
| CDK2 | CDK | CMGC | 6q4c | A | C | 4-bromanyl-1,8-naphthyridine | Human | 11201 | |
| CDK2 | CDK | CMGC | 5anj | A | | n-(9h-purin-6-yl)thiophene-2-carboxamide | Human | 6541 | |
| CDK8 | CDK | CMGC | 6tpa | A | | 1-[4-chloranyl-3-(trifluoromethyl)phenyl]-3-(5-oxidanylidene-6-pyridin-4-yl-pyrido[2,3-b][1,5]benzoxazepin-9-yl)urea | Human | 13160 | |
| CDK2 | CDK | CMGC | 2v22 | A | | - | Human | 4077 | |
| CDK2 | CDK | CMGC | 7b5r | L | | - | Human | 13265 | |
| CDK2 | CDK | CMGC | 4fki | A | B | n-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamide | Human | 4272 | |
| CDK8 | CDK | CMGC | 5xs2 | A | B | 3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamide | Human | 8314 | |
| CDK2 | CDK | CMGC | 2iw6 | A | | [(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrile | Human | 4019 | |
| CDK8 | CDK | CMGC | 4crl | A | | cortistatin a | Human | 6096 | |
| CDK8 | CDK | CMGC | 4g6l | A | | - | Human | 3851 | |
| CLK1 | CLK | CMGC | 6khd | B | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11644 | |
| CDK2 | CDK | CMGC | 4eon | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4153 | |
| CLK1 | CLK | CMGC | 7ak3 | A | A | ~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 13142 | |
| MAPK14 (p38a) | MAPK | CMGC | 3obg | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5211 | |
| CDK8 | CDK | CMGC | 5idp | A | A | (3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanone | Human | 7317 | |
| CDK8 | CDK | CMGC | 5fgk | A | A | 8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-one | Human | 6391 | |
| CDK8 | CDK | CMGC | 6r3s | A | B | 6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamide | Human | 12141 | |
| CDK8 | CDK | CMGC | 5hvy | A | A | n-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}urea | Human | 6553 | |
| CLK1 | CLK | CMGC | 7opg | A | B | 4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenol | Human | 13809 | |
| CDK2 | CDK | CMGC | 8bya | A | | - | Human | 14814 | |
| CDK2 | CDK | CMGC | 8bzo | A | | - | Human | 14815 | |
| CDK2 | CDK | CMGC | 3rni | A | B | 3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 4420 | |
| CDK2 | CDK | CMGC | 3qhr | A | | adenosine-5'-diphosphate | Human | 4458 | |
| CDK2 | CDK | CMGC | 2v0d | A | | 2-imino-5-(1-pyridin-2-yl-meth-(e)-ylidene)-1,3-thiazolidin-4-one | Human | 4327 | |
| CDK2 | CDK | CMGC | 2wih | A | | n,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4163 | |
| CDK2 | CDK | CMGC | 5oo1 | A | | ~{n}-(4-pyrimidin-2-ylphenyl)propanamide | Human | 10566 | |
| DYRK2 | DYRK | CMGC | 7dh9 | A | | [2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridin-4-yl]methanol | Human | 13976 | |
| CDK8 | CDK | CMGC | 5hbj | A | A | 8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-one | Human | 6390 | |
| CDK8 | CDK | CMGC | 4f6u | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]urea | Human | 3849 | |
| CDK8 | CDK | CMGC | 4f7j | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)urea | Human | 3843 | |
| CDK8 | CDK | CMGC | 4f7s | A | B | n-(2-phenylethyl)quinazolin-4-amine | Human | 3853 | |
| CDK8 | CDK | CMGC | 5bnj | A | | 8-{3-chloro-5-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]pyridin-4-yl}-2,8-diazaspiro[4.5]decan-1-one | Human | 6152 | |
| CDK9 | CDK | CMGC | 6cyt | A | | - | Human | 10797 | |
| CDK9 | CDK | CMGC | 4bci | A | | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 2243 | |
| CDK9 | CDK | CMGC | 3mia | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2242 | |
| MAPK7 (Erk5) | MAPK | CMGC | 6hkm | A | | [4-(6,7-dimethoxyquinazolin-4-yl)piperidin-1-yl]-[4-(trifluoromethyloxy)phenyl]methanone | Human | 10917 | |
| CDK9 | CDK | CMGC | 3mi9 | A | | - | Human | 2239 | |
| CLK1 | CLK | CMGC | 5j1v | B | | pyrido[3,4-g]quinazoline-2,10-diamine | Human | 6580 | |
| CDK2 | CDK | CMGC | 3ddp | A | B | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 6780 | |
| CDK2 | CDK | CMGC | 5ane | A | | 6-methoxy-9h-purine | Human | 6542 | |
| CDK2 | CDK | CMGC | 1h1q | A | | 2-anilino-6-cyclohexylmethoxypurine | Human | 4195 | |
| CDK2 | CDK | CMGC | 3ezv | A | | 4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}aniline | Human | 4083 | |
| CDK8 | CDK | CMGC | 3rgf | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 3841 | |
| CDK9 | CDK | CMGC | 4ogr | I | | adenosine | Human | 2241 | |
| CDK8 | CDK | CMGC | 5hnb | A | A | [6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanone | Human | 6562 | |
| CDK8 | CDK | CMGC | 6qtg | A | | 2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]-~{n},~{n}-dimethyl-ethanamide | Human | 12094 | |
| CLK1 | CLK | CMGC | 6r6e | A | | 5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amine | Human | 12232 | |
| CDK2 | CDK | CMGC | 1h1s | A | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4400 | |
| CDK8 | CDK | CMGC | 4f7n | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(5-hydroxypentyl)urea | Human | 3847 | |
| CDK9 | CDK | CMGC | 3tn8 | A | | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 2240 | |
| CDK9 | CDK | CMGC | 4ec9 | A | | - | Human | 2234 | |
| CDK9 | CDK | CMGC | 4imy | A | B | adenosine monophosphate | Human | 2252 | |
| CDK9 | CDK | CMGC | 5l1z | A | | - | Human | 7121 | |
| CDK9 | CDK | CMGC | 6w9e | A | A | (4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone | Human | 13859 | |
| CLK1 | CLK | CMGC | 1z57 | A | A | debromohymenialdisine | Human | 106 | |
| CLK1 | CLK | CMGC | 6i5k | C | A | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10834 | |
| CDK8 | CDK | CMGC | 5i5z | A | | n-methyl-8-(1-methyl-2,2-dioxo-2,3-dihydro-1h-2lambda~6~,1-benzothiazol-5-yl)-1,6-naphthyridine-2-carboxamide | Human | 6536 | |
| CDK8 | CDK | CMGC | 5idn | A | A | [(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanone | Human | 7322 | |
| CDK9 | CDK | CMGC | 6z45 | A | | (1~{s},3~{r})-3-acetamido-~{n}-[5-chloranyl-4-(5,5-dimethyl-4,6-dihydropyrrolo[1,2-b]pyrazol-3-yl)pyridin-2-yl]cyclohexane-1-carboxamide | Human | 13115 | |
| CDK9 | CDK | CMGC | 3blr | A | | 2-(2-chloro-phenyl)-5,7-dihydroxy-8-(3-hydroxy-1-methyl-piperidin-4-yl)-4h-benzopyran-4-one | Human | 2236 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mz3 | A | B | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | 8681 | |
| MAPK14 (p38a) | MAPK | CMGC | 5wjj | A | A | n-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamide | Human | 9514 | |
| CDK2 | CDK | CMGC | 3r8z | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanone | Human | 4137 | |
| CDK8 | CDK | CMGC | 5hbh | A | | 5-[5-chloranyl-4-[1-(2-methoxyethyl)-1,8-diazaspiro[4.5]decan-8-yl]pyridin-3-yl]-1-methyl-3~{h}-2,1-benzothiazole 2,2-dioxide | Human | 6387 | |
| CDK8 | CDK | CMGC | 5icp | A | B | [(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanone | Human | 7321 | |
| CDK8 | CDK | CMGC | 6y0a | A | A | 6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamide | Human | 13306 | |
| CDK8 | CDK | CMGC | 5hbe | A | A | 8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one | Human | 6389 | |
| CDK2 | CDK | CMGC | 1vyz | A | | n-(5-cyclopropyl-1h-pyrazol-3-yl)benzamide | Human | 4325 | |
| CDK9 | CDK | CMGC | 4imy | E | B | adenosine monophosphate | Human | 2256 | |
| CDK9 | CDK | CMGC | 6gzh | A | | [4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azanium | Human | 10427 | |
| CDK9 | CDK | CMGC | 3blq | A | | adenosine-5'-triphosphate | Human | 2248 | |
| CDK9 | CDK | CMGC | 6w9e | A | C | (4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone | Human | 13861 | |
| MAPK9 (JNK2) | MAPK | CMGC | 8elc | A | | 4-(dimethylamino)-n-{4-[(3s)-3-({4-[(8r)-2-phenylpyrazolo[1,5-a]pyridin-3-yl]pyrimidin-2-yl}amino)pyrrolidine-1-carbonyl]phenyl}butanamide | Human | 14816 | |
| CDK2 | CDK | CMGC | 2x1n | A | B | 2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amine | Human | 4078 | |
| CDK1 (CDC2) | CDK | CMGC | 5lqf | A | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 7364 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | A | B | - | Human | 4616 | |
| CDK1 (CDC2) | CDK | CMGC | 5lqf | D | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 7367 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu7 | C | | - | Human | 10775 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc3 | A | B | - | Human | 6554 | |
| CDK2 | CDK | CMGC | 4ii5 | A | A | adenosine-5'-diphosphate | Human | 3930 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4awi | A | A | n-(1,1-dioxidotetrahydro-2h-thiopyran-4-yl)-4-[2-(1-methylethyl)-1h-pyrrolo[2,3-b]pyridin-4-yl]benzenesulfonamide | Human | 4661 | |
| MAPK8 (JNK1) | MAPK | CMGC | 6f5e | B | | - | Human | 9078 | |
| DYRK1A | DYRK | CMGC | 6eip | C | | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | 10533 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fso | X | | - | Human | 5117 | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | A | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | 5006 | |
| MAPK8 (JNK1) | MAPK | CMGC | 5lw1 | H | | adenosine | Human | 9080 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 4656 | |
| MAPK8 (JNK1) | MAPK | CMGC | 11zl | A | A | (4m)-n-[4-hydroxy-3-(pyrrolidine-1-carbonyl)phenyl]-4-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1-benzothiophene-2-carboxamide | Human | 15534 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4e73 | A | B | methyl 3-(4-{[(1r,2s,3s,5s,7s)-5-aminotricyclo[3.3.1.1~3,7~]dec-2-yl]carbamoyl}benzyl)-4-oxo-1-phenyl-1,4-dihydro-1,8-naphthyridine-2-carboxylate | Human | 4669 | |
| MAPK8 (JNK1) | MAPK | CMGC | 5lw1 | E | | adenosine | Human | 9079 | |
| CDK2 | CDK | CMGC | 4eos | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4181 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | E | B | - | Human | 6454 | |
| CLK1 | CLK | CMGC | 6i5l | B | B | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10839 | |
| CDK2 | CDK | CMGC | 2r3i | A | C | - | Human | 4317 | |
| CDK2 | CDK | CMGC | 3ql8 | A | B | 3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrile | Human | 4306 | |
| CDK2 | CDK | CMGC | 3r8u | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanone | Human | 3864 | |
| CDK2 | CDK | CMGC | 3tiz | A | | 1-{(e)-[(4-hydroxyphenyl)imino]methyl}naphthalen-2-ol | Human | 4136 | |
| CDK2 | CDK | CMGC | 4eos | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4340 | |
| CDK2 | CDK | CMGC | 3qtu | A | B | 4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4323 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | C | B | - | Human | 4611 | |
| DYRK1A | DYRK | CMGC | 6t6a | A | B | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11858 | |
| DYRK1A | DYRK | CMGC | 6eij | B | | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | 10516 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh2 | A | | - | Human | 4985 | |
| CDK2 | CDK | CMGC | 3ej1 | C | | n-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amine | Human | 4092 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otd | B | B | [2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azanium | Human | 9632 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cs6 | A | A | - | Human | 6915 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osr | A | A | adenosine-5'-triphosphate | Human | 10601 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5wp1 | A | B | 5,7-dihydroxy-4h-1-benzopyran-4-one | Human | 10440 | |
| CDK2 | CDK | CMGC | 3qqk | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 4514 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3o17 | B | | - | Human | 4667 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | A | B | - | Human | 6448 | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | B | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 1717 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mov | A | A | 4'-hydroxycinnamic acid | Human | 7655 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3at4 | A | | [1-(6-{6-[(1-methylethyl)amino]-1h-indazol-1-yl}pyrazin-2-yl)-1h-pyrrol-3-yl]acetic acid | Human | 5413 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6fvg | A | B | adenosine-5'-triphosphate | Human | 11339 | |
| CDK5 | CDK | CMGC | 1unh | B | | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | 2787 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3o2m | A | | - | Human | 4676 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | D | A | phosphoaminophosphonic acid-adenylate ester | Human | 4627 | |
| CDK2 | CDK | CMGC | 2vti | A | | n-(4-sulfamoylphenyl)-1h-indazole-3-carboxamide | Human | 4177 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgb | A | A | 5,6-dibromobenzotriazole | Human | 14468 | |
| DYRK1A | DYRK | CMGC | 7ak2 | A | | 4-[2-methyl-3-(2-pyridin-2-yloxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13593 | |
| CDK2 | CDK | CMGC | 3r8p | A | A | (5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4232 | |
| CDK8 | CDK | CMGC | 4f6s | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 3848 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgb | A | B | 5,6-dibromobenzotriazole | Human | 14470 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgd | A | B | 5,6-dibromobenzotriazole | Human | 14471 | |
| CDK2 | CDK | CMGC | 3bhu | A | A | 4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4105 | |
| CDK2 | CDK | CMGC | 1f5q | A | A | - | Human | 4194 | |
| SRPK2 | SRPK | CMGC | 5myv | C | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7571 | |
| SRPK2 | SRPK | CMGC | 5myv | D | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7578 | |
| SRPK2 | SRPK | CMGC | 5myv | A | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7579 | |
| CDK2 | CDK | CMGC | 1ol1 | A | | - | Human | 4429 | |
| CDK2 | CDK | CMGC | 6q4h | A | B | 2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acid | Human | 11190 | |
| CLK1 | CLK | CMGC | 6ft9 | B | B | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9894 | |
| CLK1 | CLK | CMGC | 6i5l | A | A | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10837 | |
| CLK1 | CLK | CMGC | 6g33 | C | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9825 | |
| CLK1 | CLK | CMGC | 6i5l | B | A | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10846 | |
| CLK1 | CLK | CMGC | 6ft9 | B | A | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9897 | |
| CLK1 | CLK | CMGC | 6z50 | A | B | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12308 | |
| CLK1 | CLK | CMGC | 8p04 | A | | (4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-one | Human | 14741 | |
| CDK2 | CDK | CMGC | 2c6o | A | | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 6783 | |
| CDK2 | CDK | CMGC | 5osm | A | B | methyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylate | Human | 9740 | |
| CDK7 | CDK | CMGC | 7b5q | J | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13277 | |
| CLK3 | CLK | CMGC | 2wu7 | A | B | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 1827 | |
| CLK1 | CLK | CMGC | 5j1w | B | B | pyrido[3,4-g]quinazolin-2-amine | Human | 6583 | |
| CLK1 | CLK | CMGC | 5j1v | C | | pyrido[3,4-g]quinazoline-2,10-diamine | Human | 6577 | |
| CLK1 | CLK | CMGC | 6g33 | C | C | - | Human | 9820 | |
| CLK1 | CLK | CMGC | 6r3d | A | | 4-[6,7-bis(chloranyl)-1~{h}-indol-3-yl]pyrimidin-2-amine | Human | 12128 | |
| CDK5 | CDK | CMGC | 3o0g | B | | {4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanone | Human | 2783 | |
| CLK1 | CLK | CMGC | 6ft8 | A | A | 3-(3-hydroxyphenyl)-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9895 | |
| CLK1 | CLK | CMGC | 6g33 | B | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9822 | |
| CLK1 | CLK | CMGC | 6i5l | C | A | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10833 | |
| CLK1 | CLK | CMGC | 6raa | A | A | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11014 | |
| CLK1 | CLK | CMGC | 6i5k | B | B | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10835 | |
| CLK1 | CLK | CMGC | 6r8j | A | A | 4-(1-methylindol-3-yl)pyrimidin-2-amine | Human | 12632 | |
| CLK1 | CLK | CMGC | 6z4z | B | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12311 | |
| CLK1 | CLK | CMGC | 6i5k | B | A | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10842 | |
| CDK2 | CDK | CMGC | 3qu0 | A | A | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4427 | |
| CDK2 | CDK | CMGC | 2r3m | A | A | n-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amine | Human | 4286 | |
| CDK2 | CDK | CMGC | 5oo0 | A | A | - | Human | 9744 | |
| DYRK2 | DYRK | CMGC | 5ztn | A | | (1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | Human | 10482 | |
| DYRK2 | DYRK | CMGC | 7dhn | A | | 7-methoxy-2-methylsulfanyl-9-(piperidin-4-ylmethylsulfanyl)-[1,3]thiazolo[5,4-b]quinoline | Human | 13971 | |
| DYRK2 | DYRK | CMGC | 5lxd | A | B | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7128 | |
| CLK1 | CLK | CMGC | 5j1w | C | B | pyrido[3,4-g]quinazolin-2-amine | Human | 6581 | |
| CLK1 | CLK | CMGC | 5x8i | B | | 5-[1-[(1s)-1-(4-fluorophenyl)ethyl]-[1,2,3]triazolo[4,5-c]quinolin-8-yl]-1,3-benzoxazole | Human | 8317 | |
| CLK1 | CLK | CMGC | 6fyo | A | A | 6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamide | Human | 10324 | |
| CDK2 | CDK | CMGC | 3ig7 | A | | n-{1-[cis-3-(acetylamino)cyclobutyl]-1h-imidazol-4-yl}-2-(4-methoxyphenyl)acetamide | Human | 4021 | |
| DYRK2 | DYRK | CMGC | 4azf | A | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3146 | |
| CLK1 | CLK | CMGC | 7oa0 | A | | 5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amine | Human | 14207 | |
| CLK1 | CLK | CMGC | 6i5k | A | A | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10844 | |
| CLK1 | CLK | CMGC | 6yte | C | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12422 | |
| CLK1 | CLK | CMGC | 6z50 | A | A | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12314 | |
| CLK1 | CLK | CMGC | 6i5k | C | B | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10838 | |
| CDK2 | CDK | CMGC | 3qx2 | A | A | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamide | Human | 4031 | |
| CDK2 | CDK | CMGC | 4eoj | C | B | adenosine-5'-triphosphate | Human | 4311 | |
| CDK2 | CDK | CMGC | 4fkp | A | B | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4313 | |
| DYRK2 | DYRK | CMGC | 3k2l | A | B | - | Human | 3145 | |
| DYRK2 | DYRK | CMGC | 3k2l | A | A | - | Human | 3147 | |
| DYRK2 | DYRK | CMGC | 7dho | A | | 2-methoxy-9-(piperidin-4-ylmethylsulfanyl)-7-propan-2-yloxy-acridine | Human | 13972 | |
| DYRK2 | DYRK | CMGC | 7ejv | A | B | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | 14181 | |
| DYRK2 | DYRK | CMGC | 7ejv | A | A | [6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanone | Human | 14180 | |
| CLK1 | CLK | CMGC | 6khd | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11646 | |
| CLK1 | CLK | CMGC | 6tw2 | E | B | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 11963 | |
| CLK1 | CLK | CMGC | 6i5i | A | A | 5-(1-methylpyrazol-4-yl)-3-[1-(phenylmethyl)pyrazol-4-yl]furo[3,2-b]pyridine | Human | 10845 | |
| CLK1 | CLK | CMGC | 6z4z | A | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12315 | |
| CLK1 | CLK | CMGC | 6q8k | A | B | ~{n}2-(3-morpholin-4-ylpropyl)pyrido[3,4-g]quinazoline-2,10-diamine | Human | 10903 | |
| CLK1 | CLK | CMGC | 6ft9 | C | A | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9896 | |
| CLK1 | CLK | CMGC | 8p08 | A | | (4~{z})-4-(1,3-benzothiazol-6-ylmethylidene)-2-[[(2~{r})-1-methoxy-4-methyl-pentan-2-yl]amino]-1~{h}-imidazol-5-one | Human | 14742 | |
| CLK1 | CLK | CMGC | 6q8p | A | | ~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amine | Human | 10899 | |
| DYRK2 | DYRK | CMGC | 4azf | A | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3144 | |
| CDK2 | CDK | CMGC | 3qru | A | B | (5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 4516 | |
| CDK2 | CDK | CMGC | 2wma | A | | - | Human | 4435 | |
| CDK2 | CDK | CMGC | 6guc | A | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 10767 | |
| DYRK2 | DYRK | CMGC | 7dg4 | A | | 2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine | Human | 13967 | |
| DYRK2 | DYRK | CMGC | 6hdr | A | B | curcumin | Human | 11571 | |
| DYRK2 | DYRK | CMGC | 5lxd | A | A | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7124 | |
| DYRK2 | DYRK | CMGC | 7akf | A | B | 4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13614 | |
| DYRK2 | DYRK | CMGC | 5lxc | A | A | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7122 | |
| CDK2 | CDK | CMGC | 2r3g | A | B | 6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amine | Human | 3923 | |
| CDK2 | CDK | CMGC | 3r28 | A | B | 4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamide | Human | 4293 | |
| DYRK2 | DYRK | CMGC | 7akf | A | A | 4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13613 | |
| DYRK2 | DYRK | CMGC | 5lxc | A | B | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7129 | |
| DYRK2 | DYRK | CMGC | 6k0j | A | | 3-(2,7-dimethoxyacridin-9-yl)sulfanylpropan-1-amine | Human | 11817 | |
| MAPK12 (p38g) | MAPK | CMGC | 7cga | A | | - | Human | 13762 | |
| SRPK2 | SRPK | CMGC | 5myv | D | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7572 | |
| CDK2 | CDK | CMGC | 3r1q | A | B | 4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamide | Human | 4507 | |
| CDK2 | CDK | CMGC | 4bzd | A | B | 6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amine | Human | 4490 | |
| CDK2 | CDK | CMGC | 4eor | A | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4205 | |
| CDKL5 | CDKL | CMGC | 4bgq | A | A | [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 1425 | |
| CDKL5 | CDKL | CMGC | 4bgq | A | B | [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 1426 | |
| CDK2 | CDK | CMGC | 3rpo | A | B | 4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acid | Human | 4098 | |
| CDK2 | CDK | CMGC | 2wip | C | | 1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acid | Human | 4190 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc3 | A | A | - | Human | 6555 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4l7f | A | C | n-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamide | Human | 4648 | |
| CDK2 | CDK | CMGC | 3bhu | C | A | 4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4087 | |
| CLK3 | CLK | CMGC | 2eu9 | A | A | - | Human | 1826 | |
| CLK3 | CLK | CMGC | 6khf | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11649 | |
| CLK3 | CLK | CMGC | 6rct | B | B | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11129 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vuk | A | | - | Human | 4659 | |
| CDK2 | CDK | CMGC | 3rjc | A | B | {4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanone | Human | 4469 | |
| CDK2 | CDK | CMGC | 1y8y | A | | (5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-(4-methanesulfonylphenyl)amine | Human | 3914 | |
| CLK3 | CLK | CMGC | 6ytw | A | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12404 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15298 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6slg | A | B | (6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-one | Human | 11816 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6ge0 | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamide | Human | 9961 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7k | A | | 1h-imidazol-2-amine | Human | 10985 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g8x | A | A | 4-chloranyl-1~{h}-indazol-3-amine | Human | 9957 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9d | A | A | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamide | Human | 9972 | |
| MAPK9 (JNK2) | MAPK | CMGC | 3npc | B | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 1237 | |
| CLK3 | CLK | CMGC | 6z55 | B | C | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12297 | |
| CLK3 | CLK | CMGC | 6ft7 | A | A | 3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9905 | |
| CLK3 | CLK | CMGC | 6z52 | A | B | 11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12627 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2h96 | B | | 5-cyano-n-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamide | Human | 4668 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pst | A | B | amp phosphoramidate | Human | 15299 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp3 | A | | (2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-ol | Human | 6084 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp7 | A | | 2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6082 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zxt | A | A | catechol | Human | 6654 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9h | A | A | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamide | Human | 9971 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao2 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)propanamide | Human | 14394 | |
| CDK2 | CDK | CMGC | 6gub | C | | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | 10763 | |
| CDK2 | CDK | CMGC | 4fkj | A | A | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamide | Human | 4387 | |
| CDK2 | CDK | CMGC | 4fks | A | B | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4489 | |
| CLK3 | CLK | CMGC | 6rct | A | B | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11126 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | D | | adenosine-5'-diphosphate | Human | 2578 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvf | A | A | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6031 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lck | A | B | ~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 6836 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9n | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamide | Human | 11413 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fuy | A | A | {4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanone | Human | 2622 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qah | A | B | 1-azanylpropylideneazanium | Human | 11348 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp8 | A | | 2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6087 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7opm | A | B | 1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]urea | Human | 14083 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao7 | A | B | ~{n}-[(1-methylindazol-6-yl)methyl]propanamide | Human | 14398 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao4 | A | B | ~{n}-(1~{h}-indazol-5-yl)ethanesulfonamide | Human | 14399 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zxt | A | B | catechol | Human | 6653 | |
| CDK2 | CDK | CMGC | 1h27 | A | | - | Human | 4116 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | C | B | - | Human | 2627 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7t | A | A | 1,2-oxazol-3-amine | Human | 11350 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g91 | A | B | 5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amine | Human | 9956 | |
| CDK2 | CDK | CMGC | 3r7v | A | A | 5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamide | Human | 4380 | |
| CDK2 | CDK | CMGC | 2c6l | A | | 4-({5-[(4-aminocyclohexyl)amino][1,2,4]triazolo[1,5-a]pyrimidin-7-yl}amino)benzenesulfonamide | Human | 6779 | |
| CDK2 | CDK | CMGC | 1oi9 | A | A | 6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purine | Human | 4033 | |
| CDK2 | CDK | CMGC | 5lmk | A | B | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | 7398 | |
| CDK2 | CDK | CMGC | 4cfu | C | A | 3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acid | Human | 3967 | |
| CDK2 | CDK | CMGC | 4cfv | C | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenol | Human | 3999 | |
| CDK2 | CDK | CMGC | 5uq3 | A | | - | Human | 8222 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6opg | A | | phosphoaminophosphonic acid-adenylate ester | Human | 11507 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao5 | A | B | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamide | Human | 14400 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3tei | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2608 | |
| CDK2 | CDK | CMGC | 6q3c | A | A | 4-bromo-1h-pyrazole | Human | 11191 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g54 | A | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10938 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 2602 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoc | A | B | ~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamide | Human | 14406 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7e75 | A | | - | Human | 14115 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdq | A | A | 4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamide | Human | 9948 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bve | A | B | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6026 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoa | A | B | ~{n}-pyridin-3-ylprop-2-enamide | Human | 14407 | |
| CDK2 | CDK | CMGC | 4erw | A | | staurosporine | Human | 4370 | |
| CDK2 | CDK | CMGC | 2i40 | A | B | 5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamide | Human | 4470 | |
| CDK2 | CDK | CMGC | 4ek5 | A | A | n-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamide | Human | 4037 | |
| CDK2 | CDK | CMGC | 3eid | A | B | (2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-ol | Human | 4424 | |
| CLK3 | CLK | CMGC | 3raw | B | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 1825 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9a | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-one | Human | 11408 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lck | A | A | ~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 6835 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3w55 | A | | (3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dione | Human | 2573 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bue | A | | 1-benzyl-4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-one | Human | 2574 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7xc1 | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14665 | |
| CDK2 | CDK | CMGC | 3rpr | A | A | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanone | Human | 4452 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhf | A | | 2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-5-(phenylmethyl)-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7997 | |
| CDK2 | CDK | CMGC | 5fp6 | A | A | 3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-ol | Human | 6302 | |
| CDK2 | CDK | CMGC | 3r1s | A | A | 2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamide | Human | 4263 | |
| CDK2 | CDK | CMGC | 3qqj | A | A | 2-(4,6-diamino-1,3,5-triazin-2-yl)phenol | Human | 4113 | |
| CLK3 | CLK | CMGC | 6ft7 | B | A | 3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9904 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjb | A | A | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 10832 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoe | A | B | ~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamide | Human | 14411 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v61 | A | B | - | Human | 8266 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2y9q | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 2567 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa3 | A | A | pyrazole | Human | 11353 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rfo | A | | - | Human | 12341 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4xj0 | B | | 1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-one | Human | 6049 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | A | B | - | Human | 2607 | |
| CDK2 | CDK | CMGC | 3s0o | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanone | Human | 3898 | |
| CDK2 | CDK | CMGC | 2g9x | C | | 3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-ol | Human | 4082 | |
| CDK2 | CDK | CMGC | 3rjc | A | A | {4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanone | Human | 4032 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v62 | A | A | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 8264 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp2 | B | | - | Human | 6081 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4n0s | A | B | caffeic acid | Human | 2555 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzm | A | | 7-ethylsulfonyl-n-(oxan-4-yl)-6,8-dihydro-5h-pyrido[3,4-d]pyrimidin-2-amine | Human | 2616 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao3 | A | B | 2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14414 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7t | A | B | 1,2-oxazol-3-amine | Human | 11347 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5k4i | A | | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 6744 | |
| CDK2 | CDK | CMGC | 2iw6 | C | | [(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrile | Human | 4108 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9j | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamide | Human | 9949 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | A | A | - | Human | 2615 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qta | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 2576 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aof | A | A | ~{n}-(2-methylpyrimidin-5-yl)propanamide | Human | 14419 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qf1 | A | A | - | Human | 15020 | |
| CDK2 | CDK | CMGC | 6ath | A | A | - | Human | 10567 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5m4u | A | A | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7390 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmd | A | C | - | Human | 10990 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6te2 | A | A | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12444 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qf1 | A | B | - | Human | 15021 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 3ofm | A | B | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 2730 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7at9 | A | B | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 13829 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8q77 | A | A | (2~{s})-2-[[(2~{s})-2-[[(2~{s})-2-[12-[[4-[[5-(4-carboxyphenyl)-1,3-thiazol-2-yl]amino]-4-oxidanylidene-butanoyl]-(2-hydroxy-2-oxoethyl)amino]dodecanoylamino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]butanedioic acid | Human | 15024 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5yf9 | B | A | nicotinic acid | Human | 11415 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a1z | A | B | 6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13147 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | A | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12117 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qbu | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 15025 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7at9 | A | C | 2-(3,4-dichlorophenyl)ethanamine | Human | 13830 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcg | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15026 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5y9m | A | | nicotinic acid | Human | 9908 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgd | A | A | 5,6-dibromobenzotriazole | Human | 14472 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 9fbi | A | A | nicotinic acid | Human | 15561 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcg | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 15027 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5yf9 | X | A | nicotinic acid | Human | 11417 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6l20 | G | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 11995 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8q9s | A | A | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamide | Human | 15028 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy9 | A | B | 3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrile | Human | 11011 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6l20 | D | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 11996 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy9 | A | A | 3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrile | Human | 11012 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmc | A | B | - | Human | 10993 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmb | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10994 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmq | A | A | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 10991 | |
| CDK2 | CDK | CMGC | 1pye | A | | [2-amino-6-(2,6-difluoro-benzoyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl-methanone | Human | 4284 | |
| CDK2 | CDK | CMGC | 2uue | C | | 4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amine | Human | 4321 | |
| CDK2 | CDK | CMGC | 2r3j | A | A | 3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4185 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmd | A | B | - | Human | 10992 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6l20 | A | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 11993 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcg | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15030 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmd | A | A | 5-[2-(diethylamino)ethyl]-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 10997 | |
| CLK1 | CLK | CMGC | 6khd | B | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11647 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3i5z | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamide | Human | 2579 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoe | A | A | ~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamide | Human | 14395 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5m56 | B | | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7389 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | B | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12114 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7atv | A | A | ~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamide | Human | 13831 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 2585 | |
