Search results (3682 entries covering 1836 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
CSNK2A1 (CK2a1)CK2CMGC8p07A7-(cyclopropylamino)-5-[[3-(1,2,4-triazol-4-yl)phenyl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman14743
CDK2CDKCMGC9espAB4-bromo-1-(2-methoxyethyl)-1h-pyrazoleHuman15901
CDK2CDKCMGC2wxvCn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4504
CDK2CDKCMGC5anoA-Human6537
CDK2CDKCMGC4eopAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4258
CDK2CDKCMGC3rakAB4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4331
CDK2CDKCMGC9et2AB~{n}-(4-bromophenyl)ethanamideHuman15902
CDK2CDKCMGC8ru8AA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman15329
CDK2CDKCMGC3unkA4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman4374
CDK2CDKCMGC2vu3AB4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman3884
SRPK1SRPKCMGC1wbpAadenosine-5'-diphosphateHuman119
CDK2CDKCMGC1r78AA4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman4253
MAPK3 (Erk1)MAPKCMGC2zoqA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman1716
CLK3CLKCMGC2wu6AA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman1823
GSK3BGSKCMGC8qjiAn-[4-[5-(1,2,4-oxadiazol-3-yl)thiophen-2-yl]pyridin-2-yl]cyclopropanecarboxamideHuman15386
MAPK1 (Erk2)MAPKCMGC8pt5AAphosphoaminophosphonic acid-adenylate esterHuman15306
MAPK1 (Erk2)MAPKCMGC8pstAAamp phosphoramidateHuman15311
MAPK14 (p38a)MAPKCMGC3k3iAA(3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinolineHuman5212
CDK2CDKCMGC1h00AB(2r)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4428
DYRK1ADYRKCMGC6eisCB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10548
CDK2CDKCMGC2ds1A(13r,15s)-13-methyl-16-oxa-8,9,12,22,24-pentaazahexacyclo[15.6.2.16,9.1,12,15.0,2,7.0,21,25]heptacosa-1(24),2,4,6,17(25),18,20-heptaene-23,26-dioneHuman4513
CDK2CDKCMGC4ek5ABn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHuman4145
CDK2CDKCMGC9eszAD5-iodanylpyrimidineHuman15903
CDK1 (CDC2)CDKCMGC6gu6A3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman10774
CDK2CDKCMGC2wevCA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4503
CDK2CDKCMGC6q4fABpyridine-2,6-diamineHuman11211
CDK2CDKCMGC2uzoA4-{5-[(z)-(2,4-dioxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3862
DYRK1ADYRKCMGC2vx3CAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3740
DYRK1ADYRKCMGC6eivB~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10536
DYRK1ADYRKCMGC7a52AB3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-oneHuman13750
DYRK1ADYRKCMGC4mq1ABn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3736
CDK1 (CDC2)CDKCMGC4yc6EA-Human4612
DYRK1ADYRKCMGC2vx3CBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3735
MAPK1 (Erk2)MAPKCMGC8pt0AAphosphoaminophosphonic acid-adenylate esterHuman15297
CDK1 (CDC2)CDKCMGC6gu4A~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10777
CDK2CDKCMGC3s0oAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHuman4123
CDK2CDKCMGC3qhwCBadenosine-5'-diphosphateHuman4143
CLK2CLKCMGC6fylAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10403
CLK2CLKCMGC6kheA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11651
CLK2CLKCMGC3nr9C(5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman1929
CLK2CLKCMGC3nr9B(5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman1928
CDK2CDKCMGC4fx3AB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman3931
CSNK2A2 (CK2a2)CK2CMGC5ooiAA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9447
CDK2CDKCMGC3qhwABadenosine-5'-diphosphateHuman4156
CDK2CDKCMGC4cfxAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4086
CDK2CDKCMGC3qqhAA2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenolHuman4393
CDK2CDKCMGC3raiAA4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4441
CDK2CDKCMGC3sqqAB4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3925
CDK2CDKCMGC6gueC4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10772
CDK2CDKCMGC1fvvA4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman4065
PRPF4B (PRP4)DYRKCMGC4ijpBB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5534
PRPF4B (PRP4)DYRKCMGC4iirAAphosphoaminophosphonic acid-adenylate esterHuman5545
CDK2CDKCMGC1pxoAB-Human3860
PRPF4B (PRP4)DYRKCMGC4ianA-Human5543
PRPF4B (PRP4)DYRKCMGC4ijpBA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5541
CDK2CDKCMGC3r9hAB4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4336
CDK2CDKCMGC1e1vA6-o-cyclohexylmethyl guanineHuman3886
CDK2CDKCMGC4bcnCA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4436
PRPF4B (PRP4)DYRKCMGC6pjjAB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11577
PRPF4B (PRP4)DYRKCMGC4ifcAAadenosine-5'-diphosphateHuman5538
CLK1CLKCMGC6qtyAAethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman12083
CDK2CDKCMGC4eolAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4089
CDK2CDKCMGC4kd1AA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman4585
CDK2CDKCMGC4bcpCA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman3872
CDK2CDKCMGC4bcnAB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4298
PRPF4B (PRP4)DYRKCMGC4iirABphosphoaminophosphonic acid-adenylate esterHuman5539
PRPF4B (PRP4)DYRKCMGC6pjjAA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11585
PRPF4B (PRP4)DYRKCMGC6pjjBA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11583
PRPF4B (PRP4)DYRKCMGC4iirBBphosphoaminophosphonic acid-adenylate esterHuman5537
PRPF4B (PRP4)DYRKCMGC4ifcBBadenosine-5'-diphosphateHuman5540
PRPF4B (PRP4)DYRKCMGC6pjjCB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11586
CDK2CDKCMGC1h1sCo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4572
CDK2CDKCMGC3ti1AAn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4201
CDK1 (CDC2)CDKCMGC5hq0AB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman6421
CDK2CDKCMGC4cfmAA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4207
CDK2CDKCMGC5ievABroniciclibHuman6570
CDK2CDKCMGC4eosCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4008
CDK2CDKCMGC1pxkAB-Human3980
CDK2CDKCMGC3tnwCB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman4493
CDK2CDKCMGC4fksAAn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4412
CSNK2A1 (CK2a1)CK2CMGC8bgcA5-[(phenylmethyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acidHuman14545
CSNK2A2 (CK2a2)CK2CMGC6hmqAB3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman10998
CSNK2A1 (CK2a1)CK2CMGC5clpAB2-(3,4-dichlorophenyl)ethanamineHuman6920
CSNK2A1 (CK2a1)CK2CMGC7b8hABnicotinic acidHuman13259
CDK8CDKCMGC6qtjA~{n},~{n}-dimethyl-2-[4-[4-(2,6-naphthyridin-4-yl)phenyl]pyrazol-1-yl]ethanamideHuman12093
CSNK2A1 (CK2a1)CK2CMGC5owlBB3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10592
CSNK2A1 (CK2a1)CK2CMGC7x4hAA5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrileHuman14595
CSNK2A1 (CK2a1)CK2CMGC6ehuAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamineHuman9684
CSNK2A1 (CK2a1)CK2CMGC4ubaA4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acidHuman5432
CSNK2A2 (CK2a2)CK2CMGC6qy8DA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12116
CSNK2A1 (CK2a1)CK2CMGC8ae7AAadenosine-5'-diphosphateHuman14682
CSNK2A1 (CK2a1)CK2CMGC5mo6AB3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoic acidHuman7665
CDK8CDKCMGC5hvyABn-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}ureaHuman6552
CSNK2A1 (CK2a1)CK2CMGC4md9L-Human5414
GSK3BGSKCMGC3zrlBB7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman691
CDK2CDKCMGC1urcCA-Human4006
CSNK2A1 (CK2a1)CK2CMGC5moeBAadenosine-5'-diphosphateHuman7693
CSNK2A1 (CK2a1)CK2CMGC6ypkAA-Human12430
CSNK2A1 (CK2a1)CK2CMGC5os7BAadenosine-5'-triphosphateHuman9626
CSNK2A1 (CK2a1)CK2CMGC4md7H-Human5481
CSNK2A1 (CK2a1)CK2CMGC6ehkAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[3,5-bis(chloranyl)-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9641
CSNK2A1 (CK2a1)CK2CMGC5cu3BAn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6921
DYRK1ADYRKCMGC4yu2BA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3737
CSNK2A1 (CK2a1)CK2CMGC3juhABphosphoaminophosphonic acid-adenylate esterHuman5456
CDK2CDKCMGC1pxoAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4512
CDK2CDKCMGC6guhAB4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10769
CDK2CDKCMGC2c5xCBhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4418
CDK2CDKCMGC2cchCC-Human4431
CSNK2A1 (CK2a1)CK2CMGC5otiAA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9672
CSNK2A1 (CK2a1)CK2CMGC3at2AA-Human5428
CSNK2A1 (CK2a1)CK2CMGC6eiiAA(3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azaniumHuman9687
DYRK1ADYRKCMGC5a4qAn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6717
DYRK1ADYRKCMGC4yljCA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3777
CSNK2A1 (CK2a1)CK2CMGC5oniAB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9459
CSNK2A1 (CK2a1)CK2CMGC6fvfAB-Human11341
CSNK2A1 (CK2a1)CK2CMGC6hbnBA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11270
CSNK2A1 (CK2a1)CK2CMGC5n9lAA(4~{z})-6,7-bis(chloranyl)-4-[[(4-methylphenyl)amino]methylidene]-8-oxidanyl-1,2-dihydrodibenzofuran-3-oneHuman9652
CSNK2A1 (CK2a1)CK2CMGC5oslABadenosine-5'-diphosphateHuman9629
CSNK2A1 (CK2a1)CK2CMGC5mohAA2-(3-methoxy-4-oxidanyl-phenyl)ethanoic acidHuman7658
CSNK2A1 (CK2a1)CK2CMGC4gubAn-[5-({3-cyano-7-[(1-methyl-1h-imidazol-4-yl)amino]pyrazolo[1,5-a]pyrimidin-5-yl}amino)-2-methylphenyl]acetamideHuman5491
CSNK2A1 (CK2a1)CK2CMGC5osuAB-Human10598
MAPK14 (p38a)MAPKCMGC1bl7A4-(4-fluorophenyl)-1-(4-piperidinyl)-5-(2-amino-4-pyrimidinyl)-imidazoleHuman5193
CSNK2A1 (CK2a1)CK2CMGC5mpjAAadenosine-5'-diphosphateHuman7677
CSNK2A1 (CK2a1)CK2CMGC4md9K-Human5477
CSNK2A1 (CK2a1)CK2CMGC5othBA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9625
CSNK2A1 (CK2a1)CK2CMGC3warAAnicotinic acidHuman5429
CSNK2A1 (CK2a1)CK2CMGC5mo8BB3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acidHuman7688
CDK2CDKCMGC1ke9A3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4250
CDK2CDKCMGC2b54A6-(3,4-dihydroxybenzyl)-3-ethyl-1-(2,4,6-trichlorophenyl)-1h-pyrazolo[3,4-d]pyrimidin-4(5h)-oneHuman4292
CSNK2A1 (CK2a1)CK2CMGC7a4qAA2-methoxyimino-5-(quinolin-6-ylmethyl)-1,3-thiazol-4-oneHuman14238
CSNK2A1 (CK2a1)CK2CMGC6gmdBBadenosine-5'-triphosphateHuman9992
CSNK2A1 (CK2a1)CK2CMGC3u4uA3-{5-(acetylamino)-3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1h-indol-1-yl}propanoic acidHuman5527
CDK2CDKCMGC2iw8ABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4377
CDK2CDKCMGC2bhhA(2e,3s)-3-hydroxy-5'-[(4-hydroxypiperidin-1-yl)sulfonyl]-3-methyl-1,3-dihydro-2,3'-biindol-2'(1'h)-oneHuman4417
CSNK2A1 (CK2a1)CK2CMGC5n1vABpyrazolo-pyrimidine macrocycleHuman7589
CSNK2A1 (CK2a1)CK2CMGC7zwgAA(5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dioneHuman14772
CSNK2A1 (CK2a1)CK2CMGC5cu3ABn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6903
CSNK2A1 (CK2a1)CK2CMGC5osuAA-Human10595
CSNK2A1 (CK2a1)CK2CMGC4fbxA-Human5415
CSNK2A1 (CK2a1)CK2CMGC7zykAAadenosine-5'-diphosphateHuman14547
CSNK2A1 (CK2a1)CK2CMGC7zwgAC(5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dioneHuman14773
CSNK2A1 (CK2a1)CK2CMGC5ctpBBn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7291
CDK2CDKCMGC3r8vAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3938
CSNK2A1 (CK2a1)CK2CMGC6hoqAA3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acidHuman11669
CSNK2A1 (CK2a1)CK2CMGC3qa0AA-Human5425
CSNK2A1 (CK2a1)CK2CMGC5cx9ABmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7290
CSNK2A1 (CK2a1)CK2CMGC5mpjBB-Human7683
CDK2CDKCMGC3bhuAB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4446
CSNK2A1 (CK2a1)CK2CMGC7at5AA~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamideHuman13840
CSNK2A1 (CK2a1)CK2CMGC5nqcAA(3e)-6,7-dichloro-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-oneHuman8112
CDK2CDKCMGC4fkoAB2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHuman4534
CDK2CDKCMGC4eoiCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4011
CSNK2A1 (CK2a1)CK2CMGC5otzABtrifluoroacetic acidHuman9618
CSNK2A1 (CK2a1)CK2CMGC6tlpAA5,6-dibromobenzotriazoleHuman13080
CSNK2A1 (CK2a1)CK2CMGC4ib5BB-Human5438
CSNK2A1 (CK2a1)CK2CMGC5owhA3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10597
CSNK2A1 (CK2a1)CK2CMGC3q9yAB1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5526
CSNK2A1 (CK2a1)CK2CMGC5otqAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methoxy-phenyl]methyl]ethanamineHuman9651
CSNK2A1 (CK2a1)CK2CMGC6rfeAB(~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12147
CSNK2A1 (CK2a1)CK2CMGC3wowAphosphoaminophosphonic acid-adenylate esterHuman5445
CSNK2A1 (CK2a1)CK2CMGC6rb1AA(~{e})-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)-~{n}-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]prop-2-enamideHuman12145
CSNK2A1 (CK2a1)CK2CMGC6tllAB4,5,6,7-tetrabromobenzotriazoleHuman13081
CSNK2A1 (CK2a1)CK2CMGC5n1vBBpyrazolo-pyrimidine macrocycleHuman7586
CSNK2A1 (CK2a1)CK2CMGC7qgeAA4,5,6,7-tetrabromobenzotriazoleHuman14469
CSNK2A1 (CK2a1)CK2CMGC5mowBA-Human7671
CSNK2A1 (CK2a1)CK2CMGC8c5qAB2-methylpropyl 5-fluoranyl-3-[1-[[1-[2-[[4-(2-methylpropyl)phenyl]sulfonylamino]ethyl]piperidin-4-yl]methyl]-1,2,3-triazol-4-yl]-1~{h}-indole-2-carboxylateHuman15175
CSNK2A1 (CK2a1)CK2CMGC7psuAB-Human14164
CSNK2A1 (CK2a1)CK2CMGC3owjAB9-hydroxy-5,11-dimethyl-4,6-dihydro-1h-pyrido[4,3-b]carbazol-1-oneHuman5470
CSNK2A1 (CK2a1)CK2CMGC5n1vAApyrazolo-pyrimidine macrocycleHuman7588
CSNK2A1 (CK2a1)CK2CMGC5otpBB-Human10591
CDK2CDKCMGC2c5vAA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4012
CSNK2A1 (CK2a1)CK2CMGC5modAB-Human7667
CSNK2A1 (CK2a1)CK2CMGC5zn5AA-Human10705
CSNK2A1 (CK2a1)CK2CMGC7a49A6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13169
CSNK2A1 (CK2a1)CK2CMGC3pe1AA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5487
CSNK2A1 (CK2a1)CK2CMGC3q9zAB1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5437
CSNK2A1 (CK2a1)CK2CMGC5ku8B~{n}-[2-[(1~{s},2~{s})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman8663
CSNK2A1 (CK2a1)CK2CMGC6tlsAB5,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13082
CSNK2A1 (CK2a1)CK2CMGC5otoBA2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9688
CSNK2A1 (CK2a1)CK2CMGC5zn0AA-Human10697
CDK2CDKCMGC4fx3CA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4349
MAPK1 (Erk2)MAPKCMGC8ao6AB~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14396
CDK2CDKCMGC3qqkAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4568
CSNK2A1 (CK2a1)CK2CMGC3c13AA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5530
CSNK2A1 (CK2a1)CK2CMGC6tlvAB6-bromanyl-1~{h}-benzotriazoleHuman13084
CDK2CDKCMGC1oiuCB3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4049
CSNK2A1 (CK2a1)CK2CMGC5ouuAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman9610
CSNK2A1 (CK2a1)CK2CMGC5otoAA2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9648
CSNK2A1 (CK2a1)CK2CMGC3ngaBA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5441
CSNK2A1 (CK2a1)CK2CMGC5movAB4'-hydroxycinnamic acidHuman7674
CSNK2A1 (CK2a1)CK2CMGC4dglD-Human5521
CSNK2A1 (CK2a1)CK2CMGC4ib5CB-Human5476
CSNK2A1 (CK2a1)CK2CMGC6jwaA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman11467
CSNK2A1 (CK2a1)CK2CMGC5os7ABadenosine-5'-triphosphateHuman9609
CSNK2A1 (CK2a1)CK2CMGC4md7G-Human5409
CSNK2A1 (CK2a1)CK2CMGC5modBB-Human7694
CDK2CDKCMGC1h1qC2-anilino-6-cyclohexylmethoxypurineHuman4053
CDK2CDKCMGC1e9hA2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHuman4302
CSNK2A1 (CK2a1)CK2CMGC4grbA5-(2-{[4-(dimethylcarbamoyl)phenyl]amino}-4-methoxypyrimidin-5-yl)thiophene-3-carboxylic acidHuman5443
CSNK2A1 (CK2a1)CK2CMGC6houAA4-hydroxy-3-methoxybenzaldehydeHuman11671
CSNK2A1 (CK2a1)CK2CMGC5cx9AAmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7287
CSNK2A1 (CK2a1)CK2CMGC6rcbA(~{e})-2-cyano-~{n}-(2-hydroxyphenyl)-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12144
CSNK2A1 (CK2a1)CK2CMGC3owjAA9-hydroxy-5,11-dimethyl-4,6-dihydro-1h-pyrido[4,3-b]carbazol-1-oneHuman5452
CSNK2A1 (CK2a1)CK2CMGC5mo6BA-Human7664
CSNK2A1 (CK2a1)CK2CMGC4ib5AB-Human5522
CSNK2A1 (CK2a1)CK2CMGC3q9xBB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5417
CDK4CDKCMGC7sj3An-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman14485
CLK3CLKCMGC6z53AB6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12305
CSNK2A1 (CK2a1)CK2CMGC3u87Aphosphoaminophosphonic acid-adenylate esterHuman5442
CSNK2A1 (CK2a1)CK2CMGC3rpsA3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman5463
CSNK2A1 (CK2a1)CK2CMGC4md9E-Human5411
CSNK2A1 (CK2a1)CK2CMGC5ot6BA-Human9613
CSNK2A1 (CK2a1)CK2CMGC6tlwAC7-bromanyl-1~{h}-benzotriazoleHuman13086
CSNK2A1 (CK2a1)CK2CMGC6teiAB3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12459
CSNK2A1 (CK2a1)CK2CMGC6tlwAA7-bromanyl-1~{h}-benzotriazoleHuman13088
CSNK2A1 (CK2a1)CK2CMGC5kwhBB~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman8620
MAPK9 (JNK2)MAPKCMGC7n8tABadenosine monophosphateHuman14242
MAPK11 (p38b)MAPKCMGC3gc8A5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman2766
MAPK11 (p38b)MAPKCMGC3gc9B5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman2767
MAPK11 (p38b)MAPKCMGC3gc9A5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman2765
MAPK11 (p38b)MAPKCMGC3gc8B5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman2769
MAPK11 (p38b)MAPKCMGC3gp0ABnilotinibHuman2764
MAPK11 (p38b)MAPKCMGC3gp0AAnilotinibHuman2768
CDKL1CDKLCMGC4aguCn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman762
PRPF4B (PRP4)DYRKCMGC8h6jHA-Human15281
PRPF4B (PRP4)DYRKCMGC6pjjCA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11578
PRPF4B (PRP4)DYRKCMGC6pk6AB4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11584
PRPF4B (PRP4)DYRKCMGC4ijpAA4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5547
PRPF4B (PRP4)DYRKCMGC8h6eH-Human15282
PRPF4B (PRP4)DYRKCMGC4ifcABadenosine-5'-diphosphateHuman5544
PRPF4B (PRP4)DYRKCMGC4ijpAB4-(5-{[(2-chloropyridin-4-yl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman5535
PRPF4B (PRP4)DYRKCMGC6cnhAB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman9775
PRPF4B (PRP4)DYRKCMGC6pjjDB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11579
PRPF4B (PRP4)DYRKCMGC6cnhAA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman9776
PRPF4B (PRP4)DYRKCMGC6pjjBB4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11581
PRPF4B (PRP4)DYRKCMGC6pk6AA4-(5-{[(2-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11582
PRPF4B (PRP4)DYRKCMGC8h6jHB-Human15283
PRPF4B (PRP4)DYRKCMGC4ianB-Human5546
PRPF4B (PRP4)DYRKCMGC6pjjDA4-(5-{[(3-aminophenyl)methyl]carbamoyl}thiophen-2-yl)-1-benzothiophene-2-carboxamideHuman11580
PRPF4B (PRP4)DYRKCMGC4iirBAphosphoaminophosphonic acid-adenylate esterHuman5536
PRPF4B (PRP4)DYRKCMGC4ifcBAadenosine-5'-diphosphateHuman5542
SRPK2SRPKCMGC5myvBB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7573
MAPK7 (Erk5)MAPKCMGC5byyAA2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman6591
CDK2CDKCMGC2r3qAA3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman4038
CSNK2A1 (CK2a1)CK2CMGC7ayaAB~{n}-[2-[(1~{r},2~{r})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman13992
CSNK2A1 (CK2a1)CK2CMGC5orkABadenosine-5'-diphosphateHuman9655
CDK5CDKCMGC4au8AB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2786
CLK3CLKCMGC6yu1aA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12403
CLK3CLKCMGC6z2vAB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12636
CSNK2A1 (CK2a1)CK2CMGC7b8iBA-Human13264
MAPK7 (Erk5)MAPKCMGC5o7iAA4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamideHuman9995
MAPK7 (Erk5)MAPKCMGC7pusAB4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamideHuman14219
CDK2CDKCMGC2c5nCBn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman3903
CDK2CDKCMGC7ackCA8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13450
CDK2CDKCMGC2xnbAA3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHuman4217
CDK2CDKCMGC6q49AC-Human11193
CDK2CDKCMGC2wfyAA-Human4324
CDK2CDKCMGC4bcpAB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4304
CDK2CDKCMGC4i3zCadenosine-5'-diphosphateHuman3961
MAPK1 (Erk2)MAPKCMGC4iz7AB-Human2577
CDK2CDKCMGC2r3nAB3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4046
CDK2CDKCMGC3qtqAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4103
CDK2CDKCMGC9esuAC-Human15904
CDK2CDKCMGC6q4aAB5-iodanylpyrimidineHuman11200
CDK2CDKCMGC2fvdA(4-amino-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrimidin-5-yl)(2,3-difluoro-6-methoxyphenyl)methanoneHuman4408
CDK2CDKCMGC6ylkABmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12494
CDK2CDKCMGC3qx4AA4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4409
CDK2CDKCMGC1e1xA6-cyclohexylmethyloxy-5-nitroso-pyrimidine-2,4-diamineHuman4114
CDK2CDKCMGC4cfvAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman4328
CDK2CDKCMGC2bpmC(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHuman4128
CDK5CDKCMGC1h4lA-Human2788
CDK5CDKCMGC7vdrA(1r)-1-[7-[(2-fluoranyl-4-pyrazol-1-yl-phenyl)amino]-1,6-naphthyridin-2-yl]-1-(1-methylpiperidin-4-yl)ethanolHuman14146
CDK2CDKCMGC3eidCA-Human4072
CDK2CDKCMGC2r3kAA3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman3953
CDK2CDKCMGC3s1hAA4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4068
CDK2CDKCMGC3ddqCAr-roscovitineHuman4364
CDK2CDKCMGC3ralAB4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3984
CDK2CDKCMGC2vttA4-{[(2,6-difluorophenyl)carbonyl]amino}-n-[(3s)-piperidin-3-yl]-1h-pyrazole-3-carboxamideHuman4100
CSNK2A1 (CK2a1)CK2CMGC6yumA4-[5-[2-(2-hydroxyethyloxy)ethyl-[(2-methylpropan-2-yl)oxycarbonyl]amino]pyrazolo[1,5-a]pyrimidin-3-yl]-2-oxidanyl-benzoic acidHuman12462
CDK1 (CDC2)CDKCMGC4yc6GA-Human4613
MAPK1 (Erk2)MAPKCMGC7nr5AB(2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13934
MAPK1 (Erk2)MAPKCMGC1wzyA1-allyl-5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman2618
CDK2CDKCMGC1giiA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHuman4448
CDK2CDKCMGC6q4bAB5-bromanylpyrimidineHuman11210
CDK1 (CDC2)CDKCMGC6gu2AB2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10776
CDK2CDKCMGC2r3hAB3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman3970
GSK3BGSKCMGC6y9sBA~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12285
CDK2CDKCMGC5nevA4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHuman8020
CDK2CDKCMGC5mhqAB(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHuman9408
CDK2CDKCMGC2c5vCA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4384
GSK3BGSKCMGC4j1rD(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman736
CDK2CDKCMGC3rprAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanoneHuman4241
CDK8CDKCMGC4f7jAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)ureaHuman3842
CDK2CDKCMGC7rwfA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHuman14344
GSK3BGSKCMGC4j71BB(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman739
CDK2CDKCMGC4ek4AC4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman4369
CDK2CDKCMGC2c5yABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman6777
CDK2CDKCMGC2wmbC-Human4474
CDK2CDKCMGC3qtuAA4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4009
CDK2CDKCMGC3dogCA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4382
DYRK2DYRKCMGC5lxdBAmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7123
GSK3BGSKCMGC4iq6B6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amineHuman750