| CDK2 | CDK | CMGC | 1pxi | A | A | 4-(2,5-dichlorothien-3-yl)pyrimidin-2-amine | Human | 4381 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv5 | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-(5-methyl-2-phenylpyrimidin-4-yl)-1h-pyrrole-2-carboxamide | Human | 2598 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao6 | A | A | ~{n}-(1~{h}-indazol-5-ylmethyl)ethanamide | Human | 14397 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv8 | A | A | 6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-one | Human | 2625 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6dmg | A | A | - | Human | 10811 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5m56 | A | | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7388 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8q9s | A | B | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamide | Human | 15031 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmb | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10995 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 9r57 | A | B | 5,6-dibromobenzotriazole | Human | 15562 | |
| CDK2 | CDK | CMGC | 1okw | C | | - | Human | 3896 | |
| CDK2 | CDK | CMGC | 1pxp | A | A | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 4316 | |
| CDK2 | CDK | CMGC | 1pxl | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4233 | |
| CDK2 | CDK | CMGC | 3le6 | A | | 5-(2-chlorophenyl)-3-methyl-7-nitropyrazolo[3,4-b][1,4]benzodiazepine | Human | 4125 | |
| CDK8 | CDK | CMGC | 3rgf | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 3846 | |
| CLK3 | CLK | CMGC | 6fyr | A | A | 6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamide | Human | 11407 | |
| CLK3 | CLK | CMGC | 6yu1 | c | B | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12411 | |
| CLK3 | CLK | CMGC | 6ytw | B | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12412 | |
| CLK3 | CLK | CMGC | 6ft7 | B | B | 3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9902 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qbu | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 15029 | |
| CDK2 | CDK | CMGC | 3ns9 | A | | (2s,3s)-3-{[7-(benzylamino)-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-5-yl]amino}butane-1,2,4-triol | Human | 4575 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzn | A | A | 2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamide | Human | 2605 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9h | A | B | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamide | Human | 9958 | |
| CDK8 | CDK | CMGC | 5cei | A | B | 4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamide | Human | 6403 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6slg | A | A | (6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-one | Human | 11815 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjb | A | B | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 10831 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aob | A | B | ~{n}-[(1-methylindazol-3-yl)methyl]propanamide | Human | 14413 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rq4 | A | A | 6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-one | Human | 11854 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zyk | A | B | adenosine-5'-diphosphate | Human | 14546 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qgc | A | B | 5,6-dibromobenzotriazole | Human | 14434 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | C | A | phosphoaminophosphonic acid-adenylate ester | Human | 4644 | |
| CDK2 | CDK | CMGC | 5cyi | C | B | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | 6053 | |
| CDK2 | CDK | CMGC | 3qxp | A | B | 4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4482 | |
| CDK2 | CDK | CMGC | 4ek8 | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amine | Human | 4079 | |
| CDK2 | CDK | CMGC | 3rm7 | A | A | 2-[(4-hydroxybenzyl)amino]-5-nitrobenzamide | Human | 3893 | |
| CDK2 | CDK | CMGC | 2uzb | A | C | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamide | Human | 4099 | |
| CDK2 | CDK | CMGC | 3pxy | A | A | 2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenol | Human | 4057 | |
| CDK2 | CDK | CMGC | 4cfw | A | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4280 | |
| CDK2 | CDK | CMGC | 1oi9 | A | B | 6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purine | Human | 4492 | |
| CDK2 | CDK | CMGC | 3qzi | A | A | 4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamide | Human | 4094 | |
| CDK2 | CDK | CMGC | 3qrt | A | B | (5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 4536 | |
| CDK2 | CDK | CMGC | 5uq1 | C | | - | Human | 8223 | |
| CDK2 | CDK | CMGC | 3r7i | A | A | 4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acid | Human | 4450 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 3e3b | X | | [1-(6-{6-[(1-methylethyl)amino]-1h-indazol-1-yl}pyrazin-2-yl)-1h-pyrrol-3-yl]acetic acid | Human | 2729 | |
| CDK2 | CDK | CMGC | 4fkl | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4583 | |
| CDK2 | CDK | CMGC | 6yl6 | A | A | - | Human | 12498 | |
| CDK2 | CDK | CMGC | 2r3l | A | B | 3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amine | Human | 4085 | |
| CDK2 | CDK | CMGC | 8fp0 | A | B | r-roscovitine | Human | 14756 | |
| CDK2 | CDK | CMGC | 8fp5 | A | B | adenosine-5'-triphosphate | Human | 14757 | |
| CDK2 | CDK | CMGC | 8fp0 | A | A | r-roscovitine | Human | 14758 | |
| CDK2 | CDK | CMGC | 8fow | A | A | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 14759 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a2h | A | B | 5,6,7-tris(bromanyl)-1~{h}-imidazo[4,5-b]pyridine | Human | 13146 | |
| CDK2 | CDK | CMGC | 8fow | A | B | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 14760 | |
| CDK2 | CDK | CMGC | 8fp5 | A | A | adenosine-5'-triphosphate | Human | 14761 | |
| CDK2 | CDK | CMGC | 3f5x | A | | 4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}aniline | Human | 3882 | |
| CDK2 | CDK | CMGC | 3qhr | C | | adenosine-5'-diphosphate | Human | 3879 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | D | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12118 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | C | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12119 | |
| CDK2 | CDK | CMGC | 4bcq | C | B | 4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrile | Human | 4120 | |
| CDK2 | CDK | CMGC | 3bht | A | A | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 3950 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3oxi | A | | methyl 3-[(thiophen-2-ylacetyl)amino]thiophene-2-carboxylate | Human | 3423 | |
| CDK2 | CDK | CMGC | 2r3r | A | A | 3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4040 | |
| CDK2 | CDK | CMGC | 1ogu | A | A | 4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamide | Human | 3965 | |
| CDK2 | CDK | CMGC | 2wev | C | B | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 3859 | |
| CDK2 | CDK | CMGC | 3r8m | A | A | 1h-indazole-3-carbohydrazide | Human | 4111 | |
| CLK3 | CLK | CMGC | 6z2v | A | A | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12637 | |
| CLK3 | CLK | CMGC | 6z55 | A | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12302 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | C | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10505 | |
| CDK2 | CDK | CMGC | 1oiy | A | A | 4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamide | Human | 4225 | |
| CDK2 | CDK | CMGC | 2j9m | A | A | 6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxide | Human | 4154 | |
| CDK1 (CDC2) | CDK | CMGC | 5lqf | A | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 7366 | |
| CDK2 | CDK | CMGC | 3py0 | A | A | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 3995 | |
| CDK2 | CDK | CMGC | 2vv9 | A | B | 2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanol | Human | 3881 | |
| CDK2 | CDK | CMGC | 3qzg | A | A | 2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenol | Human | 4144 | |
| CDK2 | CDK | CMGC | 2vv9 | A | A | 2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanol | Human | 3989 | |
| CDK2 | CDK | CMGC | 1h25 | A | | - | Human | 4273 | |
| CDK2 | CDK | CMGC | 3r7e | A | A | 5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamide | Human | 4159 | |
| CDK2 | CDK | CMGC | 2r3n | A | A | 3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4101 | |
| CDK2 | CDK | CMGC | 1fvt | A | | 4-(5-bromo-2-oxo-2h-indol-3-ylazo)-benzenesulfonamide | Human | 4480 | |
| CDK1 (CDC2) | CDK | CMGC | 4y72 | A | B | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4609 | |
| CLK4 | CLK | CMGC | 6fyv | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10511 | |
| CDK2 | CDK | CMGC | 2vto | A | A | n-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamide | Human | 4421 | |
| CDK2 | CDK | CMGC | 1ke7 | A | | 3-{[(2,2-dioxido-1,3-dihydro-2-benzothien-5-yl)amino]methylene}-5-(1,3-oxazol-5-yl)-1,3-dihydro-2h-indol-2-one | Human | 4295 | |
| CDK2 | CDK | CMGC | 3bhv | C | B | 9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-ol | Human | 4529 | |
| CDK2 | CDK | CMGC | 1h24 | C | | - | Human | 4296 | |
| CDK2 | CDK | CMGC | 3bht | C | A | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4151 | |
| CDK2 | CDK | CMGC | 4ek6 | A | A | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamide | Human | 4359 | |
| CDK2 | CDK | CMGC | 4fkw | A | B | 2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylate | Human | 4277 | |
| CDK2 | CDK | CMGC | 3tiy | A | B | 2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-one | Human | 4488 | |
| CDK2 | CDK | CMGC | 1ol2 | A | | - | Human | 4305 | |
| CDK2 | CDK | CMGC | 6q4h | A | A | 2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acid | Human | 11194 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | A | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12120 | |
| CDK2 | CDK | CMGC | 2cci | C | | adenosine-5'-triphosphate | Human | 4532 | |
| CLK1 | CLK | CMGC | 6r6x | A | | 5-(1-methylindol-3-yl)pyrimidin-4-amine | Human | 12231 | |
| CDK2 | CDK | CMGC | 1fin | C | | adenosine-5'-triphosphate | Human | 4479 | |
| CDK2 | CDK | CMGC | 2r3o | A | C | (5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanol | Human | 4229 | |
| DYRK1A | DYRK | CMGC | 6s11 | A | A | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11361 | |
| DYRK1A | DYRK | CMGC | 6eip | A | | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | 10555 | |
| DYRK1A | DYRK | CMGC | 6eiq | D | | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | 10541 | |
| DYRK1A | DYRK | CMGC | 7ajm | A | A | ~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamide | Human | 13590 | |
| DYRK1A | DYRK | CMGC | 6uwy | A | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11989 | |
| DYRK1A | DYRK | CMGC | 7aj5 | A | B | 4-(1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13591 | |
| DYRK1A | DYRK | CMGC | 6eip | D | | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | 10531 | |
| DYRK1A | DYRK | CMGC | 6t6a | D | A | - | Human | 11862 | |
| DYRK1A | DYRK | CMGC | 7a4o | A | | phosphoaminophosphonic acid-adenylate ester | Human | 13744 | |
| DYRK1A | DYRK | CMGC | 2vx3 | D | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3786 | |
| DYRK1A | DYRK | CMGC | 6uwy | C | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11984 | |
| DYRK1A | DYRK | CMGC | 6a1g | A | | 5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amine | Human | 10530 | |
| DYRK1A | DYRK | CMGC | 6eir | D | | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10549 | |
| DYRK1A | DYRK | CMGC | 7a5d | A | B | 4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13745 | |
| DYRK1A | DYRK | CMGC | 4yu2 | C | B | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3775 | |
| MAPK9 (JNK2) | MAPK | CMGC | 3e7o | A | | n-{3-[5-(1h-1,2,4-triazol-3-yl)-1h-indazol-3-yl]phenyl}furan-2-carboxamide | Human | 1238 | |
| CLK1 | CLK | CMGC | 6r8j | A | B | 4-(1-methylindol-3-yl)pyrimidin-2-amine | Human | 12631 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6te2 | A | B | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12446 | |
| DYRK1A | DYRK | CMGC | 5a4t | C | | n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide | Human | 6734 | |
| DYRK1A | DYRK | CMGC | 7ajm | A | B | ~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamide | Human | 13598 | |
| DYRK1A | DYRK | CMGC | 6eip | B | | 4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamide | Human | 10517 | |
| DYRK1A | DYRK | CMGC | 6s1b | A | A | ~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11359 | |
| DYRK1A | DYRK | CMGC | 7aj8 | A | B | 4-(1-benzofuran-5-yl)pyridin-2-amine | Human | 13603 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7x4u | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14661 | |
| DYRK1A | DYRK | CMGC | 6uwy | C | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11985 | |
| DYRK1A | DYRK | CMGC | 5aik | B | | 4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine | Human | 3759 | |
| DYRK1A | DYRK | CMGC | 5a4l | C | A | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6721 | |
| DYRK1A | DYRK | CMGC | 6eis | B | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10556 | |
| DYRK1A | DYRK | CMGC | 4nct | D | | pkc412 | Human | 3751 | |
| CDK5 | CDK | CMGC | 7vds | A | B | 5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrile | Human | 14147 | |
| DYRK1A | DYRK | CMGC | 5a4q | D | | n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6737 | |
| DYRK1A | DYRK | CMGC | 4yu2 | A | B | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3765 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7cml | A | B | - | Human | 12705 | |
| CDK9 | CDK | CMGC | 4imy | A | A | adenosine monophosphate | Human | 2238 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7x4u | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14660 | |
| CDK9 | CDK | CMGC | 8k5r | A | | (1s,3s)-n3-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamine | Human | 15081 | |
| CDK5 | CDK | CMGC | 1ung | B | | 6-phenyl[5h]pyrrolo[2,3-b]pyrazine | Human | 2789 | |
| DYRK2 | DYRK | CMGC | 8hlt | A | | (6-{[(4p)-4-(1,3-benzothiazol-5-yl)-5-fluoropyrimidin-2-yl]amino}pyridin-3-yl)(piperazin-1-yl)methanone | Human | 15091 | |
| DYRK1A | DYRK | CMGC | 7ajs | A | B | 4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamine | Human | 13607 | |
| CLK1 | CLK | CMGC | 6ytg | A | B | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12424 | |
| DYRK1A | DYRK | CMGC | 5a4e | A | B | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6740 | |
| DYRK1A | DYRK | CMGC | 4ylj | C | B | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3748 | |
| DYRK1A | DYRK | CMGC | 5a4e | C | A | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6725 | |
| DYRK1A | DYRK | CMGC | 6s1i | A | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11370 | |
| DYRK1A | DYRK | CMGC | 5a4e | A | A | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6741 | |
| DYRK1A | DYRK | CMGC | 6s1i | A | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11376 | |
| CDK9 | CDK | CMGC | 4ogr | E | | adenosine | Human | 2235 | |
| DYRK1A | DYRK | CMGC | 3anq | C | | (1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one | Human | 3791 | |
| DYRK1A | DYRK | CMGC | 4mq2 | C | B | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3780 | |
| DYRK1A | DYRK | CMGC | 7fhs | A | A | (5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | 14160 | |
| DYRK1A | DYRK | CMGC | 6s11 | A | B | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11364 | |
| DYRK1A | DYRK | CMGC | 6qu2 | A | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12085 | |
| DYRK1A | DYRK | CMGC | 4aze | A | | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3761 | |
| DYRK1A | DYRK | CMGC | 6s1b | A | B | ~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11377 | |
| DYRK1A | DYRK | CMGC | 4yll | A | C | 10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3731 | |
| DYRK1A | DYRK | CMGC | 6eiq | C | | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | 10524 | |
| DYRK1A | DYRK | CMGC | 5a4t | D | | n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide | Human | 6712 | |
| DYRK1A | DYRK | CMGC | 7a53 | A | A | (3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-one | Human | 13755 | |
| DYRK1A | DYRK | CMGC | 4yu2 | D | B | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3733 | |
| DYRK1A | DYRK | CMGC | 4mq1 | C | A | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3781 | |
| DYRK1A | DYRK | CMGC | 6s1i | B | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11371 | |
| DYRK1A | DYRK | CMGC | 6ej4 | C | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10519 | |
| DYRK1A | DYRK | CMGC | 2wo6 | B | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3749 | |
| DYRK1A | DYRK | CMGC | 7a5b | A | | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 13756 | |
| DYRK1A | DYRK | CMGC | 5a54 | C | | n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide | Human | 6720 | |
| DYRK1A | DYRK | CMGC | 6yf8 | A | | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | 13462 | |
| GSK3B | GSK | CMGC | 6tcu | A | A | 5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamide | Human | 12780 | |
| CDK2 | CDK | CMGC | 1gij | A | | 1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-(5-pyrrolidin-2-yl-1h-pyrazol-3-yl)-urea | Human | 4542 | |
| CDK2 | CDK | CMGC | 4eoo | C | B | adenosine-5'-triphosphate | Human | 4139 | |
| CDK2 | CDK | CMGC | 2r3k | A | C | 3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amine | Human | 4022 | |
| CDK2 | CDK | CMGC | 4eor | C | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4487 | |
| CDK2 | CDK | CMGC | 2vtq | A | | {[(2,6-difluorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamide | Human | 3891 | |
| CDK2 | CDK | CMGC | 9ess | A | A | (4-bromo-2-methoxyphenyl)methanol | Human | 15908 | |
| CDK2 | CDK | CMGC | 4eon | A | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 3902 | |
| CDK2 | CDK | CMGC | 3s00 | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanone | Human | 4208 | |
| CDK2 | CDK | CMGC | 3dog | A | A | (2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol | Human | 4541 | |
| CDK2 | CDK | CMGC | 4fkq | A | A | 4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamide | Human | 3972 | |
| CDK2 | CDK | CMGC | 9esj | A | C | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid | Human | 15909 | |
| CDK2 | CDK | CMGC | 1dm2 | A | B | 4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-one | Human | 4024 | |
| CDK2 | CDK | CMGC | 2r3p | A | B | 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amine | Human | 4392 | |
| CDK2 | CDK | CMGC | 2i40 | A | A | 5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamide | Human | 4363 | |
| CDK13 (CHED) | CDK | CMGC | 5efq | C | | adenosine-5'-diphosphate | Human | 6324 | |
| DYRK1A | DYRK | CMGC | 7a51 | A | | 4-azanyl-6-bromanyl-7-methyl-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13753 | |
| DYRK1A | DYRK | CMGC | 6eiv | C | | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10542 | |
| DYRK1A | DYRK | CMGC | 3anq | A | | (1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one | Human | 3767 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7opm | A | A | 1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]urea | Human | 14084 | |
| DYRK1A | DYRK | CMGC | 5a4e | B | B | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6726 | |
| DYRK1A | DYRK | CMGC | 2vx3 | B | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3766 | |
| DYRK1A | DYRK | CMGC | 4ylj | B | A | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3753 | |
| DYRK1A | DYRK | CMGC | 7aja | A | A | 1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazine | Human | 13610 | |
| DYRK1A | DYRK | CMGC | 4ylk | A | A | 10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3789 | |
| DYRK1A | DYRK | CMGC | 4ylj | D | B | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3793 | |
| DYRK1A | DYRK | CMGC | 6s14 | A | A | ~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11418 | |
| CDK2 | CDK | CMGC | 3eoc | C | | 5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine | Human | 3969 | |
| CDK2 | CDK | CMGC | 9ess | A | B | (4-bromo-2-methoxyphenyl)methanol | Human | 15911 | |
| CDK2 | CDK | CMGC | 5d1j | A | | n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamide | Human | 4058 | |
| CDK2 | CDK | CMGC | 6q4e | A | C | 6-iodanyl-7~{h}-purin-2-amine | Human | 11219 | |
| CDK2 | CDK | CMGC | 3qtw | A | A | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4397 | |
| CDK2 | CDK | CMGC | 2w05 | A | A | n-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamide | Human | 4547 | |
| CDK2 | CDK | CMGC | 5oo3 | A | B | 1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-one | Human | 10568 | |
| CDK2 | CDK | CMGC | 3f5x | C | | 4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}aniline | Human | 3894 | |
| CDK2 | CDK | CMGC | 3ti1 | A | B | n-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamide | Human | 4213 | |
| CDK2 | CDK | CMGC | 6q49 | A | B | - | Human | 11220 | |
| DYRK1A | DYRK | CMGC | 4yu2 | B | B | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3738 | |
| DYRK1A | DYRK | CMGC | 6eis | D | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10547 | |
| DYRK1A | DYRK | CMGC | 6ln1 | A | | 1,3,5,8-tetrakis(oxidanyl)xanthen-9-one | Human | 13935 | |
| DYRK1A | DYRK | CMGC | 6t6a | B | A | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11860 | |
| DYRK1A | DYRK | CMGC | 6qu2 | D | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12089 | |
| DYRK1A | DYRK | CMGC | 5a54 | B | | n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide | Human | 6716 | |
| DYRK1A | DYRK | CMGC | 2wo6 | B | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3739 | |
| DYRK1A | DYRK | CMGC | 7fht | A | B | (5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | 14162 | |
| DYRK1A | DYRK | CMGC | 7ajw | A | B | 4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13611 | |
| DYRK1A | DYRK | CMGC | 7ajw | A | A | 4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13612 | |
| DYRK1A | DYRK | CMGC | 6eij | D | | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | 10559 | |
| DYRK1A | DYRK | CMGC | 7a5n | A | | 5-(2-azanylpyridin-4-yl)-~{n}-[[2,6-bis(fluoranyl)phenyl]methyl]-2-methyl-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amine | Human | 13757 | |
| DYRK1A | DYRK | CMGC | 6qu2 | B | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12086 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fko | A | | 3-(2-chlorophenyl)-6-(2-fluorophenoxy)-2h-indazole | Human | 5075 | |
| GSK3B | GSK | CMGC | 1j1c | B | | adenosine-5'-diphosphate | Human | 677 | |
| CDK2 | CDK | CMGC | 2bkz | A | | 1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 3942 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | C | | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | 12794 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hme | A | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11275 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 2pvr | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5505 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oqu | B | B | adenosine-5'-diphosphate | Human | 9678 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h36 | A | A | - | Human | 3459 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4kke | A | | adenosine monophosphate | Human | 3448 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | D | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10496 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | B | A | phosphomethylphosphonic acid adenylate ester | Human | 10504 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3cgf | A | | n-cyclohexyl-4-imidazo[1,2-a]pyridin-3-yl-n-methylpyrimidin-2-amine | Human | 6770 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4y5h | A | | 1-(trans-4-{[7-oxo-8-(propan-2-yl)-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}cyclohexyl)-3-propan-2-ylurea | Human | 3431 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4whz | A | A | 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamide | Human | 3429 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8vo4 | A | | (4p)-4-{6-[(azetidin-1-yl)methyl]-5-(2-chloro-6-fluoroanilino)-1h-indazol-1-yl}-n-methylthiophene-2-carboxamide | Human | 15637 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4w4w | A | | n-(2-methylpyridin-4-yl)-3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}benzamide | Human | 3418 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6r | A | B | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3436 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2exc | X | | n-{2'-[(4-fluorophenyl)amino]-4,4'-bipyridin-2-yl}-4-methoxycyclohexanecarboxamide | Human | 3478 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8vnx | A | A | (4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamide | Human | 15638 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3rtp | A | | n-[4-cyano-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamide | Human | 3467 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2waj | A | A | 1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinoline | Human | 3472 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4w4v | A | | 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamide | Human | 3437 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3ttj | A | A | 9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamine | Human | 3458 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6r | B | B | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3417 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4x21 | B | | n-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamide | Human | 6239 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8wgf | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15046 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4z9l | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 3438 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | B | B | phosphomethylphosphonic acid adenylate ester | Human | 10499 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2p33 | A | | 4-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-n-ethylpiperidine-1-carboxamide | Human | 3455 | |
| HIPK3 | DYRK | CMGC | 7o7i | A | | - | Human | 13996 | |
| CDK2 | CDK | CMGC | 4acm | A | A | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 4247 | |
| CDK2 | CDK | CMGC | 3wbl | A | | n~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamine | Human | 3895 | |
| CDK2 | CDK | CMGC | 3rm7 | A | B | 2-[(4-hydroxybenzyl)amino]-5-nitrobenzamide | Human | 4499 | |
| CDK2 | CDK | CMGC | 4cfx | C | C | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4442 | |
| CDK2 | CDK | CMGC | 3pxr | A | B | - | Human | 4173 | |
| CDK2 | CDK | CMGC | 2r3h | A | A | 3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amine | Human | 4152 | |
| CDK2 | CDK | CMGC | 6q4e | A | A | 6-iodanyl-7~{h}-purin-2-amine | Human | 11199 | |
| CDK2 | CDK | CMGC | 2r3j | A | B | 3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4544 | |
| CDK2 | CDK | CMGC | 3s1h | A | B | 4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4226 | |
| CDK2 | CDK | CMGC | 5if1 | A | A | - | Human | 6568 | |
| CDK2 | CDK | CMGC | 2iw9 | C | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 3858 | |
| CDK2 | CDK | CMGC | 5lmk | C | B | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | 7397 | |
| CDK2 | CDK | CMGC | 4cfw | C | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4549 | |
| CDK2 | CDK | CMGC | 8cur | A | B | 6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | 14692 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ksk | A | | 4-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13386 | |
| MAPK10 (JNK3) | MAPK | CMGC | 1pmv | A | | 2,6-dihydroanthra/1,9-cd/pyrazol-6-one | Human | 3434 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | C | C | - | Human | 3446 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | A | B | - | Human | 3454 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8bzp | A | B | 2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamide | Human | 14858 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3tti | A | | trans-4-({9-[(3s)-tetrahydrofuran-3-yl]-8-[(2,4,6-trifluorophenyl)amino]-9h-purin-2-yl}amino)cyclohexanol | Human | 3456 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4whz | A | B | 3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamide | Human | 3422 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | B | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10506 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3g9l | X | | (3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-[(e)-2-phenylethenyl]-1h-indole-2,3-dione 3-oxime | Human | 3435 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8vnx | A | B | (4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamide | Human | 15639 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h39 | A | B | - | Human | 3462 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6s | A | B | 3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3449 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fi2 | A | B | 3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | 3452 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | D | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10497 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2zdu | A | | 4-[(4-{[6-bromo-3-(methoxycarbonyl)-1-oxo-4-phenylisoquinolin-2(1h)-yl]methyl}phenyl)amino]-4-oxobutanoic acid | Human | 3479 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | A | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10503 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2zdt | A | B | 4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acid | Human | 3424 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7orf | A | B | n-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamide | Human | 13814 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4u79 | A | | n-{4-[(3-{2-[(trans-4-aminocyclohexyl)amino]pyrimidin-4-yl}pyridin-2-yl)oxy]naphthalen-1-yl}benzenesulfonamide | Human | 3466 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6s | B | B | 3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3425 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3kvx | A | A | n-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)aniline | Human | 3433 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8enj | A | | n-[3-({(4p)-4-[(3m)-1-tert-butyl-3-(3-hydroxyphenyl)-1h-pyrazol-4-yl]pyridin-2-yl}amino)propyl]-4-hydroxybenzene-1-sulfonamide | Human | 14884 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2zdt | A | A | 4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acid | Human | 3421 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | C | B | - | Human | 3465 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8bzp | A | A | 2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamide | Human | 14859 | |
| DYRK1A | DYRK | CMGC | 6yf8 | B | | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | 13461 | |
| SRPK1 | SRPK | CMGC | 6fad | D | | - | Human | 11637 | |
| SRPK1 | SRPK | CMGC | 7zks | A | B | n-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamide | Human | 14618 | |
| SRPK1 | SRPK | CMGC | 7pqs | A | B | ~{n}-[3-[[[2-(6-chloranyl-7-fluoranyl-1~{h}-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-~{n}-methyl-methanesulfonamide | Human | 14015 | |
| SRPK1 | SRPK | CMGC | 6fad | A | | - | Human | 11638 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7yl1 | A | | 7-hexyl-3-methyl-8-sulfanylidene-9h-purine-2,6-dione | Human | 14845 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6r | A | A | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3441 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8wgf | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15047 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2o0u | A | | n-{3-cyano-6-[3-(1-piperidinyl)propanoyl]-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-yl}1-naphthalenecarboxamide | Human | 3415 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fi3 | A | A | 3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | 3442 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fi3 | A | B | 3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | 3445 | |
| SRPK1 | SRPK | CMGC | 7pqs | A | A | ~{n}-[3-[[[2-(6-chloranyl-7-fluoranyl-1~{h}-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-~{n}-methyl-methanesulfonamide | Human | 14014 | |
| SRPK1 | SRPK | CMGC | 5xv7 | A | | 9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrile | Human | 9727 | |
| CDK9 | CDK | CMGC | 4imy | C | A | adenosine monophosphate | Human | 2237 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g97 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-one | Human | 9960 | |
| CDK2 | CDK | CMGC | 2cch | A | B | adenosine-5'-triphosphate | Human | 4553 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4q | A | B | 2-methoxyimino-5-(quinolin-6-ylmethyl)-1,3-thiazol-4-one | Human | 14239 | |
| CDK2 | CDK | CMGC | 8oy2 | A | | (1s,2s,11as)-1-methoxy-1,4,7,10-tetramethyl-2,9-bis(oxidanyl)-2,11a-dihydrobenzo[b][1,4]benzodioxepine-3,6-dione | Human | 15078 | |
| CDK13 (CHED) | CDK | CMGC | 5efq | A | | adenosine-5'-diphosphate | Human | 6323 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4b99 | A | | 11-cyclopentyl-2-[[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl-phenyl]amino]-5-methyl-pyrimido[4,5-b][1,4]benzodiazepin-6-one | Human | 388 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8x5m | A | B | 3-[4-(dimethylamino)butanoylamino]-~{n}-[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide | Human | 15100 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv3 | A | A | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 2617 | |
| CDK7 | CDK | CMGC | 1ua2 | D | | adenosine-5'-triphosphate | Human | 543 | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | A | - | Human | 5163 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | B | - | Human | 5222 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qdz | A | B | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | 11958 | |
| HIPK2 | DYRK | CMGC | 7ncf | A | | 3-(4-tert-butylphenyl)-5-(1h-pyrazol-4-yl)furo[3,2-b]pyridine | Human | 13393 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5yf9 | X | B | nicotinic acid | Human | 11414 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | B | 2-amino-phenylamino-dibenzosuberone | Human | 5089 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ewq | A | A | 3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazine | Human | 5200 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | B | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5013 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | B | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 4983 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp2 | A | B | 1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-one | Human | 5031 | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | A | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | 5081 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | B | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | 5214 | |
| MAPK14 (p38a) | MAPK | CMGC | 5omh | A | | 1-(3-chlorophenyl)-3-methyl-4~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | 11251 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ehv | A | A | - | Human | 4997 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mw1 | A | | 8-(2,6-dichlorophenyl)-4-(2,4-difluorophenyl)-2-piperidin-4-yl-1,7-naphthyridine 7-oxide | Human | 5072 | |
| MAPK14 (p38a) | MAPK | CMGC | 1zzl | A | | 6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-3-isopropyl[1,2,4]triazolo[4,3-a]pyridine | Human | 5249 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gfe | A | | n-cyclopropyl-3-{[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-4-yl]amino}-4-methylbenzamide | Human | 4991 | |
| MAPK14 (p38a) | MAPK | CMGC | 1bmk | A | | 4-(fluorophenyl)-1-cyclopropylmethyl-5-(2-amino-4-pyrimidinyl)imidazole | Human | 5235 | |
| MAPK1 (Erk2) | MAPK | CMGC | 1tvo | A | | 5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amine | Human | 2581 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fly | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-[(1-methylethyl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5113 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | B | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | 5120 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfe | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-4-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | 5173 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qdz | A | A | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | 11956 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh8 | A | A | [3-(benzyloxy)phenyl]methanol | Human | 4978 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 8 | - | Human | 5078 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfa | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 5018 | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | B | | - | Human | 5007 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | B | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | 5132 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh1 | A | | - | Human | 5003 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | B | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | 5246 | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyy | A | | 3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-4h-1,2,4-triazol-3-yl)phenol | Human | 9513 | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | A | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | 5247 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nww | A | | 1-[2-(2-{[2-(dimethylamino)ethyl]amino}-6-{2-[(1-methylethyl)amino]-1,3-thiazol-5-yl}pyrimidin-4-yl)benzyl]-3-ethylurea | Human | 5068 | |
| MAPK14 (p38a) | MAPK | CMGC | 5wjj | A | B | n-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamide | Human | 9516 | |
| MAPK14 (p38a) | MAPK | CMGC | 2okr | A | | - | Human | 5136 | |
| MAPK14 (p38a) | MAPK | CMGC | 3kf7 | A | | 3-{6-[2-(2,4-difluorophenyl)ethyl][1,2,4]triazolo[4,3-a]pyridin-3-yl}-4-methylbenzamide | Human | 5201 | |
| MAPK14 (p38a) | MAPK | CMGC | 3huc | A | B | n-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamide | Human | 5111 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gc7 | A | B | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 5256 | |
| MAPK14 (p38a) | MAPK | CMGC | 6zwp | A | B | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 12698 | |
| MAPK14 (p38a) | MAPK | CMGC | 1oz1 | A | A | 3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-ol | Human | 5230 | |
| MAPK14 (p38a) | MAPK | CMGC | 2baq | A | | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | 5184 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | B | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | 5155 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mgy | A | | - | Human | 5171 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | 4998 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | B | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | 5046 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 4977 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv3 | A | A | 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5012 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | A | | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 4993 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | A | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5237 | |
| MAPK14 (p38a) | MAPK | CMGC | 6zqs | A | | 2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-one | Human | 12986 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmm | A | | 6-(2,4-difluorophenoxy)-n-[(1r)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 5186 | |
| CDK2 | CDK | CMGC | 3qwk | A | B | 4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamide | Human | 4155 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | B | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12121 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | D | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5144 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfk | A | A | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | Human | 11617 | |
| MAPK14 (p38a) | MAPK | CMGC | 3odz | X | | - | Human | 5069 | |
| MAPK14 (p38a) | MAPK | CMGC | 4fa2 | A | A | trans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanol | Human | 5150 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fc1 | X | | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 5110 | |
| MAPK14 (p38a) | MAPK | CMGC | 3e92 | A | | n-cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamide | Human | 5149 | |
| MAPK14 (p38a) | MAPK | CMGC | 8yd9 | A | B | - | Human | 15696 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv4 | B | | 1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5064 | |
| MAPK14 (p38a) | MAPK | CMGC | 9r27 | A | | 4-[4-[[4-chloranyl-3-(trifluoromethyl)phenyl]carbamoylamino]-3-fluoranyl-phenoxy]-~{n}-methyl-pyridine-2-carboxamide | Human | 15697 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbn | A | | n-(3-tert-butyl-1h-pyrazol-5-yl)-n'-{4-chloro-3-[(pyridin-3-yloxy)methyl]phenyl}urea | Human | 5257 | |
| MAPK14 (p38a) | MAPK | CMGC | 3roc | A | | 3-{5-chloro-4-[(2,4-difluorobenzyl)oxy]-6-oxopyrimidin-1(6h)-yl}-n-(2-hydroxyethyl)-4-methylbenzamide | Human | 5011 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcp | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5194 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv6 | A | | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(2-morpholin-4-ylethoxy)phenyl]urea | Human | 5101 | |
| MAPK14 (p38a) | MAPK | CMGC | 2yiw | A | | 1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | 4988 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6c | A | | - | Human | 5015 | |
| MAPK14 (p38a) | MAPK | CMGC | 1di9 | A | | 4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazoline | Human | 5251 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcq | A | B | 1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5053 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 5 | - | Human | 5107 | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8x | A | | n,4-dimethyl-3-[(1-phenyl-1h-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamide | Human | 5041 | |
| MAPK14 (p38a) | MAPK | CMGC | 8a8m | A | | phosphomethylphosphonic acid adenosyl ester | Human | 14289 | |
| MAPK14 (p38a) | MAPK | CMGC | 5etc | A | | - | Human | 6361 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wfc | A | | - | Human | 4989 | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | B | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | 5004 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | B | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5175 | |
| DYRK1A | DYRK | CMGC | 8c3g | A | A | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 15155 | |
| DYRK1A | DYRK | CMGC | 8c3r | A | A | gossypin | Human | 15156 | |
| DYRK1A | DYRK | CMGC | 8c3r | A | B | gossypin | Human | 15157 | |
| DYRK1A | DYRK | CMGC | 8c3g | A | B | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 15153 | |
| DYRK1A | DYRK | CMGC | 8c3q | A | B | rutin | Human | 15154 | |
| MAPK14 (p38a) | MAPK | CMGC | 1yqj | A | | 6((s)-3-benzylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyrazine | Human | 5152 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj5 | A | | pexmetinib | Human | 15698 | |
| MAPK14 (p38a) | MAPK | CMGC | 5o8u | A | | - | Human | 8381 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e8a | A | | - | Human | 4979 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpa | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5026 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | H | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12487 | |
| MAPK14 (p38a) | MAPK | CMGC | 2npq | A | | - | Human | 5205 | |
| CLK3 | CLK | CMGC | 6khf | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11650 | |
| DYRK1A | DYRK | CMGC | 8c3q | A | A | rutin | Human | 15158 | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyx | A | B | n-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amine | Human | 9517 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | A | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5032 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hvc | A | | 4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridine | Human | 5054 | |
| MAPK14 (p38a) | MAPK | CMGC | 4a9y | A | | n-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamide | Human | 5073 | |
| MAPK14 (p38a) | MAPK | CMGC | 4r3c | A | B | 6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine | Human | 5036 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbw | A | | 3-(1-naphthylmethoxy)pyridin-2-amine | Human | 5179 | |
| CDK6 | CDK | CMGC | 8i0m | A | | 2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamide | Human | 15164 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh7 | A | A | (3-phenoxyphenyl)methanol | Human | 5208 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ody | X | | - | Human | 5233 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbo | A | | 2-chlorophenol | Human | 5039 | |
| DYRK1B | DYRK | CMGC | 8c2z | A | A | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 15180 | |
| DYRK1B | DYRK | CMGC | 8c2z | A | B | n-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amine | Human | 15181 | |
| MAPK14 (p38a) | MAPK | CMGC | 8yd9 | A | A | - | Human | 15699 | |
| MAPK14 (p38a) | MAPK | CMGC | 3d83 | A | | n-{4'-[(cyclopropylmethyl)carbamoyl]-6-methylbiphenyl-3-yl}-2-morpholin-4-ylpyridine-4-carboxamide | Human | 5028 | |
| MAPK14 (p38a) | MAPK | CMGC | 6anl | A | A | tak-715 | Human | 9515 | |
| DYRK3 | DYRK | CMGC | 5y86 | A | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 9876 | |
| CLK1 | CLK | CMGC | 6g33 | B | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9821 | |
| CLK1 | CLK | CMGC | 6zln | A | B | 4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 12710 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | A | | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5060 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 3 | - | Human | 5040 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5a | X | A | - | Human | 5189 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw5 | A | | n-[2-(3-{[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl}-1h-indol-1-yl)ethyl]-3-(trifluoromethyl)benzamide | Human | 5076 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | C | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5142 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fsk | A | | 3-(2-chlorophenyl)-7-[(trans-4-hydroxycyclohexyl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 5008 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | C | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | 5199 | |
| MAPK14 (p38a) | MAPK | CMGC | 6zwp | A | A | 5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 12699 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lhj | A | | n-cyclopropyl-3-[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamide | Human | 5234 | |
| CLK1 | CLK | CMGC | 6i5k | A | B | 5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridine | Human | 10836 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kip | B | | 2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamide | Human | 5180 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fl4 | A | | 6-(2,4-difluorophenoxy)-3-(2-methylphenyl)-1h-pyrazolo[3,4-d]pyrimidine | Human | 5151 | |
| MAPK14 (p38a) | MAPK | CMGC | 3s4q | A | | 3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-n-cyclopropyl-4-methylbenzamide | Human | 5133 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | B | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | 5034 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfc | A | | (4-{5-[({4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}carbamoyl)amino]-3-tert-butyl-1h-pyrazol-1-yl}phenyl)acetic acid | Human | 5160 | |
| CLK1 | CLK | CMGC | 6i5i | A | B | 5-(1-methylpyrazol-4-yl)-3-[1-(phenylmethyl)pyrazol-4-yl]furo[3,2-b]pyridine | Human | 10840 | |
| CLK1 | CLK | CMGC | 6khd | C | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11643 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | A | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | 5038 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9y | A | B | n,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5017 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ocg | A | | 5-amino-n-[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]-1-phenyl-1h-pyrazole-4-carboxamide | Human | 4984 | |
| MAPK14 (p38a) | MAPK | CMGC | 2bal | A | | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl][3-(piperidin-4-yloxy)phenyl]methanone | Human | 5260 | |
| MAPK14 (p38a) | MAPK | CMGC | 5eta | B | | - | Human | 7137 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fst | X | B | - | Human | 5195 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv3 | A | B | 1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5232 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa0 | A | A | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamide | Human | 5213 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fln | C | | 6-(2,4-difluorophenoxy)-8-methyl-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5090 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | B | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5137 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gi3 | A | | n-{5-tert-butyl-2-methoxy-3-[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]naphthalen-1-yl}carbamoyl)amino]phenyl}methanesulfonamide | Human | 5226 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfi | A | B | ~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamide | Human | 11619 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | F | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12489 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp2 | A | A | 1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-one | Human | 5217 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mtx | A | A | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamide | Human | 8382 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnx | A | | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | 5002 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | B | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5188 | |
| MAPK14 (p38a) | MAPK | CMGC | 4l8m | A | A | n-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamide | Human | 5005 | |
| MAPK14 (p38a) | MAPK | CMGC | 2bak | A | | n-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamide | Human | 5114 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fsm | X | | - | Human | 5044 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj2 | A | A | - | Human | 15700 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | A | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | 5216 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5263 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ouk | A | | 4-[5-[2-(1-phenyl-ethylamino)-pyrimidin-4-yl]-1-methyl-4-(3-trifluoromethylphenyl)-1h-imidazol-2-yl]-piperidine | Human | 5146 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hl7 | A | | 2-{4-[5-(4-chlorophenyl)-4-pyrimidin-4-yl-1h-pyrazol-3-yl]piperidin-1-yl}-2-oxoethanol | Human | 5236 | |
| MAPK14 (p38a) | MAPK | CMGC | 6ohd | A | B | 3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamide | Human | 11819 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kip | A | | 2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamide | Human | 5159 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | C | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5182 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 9 | - | Human | 5127 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hll | A | A | 3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamide | Human | 5115 | |
| MAPK14 (p38a) | MAPK | CMGC | 4l8m | A | B | n-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamide | Human | 4992 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fml | A | | 6-(2,4-difluorophenoxy)-n-[(1s)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 5010 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmj | A | | 4-(5-methyl-3-phenylisoxazol-4-yl)pyrimidin-2-amine | Human | 5129 | |
| MAPK14 (p38a) | MAPK | CMGC | 6m9l | A | | 3-benzyl-6-[(2,4-difluorophenyl)amino]-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-one | Human | 11255 | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | B | - | Human | 5030 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmn | A | B | 6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amine | Human | 4995 | |
| CDK4 | CDK | CMGC | 3g33 | A | | - | Human | 3387 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hp5 | A | | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 5158 | |
| MAPK14 (p38a) | MAPK | CMGC | 3heg | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5218 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj4 | A | C | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 15706 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kin | B | | 5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamide | Human | 5131 | |
| MAPK14 (p38a) | MAPK | CMGC | 1kv2 | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 5255 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmh | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5024 | |
| MAPK14 (p38a) | MAPK | CMGC | 3flw | A | | 6-(2,4-difluorophenoxy)-2-{[3-hydroxy-1-(2-hydroxyethyl)propyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5153 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | D | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5016 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ehv | A | B | - | Human | 4981 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh0 | A | | - | Human | 5124 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hec | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 5035 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa1 | A | A | pyridin-2-amine | Human | 11352 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nho | A | | (6~{s})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7993 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4h3p | D | | phosphoaminophosphonic acid-adenylate ester | Human | 2575 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvd | A | A | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-one | Human | 6030 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4i | A | | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7400 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mod | A | A | - | Human | 7678 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr3 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13922 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqw | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13927 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqq | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamide | Human | 13928 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr8 | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamide | Human | 13929 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7w5o | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 14110 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7auv | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13930 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr9 | A | B | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamide | Human | 13931 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp7 | B | | 2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6093 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9a | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-one | Human | 11412 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | A | C | benzoic acid | Human | 11277 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otp | B | A | - | Human | 10602 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | E | B | phosphoaminophosphonic acid-adenylate ester | Human | 2591 | |
| CDK6 | CDK | CMGC | 2f2c | B | | (2s)-2-({6-[(3-amino-5-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-ol | Human | 2795 | |
| CDK6 | CDK | CMGC | 4aua | A | | 1h-benzimidazol-2-yl(1h-pyrrol-2-yl)methanone | Human | 2801 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oue | B | A | (3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-imidazol-4-yl)ethyl]azanium | Human | 9635 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehu | B | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamine | Human | 9630 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oty | A | A | trifluoroacetic acid | Human | 9692 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ouu | B | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 9657 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3qa0 | B | B | - | Human | 5528 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7auv | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13925 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3h30 | B | B | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 5480 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8i | B | B | - | Human | 13262 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ctp | A | A | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7304 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hot | A | A | (2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enal | Human | 11667 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md8 | E | | - | Human | 5439 | |
| CLK1 | CLK | CMGC | 7o9y | A | | 4-(1~{h}-indol-3-yl)pyrimidin-2-amine | Human | 14208 | |
| DYRK1A | DYRK | CMGC | 7fhs | A | B | (5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | 14159 | |
| DYRK1A | DYRK | CMGC | 6qu2 | C | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12090 | |
| DYRK1A | DYRK | CMGC | 4aze | B | | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3768 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fi2 | A | A | 3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamide | Human | 3463 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | A | C | - | Human | 3453 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fv8 | A | A | 5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamide | Human | 3468 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | C | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10507 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tll | A | A | 4,5,6,7-tetrabromobenzotriazole | Human | 13093 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otp | A | A | 2-[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 10588 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5clp | A | A | 2-(3,4-dichlorophenyl)ethanamine | Human | 6922 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3kvx | A | B | n-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)aniline | Human | 3430 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3pze | A | | 3-(carbamoylamino)-5-phenylthiophene-2-carboxamide | Human | 4642 | |
| GSK3B | GSK | CMGC | 6hk3 | B | B | 3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11424 | |
| GSK3B | GSK | CMGC | 3f7z | A | A | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 743 | |
| GSK3B | GSK | CMGC | 9hm1 | A | | n-(4-{5-[(2-aminoethyl)sulfamoyl]thiophen-2-yl}pyridin-2-yl)cyclopropanecarboxamide | Human | 15792 | |
| GSK3B | GSK | CMGC | 6hk4 | B | A | 3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamide | Human | 11430 | |
| GSK3B | GSK | CMGC | 1q3d | A | | staurosporine | Human | 705 | |
| GSK3B | GSK | CMGC | 3zrm | B | A | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 753 | |
| CDK2 | CDK | CMGC | 6yl6 | A | B | - | Human | 12495 | |
| CDK2 | CDK | CMGC | 1pxm | A | B | - | Human | 3936 | |
| CDK2 | CDK | CMGC | 8cur | A | A | 6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | 14693 | |
| CDK2 | CDK | CMGC | 4cfm | C | A | 6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amine | Human | 4260 | |
| CDK2 | CDK | CMGC | 4d1x | A | | (4s)-2-(6-hydroxy-1,3-benzothiazol-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acid | Human | 4344 | |
| CDK2 | CDK | CMGC | 8ru8 | A | B | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 15328 | |
| CDK2 | CDK | CMGC | 4bck | A | C | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4433 | |
| CDK2 | CDK | CMGC | 4cfx | A | C | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 3963 | |
| CDK2 | CDK | CMGC | 1oiy | A | B | 4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamide | Human | 3945 | |
| CDK2 | CDK | CMGC | 4cfw | A | C | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4141 | |
| CDK2 | CDK | CMGC | 2vth | A | | 5-hydroxynaphthalene-1-sulfonamide | Human | 4274 | |
| CDK2 | CDK | CMGC | 2x1n | A | A | 2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amine | Human | 4579 | |
| CDK2 | CDK | CMGC | 4bck | A | A | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4095 | |
| CDK2 | CDK | CMGC | 1hcl | A | B | - | Human | 4540 | |
| CDK2 | CDK | CMGC | 4bcn | A | A | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4084 | |
| CDK2 | CDK | CMGC | 3r9n | A | B | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanone | Human | 3867 | |
| CDK2 | CDK | CMGC | 3qql | A | B | (5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4378 | |
| CDK2 | CDK | CMGC | 7nvq | A | | staurosporine | Human | 13627 | |
| CDK2 | CDK | CMGC | 1h07 | A | B | ((2-bromo-4-methylphenyl){6-[(4-{[(2s)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrile | Human | 3908 | |
| CDK2 | CDK | CMGC | 5uq1 | A | | - | Human | 8220 | |
| CDK2 | CDK | CMGC | 2uue | A | | 4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amine | Human | 4515 | |
| CDK2 | CDK | CMGC | 4fki | A | A | n-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamide | Human | 4430 | |
| CDK2 | CDK | CMGC | 4cfm | A | B | 6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amine | Human | 3986 | |
| CDK2 | CDK | CMGC | 2c6t | A | | 4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamide | Human | 4371 | |
| CDK2 | CDK | CMGC | 6guh | A | A | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10765 | |
| CDK2 | CDK | CMGC | 2xnb | A | B | 3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-one | Human | 4034 | |
| CDK2 | CDK | CMGC | 4bcq | C | A | 4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrile | Human | 3996 | |
| CDK2 | CDK | CMGC | 5osj | A | B | - | Human | 9742 | |
| CDK2 | CDK | CMGC | 6yl1 | A | B | methyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | 12496 | |
| CDK2 | CDK | CMGC | 3rzb | A | A | 4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamide | Human | 4264 | |
| CDK2 | CDK | CMGC | 2xmy | A | A | 4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamide | Human | 4526 | |
| CDK2 | CDK | CMGC | 2cch | A | C | - | Human | 4566 | |
| CDK2 | CDK | CMGC | 3rai | A | B | 4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4002 | |
| GSK3B | GSK | CMGC | 3f7z | B | B | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 670 | |
| GSK3B | GSK | CMGC | 6v6l | A | A | 1-(6-((2-((6-amino-5-nitropyridin-2-yl)amino)ethyl)amino)-2-(2,4-dichlorophenyl)pyridin-3-yl)-4-methylpiperazin-2-one | Human | 11913 | |
| GSK3B | GSK | CMGC | 3f88 | B | A | 5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 744 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu6 | B | | ~{n}-(1~{h}-benzimidazol-2-ylmethyl)-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amine | Human | 14921 | |
| CDK12 (CRK7) | CDK | CMGC | 9fmr | B | | ~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amine | Human | 15854 | |
| MAPK13 (p38d) | MAPK | CMGC | 4yno | A | | - | Human | 2947 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8pt9 | A | | methyl (1s,3s)-1-methyl-3-[[3-[[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]carbamoyl]-4-oxidanylidene-cyclohexane-1-carboxylate | Human | 15293 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8pta | A | | methyl (1r,3s)-1-methyl-3-[[3-[[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]carbamoyl]-4-oxidanylidene-cyclohexane-1-carboxylate | Human | 15294 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8pt8 | A | | methyl (1r,3r)-1-methyl-3-[[3-[[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methylcarbamoyl]-4-oxidanylidene-cyclohexane-1-carboxylate | Human | 15295 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psw | A | B | amp phosphoramidate | Human | 15303 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt3 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15304 | |
| CDK6 | CDK | CMGC | 6oqo | A | | n-[5-(6-ethyl-2,6-diazaspiro[3.3]heptan-2-yl)pyridin-2-yl]-5-fluoro-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amine | Human | 12646 | |
| CDK6 | CDK | CMGC | 9d8u | A | | atirmociclib | Human | 15857 | |
| CDK6 | CDK | CMGC | 1g3n | A | | - | Human | 2806 | |
| CDK6 | CDK | CMGC | 1bi7 | A | | - | Human | 2798 | |
| CDK6 | CDK | CMGC | 1blx | A | | - | Human | 2802 | |
| CDK6 | CDK | CMGC | 1bi8 | A | | - | Human | 2796 | |
| CDK6 | CDK | CMGC | 6oql | A | | 5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amine | Human | 12647 | |
| CDK6 | CDK | CMGC | 9pe7 | A | | (3r,4r)-4-({(4m)-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-1,3-benzimidazol-6-yl]pyrimidin-2-yl}amino)-1-(methanesulfonyl)piperidin-3-ol | Human | 15858 | |
| CDK6 | CDK | CMGC | 1jow | B | | - | Human | 2793 | |
| CDK6 | CDK | CMGC | 1bi8 | C | | - | Human | 2799 | |
| CDK6 | CDK | CMGC | 4ez5 | A | | {5-[4-(dimethylamino)piperidin-1-yl]-1h-imidazo[4,5-b]pyridin-2-yl}[2-(isoquinolin-4-yl)pyridin-4-yl]methanone | Human | 2800 | |
| CDK6 | CDK | CMGC | 2euf | B | | 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 2804 | |
| CDK6 | CDK | CMGC | 1xo2 | B | | 3,7,3',4'-tetrahydroxyflavone | Human | 2794 | |
| CDK2 | CDK | CMGC | 1w0x | C | B | olomoucine | Human | 4478 | |
| CDK2 | CDK | CMGC | 1h01 | A | A | (2r)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | 3974 | |
| CDK2 | CDK | CMGC | 6p3w | C | B | - | Human | 11516 | |
| CDK2 | CDK | CMGC | 1h07 | A | A | ((2-bromo-4-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrile | Human | 3918 | |
| CDK2 | CDK | CMGC | 1pxj | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 3927 | |
| CDK2 | CDK | CMGC | 2iw9 | C | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4218 | |
| CDK2 | CDK | CMGC | 4bcp | A | A | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4552 | |
| CDK2 | CDK | CMGC | 2b55 | A | | 2-(4-(aminomethyl)piperidin-1-yl)-n-(3_cyclohexyl-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)acetamide | Human | 4216 | |
| CDK2 | CDK | CMGC | 6q4d | A | A | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid | Human | 11184 | |
| CDK2 | CDK | CMGC | 3roy | A | A | 4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4131 | |
| CDK2 | CDK | CMGC | 4ii5 | A | B | adenosine-5'-diphosphate | Human | 4456 | |
| CDK2 | CDK | CMGC | 3uli | A | A | 1-(aminomethyl)-n-(3-{[6-bromo-2-(4-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-7-yl]amino}propyl)cyclopropanecarboxamide | Human | 4115 | |
| CDK2 | CDK | CMGC | 3bht | A | B | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4491 | |
| CDK2 | CDK | CMGC | 3r8m | A | B | 1h-indazole-3-carbohydrazide | Human | 4451 | |
| CDK2 | CDK | CMGC | 2w06 | A | | 4-{[4-(1-cyclopropyl-2-methyl-1h-imidazol-5-yl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamide | Human | 3982 | |
| CDK2 | CDK | CMGC | 2uzd | A | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamide | Human | 3877 | |
| CDK2 | CDK | CMGC | 5ang | A | | 7-hydroxy-4-(morpholinomethyl)chromen-2-one | Human | 6540 | |
| CDK2 | CDK | CMGC | 5k4j | A | A | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 6751 | |
| CDK2 | CDK | CMGC | 2c5o | C | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4050 | |
| CDK2 | CDK | CMGC | 4fks | A | C | n-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamide | Human | 4315 | |
| CDK2 | CDK | CMGC | 2iw9 | A | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4174 | |
| CDK2 | CDK | CMGC | 3r71 | A | B | 4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4345 | |
| CDK2 | CDK | CMGC | 2btr | A | | n-(5-isopropyl-thiazol-2-yl)-2-pyridin-3-yl-acetamide | Human | 3998 | |
| CDK2 | CDK | CMGC | 9d0w | C | | - | Human | 15925 | |
| CDK2 | CDK | CMGC | 2r3f | A | B | 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4291 | |
| CDK2 | CDK | CMGC | 1p2a | A | | 5-[(2-aminoethyl)amino]-6-fluoro-3-(1h-pyrrol-2-yl)benzo[cd]indol-2(1h)-one | Human | 4422 | |
| CDK2 | CDK | CMGC | 3rpo | A | A | 4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acid | Human | 3966 | |
| CDK2 | CDK | CMGC | 1urc | C | B | - | Human | 3937 | |
| CDK2 | CDK | CMGC | 4cfw | C | C | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4102 | |
| CDK2 | CDK | CMGC | 2r3p | A | A | 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amine | Human | 4176 | |
| CDK2 | CDK | CMGC | 5oo0 | A | C | - | Human | 9745 | |
| CDK2 | CDK | CMGC | 1v1k | A | B | (2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-ol | Human | 3928 | |
| CDK2 | CDK | CMGC | 1jsu | A | | - | Human | 4146 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu7 | E | | - | Human | 10782 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu2 | A | A | 2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-one | Human | 10780 | |
| CDK1 (CDC2) | CDK | CMGC | 6gu3 | A | | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10778 | |
| MAPK10 (JNK3) | MAPK | CMGC | 1pmn | A | | cyclopropyl-{4-[5-(3,4-dichlorophenyl)-2-[(1-methyl)-piperidin]-4-yl-3-propyl-3h-imidazol-4-yl]-pyrimidin-2-yl}amine | Human | 3439 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2ok1 | A | A | n-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamide | Human | 3444 | |
| CDK2 | CDK | CMGC | 6oqi | A | | 5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4s)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amine | Human | 12648 | |
| CDK12 (CRK7) | CDK | CMGC | 6ckx | A | | n-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamide | Human | 10578 | |
| CDK6 | CDK | CMGC | 5l2s | A | | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 6990 | |
| CDK2 | CDK | CMGC | 2wpa | C | | n-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamide | Human | 4162 | |
| CDK2 | CDK | CMGC | 9et7 | A | B | 4-bromanyl-1~{h}-pyridin-2-one | Human | 15907 | |
| CDK2 | CDK | CMGC | 2exm | A | | n-(3-methylbut-2-en-1-yl)-9h-purin-6-amine | Human | 4055 | |
| CDK2 | CDK | CMGC | 1h1r | C | B | 6-cyclohexylmethoxy-2-(3'-chloroanilino) purine | Human | 4081 | |
| CDK2 | CDK | CMGC | 1pxo | A | D | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4167 | |
| CDK2 | CDK | CMGC | 3bhv | A | B | 9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-ol | Human | 4001 | |
| CDK2 | CDK | CMGC | 4fku | A | A | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 3863 | |
| CDK2 | CDK | CMGC | 6q4a | A | A | 5-iodanylpyrimidine | Human | 11195 | |
| CDK2 | CDK | CMGC | 4ek8 | A | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amine | Human | 3871 | |
| CDK2 | CDK | CMGC | 9d0x | B | | - | Human | 15910 | |
| CDK2 | CDK | CMGC | 4bco | A | A | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 3988 | |
| CDK2 | CDK | CMGC | 5iex | A | A | (2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-ol | Human | 6565 | |
| CDK2 | CDK | CMGC | 8b54 | A | B | ~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | 14680 | |
| CDK2 | CDK | CMGC | 1urc | A | B | - | Human | 4010 | |
| CDK2 | CDK | CMGC | 3r28 | A | A | 4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamide | Human | 4052 | |
| CDK2 | CDK | CMGC | 4bcp | C | B | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4501 | |
| CDK2 | CDK | CMGC | 9hiu | B | | - | Human | 15912 | |
| CDK2 | CDK | CMGC | 2b52 | A | | 1-(3-(2,4-dimethylthiazol-5-yl)-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)-3-(4-methylpiperazin-1-yl)urea | Human | 3997 | |
| CDK2 | CDK | CMGC | 6gva | A | A | 5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | 11206 | |
| CDK2 | CDK | CMGC | 3r1y | A | A | 2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4319 | |
| CDK2 | CDK | CMGC | 6yl1 | A | A | methyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | 12497 | |
| CDK2 | CDK | CMGC | 4cfu | A | A | 3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acid | Human | 3905 | |
| CDK2 | CDK | CMGC | 2c4g | A | | (3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-ium | Human | 4088 | |
| CDK2 | CDK | CMGC | 4rj3 | A | A | 1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amine | Human | 4244 | |
| CDK2 | CDK | CMGC | 1h26 | C | | - | Human | 4179 | |
| CDK2 | CDK | CMGC | 6q4b | A | C | 5-bromanylpyrimidine | Human | 11180 | |
| CDK2 | CDK | CMGC | 9esl | A | B | 4-bromanyl-1-(2-methoxyethyl)pyridin-2-one | Human | 15931 | |
| CDK2 | CDK | CMGC | 3r7u | A | A | 2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamide | Human | 4510 | |
| CDK2 | CDK | CMGC | 4eom | A | B | adenosine-5'-triphosphate | Human | 4472 | |
| CDK2 | CDK | CMGC | 3qwk | A | A | 4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamide | Human | 4091 | |
| CDK2 | CDK | CMGC | 1pxj | A | B | - | Human | 3911 | |
| CDK2 | CDK | CMGC | 2whb | C | A | - | Human | 4132 | |
| CDK2 | CDK | CMGC | 4fkp | A | A | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4035 | |
| CDK2 | CDK | CMGC | 6inl | A | | 2,2'-{[6-{[(4-methoxyphenyl)methyl]amino}-9-(propan-2-yl)-9h-purin-2-yl]azanediyl}di(ethan-1-ol) | Human | 11794 | |
| CDK2 | CDK | CMGC | 4eol | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4270 | |
| CDK2 | CDK | CMGC | 3dog | C | B | (2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol | Human | 4121 | |
| CDK2 | CDK | CMGC | 3r7i | A | B | 4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acid | Human | 4070 | |
| CDK2 | CDK | CMGC | 9esq | A | B | 4-bromanyl-2-oxidanyl-benzoic acid | Human | 15933 | |
| CDK2 | CDK | CMGC | 3rpv | A | A | 4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4348 | |
| CDK2 | CDK | CMGC | 3qzi | A | B | 4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamide | Human | 4500 | |
| CDK2 | CDK | CMGC | 4fkq | A | B | 4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamide | Human | 4026 | |
| CDK2 | CDK | CMGC | 4eop | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4463 | |
| CDK2 | CDK | CMGC | 2bts | A | | 4-[(5-isopropyl-1,3-thiazol-2-yl)amino]benzenesulfonamide | Human | 4443 | |
| CDK2 | CDK | CMGC | 3tnw | A | A | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 4254 | |
| CDK2 | CDK | CMGC | 1h08 | A | B | (2s)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-ol | Human | 4411 | |
| CDK2 | CDK | CMGC | 3r1q | A | A | 4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamide | Human | 4224 | |
| CDK2 | CDK | CMGC | 3pxz | A | | 8-anilino-1-naphthalene sulfonate | Human | 4251 | |
| CDK2 | CDK | CMGC | 1qmz | C | | adenosine-5'-triphosphate | Human | 4527 | |
| CDK2 | CDK | CMGC | 1pxk | A | A | n-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n'-hydroxyimidoformamide | Human | 3915 | |
| CDK2 | CDK | CMGC | 4cfx | C | A | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4166 | |
| CDK2 | CDK | CMGC | 3my5 | C | A | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 4473 | |
| CDK2 | CDK | CMGC | 3sw4 | A | B | n'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamine | Human | 4439 | |
| CDK2 | CDK | CMGC | 2r3g | A | A | 6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amine | Human | 4276 | |
| CDK2 | CDK | CMGC | 9esu | A | D | - | Human | 15934 | |
| CDK2 | CDK | CMGC | 4eos | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4028 | |
| CDK2 | CDK | CMGC | 2c5y | A | A | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 6785 | |
| CDK2 | CDK | CMGC | 4eol | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4235 | |
| CDK2 | CDK | CMGC | 9esn | A | B | 4-bromo-1-(2-hydroxyethyl)pyridin-2(1h)-one | Human | 15923 | |
| CDK2 | CDK | CMGC | 3bhv | A | A | 9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-ol | Human | 4531 | |
| CDK2 | CDK | CMGC | 3my5 | A | B | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 3887 | |
| CDK2 | CDK | CMGC | 6q4f | A | A | pyridine-2,6-diamine | Human | 11202 | |
| CDK2 | CDK | CMGC | 5if1 | C | B | - | Human | 6571 | |
| CDK2 | CDK | CMGC | 6sg4 | A | A | - | Human | 13246 | |
| CDK2 | CDK | CMGC | 4eoq | A | A | adenosine-5'-triphosphate | Human | 4402 | |
| CDK2 | CDK | CMGC | 5a14 | A | B | 1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea | Human | 3901 | |
| CDK2 | CDK | CMGC | 5cyi | C | A | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | 6055 | |
| CDK2 | CDK | CMGC | 3sw4 | A | A | n'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamine | Human | 4076 | |
| CDK2 | CDK | CMGC | 4bck | C | B | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4506 | |
| CDK2 | CDK | CMGC | 2vts | A | | 5-[(4-aminocyclohexyl)amino]-7-(propan-2-ylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 4300 | |
| CDK2 | CDK | CMGC | 9et2 | A | A | ~{n}-(4-bromophenyl)ethanamide | Human | 15924 | |
| DYRK1A | DYRK | CMGC | 2wo6 | A | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3764 | |
| CDK2 | CDK | CMGC | 1f5q | C | B | - | Human | 3952 | |
| CDK2 | CDK | CMGC | 3r1y | A | B | 2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4405 | |