CDK2CDKCMGC2cjmAadenosine-5'-triphosphateHuman4406
CDK2CDKCMGC4eokAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3913
CDK2CDKCMGC2vtrAA5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4391
CDK2CDKCMGC3eidCB-Human4467
CDK2CDKCMGC3pj8AB(2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-olHuman4454
CDK2CDKCMGC2c5vAB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4338
CDK2CDKCMGC4bcmAA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4290
CDK2CDKCMGC2r3rAB3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4215
CDK2CDKCMGC7m2fAB[(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acidHuman13796
CDK2CDKCMGC3tnwCA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3940
CDK2CDKCMGC3qhwCAadenosine-5'-diphosphateHuman4129
CDK2CDKCMGC2wfyCB-Human4096
CDK2CDKCMGC2wevCC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4288
CDK2CDKCMGC3ddpCB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6778
CDK2CDKCMGC1jsvA4-[(6-amino-4-pyrimidinyl)amino]benzenesulfonamideHuman4171
CDK2CDKCMGC3qtzAA4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4109
CDK2CDKCMGC1pxnAA4-[4-(4-methyl-2-methylamino-thiazol-5-yl)-pyrimidin-2-ylamino]-phenolHuman4383
CDK2CDKCMGC1h0wAB1-amino-6-cyclohex-3-enylmethyloxypurineHuman4016
CDK2CDKCMGC3r9dAA4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4562
CDK1 (CDC2)CDKCMGC6gu7G-Human10779
MAPK1 (Erk2)MAPKCMGC4g6nAB3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazoleHuman2593
CDK2CDKCMGC2cchAAadenosine-5'-triphosphateHuman4303
CDK2CDKCMGC2cchCAadenosine-5'-triphosphateHuman3932
CDK2CDKCMGC1fvvC4-[(7-oxo-7h-thiazolo[5,4-e]indol-8-ylmethyl)-amino]-n-pyridin-2-yl-benzenesulfonamideHuman4461
CDK2CDKCMGC6q4dAB2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11215
CDK2CDKCMGC4eoqCBadenosine-5'-triphosphateHuman3912
CDK2CDKCMGC1ol1C-Human3951
CDK2CDKCMGC3rzbAB4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamideHuman4395
CDK16 (PCTAIRE1)CDKCMGC3mtlAB(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human1702
CDK2CDKCMGC6q4kAA-Human11179
CDK2CDKCMGC1h27C-Human4030
CDK2CDKCMGC1oiuAB3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4556
CDK2CDKCMGC4eorABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3934
CDK2CDKCMGC4bcmCB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4124
CDK2CDKCMGC3pxqA8-anilino-1-naphthalene sulfonateHuman3947
CDK2CDKCMGC1h0vAB5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHuman3933
CDK2CDKCMGC1w8cAA6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHuman4332
CDK2CDKCMGC4eokCo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4385
CDK2CDKCMGC3qtwAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman3890
CDK2CDKCMGC4bckAB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman3960
CDK2CDKCMGC4eooAAadenosine-5'-triphosphateHuman4403
CDK2CDKCMGC2c6mA4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6782
CDK2CDKCMGC3qwjAB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamideHuman4182
DYRK2DYRKCMGC6hdrAAcurcuminHuman11570
DYRK2DYRKCMGC5lxcBAmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7125
DYRK2DYRKCMGC3kvwAB(2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acidHuman3149
MAPK8 (JNK1)MAPKCMGC3o2mB-Human4649
DYRK2DYRKCMGC7dh3A2,7-dimethoxy-9-piperidin-4-ylsulfanyl-acridineHuman13978
DYRK2DYRKCMGC5ztnB(1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneHuman10483
DYRK2DYRKCMGC7ejvBB[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14182
DYRK2DYRKCMGC7ejvBA[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14183
DYRK2DYRKCMGC7dhkA2-methoxy-7-phenylmethoxy-9-(piperidin-4-ylmethylsulfanyl)acridineHuman13977
CDK1 (CDC2)CDKCMGC6gu7A4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10781
MAPK8 (JNK1)MAPKCMGC2xrwAAphosphoaminophosphonic acid-adenylate esterHuman4675
CDK16 (PCTAIRE1)CDKCMGC5g6vB4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman7274
CDK2CDKCMGC7ackAA8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13451
MAPK8 (JNK1)MAPKCMGC3vulA-Human4633
CLK1CLKCMGC6khdAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11645
CDK2CDKCMGC7s4tAA2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHuman14374
DYRK1ADYRKCMGC7aj2AB4-(4-methoxyphenyl)pyridin-2-amineHuman13592
DYRK1ADYRKCMGC7ajaAB1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazineHuman13597
DYRK1ADYRKCMGC7aj2AA4-(4-methoxyphenyl)pyridin-2-amineHuman13609
CLK1CLKCMGC6khdCA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11648
CDK2CDKCMGC2r3lAC3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4496
MAPK1 (Erk2)MAPKCMGC5wp1AA5,7-dihydroxy-4h-1-benzopyran-4-oneHuman10441
CSNK2A2 (CK2a2)CK2CMGC7atvAB~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamideHuman13828
CDK2CDKCMGC7s4tAB2-{[2-(6-chloro-1h-indol-3-yl)ethyl]amino}-5-nitrobenzoic acidHuman14373
CDK2CDKCMGC8h6pA(7s,10r)-11-oxa-2,4,5,13,17,23-hexaazatetracyclo[17.3.1.1~3,6~.1~7,10~]pentacosa-1(23),3(25),5,19,21-pentaene-12,18-dioneHuman14625
CDK2CDKCMGC5nevC4-[[6-(3-phenylphenyl)-7~{h}-purin-2-yl]amino]benzenesulfonamideHuman8019
CDK2CDKCMGC3rm6AB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamideHuman4357
CDK2CDKCMGC8h6tA(1r,3s)-3-{3-[(pyridin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl propan-2-ylcarbamateHuman14626
CSNK2A1 (CK2a1)CK2CMGC6q4qABbenzoic acidHuman11276
CSNK2A1 (CK2a1)CK2CMGC6q4qBBbenzoic acidHuman11278
CSNK2A1 (CK2a1)CK2CMGC6q4qBAbenzoic acidHuman11274
MAPK8 (JNK1)MAPKCMGC4ux9DBphosphoaminophosphonic acid-adenylate esterHuman4666
MAPK8 (JNK1)MAPKCMGC4yr8CB-Human6447
CLK1CLKCMGC6i5lCB3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10841
MAPK1 (Erk2)MAPKCMGC7nqqAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamideHuman13926
MAPK1 (Erk2)MAPKCMGC7nr9AA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamideHuman13932
CDK2CDKCMGC4fktABn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4322
CDK2CDKCMGC6p3wAA-Human11515
CDK2CDKCMGC2c5nAAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4063
CDK2CDKCMGC7m2fAA[(1r,4r)-4-{4-[4-(5-fluoro-2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-2-yl]-3,6-dihydropyridin-1(2h)-yl}cyclohexyl]acetic acidHuman13797
CSNK2A1 (CK2a1)CK2CMGC8c6mAA(5~{z})-5-[(3-methoxy-4-oxidanyl-phenyl)methylidene]-1,3-thiazolidine-2,4-dioneHuman15277
CDK2CDKCMGC1urcAA-Human4334
CDK2CDKCMGC6p3wCA-Human11514
MAPK1 (Erk2)MAPKCMGC8ao3AA2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14386
MAPK1 (Erk2)MAPKCMGC8aoiAA1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-oneHuman14387
MAPK1 (Erk2)MAPKCMGC8aodAA1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-oneHuman14417
CDK2CDKCMGC7ra5AB4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman13959
CDK2CDKCMGC3qtzAB4-{[4-amino-5-(3-fluorobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4337
CDK2CDKCMGC6rijAA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12623
CDK2CDKCMGC4ez7AstaurosporineHuman4240
MAPK8 (JNK1)MAPKCMGC4ux9CBphosphoaminophosphonic acid-adenylate esterHuman4647
MAPK8 (JNK1)MAPKCMGC4l7fABn-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamideHuman4637
CSNK2A1 (CK2a1)CK2CMGC8c6mAB(5~{z})-5-[(3-methoxy-4-oxidanyl-phenyl)methylidene]-1,3-thiazolidine-2,4-dioneHuman15278
MAPK1 (Erk2)MAPKCMGC8pt5ABphosphoaminophosphonic acid-adenylate esterHuman15301
MAPK8 (JNK1)MAPKCMGC2g01A6-chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4h-pyrazolo[3,4-b]quinolin-4-oneHuman4662
MAPK8 (JNK1)MAPKCMGC3o17A-Human4670
CDK2CDKCMGC1di8A4-[3-hydroxyanilino]-6,7-dimethoxyquinazolineHuman4577
CDK2CDKCMGC3rahAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman4438
CDK2CDKCMGC2uzlA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHuman3917
CDK2CDKCMGC3lfsAn-(6-chloro-5-phenyl-1h-indazol-3-yl)butanamideHuman4069
CDK2CDKCMGC4fklAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4134
CLK1CLKCMGC6q8kAA~{n}2-(3-morpholin-4-ylpropyl)pyrido[3,4-g]quinazoline-2,10-diamineHuman10902
CDK2CDKCMGC1oiqAn-[4-(2-methylimidazo[1,2-a]pyridin-3-yl)-2-pyrimidinyl]acetamideHuman4379
CDK2CDKCMGC4eomAAadenosine-5'-triphosphateHuman4528
CDK2CDKCMGC2w05ABn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHuman4256
CDK2CDKCMGC2vu3AA4-{[(2,6-dichlorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman4582
CDK2CDKCMGC6q4eAB6-iodanyl-7~{h}-purin-2-amineHuman11205
CDK2CDKCMGC1h00AA(2s)-1-[4-({6-[(2,6-difluorophenyl)amino]pyrimidin-4-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4484
CDK9CDKCMGC7nwkAn-((1r,3r)-3-(7-(4-fluoro-2-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-2-yl)cyclopentyl)acetamideHuman13951
CSNK2A2 (CK2a2)CK2CMGC6tguAB4-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxidanyl-benzoic acidHuman12445
DYRK2DYRKCMGC7akhA4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13615
DYRK2DYRKCMGC6hdpABscorzodihydrostilbene aHuman11573
DYRK1ADYRKCMGC7aj4AB4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amineHuman13588
CDK2CDKCMGC2c5xABhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman3892
CDK2CDKCMGC3ddqAAr-roscovitineHuman4477
CDK2CDKCMGC1vywCn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamideHuman4133
CDK2CDKCMGC2c5oCA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4414
CDK2CDKCMGC7zpcAA~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamideHuman14606
MAPK1 (Erk2)MAPKCMGC8ao9AC1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-oneHuman14401
CSNK2A1 (CK2a1)CK2CMGC8c6nAB(2~{z},5~{z})-5-[(4-methoxy-3-oxidanyl-phenyl)methylidene]-2-phenylimino-1,3-thiazolidin-4-oneHuman15279
MAPK8 (JNK1)MAPKCMGC2no3B2-({2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}amino)benzamideHuman4657
MAPK1 (Erk2)MAPKCMGC8ao9AB1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-oneHuman14390
MAPK1 (Erk2)MAPKCMGC8aojAA1-[(2~{s})-2-(5-methyl-3-pyridin-4-yl-1~{h}-pyrazol-4-yl)pyrrolidin-1-yl]propan-1-oneHuman14412
SRPK2SRPKCMGC7zkxABn-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamideHuman14616
CDK2CDKCMGC7s85A2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethoxy)benzoic acidHuman14425
CDK2CDKCMGC4i3zAadenosine-5'-diphosphateHuman4148
MAPK1 (Erk2)MAPKCMGC8aojAB-Human14418
MAPK1 (Erk2)MAPKCMGC8ao9AA1-(6,7-dihydro-4~{h}-[1,3]thiazolo[5,4-c]pyridin-5-yl)propan-1-oneHuman14420
MAPK1 (Erk2)MAPKCMGC8psyAamp phosphoramidateHuman15308
CDK2CDKCMGC7ug1AA8-(4-chloroanilino)naphthalene-1-sulfonic acidHuman14700
CDK2CDKCMGC7ug1AB8-(4-chloroanilino)naphthalene-1-sulfonic acidHuman14701
CDK2CDKCMGC4fkrAA(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman4149
CDK2CDKCMGC1h26A-Human4122
CSNK2A1 (CK2a1)CK2CMGC8qwyA4-[6-[(2-methoxy-5-propan-2-yloxy-phenyl)amino]pyrazin-2-yl]benzoic acidHuman15174
CDK2CDKCMGC5ieyAA4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHuman6566
MAPK8 (JNK1)MAPKCMGC3v3vA3,5,6,7-tetrahydroxy-2-(3,4-dihydroxyphenyl)-4h-chromen-4-oneHuman4653
CDK2CDKCMGC6gubA2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10764
CDK2CDKCMGC3qzhA4-methoxy-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3954
CDK2CDKCMGC2wmbA-Human4060
MAPK8 (JNK1)MAPKCMGC4yr8FB-Human6453
CDK2CDKCMGC3rmfAA4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman3873
CDK2CDKCMGC6q4iAA2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHuman11183
CDK2CDKCMGC6rijCA4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12625
MAPK14 (p38a)MAPKCMGC3hegAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5112
CDK2CDKCMGC3r6xAB4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4107
DYRK1ADYRKCMGC7ajsAA4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13599
DYRK1ADYRKCMGC7aj5AA4-(1-benzofuran-5-yl)pyridine-2,6-diamineHuman13602
CDK2CDKCMGC1e9hC2',3-dioxo-1,1',2',3-tetrahydro-2,3'-biindole-5'-sulfonic acidHuman4570
MAPK8 (JNK1)MAPKCMGC3vugA-Human4665
DYRK1ADYRKCMGC7aklA4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13589
CDK2CDKCMGC1b39Aadenosine-5'-triphosphateHuman4407
CDK2CDKCMGC5oo3AA1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHuman10569
CDK2CDKCMGC2v22C-Human4255
DYRK1ADYRKCMGC7akaAB4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13595
CDK2CDKCMGC3py1AB(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman4444
CDK2CDKCMGC2bpmA(2s)-n-[(3z)-5-cyclopropyl-3h-pyrazol-3-ylidene]-2-[4-(2-oxoimidazolidin-1-yl)phenyl]propanamideHuman4042
CDK12 (CRK7)CDKCMGC7nxkA(e)-n-[4-[(1r,3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]cyclohexyl]oxyphenyl]-4-(dimethylamino)but-2-enamideHuman13547
MAPK1 (Erk2)MAPKCMGC8aoaAA~{n}-pyridin-3-ylprop-2-enamideHuman14391
CDK2CDKCMGC2cciAadenosine-5'-triphosphateHuman4373
CDK2CDKCMGC1ke6An-methyl-{4-[2-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)hydrazino]phenyl}methanesulfonamideHuman4219
MAPK1 (Erk2)MAPKCMGC8ao5AA~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamideHuman14392
CDK2CDKCMGC1oguAB4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3935
CDK2CDKCMGC7b7sAA7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxideHuman13833
CDK2CDKCMGC2r3lAA3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4200
CDK9CDKCMGC8i0lA2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman15170
CDK2CDKCMGC6gukAA~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10773
CDK2CDKCMGC2w1hAn-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamideHuman4228
CDK2CDKCMGC4cfwAB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4557
CDK2CDKCMGC3my5CC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3929
CDK2CDKCMGC2uznA4-{5-[(1z)-1-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)ethyl]-2-furyl}benzenesulfonamideHuman4064
CSNK2A1 (CK2a1)CK2CMGC8qwzA4-[6-(6-propan-2-yloxyindol-1-yl)pyrazin-2-yl]benzoic acidHuman15176
DYRK1ADYRKCMGC7akbAB4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13604
CDK2CDKCMGC3sw7AAn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHuman4198
CDK2CDKCMGC4bcoAB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4051
CDK2CDKCMGC3lfnAn-[6-(4-hydroxyphenyl)-5-phenyl-1h-indazol-3-yl]butanamideHuman4330
CDK2CDKCMGC5ankA2,4,6-trioxo-1-phenyl-hexahydropyrimidine-5-carboxamideHuman6538
CSNK2A1 (CK2a1)CK2CMGC6q38ABbenzoic acidHuman11285
MAPK10 (JNK3)MAPKCMGC7s1nAA4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13958
CDK2CDKCMGC3rmfAB4-{[4-amino-5-(naphthalen-2-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4014
CDK2CDKCMGC3qtxAA4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4339
CDK2CDKCMGC1h1rAA6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman3906
MAPK1 (Erk2)MAPKCMGC8pt1AAphosphoaminophosphonic acid-adenylate esterHuman15302
MAPK1 (Erk2)MAPKCMGC8aogAB~{n}-(5-methyl-1,2-oxazol-3-yl)propanamideHuman14421
MAPK10 (JNK3)MAPKCMGC7s1nAB4-[5-(2-chloro-6-fluoroanilino)-6-methyl-1h-pyrazolo[3,4-b]pyridin-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13957
DYRK2DYRKCMGC7dhvA2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine-4-carboxylic acidHuman13974
CDK2CDKCMGC4cfnAB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4437
CDK2CDKCMGC4eomCAadenosine-5'-triphosphateHuman4481
CDK2CDKCMGC2wevAB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4580
DYRK1ADYRKCMGC7aj8AA4-(1-benzofuran-5-yl)pyridin-2-amineHuman13587
DYRK1ADYRKCMGC7akeA4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13601
GSK3BGSKCMGC7oy5AB~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHuman14119
MAPK1 (Erk2)MAPKCMGC7nr8AA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamideHuman13933
GSK3BGSKCMGC7oy5AA~{n}4-(3-cyclopropyl-1~{h}-pyrazol-5-yl)-~{n}2-(phenylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHuman14118
CDK2CDKCMGC7kjsA6-(difluoromethyl)-8-[(1r,2r)-2-hydroxy-2-methylcyclopentyl]-2-{[1-(methylsulfonyl)piperidin-4-yl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman13740
DYRK2DYRKCMGC7dhhA[9-(azetidin-3-ylmethylsulfanyl)-2,7-dimethoxy-acridin-4-yl]methanolHuman13975
CDK2CDKCMGC7b7sAB7-(3-(trifluoromethyl)-1h-pyrazol-4yl)-3,8,10,11-tetrahydropyrazolo[4,3-f]thiopyrano[3,4-c]quinoline 9-oxideHuman13834
CDK2CDKCMGC1pxlAB-Human4074
CDK2CDKCMGC3eocA5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman4390
CSNK2A1 (CK2a1)CK2CMGC8c6lAB5-azanyl-3-[(~{z})-1-cyano-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]-3~{h}-pyrazole-4-carbonitrileHuman15280
GSK3BGSKCMGC5t31B(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9564
MAPK1 (Erk2)MAPKCMGC8aohAB~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamideHuman14404
MAPK1 (Erk2)MAPKCMGC8pt3ABphosphoaminophosphonic acid-adenylate esterHuman15305
SRPK1SRPKCMGC3begAphosphoaminophosphonic acid-adenylate esterHuman9472
CDK2CDKCMGC4bckCD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4080
CDK2CDKCMGC7mkxA2-[(5-bromo-2-{4-[(cyanomethyl)sulfamoyl]anilino}pyrimidin-4-yl)amino]-6-fluorobenzamideHuman14490
CDK2CDKCMGC1jvpP13-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazoleHuman3919
MAPK8 (JNK1)MAPKCMGC4awiABn-(1,1-dioxidotetrahydro-2h-thiopyran-4-yl)-4-[2-(1-methylethyl)-1h-pyrrolo[2,3-b]pyridin-4-yl]benzenesulfonamideHuman4634
CDK2CDKCMGC2vtoABn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHuman3946
CDK2CDKCMGC3rniAA3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman3993
CDK2CDKCMGC3ralAA4-{[4-amino-5-(3-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4017
CDK2CDKCMGC4eojABadenosine-5'-triphosphateHuman4015
CDK2CDKCMGC3py1AA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman4361
CDK1 (CDC2)CDKCMGC4y72AA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4610
MAPK8 (JNK1)MAPKCMGC6zr5Aphosphoaminophosphonic acid-adenylate esterHuman12984
CDK2CDKCMGC6q4iAB2-[4-[(2-oxidanylidene-3~{h}-pyridin-4-yl)oxy]phenyl]ethanoic acidHuman11197
CDK2CDKCMGC1oiuCA3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4524
DYRK1ADYRKCMGC6s17AA~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11369
MAPK7 (Erk5)MAPKCMGC9ltaA4-[5-chloranyl-2-[[3-[(dimethylamino)methyl]phenyl]amino]pyrimidin-4-yl]-~{n}-morpholin-4-yl-thiophene-2-carboxamideHuman15439
CDKL5CDKLCMGC9epuA~{n}-[5-[(5-propan-2-yl-1,3-oxazol-2-yl)methylsulfanyl]-1,3-thiazol-2-yl]piperidine-4-carboxamideHuman15440
CLK3CLKCMGC29moA3^{3}-methoxy-1^{7}-(2-(2-(4-methylpiperazin-1-yl)ethoxy)ethoxy)-4,7,10-trioxa-2-aza-1(4,6)-quinolina-3(1,2)-benzenacyclodecaphane-1^{3}-carbonitrileHuman15441
CLK3CLKCMGC29mpA1^{7}-methoxy-4,7,10-trioxa-2-aza-1(4,6)-quinolina-3(1,2)-benzenacyclodecaphane-1^{3}-carbonitrileHuman15442
CLK3CLKCMGC9ez3A1-(5-~{tert}-butyl-2-quinolin-6-yl-pyrazol-3-yl)-3-[3-(4-morpholin-4-yl-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl)phenyl]ureaHuman15443
CDK16 (PCTAIRE1)CDKCMGC9r2iCphosphothiophosphoric acid-adenylate esterHuman15481
CDK2CDKCMGC3r7yAA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamideHuman4476
CDK2CDKCMGC4ii5CAadenosine-5'-diphosphateHuman4530
CDK2CDKCMGC1oiyCA4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4465
CDK2CDKCMGC1pxiAB-Human3924
CDK2CDKCMGC5andA2-imidazol-1-yl-1h-benzimidazoleHuman6543
CDK2CDKCMGC4bcoCB2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4018
MAPK1 (Erk2)MAPKCMGC8u8jA(4m)-4-{(4r)-3-[(2s)-2-methylbutyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(1-methyl-1h-pyrazol-5-yl)pyrimidin-2-amineHuman15224
MAPK1 (Erk2)MAPKCMGC8u8kA(4m)-4-{(4s)-3-[(2-chloropyridin-3-yl)methyl][1,2,4]triazolo[4,3-a]pyridin-7-yl}-n-(oxan-4-yl)pyrimidin-2-amineHuman15225
MAPK1 (Erk2)MAPKCMGC9tyhAadenosine-5'-diphosphateHuman15552
MAPK1 (Erk2)MAPKCMGC9tygBadenosine-5'-diphosphateHuman15553
MAPK1 (Erk2)MAPKCMGC9tyiA-Human15554
CSNK2A2 (CK2a2)CK2CMGC9ihiAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman15555
CSNK2A2 (CK2a2)CK2CMGC9fbiABnicotinic acidHuman15556
CSNK2A2 (CK2a2)CK2CMGC9r57AA5,6-dibromobenzotriazoleHuman15557
CSNK2A2 (CK2a2)CK2CMGC9r5cAB3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman15558
CSNK2A2 (CK2a2)CK2CMGC9hk5AA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman15559
CSNK2A2 (CK2a2)CK2CMGC9hk5AB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman15560
DYRK1ADYRKCMGC9ft2A3-[[[4-[(3-cyclobutyl-1~{h}-pyrazol-5-yl)amino]furo[3,2-d]pyrimidin-2-yl]amino]methyl]benzamideHuman15583
MAPK11 (p38b)MAPKCMGC8ygwA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman15234
CDK7CDKCMGC8p4zAA2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHuman14796
DYRK1ADYRKCMGC9ft6A~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)furo[3,2-d]pyrimidine-2,4-diamineHuman15584
DYRK1ADYRKCMGC9ft4A~{n}4-(5-cyclopropyl-1~{h}-pyrazol-3-yl)-~{n}2-(phenylmethyl)furo[3,2-d]pyrimidine-2,4-diamineHuman15585
DYRK1ADYRKCMGC8yevAcoumestrolHuman15586
DYRK1ADYRKCMGC9fpxAcurcuminHuman15587
DYRK1ADYRKCMGC7fhtAC(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman15588
DYRK1ADYRKCMGC9fufA3-[[[4-[(3-cyclopropyl-1~{h}-pyrazol-5-yl)amino]thieno[3,2-d]pyrimidin-2-yl]amino]methyl]benzamideHuman15589
DYRK1ADYRKCMGC9ft3A~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHuman15590
DYRK1ADYRKCMGC9ykoA(5,6-dihydroxy-1,3-benzothiazol-2-yl)(3,4-dihydroxyphenyl)methanoneHuman15591
CDK7CDKCMGC8p4zAB2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHuman14797
CDK2CDKCMGC8uv0AA1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-olHuman15238
CLK2CLKCMGC3nr9A(5z)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman1927
CDK2CDKCMGC3r9nAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3885
CDK2CDKCMGC8uv0AB1-{(4m)-4-[2-{[1-(cyclopropanesulfonyl)piperidin-4-yl]amino}-5-(trifluoromethyl)pyrimidin-4-yl]-1h-pyrazol-1-yl}-2-methylpropan-2-olHuman15239
CDK1 (CDC2)CDKCMGC4yc6AA-Human4607
MAPK1 (Erk2)MAPKCMGC5v61AA-Human8265
CDK2CDKCMGC4fkvAB(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHuman3939
CSNK2A1 (CK2a1)CK2CMGC5otoBB2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9611
CDK2CDKCMGC3qx2AB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamideHuman4297
CDK2CDKCMGC1gy3Cadenosine-5'-triphosphateHuman4445
CSNK2A1 (CK2a1)CK2CMGC7a4bAB 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13165
CSNK2A1 (CK2a1)CK2CMGC7l1xAA(2~{z})-6-[[2,6-bis(chloranyl)phenyl]methylsulfonyl]-2-[[4-oxidanyl-3-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methylidene]-4~{h}-1,4-benzothiazin-3-oneHuman13847
MAPK1 (Erk2)MAPKCMGC6nbsAA-Human11510
CDK2CDKCMGC5jq8A(3s,4s)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman7417
CDK2CDKCMGC3rm6AA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitro-4-{[2-(piperazin-1-yl)ethyl]amino}benzamideHuman4262
CDK2CDKCMGC7qhlAA5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidineHuman14275
CDK2CDKCMGC3qqjAB2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4204
CDK2CDKCMGC3qqgAB4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4310
CDK2CDKCMGC3qqfAA5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4211
CDK2CDKCMGC2iw8CBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4350
CDK7CDKCMGC8pyrAB-Human15253
CDK2CDKCMGC2c4gC(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHuman4453
CDK2CDKCMGC1okwA-Human4314
CDK2CDKCMGC1w0xCAolomoucineHuman4537
CLK3CLKCMGC6ft7AB3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9903
CLK3CLKCMGC6z52BB11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12626
CSNK2A1 (CK2a1)CK2CMGC7bu4AA4-(6-aminocarbonyl-8-oxidanylidene-9-phenyl-7h-purin-2-yl)benzoic acidHuman13486
CLK3CLKCMGC6z53AA6-(2-methoxyethoxy)-11,15-dimethyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12300
MAPK1 (Erk2)MAPKCMGC8ao8AB1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-oneHuman14405
CSNK2A1 (CK2a1)CK2CMGC5mp8BAadenosine-5'-diphosphateHuman7695
CDK2CDKCMGC6gukAB~{n}2-[(1~{r},2~{s})-2-azanylcyclohexyl]-~{n}6-(3-chlorophenyl)-9-ethyl-purine-2,6-diamineHuman10768
CSNK2A1 (CK2a1)CK2CMGC1jwhB-Human5524
CSNK2A1 (CK2a1)CK2CMGC5otiAB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9667
CSNK2A1 (CK2a1)CK2CMGC5moeBBadenosine-5'-diphosphateHuman7687
MAPK1 (Erk2)MAPKCMGC8ao8AA1-[(2~{r})-2-(3-methylimidazol-4-yl)piperidin-1-yl]propan-1-oneHuman14410
CSNK2A1 (CK2a1)CK2CMGC3owkAA7-chloro-10-methyl-11h-benzo[g]pyrido[4,3-b]indol-3-olHuman5467
CSNK2A1 (CK2a1)CK2CMGC3q9yAA1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5493
CSNK2A1 (CK2a1)CK2CMGC5oniBA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9458
CSNK2A1 (CK2a1)CK2CMGC5cvhAAadenosine-5'-diphosphateHuman6896
CLK3CLKCMGC3rawBA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman1824
MAPK1 (Erk2)MAPKCMGC8ao2AA~{n}-(1~{h}-indazol-5-ylmethyl)propanamideHuman14415
GSK3BGSKCMGC9hv3A2-oxidanylidene-~{n}-[3-(4-phenylpiperazin-1-yl)propyl]-6-pyridin-3-yl-3~{h}-benzimidazole-1-carboxamideHuman15794
GSK3BGSKCMGC9x2yAA-Human15795
GSK3BGSKCMGC9hulA~{n}-[3-[4-[2,3-bis(chloranyl)phenyl]piperazin-1-yl]propyl]-2-oxidanylidene-6-pyridin-3-yl-3~{h}-benzimidazole-1-carboxamideHuman15796
GSK3BGSKCMGC9fr6A3-[[[4-[(3-cyclopropyl-1~{h}-pyrazol-5-yl)amino]thieno[3,2-d]pyrimidin-2-yl]amino]methyl]benzamideHuman15797
CLK3CLKCMGC6ytyAA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12409
GSK3BGSKCMGC9hukA~{n}-[4-[4-[2,3-bis(chloranyl)phenyl]piperazin-1-yl]butyl]-2-oxidanylidene-6-pyridin-3-yl-3~{h}-benzimidazole-1-carboxamideHuman15800
GSK3BGSKCMGC9fr7A~{n}4-(5-cyclopropyl-1~{h}-pyrazol-3-yl)-~{n}2-(phenylmethyl)furo[3,2-d]pyrimidine-2,4-diamineHuman15801
GSK3BGSKCMGC9x2yAB-Human15802
CDK2CDKCMGC2vtnA4-(acetylamino)-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4027
MAPK7 (Erk5)MAPKCMGC7pusAA4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamideHuman14218
MAPK7 (Erk5)MAPKCMGC6hknAA[2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanoneHuman10918
MAPK7 (Erk5)MAPKCMGC4ic7Dphosphoaminophosphonic acid-adenylate esterHuman391
CLK3CLKCMGC2wu7AAethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman1828
GSK3BGSKCMGC9fr9A3-[[[4-[(3-cyclobutyl-1~{h}-pyrazol-5-yl)amino]furo[3,2-d]pyrimidin-2-yl]amino]methyl]benzamideHuman15798
GSK3BGSKCMGC9x2qAA-Human15799
CDK2CDKCMGC2c6tC4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman3994
MAPK1 (Erk2)MAPKCMGC4g6nAA3-(4-chlorophenyl)-4,5,6,7-tetrahydro-1h-indazoleHuman2609
GSK3BGSKCMGC9x2xAA-Human15803
GSK3BGSKCMGC9x2vAA-Human15804
GSK3BGSKCMGC9x2uAB-Human15805
GSK3BGSKCMGC9x2vAB-Human15806
GSK3BGSKCMGC9x2wA-Human15807
GSK3BGSKCMGC9x2xAB-Human15808
CDK2CDKCMGC2xmyAB4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHuman3985
CLK1CLKCMGC6i5hAA5-(1-methylpyrazol-4-yl)-3-(3-phenoxyphenyl)furo[3,2-b]pyridineHuman10848
DYRK1ADYRKCMGC7aj4AA4-(4-chloranyl-3-methoxy-phenyl)pyridin-2-amineHuman13605
CDK2CDKCMGC9qjjBots964Human15914
CDK2CDKCMGC13gkAC-Human15915
CDK2CDKCMGC9nyrAB-Human15916
CDK2CDKCMGC9et1AA4-iodanylbenzamideHuman15917
CDK2CDKCMGC9glaAA7-dimethylphosphoryl-3-[2-[[(3~{s})-6,6-dimethylpiperidin-3-yl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]-1~{h}-indole-6-carbonitrileHuman15918
CDK2CDKCMGC9fr2A4-[[6-(cyclohexylmethoxy)-7~{h}-purin-2-yl]amino]benzenesulfonyl fluorideHuman15919
CDK2CDKCMGC9eswAD-Human15920
CDK2CDKCMGC9eskAB(4-bromo-2-oxopyridin-1(2h)-yl)acetic acidHuman15913
CDK2CDKCMGC9esjAA2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman15953
CDK2CDKCMGC9eswAB(4-bromanylpyridin-2-yl)methanolHuman15954
CDK2CDKCMGC9esuAB4-bromanyl-2-(methoxymethyl)pyridineHuman15955
CDK2CDKCMGC9esoAB-Human15956
MAPK1 (Erk2)MAPKCMGC5bveAA2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6029
CDK2CDKCMGC7s7aAA2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14427
CDK2CDKCMGC9esyAA4-bromanyl-1,8-naphthyridineHuman15930
CDK2CDKCMGC9et1AB4-iodanylbenzamideHuman15951
CDK2CDKCMGC9etpAA4-bromo-1h-pyrazoleHuman15952
CDK2CDKCMGC2r3kAB3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman3876
CDK2CDKCMGC7sa0AA2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acidHuman14428
CDK2CDKCMGC7sa0AB2-{[(3r)-2,3,4,9-tetrahydro-1h-carbazol-3-yl]amino}-5-(trifluoromethyl)benzoic acidHuman14429
CDK2CDKCMGC7s84AB2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14432
CDK2CDKCMGC9nyqA4-({4-[(1s,4s)-4-hydroxy-4-methylcyclohexyl]-5-(trifluoromethyl)pyrimidin-2-yl}amino)-n,3-dimethylbenzene-1-sulfonamideHuman15957
CDK2CDKCMGC9gp3A(3~{s})-~{n}-ethyl-3-[[9-ethyl-2-[[(2~{r},3~{s})-2-oxidanylpentan-3-yl]amino]purin-6-yl]amino]pyrrolidine-1-sulfonamideHuman15958
CDK2CDKCMGC9esqAA4-bromanyl-2-oxidanyl-benzoic acidHuman15959
CSNK2A1 (CK2a1)CK2CMGC7qgcAA5,6-dibromobenzotriazoleHuman14433
MAPK1 (Erk2)MAPKCMGC5bvdAB2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-oneHuman6028
CDK2CDKCMGC7s9xAA2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acidHuman14430
CDK9CDKCMGC32awA4-[[[6-[5-chloranyl-2-[[4-[[(2~{r})-1-methoxypropan-2-yl]amino]phenyl]amino]pyridin-4-yl]pyridin-2-yl]amino]methyl]oxane-4-carbonitrileHuman15994
CDK13 (CHED)CDKCMGC7nxjAn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman13544
MAPK7 (Erk5)MAPKCMGC6hknAB[2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanoneHuman10919
CSNK2A1 (CK2a1)CK2CMGC9qsrA5-[7-[(3-chloranyl-4-phenyl-phenyl)methylamino]heptylamino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman16063
CSNK2A1 (CK2a1)CK2CMGC9s6gABphosphoaminophosphonic acid-adenylate esterHuman16064
CSNK2A1 (CK2a1)CK2CMGC9qssA5-[8-[(3-chloranyl-4-phenyl-phenyl)methylamino]octylamino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman16065
CSNK2A1 (CK2a1)CK2CMGC9fblABnicotinic acidHuman16066
CSNK2A1 (CK2a1)CK2CMGC9rcyAB-Human16067
CSNK2A1 (CK2a1)CK2CMGC9fbmAAnicotinic acidHuman16068
CSNK2A1 (CK2a1)CK2CMGC9s77AAnicotinic acidHuman16069
CSNK2A1 (CK2a1)CK2CMGC9s7iABphosphoaminophosphonic acid-adenylate esterHuman16070
MAPK3 (Erk1)MAPKCMGC9uuxBphosphoaminophosphonic acid-adenylate esterHuman16039
MAPK3 (Erk1)MAPKCMGC9uurBphosphoaminophosphonic acid-adenylate esterHuman16040
MAPK3 (Erk1)MAPKCMGC9tu0A-Human16041
CSNK2A1 (CK2a1)CK2CMGC9qrhA5-[[(3~{e})-3-[4-[2-(3,4-dichlorophenyl)ethylamino]-4-oxidanylidene-butanoyl]iminopropyl]amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman16061
CSNK2A1 (CK2a1)CK2CMGC7i85AA5-(ethylamino)benzo[c][2,6]naphthyridine-8-carboxamideHuman16062
MAPK8 (JNK1)MAPKCMGC4yr8CA-Human6449
CSNK2A1 (CK2a1)CK2CMGC9rfnAA-Human16071
CSNK2A1 (CK2a1)CK2CMGC9rcxAB-Human16072
DYRK2DYRKCMGC9kqyA-Human16123
DYRK2DYRKCMGC9mc0A[2-[[4-(1,3-benzothiazol-5-yl)-5-fluoranyl-pyrimidin-2-yl]amino]-1,3-thiazol-5-yl]-piperazin-1-yl-methanoneHuman16124
CDK2CDKCMGC3pxrAA-Human3941
CDK2CDKCMGC7s7aAB2-{[2-(2h-indazol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14426
CDK2CDKCMGC2clxAA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3909
CSNK2A1 (CK2a1)CK2CMGC5h8eA~{n}-[2-[2-azanylethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman6409
CSNK2A1 (CK2a1)CK2CMGC5otrABadenosine-5'-triphosphateHuman9634
MAPK10 (JNK3)MAPKCMGC4x21An-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamideHuman6240
CDK2CDKCMGC4eojAAadenosine-5'-triphosphateHuman4271
CDK2CDKCMGC4eomCBadenosine-5'-triphosphateHuman4423
CDK2CDKCMGC3r71AA4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3962
CDK2CDKCMGC1pxoAC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4546
CSNK2A1 (CK2a1)CK2CMGC6rffAA(~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-nitro-4-oxidanyl-phenyl)prop-2-enamideHuman12146
MAPK1 (Erk2)MAPKCMGC8aodAB1-(3-oxidanyl-2~{h}-quinoxalin-1-yl)propan-1-oneHuman14388
CSNK2A1 (CK2a1)CK2CMGC6horAB(~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-oneHuman11663
CSNK2A1 (CK2a1)CK2CMGC1pjkABphosphoaminophosphonic acid-adenylate esterHuman5410
CSNK2A1 (CK2a1)CK2CMGC6l23AB(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman13454
CDK2CDKCMGC4eopCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4061
CDK2CDKCMGC3r8lAB(5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4523
CDK2CDKCMGC6athAB-Human10570
CSNK2A1 (CK2a1)CK2CMGC3ngaAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5515
CSNK2A1 (CK2a1)CK2CMGC5mmfAB(3-chloranyl-4-phenyl-phenyl)methyl-propyl-azaniumHuman7666
CSNK2A1 (CK2a1)CK2CMGC3qa0BA-Human5495
CSNK2A1 (CK2a1)CK2CMGC5clpBA2-(3,4-dichlorophenyl)ethanamineHuman6909
CSNK2A1 (CK2a1)CK2CMGC5n9kAA1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diolHuman9682
CSNK2A1 (CK2a1)CK2CMGC3u87Bphosphoaminophosphonic acid-adenylate esterHuman5513
MAPK12 (p38g)MAPKCMGC6unaAB-Human11900
CSNK2A1 (CK2a1)CK2CMGC6rb1AB(~{e})-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)-~{n}-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]prop-2-enamideHuman12142
CSNK2A1 (CK2a1)CK2CMGC6hotAB(2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enalHuman11670
CSNK2A1 (CK2a1)CK2CMGC5t1hAA7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman8685
MAPK12 (p38g)MAPKCMGC6unaBA-Human11901
CDK2CDKCMGC3qqgAA4-chloro-2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4130
MAPK1 (Erk2)MAPKCMGC5bujAA4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-oneHuman2560
CDK2CDKCMGC4bckCC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4029
CDK2CDKCMGC7qhlAB5-(2-amino-1-ethyl)thio-3-cyclobutyl-7-[4-(pyrazol-1-yl)benzyl]amino-1(2)h-pyrazolo[4,3-d]pyrimidineHuman14276
CDK2CDKCMGC4eolCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4521
CDK2CDKCMGC6q4kAC-Human11189
CDK1 (CDC2)CDKCMGC4yc6EB-Human4614
CDK7CDKCMGC1ua2Cadenosine-5'-triphosphateHuman542
CDK7CDKCMGC7b5oJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13278
MAPK1 (Erk2)MAPKCMGC8aocAA~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamideHuman14409
MAPK1 (Erk2)MAPKCMGC2y9qAAphosphoaminophosphonic acid-adenylate esterHuman2626
CDK2CDKCMGC7zpcAB~{n}-(1-methylpyrazol-4-yl)-5-phenyl-pyrazolo[1,5-a]pyrimidine-7-carboxamideHuman14607
CDK7CDKCMGC7nvr8-Human13543
CDK2CDKCMGC1fq1Badenosine-5'-triphosphateHuman4266
CDK2CDKCMGC4cfvAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman4180
MAPK10 (JNK3)MAPKCMGC4h36AB-Human3461
CDK8CDKCMGC5hnbAB[6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanoneHuman6563
MAPK14 (p38a)MAPKCMGC6hwuAB-Human11249
MAPK14 (p38a)MAPKCMGC4zthAB6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazineHuman6707
MAPK8 (JNK1)MAPKCMGC1ukhA-Human4628
CSNK2A1 (CK2a1)CK2CMGC4md9G-Human5483
CSNK2A1 (CK2a1)CK2CMGC6horAA(~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-oneHuman11668
CSNK2A1 (CK2a1)CK2CMGC6ypnBBadenosine-5'-diphosphateHuman12436
CDK5CDKCMGC7vdqA2-[[7-[[2-fluoranyl-4-[3-(hydroxymethyl)pyrazol-1-yl]phenyl]amino]-1,6-naphthyridin-2-yl]-(1-methylpiperidin-4-yl)amino]ethanoic acidHuman14144
CDK5CDKCMGC7vdsAA5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHuman14148
MAPK8 (JNK1)MAPKCMGC2h96A5-cyano-n-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamideHuman4655
CDK5CDKCMGC1unhA(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2780
CDK5CDKCMGC3o0gA-Human2782
CDK5CDKCMGC1unlB-Human2790
CDK2CDKCMGC7rxoAB2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acidHuman14351
CSNK2A1 (CK2a1)CK2CMGC5cshAAadenosine-5'-triphosphateHuman6918
CSNK2A1 (CK2a1)CK2CMGC5oszAA2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azaniumHuman9669
CSNK2A1 (CK2a1)CK2CMGC5kwhAB~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman8619
CDK2CDKCMGC7uxkA-Human14570
CDK2CDKCMGC7uxiAA-Human14571
CDK2CDKCMGC7rxoAA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(methoxycarbonyl)benzoic acidHuman14352
MAPK8 (JNK1)MAPKCMGC4qtdAA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman4651
MAPK8 (JNK1)MAPKCMGC4g1wAmethyl 7-fluoro-3-{4-[(2-hydroxyethyl)sulfonyl]benzyl}-4-oxo-1-phenyl-1,4-dihydroquinoline-2-carboxylateHuman4631
MAPK8 (JNK1)MAPKCMGC2xs0Aphosphoaminophosphonic acid-adenylate esterHuman4629
MAPK8 (JNK1)MAPKCMGC2gmxBn-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-bromo-2,5-dimethoxyphenyl)acetamideHuman4638
CDK2CDKCMGC7uxiAB-Human14572
CSNK2A1 (CK2a1)CK2CMGC7quxABadenosine-5'-diphosphateHuman14573
CSNK2A1 (CK2a1)CK2CMGC5mo6BB-Human7652
CSNK2A1 (CK2a1)CK2CMGC7quxAAadenosine-5'-diphosphateHuman14574
CSNK2A1 (CK2a1)CK2CMGC6tlrAA4,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13089
CSNK2A1 (CK2a1)CK2CMGC5m4cAB3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acidHuman7403
MAPK8 (JNK1)MAPKCMGC1ukiA2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHuman4630
CSNK2A1 (CK2a1)CK2CMGC7b8iAA-Human13263
MAPK8 (JNK1)MAPKCMGC4yr8EA-Human6451
CSNK2A1 (CK2a1)CK2CMGC8aekAAadenosine-5'-triphosphateHuman14442
CSNK2A1 (CK2a1)CK2CMGC6hnwABcoumestrolHuman11521
MAPK8 (JNK1)MAPKCMGC6zr5Bphosphoaminophosphonic acid-adenylate esterHuman12985
MAPK8 (JNK1)MAPKCMGC4hysAtrans-4-{[4-(1h-indazol-1-yl)pyrimidin-2-yl]amino}cyclohexanolHuman4672
CSNK2A1 (CK2a1)CK2CMGC7zydAAadenosine-5'-triphosphateHuman14438
CSNK2A1 (CK2a1)CK2CMGC7zy0ABadenosine-5'-diphosphateHuman14439
CSNK2A1 (CK2a1)CK2CMGC7zyoABadenosine-5'-triphosphateHuman14440
CSNK2A1 (CK2a1)CK2CMGC7zyrABadenosine-5'-triphosphateHuman14456
CSNK2A1 (CK2a1)CK2CMGC5cu0ABn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7293
CSNK2A1 (CK2a1)CK2CMGC5cshBAadenosine-5'-triphosphateHuman6923
MAPK8 (JNK1)MAPKCMGC3vuiA-Human4652
CSNK2A1 (CK2a1)CK2CMGC7zy2AAadenosine-5'-triphosphateHuman14443
CSNK2A1 (CK2a1)CK2CMGC7zyrAAadenosine-5'-triphosphateHuman14444
CSNK2A1 (CK2a1)CK2CMGC8aecACadenosine-5'-triphosphateHuman14446
CSNK2A1 (CK2a1)CK2CMGC8aekABadenosine-5'-triphosphateHuman14447
CSNK2A1 (CK2a1)CK2CMGC7zy0AAadenosine-5'-diphosphateHuman14452
CSNK2A1 (CK2a1)CK2CMGC8aecAAadenosine-5'-triphosphateHuman14455
MAPK8 (JNK1)MAPKCMGC4ux9ABphosphoaminophosphonic acid-adenylate esterHuman4646
CDK2CDKCMGC7vduAB[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14137
CDK2CDKCMGC1gz8AB1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHuman3956
CDK2CDKCMGC4eojCAadenosine-5'-triphosphateHuman4041
CSNK2A1 (CK2a1)CK2CMGC7zyoAAadenosine-5'-triphosphateHuman14448
MAPK8 (JNK1)MAPKCMGC2xrwACphosphoaminophosphonic acid-adenylate esterHuman4660
MAPK8 (JNK1)MAPKCMGC3vudA-Human4664
MAPK14 (p38a)MAPKCMGC3fmnAA6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman5196
CDK2CDKCMGC4fkrAB(8z)-8-{[(2,2-dioxido-1,3-dihydro-2-benzothiophen-5-yl)amino]methylidene}-6,8-dihydro-7h-[1,3]thiazolo[5,4-e]indol-7-oneHuman4535
CDK2CDKCMGC3eidAA(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4386
CSNK2A1 (CK2a1)CK2CMGC7l1xAB(2~{z})-6-[[2,6-bis(chloranyl)phenyl]methylsulfonyl]-2-[[4-oxidanyl-3-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenyl]methylidene]-4~{h}-1,4-benzothiazin-3-oneHuman13848
CSNK2A1 (CK2a1)CK2CMGC6a1cAB5-bromanyl-2-methoxy-4-[(e)-(3-methylsulfanyl-5-phenyl-1,2,4-triazol-4-yl)iminomethyl]phenolHuman11286
CSNK2A1 (CK2a1)CK2CMGC5ct0BA3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-olHuman7288
CSNK2A1 (CK2a1)CK2CMGC3q9wAA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5436
DYRK1ADYRKCMGC2wo6AAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3758
CDK2CDKCMGC6p3wAB-Human11517
CDK2CDKCMGC4bcmAB4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4203
CDK2CDKCMGC1h24A-Human4199
CDK2CDKCMGC1oguCB4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman4560
CSNK2A1 (CK2a1)CK2CMGC7zydABadenosine-5'-triphosphateHuman14450
MAPK7 (Erk5)MAPKCMGC4zsjAB3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6585
MAPK7 (Erk5)MAPKCMGC4ic7Aphosphoaminophosphonic acid-adenylate esterHuman392
MAPK14 (p38a)MAPKCMGC2lgcA4-Human5067
CDK2CDKCMGC4bghAB4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHuman4509
CSNK2A1 (CK2a1)CK2CMGC8aecABadenosine-5'-triphosphateHuman14451
CSNK2A1 (CK2a1)CK2CMGC3bqcAB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5490
MAPK7 (Erk5)MAPKCMGC5o7iAB4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamideHuman9994
MAPK7 (Erk5)MAPKCMGC5byyAB2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman6587
MAPK7 (Erk5)MAPKCMGC4zslA3-amino-5-[(4-chlorophenyl)amino]-n-[(1s)-1-phenylethyl]-1h-1,2,4-triazole-1-carboxamideHuman6586
MAPK7 (Erk5)MAPKCMGC4zsgAB3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6584
CDK16 (PCTAIRE1)CDKCMGC5g6vA4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamideHuman7273
CDK2CDKCMGC2c6iA4-{[5-(cyclohexylmethoxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6774
CDK2CDKCMGC2wfyCA-Human4329
CDK2CDKCMGC3r8lAA(5r)-5-tert-butyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4186
CSNK2A1 (CK2a1)CK2CMGC3mb7AAnaphtho[2,1-b:7,8-b']difuran-2,9-dicarboxylic acidHuman5448
CSNK2A1 (CK2a1)CK2CMGC5mmrAA~{n}'-[(3-chloranyl-4-phenyl-phenyl)methyl]butane-1,4-diamineHuman7668
CSNK2A1 (CK2a1)CK2CMGC6teiBA3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12460
CSNK2A1 (CK2a1)CK2CMGC5zn2AA-Human10698
CSNK2A1 (CK2a1)CK2CMGC5n9kAB1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diolHuman9695
CDK2CDKCMGC1gihA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-pyridin-2-yl-ureaHuman3922
CSNK2A1 (CK2a1)CK2CMGC3rpsB-Human5450
CLK3CLKCMGC2exeAB-Human1819
CLK3CLKCMGC6rctBA4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11128
CLK3CLKCMGC6z55AB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12298
CLK3CLKCMGC6yu1cA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12405
CDK2CDKCMGC1f5qCA-Human4281
CLK3CLKCMGC6ytyAB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12406
CLK3CLKCMGC6ytwAB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12407
CDK2CDKCMGC8erdAA(2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanoneHuman14949
CSNK2A1 (CK2a1)CK2CMGC5kwhBA~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman8618
MAPK14 (p38a)MAPKCMGC3hv7A1-[1-(3-aminophenyl)-3-tert-butyl-1h-pyrazol-5-yl]-3-naphthalen-1-ylureaHuman5223
CDK2CDKCMGC8ernAAn,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamideHuman14948
CDK2CDKCMGC8ernABn,3-dimethyl-4-({7-[(2s)-2-methylpyrrolidine-1-carbonyl]quinazolin-2-yl}amino)benzene-1-sulfonamideHuman14950
CDK2CDKCMGC3pxfAA8-anilino-1-naphthalene sulfonateHuman4047
CDK2CDKCMGC8erdAB(2-{[1-(methanesulfonyl)piperidin-4-yl]amino}quinazolin-7-yl)[(2s)-2-methylpyrrolidin-1-yl]methanoneHuman14951
SRPK2SRPKCMGC7zkxAAn-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamideHuman14617
MAPK8 (JNK1)MAPKCMGC2no3A2-({2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}amino)benzamideHuman4640
SRPK2SRPKCMGC5myvCA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7580
CDK2CDKCMGC4eoqCAadenosine-5'-triphosphateHuman4004
CDK2CDKCMGC5fp5A4-fluorobenzoic acidHuman6285
CDK2CDKCMGC2vtjA4-[(6-chloropyrazin-2-yl)amino]benzenesulfonamideHuman3959
CDK2CDKCMGC7s9xAB2-[(9h-carbazol-3-yl)amino]-5-(trifluoromethyl)benzoic acidHuman14431
CDK2CDKCMGC6gufCn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman10762
CDK2CDKCMGC2uzbAD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman3866
CDK2CDKCMGC6gvaAB5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman11204
CDK2CDKCMGC2c6kA4-{[5-(cyclohexylamino)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman6773
CDK2CDKCMGC1pkdA7-hydroxystaurosporineHuman4170
CDK2CDKCMGC6q48AC4-iodanyl-3~{h}-pyridin-2-oneHuman11196
CDK2CDKCMGC6q3bAA4-iodopyrazoleHuman11177
CDK2CDKCMGC1h25C-Human4112
CDK2CDKCMGC3pj8AA(2r)-2-{[7-(benzylamino)-3-(propan-2-yl)-1h-pyrazolo[4,3-d]pyrimidin-5-yl]amino}butan-1-olHuman4375
CDK2CDKCMGC2c5xAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4312
CDK2CDKCMGC3sw7ABn~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethyl-2-nitrobenzene-1,4-diamineHuman4584
CDK2CDKCMGC3rahAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman4206
CSNK2A1 (CK2a1)CK2CMGC8pvoA2-[1-(1,3-benzothiazol-6-ylsulfonyl)piperidin-4-yl]-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman14976
MAPK1 (Erk2)MAPKCMGC5v62AB5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman8262
DYRK1ADYRKCMGC4mq2DAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3757
CDK2CDKCMGC1pxmAA3-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-ylamino]-phenolHuman3944
CDK2CDKCMGC4bghAA4-((5-bromo-4-(prop-2-yn-1-ylamino)pyrimidin-2-yl)amino)benzenesulfonamideHuman4073
CDK2CDKCMGC3bhvCA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4353
CDK2CDKCMGC2x1nCB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4062
CDK8CDKCMGC5fgkAB8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6388
CSNK2A1 (CK2a1)CK2CMGC8pvpA~{n}-[5-[(3-chloranyl-4-phenyl-phenyl)methylamino]pentyl]isoquinoline-5-sulfonamideHuman14977
CDK2CDKCMGC3qrtAA(5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4586
CDK2CDKCMGC3rakAA4-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4574
CDK8CDKCMGC4f70A1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[2-(morpholin-4-yl)ethyl]ureaHuman3852
CDK6CDKCMGC3nuxA4-[5-chloro-3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(5-piperazin-1-ylpyridin-2-yl)pyrimidin-2-amineHuman2807
MAPK14 (p38a)MAPKCMGC2bajA1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2,3-dichlorophenyl)ureaHuman5176
CDK8CDKCMGC5xqxAn-methyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHuman8313
CDK6CDKCMGC5l2tA7-cyclopentyl-n,n-dimethyl-2-{[5-(piperazin-1-yl)pyridin-2-yl]amino}-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman6992
MAPK14 (p38a)MAPKCMGC3objA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman4994
MAPK1 (Erk2)MAPKCMGC4g6oA4-{4-[4-(aminomethyl)-3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHuman2565
MAPK14 (p38a)MAPKCMGC3zsgAAtak-715Human5033
DYRK1ADYRKCMGC5a4lBBn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6735
MAPK14 (p38a)MAPKCMGC2i0hAA2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dioneHuman5062
CDK2CDKCMGC5ievAAroniciclibHuman6567
MAPK1 (Erk2)MAPKCMGC8ao7AA~{n}-[(1-methylindazol-6-yl)methyl]propanamideHuman14389
MAPK1 (Erk2)MAPKCMGC8aoiAB1-(2,3-dihydropyrido[2,3-b][1,4]oxazin-1-yl)propan-1-oneHuman14393
MAPK14 (p38a)MAPKCMGC4aacAn-isoxazol-3-yl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxo-quinazolin-3-yl]benzamideHuman5048
MAPK14 (p38a)MAPKCMGC1r3cAB-Human4996
CDK2CDKCMGC3qqhAB2-[4-amino-6-(phenylamino)-1,3,5-triazin-2-yl]-4-chlorophenolHuman4533
CSNK2A1 (CK2a1)CK2CMGC8p06A7-(cyclopropylamino)-5-[[2-(1,2,4-triazol-4-yl)pyridin-4-yl]amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman14813
MAPK14 (p38a)MAPKCMGC3c5uA6-[4-(2-fluorophenyl)-1,3-oxazol-5-yl]-n-(1-methylethyl)-1,3-benzothiazol-2-amineHuman5125
CDK2CDKCMGC3rkbAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4039
CDK2CDKCMGC4ek6ABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHuman4056
CDK2CDKCMGC4eorCAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4221
CDK2CDKCMGC3r83AA4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4234
CDK2CDKCMGC2clxAB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3880
MAPK14 (p38a)MAPKCMGC3oc1A1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5019
CDK2CDKCMGC5uq2A-Human8221
CDK2CDKCMGC3r1sAB2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4358
MAPK1 (Erk2)MAPKCMGC4fv4AA9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrileHuman2623
CDK2CDKCMGC3pxyAB2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenolHuman3904
CDK2CDKCMGC6q3fAA-Human11181
CDK2CDKCMGC3qx4AB4-chloro-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3990