| CDK2 | CDK | CMGC | 1ckp | A | B | purvalanol b | Human | 4214 | |
| CDK2 | CDK | CMGC | 4kd1 | A | B | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 4525 | |
| CDK2 | CDK | CMGC | 3igg | A | | n-[1-(cis-3-hydroxycyclobutyl)-1h-imidazol-4-yl]-2-(4-methoxyphenyl)acetamide | Human | 4360 | |
| CDK2 | CDK | CMGC | 3qxp | A | A | 4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4343 | |
| CDK2 | CDK | CMGC | 3r9d | A | B | 4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4565 | |
| CDK2 | CDK | CMGC | 2r3i | A | B | 5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4059 | |
| CDK2 | CDK | CMGC | 1h28 | C | | - | Human | 4351 | |
| CDK2 | CDK | CMGC | 2whb | A | B | - | Human | 4457 | |
| CDK2 | CDK | CMGC | 1v1k | A | A | (2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-ol | Human | 4189 | |
| CDK2 | CDK | CMGC | 11gv | A | A | (1r,3s)-3-{3-[(1-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl bicyclo[1.1.1]pentan-1-ylcarbamate | Human | 15932 | |
| CDK2 | CDK | CMGC | 6q4f | A | C | pyridine-2,6-diamine | Human | 11212 | |
| CDK2 | CDK | CMGC | 3r8z | A | B | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanone | Human | 4140 | |
| CDK2 | CDK | CMGC | 5lmk | A | A | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | 7399 | |
| CDK2 | CDK | CMGC | 3bhu | C | B | 4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 4464 | |
| CDK2 | CDK | CMGC | 2uzb | C | D | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamide | Human | 4502 | |
| CDK2 | CDK | CMGC | 6q4d | A | C | 2-(4-bromanyl-2-methoxy-phenyl)ethanoic acid | Human | 11188 | |
| CDK2 | CDK | CMGC | 2w17 | A | B | n-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 4165 | |
| CDK2 | CDK | CMGC | 3qhw | A | A | adenosine-5'-diphosphate | Human | 4346 | |
| CDK2 | CDK | CMGC | 2uze | C | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acid | Human | 4071 | |
| CDK2 | CDK | CMGC | 1oi9 | C | A | 6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purine | Human | 4571 | |
| CDK2 | CDK | CMGC | 3rk7 | A | | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzamide | Human | 4236 | |
| CDK2 | CDK | CMGC | 1f5q | A | B | - | Human | 4517 | |
| CDK2 | CDK | CMGC | 3r8p | A | B | (5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4538 | |
| CDK2 | CDK | CMGC | 3rk9 | A | A | [4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4158 | |
| CDK2 | CDK | CMGC | 3tnw | A | B | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 3948 | |
| CDK2 | CDK | CMGC | 9nyr | A | A | - | Human | 15939 | |
| CDK2 | CDK | CMGC | 3s2p | A | | (3s,4s)-1-{3-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-4-hydroxyphenyl}pyrrolidine-3,4-diol | Human | 4404 | |
| CDK2 | CDK | CMGC | 5jq5 | A | | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 7416 | |
| CDK2 | CDK | CMGC | 4eop | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4044 | |
| CDK2 | CDK | CMGC | 2vtp | A | A | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4511 | |
| CDK2 | CDK | CMGC | 2cjm | C | | adenosine-5'-triphosphate | Human | 4126 | |
| CDK2 | CDK | CMGC | 9et7 | A | A | 4-bromanyl-1~{h}-pyridin-2-one | Human | 15940 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u9c | B | | 7-hydroxy-3h-phenoxazin-3-one | Human | 5523 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu6 | A | B | adenosine-5'-triphosphate | Human | 6906 | |
| DYRK2 | DYRK | CMGC | 5lxc | B | B | methyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7126 | |
| CDK2 | CDK | CMGC | 2c5n | C | A | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 4161 | |
| CDK2 | CDK | CMGC | 3my5 | A | A | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 4554 | |
| CDK2 | CDK | CMGC | 4cfu | C | B | 3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acid | Human | 4539 | |
| CDK2 | CDK | CMGC | 9esk | A | A | (4-bromo-2-oxopyridin-1(2h)-yl)acetic acid | Human | 15945 | |
| CDK2 | CDK | CMGC | 2duv | A | | 2-(3,4-dihydroxyphenyl)-8-(1,1-dioxidoisothiazolidin-2-yl)-3-hydroxy-6-methyl-4h-chromen-4-one | Human | 4193 | |
| CDK2 | CDK | CMGC | 3qql | A | A | (5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazide | Human | 4341 | |
| CDK2 | CDK | CMGC | 1pkd | C | | 7-hydroxystaurosporine | Human | 3973 | |
| CDK2 | CDK | CMGC | 3r9h | A | A | 4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 3958 | |
| CDK2 | CDK | CMGC | 4fx3 | C | B | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 4495 | |
| CDK2 | CDK | CMGC | 7ra5 | A | A | 4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amine | Human | 13960 | |
| CDK2 | CDK | CMGC | 9etp | A | B | 4-bromo-1h-pyrazole | Human | 15949 | |
| CDK2 | CDK | CMGC | 6q3f | A | B | - | Human | 11187 | |
| CDK2 | CDK | CMGC | 2c5n | A | B | n-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamine | Human | 4223 | |
| CDK2 | CDK | CMGC | 4fkw | A | A | 2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylate | Human | 4252 | |
| CDK2 | CDK | CMGC | 5if1 | C | A | - | Human | 6564 | |
| CLK3 | CLK | CMGC | 6fyr | A | B | 6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamide | Human | 11406 | |
| CDK2 | CDK | CMGC | 4acm | A | B | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 3983 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qte | A | B | 4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamide | Human | 2564 | |
| CDK2 | CDK | CMGC | 2whb | A | A | - | Human | 4471 | |
| CDK2 | CDK | CMGC | 1okv | C | | - | Human | 4093 | |
| CDK2 | CDK | CMGC | 4bco | C | A | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4333 | |
| CDK2 | CDK | CMGC | 2c68 | A | | (5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydropyrazolo[1,5-a]pyrimidin-7-amine | Human | 6776 | |
| CDK2 | CDK | CMGC | 2vtm | A | | pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 4283 | |
| CDK2 | CDK | CMGC | 1oit | A | | 4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]benzenesulfonamide | Human | 4025 | |
| CDK2 | CDK | CMGC | 4gcj | A | B | 4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4362 | |
| CDK2 | CDK | CMGC | 3qts | A | A | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanone | Human | 4275 | |
| CDK2 | CDK | CMGC | 3fz1 | A | | (3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-one | Human | 4335 | |
| CDK2 | CDK | CMGC | 4fku | A | B | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 4573 | |
| CDK2 | CDK | CMGC | 2uze | A | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acid | Human | 3949 | |
| CDK2 | CDK | CMGC | 2vtp | A | B | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 4401 | |
| CDK2 | CDK | CMGC | 6q4c | A | A | 4-bromanyl-1,8-naphthyridine | Human | 11182 | |
| MAPK8 (JNK1) | MAPK | CMGC | 5lw1 | B | | adenosine | Human | 9081 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | A | A | - | Human | 6452 | |
| CDK8 | CDK | CMGC | 4f6w | A | | n-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-4-[2-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)ethyl]piperazine-1-carboxamide | Human | 3845 | |
| CDK8 | CDK | CMGC | 4f7l | A | | tert-butyl [3-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)propyl]carbamate | Human | 3840 | |
| CDK8 | CDK | CMGC | 4f6u | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]urea | Human | 3844 | |
| CDK2 | CDK | CMGC | 2wip | A | | 1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acid | Human | 4520 | |
| CDK2 | CDK | CMGC | 2i40 | C | A | 5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamide | Human | 4222 | |
| CDK2 | CDK | CMGC | 4cfm | C | B | 6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amine | Human | 4005 | |
| CDK2 | CDK | CMGC | 6q4j | A | B | 2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acid | Human | 11213 | |
| CDK2 | CDK | CMGC | 4bcq | A | B | 4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrile | Human | 4415 | |
| CDK2 | CDK | CMGC | 2j9m | A | B | 6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxide | Human | 4246 | |
| CDK2 | CDK | CMGC | 1p5e | C | | 4,5,6,7-tetrabromobenzotriazole | Human | 4434 | |
| CDK2 | CDK | CMGC | 2iw8 | A | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4142 | |
| CDK2 | CDK | CMGC | 3ddq | A | B | r-roscovitine | Human | 4269 | |
| CDK2 | CDK | CMGC | 1w8c | A | B | 6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amine | Human | 4197 | |
| CDK2 | CDK | CMGC | 3rk5 | A | | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzoic acid | Human | 4160 | |
| CDK2 | CDK | CMGC | 9esw | A | A | (4-bromanylpyridin-2-yl)methanol | Human | 15935 | |
| CLK1 | CLK | CMGC | 6z4z | B | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12310 | |
| CDK2 | CDK | CMGC | 1h1p | C | | 6-o-cyclohexylmethyl guanine | Human | 4581 | |
| CDK2 | CDK | CMGC | 3rk9 | A | B | [4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4259 | |
| CDK2 | CDK | CMGC | 9esw | A | C | - | Human | 15936 | |
| CDK2 | CDK | CMGC | 1buh | A | | - | Human | 4178 | |
| CDK2 | CDK | CMGC | 3sqq | A | A | 4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4231 | |
| CDK2 | CDK | CMGC | 2wxv | A | | n,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4318 | |
| CDK2 | CDK | CMGC | 4fkv | A | A | (3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamide | Human | 4299 | |
| CDK2 | CDK | CMGC | 9hj1 | B | | - | Human | 15937 | |
| CDK2 | CDK | CMGC | 3bht | C | B | 4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 3889 | |
| CDK2 | CDK | CMGC | 9esu | A | A | 4-bromanyl-2-(methoxymethyl)pyridine | Human | 15938 | |
| CDK2 | CDK | CMGC | 4bcn | C | B | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 4150 | |
| CDK2 | CDK | CMGC | 4eoo | C | A | adenosine-5'-triphosphate | Human | 4188 | |
| CDK2 | CDK | CMGC | 3r7e | A | B | 5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamide | Human | 4447 | |
| CDK2 | CDK | CMGC | 9ob3 | A | | (1r,3r)-3-{3-[(pyrazine-2-carbonyl)amino]-1h-pyrazol-5-yl}cyclopentyl [(1s)-1-cyclopropylethyl]carbamate | Human | 15941 | |
| CDK2 | CDK | CMGC | 5osm | A | A | methyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylate | Human | 9741 | |
| CDK2 | CDK | CMGC | 2r3m | A | B | n-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amine | Human | 4576 | |
| CDK2 | CDK | CMGC | 2c5x | C | A | hydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammonium | Human | 4466 | |
| CDK2 | CDK | CMGC | 4bcq | A | A | 4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrile | Human | 4396 | |
| CDK2 | CDK | CMGC | 3r73 | A | B | 4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 3899 | |
| CDK2 | CDK | CMGC | 5fp6 | A | B | 3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-ol | Human | 6301 | |
| CDK2 | CDK | CMGC | 2wma | C | | - | Human | 4410 | |
| CDK2 | CDK | CMGC | 9jj5 | A | | ~{n}-(4-azanylcyclohexyl)-4-[[2,6-bis(fluoranyl)-3-[4-(methylcarbamoyl)phenyl]phenyl]carbonylamino]-1~{h}-pyrazole-3-carboxamide | Human | 15942 | |
| CDK2 | CDK | CMGC | 3ql8 | A | A | 3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrile | Human | 3916 | |
| CDK2 | CDK | CMGC | 2c5o | A | A | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4388 | |
| CDK2 | CDK | CMGC | 5iex | A | B | (2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-ol | Human | 6572 | |
| CDK2 | CDK | CMGC | 3qzf | A | | 2-(4,6-diamino-1,3,5-triazin-2-yl)benzene-1,4-diol | Human | 4569 | |
| CDK2 | CDK | CMGC | 2a0c | X | A | 2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenol | Human | 4157 | |
| CDK2 | CDK | CMGC | 5a14 | A | A | 1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea | Human | 3977 | |
| CDK2 | CDK | CMGC | 4gcj | A | A | 4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4138 | |
| CDK2 | CDK | CMGC | 1urw | A | B | 2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]- | Human | 4196 | |
| CDK2 | CDK | CMGC | 8b54 | A | A | ~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amine | Human | 14681 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7cml | B | A | - | Human | 12706 | |
| CDK2 | CDK | CMGC | 9hiw | B | | - | Human | 15943 | |
| CDK2 | CDK | CMGC | 4bck | A | D | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4563 | |
| CDK2 | CDK | CMGC | 5ani | A | | 6-chloro-9h-purine | Human | 6539 | |
| CDK9 | CDK | CMGC | 4ec8 | A | | - | Human | 2244 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | A | | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | 12791 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | B | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12792 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yll | A | | ~{n}4-[3-(4-methoxyphenyl)-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]cyclohexane-1,4-diamine | Human | 12793 | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | A | A | - | Human | 12982 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | D | | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | 12795 | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | B | B | - | Human | 12983 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | D | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12796 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6ylc | B | | 5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrile | Human | 12797 | |
| DYRK1A | DYRK | CMGC | 6yf8 | C | | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | 13463 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6l | A | A | 5-azanyl-3-[(~{z})-1-cyano-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]-3~{h}-pyrazole-4-carbonitrile | Human | 15275 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c6n | A | A | (2~{z},5~{z})-5-[(4-methoxy-3-oxidanyl-phenyl)methylidene]-2-phenylimino-1,3-thiazolidin-4-one | Human | 15276 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | A | A | benzoic acid | Human | 11281 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moe | A | A | adenosine-5'-diphosphate | Human | 7650 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmr | B | B | - | Human | 7680 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3wik | A | | n-[5-(4-nitrophenyl)-1,3,4-thiadiazol-2-yl]acetamide | Human | 5459 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4w4x | A | | 3-(4-{[(4-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamide | Human | 3440 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ots | A | B | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3,5-bis(chloranyl)-4-phenyl-phenyl]methyl]azanium | Human | 10599 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot6 | A | A | (3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-pyrrol-2-yl)ethyl]azanium | Human | 9619 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9gcw | A | B | - | Human | 16073 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oni | B | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9454 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvg | A | B | - | Human | 6908 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hop | A | C | (~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-one | Human | 11662 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yzh | A | A | adenosine-5'-diphosphate | Human | 13559 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlw | A | B | 7-bromanyl-1~{h}-benzotriazole | Human | 13085 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owk | A | B | 7-chloro-10-methyl-11h-benzo[g]pyrido[4,3-b]indol-3-ol | Human | 5433 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | F | | - | Human | 5473 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4c | A | A | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13170 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rfe | A | A | (~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12148 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlu | A | B | 6,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13090 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo5 | B | B | - | Human | 7656 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otl | B | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9616 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csp | A | A | 2-hydroxy-5-methylbenzoic acid | Human | 6904 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s9y | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 16087 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu6 | A | A | adenosine-5'-triphosphate | Human | 6899 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe2 | A | B | 5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5519 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csp | A | B | 2-hydroxy-5-methylbenzoic acid | Human | 6905 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s7a | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 16088 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlu | A | A | 6,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13091 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot5 | B | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9605 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mow | A | B | 5-bromopyridine-2,3-diamine | Human | 7684 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4c | B | B | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13171 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s7a | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 16089 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9h97 | A | | 1,2,3,4-tetrakis(bromanyl)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 16090 | |
| CDK2 | CDK | CMGC | 2c69 | A | | (5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-7-amine | Human | 6775 | |
| CDK2 | CDK | CMGC | 1pw2 | A | | - | Human | 4432 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3war | A | B | nicotinic acid | Human | 5464 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s7h | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 16097 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4c | B | A | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13173 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe2 | A | A | 5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5508 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmf | A | A | (3-chloranyl-4-phenyl-phenyl)methyl-propyl-azanium | Human | 7682 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4c | A | B | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13174 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9qst | A | | 5-[4-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanoylamino]butylamino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 16101 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owl | A | A | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10593 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hbn | A | B | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11284 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otz | A | A | trifluoroacetic acid | Human | 9650 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mp8 | B | B | adenosine-5'-diphosphate | Human | 7692 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqu | A | A | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6035 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8p05 | A | | (4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-one | Human | 14744 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otd | B | A | [2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azanium | Human | 9690 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu0 | B | B | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7301 | |
| CDK2 | CDK | CMGC | 1wcc | A | B | 2-amino-6-chloropyrazine | Human | 3897 | |
| CDK2 | CDK | CMGC | 3lfq | A | | n-(6,7-difluoro-5-phenyl-1h-indazol-3-yl)butanamide | Human | 4320 | |
| CDK2 | CDK | CMGC | 4ek4 | A | B | 4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamide | Human | 3957 | |
| CDK2 | CDK | CMGC | 4cfn | C | B | 6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amine | Human | 4567 | |
| CDK2 | CDK | CMGC | 4eoi | A | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4342 | |
| CDK2 | CDK | CMGC | 6ylk | A | A | methyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylate | Human | 12499 | |
| CDK2 | CDK | CMGC | 2x1n | C | A | 2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amine | Human | 3991 | |
| CDK2 | CDK | CMGC | 2c5o | A | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amine | Human | 4440 | |
| CDK2 | CDK | CMGC | 3pxf | A | B | 8-anilino-1-naphthalene sulfonate | Human | 4301 | |
| CDK8 | CDK | CMGC | 6t41 | A | | ~{n}-[(4-chlorophenyl)methyl]quinazolin-4-amine | Human | 11908 | |
| CDK2 | CDK | CMGC | 3r7y | A | B | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamide | Human | 3975 | |
| CDK2 | CDK | CMGC | 1pxn | A | B | - | Human | 4172 | |
| CDK2 | CDK | CMGC | 3tiy | A | A | 2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-one | Human | 4413 | |
| CDK2 | CDK | CMGC | 6q3b | A | B | 4-iodopyrazole | Human | 11208 | |
| CDK2 | CDK | CMGC | 1hck | A | B | adenosine-5'-triphosphate | Human | 4416 | |
| CDK2 | CDK | CMGC | 1h01 | A | B | (2s)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-ol | Human | 4561 | |
| CDK2 | CDK | CMGC | 5lmk | C | A | 4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamide | Human | 7396 | |
| CDK2 | CDK | CMGC | 1qmz | A | | adenosine-5'-triphosphate | Human | 4242 | |
| CDK8 | CDK | CMGC | 5idp | A | B | (3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanone | Human | 7320 | |
| CDK8 | CDK | CMGC | 5icp | A | A | [(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanone | Human | 7318 | |
| CDK8 | CDK | CMGC | 8tqc | C | B | - | Human | 15963 | |
| CDK8 | CDK | CMGC | 5xs2 | A | A | 3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamide | Human | 8315 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n67 | A | A | - | Human | 8523 | |
| MAPK14 (p38a) | MAPK | CMGC | 1r3c | A | A | - | Human | 5170 | |
| DYRK2 | DYRK | CMGC | 7dl6 | A | | [2,7-dimethoxy-9-[[(3r)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanol | Human | 14013 | |
| DYRK2 | DYRK | CMGC | 5lxd | B | B | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 7127 | |
| DYRK2 | DYRK | CMGC | 7dhc | A | | 4-[bis(fluoranyl)methyl]-2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine | Human | 13973 | |
| DYRK2 | DYRK | CMGC | 7djo | A | | [2,7-dimethoxy-9-[[(3s)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanol | Human | 13994 | |
| DYRK2 | DYRK | CMGC | 6hdp | A | A | scorzodihydrostilbene a | Human | 11572 | |
| DYRK2 | DYRK | CMGC | 3kvw | A | A | (2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acid | Human | 3148 | |
| CDK8 | CDK | CMGC | 8tq2 | C | B | - | Human | 15964 | |
| CDK8 | CDK | CMGC | 5idn | A | B | [(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanone | Human | 7319 | |
| CDK8 | CDK | CMGC | 5hbj | A | B | 8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-one | Human | 6385 | |
| CDK8 | CDK | CMGC | 6y0a | A | B | 6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamide | Human | 13305 | |
| CDK8 | CDK | CMGC | 8tq2 | C | A | - | Human | 15965 | |
| CDK8 | CDK | CMGC | 8tqc | C | A | - | Human | 15966 | |
| CDK8 | CDK | CMGC | 6r3s | A | A | 6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamide | Human | 12140 | |
| CDK8 | CDK | CMGC | 5cei | A | A | 4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamide | Human | 6404 | |
| CLK2 | CLK | CMGC | 5unp | A | | n~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamine | Human | 9887 | |
| GSK3B | GSK | CMGC | 1r0e | A | A | 3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 733 | |
| GSK3B | GSK | CMGC | 3zrl | A | C | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 654 | |
| GSK3B | GSK | CMGC | 1q3d | B | | staurosporine | Human | 752 | |
| MAPK13 (p38d) | MAPK | CMGC | 8x23 | A | B | - | Human | 15128 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byz | A | B | 4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamide | Human | 6592 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsg | A | A | 3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | 6589 | |
| MAPK7 (Erk5) | MAPK | CMGC | 5byz | A | A | 4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamide | Human | 6590 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4zsj | A | A | 3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamide | Human | 6588 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic8 | B | | - | Human | 389 | |
| MAPK7 (Erk5) | MAPK | CMGC | 4ic8 | A | | - | Human | 390 | |
| CDKL5 | CDKL | CMGC | 8cie | A | | 4-[[3,5-bis(fluoranyl)phenyl]carbonylamino]-~{n}-piperidin-4-yl-1~{h}-pyrazole-3-carboxamide | Human | 14778 | |
| CLK3 | CLK | CMGC | 6z54 | A | A | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12294 | |
| CLK3 | CLK | CMGC | 2eu9 | A | B | - | Human | 1830 | |
| CLK3 | CLK | CMGC | 6z54 | A | B | 11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12295 | |
| CLK3 | CLK | CMGC | 6z51 | A | A | n-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide | Human | 12296 | |
| CLK3 | CLK | CMGC | 2exe | A | A | - | Human | 1822 | |
| CLK3 | CLK | CMGC | 6fyp | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10400 | |
| CLK3 | CLK | CMGC | 6rct | A | A | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11127 | |
| CLK3 | CLK | CMGC | 6z52 | A | A | 11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12628 | |
| CLK3 | CLK | CMGC | 3raw | A | A | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 1820 | |
| CLK3 | CLK | CMGC | 6z55 | B | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12299 | |
| CLK3 | CLK | CMGC | 2wu6 | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 1821 | |
| CLK3 | CLK | CMGC | 6fyp | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10397 | |
| CLK3 | CLK | CMGC | 6z55 | A | C | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12301 | |
| CLK3 | CLK | CMGC | 3raw | A | B | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 1829 | |
| CLK3 | CLK | CMGC | 6z52 | B | A | 11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one | Human | 12629 | |
| CLK3 | CLK | CMGC | 6yu1 | a | B | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12408 | |
| CLK3 | CLK | CMGC | 6z55 | B | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12303 | |
| CLK3 | CLK | CMGC | 6z51 | A | B | n-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide | Human | 12304 | |
| CLK3 | CLK | CMGC | 6ytw | B | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12410 | |
| CDK16 (PCTAIRE1) | CDK | CMGC | 3mtl | A | A | (2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime} | Human | 1701 | |
| CDK2 | CDK | CMGC | 3qxo | A | | 5-nitro-2-[(4-sulfamoylbenzyl)amino]benzamide | Human | 4282 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | C | A | - | Human | 4608 | |
| CDK1 (CDC2) | CDK | CMGC | 4yc6 | G | B | - | Human | 4615 | |
| CDK1 (CDC2) | CDK | CMGC | 5lqf | D | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 7365 | |
| CDK1 (CDC2) | CDK | CMGC | 5hq0 | A | A | {[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamide | Human | 6422 | |
| CDK1 (CDC2) | CDK | CMGC | 7nj0 | B | | - | Human | 13827 | |
| CLK4 | CLK | CMGC | 6fyv | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10510 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 4643 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2gmx | A | | n-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-bromo-2,5-dimethoxyphenyl)acetamide | Human | 4674 | |
| MAPK8 (JNK1) | MAPK | CMGC | 9ft9 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 15532 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vuh | A | | - | Human | 4663 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2g01 | B | | 6-chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4h-pyrazolo[3,4-b]quinolin-4-one | Human | 4641 | |
| MAPK8 (JNK1) | MAPK | CMGC | 12cv | A | A | (4m)-n-[3-(dimethylcarbamoyl)-4-hydroxyphenyl]-4-(1h-pyrrolo[2,3-b]pyridin-5-yl)-3h-1lambda~4~-benzothiophene-2-carboxamide | Human | 15533 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4qtd | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 4673 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4hyu | A | | trans-4-[(4-{4-[3-(methylsulfonyl)propoxy]-1h-indazol-1-yl}pyrimidin-2-yl)amino]cyclohexanol | Human | 4632 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4l7f | A | A | n-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamide | Human | 4639 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4e73 | A | A | methyl 3-(4-{[(1r,2s,3s,5s,7s)-5-aminotricyclo[3.3.1.1~3,7~]dec-2-yl]carbamoyl}benzyl)-4-oxo-1-phenyl-1,4-dihydro-1,8-naphthyridine-2-carboxylate | Human | 4645 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4ux9 | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 4635 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4izy | A | | trans-4-[(4-{4-[4-(methylsulfonyl)piperidin-1-yl]-1h-indol-1-yl}pyrimidin-2-yl)amino]cyclohexanol | Human | 4654 | |
| MAPK8 (JNK1) | MAPK | CMGC | 11zl | A | B | (4m)-n-[4-hydroxy-3-(pyrrolidine-1-carbonyl)phenyl]-4-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1-benzothiophene-2-carboxamide | Human | 15535 | |
| MAPK8 (JNK1) | MAPK | CMGC | 4yr8 | F | A | - | Human | 6450 | |
| MAPK8 (JNK1) | MAPK | CMGC | 2xrw | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 4650 | |
| MAPK8 (JNK1) | MAPK | CMGC | 12cv | A | B | (4m)-n-[3-(dimethylcarbamoyl)-4-hydroxyphenyl]-4-(1h-pyrrolo[2,3-b]pyridin-5-yl)-3h-1lambda~4~-benzothiophene-2-carboxamide | Human | 15536 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3vum | A | | - | Human | 4671 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3elj | A | A | 2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide | Human | 4658 | |
| MAPK8 (JNK1) | MAPK | CMGC | 3elj | A | B | 2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamide | Human | 4636 | |
| MAPK8 (JNK1) | MAPK | CMGC | 8x5m | A | A | 3-[4-(dimethylamino)butanoylamino]-~{n}-[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamide | Human | 15099 | |
| SRPK2 | SRPK | CMGC | 5myv | B | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7576 | |
| SRPK2 | SRPK | CMGC | 2x7g | A | | purvalanol b | Human | 1409 | |
| CLK1 | CLK | CMGC | 1z57 | A | B | debromohymenialdisine | Human | 105 | |
| CLK1 | CLK | CMGC | 7opg | A | A | 4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenol | Human | 13808 | |
| CLK1 | CLK | CMGC | 6yti | A | A | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 12413 | |
| CLK1 | CLK | CMGC | 5j1w | A | B | pyrido[3,4-g]quinazolin-2-amine | Human | 6576 | |
| CLK1 | CLK | CMGC | 6i5h | A | B | 5-(1-methylpyrazol-4-yl)-3-(3-phenoxyphenyl)furo[3,2-b]pyridine | Human | 10849 | |
| CLK1 | CLK | CMGC | 6yti | A | B | methyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidate | Human | 12414 | |
| CLK1 | CLK | CMGC | 6g33 | A | C | - | Human | 9826 | |
| CLK1 | CLK | CMGC | 5j1w | C | A | pyrido[3,4-g]quinazolin-2-amine | Human | 6578 | |
| CLK1 | CLK | CMGC | 6ytg | A | A | (4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrile | Human | 12416 | |
| CLK1 | CLK | CMGC | 6yta | A | B | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 12417 | |
| CLK1 | CLK | CMGC | 5x8i | A | | 5-[1-[(1s)-1-(4-fluorophenyl)ethyl]-[1,2,3]triazolo[4,5-c]quinolin-8-yl]-1,3-benzoxazole | Human | 8316 | |
| CLK1 | CLK | CMGC | 6z4z | C | A | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12309 | |
| CLK1 | CLK | CMGC | 6fyo | A | B | 6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamide | Human | 10323 | |
| CLK1 | CLK | CMGC | 6tw2 | E | A | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 11962 | |
| CLK1 | CLK | CMGC | 6i5l | A | B | 3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridine | Human | 10843 | |
| CLK1 | CLK | CMGC | 6q8p | C | | ~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amine | Human | 10901 | |
| CLK1 | CLK | CMGC | 6ytd | A | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12418 | |
| CLK1 | CLK | CMGC | 6yte | C | A | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12419 | |
| CLK1 | CLK | CMGC | 6g33 | A | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9824 | |
| CLK1 | CLK | CMGC | 6ft9 | C | B | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9900 | |
| CLK1 | CLK | CMGC | 6g33 | C | B | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9823 | |
| CLK1 | CLK | CMGC | 6g33 | A | A | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 9819 | |
| CLK1 | CLK | CMGC | 6z4z | A | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12312 | |
| CLK1 | CLK | CMGC | 2vag | A | A | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 104 | |
| CLK1 | CLK | CMGC | 6ytd | A | B | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 12420 | |
| CLK1 | CLK | CMGC | 6z4z | C | B | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12313 | |
| CLK1 | CLK | CMGC | 6g33 | B | C | - | Human | 9827 | |
| CLK1 | CLK | CMGC | 2vag | A | B | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 103 | |
| CLK1 | CLK | CMGC | 6yta | A | A | 1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanone | Human | 12423 | |
| CLK1 | CLK | CMGC | 6q8p | B | | ~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amine | Human | 10900 | |
| CLK1 | CLK | CMGC | 5j1w | A | A | pyrido[3,4-g]quinazolin-2-amine | Human | 6579 | |
| CLK1 | CLK | CMGC | 6ft9 | A | B | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9898 | |
| CLK1 | CLK | CMGC | 6ft9 | A | A | 2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9901 | |
| CLK1 | CLK | CMGC | 6qty | A | B | ethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylate | Human | 12084 | |
| CLK1 | CLK | CMGC | 5j1w | B | A | pyrido[3,4-g]quinazolin-2-amine | Human | 6575 | |
| CLK1 | CLK | CMGC | 6ft8 | A | B | 3-(3-hydroxyphenyl)-1~{h}-pyrrolo[3,4-g]indol-8-one | Human | 9899 | |
| CLK1 | CLK | CMGC | 7ak3 | A | B | ~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 13143 | |
| CLK1 | CLK | CMGC | 6raa | A | B | 4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamide | Human | 11013 | |
| CLK1 | CLK | CMGC | 6zln | A | A | 4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 12711 | |
| CDK12 (CRK7) | CDK | CMGC | 8buq | B | | (2~{r})-2-[[6-[[1-(3-chlorophenyl)pyrazol-3-yl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14917 | |
| CDK12 (CRK7) | CDK | CMGC | 6td3 | H | | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 12370 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu2 | B | | ~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-propan-2-yl-purin-6-amine | Human | 14918 | |
| CDK12 (CRK7) | CDK | CMGC | 5acb | C | | n-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamide | Human | 6701 | |
| CDK12 (CRK7) | CDK | CMGC | 6b3e | A | | 2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-ol | Human | 9452 | |
| CDK12 (CRK7) | CDK | CMGC | 8buf | B | | 2-(6,7-dihydro-4~{h}-thieno[3,2-c]pyridin-5-ylmethyl)-6,7-dimethoxy-3~{h}-quinazolin-4-one | Human | 14919 | |
| CDK12 (CRK7) | CDK | CMGC | 4un0 | C | | - | Human | 4854 | |
| CDK12 (CRK7) | CDK | CMGC | 9jk1 | A | | n-[5-[[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-[(phenylmethyl)carbamoyl]amino]-2-[4-(dimethylamino)piperidin-1-yl]phenyl]propanamide | Human | 15853 | |
| CDK12 (CRK7) | CDK | CMGC | 8bur | B | B | ~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamide | Human | 14920 | |
| CDK12 (CRK7) | CDK | CMGC | 6td3 | B | | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 12371 | |
| CDK12 (CRK7) | CDK | CMGC | 8buh | B | | 6-[[[2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-9-propan-2-yl-purin-6-yl]amino]methyl]-3-pyridin-2-yl-1~{h}-pyridin-2-one | Human | 14922 | |
| CDK12 (CRK7) | CDK | CMGC | 4cxa | C | | - | Human | 4853 | |
| CDK12 (CRK7) | CDK | CMGC | 8bup | B | | (2~{r})-2-[[6-[3-(3-methylphenyl)propylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14923 | |
| CDK12 (CRK7) | CDK | CMGC | 8bum | B | | (2r)-2-[[6-(5-naphthalen-1-ylpentylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14924 | |
| CDK12 (CRK7) | CDK | CMGC | 8bui | B | | (2~{r})-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)amino]purin-2-yl]amino]butan-1-ol | Human | 14925 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu5 | B | | ~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amine | Human | 14926 | |
| CDK12 (CRK7) | CDK | CMGC | 8buk | B | | (2~{r})-2-[[6-(naphthalen-2-ylmethylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14927 | |
| CDK12 (CRK7) | CDK | CMGC | 8bub | B | | ~{n}-(5-methyl-2,3-dihydro-1,3-thiazol-2-yl)-3-(5-methylfuran-2-yl)carbonyl-1,3-thiazolidine-4-carboxamide | Human | 14928 | |
| CDK12 (CRK7) | CDK | CMGC | 9x26 | A | B | (2s)-n-[2-[4-(dimethylamino)piperidin-1-yl]-5-[[(1s)-1-(4-fluorophenyl)ethyl]carbamoyl-[4-(quinazolin-2-ylamino)cyclohexyl]amino]pyridin-3-yl]-2-fluoranyl-propanamide | Human | 15855 | |
| CDK12 (CRK7) | CDK | CMGC | 8bud | B | | ~{n}-(5-bromanylpyridin-2-yl)-3-(4-oxidanylidenequinazolin-3-yl)propanamide | Human | 14929 | |
| CDK12 (CRK7) | CDK | CMGC | 9x26 | A | A | (2s)-n-[2-[4-(dimethylamino)piperidin-1-yl]-5-[[(1s)-1-(4-fluorophenyl)ethyl]carbamoyl-[4-(quinazolin-2-ylamino)cyclohexyl]amino]pyridin-3-yl]-2-fluoranyl-propanamide | Human | 15856 | |
| CDK12 (CRK7) | CDK | CMGC | 8p81 | A | B | ~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amine | Human | 15061 | |
| CDK12 (CRK7) | CDK | CMGC | 4nst | C | | adenosine-5'-diphosphate | Human | 4851 | |
| CDK12 (CRK7) | CDK | CMGC | 6ckx | C | | n-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamide | Human | 10579 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu1 | B | | (2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-ol | Human | 14930 | |
| CDK12 (CRK7) | CDK | CMGC | 6b3e | C | | 2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-ol | Human | 9453 | |
| CDK12 (CRK7) | CDK | CMGC | 4un0 | D | | - | Human | 4855 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu3 | B | | 2-morpholin-4-yl-9-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]purin-6-amine | Human | 14931 | |
| CDK12 (CRK7) | CDK | CMGC | 8bua | B | | (2~{r})-~{n}-(1~{h}-benzimidazol-2-yl)-2-(3-oxidanylidene-1~{h}-isoindol-2-yl)propanamide | Human | 14932 | |
| CDK12 (CRK7) | CDK | CMGC | 8buj | B | | (2~{r})-2-[[6-(octylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14933 | |
| CDK12 (CRK7) | CDK | CMGC | 8buo | B | | (2~{r})-2-[[6-[(3-fluoranyl-4-pyridin-2-yl-phenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14934 | |
| CDK12 (CRK7) | CDK | CMGC | 4cxa | A | | phosphoaminophosphonic acid-adenylate ester | Human | 4856 | |
| CDK12 (CRK7) | CDK | CMGC | 8bug | B | | 2-[2-[(6-methylpyridin-2-yl)amino]-1,3-thiazol-4-yl]-~{n}-(5-methyl-1,3-thiazol-2-yl)ethanamide | Human | 14935 | |
| CDK12 (CRK7) | CDK | CMGC | 8p81 | A | A | ~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amine | Human | 15062 | |