CDK2CDKCMGC5cyiAA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6052
CDK2CDKCMGC4cfxAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4485
CDK2CDKCMGC3r6xAA4-[(3-hydroxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4398
CDK2CDKCMGC2g9xA3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-olHuman3883
CDK2CDKCMGC3r8vAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman4191
CDK2CDKCMGC2a4lAr-roscovitineHuman4238
CDK2CDKCMGC3s00AB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHuman4248
CDK2CDKCMGC1ke5An-methyl-4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4376
CDK2CDKCMGC4nj3AA6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman4075
CDK2CDKCMGC1gy3Aadenosine-5'-triphosphateHuman3978
CDK2CDKCMGC1jstCadenosine-5'-triphosphateHuman4356
CDK2CDKCMGC1h1pA6-o-cyclohexylmethyl guanineHuman4309
CDK2CDKCMGC9esjAB2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman15905
CDK2CDKCMGC9esyAB4-bromanyl-1,8-naphthyridineHuman15906
CDK2CDKCMGC6rijCB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12622
CDK2CDKCMGC7s84AA2-{[2-(1h-indol-3-yl)ethyl]amino}-5-(trifluoromethyl)benzoic acidHuman14424
CDK2CDKCMGC6q4jAA2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHuman11209
CDK2CDKCMGC2bheA(2z)-5'-bromo-2,3'-biindole-2',3(1h,1'h)-dione ammoniateHuman4184
CDK2CDKCMGC1ol2C-Human4497
CDK2CDKCMGC6q4cAB4-bromanyl-1,8-naphthyridineHuman11207
CDK2CDKCMGC4rj3AB1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4127
CDK2CDKCMGC1pf8A(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3861
CDK2CDKCMGC1hclAA-Human4545
CDK2CDKCMGC1b38Aadenosine-5'-triphosphateHuman4483
CDK2CDKCMGC1g5sA2-[trans-(4-aminocyclohexyl)amino]-6-(benzyl-amino)-9-cyclopentylpurineHuman3888
CDK2CDKCMGC4ek3AA-Human3971
CDK2CDKCMGC3r8uAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman3926
CDK2CDKCMGC4eoiAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4307
CDK2CDKCMGC1h1rAB6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman4494
CDK2CDKCMGC4eonAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4326
CDK2CDKCMGC3qtxAB4-{[4-amino-5-(3-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4419
CDK2CDKCMGC4cfuAB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman4308
CDK2CDKCMGC6q4cAC4-bromanyl-1,8-naphthyridineHuman11201
CDK2CDKCMGC5anjAn-(9h-purin-6-yl)thiophene-2-carboxamideHuman6541
CDK8CDKCMGC6tpaA1-[4-chloranyl-3-(trifluoromethyl)phenyl]-3-(5-oxidanylidene-6-pyridin-4-yl-pyrido[2,3-b][1,5]benzoxazepin-9-yl)ureaHuman13160
CDK2CDKCMGC2v22A-Human4077
CDK2CDKCMGC7b5rL-Human13265
CDK2CDKCMGC4fkiABn-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamideHuman4272
CDK8CDKCMGC5xs2AB3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHuman8314
CDK2CDKCMGC2iw6A[(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrileHuman4019
CDK8CDKCMGC4crlAcortistatin aHuman6096
CDK8CDKCMGC4g6lA-Human3851
CLK1CLKCMGC6khdBA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11644
CDK2CDKCMGC4eonCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4153
CLK1CLKCMGC7ak3AA~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman13142
MAPK14 (p38a)MAPKCMGC3obgA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5211
CDK8CDKCMGC5idpAA(3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanoneHuman7317
CDK8CDKCMGC5fgkAA8-[3-(3-azanyl-2~{h}-indazol-6-yl)-5-chloranyl-pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6391
CDK8CDKCMGC6r3sAB6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman12141
CDK8CDKCMGC5hvyAAn-{(3s)-1-[2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl}-n'-{4-[(morpholin-4-yl)methyl]-3-(trifluoromethyl)phenyl}ureaHuman6553
CLK1CLKCMGC7opgAB4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenolHuman13809
CDK2CDKCMGC8byaA-Human14814
CDK2CDKCMGC8bzoA-Human14815
CDK2CDKCMGC3rniAB3-[(4-amino-5-benzoyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4420
CDK2CDKCMGC3qhrAadenosine-5'-diphosphateHuman4458
CDK2CDKCMGC2v0dA2-imino-5-(1-pyridin-2-yl-meth-(e)-ylidene)-1,3-thiazolidin-4-oneHuman4327
CDK2CDKCMGC2wihAn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4163
CDK2CDKCMGC5oo1A~{n}-(4-pyrimidin-2-ylphenyl)propanamideHuman10566
DYRK2DYRKCMGC7dh9A[2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridin-4-yl]methanolHuman13976
CDK8CDKCMGC5hbjAA8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6390
CDK8CDKCMGC4f6uAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]ureaHuman3849
CDK8CDKCMGC4f7jAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(2-hydroxyethyl)ureaHuman3843
CDK8CDKCMGC4f7sABn-(2-phenylethyl)quinazolin-4-amineHuman3853
CDK8CDKCMGC5bnjA8-{3-chloro-5-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]pyridin-4-yl}-2,8-diazaspiro[4.5]decan-1-oneHuman6152
CDK9CDKCMGC6cytA-Human10797
CDK9CDKCMGC4bciA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman2243
CDK9CDKCMGC3miaAphosphoaminophosphonic acid-adenylate esterHuman2242
MAPK7 (Erk5)MAPKCMGC6hkmA[4-(6,7-dimethoxyquinazolin-4-yl)piperidin-1-yl]-[4-(trifluoromethyloxy)phenyl]methanoneHuman10917
CDK9CDKCMGC3mi9A-Human2239
CLK1CLKCMGC5j1vBpyrido[3,4-g]quinazoline-2,10-diamineHuman6580
CDK2CDKCMGC3ddpAB(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6780
CDK2CDKCMGC5aneA6-methoxy-9h-purineHuman6542
CDK2CDKCMGC1h1qA2-anilino-6-cyclohexylmethoxypurineHuman4195
CDK2CDKCMGC3ezvA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman4083
CDK8CDKCMGC3rgfAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3841
CDK9CDKCMGC4ogrIadenosineHuman2241
CDK8CDKCMGC5hnbAA[6-hydroxy-3-(3-methylbenzyl)-1h-indazol-5-yl][(3s)-3-hydroxypyrrolidin-1-yl]methanoneHuman6562
CDK8CDKCMGC6qtgA2-[4-(4-isoquinolin-4-ylphenyl)pyrazol-1-yl]-~{n},~{n}-dimethyl-ethanamideHuman12094
CLK1CLKCMGC6r6eA5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amineHuman12232
CDK2CDKCMGC1h1sAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4400
CDK8CDKCMGC4f7nA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(5-hydroxypentyl)ureaHuman3847
CDK9CDKCMGC3tn8A4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman2240
CDK9CDKCMGC4ec9A-Human2234
CDK9CDKCMGC4imyABadenosine monophosphateHuman2252
CDK9CDKCMGC5l1zA-Human7121
CDK9CDKCMGC6w9eAA(4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13859
CLK1CLKCMGC1z57AAdebromohymenialdisineHuman106
CLK1CLKCMGC6i5kCA5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10834
CDK8CDKCMGC5i5zAn-methyl-8-(1-methyl-2,2-dioxo-2,3-dihydro-1h-2lambda~6~,1-benzothiazol-5-yl)-1,6-naphthyridine-2-carboxamideHuman6536
CDK8CDKCMGC5idnAA[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanoneHuman7322
CDK9CDKCMGC6z45A(1~{s},3~{r})-3-acetamido-~{n}-[5-chloranyl-4-(5,5-dimethyl-4,6-dihydropyrrolo[1,2-b]pyrazol-3-yl)pyridin-2-yl]cyclohexane-1-carboxamideHuman13115
CDK9CDKCMGC3blrA2-(2-chloro-phenyl)-5,7-dihydroxy-8-(3-hydroxy-1-methyl-piperidin-4-yl)-4h-benzopyran-4-oneHuman2236
MAPK14 (p38a)MAPKCMGC5mz3AB~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8681
MAPK14 (p38a)MAPKCMGC5wjjAAn-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamideHuman9514
CDK2CDKCMGC3r8zAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanoneHuman4137
CDK8CDKCMGC5hbhA5-[5-chloranyl-4-[1-(2-methoxyethyl)-1,8-diazaspiro[4.5]decan-8-yl]pyridin-3-yl]-1-methyl-3~{h}-2,1-benzothiazole 2,2-dioxideHuman6387
CDK8CDKCMGC5icpAB[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanoneHuman7321
CDK8CDKCMGC6y0aAA6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman13306
CDK8CDKCMGC5hbeAA8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-oneHuman6389
CDK2CDKCMGC1vyzAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzamideHuman4325
CDK9CDKCMGC4imyEBadenosine monophosphateHuman2256
CDK9CDKCMGC6gzhA[4-[[4-[5-(cyclopropylmethyl)-1-methyl-pyrazol-4-yl]-5-fluoranyl-pyrimidin-2-yl]amino]cyclohexyl]azaniumHuman10427
CDK9CDKCMGC3blqAadenosine-5'-triphosphateHuman2248
CDK9CDKCMGC6w9eAC(4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13861
MAPK9 (JNK2)MAPKCMGC8elcA4-(dimethylamino)-n-{4-[(3s)-3-({4-[(8r)-2-phenylpyrazolo[1,5-a]pyridin-3-yl]pyrimidin-2-yl}amino)pyrrolidine-1-carbonyl]phenyl}butanamideHuman14816
CDK2CDKCMGC2x1nAB2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4078
CDK1 (CDC2)CDKCMGC5lqfAAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7364
CDK1 (CDC2)CDKCMGC4yc6AB-Human4616
CDK1 (CDC2)CDKCMGC5lqfDBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7367
CDK1 (CDC2)CDKCMGC6gu7C-Human10775
CDK1 (CDC2)CDKCMGC4yc3AB-Human6554
CDK2CDKCMGC4ii5AAadenosine-5'-diphosphateHuman3930
MAPK8 (JNK1)MAPKCMGC4awiAAn-(1,1-dioxidotetrahydro-2h-thiopyran-4-yl)-4-[2-(1-methylethyl)-1h-pyrrolo[2,3-b]pyridin-4-yl]benzenesulfonamideHuman4661
MAPK8 (JNK1)MAPKCMGC6f5eB-Human9078
DYRK1ADYRKCMGC6eipC4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10533
MAPK14 (p38a)MAPKCMGC2fsoX-Human5117
MAPK14 (p38a)MAPKCMGC3qudAA{4-[(2-aminophenyl)amino]phenyl}(phenyl)methanoneHuman5006
MAPK8 (JNK1)MAPKCMGC5lw1HadenosineHuman9080
MAPK8 (JNK1)MAPKCMGC4ux9BBphosphoaminophosphonic acid-adenylate esterHuman4656
MAPK8 (JNK1)MAPKCMGC11zlAA(4m)-n-[4-hydroxy-3-(pyrrolidine-1-carbonyl)phenyl]-4-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1-benzothiophene-2-carboxamideHuman15534
MAPK8 (JNK1)MAPKCMGC4e73ABmethyl 3-(4-{[(1r,2s,3s,5s,7s)-5-aminotricyclo[3.3.1.1~3,7~]dec-2-yl]carbamoyl}benzyl)-4-oxo-1-phenyl-1,4-dihydro-1,8-naphthyridine-2-carboxylateHuman4669
MAPK8 (JNK1)MAPKCMGC5lw1EadenosineHuman9079
CDK2CDKCMGC4eosCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4181
MAPK8 (JNK1)MAPKCMGC4yr8EB-Human6454
CLK1CLKCMGC6i5lBB3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10839
CDK2CDKCMGC2r3iAC-Human4317
CDK2CDKCMGC3ql8AB3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrileHuman4306
CDK2CDKCMGC3r8uAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](naphthalen-2-yl)methanoneHuman3864
CDK2CDKCMGC3tizA1-{(e)-[(4-hydroxyphenyl)imino]methyl}naphthalen-2-olHuman4136
CDK2CDKCMGC4eosAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4340
CDK2CDKCMGC3qtuAB4-{[4-amino-5-(4-sulfamoylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4323
CDK1 (CDC2)CDKCMGC4yc6CB-Human4611
DYRK1ADYRKCMGC6t6aAB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11858
DYRK1ADYRKCMGC6eijB~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10516
MAPK14 (p38a)MAPKCMGC3mh2A-Human4985
CDK2CDKCMGC3ej1Cn-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHuman4092
CSNK2A1 (CK2a1)CK2CMGC5otdBB[2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azaniumHuman9632
CSNK2A1 (CK2a1)CK2CMGC5cs6AA-Human6915
CSNK2A1 (CK2a1)CK2CMGC5osrAAadenosine-5'-triphosphateHuman10601
MAPK1 (Erk2)MAPKCMGC5wp1AB5,7-dihydroxy-4h-1-benzopyran-4-oneHuman10440
CDK2CDKCMGC3qqkAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4514
MAPK8 (JNK1)MAPKCMGC3o17B-Human4667
MAPK8 (JNK1)MAPKCMGC4yr8AB-Human6448
MAPK3 (Erk1)MAPKCMGC4qtbBA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman1717
CSNK2A1 (CK2a1)CK2CMGC5movAA4'-hydroxycinnamic acidHuman7655
CSNK2A1 (CK2a1)CK2CMGC3at4A[1-(6-{6-[(1-methylethyl)amino]-1h-indazol-1-yl}pyrazin-2-yl)-1h-pyrrol-3-yl]acetic acidHuman5413
CSNK2A1 (CK2a1)CK2CMGC6fvgABadenosine-5'-triphosphateHuman11339
CDK5CDKCMGC1unhB(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2787
MAPK8 (JNK1)MAPKCMGC3o2mA-Human4676
MAPK8 (JNK1)MAPKCMGC4ux9DAphosphoaminophosphonic acid-adenylate esterHuman4627
CDK2CDKCMGC2vtiAn-(4-sulfamoylphenyl)-1h-indazole-3-carboxamideHuman4177
CSNK2A1 (CK2a1)CK2CMGC7qgbAA5,6-dibromobenzotriazoleHuman14468
DYRK1ADYRKCMGC7ak2A4-[2-methyl-3-(2-pyridin-2-yloxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13593
CDK2CDKCMGC3r8pAA(5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4232
CDK8CDKCMGC4f6sA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman3848
CSNK2A1 (CK2a1)CK2CMGC7qgbAB5,6-dibromobenzotriazoleHuman14470
CSNK2A1 (CK2a1)CK2CMGC7qgdAB5,6-dibromobenzotriazoleHuman14471
CDK2CDKCMGC3bhuAA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4105
CDK2CDKCMGC1f5qAA-Human4194
SRPK2SRPKCMGC5myvCB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7571
SRPK2SRPKCMGC5myvDA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7578
SRPK2SRPKCMGC5myvAA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7579
CDK2CDKCMGC1ol1A-Human4429
CDK2CDKCMGC6q4hAB2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHuman11190
CLK1CLKCMGC6ft9BB2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9894
CLK1CLKCMGC6i5lAA3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10837
CLK1CLKCMGC6g33CA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9825
CLK1CLKCMGC6i5lBA3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10846
CLK1CLKCMGC6ft9BA2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9897
CLK1CLKCMGC6z50AB11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12308
CLK1CLKCMGC8p04A(4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-oneHuman14741
CDK2CDKCMGC2c6oAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman6783
CDK2CDKCMGC5osmABmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHuman9740
CDK7CDKCMGC7b5qJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13277
CLK3CLKCMGC2wu7ABethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman1827
CLK1CLKCMGC5j1wBBpyrido[3,4-g]quinazolin-2-amineHuman6583
CLK1CLKCMGC5j1vCpyrido[3,4-g]quinazoline-2,10-diamineHuman6577
CLK1CLKCMGC6g33CC-Human9820
CLK1CLKCMGC6r3dA4-[6,7-bis(chloranyl)-1~{h}-indol-3-yl]pyrimidin-2-amineHuman12128
CDK5CDKCMGC3o0gB{4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanoneHuman2783
CLK1CLKCMGC6ft8AA3-(3-hydroxyphenyl)-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9895
CLK1CLKCMGC6g33BB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9822
CLK1CLKCMGC6i5lCA3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10833
CLK1CLKCMGC6raaAA4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11014
CLK1CLKCMGC6i5kBB5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10835
CLK1CLKCMGC6r8jAA4-(1-methylindol-3-yl)pyrimidin-2-amineHuman12632
CLK1CLKCMGC6z4zBB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12311
CLK1CLKCMGC6i5kBA5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10842
CDK2CDKCMGC3qu0AA4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4427
CDK2CDKCMGC2r3mAAn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHuman4286
CDK2CDKCMGC5oo0AA-Human9744
DYRK2DYRKCMGC5ztnA(1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneHuman10482
DYRK2DYRKCMGC7dhnA7-methoxy-2-methylsulfanyl-9-(piperidin-4-ylmethylsulfanyl)-[1,3]thiazolo[5,4-b]quinolineHuman13971
DYRK2DYRKCMGC5lxdABmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7128
CLK1CLKCMGC5j1wCBpyrido[3,4-g]quinazolin-2-amineHuman6581
CLK1CLKCMGC5x8iB5-[1-[(1s)-1-(4-fluorophenyl)ethyl]-[1,2,3]triazolo[4,5-c]quinolin-8-yl]-1,3-benzoxazoleHuman8317
CLK1CLKCMGC6fyoAA6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHuman10324
CDK2CDKCMGC3ig7An-{1-[cis-3-(acetylamino)cyclobutyl]-1h-imidazol-4-yl}-2-(4-methoxyphenyl)acetamideHuman4021
DYRK2DYRKCMGC4azfAB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3146
CLK1CLKCMGC7oa0A5-[6,7-bis(chloranyl)-1-methyl-indol-3-yl]pyrimidin-4-amineHuman14207
CLK1CLKCMGC6i5kAA5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10844
CLK1CLKCMGC6yteCB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12422
CLK1CLKCMGC6z50AA11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12314
CLK1CLKCMGC6i5kCB5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10838
CDK2CDKCMGC3qx2AA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-[(2-hydroxyethyl)amino]-5-nitrobenzamideHuman4031
CDK2CDKCMGC4eojCBadenosine-5'-triphosphateHuman4311
CDK2CDKCMGC4fkpAB3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4313
DYRK2DYRKCMGC3k2lAB-Human3145
DYRK2DYRKCMGC3k2lAA-Human3147
DYRK2DYRKCMGC7dhoA2-methoxy-9-(piperidin-4-ylmethylsulfanyl)-7-propan-2-yloxy-acridineHuman13972
DYRK2DYRKCMGC7ejvAB[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14181
DYRK2DYRKCMGC7ejvAA[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14180
CLK1CLKCMGC6khdAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11646
CLK1CLKCMGC6tw2EBethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman11963
CLK1CLKCMGC6i5iAA5-(1-methylpyrazol-4-yl)-3-[1-(phenylmethyl)pyrazol-4-yl]furo[3,2-b]pyridineHuman10845
CLK1CLKCMGC6z4zAA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12315
CLK1CLKCMGC6q8kAB~{n}2-(3-morpholin-4-ylpropyl)pyrido[3,4-g]quinazoline-2,10-diamineHuman10903
CLK1CLKCMGC6ft9CA2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9896
CLK1CLKCMGC8p08A(4~{z})-4-(1,3-benzothiazol-6-ylmethylidene)-2-[[(2~{r})-1-methoxy-4-methyl-pentan-2-yl]amino]-1~{h}-imidazol-5-oneHuman14742
CLK1CLKCMGC6q8pA~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amineHuman10899
DYRK2DYRKCMGC4azfAA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3144
CDK2CDKCMGC3qruAB(5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4516
CDK2CDKCMGC2wmaA-Human4435
CDK2CDKCMGC6gucA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman10767
DYRK2DYRKCMGC7dg4A2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridineHuman13967
DYRK2DYRKCMGC6hdrABcurcuminHuman11571
DYRK2DYRKCMGC5lxdAAmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7124
DYRK2DYRKCMGC7akfAB4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13614
DYRK2DYRKCMGC5lxcAAmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7122
CDK2CDKCMGC2r3gAB6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman3923
CDK2CDKCMGC3r28AB4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamideHuman4293
DYRK2DYRKCMGC7akfAA4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13613
DYRK2DYRKCMGC5lxcABmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7129
DYRK2DYRKCMGC6k0jA3-(2,7-dimethoxyacridin-9-yl)sulfanylpropan-1-amineHuman11817
MAPK12 (p38g)MAPKCMGC7cgaA-Human13762
SRPK2SRPKCMGC5myvDB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7572
CDK2CDKCMGC3r1qAB4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4507
CDK2CDKCMGC4bzdAB6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHuman4490
CDK2CDKCMGC4eorAAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4205
CDKL5CDKLCMGC4bgqAA[4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1425
CDKL5CDKLCMGC4bgqAB[4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman1426
CDK2CDKCMGC3rpoAB4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acidHuman4098
CDK2CDKCMGC2wipC1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHuman4190
CDK1 (CDC2)CDKCMGC4yc3AA-Human6555
MAPK8 (JNK1)MAPKCMGC4l7fACn-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamideHuman4648
CDK2CDKCMGC3bhuCA4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4087
CLK3CLKCMGC2eu9AA-Human1826
CLK3CLKCMGC6khfAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11649
CLK3CLKCMGC6rctBB4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11129
MAPK8 (JNK1)MAPKCMGC3vukA-Human4659
CDK2CDKCMGC3rjcAB{4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanoneHuman4469
CDK2CDKCMGC1y8yA(5-chloropyrazolo[1,5-a]pyrimidin-7-yl)-(4-methanesulfonylphenyl)amineHuman3914
CLK3CLKCMGC6ytwAA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12404
MAPK1 (Erk2)MAPKCMGC8psrABphosphoaminophosphonic acid-adenylate esterHuman15298
MAPK1 (Erk2)MAPKCMGC6slgAB(6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-oneHuman11816
MAPK1 (Erk2)MAPKCMGC6ge0AB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamideHuman9961
MAPK1 (Erk2)MAPKCMGC6q7kA1h-imidazol-2-amineHuman10985
MAPK1 (Erk2)MAPKCMGC6g8xAA4-chloranyl-1~{h}-indazol-3-amineHuman9957
MAPK1 (Erk2)MAPKCMGC6g9dAA~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamideHuman9972
MAPK9 (JNK2)MAPKCMGC3npcB1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman1237
CLK3CLKCMGC6z55BC7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12297
CLK3CLKCMGC6ft7AA3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9905
CLK3CLKCMGC6z52AB11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12627
MAPK8 (JNK1)MAPKCMGC2h96B5-cyano-n-(2,5-dimethoxybenzyl)-6-ethoxypyridine-2-carboxamideHuman4668
MAPK1 (Erk2)MAPKCMGC8pstABamp phosphoramidateHuman15299
MAPK1 (Erk2)MAPKCMGC4qp3A(2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-olHuman6084
MAPK1 (Erk2)MAPKCMGC4qp7A2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6082
MAPK1 (Erk2)MAPKCMGC4zxtAAcatecholHuman6654
MAPK1 (Erk2)MAPKCMGC6g9hAA~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamideHuman9971
MAPK1 (Erk2)MAPKCMGC8ao2AB~{n}-(1~{h}-indazol-5-ylmethyl)propanamideHuman14394
CDK2CDKCMGC6gubC2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10763
CDK2CDKCMGC4fkjAAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHuman4387
CDK2CDKCMGC4fksABn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4489
CLK3CLKCMGC6rctAB4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11126
MAPK1 (Erk2)MAPKCMGC4iz5Dadenosine-5'-diphosphateHuman2578
MAPK1 (Erk2)MAPKCMGC5bvfAA2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6031
MAPK1 (Erk2)MAPKCMGC5lckAB~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamideHuman6836
MAPK1 (Erk2)MAPKCMGC6g9nAB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamideHuman11413
MAPK1 (Erk2)MAPKCMGC4fuyAA{4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanoneHuman2622
MAPK1 (Erk2)MAPKCMGC6qahAB1-azanylpropylideneazaniumHuman11348
MAPK1 (Erk2)MAPKCMGC4qp8A2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6087
MAPK1 (Erk2)MAPKCMGC7opmAB1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]ureaHuman14083
MAPK1 (Erk2)MAPKCMGC8ao7AB~{n}-[(1-methylindazol-6-yl)methyl]propanamideHuman14398
MAPK1 (Erk2)MAPKCMGC8ao4AB~{n}-(1~{h}-indazol-5-yl)ethanesulfonamideHuman14399
MAPK1 (Erk2)MAPKCMGC4zxtABcatecholHuman6653
CDK2CDKCMGC1h27A-Human4116
MAPK1 (Erk2)MAPKCMGC4izaCB-Human2627
MAPK1 (Erk2)MAPKCMGC6q7tAA1,2-oxazol-3-amineHuman11350
MAPK1 (Erk2)MAPKCMGC6g91AB5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amineHuman9956
CDK2CDKCMGC3r7vAA5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamideHuman4380
CDK2CDKCMGC2c6lA4-({5-[(4-aminocyclohexyl)amino][1,2,4]triazolo[1,5-a]pyrimidin-7-yl}amino)benzenesulfonamideHuman6779
CDK2CDKCMGC1oi9AA6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4033
CDK2CDKCMGC5lmkAB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7398
CDK2CDKCMGC4cfuCA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman3967
CDK2CDKCMGC4cfvCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman3999
CDK2CDKCMGC5uq3A-Human8222
MAPK1 (Erk2)MAPKCMGC6opgAphosphoaminophosphonic acid-adenylate esterHuman11507
MAPK1 (Erk2)MAPKCMGC8ao5AB~{n}-(1~{h}-indazol-5-ylmethyl)ethanesulfonamideHuman14400
MAPK1 (Erk2)MAPKCMGC3teiAphosphoaminophosphonic acid-adenylate esterHuman2608
CDK2CDKCMGC6q3cAA4-bromo-1h-pyrazoleHuman11191
MAPK1 (Erk2)MAPKCMGC6g54AAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10938
MAPK1 (Erk2)MAPKCMGC4qtaAA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman2602
MAPK1 (Erk2)MAPKCMGC8aocAB~{n}-(3-methyl-[1,2]oxazolo[5,4-b]pyridin-5-yl)propanamideHuman14406
MAPK1 (Erk2)MAPKCMGC7e75A-Human14115
MAPK1 (Erk2)MAPKCMGC6gdqAA4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamideHuman9948
MAPK1 (Erk2)MAPKCMGC5bveAB2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6026
MAPK1 (Erk2)MAPKCMGC8aoaAB~{n}-pyridin-3-ylprop-2-enamideHuman14407
CDK2CDKCMGC4erwAstaurosporineHuman4370
CDK2CDKCMGC2i40AB5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4470
CDK2CDKCMGC4ek5AAn-(5-cyclopropyl-1h-pyrazol-3-yl)benzene-1,4-dicarboxamideHuman4037
CDK2CDKCMGC3eidAB(2s)-1-(dimethylamino)-3-(4-{[4-(6-morpholin-4-ylpyrazolo[1,5-b]pyridazin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4424
CLK3CLKCMGC3rawBB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman1825
MAPK1 (Erk2)MAPKCMGC6g9aAA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-oneHuman11408
MAPK1 (Erk2)MAPKCMGC5lckAA~{n}-[2-[[2-[(5-methoxypyridin-3-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]phenyl]propanamideHuman6835
MAPK1 (Erk2)MAPKCMGC3w55A(3s,5z,8s,9s,11e)-8,9,16-trihydroxy-14-methoxy-3-methyl-3,4,9,10-tetrahydro-1h-2-benzoxacyclotetradecine-1,7(8h)-dioneHuman2573
MAPK1 (Erk2)MAPKCMGC5bueA1-benzyl-4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-oneHuman2574
MAPK1 (Erk2)MAPKCMGC7xc1A(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14665
CDK2CDKCMGC3rprAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl][3-(trifluoromethyl)phenyl]methanoneHuman4452
MAPK1 (Erk2)MAPKCMGC5nhfA2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-5-(phenylmethyl)-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7997
CDK2CDKCMGC5fp6AA3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHuman6302
CDK2CDKCMGC3r1sAA2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4263
CDK2CDKCMGC3qqjAA2-(4,6-diamino-1,3,5-triazin-2-yl)phenolHuman4113
CLK3CLKCMGC6ft7BA3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9904
MAPK1 (Erk2)MAPKCMGC6gjbAA[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman10832
MAPK1 (Erk2)MAPKCMGC8aoeAB~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamideHuman14411
MAPK1 (Erk2)MAPKCMGC5v61AB-Human8266
MAPK1 (Erk2)MAPKCMGC2y9qACphosphoaminophosphonic acid-adenylate esterHuman2567
MAPK1 (Erk2)MAPKCMGC6qa3AApyrazoleHuman11353
MAPK1 (Erk2)MAPKCMGC6rfoA-Human12341
MAPK1 (Erk2)MAPKCMGC4xj0B1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-oneHuman6049
MAPK1 (Erk2)MAPKCMGC4izaAB-Human2607
CDK2CDKCMGC3s0oAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-2-yl)methanoneHuman3898
CDK2CDKCMGC2g9xC3-({2-[(4-{[6-(cyclohexylmethoxy)-9h-purin-2-yl]amino}phenyl)sulfonyl]ethyl}amino)propan-1-olHuman4082
CDK2CDKCMGC3rjcAA{4-amino-2-[(3-fluorophenyl)amino]-1,3-thiazol-5-yl}(phenyl)methanoneHuman4032
MAPK1 (Erk2)MAPKCMGC5v62AA5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman8264
MAPK1 (Erk2)MAPKCMGC4qp2B-Human6081
MAPK1 (Erk2)MAPKCMGC4n0sABcaffeic acidHuman2555
MAPK1 (Erk2)MAPKCMGC4zzmA7-ethylsulfonyl-n-(oxan-4-yl)-6,8-dihydro-5h-pyrido[3,4-d]pyrimidin-2-amineHuman2616
MAPK1 (Erk2)MAPKCMGC8ao3AB2-chloranyl-~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14414
MAPK1 (Erk2)MAPKCMGC6q7tAB1,2-oxazol-3-amineHuman11347
MAPK1 (Erk2)MAPKCMGC5k4iA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6744
CDK2CDKCMGC2iw6C[(2-chloro-5-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino]acetonitrileHuman4108
MAPK1 (Erk2)MAPKCMGC6g9jAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamideHuman9949
MAPK1 (Erk2)MAPKCMGC4iz7AA-Human2615
MAPK1 (Erk2)MAPKCMGC4qtaAB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman2576
MAPK1 (Erk2)MAPKCMGC8aofAA~{n}-(2-methylpyrimidin-5-yl)propanamideHuman14419
CSNK2A2 (CK2a2)CK2CMGC8qf1AA-Human15020
CDK2CDKCMGC6athAA-Human10567
CSNK2A2 (CK2a2)CK2CMGC5m4uAA4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7390
CSNK2A2 (CK2a2)CK2CMGC6hmdAC-Human10990
CSNK2A2 (CK2a2)CK2CMGC6te2AA3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12444
CSNK2A2 (CK2a2)CK2CMGC8qf1AB-Human15021
CSNK2A2 (CK2a2)CK2CMGC3ofmAB3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman2730
CSNK2A2 (CK2a2)CK2CMGC7at9AB3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman13829
CSNK2A2 (CK2a2)CK2CMGC8q77AA(2~{s})-2-[[(2~{s})-2-[[(2~{s})-2-[12-[[4-[[5-(4-carboxyphenyl)-1,3-thiazol-2-yl]amino]-4-oxidanylidene-butanoyl]-(2-hydroxy-2-oxoethyl)amino]dodecanoylamino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]butanedioic acidHuman15024
CSNK2A2 (CK2a2)CK2CMGC5yf9BAnicotinic acidHuman11415
CSNK2A2 (CK2a2)CK2CMGC7a1zAB6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13147
CSNK2A2 (CK2a2)CK2CMGC6qy8AA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12117
CSNK2A2 (CK2a2)CK2CMGC8qbuAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman15025
CSNK2A2 (CK2a2)CK2CMGC7at9AC2-(3,4-dichlorophenyl)ethanamineHuman13830
CSNK2A2 (CK2a2)CK2CMGC8qcgAAphosphoaminophosphonic acid-adenylate esterHuman15026
CSNK2A2 (CK2a2)CK2CMGC5y9mAnicotinic acidHuman9908
CSNK2A1 (CK2a1)CK2CMGC7qgdAA5,6-dibromobenzotriazoleHuman14472
CSNK2A2 (CK2a2)CK2CMGC9fbiAAnicotinic acidHuman15561
CSNK2A2 (CK2a2)CK2CMGC8qcgACphosphoaminophosphonic acid-adenylate esterHuman15027
CSNK2A2 (CK2a2)CK2CMGC5yf9XAnicotinic acidHuman11417
CSNK2A2 (CK2a2)CK2CMGC6l20G(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman11995
CSNK2A2 (CK2a2)CK2CMGC8q9sAA~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamideHuman15028
CSNK2A2 (CK2a2)CK2CMGC6qy9AB3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrileHuman11011
CSNK2A2 (CK2a2)CK2CMGC6l20D(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman11996
CSNK2A2 (CK2a2)CK2CMGC6qy9AA3-[3-[2-[(3,4,5-trimethoxyphenyl)amino]pyrrolo[2,3-d]pyrimidin-7-yl]phenyl]propanenitrileHuman11012
CSNK2A2 (CK2a2)CK2CMGC6hmcAB-Human10993
CSNK2A2 (CK2a2)CK2CMGC6hmbAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10994
CSNK2A2 (CK2a2)CK2CMGC6hmqAA3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman10991
CDK2CDKCMGC1pyeA[2-amino-6-(2,6-difluoro-benzoyl)-imidazo[1,2-a]pyridin-3-yl]-phenyl-methanoneHuman4284
CDK2CDKCMGC2uueC4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHuman4321
CDK2CDKCMGC2r3jAA3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4185
CSNK2A2 (CK2a2)CK2CMGC6hmdAB-Human10992
CSNK2A2 (CK2a2)CK2CMGC6l20A(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman11993
CSNK2A2 (CK2a2)CK2CMGC8qcgABphosphoaminophosphonic acid-adenylate esterHuman15030
CSNK2A2 (CK2a2)CK2CMGC6hmdAA5-[2-(diethylamino)ethyl]-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman10997
CLK1CLKCMGC6khdBB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11647
MAPK1 (Erk2)MAPKCMGC3i5zAn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHuman2579
MAPK1 (Erk2)MAPKCMGC8aoeAA~{n}-(1~{h}-pyrrolo[2,3-b]pyridin-4-yl)ethanesulfonamideHuman14395
CSNK2A2 (CK2a2)CK2CMGC5m56B4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7389
CSNK2A2 (CK2a2)CK2CMGC6qy8BA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12114
CSNK2A2 (CK2a2)CK2CMGC7atvAA~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamideHuman13831
MAPK1 (Erk2)MAPKCMGC4nifBAphosphoaminophosphonic acid-adenylate esterHuman2585
CDK2CDKCMGC1pxiAA4-(2,5-dichlorothien-3-yl)pyrimidin-2-amineHuman4381
MAPK1 (Erk2)MAPKCMGC4fv5An-[(1s)-2-hydroxy-1-phenylethyl]-4-(5-methyl-2-phenylpyrimidin-4-yl)-1h-pyrrole-2-carboxamideHuman2598
MAPK1 (Erk2)MAPKCMGC8ao6AA~{n}-(1~{h}-indazol-5-ylmethyl)ethanamideHuman14397
MAPK1 (Erk2)MAPKCMGC4fv8AA6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-oneHuman2625
MAPK1 (Erk2)MAPKCMGC6dmgAA-Human10811
CSNK2A2 (CK2a2)CK2CMGC5m56A4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7388
CSNK2A2 (CK2a2)CK2CMGC8q9sAB~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamideHuman15031
CSNK2A2 (CK2a2)CK2CMGC6hmbAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10995
CSNK2A2 (CK2a2)CK2CMGC9r57AB5,6-dibromobenzotriazoleHuman15562
CDK2CDKCMGC1okwC-Human3896
CDK2CDKCMGC1pxpAAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4316
CDK2CDKCMGC1pxlAA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4233
CDK2CDKCMGC3le6A5-(2-chlorophenyl)-3-methyl-7-nitropyrazolo[3,4-b][1,4]benzodiazepineHuman4125
CDK8CDKCMGC3rgfAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman3846
CLK3CLKCMGC6fyrAA6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHuman11407
CLK3CLKCMGC6yu1cB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12411
CLK3CLKCMGC6ytwBA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12412
CLK3CLKCMGC6ft7BB3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9902
CSNK2A2 (CK2a2)CK2CMGC8qbuAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman15029
CDK2CDKCMGC3ns9A(2s,3s)-3-{[7-(benzylamino)-3-(1-methylethyl)pyrazolo[1,5-a]pyrimidin-5-yl]amino}butane-1,2,4-triolHuman4575
MAPK1 (Erk2)MAPKCMGC4zznAA2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamideHuman2605
MAPK1 (Erk2)MAPKCMGC6g9hAB~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-methyl-ethanamideHuman9958
CDK8CDKCMGC5ceiAB4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamideHuman6403
MAPK1 (Erk2)MAPKCMGC6slgAA(6~{r})-7-[[3,4-bis(fluoranyl)phenyl]methyl]-6-(methoxymethyl)-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5,6-dihydroimidazo[1,2-a]pyrazin-8-oneHuman11815
MAPK1 (Erk2)MAPKCMGC6gjbAB[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[4-[1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-2-oxidanylidene-pyridin-4-yl]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman10831
MAPK1 (Erk2)MAPKCMGC8aobAB~{n}-[(1-methylindazol-3-yl)methyl]propanamideHuman14413
MAPK1 (Erk2)MAPKCMGC6rq4AA6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-oneHuman11854
CSNK2A1 (CK2a1)CK2CMGC7zykABadenosine-5'-diphosphateHuman14546
CSNK2A1 (CK2a1)CK2CMGC7qgcAB5,6-dibromobenzotriazoleHuman14434
MAPK8 (JNK1)MAPKCMGC4ux9CAphosphoaminophosphonic acid-adenylate esterHuman4644
CDK2CDKCMGC5cyiCB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6053
CDK2CDKCMGC3qxpAB4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4482
CDK2CDKCMGC4ek8AA4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amineHuman4079
CDK2CDKCMGC3rm7AA2-[(4-hydroxybenzyl)amino]-5-nitrobenzamideHuman3893
CDK2CDKCMGC2uzbAC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4099
CDK2CDKCMGC3pxyAA2-(4,6-diamino-1,3,5-triazin-2-yl)-4-methoxyphenolHuman4057
CDK2CDKCMGC4cfwAA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4280
CDK2CDKCMGC1oi9AB6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4492
CDK2CDKCMGC3qziAA4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamideHuman4094
CDK2CDKCMGC3qrtAB(5r)-5-(2-methylbutan-2-yl)-n-(4-sulfamoylbenzyl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4536
CDK2CDKCMGC5uq1C-Human8223
CDK2CDKCMGC3r7iAA4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acidHuman4450
CSNK2A2 (CK2a2)CK2CMGC3e3bX[1-(6-{6-[(1-methylethyl)amino]-1h-indazol-1-yl}pyrazin-2-yl)-1h-pyrrol-3-yl]acetic acidHuman2729
CDK2CDKCMGC4fklAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4583
CDK2CDKCMGC6yl6AA-Human12498
CDK2CDKCMGC2r3lAB3-bromo-6-phenyl-n-(pyrimidin-5-ylmethyl)imidazo[1,2-a]pyridin-8-amineHuman4085
CDK2CDKCMGC8fp0ABr-roscovitineHuman14756
CDK2CDKCMGC8fp5ABadenosine-5'-triphosphateHuman14757
CDK2CDKCMGC8fp0AAr-roscovitineHuman14758
CDK2CDKCMGC8fowAA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman14759
CSNK2A2 (CK2a2)CK2CMGC7a2hAB5,6,7-tris(bromanyl)-1~{h}-imidazo[4,5-b]pyridineHuman13146
CDK2CDKCMGC8fowAB3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman14760
CDK2CDKCMGC8fp5AAadenosine-5'-triphosphateHuman14761
CDK2CDKCMGC3f5xA4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman3882
CDK2CDKCMGC3qhrCadenosine-5'-diphosphateHuman3879
CSNK2A2 (CK2a2)CK2CMGC6qy8DB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12118
CSNK2A2 (CK2a2)CK2CMGC6qy8CB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12119
CDK2CDKCMGC4bcqCB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4120
CDK2CDKCMGC3bhtAA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman3950
MAPK10 (JNK3)MAPKCMGC3oxiAmethyl 3-[(thiophen-2-ylacetyl)amino]thiophene-2-carboxylateHuman3423
CDK2CDKCMGC2r3rAA3-bromo-5-phenyl-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4040
CDK2CDKCMGC1oguAA4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3965
CDK2CDKCMGC2wevCB[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman3859
CDK2CDKCMGC3r8mAA1h-indazole-3-carbohydrazideHuman4111
CLK3CLKCMGC6z2vAA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12637
CLK3CLKCMGC6z55AA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12302
MAPK10 (JNK3)MAPKCMGC6emhCB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10505
CDK2CDKCMGC1oiyAA4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4225
CDK2CDKCMGC2j9mAA6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxideHuman4154
CDK1 (CDC2)CDKCMGC5lqfABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7366
CDK2CDKCMGC3py0AA(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3995
CDK2CDKCMGC2vv9AB2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHuman3881
CDK2CDKCMGC3qzgAA2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenolHuman4144
CDK2CDKCMGC2vv9AA2-{4-[4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)phenyl]piperazin-1-yl}-2-oxoethanolHuman3989
CDK2CDKCMGC1h25A-Human4273
CDK2CDKCMGC3r7eAA5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamideHuman4159
CDK2CDKCMGC2r3nAA3-cyclopropyl-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4101
CDK2CDKCMGC1fvtA4-(5-bromo-2-oxo-2h-indol-3-ylazo)-benzenesulfonamideHuman4480
CDK1 (CDC2)CDKCMGC4y72AB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4609
CLK4CLKCMGC6fyvAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10511
CDK2CDKCMGC2vtoAAn-(4-fluorophenyl)-4-[(phenylcarbonyl)amino]-1h-pyrazole-3-carboxamideHuman4421
CDK2CDKCMGC1ke7A3-{[(2,2-dioxido-1,3-dihydro-2-benzothien-5-yl)amino]methylene}-5-(1,3-oxazol-5-yl)-1,3-dihydro-2h-indol-2-oneHuman4295
CDK2CDKCMGC3bhvCB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4529
CDK2CDKCMGC1h24C-Human4296
CDK2CDKCMGC3bhtCA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4151
CDK2CDKCMGC4ek6AAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(thiophen-2-yl)phenyl]acetamideHuman4359
CDK2CDKCMGC4fkwAB2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHuman4277
CDK2CDKCMGC3tiyAB2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHuman4488
CDK2CDKCMGC1ol2A-Human4305
CDK2CDKCMGC6q4hAA2-[3-[(2-azanyl-9~{h}-purin-6-yl)oxy]phenyl]ethanoic acidHuman11194
CSNK2A2 (CK2a2)CK2CMGC6qy8AB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12120
CDK2CDKCMGC2cciCadenosine-5'-triphosphateHuman4532
CLK1CLKCMGC6r6xA5-(1-methylindol-3-yl)pyrimidin-4-amineHuman12231
CDK2CDKCMGC1finCadenosine-5'-triphosphateHuman4479
CDK2CDKCMGC2r3oAC(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4229
DYRK1ADYRKCMGC6s11AA6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11361
DYRK1ADYRKCMGC6eipA4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10555
DYRK1ADYRKCMGC6eiqD[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10541
DYRK1ADYRKCMGC7ajmAA~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamideHuman13590
DYRK1ADYRKCMGC6uwyAA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11989
DYRK1ADYRKCMGC7aj5AB4-(1-benzofuran-5-yl)pyridine-2,6-diamineHuman13591
DYRK1ADYRKCMGC6eipD4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10531
DYRK1ADYRKCMGC6t6aDA-Human11862
DYRK1ADYRKCMGC7a4oAphosphoaminophosphonic acid-adenylate esterHuman13744
DYRK1ADYRKCMGC2vx3DAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3786
DYRK1ADYRKCMGC6uwyCA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11984
DYRK1ADYRKCMGC6a1gA5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10530
DYRK1ADYRKCMGC6eirD~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10549
DYRK1ADYRKCMGC7a5dAB4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13745
DYRK1ADYRKCMGC4yu2CB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3775
MAPK9 (JNK2)MAPKCMGC3e7oAn-{3-[5-(1h-1,2,4-triazol-3-yl)-1h-indazol-3-yl]phenyl}furan-2-carboxamideHuman1238
CLK1CLKCMGC6r8jAB4-(1-methylindol-3-yl)pyrimidin-2-amineHuman12631
CSNK2A2 (CK2a2)CK2CMGC6te2AB3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12446
DYRK1ADYRKCMGC5a4tCn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6734
DYRK1ADYRKCMGC7ajmAB~{n}-[6-azanyl-4-(1-benzofuran-5-yl)pyridin-2-yl]-2-(methylamino)ethanamideHuman13598
DYRK1ADYRKCMGC6eipB4-[[(3~{r},7~{s})-2-cyclopentyl-9-methyl-8-oxidanylidene-2,9,12,14-tetrazatricyclo[8.4.0.0^{3,7}]tetradeca-1(14),10,12-trien-13-yl]amino]benzamideHuman10517
DYRK1ADYRKCMGC6s1bAA~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11359
DYRK1ADYRKCMGC7aj8AB4-(1-benzofuran-5-yl)pyridin-2-amineHuman13603
MAPK1 (Erk2)MAPKCMGC7x4uAB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14661
DYRK1ADYRKCMGC6uwyCB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11985
DYRK1ADYRKCMGC5aikB4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3759
DYRK1ADYRKCMGC5a4lCAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6721
DYRK1ADYRKCMGC6eisBA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10556
DYRK1ADYRKCMGC4nctDpkc412Human3751
CDK5CDKCMGC7vdsAB5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHuman14147
DYRK1ADYRKCMGC5a4qDn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6737
DYRK1ADYRKCMGC4yu2AB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3765
MAPK9 (JNK2)MAPKCMGC7cmlAB-Human12705
CDK9CDKCMGC4imyAAadenosine monophosphateHuman2238
MAPK1 (Erk2)MAPKCMGC7x4uAA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14660
CDK9CDKCMGC8k5rA(1s,3s)-n3-(5-pentan-3-ylpyrazolo[1,5-a]pyrimidin-7-yl)cyclopentane-1,3-diamineHuman15081
CDK5CDKCMGC1ungB6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2789
DYRK2DYRKCMGC8hltA(6-{[(4p)-4-(1,3-benzothiazol-5-yl)-5-fluoropyrimidin-2-yl]amino}pyridin-3-yl)(piperazin-1-yl)methanoneHuman15091
DYRK1ADYRKCMGC7ajsAB4-(2-methyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13607
CLK1CLKCMGC6ytgAB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12424
DYRK1ADYRKCMGC5a4eABn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6740
DYRK1ADYRKCMGC4yljCB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3748
DYRK1ADYRKCMGC5a4eCAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6725
DYRK1ADYRKCMGC6s1iAA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11370
DYRK1ADYRKCMGC5a4eAAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6741
DYRK1ADYRKCMGC6s1iAB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11376
CDK9CDKCMGC4ogrEadenosineHuman2235
DYRK1ADYRKCMGC3anqC(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3791
DYRK1ADYRKCMGC4mq2CBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3780
DYRK1ADYRKCMGC7fhsAA(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14160
DYRK1ADYRKCMGC6s11AB6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11364
DYRK1ADYRKCMGC6qu2AA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12085
DYRK1ADYRKCMGC4azeA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3761
DYRK1ADYRKCMGC6s1bAB~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11377
DYRK1ADYRKCMGC4yllAC10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3731
DYRK1ADYRKCMGC6eiqC[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10524
DYRK1ADYRKCMGC5a4tDn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6712
DYRK1ADYRKCMGC7a53AA(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-oneHuman13755
DYRK1ADYRKCMGC4yu2DB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3733
DYRK1ADYRKCMGC4mq1CAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3781
DYRK1ADYRKCMGC6s1iBA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11371
DYRK1ADYRKCMGC6ej4C3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10519
DYRK1ADYRKCMGC2wo6BAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3749
DYRK1ADYRKCMGC7a5bA4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman13756
DYRK1ADYRKCMGC5a54Cn-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6720
DYRK1ADYRKCMGC6yf8A~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13462
GSK3BGSKCMGC6tcuAA5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamideHuman12780
CDK2CDKCMGC1gijA1-(5-oxo-2,3,5,9b-tetrahydro-1h-pyrrolo[2,1-a]isoindol-9-yl)-3-(5-pyrrolidin-2-yl-1h-pyrazol-3-yl)-ureaHuman4542
CDK2CDKCMGC4eooCBadenosine-5'-triphosphateHuman4139
CDK2CDKCMGC2r3kAC3-bromo-5-phenyl-n-(pyrimidin-5-ylmethyl)pyrazolo[1,5-a]pyridin-7-amineHuman4022
CDK2CDKCMGC4eorCBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4487
CDK2CDKCMGC2vtqA{[(2,6-difluorophenyl)carbonyl]amino}-n-piperidin-4-yl-1h-pyrazole-3-carboxamideHuman3891
CDK2CDKCMGC9essAA(4-bromo-2-methoxyphenyl)methanolHuman15908
CDK2CDKCMGC4eonAA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman3902
CDK2CDKCMGC3s00AA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](5-chlorothiophen-2-yl)methanoneHuman4208
CDK2CDKCMGC3dogAA(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4541
CDK2CDKCMGC4fkqAA4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHuman3972
CDK2CDKCMGC9esjAC2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman15909
CDK2CDKCMGC1dm2AB4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHuman4024
CDK2CDKCMGC2r3pAB5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHuman4392
CDK2CDKCMGC2i40AA5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4363
CDK13 (CHED)CDKCMGC5efqCadenosine-5'-diphosphateHuman6324
DYRK1ADYRKCMGC7a51A4-azanyl-6-bromanyl-7-methyl-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13753
DYRK1ADYRKCMGC6eivC~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10542
DYRK1ADYRKCMGC3anqA(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3767
MAPK1 (Erk2)MAPKCMGC7opmAA1-[4-(hydroxymethyl)-1h-pyrazolo[4,3-c]pyridin-6-yl]-3-[(1s)-1-phenylethyl]ureaHuman14084
DYRK1ADYRKCMGC5a4eBBn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6726
DYRK1ADYRKCMGC2vx3BAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3766
DYRK1ADYRKCMGC4yljBA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3753
DYRK1ADYRKCMGC7ajaAA1-[4-(1-benzofuran-5-yl)pyridin-2-yl]piperazineHuman13610
DYRK1ADYRKCMGC4ylkAA10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3789
DYRK1ADYRKCMGC4yljDB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3793
DYRK1ADYRKCMGC6s14AA~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11418
CDK2CDKCMGC3eocC5-methyl-7-phenyl-n-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman3969
CDK2CDKCMGC9essAB(4-bromo-2-methoxyphenyl)methanolHuman15911
CDK2CDKCMGC5d1jAn-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)piperidine-4-carboxamideHuman4058
CDK2CDKCMGC6q4eAC6-iodanyl-7~{h}-purin-2-amineHuman11219
CDK2CDKCMGC3qtwAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4397
CDK2CDKCMGC2w05AAn-(2-methoxyethyl)-4-({4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)benzenesulfonamideHuman4547
CDK2CDKCMGC5oo3AB1-(4-ethyl-2,3-dihydroquinoxalin-1-yl)propan-1-oneHuman10568
CDK2CDKCMGC3f5xC4-{3-[7-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman3894
CDK2CDKCMGC3ti1ABn-[2-(diethylamino)ethyl]-5-[(z)-(5-fluoro-2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-2,4-dimethyl-1h-pyrrole-3-carboxamideHuman4213
CDK2CDKCMGC6q49AB-Human11220
DYRK1ADYRKCMGC4yu2BB(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3738
DYRK1ADYRKCMGC6eisDA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10547
DYRK1ADYRKCMGC6ln1A1,3,5,8-tetrakis(oxidanyl)xanthen-9-oneHuman13935