| CDK12 (CRK7) | CDK | CMGC | 8but | B | | 2-[[6-[[4-(2-hydroxyethyloxy)phenyl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14936 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | B | A | n-cyclohexyl-9h-purin-6-amine | Human | 6086 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv0 | A | A | n-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amine | Human | 2562 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aoh | A | A | ~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamide | Human | 14385 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhp | A | | 5-(2-methoxyethyl)-1-methyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydropyrrolo[3,2-c]pyridin-4-one | Human | 7998 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp1 | B | | n-benzyl-9h-purin-6-amine | Human | 6080 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7cml | B | B | - | Human | 12704 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6oph | A | | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 11509 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4h3q | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2611 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2ojj | A | | (s)-n-(1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamide | Human | 2612 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g97 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-one | Human | 9970 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr5 | A | A | (2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamide | Human | 13921 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | C | A | - | Human | 2569 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7s | A | A | - | Human | 11349 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | A | | adenosine-5'-diphosphate | Human | 2554 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qpa | A | | 7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6077 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz7 | C | B | - | Human | 2597 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fux | A | | trans-4-{[4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)pyrimidin-2-yl]amino}cyclohexanol | Human | 2568 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9m | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamide | Human | 9944 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaq | A | B | thiophen-3-ylmethylazanium | Human | 10989 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nr3 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13923 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g93 | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-one | Human | 9959 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | A | A | n-cyclohexyl-9h-purin-6-amine | Human | 6088 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5ngu | A | | 2-[2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-one | Human | 7991 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaq | A | A | thiophen-3-ylmethylazanium | Human | 10983 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7nqw | A | B | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-one | Human | 13924 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa3 | A | B | pyrazole | Human | 11345 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4n0s | A | A | caffeic acid | Human | 2589 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhh | A | | 5-(2-methoxyethyl)-2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7996 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzn | A | B | 2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamide | Human | 2610 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4o6e | A | A | n-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamide | Human | 2559 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | E | A | phosphoaminophosphonic acid-adenylate ester | Human | 2621 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g54 | A | B | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10937 | |
| MAPK1 (Erk2) | MAPK | CMGC | 7e73 | A | | - | Human | 14114 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdm | A | A | (3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamide | Human | 9968 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9m | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamide | Human | 9964 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv1 | A | A | n-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamide | Human | 2594 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9d | A | B | ~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamide | Human | 9953 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qag | A | A | 1~{h}-1,2,3-triazole | Human | 10988 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9k | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamide | Human | 9966 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp6 | A | | 5h-pyrrolo[2,3-b]pyrazine | Human | 6089 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fmq | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 2604 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2ojg | A | | n,n-dimethyl-4-(4-phenyl-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamide | Human | 2603 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g8x | A | B | 4-chloranyl-1~{h}-indazol-3-amine | Human | 9954 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9n | A | A | (2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamide | Human | 11410 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv3 | A | B | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 2580 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4xj0 | A | | 1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-one | Human | 6048 | |
| MAPK1 (Erk2) | MAPK | CMGC | 1pme | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 2583 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv2 | A | B | 4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamide | Human | 2571 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4h3p | A | | phosphoaminophosphonic acid-adenylate ester | Human | 2624 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aob | A | A | ~{n}-[(1-methylindazol-3-yl)methyl]propanamide | Human | 14402 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | C | A | - | Human | 2588 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa4 | A | A | 1~{h}-pyridin-2-one | Human | 11344 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 15300 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5buj | A | B | 4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-one | Human | 2561 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5ax3 | A | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 6398 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdm | A | B | (3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamide | Human | 9946 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6dmg | A | B | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 10810 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aog | A | A | ~{n}-(5-methyl-1,2-oxazol-3-yl)propanamide | Human | 14403 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv8 | A | B | 6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-one | Human | 2601 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3i60 | A | | 4-{2-[(2-chlorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-phenylethyl]-1h-pyrrole-2-carboxamide | Human | 2584 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv6 | A | | n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-4-(2-{[(2s)-1-hydroxybutan-2-yl]amino}-5-methylpyrimidin-4-yl)-1h-pyrrole-2-carboxamide | Human | 2551 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhv | A | | 7-[2-(oxan-4-ylamino)pyrimidin-4-yl]-3,4-dihydro-2~{h}-pyrrolo[1,2-a]pyrazin-1-one | Human | 7995 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qal | A | A | 1,1-bis(oxidanylidene)thietan-3-ol | Human | 10987 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv9 | A | A | 3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 2582 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | C | | adenosine-5'-diphosphate | Human | 2595 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g92 | A | A | ~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amine | Human | 11409 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3sa0 | A | B | norathyriol | Human | 2557 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lcj | A | B | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 6834 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v60 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 8263 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6opi | A | | (3r)-n-[3-(2-cyclopropylpyridin-4-yl)-1h-indazol-5-yl]-3-(methoxymethyl)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]-3,6-dihydropyridin-1(2h)-yl}ethyl)pyrrolidine-3-carboxamide | Human | 11511 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9k | A | B | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamide | Human | 9947 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2oji | A | | n-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamide | Human | 2570 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaw | A | B | [1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazanium | Human | 10986 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bvf | A | B | 2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-one | Human | 6027 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | A | B | n-cyclohexyl-9h-purin-6-amine | Human | 6075 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp8 | B | | 2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6076 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv2 | A | A | 4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamide | Human | 2592 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt0 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15307 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8aof | A | B | ~{n}-(2-methylpyrimidin-5-yl)propanamide | Human | 14408 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g9j | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamide | Human | 9952 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp3 | B | | (2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-ol | Human | 6079 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv7 | A | A | 4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrile | Human | 2572 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4nif | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 2566 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fuy | A | B | {4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanone | Human | 2587 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iza | A | A | - | Human | 2586 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp9 | A | | 7-(1-propyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6085 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qpa | B | | 7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazine | Human | 6090 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qte | A | A | 4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamide | Human | 2590 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8pt1 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 15309 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8psw | A | A | amp phosphoramidate | Human | 15310 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6dmg | A | C | ethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinate | Human | 10809 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa1 | A | B | pyridin-2-amine | Human | 11346 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv9 | A | B | 3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridine | Human | 2552 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp4 | B | B | n-cyclohexyl-9h-purin-6-amine | Human | 6083 | |
| MAPK1 (Erk2) | MAPK | CMGC | 8ao4 | A | A | ~{n}-(1~{h}-indazol-5-yl)ethanesulfonamide | Human | 14416 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g93 | A | A | 6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-one | Human | 9955 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp6 | B | | 5h-pyrrolo[2,3-b]pyrazine | Human | 6091 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhl | A | | (6~{r})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7992 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6d5y | A | | - | Human | 10939 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv4 | A | B | 9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrile | Human | 2558 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6q7s | A | B | - | Human | 11343 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g92 | A | B | ~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amine | Human | 11411 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp1 | A | | n-benzyl-9h-purin-6-amine | Human | 6092 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6ge0 | A | A | 2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamide | Human | 9950 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6rq4 | A | B | 6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-one | Human | 11855 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv7 | A | B | 4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrile | Human | 2614 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6nbs | A | B | - | Human | 11508 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qag | A | B | 1~{h}-1,2,3-triazole | Human | 10982 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4qp2 | A | | 5-chloro-1,3-benzoxazol-2-amine | Human | 6078 | |
| MAPK1 (Erk2) | MAPK | CMGC | 2y9q | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2556 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv1 | A | B | n-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamide | Human | 2613 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5lcj | A | A | [(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamate | Human | 6833 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5nhj | A | | 5-(2-methoxyethyl)-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-one | Human | 7994 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4iz5 | B | | adenosine-5'-diphosphate | Human | 2600 | |
| MAPK1 (Erk2) | MAPK | CMGC | 3sa0 | A | A | norathyriol | Human | 2596 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qah | A | A | 1-azanylpropylideneazanium | Human | 11354 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qaw | A | A | [1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazanium | Human | 10984 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5bui | A | | 3-(4-fluorophenyl)-5-(pyridin-2-yl)-4,5,6,7-tetrahydro-2h-pyrazolo[4,3-c]pyridine | Human | 2563 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjd | A | B | cyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamate | Human | 10830 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzo | A | A | n-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 2620 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4o6e | A | B | n-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamide | Human | 2553 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a1b | A | B | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13144 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a1z | A | A | 6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13145 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcd | A | B | 4,5,6,7-tetrabromobenzotriazole | Human | 15019 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5m4u | A | B | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7391 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6tew | A | A | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12443 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6hmc | A | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 10996 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6qy8 | C | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12115 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ywm | X | | nicotinic acid | Human | 10759 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8qcd | A | A | 4,5,6,7-tetrabromobenzotriazole | Human | 15023 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 3ofm | A | A | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 2728 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6l20 | J | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 11994 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5yf9 | B | B | nicotinic acid | Human | 11416 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6tew | A | B | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12447 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a22 | A | A | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13148 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ooi | A | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9446 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ooi | B | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9445 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a1b | A | A | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13149 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a2h | A | A | 5,6,7-tris(bromanyl)-1~{h}-imidazo[4,5-b]pyridine | Human | 13150 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7xyh | A | | 5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrile | Human | 14587 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 6tgu | A | A | 4-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxidanyl-benzoic acid | Human | 12448 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7at9 | A | A | 3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-ol | Human | 13832 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5y9m | X | | nicotinic acid | Human | 9909 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 7a22 | A | B | 5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13151 | |
| MAPK13 (p38d) | MAPK | CMGC | 4myg | A | | - | Human | 2951 | |
| MAPK13 (p38d) | MAPK | CMGC | 4myg | B | | - | Human | 2950 | |
| MAPK13 (p38d) | MAPK | CMGC | 8x23 | A | A | - | Human | 15129 | |
| MAPK13 (p38d) | MAPK | CMGC | 5eko | A | | 3-(4-methyl-1h-imidazol-1-yl)-n-[4-(pyridin-4-yloxy)phenyl]benzamide | Human | 6746 | |
| MAPK13 (p38d) | MAPK | CMGC | 3coi | A | A | - | Human | 2948 | |
| MAPK13 (p38d) | MAPK | CMGC | 4eyj | A | | 1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-yloxy)phenyl]urea | Human | 2949 | |
| MAPK13 (p38d) | MAPK | CMGC | 5ekn | A | | 1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-ylsulfanyl)phenyl]urea | Human | 6745 | |
| MAPK13 (p38d) | MAPK | CMGC | 4eym | A | | 2-(morpholin-4-yl)-n-[4-(pyridin-4-yloxy)phenyl]pyridine-4-carboxamide | Human | 2945 | |
| MAPK13 (p38d) | MAPK | CMGC | 3coi | A | B | - | Human | 2946 | |
| CDK4 | CDK | CMGC | 5fwm | K | | - | Human | 6749 | |
| CDK4 | CDK | CMGC | 5fwk | K | | - | Human | 6747 | |
| CDK4 | CDK | CMGC | 6p8f | B | | - | Human | 11892 | |
| CDK4 | CDK | CMGC | 3g33 | C | | - | Human | 3384 | |
| CDK4 | CDK | CMGC | 6p8e | B | | - | Human | 11891 | |
| CDK4 | CDK | CMGC | 2w9z | B | B | - | Human | 3383 | |
| DYRK1A | DYRK | CMGC | 3anr | B | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 3729 | |
| DYRK1A | DYRK | CMGC | 5a4e | D | B | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6733 | |
| DYRK1A | DYRK | CMGC | 6a1f | A | B | 8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amine | Human | 10521 | |
| DYRK1A | DYRK | CMGC | 6s1j | A | A | 3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazine | Human | 11365 | |
| DYRK1A | DYRK | CMGC | 6s11 | B | B | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11372 | |
| DYRK1A | DYRK | CMGC | 6t6a | A | A | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11857 | |
| DYRK1A | DYRK | CMGC | 6eiq | B | | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | 10529 | |
| DYRK1A | DYRK | CMGC | 6eif | D | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10532 | |
| DYRK1A | DYRK | CMGC | 7a53 | A | B | (3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-one | Human | 13741 | |
| DYRK1A | DYRK | CMGC | 7a5d | A | A | 4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrile | Human | 13742 | |
| DYRK1A | DYRK | CMGC | 6ej4 | D | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10545 | |
| DYRK1A | DYRK | CMGC | 4nct | A | | pkc412 | Human | 3794 | |
| DYRK1A | DYRK | CMGC | 5a3x | A | | n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6723 | |
| DYRK1A | DYRK | CMGC | 7zh8 | A | B | 6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridine | Human | 14488 | |
| DYRK1A | DYRK | CMGC | 6yf8 | D | | ~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamide | Human | 13460 | |
| DYRK1A | DYRK | CMGC | 4mq1 | A | A | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3796 | |
| DYRK1A | DYRK | CMGC | 5a4t | A | | n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide | Human | 6732 | |
| DYRK1A | DYRK | CMGC | 7zh8 | A | A | 6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridine | Human | 14489 | |
| DYRK1A | DYRK | CMGC | 4mq1 | D | B | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3763 | |
| DYRK1A | DYRK | CMGC | 6s1i | C | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11373 | |
| DYRK1A | DYRK | CMGC | 7a4r | A | B | 2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-one | Human | 13743 | |
| DYRK1A | DYRK | CMGC | 5a4e | D | A | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6714 | |
| DYRK1A | DYRK | CMGC | 5aik | D | | 4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine | Human | 3742 | |
| DYRK1A | DYRK | CMGC | 7o7k | A | B | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 13987 | |
| DYRK1A | DYRK | CMGC | 5a3x | C | | n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6722 | |
| DYRK1A | DYRK | CMGC | 4ylj | B | B | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3785 | |
| DYRK1A | DYRK | CMGC | 6a1g | B | | 5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amine | Human | 10539 | |
| DYRK1A | DYRK | CMGC | 5a4l | B | A | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6719 | |
| DYRK1A | DYRK | CMGC | 4mq2 | C | A | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3730 | |
| DYRK1A | DYRK | CMGC | 4aze | C | | 5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-one | Human | 3788 | |
| DYRK1A | DYRK | CMGC | 5aik | A | | 4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine | Human | 3732 | |
| DYRK1A | DYRK | CMGC | 6eis | A | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10553 | |
| DYRK1A | DYRK | CMGC | 6eiv | A | | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10540 | |
| DYRK1A | DYRK | CMGC | 4mq1 | D | A | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3744 | |
| DYRK1A | DYRK | CMGC | 6uwy | D | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11988 | |
| DYRK1A | DYRK | CMGC | 5a4l | D | B | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6730 | |
| DYRK1A | DYRK | CMGC | 6uwy | B | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11982 | |
| DYRK1A | DYRK | CMGC | 6s1j | A | B | 3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazine | Human | 11360 | |
| DYRK1A | DYRK | CMGC | 6t6a | C | B | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11859 | |
| DYRK1A | DYRK | CMGC | 6qu2 | D | A | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12091 | |
| DYRK1A | DYRK | CMGC | 6uip | B | | 4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide | Human | 12025 | |
| DYRK1A | DYRK | CMGC | 6eir | C | | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10528 | |
| DYRK1A | DYRK | CMGC | 6t6a | C | A | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11863 | |
| DYRK1A | DYRK | CMGC | 4mq1 | C | B | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3750 | |
| DYRK1A | DYRK | CMGC | 2vx3 | A | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3762 | |
| DYRK1A | DYRK | CMGC | 7ajv | A | | 4-(2,3-dibutylimidazo[4,5-b]pyridin-5-yl)pyridine-2,6-diamine | Human | 13594 | |
| DYRK1A | DYRK | CMGC | 7a55 | A | | 3-(1-methylpyrazol-4-yl)-1~{h}-pyrazole-5-carboxylic acid | Human | 13746 | |
| DYRK1A | DYRK | CMGC | 6eil | A | | [3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone | Human | 10546 | |
| DYRK1A | DYRK | CMGC | 6eiq | A | | [4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanone | Human | 10554 | |
| DYRK1A | DYRK | CMGC | 6eil | C | | - | Human | 10552 | |
| DYRK1A | DYRK | CMGC | 7a5l | A | A | 4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amine | Human | 13747 | |
| DYRK1A | DYRK | CMGC | 3anq | D | | (1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one | Human | 3795 | |
| DYRK1A | DYRK | CMGC | 3anr | A | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 3778 | |
| DYRK1A | DYRK | CMGC | 6eis | A | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10526 | |
| DYRK1A | DYRK | CMGC | 6eil | B | | [3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone | Human | 10557 | |
| DYRK1A | DYRK | CMGC | 5a54 | A | | n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide | Human | 6736 | |
| DYRK1A | DYRK | CMGC | 6uwy | B | A | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11983 | |
| DYRK1A | DYRK | CMGC | 5a4l | A | B | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6728 | |
| DYRK1A | DYRK | CMGC | 5a4e | B | A | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6713 | |
| DYRK1A | DYRK | CMGC | 6eis | C | A | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10535 | |
| DYRK1A | DYRK | CMGC | 7aka | A | A | 4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13596 | |
| DYRK1A | DYRK | CMGC | 4ylk | A | B | 10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3756 | |
| DYRK1A | DYRK | CMGC | 3anr | D | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 3755 | |
| DYRK1A | DYRK | CMGC | 6s11 | B | A | 6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazine | Human | 11378 | |
| DYRK1A | DYRK | CMGC | 5a4q | C | | n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6738 | |
| DYRK1A | DYRK | CMGC | 4nct | C | | pkc412 | Human | 3779 | |
| DYRK1A | DYRK | CMGC | 6qu2 | A | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12092 | |
| DYRK1A | DYRK | CMGC | 4yll | A | A | 10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3747 | |
| DYRK1A | DYRK | CMGC | 4mq1 | B | A | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3773 | |
| DYRK1A | DYRK | CMGC | 6s1i | D | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11362 | |
| DYRK1A | DYRK | CMGC | 4yu2 | C | A | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3741 | |
| DYRK1A | DYRK | CMGC | 6ej4 | A | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10520 | |
| DYRK1A | DYRK | CMGC | 3anr | C | | 7-methoxy-1-methyl-9h-beta-carboline | Human | 3783 | |
| DYRK1A | DYRK | CMGC | 6s1i | D | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11379 | |
| DYRK1A | DYRK | CMGC | 6s17 | A | B | ~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11375 | |
| DYRK1A | DYRK | CMGC | 6s1i | C | A | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11366 | |
| DYRK1A | DYRK | CMGC | 7a52 | A | A | 3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-one | Human | 13748 | |
| DYRK1A | DYRK | CMGC | 2vx3 | A | A | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3776 | |
| DYRK1A | DYRK | CMGC | 6eil | D | | [3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanone | Human | 10551 | |
| DYRK1A | DYRK | CMGC | 7a4s | A | | 7-chlorothieno[3,2-c]pyridin-4-amine | Human | 13749 | |
| DYRK1A | DYRK | CMGC | 7aj7 | A | | 4-(3-methylbenzimidazol-5-yl)pyridine-2,6-diamine | Human | 13600 | |
| DYRK1A | DYRK | CMGC | 6s1h | A | A | ~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 11419 | |
| DYRK1A | DYRK | CMGC | 6eir | B | | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10558 | |
| DYRK1A | DYRK | CMGC | 6eis | B | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10537 | |
| DYRK1A | DYRK | CMGC | 5a4q | B | | n-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6729 | |
| DYRK1A | DYRK | CMGC | 6t6a | D | B | - | Human | 11856 | |
| DYRK1A | DYRK | CMGC | 6eiv | D | | ~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10527 | |
| DYRK1A | DYRK | CMGC | 6eis | D | B | 1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-one | Human | 10543 | |
| DYRK1A | DYRK | CMGC | 6eir | A | | ~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamide | Human | 10550 | |
| DYRK1A | DYRK | CMGC | 4yu2 | A | A | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3774 | |
| DYRK1A | DYRK | CMGC | 4ylj | A | A | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3782 | |
| DYRK1A | DYRK | CMGC | 7z5n | A | | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 14667 | |
| DYRK1A | DYRK | CMGC | 4mq2 | A | B | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3771 | |
| DYRK1A | DYRK | CMGC | 6uip | C | | 4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide | Human | 12026 | |
| DYRK1A | DYRK | CMGC | 5a3x | D | | n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6718 | |
| DYRK1A | DYRK | CMGC | 4mq2 | B | A | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3792 | |
| DYRK1A | DYRK | CMGC | 4mq1 | B | B | n-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamide | Human | 3770 | |
| DYRK1A | DYRK | CMGC | 2vx3 | D | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3790 | |
| DYRK1A | DYRK | CMGC | 4ylj | A | B | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3746 | |
| DYRK1A | DYRK | CMGC | 2vx3 | B | B | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 3769 | |
| DYRK1A | DYRK | CMGC | 6eif | A | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10534 | |
| DYRK1A | DYRK | CMGC | 6s1h | A | B | ~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amine | Human | 11420 | |
| DYRK1A | DYRK | CMGC | 7a4r | A | A | 2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-one | Human | 13751 | |
| DYRK1A | DYRK | CMGC | 5a4l | C | B | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6711 | |
| DYRK1A | DYRK | CMGC | 6qu2 | C | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12087 | |
| DYRK1A | DYRK | CMGC | 6uip | A | | 4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamide | Human | 12027 | |
| DYRK1A | DYRK | CMGC | 5a54 | D | | n-(6-nitro-1,3-benzothiazol-2-yl)ethanamide | Human | 6710 | |
| DYRK1A | DYRK | CMGC | 5a4l | A | A | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6731 | |
| DYRK1A | DYRK | CMGC | 4mq2 | D | B | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3734 | |
| DYRK1A | DYRK | CMGC | 4nct | B | | pkc412 | Human | 3743 | |
| DYRK1A | DYRK | CMGC | 6eij | C | | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | 10538 | |
| DYRK1A | DYRK | CMGC | 6qu2 | B | B | 8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-one | Human | 12088 | |
| DYRK1A | DYRK | CMGC | 7ajy | A | | 4-[2-methyl-3-[(2~{r})-2-phenoxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13606 | |
| DYRK1A | DYRK | CMGC | 5a4t | B | | n-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamide | Human | 6715 | |
| DYRK1A | DYRK | CMGC | 5a3x | B | | n-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6724 | |
| DYRK1A | DYRK | CMGC | 7akb | A | A | 4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamine | Human | 13608 | |
| DYRK1A | DYRK | CMGC | 6s1i | B | B | ~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11367 | |
| DYRK1A | DYRK | CMGC | 7a4z | A | | 3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amine | Human | 13752 | |
| DYRK1A | DYRK | CMGC | 7a4w | A | | 6-(4-methoxyphenyl)pyrimidine-2,4-diamine | Human | 13754 | |
| DYRK1A | DYRK | CMGC | 4mq2 | B | B | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3787 | |
| DYRK1A | DYRK | CMGC | 5aik | C | | 4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amine | Human | 3754 | |
| DYRK1A | DYRK | CMGC | 6t6a | B | B | 4-chloranyl-5~{h}-cyclohepta[b]indol-10-one | Human | 11861 | |
| DYRK1A | DYRK | CMGC | 4yll | A | B | 10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3772 | |
| DYRK1A | DYRK | CMGC | 4yu2 | D | A | (1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrile | Human | 3760 | |
| DYRK1A | DYRK | CMGC | 6a1f | A | A | 8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amine | Human | 10522 | |
| DYRK1A | DYRK | CMGC | 6ej4 | B | | 3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)aniline | Human | 10523 | |
| DYRK1A | DYRK | CMGC | 5a4l | D | A | n-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamide | Human | 6739 | |
| DYRK1A | DYRK | CMGC | 6uwy | A | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11987 | |
| DYRK1A | DYRK | CMGC | 4mq2 | A | A | methyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoate | Human | 3752 | |
| DYRK1A | DYRK | CMGC | 7o7k | A | A | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 13988 | |
| DYRK1A | DYRK | CMGC | 3anq | B | | (1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-one | Human | 3745 | |
| DYRK1A | DYRK | CMGC | 6eif | C | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10525 | |
| DYRK1A | DYRK | CMGC | 6eij | A | | ~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamide | Human | 10518 | |
| DYRK1A | DYRK | CMGC | 4ylj | D | A | 10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acid | Human | 3784 | |
| DYRK1A | DYRK | CMGC | 5a4e | C | B | n-(5-methoxy-1,3-benzothiazol-2-yl)ethanamide | Human | 6727 | |
| DYRK1A | DYRK | CMGC | 6s14 | A | B | ~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amine | Human | 11421 | |
| DYRK1A | DYRK | CMGC | 7fht | A | A | (5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one | Human | 14161 | |
| DYRK1A | DYRK | CMGC | 6eif | B | | 4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamide | Human | 10544 | |
| DYRK1A | DYRK | CMGC | 6uwy | D | B | 4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamide | Human | 11986 | |
| DYRK1A | DYRK | CMGC | 7a5l | A | B | 4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amine | Human | 13758 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3v6r | B | A | 4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamide | Human | 3427 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2o2u | A | | n-(3-cyano-4,5,6,7-tetrahydro-1-benzothien-2-yl)-2-fluorobenzamide | Human | 3457 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3g90 | X | | (3e)-5-fluoro-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-1h-indole-2,3-dione 3-oxime | Human | 3477 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | A | B | phosphomethylphosphonic acid adenylate ester | Human | 10509 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3fv8 | A | B | 5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamide | Human | 3426 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3da6 | A | | n-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)naphthalen-1-yl]-1h-benzimidazol-2-amine | Human | 3476 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | B | B | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10501 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8vs0 | A | | (4p)-4-[6-fluoro-5-(2-methoxyanilino)-1h-indazol-1-yl]-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 15635 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2r9s | A | | n-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamide | Human | 3450 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h39 | A | A | - | Human | 3460 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4kkg | A | | - | Human | 3443 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3cgo | A | | 2-{4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidin-1-yl}-n-methylacetamide | Human | 6771 | |
| MAPK10 (JNK3) | MAPK | CMGC | 8vtf | A | | (4p)-4-[6-fluoro-5-(2-methoxyanilino)-1h-indazol-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 15636 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3oy1 | A | | 5-[2-(cyclohexylamino)pyridin-4-yl]-4-naphthalen-2-yl-2-(tetrahydro-2h-pyran-4-yl)-2,4-dihydro-3h-1,2,4-triazol-3-one | Human | 3469 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | C | A | - | Human | 3475 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ore | A | B | 4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamide | Human | 13810 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6ekd | A | B | 4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10502 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4y46 | A | | 1-{trans-4-[(8-cyclopentyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]cyclohexyl}-3-propan-2-ylurea | Human | 3414 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ore | A | A | 4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamide | Human | 13811 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2b1p | A | | 3-{6-[(2-chlorophenyl)amino]-1h-indazol-3-yl}-5-{[4-(dimethylamino)butanoyl]amino}benzoic acid | Human | 3464 | |
| MAPK10 (JNK3) | MAPK | CMGC | 1pmu | A | | 9-(4-hydroxyphenyl)-2,7-phenanthroline | Human | 3474 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4h3b | A | A | - | Human | 3480 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4z9l | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 3432 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7orf | A | A | n-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamide | Human | 13812 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6emh | A | A | 4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10508 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3ttj | A | B | 9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamine | Human | 3428 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2r9s | B | | n-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamide | Human | 3420 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ksi | A | | 4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13387 | |
| MAPK10 (JNK3) | MAPK | CMGC | 1jnk | A | | phosphoaminophosphonic acid-adenylate ester | Human | 3451 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6eq9 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 10500 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3g9n | A | | (3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-phenyl-1h-indole-2,3-dione 3-oxime | Human | 3416 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ore | A | C | 4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamide | Human | 13813 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4kkh | A | | cyclopropyl[(3r)-3-({4-[6-hydroxy-2-(naphthalen-2-yl)-1h-benzimidazol-1-yl]pyrimidin-2-yl}amino)piperidin-1-yl]methanone | Human | 3419 | |
| MAPK10 (JNK3) | MAPK | CMGC | 3ptg | A | | n-[4-methyl-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamide | Human | 3470 | |
| MAPK10 (JNK3) | MAPK | CMGC | 7ksj | A | | 4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamide | Human | 13388 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2waj | A | B | 1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinoline | Human | 3471 | |
| MAPK10 (JNK3) | MAPK | CMGC | 2ok1 | A | B | n-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamide | Human | 3473 | |
| MAPK10 (JNK3) | MAPK | CMGC | 4w4y | A | | 3-(4-{[(4-methylphenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamide | Human | 3447 | |
| MAPK10 (JNK3) | MAPK | CMGC | 6ekd | A | A | 4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amine | Human | 10498 | |
| SRPK1 | SRPK | CMGC | 4wua | A | A | n-[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamide | Human | 9471 | |
| SRPK1 | SRPK | CMGC | 6fad | B | | - | Human | 11640 | |
| SRPK1 | SRPK | CMGC | 4wua | A | B | n-[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamide | Human | 9469 | |
| SRPK1 | SRPK | CMGC | 6fad | C | | - | Human | 11639 | |
| SRPK1 | SRPK | CMGC | 5my8 | A | A | sphinx31 | Human | 9466 | |
| SRPK1 | SRPK | CMGC | 5my8 | A | B | sphinx31 | Human | 9468 | |
| SRPK1 | SRPK | CMGC | 7zks | A | A | n-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamide | Human | 14619 | |
| SRPK1 | SRPK | CMGC | 5mxx | A | A | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 9470 | |
| SRPK1 | SRPK | CMGC | 7dd1 | A | | - | Human | 13510 | |
| SRPK1 | SRPK | CMGC | 5mxx | A | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 9467 | |
| GSK3A | GSK | CMGC | 7sxf | A | B | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 14780 | |
| GSK3A | GSK | CMGC | 7sxf | A | A | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 14781 | |
| GSK3A | GSK | CMGC | 7sxg | A | B | (4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-ol | Human | 14782 | |
| GSK3A | GSK | CMGC | 7sxg | A | A | (4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-ol | Human | 14783 | |
| CDKL3 | CDKL | CMGC | 3zdu | A | | [4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrile | Human | 4677 | |
| CDKL1 | CDKL | CMGC | 4agu | A | | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 761 | |
| CDKL1 | CDKL | CMGC | 4agu | B | | n-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamide | Human | 760 | |
| MAPK14 (p38a) | MAPK | CMGC | 4r3c | A | A | 6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine | Human | 5198 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ctq | A | | n-benzyl-1-[5-({5-tert-butyl-2-methoxy-3-[(methylsulfonyl)amino]phenyl}carbamoyl)-2-methylphenyl]-1h-1,2,3-triazole-4-carboxamide | Human | 5220 | |
| MAPK14 (p38a) | MAPK | CMGC | 5tco | A | | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulene-9-carboxamide | Human | 8031 | |
| MAPK14 (p38a) | MAPK | CMGC | 2gfs | A | B | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | 5050 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5203 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnv | A | A | 1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylurea | Human | 5037 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | A | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5074 | |
| MAPK14 (p38a) | MAPK | CMGC | 4dli | A | | - | Human | 5092 | |
| MAPK14 (p38a) | MAPK | CMGC | 2y8o | A | A | - | Human | 5079 | |
| MAPK14 (p38a) | MAPK | CMGC | 3oef | X | B | - | Human | 5231 | |
| MAPK14 (p38a) | MAPK | CMGC | 5tbe | A | | ~{n}-[2,4-bis(fluoranyl)-5-[[9-(2-morpholin-4-ylethylcarbamoyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulen-3-yl]amino]phenyl]thiophene-2-carboxamide | Human | 8032 | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3j | A | | 2-(4-fluorophenyl)-3-oxo-6-pyridin-4-yl-n-[2-(trifluoromethyl)benzyl]-2,3-dihydropyridazine-4-carboxamide | Human | 5047 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | C | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | 11618 | |
| MAPK14 (p38a) | MAPK | CMGC | 5omg | A | A | 3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | 11246 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hrb | A | | [3-amino-2-(2-methylphenyl)-1-oxidopyridin-4-yl](2,4-difluorophenyl)methanone | Human | 5202 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w84 | A | | 3-(2-pyridin-4-ylethyl)-1h-indole | Human | 5065 | |
| MAPK14 (p38a) | MAPK | CMGC | 2gfs | A | A | [5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanone | Human | 5227 | |
| MAPK14 (p38a) | MAPK | CMGC | 3u8w | A | | 3-[3-(2-chloro-6-fluorophenyl)-5-ethyl-6-oxo-5,6-dihydro[1,2,4]triazolo[4,3-b]pyridazin-7-yl]-n-cyclopropyl-4-methylbenzamide | Human | 5192 | |
| MAPK14 (p38a) | MAPK | CMGC | 3huc | A | A | n-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamide | Human | 5027 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | A | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5141 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbt | A | | 3-fluoro-5-morpholin-4-yl-n-[1-(2-pyridin-4-ylethyl)-1h-indol-6-yl]benzamide | Human | 5082 | |
| MAPK14 (p38a) | MAPK | CMGC | 3k3i | A | B | (3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinoline | Human | 5022 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | B | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | 5138 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mtx | A | B | 3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamide | Human | 8379 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfi | A | A | ~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamide | Human | 11613 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfo | A | B | 5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 11621 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w83 | A | | n-[4-chloro-3-(pyridin-3-yloxymethyl)-phenyl]-3-fluoro- | Human | 4986 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mty | A | | ~{n}-[2,4-bis(fluoranyl)-5-[[14-(2-hydroxyethylcarbamoyl)-2-oxidanylidene-6-tricyclo[9.4.0.0^{3,8}]pentadeca-1(15),3(8),4,6,11,13-hexaenyl]amino]phenyl]thiophene-2-carboxamide | Human | 8383 | |
| MAPK14 (p38a) | MAPK | CMGC | 5o8v | A | | - | Human | 8380 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfb | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)urea | Human | 5001 | |
| MAPK14 (p38a) | MAPK | CMGC | 5etf | A | A | - | Human | 7134 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fsf | A | | 3-(2,6-dichlorophenyl)-7-({4-[(diethylamino)methoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-one | Human | 5097 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fmk | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5209 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvq | A | A | n-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamide | Human | 5183 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh9 | A | | - | Human | 4982 | |
| MAPK14 (p38a) | MAPK | CMGC | 1bl6 | A | | 4-(4-fluorophenyl)-1-cycloropropylmethyl-5-(4-pyridyl)-imidazole | Human | 5243 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | D | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12486 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfk | A | B | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamide | Human | 11620 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iph | A | B | 6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamide | Human | 5156 | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | 5122 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fls | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5119 | |
| MAPK14 (p38a) | MAPK | CMGC | 3que | A | | 2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-one | Human | 5095 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwt | A | B | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamide | Human | 11254 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | B | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | 5059 | |
| MAPK14 (p38a) | MAPK | CMGC | 4kiq | C | | ethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylate | Human | 5215 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mh3 | A | | - | Human | 5109 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsg | A | B | tak-715 | Human | 5098 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | B | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | 11616 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qyx | A | | - | Human | 12127 | |
| MAPK14 (p38a) | MAPK | CMGC | 3flz | A | | 8-methyl-6-phenoxy-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5204 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hub | A | | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | 5029 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwv | A | A | - | Human | 11253 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 2 | - | Human | 5093 | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | A | - | Human | 5025 | |
| MAPK14 (p38a) | MAPK | CMGC | 3qud | A | B | {4-[(2-aminophenyl)amino]phenyl}(phenyl)methanone | Human | 5262 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gc7 | A | A | 5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-one | Human | 5061 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh3 | A | | naringenin | Human | 5042 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | 6880 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwu | A | A | - | Human | 11247 | |
| MAPK14 (p38a) | MAPK | CMGC | 5mz3 | A | A | ~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamide | Human | 8680 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh2 | A | | 3-phenylquinazolin-4(3h)-one | Human | 5244 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fsl | X | | - | Human | 5264 | |
| MAPK14 (p38a) | MAPK | CMGC | 2onl | A | | - | Human | 5177 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ha8 | A | B | n~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamide | Human | 5187 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvm | B | | 4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5210 | |
| MAPK14 (p38a) | MAPK | CMGC | 3itz | A | | 4-chloro-n-cyclopropyl-3-{[1-(2,6-difluorophenyl)-1h-pyrazolo[3,4-d]pyridazin-4-yl]amino}benzamide | Human | 5135 | |
| MAPK14 (p38a) | MAPK | CMGC | 3kq7 | A | B | n-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamide | Human | 5057 | |
| MAPK14 (p38a) | MAPK | CMGC | 6qe1 | A | | 1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{r})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]urea | Human | 11957 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvp | A | A | n-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamide | Human | 5070 | |
| MAPK14 (p38a) | MAPK | CMGC | 3new | A | B | - | Human | 5248 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv4 | A | | 1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5121 | |
| MAPK14 (p38a) | MAPK | CMGC | 3bx5 | A | | n-[2-methyl-5-(methylcarbamoyl)phenyl]-2-{[(1r)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamide | Human | 5000 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnw | A | A | 2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamide | Human | 5139 | |
| MAPK14 (p38a) | MAPK | CMGC | 2fst | X | A | - | Human | 5080 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | B | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12488 | |
| MAPK14 (p38a) | MAPK | CMGC | 1kv1 | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5252 | |
| MAPK14 (p38a) | MAPK | CMGC | 2i0h | A | B | 2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dione | Human | 5009 | |
| MAPK14 (p38a) | MAPK | CMGC | 3pg3 | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}urea | Human | 5096 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa4 | A | | n-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]furan-3-carboxamide | Human | 5045 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbs | A | | 3-fluoro-5-morpholin-4-yl-n-[3-(2-pyridin-4-ylethyl)-1h-indol-5-yl]benzamide | Human | 5258 | |
| MAPK14 (p38a) | MAPK | CMGC | 1m7q | A | | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2(1h)-one | Human | 5128 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e6a | A | | - | Human | 5238 | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv3 | A | | 5-methyl-4-[(2-methyl-5-{[(3-morpholin-4-ylphenyl)carbonyl]amino}phenyl)amino]-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5207 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | F | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12490 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hec | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 5166 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lff | A | A | (4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acid | Human | 5140 | |
| MAPK14 (p38a) | MAPK | CMGC | 5eti | A | | - | Human | 6362 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | B | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12491 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w82 | A | | n-[(3z)-5-tert-butyl-2-phenyl-1,2-dihydro-3h-pyrazol-3-ylidene]-n'-(4-chlorophenyl)urea | Human | 5165 | |
| MAPK14 (p38a) | MAPK | CMGC | 4geo | A | | - | Human | 5190 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | D | B | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12492 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcs | A | A | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5077 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw7 | A | | 2-({4-[(4-benzylpiperidin-1-yl)carbonyl]benzyl}sulfanyl)-3h-imidazo[4,5-c]pyridine | Human | 5084 | |
| MAPK14 (p38a) | MAPK | CMGC | 3d7z | A | B | n~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamide | Human | 5108 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfo | A | A | 5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamide | Human | 11615 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zaz | A | A | 4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehyde | Human | 4980 | |
| MAPK14 (p38a) | MAPK | CMGC | 1r39 | A | | - | Human | 5116 | |
| MAPK14 (p38a) | MAPK | CMGC | 5omg | A | B | 3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxide | Human | 11245 | |
| MAPK14 (p38a) | MAPK | CMGC | 1a9u | A | | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5229 | |
| MAPK14 (p38a) | MAPK | CMGC | 3flq | A | | 6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 5168 | |
| MAPK14 (p38a) | MAPK | CMGC | 3uvr | A | B | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}urea | Human | 6879 | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8t | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5167 | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8p | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5071 | |
| MAPK14 (p38a) | MAPK | CMGC | 2yis | A | | 1-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1h-pyrazol-5-yl]-3-{2-[(3-{2-[(2-hydroxyethyl)sulfanyl]phenyl}[1,2,4]triazolo[4,3-a]pyridin-6-yl)sulfanyl]benzyl}urea | Human | 5240 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | B | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | 5154 | |
| MAPK14 (p38a) | MAPK | CMGC | 2qd9 | A | | 1-[(3ar)-5-{[3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8h)-yl]carbonyl}-6-methoxy-3ah-pyrrolo[2,3-b]pyridin-3-yl]-2-[(3r)-3-hydroxypyrrolidin-1-yl]-2-oxoethanone | Human | 5197 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mvl | B | | 4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5091 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | A | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | 5178 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iph | A | A | 6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamide | Human | 4999 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwt | A | A | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamide | Human | 11248 | |
| MAPK14 (p38a) | MAPK | CMGC | 3l8s | A | | 3-[(4-bromo-2,6-difluorobenzyl)oxy]-5-{[(4-pyrrolidin-1-ylbutyl)carbamoyl]amino}isothiazole-4-carboxamide | Human | 5055 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9w | A | B | n,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5106 | |
| MAPK14 (p38a) | MAPK | CMGC | 6tca | H | A | n-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamide | Human | 12493 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fi4 | A | | (2s)-1-{[3-(2-chlorophenyl)-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-ol | Human | 5051 | |
| MAPK14 (p38a) | MAPK | CMGC | 3o8u | A | | 1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-urea | Human | 5250 | |
| MAPK14 (p38a) | MAPK | CMGC | 3s3i | A | | 3-(3-tert-butyl[1,2,4]triazolo[4,3-a]pyridin-7-yl)-n-cyclopropyl-4-methylbenzamide | Human | 5169 | |
| MAPK14 (p38a) | MAPK | CMGC | 3dt1 | A | | n-cyclopropyl-4-methyl-3-{2-[(2-morpholin-4-ylethyl)amino]quinazolin-6-yl}benzamide | Human | 5086 | |
| MAPK14 (p38a) | MAPK | CMGC | 3lfd | A | | 1-{4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5102 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcv | A | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5174 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ouy | A | | 1-(2,6-dichlorophenyl)-6-[(2,4-difluorophenyl)sulfanyl]-7-(1,2,3,6-tetrahydro-4-pyridinyl)-3,4-dihydropyrido[3,2-d]pyrimidin-2(1h)-one | Human | 7258 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb1 | A | B | n-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamide | Human | 5103 | |
| MAPK14 (p38a) | MAPK | CMGC | 5eta | A | | - | Human | 7136 | |
| MAPK14 (p38a) | MAPK | CMGC | 2yix | A | | 1-ethyl-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)urea | Human | 5143 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zs5 | A | A | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 4987 | |
| MAPK14 (p38a) | MAPK | CMGC | 8x3m | A | A | - | Human | 15701 | |
| MAPK14 (p38a) | MAPK | CMGC | 3rin | A | | n-cyclopropyl-4-methyl-3-(2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indol]-6'-yl)benzamide | Human | 5239 | |
| MAPK14 (p38a) | MAPK | CMGC | 1wbv | A | | 3-fluoro-n-1h-indol-5-yl-5-morpholin-4-ylbenzamide | Human | 5148 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9y | A | A | n,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5225 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | B | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | 5147 | |
| MAPK14 (p38a) | MAPK | CMGC | 3nnu | A | A | 2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamide | Human | 5094 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zya | A | A | 2-amino-phenylamino-dibenzosuberone | Human | 5105 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh7 | A | B | (3-phenoxyphenyl)methanol | Human | 5020 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw6 | A | A | ethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylate | Human | 4990 | |
| MAPK14 (p38a) | MAPK | CMGC | 1w7h | A | | 3-(benzyloxy)pyridin-2-amine | Human | 5023 | |
| MAPK14 (p38a) | MAPK | CMGC | 2okr | D | | - | Human | 5100 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj2 | A | B | - | Human | 15702 | |
| MAPK14 (p38a) | MAPK | CMGC | 4aa5 | A | | n-cyclopropyl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]benzamide | Human | 5206 | |
| MAPK14 (p38a) | MAPK | CMGC | 4fa2 | A | B | trans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanol | Human | 5145 | |
| MAPK14 (p38a) | MAPK | CMGC | 6hwv | A | B | - | Human | 11250 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n66 | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 8524 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 1 | - | Human | 5021 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | A | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5162 | |
| MAPK14 (p38a) | MAPK | CMGC | 6m95 | A | | (4-benzylpiperidin-1-yl)[2-methoxy-4-(methylsulfanyl)phenyl]methanone | Human | 11252 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh8 | A | B | [3-(benzyloxy)phenyl]methanol | Human | 5014 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 10 | - | Human | 5063 | |
| MAPK14 (p38a) | MAPK | CMGC | 2zb0 | A | A | n-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamide | Human | 5099 | |
| MAPK14 (p38a) | MAPK | CMGC | 6anl | A | B | tak-715 | Human | 9518 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ds6 | D | | n-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamide | Human | 5123 | |
| MAPK14 (p38a) | MAPK | CMGC | 5ml5 | A | | 3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-methylsulfanyl-1~{h}-imidazol-5-yl]pyridin-2-yl]propanamide | Human | 7544 | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg6 | A | | 4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methyl-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5228 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj4 | A | A | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 15703 | |
| MAPK14 (p38a) | MAPK | CMGC | 3ha8 | A | A | n~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamide | Human | 5253 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 6 | - | Human | 5219 | |
| MAPK14 (p38a) | MAPK | CMGC | 3e93 | A | A | 4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamide | Human | 5241 | |
| MAPK14 (p38a) | MAPK | CMGC | 9cj4 | A | B | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 15704 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcs | A | B | 4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamide | Human | 5052 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh6 | A | | n-phenylpyridine-3-carboxamide | Human | 5083 | |
| MAPK14 (p38a) | MAPK | CMGC | 3bv2 | A | | 5-methyl-4-[(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)amino]-n-(1-phenylethenyl)pyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5191 | |
| MAPK14 (p38a) | MAPK | CMGC | 8x3m | A | B | - | Human | 15705 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hll | A | B | 3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamide | Human | 5104 | |
| MAPK14 (p38a) | MAPK | CMGC | 3mpt | A | A | n-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamide | Human | 5224 | |
| MAPK14 (p38a) | MAPK | CMGC | 4e5b | A | | - | Human | 5221 | |
| MAPK14 (p38a) | MAPK | CMGC | 2lgc | A | 7 | - | Human | 5161 | |
| MAPK14 (p38a) | MAPK | CMGC | 5xyx | A | A | n-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amine | Human | 9519 | |
| MAPK14 (p38a) | MAPK | CMGC | 4f9w | A | A | n,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amine | Human | 5130 | |
| MAPK14 (p38a) | MAPK | CMGC | 1zz2 | A | | n-[3-(4-fluorophenoxy)phenyl]-4-[(2-hydroxybenzyl)amino]piperidine-1-sulfonamide | Human | 5164 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcu | B | B | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5126 | |
| MAPK14 (p38a) | MAPK | CMGC | 3iw8 | A | | 1-{4-[(1s)-1-amino-2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-(3-chloro-4-fluorophenyl)urea | Human | 5181 | |
| MAPK14 (p38a) | MAPK | CMGC | 4ewq | A | B | 3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazine | Human | 5245 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh4 | A | | phenyl(piperidin-1-yl)methanone | Human | 5043 | |
| MAPK14 (p38a) | MAPK | CMGC | 5etf | A | B | - | Human | 7135 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkl | A | | n-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-2h-pyran-4-ylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]benzamide | Human | 5172 | |
| MAPK14 (p38a) | MAPK | CMGC | 4eh5 | A | | benzyl pyridine-3-carboxylate | Human | 5185 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n67 | A | B | - | Human | 8521 | |
| MAPK14 (p38a) | MAPK | CMGC | 4zth | A | A | 6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazine | Human | 6706 | |
| MAPK14 (p38a) | MAPK | CMGC | 1zyj | A | | 4-phenoxy-n-(pyridin-2-ylmethyl)benzamide | Human | 5058 | |
| MAPK14 (p38a) | MAPK | CMGC | 3fkn | A | | 3-[2-chloro-5-(methylsulfonyl)phenyl]-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidine | Human | 5049 | |
| MAPK14 (p38a) | MAPK | CMGC | 6sfj | A | A | ~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamide | Human | 11614 | |
| MAPK14 (p38a) | MAPK | CMGC | 1ove | A | B | 1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-one | Human | 5087 | |
| MAPK14 (p38a) | MAPK | CMGC | 2rg5 | A | | n-ethyl-4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamide | Human | 5254 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n65 | A | | 2-phenyl-~{n}4-(2-thiophen-2-ylethyl)quinazoline-4,7-diamine | Human | 8525 | |
| MAPK14 (p38a) | MAPK | CMGC | 4dlj | A | | 2-phenyl-n~4~-(2-phenylethyl)quinazoline-4,7-diamine | Human | 5242 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n63 | A | | - | Human | 8526 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcp | A | B | 4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridine | Human | 5157 | |
| MAPK14 (p38a) | MAPK | CMGC | 3hv5 | B | A | 1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}urea | Human | 5085 | |
| MAPK14 (p38a) | MAPK | CMGC | 1oz1 | A | B | 3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-ol | Human | 5261 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsh | A | B | 2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamide | Human | 5118 | |
| MAPK14 (p38a) | MAPK | CMGC | 6ohd | A | A | 3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamide | Human | 11818 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcv | A | A | 1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5088 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n64 | A | | - | Human | 8527 | |
| MAPK14 (p38a) | MAPK | CMGC | 3gcq | A | A | 1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]urea | Human | 5066 | |
| GSK3B | GSK | CMGC | 9x2q | A | B | - | Human | 15789 | |
| GSK3B | GSK | CMGC | 4acg | A | | 2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamide | Human | 681 | |
| GSK3B | GSK | CMGC | 9fr5 | A | | ~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)furo[3,2-d]pyrimidine-2,4-diamine | Human | 15790 | |
| GSK3B | GSK | CMGC | 4ptg | B | B | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamide | Human | 754 | |
| GSK3B | GSK | CMGC | 6hk4 | B | B | 3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamide | Human | 11427 | |
| GSK3B | GSK | CMGC | 1gng | B | | - | Human | 700 | |
| GSK3B | GSK | CMGC | 5f94 | B | A | 2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamide | Human | 6372 | |
| GSK3B | GSK | CMGC | 3sd0 | B | | 3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dione | Human | 673 | |
| GSK3B | GSK | CMGC | 4ptg | A | A | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamide | Human | 735 | |
| GSK3B | GSK | CMGC | 8djd | A | B | 2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamide | Human | 14668 | |
| GSK3B | GSK | CMGC | 5kpk | B | | (4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9731 | |
| GSK3B | GSK | CMGC | 3pup | A | | ruthenium octasporine | Human | 7207 | |
| GSK3B | GSK | CMGC | 6y9s | A | A | ~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamide | Human | 12286 | |
| GSK3B | GSK | CMGC | 8djc | A | B | (4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamide | Human | 14669 | |
| GSK3B | GSK | CMGC | 4ach | A | | 3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamide | Human | 653 | |
| GSK3B | GSK | CMGC | 3gb2 | A | B | 2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazole | Human | 734 | |
| GSK3B | GSK | CMGC | 3zrl | B | A | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 718 | |
| GSK3B | GSK | CMGC | 3zrl | B | C | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 676 | |
| GSK3B | GSK | CMGC | 3f88 | A | B | 5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 679 | |
| GSK3B | GSK | CMGC | 4j71 | A | A | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 642 | |
| GSK3B | GSK | CMGC | 5hlp | B | A | 4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-one | Human | 6646 | |
| GSK3B | GSK | CMGC | 1o9u | A | | 9-methyl-9h-purin-6-amine | Human | 708 | |
| GSK3B | GSK | CMGC | 4acd | A | | 3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 723 | |
| GSK3B | GSK | CMGC | 1q4l | A | | 2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acid | Human | 714 | |
| GSK3B | GSK | CMGC | 5hlp | A | B | 4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-one | Human | 6648 | |
| GSK3B | GSK | CMGC | 4ach | B | | 3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamide | Human | 702 | |
| GSK3B | GSK | CMGC | 9x2u | A | A | - | Human | 15791 | |
| GSK3B | GSK | CMGC | 7u33 | A | A | 3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamide | Human | 14198 | |
| GSK3B | GSK | CMGC | 3i4b | B | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamide | Human | 629 | |
| GSK3B | GSK | CMGC | 1j1c | A | | adenosine-5'-diphosphate | Human | 696 | |
| GSK3B | GSK | CMGC | 3m1s | B | B | ruthenium pyridocarbazole | Human | 7208 | |
| GSK3B | GSK | CMGC | 7z1g | A | | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 14662 | |
| GSK3B | GSK | CMGC | 3f7z | B | C | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 686 | |
| GSK3B | GSK | CMGC | 1pyx | B | | phosphoaminophosphonic acid-adenylate ester | Human | 663 | |
| GSK3B | GSK | CMGC | 3zrk | A | C | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 697 | |
| GSK3B | GSK | CMGC | 4pte | A | A | n-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamide | Human | 716 | |
| GSK3B | GSK | CMGC | 1r0e | A | B | 3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 672 | |
| GSK3B | GSK | CMGC | 3pup | B | | ruthenium octasporine | Human | 7211 | |
| GSK3B | GSK | CMGC | 5t31 | A | | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9565 | |
| GSK3B | GSK | CMGC | 5k5n | B | | 5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamide | Human | 7410 | |
| GSK3B | GSK | CMGC | 6gjo | A | | (3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-one | Human | 10974 | |
| GSK3B | GSK | CMGC | 3l1s | B | | (4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-one | Human | 713 | |
| GSK3B | GSK | CMGC | 1q41 | A | | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | 628 | |
| GSK3B | GSK | CMGC | 6v6l | A | B | 1-(6-((2-((6-amino-5-nitropyridin-2-yl)amino)ethyl)amino)-2-(2,4-dichlorophenyl)pyridin-3-yl)-4-methylpiperazin-2-one | Human | 11912 | |
| GSK3B | GSK | CMGC | 9fr8 | A | | ~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)thieno[3,2-d]pyrimidine-2,4-diamine | Human | 15793 | |
| GSK3B | GSK | CMGC | 4nm0 | A | B | adenosine-5'-diphosphate | Human | 671 | |
| GSK3B | GSK | CMGC | 4ptc | A | A | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | 664 | |
| GSK3B | GSK | CMGC | 7sxh | A | B | (4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-ol | Human | 14784 | |
| GSK3B | GSK | CMGC | 3gb2 | A | A | 2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazole | Human | 727 | |
| GSK3B | GSK | CMGC | 4nm3 | A | B | adenosine-5'-diphosphate | Human | 640 | |
| GSK3B | GSK | CMGC | 4acc | B | | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 669 | |
| GSK3B | GSK | CMGC | 3zdi | A | | 3,6-diamino-4-(2-chlorophenyl)thieno[2,3-b]pyridine-2,5-dicarbonitrile | Human | 748 | |
| GSK3B | GSK | CMGC | 4nm5 | A | A | adenosine-5'-diphosphate | Human | 755 | |
| GSK3B | GSK | CMGC | 5hln | A | | chir99021 | Human | 6649 | |
| GSK3B | GSK | CMGC | 7b6f | A | A | 3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrile | Human | 13069 | |
| GSK3B | GSK | CMGC | 7sxj | A | A | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 14785 | |
| GSK3B | GSK | CMGC | 3say | A | B | (3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamide | Human | 661 | |
| GSK3B | GSK | CMGC | 6hk4 | A | A | 3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamide | Human | 11429 | |
| GSK3B | GSK | CMGC | 4j71 | B | A | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 641 | |
| GSK3B | GSK | CMGC | 6y9r | A | A | ~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamide | Human | 12287 | |
| GSK3B | GSK | CMGC | 4pte | B | A | n-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamide | Human | 722 | |
| GSK3B | GSK | CMGC | 6hk4 | A | B | 3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamide | Human | 11423 | |
| GSK3B | GSK | CMGC | 5k5n | A | | 5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamide | Human | 7411 | |
| GSK3B | GSK | CMGC | 2jld | B | A | ruthenium pyridocarbazole | Human | 7205 | |
| GSK3B | GSK | CMGC | 2jld | A | B | ruthenium pyridocarbazole | Human | 7214 | |
| GSK3B | GSK | CMGC | 6h0u | A | | (2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamide | Human | 11049 | |
| GSK3B | GSK | CMGC | 3say | A | A | (3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamide | Human | 738 | |
| GSK3B | GSK | CMGC | 3f88 | A | A | 5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 741 | |
| GSK3B | GSK | CMGC | 8av1 | A | A | 2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxaline | Human | 14706 | |
| GSK3B | GSK | CMGC | 8auz | A | A | 8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxaline | Human | 14707 | |
| GSK3B | GSK | CMGC | 3zrl | A | A | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 712 | |
| GSK3B | GSK | CMGC | 5hlp | A | A | 4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-one | Human | 6647 | |
| GSK3B | GSK | CMGC | 5kpl | B | A | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9728 | |
| GSK3B | GSK | CMGC | 8dje | A | A | (4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamide | Human | 14670 | |
| GSK3B | GSK | CMGC | 5oy4 | A | | ~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamide | Human | 8621 | |
| GSK3B | GSK | CMGC | 3zrm | B | B | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 652 | |
| GSK3B | GSK | CMGC | 5f95 | A | | 2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamide | Human | 6373 | |
| GSK3B | GSK | CMGC | 2jld | A | A | ruthenium pyridocarbazole | Human | 7213 | |
| GSK3B | GSK | CMGC | 4afj | B | A | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 678 | |
| GSK3B | GSK | CMGC | 3zrm | A | C | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 724 | |
| GSK3B | GSK | CMGC | 4b7t | A | | (5z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-methyl-2-(propan-2-ylamino)imidazol-4-one | Human | 732 | |
| GSK3B | GSK | CMGC | 3zrk | A | A | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 675 | |
| GSK3B | GSK | CMGC | 1uv5 | A | | 6-bromoindirubin-3'-oxime | Human | 759 | |
| GSK3B | GSK | CMGC | 4j71 | A | B | (2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 690 | |
| GSK3B | GSK | CMGC | 1q5k | A | | n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea | Human | 680 | |
| GSK3B | GSK | CMGC | 8auz | A | B | 8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxaline | Human | 14708 | |
| GSK3B | GSK | CMGC | 5kpm | B | | (4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9734 | |
| GSK3B | GSK | CMGC | 3zrl | A | B | 7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 725 | |
| GSK3B | GSK | CMGC | 6hk3 | B | A | 3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11422 | |
| GSK3B | GSK | CMGC | 7u31 | A | A | 5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amine | Human | 14199 | |
| GSK3B | GSK | CMGC | 6hk7 | A | | 3-azanyl-~{n}-(2-methoxyethyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11428 | |
| GSK3B | GSK | CMGC | 4ptc | B | A | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | 747 | |
| GSK3B | GSK | CMGC | 4pte | A | B | n-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamide | Human | 717 | |
| GSK3B | GSK | CMGC | 3zrk | B | A | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 637 | |
| GSK3B | GSK | CMGC | 1r0e | B | A | 3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 687 | |
| GSK3B | GSK | CMGC | 1h8f | A | | - | Human | 745 | |
| GSK3B | GSK | CMGC | 6y9s | B | B | ~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamide | Human | 12288 | |
| GSK3B | GSK | CMGC | 5f94 | B | B | 2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamide | Human | 6371 | |
| GSK3B | GSK | CMGC | 4ptg | B | A | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamide | Human | 740 | |
| GSK3B | GSK | CMGC | 3l1s | A | | (4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-one | Human | 757 | |
| GSK3B | GSK | CMGC | 7u33 | A | B | 3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamide | Human | 14200 | |
| GSK3B | GSK | CMGC | 5f94 | A | B | 2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamide | Human | 6369 | |
| GSK3B | GSK | CMGC | 6y9r | A | B | ~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamide | Human | 12289 | |
| GSK3B | GSK | CMGC | 4afj | A | A | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 632 | |
| GSK3B | GSK | CMGC | 3f7z | A | C | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 685 | |
| GSK3B | GSK | CMGC | 4acd | B | | 3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 692 | |
| GSK3B | GSK | CMGC | 3zrm | A | A | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 751 | |
| GSK3B | GSK | CMGC | 4afj | A | C | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 742 | |
| GSK3B | GSK | CMGC | 1q41 | B | | (z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oxime | Human | 658 | |
| GSK3B | GSK | CMGC | 1j1b | B | | phosphoaminophosphonic acid-adenylate ester | Human | 657 | |
| GSK3B | GSK | CMGC | 1gng | A | | - | Human | 665 | |
| GSK3B | GSK | CMGC | 6hk3 | A | A | 3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11425 | |
| GSK3B | GSK | CMGC | 4j1r | C | | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 688 | |
| GSK3B | GSK | CMGC | 4afj | B | C | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 711 | |
| GSK3B | GSK | CMGC | 4dit | A | | n-(pyridin-3-yl)-2-(thiophen-3-yl)-3h-imidazo[4,5-b]pyridine-7-carboxamide | Human | 689 | |
| GSK3B | GSK | CMGC | 7u31 | A | B | 5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amine | Human | 14201 | |
| GSK3B | GSK | CMGC | 3m1s | B | A | ruthenium pyridocarbazole | Human | 7210 | |
| GSK3B | GSK | CMGC | 4afj | A | B | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 683 | |
| GSK3B | GSK | CMGC | 1h8f | B | | - | Human | 666 | |
| GSK3B | GSK | CMGC | 4acg | B | | 2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamide | Human | 721 | |
| GSK3B | GSK | CMGC | 4ptc | B | B | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | 758 | |
| GSK3B | GSK | CMGC | 4nm7 | A | B | adenosine-5'-diphosphate | Human | 684 | |
| GSK3B | GSK | CMGC | 3zrm | A | B | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 648 | |