DYRK1ADYRKCMGC6t6aBA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11860
DYRK1ADYRKCMGC6qu2DB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12089
DYRK1ADYRKCMGC5a54Bn-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6716
DYRK1ADYRKCMGC2wo6BBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3739
DYRK1ADYRKCMGC7fhtAB(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14162
DYRK1ADYRKCMGC7ajwAB4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13611
DYRK1ADYRKCMGC7ajwAA4-[2-methyl-3-(2-phenoxyethyl)imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13612
DYRK1ADYRKCMGC6eijD~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10559
DYRK1ADYRKCMGC7a5nA5-(2-azanylpyridin-4-yl)-~{n}-[[2,6-bis(fluoranyl)phenyl]methyl]-2-methyl-7~{h}-pyrrolo[2,3-d]pyrimidin-4-amineHuman13757
DYRK1ADYRKCMGC6qu2BA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12086
MAPK14 (p38a)MAPKCMGC3fkoA3-(2-chlorophenyl)-6-(2-fluorophenoxy)-2h-indazoleHuman5075
GSK3BGSKCMGC1j1cBadenosine-5'-diphosphateHuman677
CDK2CDKCMGC2bkzA1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHuman3942
MAPK6 (Erk3)MAPKCMGC6ylcC5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12794
CSNK2A1 (CK2a1)CK2CMGC6hmeAA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11275
CSNK2A1 (CK2a1)CK2CMGC2pvrABphosphoaminophosphonic acid-adenylate esterHuman5505
CSNK2A1 (CK2a1)CK2CMGC5oquBBadenosine-5'-diphosphateHuman9678
MAPK10 (JNK3)MAPKCMGC4h36AA-Human3459
MAPK10 (JNK3)MAPKCMGC4kkeAadenosine monophosphateHuman3448
MAPK10 (JNK3)MAPKCMGC6emhDB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10496
MAPK10 (JNK3)MAPKCMGC6eq9BAphosphomethylphosphonic acid adenylate esterHuman10504
MAPK10 (JNK3)MAPKCMGC3cgfAn-cyclohexyl-4-imidazo[1,2-a]pyridin-3-yl-n-methylpyrimidin-2-amineHuman6770
MAPK10 (JNK3)MAPKCMGC4y5hA1-(trans-4-{[7-oxo-8-(propan-2-yl)-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl]amino}cyclohexyl)-3-propan-2-ylureaHuman3431
MAPK10 (JNK3)MAPKCMGC4whzAA3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamideHuman3429
MAPK10 (JNK3)MAPKCMGC8vo4A(4p)-4-{6-[(azetidin-1-yl)methyl]-5-(2-chloro-6-fluoroanilino)-1h-indazol-1-yl}-n-methylthiophene-2-carboxamideHuman15637
MAPK10 (JNK3)MAPKCMGC4w4wAn-(2-methylpyridin-4-yl)-3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}benzamideHuman3418
MAPK10 (JNK3)MAPKCMGC3v6rAB4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3436
MAPK10 (JNK3)MAPKCMGC2excXn-{2'-[(4-fluorophenyl)amino]-4,4'-bipyridin-2-yl}-4-methoxycyclohexanecarboxamideHuman3478
MAPK10 (JNK3)MAPKCMGC8vnxAA(4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamideHuman15638
MAPK10 (JNK3)MAPKCMGC3rtpAn-[4-cyano-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamideHuman3467
MAPK10 (JNK3)MAPKCMGC2wajAA1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinolineHuman3472
MAPK10 (JNK3)MAPKCMGC4w4vA3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamideHuman3437
MAPK10 (JNK3)MAPKCMGC3ttjAA9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamineHuman3458
MAPK10 (JNK3)MAPKCMGC3v6rBB4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3417
MAPK10 (JNK3)MAPKCMGC4x21Bn-ethyl-4-{[4-(1h-indol-3-yl)-5-iodopyrimidin-2-yl]amino}piperidine-1-carboxamideHuman6239
MAPK10 (JNK3)MAPKCMGC8wgfAAphosphoaminophosphonic acid-adenylate esterHuman15046
MAPK10 (JNK3)MAPKCMGC4z9lABphosphoaminophosphonic acid-adenylate esterHuman3438
MAPK10 (JNK3)MAPKCMGC6eq9BBphosphomethylphosphonic acid adenylate esterHuman10499
MAPK10 (JNK3)MAPKCMGC2p33A4-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}-n-ethylpiperidine-1-carboxamideHuman3455
HIPK3DYRKCMGC7o7iA-Human13996
CDK2CDKCMGC4acmAA3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman4247
CDK2CDKCMGC3wblAn~7~-(4-ethoxyphenyl)-6-methyl-n~5~-[(3s)-piperidin-3-yl]pyrazolo[1,5-a]pyrimidine-5,7-diamineHuman3895
CDK2CDKCMGC3rm7AB2-[(4-hydroxybenzyl)amino]-5-nitrobenzamideHuman4499
CDK2CDKCMGC4cfxCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4442
CDK2CDKCMGC3pxrAB-Human4173
CDK2CDKCMGC2r3hAA3-methyl-n-(pyridin-4-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman4152
CDK2CDKCMGC6q4eAA6-iodanyl-7~{h}-purin-2-amineHuman11199
CDK2CDKCMGC2r3jAB3-bromo-5-phenyl-n-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4544
CDK2CDKCMGC3s1hAB4-{[4-amino-5-(4-methoxybenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4226
CDK2CDKCMGC5if1AA-Human6568
CDK2CDKCMGC2iw9CBo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3858
CDK2CDKCMGC5lmkCB4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7397
CDK2CDKCMGC4cfwCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4549
CDK2CDKCMGC8curAB6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman14692
MAPK10 (JNK3)MAPKCMGC7kskA4-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13386
MAPK10 (JNK3)MAPKCMGC1pmvA2,6-dihydroanthra/1,9-cd/pyrazol-6-oneHuman3434
MAPK10 (JNK3)MAPKCMGC4h3bCC-Human3446
MAPK10 (JNK3)MAPKCMGC4h3bAB-Human3454
MAPK10 (JNK3)MAPKCMGC8bzpAB2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamideHuman14858
MAPK10 (JNK3)MAPKCMGC3ttiAtrans-4-({9-[(3s)-tetrahydrofuran-3-yl]-8-[(2,4,6-trifluorophenyl)amino]-9h-purin-2-yl}amino)cyclohexanolHuman3456
MAPK10 (JNK3)MAPKCMGC4whzAB3-(4-{[(2-chlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-{1-[(3s)-pyrrolidin-3-yl]-1h-pyrazol-4-yl}benzamideHuman3422
MAPK10 (JNK3)MAPKCMGC6emhBA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10506
MAPK10 (JNK3)MAPKCMGC3g9lX(3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-[(e)-2-phenylethenyl]-1h-indole-2,3-dione 3-oximeHuman3435
MAPK10 (JNK3)MAPKCMGC8vnxAB(4p)-4-[5-(2-chloro-6-fluoroanilino)-6-(methoxymethyl)-1h-indazol-1-yl]-n-methylthiophene-2-carboxamideHuman15639
MAPK10 (JNK3)MAPKCMGC4h39AB-Human3462
MAPK10 (JNK3)MAPKCMGC3v6sAB3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3449
MAPK10 (JNK3)MAPKCMGC3fi2AB3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHuman3452
MAPK10 (JNK3)MAPKCMGC6emhDA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10497
MAPK10 (JNK3)MAPKCMGC2zduA4-[(4-{[6-bromo-3-(methoxycarbonyl)-1-oxo-4-phenylisoquinolin-2(1h)-yl]methyl}phenyl)amino]-4-oxobutanoic acidHuman3479
MAPK10 (JNK3)MAPKCMGC6emhAB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10503
MAPK10 (JNK3)MAPKCMGC2zdtAB4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acidHuman3424
MAPK10 (JNK3)MAPKCMGC7orfABn-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamideHuman13814
MAPK10 (JNK3)MAPKCMGC4u79An-{4-[(3-{2-[(trans-4-aminocyclohexyl)amino]pyrimidin-4-yl}pyridin-2-yl)oxy]naphthalen-1-yl}benzenesulfonamideHuman3466
MAPK10 (JNK3)MAPKCMGC3v6sBB3-{[4-(dimethylamino)butanoyl]amino}-n-(4-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3425
MAPK10 (JNK3)MAPKCMGC3kvxAAn-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)anilineHuman3433
MAPK10 (JNK3)MAPKCMGC8enjAn-[3-({(4p)-4-[(3m)-1-tert-butyl-3-(3-hydroxyphenyl)-1h-pyrazol-4-yl]pyridin-2-yl}amino)propyl]-4-hydroxybenzene-1-sulfonamideHuman14884
MAPK10 (JNK3)MAPKCMGC2zdtAA4-[(6-chloro-1-oxo-4-phenyl-3-propanoylisoquinolin-2(1h)-yl)methyl]benzoic acidHuman3421
MAPK10 (JNK3)MAPKCMGC4h3bCB-Human3465
MAPK10 (JNK3)MAPKCMGC8bzpAA2-bromanyl-2,2-bis(fluoranyl)-~{n}-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)ethanamideHuman14859
DYRK1ADYRKCMGC6yf8B~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13461
SRPK1SRPKCMGC6fadD-Human11637
SRPK1SRPKCMGC7zksABn-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamideHuman14618
SRPK1SRPKCMGC7pqsAB~{n}-[3-[[[2-(6-chloranyl-7-fluoranyl-1~{h}-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-~{n}-methyl-methanesulfonamideHuman14015
SRPK1SRPKCMGC6fadA-Human11638
MAPK10 (JNK3)MAPKCMGC7yl1A7-hexyl-3-methyl-8-sulfanylidene-9h-purine-2,6-dioneHuman14845
MAPK10 (JNK3)MAPKCMGC3v6rAA4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3441
MAPK10 (JNK3)MAPKCMGC8wgfABphosphoaminophosphonic acid-adenylate esterHuman15047
MAPK10 (JNK3)MAPKCMGC2o0uAn-{3-cyano-6-[3-(1-piperidinyl)propanoyl]-4,5,6,7-tetrahydrothieno[2,3-c]pyridin-2-yl}1-naphthalenecarboxamideHuman3415
MAPK10 (JNK3)MAPKCMGC3fi3AA3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHuman3442
MAPK10 (JNK3)MAPKCMGC3fi3AB3-{5-[(2-fluorophenyl)amino]-1h-indazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHuman3445
SRPK1SRPKCMGC7pqsAA~{n}-[3-[[[2-(6-chloranyl-7-fluoranyl-1~{h}-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-~{n}-methyl-methanesulfonamideHuman14014
SRPK1SRPKCMGC5xv7A9-ethyl-6,6-dimethyl-8-[4-(morpholin-4-yl)piperidin-1-yl]-11-oxo-6,11-dihydro-5h-benzo[b]carbazole-3-carbonitrileHuman9727
CDK9CDKCMGC4imyCAadenosine monophosphateHuman2237
MAPK1 (Erk2)MAPKCMGC6g97AA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-oneHuman9960
CDK2CDKCMGC2cchABadenosine-5'-triphosphateHuman4553
CSNK2A1 (CK2a1)CK2CMGC7a4qAB2-methoxyimino-5-(quinolin-6-ylmethyl)-1,3-thiazol-4-oneHuman14239
CDK2CDKCMGC8oy2A(1s,2s,11as)-1-methoxy-1,4,7,10-tetramethyl-2,9-bis(oxidanyl)-2,11a-dihydrobenzo[b][1,4]benzodioxepine-3,6-dioneHuman15078
CDK13 (CHED)CDKCMGC5efqAadenosine-5'-diphosphateHuman6323
MAPK7 (Erk5)MAPKCMGC4b99A11-cyclopentyl-2-[[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl-phenyl]amino]-5-methyl-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman388
MAPK8 (JNK1)MAPKCMGC8x5mAB3-[4-(dimethylamino)butanoylamino]-~{n}-[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamideHuman15100
MAPK1 (Erk2)MAPKCMGC4fv3AAethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman2617
CDK7CDKCMGC1ua2Dadenosine-5'-triphosphateHuman543
MAPK14 (p38a)MAPKCMGC3oefXA-Human5163
MAPK14 (p38a)MAPKCMGC4e5aXB-Human5222
MAPK14 (p38a)MAPKCMGC6qdzAB1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ureaHuman11958
HIPK2DYRKCMGC7ncfA3-(4-tert-butylphenyl)-5-(1h-pyrazol-4-yl)furo[3,2-b]pyridineHuman13393
CSNK2A2 (CK2a2)CK2CMGC5yf9XBnicotinic acidHuman11414
MAPK14 (p38a)MAPKCMGC3zyaAB2-amino-phenylamino-dibenzosuberoneHuman5089
MAPK14 (p38a)MAPKCMGC4ewqAA3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazineHuman5200
MAPK14 (p38a)MAPKCMGC4kiqBethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5013
MAPK14 (p38a)MAPKCMGC3zsiAB5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman4983
MAPK14 (p38a)MAPKCMGC3hp2AB1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-oneHuman5031
MAPK14 (p38a)MAPKCMGC3kq7AAn-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamideHuman5081
MAPK14 (p38a)MAPKCMGC3uvqABn-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamideHuman5214
MAPK14 (p38a)MAPKCMGC5omhA1-(3-chlorophenyl)-3-methyl-4~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxideHuman11251
MAPK14 (p38a)MAPKCMGC4ehvAA-Human4997
MAPK14 (p38a)MAPKCMGC3mw1A8-(2,6-dichlorophenyl)-4-(2,4-difluorophenyl)-2-piperidin-4-yl-1,7-naphthyridine 7-oxideHuman5072
MAPK14 (p38a)MAPKCMGC1zzlA6-[4-(4-fluorophenyl)-1,3-oxazol-5-yl]-3-isopropyl[1,2,4]triazolo[4,3-a]pyridineHuman5249
MAPK14 (p38a)MAPKCMGC3gfeAn-cyclopropyl-3-{[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-4-yl]amino}-4-methylbenzamideHuman4991
MAPK14 (p38a)MAPKCMGC1bmkA4-(fluorophenyl)-1-cyclopropylmethyl-5-(2-amino-4-pyrimidinyl)imidazoleHuman5235
MAPK1 (Erk2)MAPKCMGC1tvoA5-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)-1h-pyrazolo[3,4-c]pyridazin-3-amineHuman2581
MAPK14 (p38a)MAPKCMGC3flyA6-(2,4-difluorophenoxy)-8-methyl-2-[(1-methylethyl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5113
MAPK14 (p38a)MAPKCMGC3lffAB(4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acidHuman5120
MAPK14 (p38a)MAPKCMGC3lfeA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-4-ylmethoxy)ethyl]-1,3-thiazol-2-yl}ureaHuman5173
MAPK14 (p38a)MAPKCMGC6qdzAA1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{s})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ureaHuman11956
MAPK14 (p38a)MAPKCMGC4eh8AA[3-(benzyloxy)phenyl]methanolHuman4978
MAPK14 (p38a)MAPKCMGC2lgcA8-Human5078
MAPK14 (p38a)MAPKCMGC3lfaAn-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamideHuman5018
MAPK14 (p38a)MAPKCMGC2onlB-Human5007
MAPK14 (p38a)MAPKCMGC4aa0ABn-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamideHuman5132
MAPK14 (p38a)MAPKCMGC3mh1A-Human5003
MAPK14 (p38a)MAPKCMGC3mptABn-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamideHuman5246
MAPK14 (p38a)MAPKCMGC5xyyA3-(5-{[(2-chloro-6-fluorophenyl)methyl]amino}-4h-1,2,4-triazol-3-yl)phenolHuman9513
MAPK14 (p38a)MAPKCMGC3d7zAAn~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamideHuman5247
MAPK14 (p38a)MAPKCMGC3nwwA1-[2-(2-{[2-(dimethylamino)ethyl]amino}-6-{2-[(1-methylethyl)amino]-1,3-thiazol-5-yl}pyrimidin-4-yl)benzyl]-3-ethylureaHuman5068
MAPK14 (p38a)MAPKCMGC5wjjABn-{4-[2-(4-fluoro-3-methylphenyl)imidazo[1,2-b]pyridazin-3-yl]pyridin-2-yl}-2-methyl-1-oxo-1lambda~5~-pyridine-4-carboxamideHuman9516
MAPK14 (p38a)MAPKCMGC2okrA-Human5136
MAPK14 (p38a)MAPKCMGC3kf7A3-{6-[2-(2,4-difluorophenyl)ethyl][1,2,4]triazolo[4,3-a]pyridin-3-yl}-4-methylbenzamideHuman5201
MAPK14 (p38a)MAPKCMGC3hucABn-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamideHuman5111
MAPK14 (p38a)MAPKCMGC3gc7AB5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman5256
MAPK14 (p38a)MAPKCMGC6zwpAB5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman12698
MAPK14 (p38a)MAPKCMGC1oz1AA3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-olHuman5230
MAPK14 (p38a)MAPKCMGC2baqA[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanoneHuman5184
MAPK14 (p38a)MAPKCMGC3uvpABn-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamideHuman5155
MAPK14 (p38a)MAPKCMGC3mgyA-Human5171
MAPK14 (p38a)MAPKCMGC3lfbAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)ureaHuman4998
MAPK14 (p38a)MAPKCMGC3nnvAB1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylureaHuman5046
MAPK14 (p38a)MAPKCMGC3zs5AB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman4977
MAPK14 (p38a)MAPKCMGC3hv3AA1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5012
MAPK14 (p38a)MAPKCMGC3mvmA4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman4993
MAPK14 (p38a)MAPKCMGC4kinA5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5237
MAPK14 (p38a)MAPKCMGC6zqsA2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-oneHuman12986
MAPK14 (p38a)MAPKCMGC3fmmA6-(2,4-difluorophenoxy)-n-[(1r)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman5186
CDK2CDKCMGC3qwkAB4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4155
CSNK2A2 (CK2a2)CK2CMGC6qy8BB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12121
MAPK14 (p38a)MAPKCMGC4kinD5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5144
MAPK14 (p38a)MAPKCMGC6sfkAA~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamideHuman11617
MAPK14 (p38a)MAPKCMGC3odzX-Human5069
MAPK14 (p38a)MAPKCMGC4fa2AAtrans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanolHuman5150
MAPK14 (p38a)MAPKCMGC3fc1X5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman5110
MAPK14 (p38a)MAPKCMGC3e92An-cyclopropyl-2',6-dimethyl-4'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-3-carboxamideHuman5149
MAPK14 (p38a)MAPKCMGC8yd9AB-Human15696
MAPK14 (p38a)MAPKCMGC3hv4B1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5064
MAPK14 (p38a)MAPKCMGC9r27A4-[4-[[4-chloranyl-3-(trifluoromethyl)phenyl]carbamoylamino]-3-fluoranyl-phenoxy]-~{n}-methyl-pyridine-2-carboxamideHuman15697
MAPK14 (p38a)MAPKCMGC1wbnAn-(3-tert-butyl-1h-pyrazol-5-yl)-n'-{4-chloro-3-[(pyridin-3-yloxy)methyl]phenyl}ureaHuman5257
MAPK14 (p38a)MAPKCMGC3rocA3-{5-chloro-4-[(2,4-difluorobenzyl)oxy]-6-oxopyrimidin-1(6h)-yl}-n-(2-hydroxyethyl)-4-methylbenzamideHuman5011
MAPK14 (p38a)MAPKCMGC3gcpAA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5194
MAPK14 (p38a)MAPKCMGC3hv6A1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[4-(2-morpholin-4-ylethoxy)phenyl]ureaHuman5101
MAPK14 (p38a)MAPKCMGC2yiwA1-(3-tert-butyl-1-phenyl-1h-pyrazol-5-yl)-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)ureaHuman4988
MAPK14 (p38a)MAPKCMGC4e6cA-Human5015
MAPK14 (p38a)MAPKCMGC1di9A4-[3-methylsulfanylanilino]-6,7-dimethoxyquinazolineHuman5251
MAPK14 (p38a)MAPKCMGC3gcqAB1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5053
MAPK14 (p38a)MAPKCMGC2lgcA5-Human5107
MAPK14 (p38a)MAPKCMGC3l8xAn,4-dimethyl-3-[(1-phenyl-1h-pyrazolo[3,4-d]pyrimidin-4-yl)amino]benzamideHuman5041
MAPK14 (p38a)MAPKCMGC8a8mAphosphomethylphosphonic acid adenosyl esterHuman14289
MAPK14 (p38a)MAPKCMGC5etcA-Human6361
MAPK14 (p38a)MAPKCMGC1wfcA-Human4989
MAPK14 (p38a)MAPKCMGC3e93AB4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamideHuman5004
MAPK14 (p38a)MAPKCMGC3gcuBA1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5175
DYRK1ADYRKCMGC8c3gAAn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15155
DYRK1ADYRKCMGC8c3rAAgossypinHuman15156
DYRK1ADYRKCMGC8c3rABgossypinHuman15157
DYRK1ADYRKCMGC8c3gABn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15153
DYRK1ADYRKCMGC8c3qABrutinHuman15154
MAPK14 (p38a)MAPKCMGC1yqjA6((s)-3-benzylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyrazineHuman5152
MAPK14 (p38a)MAPKCMGC9cj5ApexmetinibHuman15698
MAPK14 (p38a)MAPKCMGC5o8uA-Human8381
MAPK14 (p38a)MAPKCMGC4e8aA-Human4979
MAPK14 (p38a)MAPKCMGC3mpaA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5026
MAPK14 (p38a)MAPKCMGC6tcaHBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12487
MAPK14 (p38a)MAPKCMGC2npqA-Human5205
CLK3CLKCMGC6khfAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11650
DYRK1ADYRKCMGC8c3qAArutinHuman15158
MAPK14 (p38a)MAPKCMGC5xyxABn-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amineHuman9517
MAPK14 (p38a)MAPKCMGC3gcuAA1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5032
MAPK14 (p38a)MAPKCMGC3hvcA4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridineHuman5054
MAPK14 (p38a)MAPKCMGC4a9yAn-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamideHuman5073
MAPK14 (p38a)MAPKCMGC4r3cAB6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazineHuman5036
MAPK14 (p38a)MAPKCMGC1wbwA3-(1-naphthylmethoxy)pyridin-2-amineHuman5179
CDK6CDKCMGC8i0mA2-[(4-azanylcyclohexyl)amino]-7-cyclopentyl-~{n},~{n}-dimethyl-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman15164
MAPK14 (p38a)MAPKCMGC4eh7AA(3-phenoxyphenyl)methanolHuman5208
MAPK14 (p38a)MAPKCMGC3odyX-Human5233
MAPK14 (p38a)MAPKCMGC1wboA2-chlorophenolHuman5039
DYRK1BDYRKCMGC8c2zAAn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15180
DYRK1BDYRKCMGC8c2zABn-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineHuman15181
MAPK14 (p38a)MAPKCMGC8yd9AA-Human15699
MAPK14 (p38a)MAPKCMGC3d83An-{4'-[(cyclopropylmethyl)carbamoyl]-6-methylbiphenyl-3-yl}-2-morpholin-4-ylpyridine-4-carboxamideHuman5028
MAPK14 (p38a)MAPKCMGC6anlAAtak-715Human9515
DYRK3DYRKCMGC5y86A7-methoxy-1-methyl-9h-beta-carbolineHuman9876
CLK1CLKCMGC6g33BA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9821
CLK1CLKCMGC6zlnAB4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman12710
MAPK14 (p38a)MAPKCMGC3mvlA4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5060
MAPK14 (p38a)MAPKCMGC2lgcA3-Human5040
MAPK14 (p38a)MAPKCMGC4e5aXA-Human5189
MAPK14 (p38a)MAPKCMGC3iw5An-[2-(3-{[2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-2-oxoethyl]sulfanyl}-1h-indol-1-yl)ethyl]-3-(trifluoromethyl)benzamideHuman5076
MAPK14 (p38a)MAPKCMGC4kinC5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5142
MAPK14 (p38a)MAPKCMGC3fskA3-(2-chlorophenyl)-7-[(trans-4-hydroxycyclohexyl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman5008
MAPK14 (p38a)MAPKCMGC1oveAC1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-oneHuman5199
MAPK14 (p38a)MAPKCMGC6zwpAA5-azanyl-~{n}-[[4-[[(2~{s})-4-cyclohexyl-1-[(4-fluorophenyl)amino]-1-oxidanylidene-butan-2-yl]carbamoyl]phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman12699
MAPK14 (p38a)MAPKCMGC3lhjAn-cyclopropyl-3-[1-(2,4-difluorophenyl)-7-methyl-6-oxo-6,7-dihydro-1h-pyrazolo[3,4-b]pyridin-5-yl]-4-methylbenzamideHuman5234
CLK1CLKCMGC6i5kAB5-(1-methylpyrazol-4-yl)-3-(3-propan-2-yloxyphenyl)furo[3,2-b]pyridineHuman10836
MAPK14 (p38a)MAPKCMGC4kipB2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamideHuman5180
MAPK14 (p38a)MAPKCMGC3fl4A6-(2,4-difluorophenoxy)-3-(2-methylphenyl)-1h-pyrazolo[3,4-d]pyrimidineHuman5151
MAPK14 (p38a)MAPKCMGC3s4qA3-[(6-benzoyl-5-methylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]-n-cyclopropyl-4-methylbenzamideHuman5133
MAPK14 (p38a)MAPKCMGC2zazAB4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehydeHuman5034
MAPK14 (p38a)MAPKCMGC3lfcA(4-{5-[({4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}carbamoyl)amino]-3-tert-butyl-1h-pyrazol-1-yl}phenyl)acetic acidHuman5160
CLK1CLKCMGC6i5iAB5-(1-methylpyrazol-4-yl)-3-[1-(phenylmethyl)pyrazol-4-yl]furo[3,2-b]pyridineHuman10840
CLK1CLKCMGC6khdCB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11643
MAPK14 (p38a)MAPKCMGC2zb1AAn-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamideHuman5038
MAPK14 (p38a)MAPKCMGC4f9yABn,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5017
MAPK14 (p38a)MAPKCMGC3ocgA5-amino-n-[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]-1-phenyl-1h-pyrazole-4-carboxamideHuman4984
MAPK14 (p38a)MAPKCMGC2balA[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl][3-(piperidin-4-yloxy)phenyl]methanoneHuman5260
MAPK14 (p38a)MAPKCMGC5etaB-Human7137
MAPK14 (p38a)MAPKCMGC2fstXB-Human5195
MAPK14 (p38a)MAPKCMGC3hv3AB1-{4-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5232
MAPK14 (p38a)MAPKCMGC4aa0AAn-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]-2-morpholin-4-yl-pyridine-4-carboxamideHuman5213
MAPK14 (p38a)MAPKCMGC3flnC6-(2,4-difluorophenoxy)-8-methyl-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5090
MAPK14 (p38a)MAPKCMGC3hv5BB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5137
MAPK14 (p38a)MAPKCMGC3gi3An-{5-tert-butyl-2-methoxy-3-[({4-[6-(morpholin-4-ylmethyl)pyridin-3-yl]naphthalen-1-yl}carbamoyl)amino]phenyl}methanesulfonamideHuman5226
MAPK14 (p38a)MAPKCMGC6sfiAB~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamideHuman11619
MAPK14 (p38a)MAPKCMGC6tcaFAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12489
MAPK14 (p38a)MAPKCMGC3hp2AA1-benzyl-4-(benzyloxy)-3-bromopyridin-2(1h)-oneHuman5217
MAPK14 (p38a)MAPKCMGC5mtxAA3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamideHuman8382
MAPK14 (p38a)MAPKCMGC3nnxA2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamideHuman5002
MAPK14 (p38a)MAPKCMGC3ds6Bn-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5188
MAPK14 (p38a)MAPKCMGC4l8mAAn-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamideHuman5005
MAPK14 (p38a)MAPKCMGC2bakAn-(3-{[7-methoxy-6-(2-pyrrolidin-1-ylethoxy)quinazolin-4-yl]amino}-4-methylphenyl)-2-morpholin-4-ylisonicotinamideHuman5114
MAPK14 (p38a)MAPKCMGC2fsmX-Human5044
MAPK14 (p38a)MAPKCMGC9cj2AA-Human15700
MAPK14 (p38a)MAPKCMGC3zshAA2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamideHuman5216
MAPK14 (p38a)MAPKCMGC3hv5AB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5263
MAPK14 (p38a)MAPKCMGC1oukA4-[5-[2-(1-phenyl-ethylamino)-pyrimidin-4-yl]-1-methyl-4-(3-trifluoromethylphenyl)-1h-imidazol-2-yl]-piperidineHuman5146
MAPK14 (p38a)MAPKCMGC3hl7A2-{4-[5-(4-chlorophenyl)-4-pyrimidin-4-yl-1h-pyrazol-3-yl]piperidin-1-yl}-2-oxoethanolHuman5236
MAPK14 (p38a)MAPKCMGC6ohdAB3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamideHuman11819