| GSK3B | GSK | CMGC | 1q3w | A | | 9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-one | Human | 635 | |
| GSK3B | GSK | CMGC | 5f94 | A | A | 2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamide | Human | 6374 | |
| GSK3B | GSK | CMGC | 4nm5 | A | B | adenosine-5'-diphosphate | Human | 694 | |
| GSK3B | GSK | CMGC | 5hlp | B | B | 4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-one | Human | 6645 | |
| GSK3B | GSK | CMGC | 3say | B | B | (3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamide | Human | 710 | |
| GSK3B | GSK | CMGC | 8av1 | A | B | 2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxaline | Human | 14709 | |
| GSK3B | GSK | CMGC | 1q5k | B | | n-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)urea | Human | 651 | |
| GSK3B | GSK | CMGC | 3zrk | B | C | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 731 | |
| GSK3B | GSK | CMGC | 5kpk | A | | (4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9735 | |
| GSK3B | GSK | CMGC | 6hk3 | A | B | 3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamide | Human | 11426 | |
| GSK3B | GSK | CMGC | 5oy4 | B | | ~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamide | Human | 8622 | |
| GSK3B | GSK | CMGC | 2ow3 | A | | bis-(indole)maleimide pyridinophane | Human | 698 | |
| GSK3B | GSK | CMGC | 1pyx | A | | phosphoaminophosphonic acid-adenylate ester | Human | 645 | |
| GSK3B | GSK | CMGC | 5kpl | A | B | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9730 | |
| GSK3B | GSK | CMGC | 3sd0 | A | | 3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dione | Human | 720 | |
| GSK3B | GSK | CMGC | 1q3w | B | | 9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-one | Human | 693 | |
| GSK3B | GSK | CMGC | 3f7z | A | B | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 647 | |
| GSK3B | GSK | CMGC | 3f7z | B | A | 2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazole | Human | 749 | |
| GSK3B | GSK | CMGC | 6gjo | B | | (3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-one | Human | 10973 | |
| GSK3B | GSK | CMGC | 4ptg | A | B | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamide | Human | 634 | |
| GSK3B | GSK | CMGC | 3du8 | B | | (7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 737 | |
| GSK3B | GSK | CMGC | 1i09 | B | | - | Human | 638 | |
| GSK3B | GSK | CMGC | 6b8j | A | B | chir99021 | Human | 8659 | |
| GSK3B | GSK | CMGC | 4iq6 | A | | 6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amine | Human | 728 | |
| GSK3B | GSK | CMGC | 7u2z | A | B | (3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamide | Human | 14202 | |
| GSK3B | GSK | CMGC | 4nm0 | A | A | adenosine-5'-diphosphate | Human | 715 | |
| GSK3B | GSK | CMGC | 4j1r | B | | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 656 | |
| GSK3B | GSK | CMGC | 3du8 | A | | (7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-one | Human | 701 | |
| GSK3B | GSK | CMGC | 7u2z | A | A | (3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamide | Human | 14203 | |
| GSK3B | GSK | CMGC | 5hln | B | | chir99021 | Human | 6650 | |
| GSK3B | GSK | CMGC | 4pte | B | B | n-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamide | Human | 667 | |
| GSK3B | GSK | CMGC | 2ow3 | B | | bis-(indole)maleimide pyridinophane | Human | 649 | |
| GSK3B | GSK | CMGC | 1q4l | B | | 2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acid | Human | 655 | |
| GSK3B | GSK | CMGC | 8dje | A | B | (4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamide | Human | 14671 | |
| GSK3B | GSK | CMGC | 3say | B | A | (3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamide | Human | 682 | |
| GSK3B | GSK | CMGC | 1j1b | A | | phosphoaminophosphonic acid-adenylate ester | Human | 707 | |
| GSK3B | GSK | CMGC | 6gn1 | A | | ~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamide | Human | 9997 | |
| GSK3B | GSK | CMGC | 4nm7 | A | A | adenosine-5'-diphosphate | Human | 695 | |
| GSK3B | GSK | CMGC | 5kpl | B | B | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9733 | |
| GSK3B | GSK | CMGC | 4j1r | A | | (2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-one | Human | 709 | |
| GSK3B | GSK | CMGC | 2o5k | A | | 2-(2,4-dichloro-phenyl)-7-hydroxy-1h-benzoimidazole-4-carboxylic acid [2-(4-methanesulfonylamino-phenyl)-ethyl]-amide | Human | 633 | |
| GSK3B | GSK | CMGC | 7sxj | A | B | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 14786 | |
| GSK3B | GSK | CMGC | 6y9s | A | B | ~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamide | Human | 12290 | |
| GSK3B | GSK | CMGC | 3q3b | A | | 4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-one | Human | 660 | |
| GSK3B | GSK | CMGC | 6b8j | A | A | chir99021 | Human | 8658 | |
| GSK3B | GSK | CMGC | 7z1f | A | | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 14663 | |
| GSK3B | GSK | CMGC | 3zrm | B | C | 7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-one | Human | 706 | |
| GSK3B | GSK | CMGC | 6tcu | A | B | 5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamide | Human | 12781 | |
| GSK3B | GSK | CMGC | 7u36 | A | | (3s)-1-[(2-fluorophenoxy)acetyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamide | Human | 14204 | |
| GSK3B | GSK | CMGC | 5kpl | A | A | (4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9729 | |
| GSK3B | GSK | CMGC | 5f95 | B | | 2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamide | Human | 6370 | |
| GSK3B | GSK | CMGC | 7sxh | A | A | (4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-ol | Human | 14787 | |
| GSK3B | GSK | CMGC | 8ff8 | A | | 2-(4-cyanoanilino)-n-(4-phenylpyridin-3-yl)pyrimidine-4-carboxamide | Human | 14763 | |
| GSK3B | GSK | CMGC | 3zrk | B | B | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 662 | |
| GSK3B | GSK | CMGC | 3zrk | A | B | 2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-one | Human | 644 | |
| GSK3B | GSK | CMGC | 3f88 | B | B | 5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thione | Human | 756 | |
| GSK3B | GSK | CMGC | 7b6f | A | B | 3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrile | Human | 13070 | |
| GSK3B | GSK | CMGC | 4acc | A | | 3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamide | Human | 704 | |
| GSK3B | GSK | CMGC | 6gn1 | B | | ~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamide | Human | 9996 | |
| GSK3B | GSK | CMGC | 2jld | B | B | ruthenium pyridocarbazole | Human | 7209 | |
| GSK3B | GSK | CMGC | 8djc | A | A | (4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamide | Human | 14672 | |
| GSK3B | GSK | CMGC | 3q3b | B | | 4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-one | Human | 674 | |
| GSK3B | GSK | CMGC | 3m1s | A | A | ruthenium pyridocarbazole | Human | 7212 | |
| GSK3B | GSK | CMGC | 3i4b | A | | n-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamide | Human | 646 | |
| GSK3B | GSK | CMGC | 4nm3 | A | A | adenosine-5'-diphosphate | Human | 730 | |
| GSK3B | GSK | CMGC | 3m1s | A | B | ruthenium pyridocarbazole | Human | 7206 | |
| GSK3B | GSK | CMGC | 4ptc | A | B | 2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamide | Human | 659 | |
| GSK3B | GSK | CMGC | 1i09 | A | | - | Human | 630 | |
| GSK3B | GSK | CMGC | 5kpm | A | | (4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-one | Human | 9732 | |
| GSK3B | GSK | CMGC | 1r0e | B | B | 3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dione | Human | 639 | |
| GSK3B | GSK | CMGC | 8djd | A | A | 2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamide | Human | 14673 | |
| SRPK2 | SRPK | CMGC | 5myv | A | B | 5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamide | Human | 7575 | |
| CLK1 | CLK | CMGC | 5j1v | A | | pyrido[3,4-g]quinazoline-2,10-diamine | Human | 6582 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qal | A | B | 1,1-bis(oxidanylidene)thietan-3-ol | Human | 10981 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6g91 | A | A | 5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amine | Human | 9965 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fmq | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 2619 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4zzo | A | B | n-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamide | Human | 2606 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6qa4 | A | B | 1~{h}-pyridin-2-one | Human | 11351 | |
| MAPK1 (Erk2) | MAPK | CMGC | 5v60 | A | A | phosphomethylphosphonic acid adenylate ester | Human | 8261 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gdq | A | B | 4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamide | Human | 9973 | |
| MAPK1 (Erk2) | MAPK | CMGC | 6gjd | A | A | cyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamate | Human | 10829 | |
| MAPK1 (Erk2) | MAPK | CMGC | 4fv0 | A | B | n-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amine | Human | 2599 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 8q77 | A | B | (2~{s})-2-[[(2~{s})-2-[[(2~{s})-2-[12-[[4-[[5-(4-carboxyphenyl)-1,3-thiazol-2-yl]amino]-4-oxidanylidene-butanoyl]-(2-hydroxy-2-oxoethyl)amino]dodecanoylamino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]butanedioic acid | Human | 15022 | |
| CSNK2A2 (CK2a2) | CK2 | CMGC | 5ooi | B | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9444 | |
| SRPK1 | SRPK | CMGC | 1wak | A | | - | Human | 120 | |
| MAPK14 (p38a) | MAPK | CMGC | 3od6 | X | | - | Human | 5134 | |
| MAPK14 (p38a) | MAPK | CMGC | 5n68 | A | | - | Human | 8522 | |
| MAPK14 (p38a) | MAPK | CMGC | 3zsi | A | A | 5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-one | Human | 5056 | |
| GSK3B | GSK | CMGC | 6h0u | B | | (2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamide | Human | 11050 | |
| GSK3B | GSK | CMGC | 4afj | B | B | 5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide | Human | 726 | |
| CDK12 (CRK7) | CDK | CMGC | 8bus | B | | 1,3-dimethyl-5-[[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]methyl]pyrazole-4-sulfonamide | Human | 14908 | |
| CDK12 (CRK7) | CDK | CMGC | 8buc | B | | 2-(1~{h}-benzimidazol-2-ylsulfanyl)-~{n}-(5-chloranylpyridin-2-yl)ethanamide | Human | 14909 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu4 | B | | (2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-ol | Human | 14910 | |
| CDK12 (CRK7) | CDK | CMGC | 8bul | B | | (2~{r})-2-[[6-(3-phenylpropylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14911 | |
| CDK12 (CRK7) | CDK | CMGC | 6td3 | E | | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 12369 | |
| CDK12 (CRK7) | CDK | CMGC | 8bue | B | | ~{n}-(1~{h}-benzimidazol-2-yl)-1-(2-methoxy-5-methyl-phenyl)-5-oxidanylidene-pyrrolidine-3-carboxamide | Human | 14912 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu7 | B | | - | Human | 14913 | |
| CDK12 (CRK7) | CDK | CMGC | 8bu9 | B | | r-roscovitine | Human | 14914 | |
| CDK12 (CRK7) | CDK | CMGC | 5acb | D | | n-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamide | Human | 6702 | |
| CDK12 (CRK7) | CDK | CMGC | 8bur | B | A | ~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamide | Human | 14915 | |
| CDK12 (CRK7) | CDK | CMGC | 8bun | B | | (2~{r})-2-[[6-[(4-phenylphenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-ol | Human | 14916 | |
| CDK12 (CRK7) | CDK | CMGC | 4nst | A | | adenosine-5'-diphosphate | Human | 4852 | |
| CDK6 | CDK | CMGC | 1g3n | E | | - | Human | 2805 | |
| CDK6 | CDK | CMGC | 3nup | A | | 4-[3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(1-methylpiperidin-4-yl)pyrimidin-2-amine | Human | 2797 | |
| CDK6 | CDK | CMGC | 4tth | B | | 9-cyclopentyl-n-(5-piperazin-1-ylpyridin-2-yl)pyrido[4,5]pyrrolo[1,2-d]pyrimidin-2-amine | Human | 2803 | |
| CDK6 | CDK | CMGC | 5l2i | A | | 6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-one | Human | 6991 | |
| CDK2 | CDK | CMGC | 2r3i | A | A | 5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4135 | |
| CDK2 | CDK | CMGC | 3r7u | A | B | 2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamide | Human | 4023 | |
| CDK2 | CDK | CMGC | 1h08 | A | A | (2r)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-ol | Human | 4220 | |
| CDK2 | CDK | CMGC | 2whb | C | B | - | Human | 4352 | |
| CDK2 | CDK | CMGC | 4eoi | C | A | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4522 | |
| CDK2 | CDK | CMGC | 1ckp | A | A | purvalanol b | Human | 4066 | |
| CDK2 | CDK | CMGC | 2uzd | C | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamide | Human | 3900 | |
| CDK2 | CDK | CMGC | 4fkj | A | B | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamide | Human | 4164 | |
| CDK2 | CDK | CMGC | 1pxp | A | B | - | Human | 3943 | |
| CDK2 | CDK | CMGC | 2wfy | A | B | - | Human | 4426 | |
| CDK2 | CDK | CMGC | 2wev | A | C | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4007 | |
| CDK2 | CDK | CMGC | 2b53 | A | | 6-(3-aminophenyl)-n-(tert-butyl)-2-(trifluoromethyl)quinazolin-4-amine | Human | 3875 | |
| CDK2 | CDK | CMGC | 4fkp | A | C | 3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indole | Human | 4468 | |
| CDK2 | CDK | CMGC | 4d1z | A | | (4s)-2-(8-hydroxyquinolin-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acid | Human | 4486 | |
| CDK2 | CDK | CMGC | 1h0w | A | A | 1-amino-6-cyclohex-3-enylmethyloxypurine | Human | 3987 | |
| CDK2 | CDK | CMGC | 1oir | A | | 1-(dimethylamino)-3-(4-{{4-(2-methylimidazo[1,2-a]pyridin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-ol | Human | 4389 | |
| CDK2 | CDK | CMGC | 3ezr | A | | 3-methoxy-4-{3-[4-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}aniline | Human | 4475 | |
| CDK2 | CDK | CMGC | 5l2w | A | | 3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridinium | Human | 6993 | |
| CDK2 | CDK | CMGC | 1h1r | C | A | 6-cyclohexylmethoxy-2-(3'-chloroanilino) purine | Human | 3920 | |
| CDK2 | CDK | CMGC | 3qqf | A | B | 5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4287 | |
| CDK2 | CDK | CMGC | 6q3c | A | B | 4-bromo-1h-pyrazole | Human | 11203 | |
| CDK2 | CDK | CMGC | 5iey | A | B | 4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamide | Human | 6573 | |
| CDK2 | CDK | CMGC | 4nj3 | A | B | 6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acid | Human | 4366 | |
| CDK2 | CDK | CMGC | 9gla | A | B | 7-dimethylphosphoryl-3-[2-[[(3~{s})-6,6-dimethylpiperidin-3-yl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]-1~{h}-indole-6-carbonitrile | Human | 15921 | |
| CDK2 | CDK | CMGC | 2iw8 | C | A | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 4294 | |
| CDK2 | CDK | CMGC | 6sg4 | C | B | - | Human | 13245 | |
| CDK2 | CDK | CMGC | 2vtl | A | | n-phenyl-1h-pyrazole-3-carboxamide | Human | 3870 | |
| CDK2 | CDK | CMGC | 4cfw | C | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamide | Human | 4508 | |
| CDK2 | CDK | CMGC | 1w98 | A | | - | Human | 4013 | |
| CDK2 | CDK | CMGC | 7vdu | A | A | [1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanol | Human | 14136 | |
| CDK2 | CDK | CMGC | 9esn | A | A | 4-bromo-1-(2-hydroxyethyl)pyridin-2(1h)-one | Human | 15922 | |
| CDK2 | CDK | CMGC | 2r3o | A | B | (5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanol | Human | 4354 | |
| CDK2 | CDK | CMGC | 2vta | A | | 1h-indazole | Human | 4118 | |
| CDK2 | CDK | CMGC | 4fko | A | A | 2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamine | Human | 4449 | |
| CDK2 | CDK | CMGC | 3qtr | A | A | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 3874 | |
| CDK2 | CDK | CMGC | 4bck | C | A | 3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamide | Human | 4268 | |
| CDK2 | CDK | CMGC | 3ej1 | A | | n-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amine | Human | 4168 | |
| CDK2 | CDK | CMGC | 6q4g | A | A | 2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acid | Human | 11214 | |
| CDK2 | CDK | CMGC | 2uzl | C | | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamide | Human | 4106 | |
| CDK2 | CDK | CMGC | 1dm2 | A | A | 4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-one | Human | 4104 | |
| CDK2 | CDK | CMGC | 3rpy | A | A | 4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4261 | |
| CDK2 | CDK | CMGC | 3roy | A | B | 4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4239 | |
| CDK2 | CDK | CMGC | 3py0 | A | B | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 3869 | |
| CDK2 | CDK | CMGC | 3ddq | C | B | r-roscovitine | Human | 4289 | |
| CDK2 | CDK | CMGC | 4cfn | A | A | 6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amine | Human | 4285 | |
| CDK2 | CDK | CMGC | 4eoq | A | B | adenosine-5'-triphosphate | Human | 4230 | |
| CDK2 | CDK | CMGC | 6q4b | A | A | 5-bromanylpyrimidine | Human | 11198 | |
| CDK2 | CDK | CMGC | 2a0c | X | B | 2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenol | Human | 3868 | |
| CDK2 | CDK | CMGC | 9eso | A | A | - | Human | 15926 | |
| CDK2 | CDK | CMGC | 4lyn | A | | (2s)-n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)-2-phenylpropanamide | Human | 4550 | |
| CDK2 | CDK | CMGC | 3qtr | A | B | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanone | Human | 4243 | |
| CDK2 | CDK | CMGC | 2r3f | A | A | 5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine | Human | 4175 | |
| CDK2 | CDK | CMGC | 1oiu | A | A | 3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamide | Human | 4110 | |
| CDK2 | CDK | CMGC | 6rij | A | B | 4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenol | Human | 12624 | |
| CDK2 | CDK | CMGC | 4ek4 | A | A | 4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamide | Human | 4212 | |
| CDK2 | CDK | CMGC | 3rpy | A | B | 4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4519 | |
| CDK2 | CDK | CMGC | 5osj | A | A | - | Human | 9743 | |
| CDK2 | CDK | CMGC | 5cyi | A | B | 6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amine | Human | 6054 | |
| CDK2 | CDK | CMGC | 1jst | A | | adenosine-5'-triphosphate | Human | 4455 | |
| CDK2 | CDK | CMGC | 4fkg | A | A | 4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acid | Human | 4020 | |
| CDK2 | CDK | CMGC | 2w17 | A | A | n-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amine | Human | 3968 | |
| CDK2 | CDK | CMGC | 2r64 | A | | n-[5-(1,1-dioxidoisothiazolidin-2-yl)-1h-indazol-3-yl]-2-(4-piperidin-1-ylphenyl)acetamide | Human | 4425 | |
| CDK2 | CDK | CMGC | 6guf | A | | n2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamine | Human | 10770 | |
| CDK2 | CDK | CMGC | 2r3o | A | A | (5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanol | Human | 4147 | |
| CDK2 | CDK | CMGC | 13gk | A | A | 4-[(1m)-1-{4-[(azetidin-1-yl)methyl]-2-chlorophenyl}-1h-imidazol-4-yl]-n-[1-(methanesulfonyl)piperidin-4-yl]-5-(trifluoromethyl)pyrimidin-2-amine | Human | 15927 | |
| CDK2 | CDK | CMGC | 1aq1 | A | | staurosporine | Human | 4267 | |
| CDK2 | CDK | CMGC | 2vtr | A | B | 5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 3907 | |
| CDK2 | CDK | CMGC | 8ypw | A | | methyl 3-[4-[3-[[3-[(1-ethylsulfonylpiperidin-4-yl)carbamoyl]-1~{h}-pyrazol-4-yl]carbamoyl]-2,4-bis(fluoranyl)phenyl]piperidin-1-yl]-3-oxidanylidene-propanoate | Human | 15928 | |
| CDK2 | CDK | CMGC | 3my5 | C | B | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 4003 | |
| CDK2 | CDK | CMGC | 2uzb | C | C | 4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamide | Human | 4045 | |
| CDK2 | CDK | CMGC | 1urw | A | A | 2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]- | Human | 4054 | |
| CDK2 | CDK | CMGC | 1h28 | A | | - | Human | 4169 | |
| CDK2 | CDK | CMGC | 9esp | A | A | 4-bromo-1-(2-methoxyethyl)-1h-pyrazole | Human | 15929 | |
| CDK2 | CDK | CMGC | 5if1 | A | B | - | Human | 6569 | |
| CDK2 | CDK | CMGC | 2bkz | C | | 1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamide | Human | 4555 | |
| CDK2 | CDK | CMGC | 1r78 | A | B | 4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-one | Human | 4249 | |
| CDK2 | CDK | CMGC | 2wev | A | A | [4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amine | Human | 4067 | |
| CDK2 | CDK | CMGC | 3rkb | A | A | [4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4460 | |
| CDK2 | CDK | CMGC | 4fkg | A | B | 4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acid | Human | 4559 | |
| CDK2 | CDK | CMGC | 3unj | A | | 4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acid | Human | 4498 | |
| CDK2 | CDK | CMGC | 4ez3 | A | | 4-[(e)-(6-hydroxy-2-oxo-1,2-dihydropyridin-3-yl)diazenyl]benzenesulfonamide | Human | 4551 | |
| CDK2 | CDK | CMGC | 4bcm | C | A | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 4227 | |
| CDK2 | CDK | CMGC | 6q49 | A | A | - | Human | 11185 | |
| CDK2 | CDK | CMGC | 5k4j | A | B | 1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-one | Human | 6750 | |
| CDK2 | CDK | CMGC | 1ykr | A | | 4-{[6-(2,6-dichlorobenzoyl)imidazo[1,2-a]pyridin-2-yl]amino}benzenesulfonamide | Human | 4578 | |
| CDK2 | CDK | CMGC | 6q4k | A | B | - | Human | 11186 | |
| CDK2 | CDK | CMGC | 2i40 | C | B | 5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamide | Human | 4043 | |
| CDK2 | CDK | CMGC | 1ke8 | A | | 4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}-n-(1,3-thiazol-2-yl)benzenesulfonamide | Human | 4048 | |
| CDK2 | CDK | CMGC | 2cch | C | B | adenosine-5'-triphosphate | Human | 4000 | |
| CDK2 | CDK | CMGC | 2wih | C | | n,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamide | Human | 4119 | |
| CDK2 | CDK | CMGC | 2c5v | C | B | 4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amine | Human | 4209 | |
| CDK2 | CDK | CMGC | 2r3q | A | C | 3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxide | Human | 3976 | |
| CDK2 | CDK | CMGC | 3r83 | A | B | 4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamide | Human | 4543 | |
| CDK2 | CDK | CMGC | 3r7v | A | B | 5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamide | Human | 4183 | |
| CDK2 | CDK | CMGC | 4cfx | C | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamide | Human | 4257 | |
| CDK2 | CDK | CMGC | 3r73 | A | A | 4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamide | Human | 4187 | |
| CDK2 | CDK | CMGC | 5mhq | A | A | (2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-ol | Human | 9409 | |
| CDK2 | CDK | CMGC | 9esz | A | A | - | Human | 15944 | |
| CDK2 | CDK | CMGC | 4cfn | C | A | 6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amine | Human | 4355 | |
| CDK2 | CDK | CMGC | 3qzg | A | B | 2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenol | Human | 4347 | |
| CDK2 | CDK | CMGC | 2jgz | A | | - | Human | 4117 | |
| CDK2 | CDK | CMGC | 7ack | C | B | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | 13452 | |
| CDK2 | CDK | CMGC | 6jgm | A | | 4-{[6-(cyclohexylmethoxy)-7h-purin-2-yl]amino}-n,n-diethylbenzamide | Human | 12008 | |
| CDK2 | CDK | CMGC | 4fx3 | A | A | (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acid | Human | 4518 | |
| CDK2 | CDK | CMGC | 1gz8 | A | A | 1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanol | Human | 3981 | |
| CDK2 | CDK | CMGC | 3qtq | A | A | [4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanone | Human | 4210 | |
| CDK2 | CDK | CMGC | 2iw9 | A | B | o6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purine | Human | 3955 | |
| CDK2 | CDK | CMGC | 1ogu | C | A | 4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamide | Human | 3964 | |
| CDK2 | CDK | CMGC | 3qu0 | A | B | 4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4558 | |
| CDK2 | CDK | CMGC | 7rwe | A | | 5-nitro-2-[(3-phenylpropyl)amino]benzoic acid | Human | 14345 | |
| CDK2 | CDK | CMGC | 9esz | A | B | 5-iodanylpyrimidine | Human | 15946 | |
| CDK2 | CDK | CMGC | 1p5e | A | | 4,5,6,7-tetrabromobenzotriazole | Human | 4090 | |
| CDK2 | CDK | CMGC | 2r3q | A | B | 3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxide | Human | 4459 | |
| CDK2 | CDK | CMGC | 3rpv | A | B | 4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamide | Human | 4372 | |
| CDK2 | CDK | CMGC | 4fkt | A | A | n-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamide | Human | 4548 | |
| CDK2 | CDK | CMGC | 1fin | A | | adenosine-5'-triphosphate | Human | 4367 | |
| CDK2 | CDK | CMGC | 3dog | A | B | (2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-ol | Human | 4365 | |
| CDK2 | CDK | CMGC | 3ddp | A | A | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 6781 | |
| CDK2 | CDK | CMGC | 1wcc | A | A | 2-amino-6-chloropyrazine | Human | 4394 | |
| CDK2 | CDK | CMGC | 6q48 | A | B | 4-iodanyl-3~{h}-pyridin-2-one | Human | 11218 | |
| CDK2 | CDK | CMGC | 1oi9 | C | B | 6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purine | Human | 4036 | |
| CDK2 | CDK | CMGC | 7ack | A | B | 8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-one | Human | 13453 | |
| CDK2 | CDK | CMGC | 13gk | A | B | 4-[(1m)-1-{4-[(azetidin-1-yl)methyl]-2-chlorophenyl}-1h-imidazol-4-yl]-n-[1-(methanesulfonyl)piperidin-4-yl]-5-(trifluoromethyl)pyrimidin-2-amine | Human | 15947 | |
| CDK2 | CDK | CMGC | 1jvp | P | 2 | 3-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazole | Human | 4097 | |
| CDK2 | CDK | CMGC | 4eoo | A | B | adenosine-5'-triphosphate | Human | 4278 | |
| CDK2 | CDK | CMGC | 3ddp | C | A | (2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 6784 | |
| CDK2 | CDK | CMGC | 11gv | A | B | (1r,3s)-3-{3-[(1-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl bicyclo[1.1.1]pentan-1-ylcarbamate | Human | 15948 | |
| CDK2 | CDK | CMGC | 6gue | A | | 4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amine | Human | 10771 | |
| CDK2 | CDK | CMGC | 6sg4 | A | B | - | Human | 13247 | |
| CDK2 | CDK | CMGC | 6guc | C | | (3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-one | Human | 10766 | |
| CDK2 | CDK | CMGC | 7e34 | A | | - | Human | 13497 | |
| CDK2 | CDK | CMGC | 2wpa | A | | n-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamide | Human | 4399 | |
| CDK2 | CDK | CMGC | 1okv | A | | - | Human | 3921 | |
| CDK2 | CDK | CMGC | 3qts | A | B | [4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanone | Human | 4564 | |
| CDK2 | CDK | CMGC | 1hck | A | A | adenosine-5'-triphosphate | Human | 3878 | |
| CDK2 | CDK | CMGC | 6q4g | A | B | 2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acid | Human | 11217 | |
| CDK2 | CDK | CMGC | 3my5 | A | C | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 3910 | |
| CDK2 | CDK | CMGC | 6sg4 | C | A | - | Human | 13248 | |
| CDK2 | CDK | CMGC | 9esl | A | A | 4-bromanyl-1-(2-methoxyethyl)pyridin-2-one | Human | 15950 | |
| CDK2 | CDK | CMGC | 6q3c | A | C | - | Human | 11178 | |
| CDK2 | CDK | CMGC | 4ii5 | C | B | adenosine-5'-diphosphate | Human | 4462 | |
| CDK2 | CDK | CMGC | 6q4a | A | C | 5-iodanylpyrimidine | Human | 11216 | |
| CDK2 | CDK | CMGC | 3qwj | A | A | 2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamide | Human | 4265 | |
| CDK2 | CDK | CMGC | 3r9o | A | | 4-amino-n-(3,5-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamide | Human | 4279 | |
| CDK2 | CDK | CMGC | 3qru | A | A | (5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamide | Human | 4237 | |
| CDK2 | CDK | CMGC | 1h0v | A | A | 5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinone | Human | 4368 | |
| CDK2 | CDK | CMGC | 4eon | C | B | (5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-one | Human | 4192 | |
| CDK2 | CDK | CMGC | 4ek3 | A | B | - | Human | 4202 | |
| CDK2 | CDK | CMGC | 4cfv | C | B | 3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenol | Human | 3979 | |
| CDK2 | CDK | CMGC | 1oiy | C | B | 4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamide | Human | 4245 | |
| CDK2 | CDK | CMGC | 6q48 | A | A | 4-iodanyl-3~{h}-pyridin-2-one | Human | 11192 | |
| CDK2 | CDK | CMGC | 4bzd | A | A | 6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amine | Human | 3865 | |
| CDK2 | CDK | CMGC | 1vyw | A | | n-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamide | Human | 3992 | |
| CDK2 | CDK | CMGC | 1y91 | A | | 4-[5-(trans-4-aminocyclohexylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-7-ylamino]-n,n-dimethylbenzenesulfonamide | Human | 4505 | |
| CDK2 | CDK | CMGC | 7b5l | L | | - | Human | 13266 | |
| CDK8 | CDK | CMGC | 4f7s | A | A | n-(2-phenylethyl)quinazolin-4-amine | Human | 3850 | |
| CDK8 | CDK | CMGC | 5hbe | A | B | 8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one | Human | 6386 | |
| CDKL2 | CDKL | CMGC | 4bbm | B | | 4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diol | Human | 965 | |
| CDKL2 | CDKL | CMGC | 4aaa | A | A | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 964 | |
| CDKL2 | CDKL | CMGC | 4aaa | A | B | 5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamide | Human | 962 | |
| CDKL2 | CDKL | CMGC | 4bbm | A | | 4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diol | Human | 963 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7n8t | A | A | adenosine monophosphate | Human | 14241 | |
| MAPK9 (JNK2) | MAPK | CMGC | 3npc | A | | 1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-urea | Human | 1235 | |
| MAPK9 (JNK2) | MAPK | CMGC | 3e7o | B | | n-{3-[5-(1h-1,2,4-triazol-3-yl)-1h-indazol-3-yl]phenyl}furan-2-carboxamide | Human | 1236 | |
| MAPK9 (JNK2) | MAPK | CMGC | 7cml | A | A | - | Human | 12707 | |
| CDK9 | CDK | CMGC | 3tni | A | | - | Human | 2250 | |
| CDK9 | CDK | CMGC | 4imy | E | A | adenosine monophosphate | Human | 2258 | |
| CDK9 | CDK | CMGC | 4imy | C | B | adenosine monophosphate | Human | 2245 | |
| CDK9 | CDK | CMGC | 4bch | A | | 4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrile | Human | 2246 | |
| CDK9 | CDK | CMGC | 4bcg | A | | 2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 2255 | |
| CDK9 | CDK | CMGC | 4ogr | A | | adenosine | Human | 2254 | |
| CDK9 | CDK | CMGC | 4bcj | A | | 2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 2247 | |
| CDK9 | CDK | CMGC | 6w9e | A | B | (4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone | Human | 13858 | |
| CDK9 | CDK | CMGC | 4or5 | A | | - | Human | 2233 | |
| CDK9 | CDK | CMGC | 6w9e | A | D | (4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanone | Human | 13860 | |
| CDK9 | CDK | CMGC | 3blh | A | | - | Human | 2251 | |
| CDK9 | CDK | CMGC | 3my1 | A | | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 2249 | |
| CDK9 | CDK | CMGC | 3lq5 | A | | (2s)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-ol | Human | 2253 | |
| CDK9 | CDK | CMGC | 4or5 | F | | - | Human | 2231 | |
| CDK9 | CDK | CMGC | 3tnh | A | | 4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenol | Human | 2232 | |
| CDK9 | CDK | CMGC | 4bcf | A | | 2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrile | Human | 2257 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | C | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12784 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yll | B | | - | Human | 12785 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | B | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12786 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | C | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12787 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | A | A | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12788 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | D | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12789 | |
| MAPK6 (Erk3) | MAPK | CMGC | 6yky | A | B | 3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amine | Human | 12790 | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | B | A | - | Human | 12980 | |
| MAPK6 (Erk3) | MAPK | CMGC | 7aqb | A | B | - | Human | 12981 | |
| CDK7 | CDK | CMGC | 6xd3 | J | | n-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamide | Human | 12772 | |
| CDK7 | CDK | CMGC | 8byq | I | | - | Human | 14732 | |
| CDK7 | CDK | CMGC | 6o9l | 8 | | - | Human | 11055 | |
| CDK7 | CDK | CMGC | 8pyr | A | A | - | Human | 15254 | |
| CDK7 | CDK | CMGC | 6xbz | J | | phosphothiophosphoric acid-adenylate ester | Human | 12773 | |
| CDK7 | CDK | CMGC | 1ua2 | B | | adenosine-5'-triphosphate | Human | 541 | |
| CDK7 | CDK | CMGC | 1ua2 | A | | adenosine-5'-triphosphate | Human | 540 | |
| CDK7 | CDK | CMGC | 29wd | I | | - | Human | 16031 | |
| CDK7 | CDK | CMGC | 8bvw | I | | - | Human | 14733 | |
| CDK7 | CDK | CMGC | 7b5o | J | B | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13279 | |
| CDK7 | CDK | CMGC | 7b5q | J | B | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13280 | |
| HIPK2 | DYRK | CMGC | 6p5s | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11512 | |
| HIPK2 | DYRK | CMGC | 6p5s | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 11513 | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | A | B | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10926 | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | B | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 1715 | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | A | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10923 | |
| MAPK3 (Erk1) | MAPK | CMGC | 2zoq | B | | (2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diol | Human | 1712 | |
| MAPK3 (Erk1) | MAPK | CMGC | 9uw3 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 16037 | |
| MAPK3 (Erk1) | MAPK | CMGC | 9uw4 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 16038 | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | A | B | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 1713 | |
| MAPK3 (Erk1) | MAPK | CMGC | 4qtb | A | A | (3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamide | Human | 1714 | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | B | A | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10925 | |
| MAPK3 (Erk1) | MAPK | CMGC | 6ges | B | B | n-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamide | Human | 10924 | |
| CDK4 | CDK | CMGC | 5fwp | K | | - | Human | 7132 | |
| CDK4 | CDK | CMGC | 6p8h | B | | - | Human | 11894 | |
| CDK4 | CDK | CMGC | 2w9z | B | A | - | Human | 3388 | |
| CDK4 | CDK | CMGC | 2w9f | B | | - | Human | 3386 | |
| CDK4 | CDK | CMGC | 6p8g | B | | - | Human | 11893 | |
| CDK4 | CDK | CMGC | 2w96 | B | A | - | Human | 3390 | |
| CDK4 | CDK | CMGC | 2w96 | B | B | - | Human | 3389 | |
| CDK4 | CDK | CMGC | 5fwl | K | | - | Human | 6748 | |