MAPK14 (p38a)MAPKCMGC4kipA2-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-1,3-thiazole-5-carboxamideHuman5159
MAPK14 (p38a)MAPKCMGC3ds6Cn-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5182
MAPK14 (p38a)MAPKCMGC2lgcA9-Human5127
MAPK14 (p38a)MAPKCMGC3hllAA3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamideHuman5115
MAPK14 (p38a)MAPKCMGC4l8mABn-[2-fluoro-5-({9-[2-(morpholin-4-yl)ethoxy]-11-oxo-6,11-dihydrodibenzo[b,e]oxepin-3-yl}amino)phenyl]benzamideHuman4992
MAPK14 (p38a)MAPKCMGC3fmlA6-(2,4-difluorophenoxy)-n-[(1s)-1-methyl-2-(methylsulfonyl)ethyl]-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman5010
MAPK14 (p38a)MAPKCMGC3fmjA4-(5-methyl-3-phenylisoxazol-4-yl)pyrimidin-2-amineHuman5129
MAPK14 (p38a)MAPKCMGC6m9lA3-benzyl-6-[(2,4-difluorophenyl)amino]-1,3-dihydro-2h-imidazo[4,5-b]pyridin-2-oneHuman11255
MAPK14 (p38a)MAPKCMGC2y8oAB-Human5030
MAPK14 (p38a)MAPKCMGC3fmnAB6-(2,4-difluorophenoxy)-n-(tetrahydro-2h-pyran-4-yl)-1h-pyrazolo[3,4-d]pyrimidin-3-amineHuman4995
CDK4CDKCMGC3g33A-Human3387
MAPK14 (p38a)MAPKCMGC3hp5A5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman5158
MAPK14 (p38a)MAPKCMGC3hegAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5218
MAPK14 (p38a)MAPKCMGC9cj4AC1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman15706
MAPK14 (p38a)MAPKCMGC4kinB5-(2-chlorophenyl)-n-[5-(cyclopropylcarbamoyl)-2-methylphenyl]thiophene-2-carboxamideHuman5131
MAPK14 (p38a)MAPKCMGC1kv2A1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman5255
MAPK14 (p38a)MAPKCMGC3fmhA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5024
MAPK14 (p38a)MAPKCMGC3flwA6-(2,4-difluorophenoxy)-2-{[3-hydroxy-1-(2-hydroxyethyl)propyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-oneHuman5153
MAPK14 (p38a)MAPKCMGC4kiqDethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5016
MAPK14 (p38a)MAPKCMGC4ehvAB-Human4981
MAPK14 (p38a)MAPKCMGC3mh0A-Human5124
MAPK14 (p38a)MAPKCMGC3hecAB4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman5035
MAPK1 (Erk2)MAPKCMGC6qa1AApyridin-2-amineHuman11352
MAPK1 (Erk2)MAPKCMGC5nhoA(6~{s})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7993
MAPK1 (Erk2)MAPKCMGC4h3pDphosphoaminophosphonic acid-adenylate esterHuman2575
MAPK1 (Erk2)MAPKCMGC5bvdAA2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-7-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]-3,4-dihydropyrrolo[1,2-a]pyrazin-1(2h)-oneHuman6030
CSNK2A1 (CK2a1)CK2CMGC5m4iA4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7400
CSNK2A1 (CK2a1)CK2CMGC5modAA-Human7678
MAPK1 (Erk2)MAPKCMGC7nr3AB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-oneHuman13922
MAPK1 (Erk2)MAPKCMGC7nqwAA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-oneHuman13927
MAPK1 (Erk2)MAPKCMGC7nqqAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(hydroxymethyl)-2,3-dihydroinden-1-yl]ethanamideHuman13928
MAPK1 (Erk2)MAPKCMGC7nr8AB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-[6-(4-methylpiperazin-1-yl)pyridin-2-yl]-2-oxidanyl-ethyl]propanamideHuman13929
MAPK1 (Erk2)MAPKCMGC7w5oA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman14110
MAPK1 (Erk2)MAPKCMGC7auvAB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13930
MAPK1 (Erk2)MAPKCMGC7nr9AB(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(2-methoxypyridin-4-yl)-2-oxidanyl-ethyl]propanamideHuman13931
MAPK1 (Erk2)MAPKCMGC4qp7B2-(1h-pyrazol-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6093
MAPK1 (Erk2)MAPKCMGC6g9aAB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-morpholin-4-ylethyl)-3~{h}-isoindol-1-oneHuman11412
CSNK2A1 (CK2a1)CK2CMGC6q4qACbenzoic acidHuman11277
CSNK2A1 (CK2a1)CK2CMGC5otpBA-Human10602
MAPK1 (Erk2)MAPKCMGC4nifEBphosphoaminophosphonic acid-adenylate esterHuman2591
CDK6CDKCMGC2f2cB(2s)-2-({6-[(3-amino-5-chlorophenyl)amino]-9-isopropyl-9h-purin-2-yl}amino)-3-methylbutan-1-olHuman2795
CDK6CDKCMGC4auaA1h-benzimidazol-2-yl(1h-pyrrol-2-yl)methanoneHuman2801
CSNK2A1 (CK2a1)CK2CMGC5oueBA(3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-imidazol-4-yl)ethyl]azaniumHuman9635
CSNK2A1 (CK2a1)CK2CMGC6ehuBA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamineHuman9630
CSNK2A1 (CK2a1)CK2CMGC5otyAAtrifluoroacetic acidHuman9692
CSNK2A1 (CK2a1)CK2CMGC5ouuBA2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman9657
CSNK2A1 (CK2a1)CK2CMGC3qa0BB-Human5528
MAPK1 (Erk2)MAPKCMGC7auvAA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13925
CSNK2A1 (CK2a1)CK2CMGC3h30BB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman5480
CSNK2A1 (CK2a1)CK2CMGC7b8iBB-Human13262
CSNK2A1 (CK2a1)CK2CMGC5ctpAAn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7304
CSNK2A1 (CK2a1)CK2CMGC6hotAA(2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enalHuman11667
CSNK2A1 (CK2a1)CK2CMGC4md8E-Human5439
CLK1CLKCMGC7o9yA4-(1~{h}-indol-3-yl)pyrimidin-2-amineHuman14208
DYRK1ADYRKCMGC7fhsAB(5~{z})-5-[(3-ethoxy-4-oxidanyl-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14159
DYRK1ADYRKCMGC6qu2CA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12090
DYRK1ADYRKCMGC4azeB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3768
MAPK10 (JNK3)MAPKCMGC3fi2AA3-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-1-yl}-n-(3,4,5-trimethoxyphenyl)benzamideHuman3463
MAPK10 (JNK3)MAPKCMGC4h3bAC-Human3453
MAPK10 (JNK3)MAPKCMGC3fv8AA5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamideHuman3468
MAPK10 (JNK3)MAPKCMGC6emhCA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10507
CSNK2A1 (CK2a1)CK2CMGC6tllAA4,5,6,7-tetrabromobenzotriazoleHuman13093
CSNK2A1 (CK2a1)CK2CMGC5otpAA2-[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman10588
CSNK2A1 (CK2a1)CK2CMGC5clpAA2-(3,4-dichlorophenyl)ethanamineHuman6922
MAPK10 (JNK3)MAPKCMGC3kvxABn-[(2z)-4-(3-fluoro-5-morpholin-4-ylphenyl)pyrimidin-2(1h)-ylidene]-4-(3-morpholin-4-yl-1h-1,2,4-triazol-1-yl)anilineHuman3430
MAPK8 (JNK1)MAPKCMGC3pzeA3-(carbamoylamino)-5-phenylthiophene-2-carboxamideHuman4642
GSK3BGSKCMGC6hk3BB3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11424
GSK3BGSKCMGC3f7zAA2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman743
GSK3BGSKCMGC9hm1An-(4-{5-[(2-aminoethyl)sulfamoyl]thiophen-2-yl}pyridin-2-yl)cyclopropanecarboxamideHuman15792
GSK3BGSKCMGC6hk4BA3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11430
GSK3BGSKCMGC1q3dAstaurosporineHuman705
GSK3BGSKCMGC3zrmBA7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman753
CDK2CDKCMGC6yl6AB-Human12495
CDK2CDKCMGC1pxmAB-Human3936
CDK2CDKCMGC8curAA6-[(e)-2-(4-chlorophenyl)ethenyl]-2-{[(2r)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman14693
CDK2CDKCMGC4cfmCA6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4260
CDK2CDKCMGC4d1xA(4s)-2-(6-hydroxy-1,3-benzothiazol-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHuman4344
CDK2CDKCMGC8ru8AB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman15328
CDK2CDKCMGC4bckAC3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4433
CDK2CDKCMGC4cfxAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman3963
CDK2CDKCMGC1oiyAB4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman3945
CDK2CDKCMGC4cfwAC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4141
CDK2CDKCMGC2vthA5-hydroxynaphthalene-1-sulfonamideHuman4274
CDK2CDKCMGC2x1nAA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman4579
CDK2CDKCMGC4bckAA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4095
CDK2CDKCMGC1hclAB-Human4540
CDK2CDKCMGC4bcnAA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4084
CDK2CDKCMGC3r9nAB[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](3-nitrophenyl)methanoneHuman3867
CDK2CDKCMGC3qqlAB(5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4378
CDK2CDKCMGC7nvqAstaurosporineHuman13627
CDK2CDKCMGC1h07AB((2-bromo-4-methylphenyl){6-[(4-{[(2s)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHuman3908
CDK2CDKCMGC5uq1A-Human8220
CDK2CDKCMGC2uueA4-methyl-5-{(2e)-2-[(4-morpholin-4-ylphenyl)imino]-2,5-dihydropyrimidin-4-yl}-1,3-thiazol-2-amineHuman4515
CDK2CDKCMGC4fkiAAn-(5-cyclopropyl-1h-pyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamideHuman4430
CDK2CDKCMGC4cfmAB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman3986
CDK2CDKCMGC2c6tA4-{[5-(cyclohexyloxy)[1,2,4]triazolo[1,5-a]pyrimidin-7-yl]amino}benzenesulfonamideHuman4371
CDK2CDKCMGC6guhAA4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10765
CDK2CDKCMGC2xnbAB3,4-dimethyl-5-(2-{[(1z)-4-piperazin-1-ylcyclohexa-2,4-dien-1-ylidene]amino}pyrimidin-4-yl)-1,3-thiazol-2(3h)-oneHuman4034
CDK2CDKCMGC4bcqCA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman3996
CDK2CDKCMGC5osjAB-Human9742
CDK2CDKCMGC6yl1ABmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12496
CDK2CDKCMGC3rzbAA4-amino-2-(phenylamino)-1,3-thiazole-5-carboxamideHuman4264
CDK2CDKCMGC2xmyAA4-[4-(3,4-dimethyl-2-oxo-2,3-dihydro-thiazol-5-yl)-pyrimidin-2-ylamino]-n-(2-methoxy-ethyl)-benzenesulfonamideHuman4526
CDK2CDKCMGC2cchAC-Human4566
CDK2CDKCMGC3raiAB4-{[3-(morpholin-4-yl)propyl]amino}-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4002
GSK3BGSKCMGC3f7zBB2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman670
GSK3BGSKCMGC6v6lAA1-(6-((2-((6-amino-5-nitropyridin-2-yl)amino)ethyl)amino)-2-(2,4-dichlorophenyl)pyridin-3-yl)-4-methylpiperazin-2-oneHuman11913
GSK3BGSKCMGC3f88BA5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman744
CDK12 (CRK7)CDKCMGC8bu6B~{n}-(1~{h}-benzimidazol-2-ylmethyl)-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman14921
CDK12 (CRK7)CDKCMGC9fmrB~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman15854
MAPK13 (p38d)MAPKCMGC4ynoA-Human2947
MAPK8 (JNK1)MAPKCMGC8pt9Amethyl (1s,3s)-1-methyl-3-[[3-[[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]carbamoyl]-4-oxidanylidene-cyclohexane-1-carboxylateHuman15293
MAPK8 (JNK1)MAPKCMGC8ptaAmethyl (1r,3s)-1-methyl-3-[[3-[[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]carbamoyl]-4-oxidanylidene-cyclohexane-1-carboxylateHuman15294
MAPK8 (JNK1)MAPKCMGC8pt8Amethyl (1r,3r)-1-methyl-3-[[3-[[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]carbamoyl]phenyl]methylcarbamoyl]-4-oxidanylidene-cyclohexane-1-carboxylateHuman15295
MAPK1 (Erk2)MAPKCMGC8pswABamp phosphoramidateHuman15303
MAPK1 (Erk2)MAPKCMGC8pt3AAphosphoaminophosphonic acid-adenylate esterHuman15304
CDK6CDKCMGC6oqoAn-[5-(6-ethyl-2,6-diazaspiro[3.3]heptan-2-yl)pyridin-2-yl]-5-fluoro-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12646
CDK6CDKCMGC9d8uAatirmociclibHuman15857
CDK6CDKCMGC1g3nA-Human2806
CDK6CDKCMGC1bi7A-Human2798
CDK6CDKCMGC1blxA-Human2802
CDK6CDKCMGC1bi8A-Human2796
CDK6CDKCMGC6oqlA5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4r)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12647
CDK6CDKCMGC9pe7A(3r,4r)-4-({(4m)-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-1,3-benzimidazol-6-yl]pyrimidin-2-yl}amino)-1-(methanesulfonyl)piperidin-3-olHuman15858
CDK6CDKCMGC1jowB-Human2793
CDK6CDKCMGC1bi8C-Human2799
CDK6CDKCMGC4ez5A{5-[4-(dimethylamino)piperidin-1-yl]-1h-imidazo[4,5-b]pyridin-2-yl}[2-(isoquinolin-4-yl)pyridin-4-yl]methanoneHuman2800
CDK6CDKCMGC2eufB6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman2804
CDK6CDKCMGC1xo2B3,7,3',4'-tetrahydroxyflavoneHuman2794
CDK2CDKCMGC1w0xCBolomoucineHuman4478
CDK2CDKCMGC1h01AA(2r)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman3974
CDK2CDKCMGC6p3wCB-Human11516
CDK2CDKCMGC1h07AA((2-bromo-4-methylphenyl){6-[(4-{[(2r)-3-(dimethylamino)-2-hydroxypropyl]oxy}phenyl)amino]pyrimidin-4-yl}amino)acetonitrileHuman3918
CDK2CDKCMGC1pxjAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman3927
CDK2CDKCMGC2iw9CAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4218
CDK2CDKCMGC4bcpAA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4552
CDK2CDKCMGC2b55A2-(4-(aminomethyl)piperidin-1-yl)-n-(3_cyclohexyl-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)acetamideHuman4216
CDK2CDKCMGC6q4dAA2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11184
CDK2CDKCMGC3royAA4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4131
CDK2CDKCMGC4ii5ABadenosine-5'-diphosphateHuman4456
CDK2CDKCMGC3uliAA1-(aminomethyl)-n-(3-{[6-bromo-2-(4-methoxyphenyl)-3h-imidazo[4,5-b]pyridin-7-yl]amino}propyl)cyclopropanecarboxamideHuman4115
CDK2CDKCMGC3bhtAB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4491
CDK2CDKCMGC3r8mAB1h-indazole-3-carbohydrazideHuman4451
CDK2CDKCMGC2w06A4-{[4-(1-cyclopropyl-2-methyl-1h-imidazol-5-yl)pyrimidin-2-yl]amino}-n-methylbenzenesulfonamideHuman3982
CDK2CDKCMGC2uzdA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3877
CDK2CDKCMGC5angA7-hydroxy-4-(morpholinomethyl)chromen-2-oneHuman6540
CDK2CDKCMGC5k4jAA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6751
CDK2CDKCMGC2c5oCB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4050
CDK2CDKCMGC4fksACn-[(4-{[(z)-(7-oxo-6,7-dihydro-8h-[1,3]thiazolo[5,4-e]indol-8-ylidene)methyl]amino}phenyl)sulfonyl]acetamideHuman4315
CDK2CDKCMGC2iw9AAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4174
CDK2CDKCMGC3r71AB4-[(3-methoxypropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4345
CDK2CDKCMGC2btrAn-(5-isopropyl-thiazol-2-yl)-2-pyridin-3-yl-acetamideHuman3998
CDK2CDKCMGC9d0wC-Human15925
CDK2CDKCMGC2r3fAB5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4291
CDK2CDKCMGC1p2aA5-[(2-aminoethyl)amino]-6-fluoro-3-(1h-pyrrol-2-yl)benzo[cd]indol-2(1h)-oneHuman4422
CDK2CDKCMGC3rpoAA4-({4-carbamoyl-2-nitro-5-[(pyridin-3-ylmethyl)amino]phenyl}amino)butanoic acidHuman3966
CDK2CDKCMGC1urcCB-Human3937
CDK2CDKCMGC4cfwCC3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4102
CDK2CDKCMGC2r3pAA5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)-3-thiocyanatopyrazolo[1,5-a]pyrimidin-7-amineHuman4176
CDK2CDKCMGC5oo0AC-Human9745
CDK2CDKCMGC1v1kAB(2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-olHuman3928
CDK2CDKCMGC1jsuA-Human4146
CDK1 (CDC2)CDKCMGC6gu7E-Human10782
CDK1 (CDC2)CDKCMGC6gu2AA2-(2-chlorophenyl)-8-[(3~{r},4~{r})-1-methyl-3-oxidanyl-piperidin-4-yl]-5,7-bis(oxidanyl)chromen-4-oneHuman10780
CDK1 (CDC2)CDKCMGC6gu3A4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10778
MAPK10 (JNK3)MAPKCMGC1pmnAcyclopropyl-{4-[5-(3,4-dichlorophenyl)-2-[(1-methyl)-piperidin]-4-yl-3-propyl-3h-imidazol-4-yl]-pyrimidin-2-yl}amineHuman3439
MAPK10 (JNK3)MAPKCMGC2ok1AAn-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamideHuman3444
CDK2CDKCMGC6oqiA5-fluoro-n-[5-(4-methylpiperazin-1-yl)pyridin-2-yl]-4-[(4s)-4-methyl-5,6,7,8-tetrahydro-4h-pyrazolo[1,5-a]azepin-3-yl]pyrimidin-2-amineHuman12648
CDK12 (CRK7)CDKCMGC6ckxAn-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamideHuman10578
CDK6CDKCMGC5l2sAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman6990
CDK2CDKCMGC2wpaCn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHuman4162
CDK2CDKCMGC9et7AB4-bromanyl-1~{h}-pyridin-2-oneHuman15907
CDK2CDKCMGC2exmAn-(3-methylbut-2-en-1-yl)-9h-purin-6-amineHuman4055
CDK2CDKCMGC1h1rCB6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman4081
CDK2CDKCMGC1pxoAD[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4167
CDK2CDKCMGC3bhvAB9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4001
CDK2CDKCMGC4fkuAA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman3863
CDK2CDKCMGC6q4aAA5-iodanylpyrimidineHuman11195
CDK2CDKCMGC4ek8AB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-(3-nitrophenyl)pyrimidin-2-amineHuman3871
CDK2CDKCMGC9d0xB-Human15910
CDK2CDKCMGC4bcoAA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman3988
CDK2CDKCMGC5iexAA(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHuman6565
CDK2CDKCMGC8b54AB~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman14680
CDK2CDKCMGC1urcAB-Human4010
CDK2CDKCMGC3r28AA4-chloro-5-nitro-2-[(3,4,5-trifluorobenzyl)amino]benzamideHuman4052
CDK2CDKCMGC4bcpCB2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4501
CDK2CDKCMGC9hiuB-Human15912
CDK2CDKCMGC2b52A1-(3-(2,4-dimethylthiazol-5-yl)-4-oxo-2,4-dihydroindeno[1,2-c]pyrazol-5-yl)-3-(4-methylpiperazin-1-yl)ureaHuman3997
CDK2CDKCMGC6gvaAA5-(2-azanylethylsulfanyl)-3-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman11206
CDK2CDKCMGC3r1yAA2-[(pyridin-3-ylmethyl)amino]benzamideHuman4319
CDK2CDKCMGC6yl1AAmethyl 4-(cyclopropylmethyl)-1-prop-2-enoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12497
CDK2CDKCMGC4cfuAA3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman3905
CDK2CDKCMGC2c4gA(3z)-5-acetyl-3-(benzoylimino)-3,6-dihydropyrrolo[3,4-c]pyrazol-5-iumHuman4088
CDK2CDKCMGC4rj3AA1-cyclopentyl-n-[2-(4-methoxypiperidin-1-yl)pyrimidin-4-yl]-1h-pyrrolo[3,2-c]pyridin-6-amineHuman4244
CDK2CDKCMGC1h26C-Human4179
CDK2CDKCMGC6q4bAC5-bromanylpyrimidineHuman11180
CDK2CDKCMGC9eslAB4-bromanyl-1-(2-methoxyethyl)pyridin-2-oneHuman15931
CDK2CDKCMGC3r7uAA2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamideHuman4510
CDK2CDKCMGC4eomABadenosine-5'-triphosphateHuman4472
CDK2CDKCMGC3qwkAA4-chloro-2-{[(2-chloropyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4091
CDK2CDKCMGC1pxjAB-Human3911
CDK2CDKCMGC2whbCA-Human4132
CDK2CDKCMGC4fkpAA3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4035
CDK2CDKCMGC6inlA2,2'-{[6-{[(4-methoxyphenyl)methyl]amino}-9-(propan-2-yl)-9h-purin-2-yl]azanediyl}di(ethan-1-ol)Human11794
CDK2CDKCMGC4eolAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4270
CDK2CDKCMGC3dogCB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4121
CDK2CDKCMGC3r7iAB4-{[(2-carbamoyl-4-nitrophenyl)amino]methyl}benzoic acidHuman4070
CDK2CDKCMGC9esqAB4-bromanyl-2-oxidanyl-benzoic acidHuman15933
CDK2CDKCMGC3rpvAA4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4348
CDK2CDKCMGC3qziAB4-chloro-5-nitro-2-[(pyrimidin-5-ylmethyl)amino]benzamideHuman4500
CDK2CDKCMGC4fkqAB4-[(2z)-2-(7-oxidanylidene-3,6-dihydropyrrolo[3,2-e]benzotriazol-8-ylidene)hydrazinyl]benzenesulfonamideHuman4026
CDK2CDKCMGC4eopCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4463
CDK2CDKCMGC2btsA4-[(5-isopropyl-1,3-thiazol-2-yl)amino]benzenesulfonamideHuman4443
CDK2CDKCMGC3tnwAA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman4254
CDK2CDKCMGC1h08AB(2s)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHuman4411
CDK2CDKCMGC3r1qAA4-chloro-2-{[(6-chloropyridin-3-yl)methyl]amino}-5-nitrobenzamideHuman4224
CDK2CDKCMGC3pxzA8-anilino-1-naphthalene sulfonateHuman4251
CDK2CDKCMGC1qmzCadenosine-5'-triphosphateHuman4527
CDK2CDKCMGC1pxkAAn-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n'-hydroxyimidoformamideHuman3915
CDK2CDKCMGC4cfxCA3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4166
CDK2CDKCMGC3my5CA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4473
CDK2CDKCMGC3sw4ABn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHuman4439
CDK2CDKCMGC2r3gAA6-(2-fluorophenyl)-n-(pyridin-3-ylmethyl)imidazo[1,2-a]pyrazin-8-amineHuman4276
CDK2CDKCMGC9esuAD-Human15934
CDK2CDKCMGC4eosAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4028
CDK2CDKCMGC2c5yAAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman6785
CDK2CDKCMGC4eolCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4235
CDK2CDKCMGC9esnAB4-bromo-1-(2-hydroxyethyl)pyridin-2(1h)-oneHuman15923
CDK2CDKCMGC3bhvAA9-amino-5-(2-aminopyrimidin-4-yl)pyrido[3',2':4,5]pyrrolo[1,2-c]pyrimidin-4-olHuman4531
CDK2CDKCMGC3my5AB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3887
CDK2CDKCMGC6q4fAApyridine-2,6-diamineHuman11202
CDK2CDKCMGC5if1CB-Human6571
CDK2CDKCMGC6sg4AA-Human13246
CDK2CDKCMGC4eoqAAadenosine-5'-triphosphateHuman4402
CDK2CDKCMGC5a14AB1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHuman3901
CDK2CDKCMGC5cyiCA6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6055
CDK2CDKCMGC3sw4AAn'-[4-(2-amino-4-methyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n,n-dimethylbenzene-1,4-diamineHuman4076
CDK2CDKCMGC4bckCB3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4506
CDK2CDKCMGC2vtsA5-[(4-aminocyclohexyl)amino]-7-(propan-2-ylamino)pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4300
CDK2CDKCMGC9et2AA~{n}-(4-bromophenyl)ethanamideHuman15924
DYRK1ADYRKCMGC2wo6ABn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3764
CDK2CDKCMGC1f5qCB-Human3952
CDK2CDKCMGC3r1yAB2-[(pyridin-3-ylmethyl)amino]benzamideHuman4405
CDK2CDKCMGC1ckpABpurvalanol bHuman4214
CDK2CDKCMGC4kd1AB3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman4525
CDK2CDKCMGC3iggAn-[1-(cis-3-hydroxycyclobutyl)-1h-imidazol-4-yl]-2-(4-methoxyphenyl)acetamideHuman4360
CDK2CDKCMGC3qxpAA4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4343
CDK2CDKCMGC3r9dAB4-amino-n-(3-fluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4565
CDK2CDKCMGC2r3iAB5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4059
CDK2CDKCMGC1h28C-Human4351
CDK2CDKCMGC2whbAB-Human4457
CDK2CDKCMGC1v1kAA(2r)-1-(dimethylamino)-3-{4-[(6-{[2-fluoro-5-(trifluoromethyl)phenyl]amino}pyrimidin-4-yl)amino]phenoxy}propan-2-olHuman4189
CDK2CDKCMGC11gvAA(1r,3s)-3-{3-[(1-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl bicyclo[1.1.1]pentan-1-ylcarbamateHuman15932
CDK2CDKCMGC6q4fACpyridine-2,6-diamineHuman11212
CDK2CDKCMGC3r8zAB[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-4-yl)methanoneHuman4140
CDK2CDKCMGC5lmkAA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7399
CDK2CDKCMGC3bhuCB4-(4-propoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman4464
CDK2CDKCMGC2uzbCD4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4502
CDK2CDKCMGC6q4dAC2-(4-bromanyl-2-methoxy-phenyl)ethanoic acidHuman11188
CDK2CDKCMGC2w17ABn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman4165
CDK2CDKCMGC3qhwAAadenosine-5'-diphosphateHuman4346
CDK2CDKCMGC2uzeC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHuman4071
CDK2CDKCMGC1oi9CA6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4571
CDK2CDKCMGC3rk7A4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzamideHuman4236
CDK2CDKCMGC1f5qAB-Human4517
CDK2CDKCMGC3r8pAB(5r)-5-propyl-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4538
CDK2CDKCMGC3rk9AA[4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4158
CDK2CDKCMGC3tnwAB4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman3948
CDK2CDKCMGC9nyrAA-Human15939
CDK2CDKCMGC3s2pA(3s,4s)-1-{3-[2-amino-6-(propan-2-yl)pyrimidin-4-yl]-4-hydroxyphenyl}pyrrolidine-3,4-diolHuman4404
CDK2CDKCMGC5jq5A(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman7416
CDK2CDKCMGC4eopAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4044
CDK2CDKCMGC2vtpAA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4511
CDK2CDKCMGC2cjmCadenosine-5'-triphosphateHuman4126
CDK2CDKCMGC9et7AA4-bromanyl-1~{h}-pyridin-2-oneHuman15940
CSNK2A1 (CK2a1)CK2CMGC3u9cB7-hydroxy-3h-phenoxazin-3-oneHuman5523
CSNK2A1 (CK2a1)CK2CMGC5cu6ABadenosine-5'-triphosphateHuman6906
DYRK2DYRKCMGC5lxcBBmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7126
CDK2CDKCMGC2c5nCAn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4161
CDK2CDKCMGC3my5AA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4554
CDK2CDKCMGC4cfuCB3-[2-azanyl-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methyl-benzoic acidHuman4539
CDK2CDKCMGC9eskAA(4-bromo-2-oxopyridin-1(2h)-yl)acetic acidHuman15945
CDK2CDKCMGC2duvA2-(3,4-dihydroxyphenyl)-8-(1,1-dioxidoisothiazolidin-2-yl)-3-hydroxy-6-methyl-4h-chromen-4-oneHuman4193