| CDK4 | CDK | CMGC | 2w99 | B | | - | Human | 3385 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4uba | B | | 4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acid | Human | 5525 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3w8l | A | | - | Human | 5427 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6eii | A | B | (3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azanium | Human | 9647 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mot | A | A | 4-hydroxybenzamide | Human | 7660 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu4 | A | B | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6895 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | B | A | - | Human | 5532 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5t1h | B | B | 7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 8684 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otq | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methoxy-phenyl]methyl]ethanamine | Human | 9638 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owl | A | A | 11-chloro-8-methyl-7h-benzo[e]pyrido[4,3-b]indol-3-ol | Human | 5502 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oul | A | B | [3-chloranyl-4-(3-fluorophenyl)phenyl]methanamine | Human | 9675 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvh | B | B | adenosine-5'-diphosphate | Human | 6917 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7psu | A | A | - | Human | 14163 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9z | A | A | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5510 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l21 | A | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12011 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5t1h | B | A | 7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 8683 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oni | A | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9455 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3juh | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5471 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9x | A | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5488 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oth | A | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9612 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmr | B | A | - | Human | 7651 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehu | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamine | Human | 9691 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mow | A | A | 5-bromopyridine-2,3-diamine | Human | 7670 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7aya | A | A | ~{n}-[2-[(1~{r},2~{r})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 13991 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4kwp | A | B | 4,5,6,7-tetrabromo-1-(2-deoxy-beta-d-erythro-pentofuranosyl)-1h-benzimidazole | Human | 5482 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oth | B | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9670 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9x | A | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5446 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ouu | B | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 9636 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6qy7 | A | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12122 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4c | A | A | 3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acid | Human | 7402 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ctp | A | B | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7289 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4rll | A | A | 4-[(e)-(9h-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acid | Human | 5418 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6fvg | A | A | adenosine-5'-triphosphate | Human | 11340 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4dgl | C | | - | Human | 5474 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypg | A | A | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12425 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1jwh | A | | phosphoaminophosphonic acid-adenylate ester | Human | 5485 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3h30 | B | A | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 5484 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu3 | A | A | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6902 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlo | A | B | 5,6,7-tris(bromanyl)-1~{h}-benzotriazole | Human | 13074 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn3 | A | A | - | Human | 10703 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ub7 | A | | 4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acid | Human | 5462 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqu | A | B | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6038 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypk | A | B | - | Human | 12426 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tei | B | B | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12457 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlo | A | C | - | Human | 13075 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo5 | A | B | ~{n}-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propyl]methanesulfonamide | Human | 7661 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csh | B | B | adenosine-5'-triphosphate | Human | 6907 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo5 | A | A | ~{n}-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propyl]methanesulfonamide | Human | 7676 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot5 | A | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9676 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oqu | A | A | adenosine-5'-diphosphate | Human | 9615 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9x | B | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5516 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tll | A | C | 4,5,6,7-tetrabromobenzotriazole | Human | 13076 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nsz | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 5503 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3amy | A | | 5,7-dihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-one | Human | 5506 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otd | A | A | [2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azanium | Human | 9697 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os8 | A | A | adenosine-5'-triphosphate | Human | 9608 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oul | A | A | [3-chloranyl-4-(3-fluorophenyl)phenyl]methanamine | Human | 9622 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md8 | F | | - | Human | 5475 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypn | B | A | adenosine-5'-diphosphate | Human | 12427 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ct0 | A | A | 3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-ol | Human | 7296 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot6 | A | B | (3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-pyrrol-2-yl)ethyl]azanium | Human | 9643 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nga | B | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5511 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu4 | A | C | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6916 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo8 | A | B | 3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acid | Human | 7673 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orh | A | B | - | Human | 9671 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otl | A | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9633 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tls | A | A | 5,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13077 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu4 | A | A | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6924 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yph | B | A | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12428 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orh | A | A | - | Human | 9620 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hop | A | B | 4-hydroxy-3-methoxybenzaldehyde | Human | 11660 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlp | A | B | 5,6-dibromobenzotriazole | Human | 13078 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb7 | A | B | naphtho[2,1-b:7,8-b']difuran-2,9-dicarboxylic acid | Human | 5455 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l24 | A | A | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12013 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rff | A | B | (~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-nitro-4-oxidanyl-phenyl)prop-2-enamide | Human | 12149 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otd | A | B | [2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azanium | Human | 9696 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hbn | A | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11287 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oqu | A | B | adenosine-5'-diphosphate | Human | 9627 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 2zjw | A | | 2,3,7,8-tetrahydroxychromeno[5,4,3-cde]chromene-5,10-dione | Human | 5423 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yph | B | B | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12429 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oyf | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methyl-phenyl]methyl]ethanamine | Human | 9658 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7at5 | A | B | ~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamide | Human | 13839 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gmd | A | A | adenosine-5'-triphosphate | Human | 9993 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8b | A | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 6408 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3w8l | B | | - | Human | 5469 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvf | A | A | adenosine-5'-triphosphate | Human | 6927 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osz | A | B | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azanium | Human | 9685 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ork | A | A | adenosine-5'-diphosphate | Human | 9693 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mod | B | A | - | Human | 7679 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3bqc | A | A | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5486 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn4 | A | B | - | Human | 10708 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot5 | A | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9656 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo7 | B | B | - | Human | 7685 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn4 | A | A | - | Human | 10700 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oum | A | B | ~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]-2-(1~{h}-imidazol-2-yl)ethanamine | Human | 9677 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwe | A | B | 7-(1~{h}-indol-2-yl)-5-methyl-~{n}-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine | Human | 14771 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gmd | A | B | adenosine-5'-triphosphate | Human | 9990 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu2 | B | A | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7292 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7qge | A | B | 4,5,6,7-tetrabromobenzotriazole | Human | 14467 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4b | B | B | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13166 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mpj | B | A | - | Human | 7675 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hbn | B | B | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11272 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvh | B | A | adenosine-5'-diphosphate | Human | 6914 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cs6 | A | B | - | Human | 6901 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yul | A | | 7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acid | Human | 12458 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu0 | B | A | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7295 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8g | A | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]ethanamide | Human | 6405 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mow | B | B | - | Human | 7686 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu2 | B | B | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7286 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md8 | H | | - | Human | 5518 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hme | B | A | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11279 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 2pvr | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5509 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md8 | G | | - | Human | 5478 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlv | A | A | 6-bromanyl-1~{h}-benzotriazole | Human | 13079 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os7 | B | B | adenosine-5'-triphosphate | Human | 9645 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yph | A | B | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12431 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csv | A | A | 3-aminobenzoic acid | Human | 6898 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6z84 | B | | ~{n}-[1-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]ethanamide | Human | 12649 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn1 | A | A | - | Human | 10696 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3u9c | A | | 7-hydroxy-3h-phenoxazin-3-one | Human | 5461 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4nh1 | A | | phosphomethylphosphonic acid adenylate ester | Human | 5412 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ots | A | A | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3,5-bis(chloranyl)-4-phenyl-phenyl]methyl]azanium | Human | 10589 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oth | A | B | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9659 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md7 | E | | - | Human | 5435 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nsz | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5512 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gih | A | A | - | Human | 9941 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3c13 | A | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5472 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4f | A | A | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7405 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypg | A | B | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12432 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3owl | A | B | 11-chloro-8-methyl-7h-benzo[e]pyrido[4,3-b]indol-3-ol | Human | 5416 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9qsv | A | | 5-(methylamino)benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 16074 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9qrj | A | | 5-[6-[(3-chloranyl-4-phenyl-phenyl)methylamino]hexylamino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 16075 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yph | A | A | 4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acid | Human | 12433 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4b | A | A | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13167 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo7 | A | B | 3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanamide | Human | 7697 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s76 | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 16076 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a49 | B | | 6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridine | Human | 13168 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5nqc | A | B | (3e)-6,7-dichloro-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-one | Human | 8111 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5b0x | A | | 4-[2-[(4-methoxyphenyl)carbonylamino]-1,3-thiazol-5-yl]benzoic acid | Human | 6475 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9hyh | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 16077 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn2 | A | B | - | Human | 10702 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7i8n | A | C | - | Human | 16078 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otl | A | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9681 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy8 | A | A | - | Human | 14441 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m4f | A | B | 4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acid | Human | 7401 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8h | A | A | nicotinic acid | Human | 13260 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5clp | B | B | 2-(3,4-dichlorophenyl)ethanamine | Human | 6911 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oum | A | A | ~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]-2-(1~{h}-imidazol-2-yl)ethanamine | Human | 9668 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os7 | A | A | adenosine-5'-triphosphate | Human | 9644 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5omy | A | A | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9457 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3pe1 | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5500 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3juh | B | A | phosphoaminophosphonic acid-adenylate ester | Human | 5431 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3wil | A | | {[(2z)-2-(3,4-dimethoxybenzylidene)-3-oxo-2,3-dihydro-1-benzofuran-6-yl]oxy}acetic acid | Human | 5468 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ku8 | A | | ~{n}-[2-[(1~{s},2~{s})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 8664 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9z | B | B | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5430 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9qri | A | | 5-[4-[[4-[2-(3,4-dichlorophenyl)ethylamino]-4-oxidanylidene-butanoyl]amino]butylamino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 16079 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmf | B | B | - | Human | 7657 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gmd | B | A | adenosine-5'-triphosphate | Human | 9991 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cx9 | B | A | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7285 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn0 | A | B | - | Human | 10699 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owl | B | A | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10590 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moe | A | B | adenosine-5'-diphosphate | Human | 7662 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn1 | A | B | - | Human | 10707 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osp | A | A | adenosine-5'-triphosphate | Human | 10587 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oue | B | B | (3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-imidazol-4-yl)ethyl]azanium | Human | 9631 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hnw | A | A | coumestrol | Human | 11523 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlr | A | B | 4,7-bis(bromanyl)-1~{h}-benzotriazole | Human | 13083 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ork | B | B | adenosine-5'-diphosphate | Human | 9646 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3h30 | A | B | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 5460 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7i85 | A | B | 5-(ethylamino)benzo[c][2,6]naphthyridine-8-carboxamide | Human | 16080 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l24 | A | B | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12012 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s7i | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 16081 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ork | B | A | adenosine-5'-diphosphate | Human | 9674 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s8j | A | C | phosphoaminophosphonic acid-adenylate ester | Human | 16082 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5t1h | A | B | 7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 8682 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn3 | A | B | - | Human | 10706 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3r0t | A | B | 3-(cyclopropylamino)-5-{[3-(trifluoromethyl)phenyl]amino}pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5517 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypj | A | B | 4-[(4-phenyl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12434 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1na7 | A | | - | Human | 5533 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otp | A | B | 2-[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 10586 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6qy7 | B | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12124 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmr | A | B | ~{n}'-[(3-chloranyl-4-phenyl-phenyl)methyl]butane-1,4-diamine | Human | 7659 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oue | A | A | 3-methyl-5-oxidanyl-benzoic acid | Human | 9686 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l23 | A | A | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 13455 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5omy | A | B | 4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 9456 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orj | B | A | adenosine-5'-diphosphate | Human | 9607 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mpj | A | B | adenosine-5'-diphosphate | Human | 7663 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q38 | A | A | benzoic acid | Human | 11271 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5owl | A | B | 3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amine | Human | 10596 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | C | A | - | Human | 5498 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aem | A | B | adenosine-5'-triphosphate | Human | 14683 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oqu | B | A | adenosine-5'-diphosphate | Human | 9623 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cs6 | B | A | - | Human | 6919 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cs6 | B | B | - | Human | 6926 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 1pjk | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 5494 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ouu | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamine | Human | 9662 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3fwq | A | | - | Human | 5507 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osz | A | C | 2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azanium | Human | 9683 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3h30 | A | A | 5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazole | Human | 5496 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3juh | B | B | phosphoaminophosphonic acid-adenylate ester | Human | 5421 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5moh | A | B | 2-(3-methoxy-4-oxidanyl-phenyl)ethanoic acid | Human | 7681 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo8 | A | A | 3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acid | Human | 7653 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvg | A | A | - | Human | 6913 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oyf | A | A | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methyl-phenyl]methyl]ethanamine | Human | 9617 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo8 | B | A | 3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acid | Human | 7654 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rcm | A | B | (~{e})-~{n}-(5-~{tert}-butyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12143 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orj | A | B | adenosine-5'-diphosphate | Human | 9624 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3axw | A | | 4-(5-amino-1,3,4-thiadiazol-2-yl)benzoic acid | Human | 5440 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7b8i | A | B | - | Human | 13261 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7z39 | A | B | 2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamide | Human | 14445 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oto | A | B | 2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9637 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6z84 | A | | ~{n}-[1-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]ethanamide | Human | 12650 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n1v | B | A | pyrazolo-pyrimidine macrocycle | Human | 7587 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orj | B | B | adenosine-5'-diphosphate | Human | 9665 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9fyf | A | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-4-fluoranyl-2-[(3~{s})-3-(methylamino)piperidin-1-yl]phenyl]propanamide | Human | 16083 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6spx | A | | - | Human | 11960 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn0 | A | D | - | Human | 10709 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot5 | B | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9689 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q04 | A | A | - | Human | 5514 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mot | A | B | 4-hydroxybenzamide | Human | 7691 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3fwq | B | | - | Human | 5479 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l22 | A | B | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12014 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqw | B | A | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6039 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6q4q | B | C | benzoic acid | Human | 11280 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oum | B | B | - | Human | 9606 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9rfn | A | B | - | Human | 16084 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5m44 | A | | 3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acid | Human | 7404 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvf | A | B | adenosine-5'-triphosphate | Human | 6910 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6qy7 | A | B | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12123 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8ae7 | A | B | adenosine-5'-diphosphate | Human | 14684 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tll | A | D | 4,5,6,7-tetrabromobenzotriazole | Human | 13087 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo6 | A | A | 3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoic acid | Human | 7672 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6spw | A | B | - | Human | 11959 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6fvf | A | A | - | Human | 11342 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ypj | A | A | 4-[(4-phenyl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12435 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s8j | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 16085 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osl | A | A | adenosine-5'-diphosphate | Human | 9673 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo7 | A | A | 3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanamide | Human | 7669 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hny | A | A | boldine | Human | 11520 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otl | B | A | ~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamine | Human | 9660 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu2 | A | A | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7303 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l22 | A | A | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12009 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwg | A | B | (5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dione | Human | 14774 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8aem | A | A | adenosine-5'-triphosphate | Human | 14685 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | M | | - | Human | 5520 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6z83 | B | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamide | Human | 12651 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oue | A | B | 3-methyl-5-oxidanyl-benzoic acid | Human | 9614 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6spw | A | A | - | Human | 11961 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3at3 | A | | (1-{6-[6-(cyclopentylamino)-1h-indazol-1-yl]pyrazin-2-yl}-1h-pyrrol-3-yl)acetic acid | Human | 5504 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s6g | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 16086 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q04 | A | B | - | Human | 5419 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hoq | A | B | 3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acid | Human | 11665 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csp | A | C | 2-hydroxy-5-methylbenzoic acid | Human | 6928 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7x4h | A | B | 5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrile | Human | 14596 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7z39 | A | A | 2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamide | Human | 14449 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn0 | A | C | - | Human | 10704 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6gih | A | B | - | Human | 9942 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9l | A | B | (4~{z})-6,7-bis(chloranyl)-4-[[(4-methylphenyl)amino]methylidene]-8-oxidanyl-1,2-dihydrodibenzofuran-3-one | Human | 9621 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 8c5q | A | A | 2-methylpropyl 5-fluoranyl-3-[1-[[1-[2-[[4-(2-methylpropyl)phenyl]sulfonylamino]ethyl]piperidin-4-yl]methyl]-1,2,3-triazol-4-yl]-1~{h}-indole-2-carboxylate | Human | 15177 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6rcm | A | A | (~{e})-~{n}-(5-~{tert}-butyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamide | Human | 12150 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3nga | A | A | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 5422 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | P | | - | Human | 5434 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu2 | A | B | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7302 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hme | A | B | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11283 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqw | A | B | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6037 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ct0 | A | B | 3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-ol | Human | 7300 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7bu4 | A | B | 4-(6-aminocarbonyl-8-oxidanylidene-9-phenyl-7h-purin-2-yl)benzoic acid | Human | 13485 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md7 | F | | - | Human | 5457 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oty | A | B | trifluoroacetic acid | Human | 9680 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s8j | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 16091 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9fbl | A | A | nicotinic acid | Human | 16092 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb6 | A | B | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 5499 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orj | A | A | adenosine-5'-diphosphate | Human | 9653 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s77 | A | B | nicotinic acid | Human | 16093 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo7 | B | A | - | Human | 7698 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3r0t | A | A | 3-(cyclopropylamino)-5-{[3-(trifluoromethyl)phenyl]amino}pyrimido[4,5-c]quinoline-8-carboxylic acid | Human | 5497 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7a4b | B | A | 5,6-dibromo-1h-triazolo[4,5-b]pyridine | Human | 13172 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s7h | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 16094 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqw | A | A | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6034 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mp8 | A | B | adenosine-5'-diphosphate | Human | 7649 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csh | A | B | adenosine-5'-triphosphate | Human | 6925 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8b | B | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 6406 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6yzh | A | B | adenosine-5'-diphosphate | Human | 13560 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehu | B | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamine | Human | 9664 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9n | A | B | 1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diol | Human | 9628 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4md9 | H | | - | Human | 5466 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5kwh | A | A | ~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamide | Human | 8617 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5oum | B | A | - | Human | 9679 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osr | A | B | adenosine-5'-triphosphate | Human | 10594 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tei | A | A | 3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acid | Human | 12461 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6a1c | A | A | 5-bromanyl-2-methoxy-4-[(e)-(3-methylsulfanyl-5-phenyl-1,2,4-triazol-4-yl)iminomethyl]phenol | Human | 11273 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5osp | A | B | adenosine-5'-triphosphate | Human | 10600 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s76 | A | B | phosphoaminophosphonic acid-adenylate ester | Human | 16095 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9rcx | A | A | - | Human | 16096 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu3 | B | B | n-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamide | Human | 6897 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9fbm | A | B | nicotinic acid | Human | 16098 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hop | A | A | 3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acid | Human | 11661 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5h8e | B | | ~{n}-[2-[2-azanylethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamide | Human | 6407 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hop | A | D | (2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enal | Human | 11666 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3at2 | A | B | - | Human | 5492 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ctp | B | A | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7297 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4ib5 | A | A | - | Human | 5501 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5n9n | A | A | 1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diol | Human | 9661 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6z83 | A | | ~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamide | Human | 12652 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mo5 | B | A | - | Human | 7689 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5zn5 | A | B | - | Human | 10701 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hny | A | B | boldine | Human | 11522 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cu0 | A | A | n-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamide | Human | 7299 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ot6 | B | B | - | Human | 9649 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy5 | A | B | - | Human | 14453 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4kwp | A | A | 4,5,6,7-tetrabromo-1-(2-deoxy-beta-d-erythro-pentofuranosyl)-1h-benzimidazole | Human | 5465 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orh | B | A | - | Human | 9694 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy8 | A | B | - | Human | 14454 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9w | A | B | 3-methyl-1,6,8-trihydroxyanthraquinone | Human | 5420 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5otr | A | A | adenosine-5'-triphosphate | Human | 9640 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6eii | B | B | (3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azanium | Human | 9642 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4rll | A | B | 4-[(e)-(9h-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acid | Human | 5449 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5ct0 | B | B | 3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-ol | Human | 7298 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9rcy | A | A | - | Human | 16099 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 9s9y | A | A | phosphoaminophosphonic acid-adenylate ester | Human | 16100 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zwe | A | A | 7-(1~{h}-indol-2-yl)-5-methyl-~{n}-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amine | Human | 14775 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5os8 | A | B | adenosine-5'-triphosphate | Human | 9666 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cx9 | B | B | methyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoate | Human | 7294 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3qa0 | A | B | - | Human | 5451 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5orh | B | B | - | Human | 9639 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6l1z | A | | (6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-one | Human | 12010 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hou | A | B | 4-hydroxy-3-methoxybenzaldehyde | Human | 11664 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mmf | B | A | - | Human | 7696 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb6 | A | A | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 5424 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6tlo | A | A | 5,6,7-tris(bromanyl)-1~{h}-benzotriazole | Human | 13092 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6hme | B | B | 5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dione | Human | 11282 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy5 | A | A | - | Human | 14457 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 4nh1 | B | | phosphomethylphosphonic acid adenylate ester | Human | 5531 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cvh | A | B | adenosine-5'-diphosphate | Human | 6912 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3mb6 | A | C | naphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acid | Human | 5529 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5mp8 | A | A | adenosine-5'-diphosphate | Human | 7690 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5cqw | B | B | 4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amine | Human | 6036 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 5csv | A | B | 3-aminobenzoic acid | Human | 6900 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 3q9z | B | A | 1,2,5,8-tetrahydroxyanthracene-9,10-dione | Human | 5426 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6qy7 | B | A | 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol | Human | 12125 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6eii | B | A | (3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azanium | Human | 9654 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7zy2 | A | B | adenosine-5'-triphosphate | Human | 14458 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 7ay9 | A | | 7-(cyclopropylamino)-5-(5-(6-oxo-1,6-dihydropyridin-3-yl)-1-(2-(piperidin-1-yl)ethyl)-1h-1,2,3-triazol-4-yl)pyrazolo[1,5-a]pyrimidine-3-carbonitrile | Human | 13993 | |
| CSNK2A1 (CK2a1) | CK2 | CMGC | 6ehk | A | B | 2-(1~{h}-benzimidazol-2-yl)-~{n}-[[3,5-bis(chloranyl)-4-(2-ethylphenyl)phenyl]methyl]ethanamine | Human | 9663 | |
| CDK5 | CDK | CMGC | 1ung | A | | 6-phenyl[5h]pyrrolo[2,3-b]pyrazine | Human | 2792 | |
| CDK5 | CDK | CMGC | 1h4l | B | | - | Human | 2779 | |
| CDK5 | CDK | CMGC | 4au8 | B | B | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | 2781 | |
| CDK5 | CDK | CMGC | 7vdp | A | | [1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanol | Human | 14145 | |
| CDK5 | CDK | CMGC | 4au8 | A | A | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | 2784 | |
| CDK5 | CDK | CMGC | 1unl | A | | r-roscovitine | Human | 2785 | |
| CDK5 | CDK | CMGC | 4au8 | B | A | 4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamide | Human | 2791 | |
| HIPK3 | DYRK | CMGC | 7o7j | A | | n-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amine | Human | 13997 | |
| CLK2 | CLK | CMGC | 6fyk | A | B | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10408 | |
| CLK2 | CLK | CMGC | 6fyk | A | A | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10406 | |
| CLK2 | CLK | CMGC | 6fyk | B | B | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10401 | |
| CLK2 | CLK | CMGC | 6fyk | B | A | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10407 | |
| CLK2 | CLK | CMGC | 6fyl | A | B | 5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acid | Human | 10404 | |
| CLK2 | CLK | CMGC | 5unp | B | | n~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamine | Human | 9888 | |
| CLK2 | CLK | CMGC | 6fyi | A | | (1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one | Human | 10405 | |
| CLK2 | CLK | CMGC | 6fyk | C | B | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10409 | |
| CLK2 | CLK | CMGC | 6fyk | C | A | (2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amine | Human | 10402 | |
| MAPK12 (p38g) | MAPK | CMGC | 1cm8 | A | | phosphoaminophosphonic acid-adenylate ester | Human | 4625 | |
| MAPK12 (p38g) | MAPK | CMGC | 6una | A | A | - | Human | 11898 | |
| MAPK12 (p38g) | MAPK | CMGC | 6una | B | B | - | Human | 11899 | |
| MAPK12 (p38g) | MAPK | CMGC | 1cm8 | B | | phosphoaminophosphonic acid-adenylate ester | Human | 4626 | |