CDK2CDKCMGC3qqlAA(5r)-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-1h-indazole-3-carbohydrazideHuman4341
CDK2CDKCMGC1pkdC7-hydroxystaurosporineHuman3973
CDK2CDKCMGC3r9hAA4-amino-n-(2,6-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman3958
CDK2CDKCMGC4fx3CB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4495
CDK2CDKCMGC7ra5AA4-[7-(methanesulfonyl)-1h-indol-3-yl]-n-[(3s)-piperidin-3-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman13960
CDK2CDKCMGC9etpAB4-bromo-1h-pyrazoleHuman15949
CDK2CDKCMGC6q3fAB-Human11187
CDK2CDKCMGC2c5nABn-[4-(2,4-dimethyl-thiazol-5-yl)-pyrimidin-2-yl]-n',n'-dimethyl-benzene-1,4-diamineHuman4223
CDK2CDKCMGC4fkwAA2-methylpropyl (3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylateHuman4252
CDK2CDKCMGC5if1CA-Human6564
CLK3CLKCMGC6fyrAB6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHuman11406
CDK2CDKCMGC4acmAB3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman3983
MAPK1 (Erk2)MAPKCMGC4qteAB4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamideHuman2564
CDK2CDKCMGC2whbAA-Human4471
CDK2CDKCMGC1okvC-Human4093
CDK2CDKCMGC4bcoCA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4333
CDK2CDKCMGC2c68A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydropyrazolo[1,5-a]pyrimidin-7-amineHuman6776
CDK2CDKCMGC2vtmApyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman4283
CDK2CDKCMGC1oitA4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]benzenesulfonamideHuman4025
CDK2CDKCMGC4gcjAB4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4362
CDK2CDKCMGC3qtsAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanoneHuman4275
CDK2CDKCMGC3fz1A(3r)-3-(aminomethyl)-9-methoxy-1,2,3,4-tetrahydro-5h-[1]benzothieno[3,2-e][1,4]diazepin-5-oneHuman4335
CDK2CDKCMGC4fkuAB(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4573
CDK2CDKCMGC2uzeA4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzoic acidHuman3949
CDK2CDKCMGC2vtpAB{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman4401
CDK2CDKCMGC6q4cAA4-bromanyl-1,8-naphthyridineHuman11182
MAPK8 (JNK1)MAPKCMGC5lw1BadenosineHuman9081
MAPK8 (JNK1)MAPKCMGC4yr8AA-Human6452
CDK8CDKCMGC4f6wAn-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-4-[2-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)ethyl]piperazine-1-carboxamideHuman3845
CDK8CDKCMGC4f7lAtert-butyl [3-({[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]carbamoyl}amino)propyl]carbamateHuman3840
CDK8CDKCMGC4f6uAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-[3-(morpholin-4-yl)propyl]ureaHuman3844
CDK2CDKCMGC2wipA1-methyl-8-(phenylamino)-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxylic acidHuman4520
CDK2CDKCMGC2i40CA5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4222
CDK2CDKCMGC4cfmCB6-(cyclohexylmethoxy)-8-(2-methylphenyl)-9h-purin-2-amineHuman4005
CDK2CDKCMGC6q4jAB2-[3-(pyrimidin-4-ylamino)phenyl]ethanoic acidHuman11213
CDK2CDKCMGC4bcqAB4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4415
CDK2CDKCMGC2j9mAB6-bromo-13-thia-2,4,8,12,19-pentaazatricyclo[12.3.1.1~3,7~]nonadeca-1(18),3(19),4,6,14,16-hexaene 13,13-dioxideHuman4246
CDK2CDKCMGC1p5eC4,5,6,7-tetrabromobenzotriazoleHuman4434
CDK2CDKCMGC2iw8AAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4142
CDK2CDKCMGC3ddqABr-roscovitineHuman4269
CDK2CDKCMGC1w8cAB6-(cyclohexylmethoxy)-8-isopropyl-9h-purin-2-amineHuman4197
CDK2CDKCMGC3rk5A4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzoic acidHuman4160
CDK2CDKCMGC9eswAA(4-bromanylpyridin-2-yl)methanolHuman15935
CLK1CLKCMGC6z4zBA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12310
CDK2CDKCMGC1h1pC6-o-cyclohexylmethyl guanineHuman4581
CDK2CDKCMGC3rk9AB[4-amino-2-(propan-2-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4259
CDK2CDKCMGC9eswAC-Human15936
CDK2CDKCMGC1buhA-Human4178
CDK2CDKCMGC3sqqAA4-{[4-amino-5-(2-methylbenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4231
CDK2CDKCMGC2wxvAn,1-dimethyl-8-{[1-(methylsulfonyl)piperidin-4-yl]amino}-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4318
CDK2CDKCMGC4fkvAA(3z)-n-[2-(1h-imidazol-4-yl)ethyl]-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxamideHuman4299
CDK2CDKCMGC9hj1B-Human15937
CDK2CDKCMGC3bhtCB4-(4-methoxy-1h-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman3889
CDK2CDKCMGC9esuAA4-bromanyl-2-(methoxymethyl)pyridineHuman15938
CDK2CDKCMGC4bcnCB2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman4150
CDK2CDKCMGC4eooCAadenosine-5'-triphosphateHuman4188
CDK2CDKCMGC3r7eAB5-nitro-2-[(pyrazin-2-ylmethyl)amino]benzamideHuman4447
CDK2CDKCMGC9ob3A(1r,3r)-3-{3-[(pyrazine-2-carbonyl)amino]-1h-pyrazol-5-yl}cyclopentyl [(1s)-1-cyclopropylethyl]carbamateHuman15941
CDK2CDKCMGC5osmAAmethyl 1-propanoyl-3,4-dihydro-2~{h}-quinoline-6-carboxylateHuman9741
CDK2CDKCMGC2r3mABn-((2-aminopyrimidin-5-yl)methyl)-5-(2,6-difluorophenyl)-3-ethylpyrazolo[1,5-a]pyrimidin-7-amineHuman4576
CDK2CDKCMGC2c5xCAhydroxy(oxo)(3-{[(2z)-4-[3-(1h-1,2,4-triazol-1-ylmethyl)phenyl]pyrimidin-2(5h)-ylidene]amino}phenyl)ammoniumHuman4466
CDK2CDKCMGC4bcqAA4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]-2-{[3-(morpholin-4-ylcarbonyl)phenyl]amino}pyrimidine-5-carbonitrileHuman4396
CDK2CDKCMGC3r73AB4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman3899
CDK2CDKCMGC5fp6AB3-(4,7-dichloro-1h-indol-3-yl)prop-2-yn-1-olHuman6301
CDK2CDKCMGC2wmaC-Human4410
CDK2CDKCMGC9jj5A~{n}-(4-azanylcyclohexyl)-4-[[2,6-bis(fluoranyl)-3-[4-(methylcarbamoyl)phenyl]phenyl]carbonylamino]-1~{h}-pyrazole-3-carboxamideHuman15942
CDK2CDKCMGC3ql8AA3-(4-amino-1,3,5-triazin-2-yl)-4-hydroxybenzonitrileHuman3916
CDK2CDKCMGC2c5oAA4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4388
CDK2CDKCMGC5iexAB(2r,3r)-3-[(5-bromo-2-{[4-(s-cyclopropylsulfonimidoyl)phenyl]amino}pyrimidin-4-yl)oxy]butan-2-olHuman6572
CDK2CDKCMGC3qzfA2-(4,6-diamino-1,3,5-triazin-2-yl)benzene-1,4-diolHuman4569
CDK2CDKCMGC2a0cXA2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHuman4157
CDK2CDKCMGC5a14AA1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]ureaHuman3977
CDK2CDKCMGC4gcjAA4-{[4-amino-5-(2-nitrobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4138
CDK2CDKCMGC1urwAB2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]-Human4196
CDK2CDKCMGC8b54AA~{n}-[(2-phenylphenyl)methyl]-5-piperidin-4-ylsulfanyl-3-propan-2-yl-2~{h}-pyrazolo[4,3-d]pyrimidin-7-amineHuman14681
MAPK9 (JNK2)MAPKCMGC7cmlBA-Human12706
CDK2CDKCMGC9hiwB-Human15943
CDK2CDKCMGC4bckAD3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4563
CDK2CDKCMGC5aniA6-chloro-9h-purineHuman6539
CDK9CDKCMGC4ec8A-Human2244
MAPK6 (Erk3)MAPKCMGC6ylcA5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12791
MAPK6 (Erk3)MAPKCMGC6ykyBA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12792
MAPK6 (Erk3)MAPKCMGC6yllA~{n}4-[3-(4-methoxyphenyl)-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]cyclohexane-1,4-diamineHuman12793
MAPK6 (Erk3)MAPKCMGC7aqbAA-Human12982
MAPK6 (Erk3)MAPKCMGC6ylcD5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12795
MAPK6 (Erk3)MAPKCMGC7aqbBB-Human12983
MAPK6 (Erk3)MAPKCMGC6ykyDA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12796
MAPK6 (Erk3)MAPKCMGC6ylcB5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12797
DYRK1ADYRKCMGC6yf8C~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13463
CSNK2A1 (CK2a1)CK2CMGC8c6lAA5-azanyl-3-[(~{z})-1-cyano-2-(3-methoxy-4-oxidanyl-phenyl)ethenyl]-3~{h}-pyrazole-4-carbonitrileHuman15275
CSNK2A1 (CK2a1)CK2CMGC8c6nAA(2~{z},5~{z})-5-[(4-methoxy-3-oxidanyl-phenyl)methylidene]-2-phenylimino-1,3-thiazolidin-4-oneHuman15276
CSNK2A1 (CK2a1)CK2CMGC6q4qAAbenzoic acidHuman11281
CSNK2A1 (CK2a1)CK2CMGC5moeAAadenosine-5'-diphosphateHuman7650
CSNK2A1 (CK2a1)CK2CMGC5mmrBB-Human7680
CSNK2A1 (CK2a1)CK2CMGC3wikAn-[5-(4-nitrophenyl)-1,3,4-thiadiazol-2-yl]acetamideHuman5459
MAPK10 (JNK3)MAPKCMGC4w4xA3-(4-{[(4-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamideHuman3440
CSNK2A1 (CK2a1)CK2CMGC5otsAB2-(1~{h}-benzimidazol-2-yl)ethyl-[[3,5-bis(chloranyl)-4-phenyl-phenyl]methyl]azaniumHuman10599
CSNK2A1 (CK2a1)CK2CMGC5ot6AA(3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-pyrrol-2-yl)ethyl]azaniumHuman9619
CSNK2A1 (CK2a1)CK2CMGC9gcwAB-Human16073
CSNK2A1 (CK2a1)CK2CMGC5oniBB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9454
CSNK2A1 (CK2a1)CK2CMGC5cvgAB-Human6908
CSNK2A1 (CK2a1)CK2CMGC6hopAC(~{e})-4-(3-methoxy-4-oxidanyl-phenyl)but-3-en-2-oneHuman11662
CSNK2A1 (CK2a1)CK2CMGC6yzhAAadenosine-5'-diphosphateHuman13559
CSNK2A1 (CK2a1)CK2CMGC6tlwAB7-bromanyl-1~{h}-benzotriazoleHuman13085
CSNK2A1 (CK2a1)CK2CMGC3owkAB7-chloro-10-methyl-11h-benzo[g]pyrido[4,3-b]indol-3-olHuman5433
CSNK2A1 (CK2a1)CK2CMGC4md9F-Human5473
CSNK2A1 (CK2a1)CK2CMGC7a4cAA5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13170
CSNK2A1 (CK2a1)CK2CMGC6rfeAA(~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12148
CSNK2A1 (CK2a1)CK2CMGC6tluAB6,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13090
CSNK2A1 (CK2a1)CK2CMGC5mo5BB-Human7656
CSNK2A1 (CK2a1)CK2CMGC5otlBB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9616
CSNK2A1 (CK2a1)CK2CMGC5cspAA2-hydroxy-5-methylbenzoic acidHuman6904
CSNK2A1 (CK2a1)CK2CMGC9s9yABphosphoaminophosphonic acid-adenylate esterHuman16087
CSNK2A1 (CK2a1)CK2CMGC5cu6AAadenosine-5'-triphosphateHuman6899
CSNK2A1 (CK2a1)CK2CMGC3pe2AB5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acidHuman5519
CSNK2A1 (CK2a1)CK2CMGC5cspAB2-hydroxy-5-methylbenzoic acidHuman6905
CSNK2A1 (CK2a1)CK2CMGC9s7aAAphosphoaminophosphonic acid-adenylate esterHuman16088
CSNK2A1 (CK2a1)CK2CMGC6tluAA6,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13091
CSNK2A1 (CK2a1)CK2CMGC5ot5BB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9605
CSNK2A1 (CK2a1)CK2CMGC5mowAB5-bromopyridine-2,3-diamineHuman7684
CSNK2A1 (CK2a1)CK2CMGC7a4cBB5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13171
CSNK2A1 (CK2a1)CK2CMGC9s7aABphosphoaminophosphonic acid-adenylate esterHuman16089
CSNK2A1 (CK2a1)CK2CMGC9h97A1,2,3,4-tetrakis(bromanyl)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman16090
CDK2CDKCMGC2c69A(5z)-5-(3-bromocyclohexa-2,5-dien-1-ylidene)-n-(pyridin-4-ylmethyl)-1,5-dihydro[1,2,4]triazolo[1,5-a]pyrimidin-7-amineHuman6775
CDK2CDKCMGC1pw2A-Human4432
CSNK2A1 (CK2a1)CK2CMGC3warABnicotinic acidHuman5464
CSNK2A1 (CK2a1)CK2CMGC9s7hABphosphoaminophosphonic acid-adenylate esterHuman16097
CSNK2A1 (CK2a1)CK2CMGC7a4cBA5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13173
CSNK2A1 (CK2a1)CK2CMGC3pe2AA5-[(3-ethynylphenyl)amino]pyrimido[4,5-c]quinoline-8-carboxylic acidHuman5508
CSNK2A1 (CK2a1)CK2CMGC5mmfAA(3-chloranyl-4-phenyl-phenyl)methyl-propyl-azaniumHuman7682
CSNK2A1 (CK2a1)CK2CMGC7a4cAB5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13174
CSNK2A1 (CK2a1)CK2CMGC9qstA5-[4-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanoylamino]butylamino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman16101
CSNK2A1 (CK2a1)CK2CMGC5owlAA3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10593
CSNK2A1 (CK2a1)CK2CMGC6hbnAB5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11284
CSNK2A1 (CK2a1)CK2CMGC5otzAAtrifluoroacetic acidHuman9650
CSNK2A1 (CK2a1)CK2CMGC5mp8BBadenosine-5'-diphosphateHuman7692
CSNK2A1 (CK2a1)CK2CMGC5cquAA4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6035
CSNK2A1 (CK2a1)CK2CMGC8p05A(4~{z})-2-(1-adamantylamino)-4-(1,3-benzothiazol-6-ylmethylidene)-1~{h}-imidazol-5-oneHuman14744
CSNK2A1 (CK2a1)CK2CMGC5otdBA[2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azaniumHuman9690
CSNK2A1 (CK2a1)CK2CMGC5cu0BBn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7301
CDK2CDKCMGC1wccAB2-amino-6-chloropyrazineHuman3897
CDK2CDKCMGC3lfqAn-(6,7-difluoro-5-phenyl-1h-indazol-3-yl)butanamideHuman4320
CDK2CDKCMGC4ek4AB4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman3957
CDK2CDKCMGC4cfnCB6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4567
CDK2CDKCMGC4eoiAB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4342
CDK2CDKCMGC6ylkAAmethyl 4-ethyl-1-propanoyl-2,3-dihydroquinoxaline-6-carboxylateHuman12499
CDK2CDKCMGC2x1nCA2-methyl-n-[(1z)-3-nitrocyclohexa-2,4-dien-1-ylidene]-4,5-dihydro[1,3]thiazolo[4,5-h]quinazolin-8-amineHuman3991
CDK2CDKCMGC2c5oAB4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-amineHuman4440
CDK2CDKCMGC3pxfAB8-anilino-1-naphthalene sulfonateHuman4301
CDK8CDKCMGC6t41A~{n}-[(4-chlorophenyl)methyl]quinazolin-4-amineHuman11908
CDK2CDKCMGC3r7yAB2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-(morpholin-4-yl)-5-nitrobenzamideHuman3975
CDK2CDKCMGC1pxnAB-Human4172
CDK2CDKCMGC3tiyAA2,3,4,6-tetrahydroxy-5h-benzo[7]annulen-5-oneHuman4413
CDK2CDKCMGC6q3bAB4-iodopyrazoleHuman11208
CDK2CDKCMGC1hckABadenosine-5'-triphosphateHuman4416
CDK2CDKCMGC1h01AB(2s)-1-[4-({4-[(2,5-dichlorophenyl)amino]pyrimidin-2-yl}amino)phenoxy]-3-(dimethylamino)propan-2-olHuman4561
CDK2CDKCMGC5lmkCA4-[4-[3-bromanyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]phenyl]benzamideHuman7396
CDK2CDKCMGC1qmzAadenosine-5'-triphosphateHuman4242
CDK8CDKCMGC5idpAB(3-amino-1h-indazol-5-yl)[(2s)-2-(4-fluorophenyl)piperidin-1-yl]methanoneHuman7320
CDK8CDKCMGC5icpAA[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](5-methylimidazo[5,1-b][1,3,4]thiadiazol-2-yl)methanoneHuman7318
CDK8CDKCMGC8tqcCB-Human15963
CDK8CDKCMGC5xs2AA3-chloranyl-4-pyridin-4-yl-1h-pyrrole-2-carboxamideHuman8315
MAPK14 (p38a)MAPKCMGC5n67AA-Human8523
MAPK14 (p38a)MAPKCMGC1r3cAA-Human5170
DYRK2DYRKCMGC7dl6A[2,7-dimethoxy-9-[[(3r)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanolHuman14013
DYRK2DYRKCMGC5lxdBBmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7127
DYRK2DYRKCMGC7dhcA4-[bis(fluoranyl)methyl]-2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridineHuman13973
DYRK2DYRKCMGC7djoA[2,7-dimethoxy-9-[[(3s)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanolHuman13994
DYRK2DYRKCMGC6hdpAAscorzodihydrostilbene aHuman11572
DYRK2DYRKCMGC3kvwAA(2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acidHuman3148
CDK8CDKCMGC8tq2CB-Human15964
CDK8CDKCMGC5idnAB[(2s)-2-(4-chlorophenyl)pyrrolidin-1-yl](3-methyl-1h-pyrazolo[3,4-b]pyridin-5-yl)methanoneHuman7319
CDK8CDKCMGC5hbjAB8-[2-azanyl-3-chloranyl-5-(1-methylindazol-5-yl)pyridin-4-yl]-2,8-diazaspiro[4.5]decan-1-oneHuman6385
CDK8CDKCMGC6y0aAB6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman13305
CDK8CDKCMGC8tq2CA-Human15965
CDK8CDKCMGC8tqcCA-Human15966
CDK8CDKCMGC6r3sAA6-[5-chloranyl-4-[(1~{s})-1-oxidanylethyl]pyridin-3-yl]-3,4-dihydro-2~{h}-1,8-naphthyridine-1-carboxamideHuman12140
CDK8CDKCMGC5ceiAA4-(4-iodophenoxy)-n-methylthieno[2,3-c]pyridine-2-carboxamideHuman6404
CLK2CLKCMGC5unpAn~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamineHuman9887
GSK3BGSKCMGC1r0eAA3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman733
GSK3BGSKCMGC3zrlAC7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman654
GSK3BGSKCMGC1q3dBstaurosporineHuman752
MAPK13 (p38d)MAPKCMGC8x23AB-Human15128
MAPK7 (Erk5)MAPKCMGC5byzAB4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamideHuman6592
MAPK7 (Erk5)MAPKCMGC4zsgAA3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6589
MAPK7 (Erk5)MAPKCMGC5byzAA4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamideHuman6590
MAPK7 (Erk5)MAPKCMGC4zsjAA3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6588
MAPK7 (Erk5)MAPKCMGC4ic8B-Human389
MAPK7 (Erk5)MAPKCMGC4ic8A-Human390
CDKL5CDKLCMGC8cieA4-[[3,5-bis(fluoranyl)phenyl]carbonylamino]-~{n}-piperidin-4-yl-1~{h}-pyrazole-3-carboxamideHuman14778
CLK3CLKCMGC6z54AA11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12294
CLK3CLKCMGC2eu9AB-Human1830
CLK3CLKCMGC6z54AB11,15-dimethyl-6-(oxan-4-yloxy)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12295
CLK3CLKCMGC6z51AAn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide Human12296
CLK3CLKCMGC2exeAA-Human1822
CLK3CLKCMGC6fypAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10400
CLK3CLKCMGC6rctAA4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11127
CLK3CLKCMGC6z52AA11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12628
CLK3CLKCMGC3rawAA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman1820
CLK3CLKCMGC6z55BB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12299
CLK3CLKCMGC2wu6AB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman1821
CLK3CLKCMGC6fypAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10397
CLK3CLKCMGC6z55AC7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12301
CLK3CLKCMGC3rawAB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman1829
CLK3CLKCMGC6z52BA11,15-dimethyl-6-(4-methylpiperazin-1-yl)-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-oneHuman12629
CLK3CLKCMGC6yu1aB(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12408
CLK3CLKCMGC6z55BA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12303
CLK3CLKCMGC6z51ABn-cyclopentyl-2-[(11,15-dimethyl-10-oxo-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-6-yl)oxy]acetamide Human12304
CLK3CLKCMGC6ytwBB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12410
CDK16 (PCTAIRE1)CDKCMGC3mtlAA(2z,3e)-2,3'-biindole-2',3(1h,1'h)-dione 3-{o-[(3r)-3,4-dihydroxybutyl]oxime}Human1701
CDK2CDKCMGC3qxoA5-nitro-2-[(4-sulfamoylbenzyl)amino]benzamideHuman4282
CDK1 (CDC2)CDKCMGC4yc6CA-Human4608
CDK1 (CDC2)CDKCMGC4yc6GB-Human4615
CDK1 (CDC2)CDKCMGC5lqfDAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman7365
CDK1 (CDC2)CDKCMGC5hq0AA{[(2,6-difluorophenyl)carbonyl]amino}-n-(4-fluorophenyl)-1h-pyrazole-3-carboxamideHuman6422
CDK1 (CDC2)CDKCMGC7nj0B-Human13827
CLK4CLKCMGC6fyvAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10510
MAPK8 (JNK1)MAPKCMGC4ux9AAphosphoaminophosphonic acid-adenylate esterHuman4643
MAPK8 (JNK1)MAPKCMGC2gmxAn-(4-amino-5-cyano-6-ethoxypyridin-2-yl)-2-(4-bromo-2,5-dimethoxyphenyl)acetamideHuman4674
MAPK8 (JNK1)MAPKCMGC9ft9Aphosphoaminophosphonic acid-adenylate esterHuman15532
MAPK8 (JNK1)MAPKCMGC3vuhA-Human4663
MAPK8 (JNK1)MAPKCMGC2g01B6-chloro-9-hydroxy-1,3-dimethyl-1,9-dihydro-4h-pyrazolo[3,4-b]quinolin-4-oneHuman4641
MAPK8 (JNK1)MAPKCMGC12cvAA(4m)-n-[3-(dimethylcarbamoyl)-4-hydroxyphenyl]-4-(1h-pyrrolo[2,3-b]pyridin-5-yl)-3h-1lambda~4~-benzothiophene-2-carboxamideHuman15533
MAPK8 (JNK1)MAPKCMGC4qtdAB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman4673
MAPK8 (JNK1)MAPKCMGC4hyuAtrans-4-[(4-{4-[3-(methylsulfonyl)propoxy]-1h-indazol-1-yl}pyrimidin-2-yl)amino]cyclohexanolHuman4632
MAPK8 (JNK1)MAPKCMGC4l7fAAn-[1-(4-fluorophenyl)cyclopropyl]-4-[(trans-4-hydroxycyclohexyl)amino]imidazo[1,2-a]quinoxaline-8-carboxamideHuman4639
MAPK8 (JNK1)MAPKCMGC4e73AAmethyl 3-(4-{[(1r,2s,3s,5s,7s)-5-aminotricyclo[3.3.1.1~3,7~]dec-2-yl]carbamoyl}benzyl)-4-oxo-1-phenyl-1,4-dihydro-1,8-naphthyridine-2-carboxylateHuman4645
MAPK8 (JNK1)MAPKCMGC4ux9BAphosphoaminophosphonic acid-adenylate esterHuman4635
MAPK8 (JNK1)MAPKCMGC4izyAtrans-4-[(4-{4-[4-(methylsulfonyl)piperidin-1-yl]-1h-indol-1-yl}pyrimidin-2-yl)amino]cyclohexanolHuman4654
MAPK8 (JNK1)MAPKCMGC11zlAB(4m)-n-[4-hydroxy-3-(pyrrolidine-1-carbonyl)phenyl]-4-(1h-pyrrolo[2,3-b]pyridin-5-yl)-1-benzothiophene-2-carboxamideHuman15535
MAPK8 (JNK1)MAPKCMGC4yr8FA-Human6450
MAPK8 (JNK1)MAPKCMGC2xrwABphosphoaminophosphonic acid-adenylate esterHuman4650
MAPK8 (JNK1)MAPKCMGC12cvAB(4m)-n-[3-(dimethylcarbamoyl)-4-hydroxyphenyl]-4-(1h-pyrrolo[2,3-b]pyridin-5-yl)-3h-1lambda~4~-benzothiophene-2-carboxamideHuman15536
MAPK8 (JNK1)MAPKCMGC3vumA-Human4671
MAPK8 (JNK1)MAPKCMGC3eljAA2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamideHuman4658
MAPK8 (JNK1)MAPKCMGC3eljAB2-fluoro-6-{[2-({2-methoxy-4-[(methylsulfonyl)methyl]phenyl}amino)-7h-pyrrolo[2,3-d]pyrimidin-4-yl]amino}benzamideHuman4636
MAPK8 (JNK1)MAPKCMGC8x5mAA3-[4-(dimethylamino)butanoylamino]-~{n}-[3-methyl-4-[(4-pyridin-3-ylpyrimidin-2-yl)amino]phenyl]benzamideHuman15099
SRPK2SRPKCMGC5myvBA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7576
SRPK2SRPKCMGC2x7gApurvalanol bHuman1409
CLK1CLKCMGC1z57ABdebromohymenialdisineHuman105
CLK1CLKCMGC7opgAA4-[2-(propylamino)imidazo[2,1-b][1,3,4]thiadiazol-5-yl]phenolHuman13808
CLK1CLKCMGC6ytiAAmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman12413
CLK1CLKCMGC5j1wABpyrido[3,4-g]quinazolin-2-amineHuman6576
CLK1CLKCMGC6i5hAB5-(1-methylpyrazol-4-yl)-3-(3-phenoxyphenyl)furo[3,2-b]pyridineHuman10849
CLK1CLKCMGC6ytiABmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman12414
CLK1CLKCMGC6g33AC-Human9826
CLK1CLKCMGC5j1wCApyrido[3,4-g]quinazolin-2-amineHuman6578
CLK1CLKCMGC6ytgAA(4~{s})-7,8-bis(chloranyl)-9-methyl-1-oxidanylidene-spiro[2,4-dihydropyrido[3,4-b]indole-3,4'-piperidine]-4-carbonitrileHuman12416
CLK1CLKCMGC6ytaAB1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman12417
CLK1CLKCMGC5x8iA5-[1-[(1s)-1-(4-fluorophenyl)ethyl]-[1,2,3]triazolo[4,5-c]quinolin-8-yl]-1,3-benzoxazoleHuman8316
CLK1CLKCMGC6z4zCA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12309
CLK1CLKCMGC6fyoAB6-~{tert}-butyl-~{n}-[6-(1~{h}-pyrazol-4-yl)-1~{h}-imidazo[1,2-a]pyridin-2-yl]pyridine-3-carboxamideHuman10323
CLK1CLKCMGC6tw2EAethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman11962
CLK1CLKCMGC6i5lAB3-(3-cyclobutylphenyl)-5-(1-methylpyrazol-4-yl)furo[3,2-b]pyridineHuman10843
CLK1CLKCMGC6q8pC~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amineHuman10901
CLK1CLKCMGC6ytdAA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12418
CLK1CLKCMGC6yteCA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12419
CLK1CLKCMGC6g33AB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9824
CLK1CLKCMGC6ft9CB2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9900
CLK1CLKCMGC6g33CB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9823
CLK1CLKCMGC6g33AA(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman9819
CLK1CLKCMGC6z4zAB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12312
CLK1CLKCMGC2vagAAethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman104
CLK1CLKCMGC6ytdAB(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman12420
CLK1CLKCMGC6z4zCB7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12313
CLK1CLKCMGC6g33BC-Human9827
CLK1CLKCMGC2vagABethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman103
CLK1CLKCMGC6ytaAA1-(3-{6-[(cyclopropylmethyl)amino]imidazo[1,2-b]pyridazin-3-yl}phenyl)ethanoneHuman12423
CLK1CLKCMGC6q8pB~{n}-methyl-10-nitro-pyrido[3,4-g]quinazolin-2-amineHuman10900
CLK1CLKCMGC5j1wAApyrido[3,4-g]quinazolin-2-amineHuman6579
CLK1CLKCMGC6ft9AB2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9898
CLK1CLKCMGC6ft9AA2-bromanyl-3-phenyl-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9901
CLK1CLKCMGC6qtyABethyl 3-[(e)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methyl-1h-indole-2-carboxylateHuman12084
CLK1CLKCMGC5j1wBApyrido[3,4-g]quinazolin-2-amineHuman6575
CLK1CLKCMGC6ft8AB3-(3-hydroxyphenyl)-1~{h}-pyrrolo[3,4-g]indol-8-oneHuman9899
CLK1CLKCMGC7ak3AB~{n}-[3-fluoranyl-4-(4-methylpiperazin-1-yl)phenyl]-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman13143
CLK1CLKCMGC6raaAB4-[2-methyl-1-(4-methylpiperazin-1-yl)-1-oxidanylidene-propan-2-yl]-~{n}-(6-pyridin-4-ylimidazo[1,2-a]pyridin-2-yl)benzamideHuman11013
CLK1CLKCMGC6zlnAA4-(6-ethoxypyrazolo[1,5-b]pyridazin-3-yl)-~{n}-[3-methoxy-5-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman12711
CDK12 (CRK7)CDKCMGC8buqB(2~{r})-2-[[6-[[1-(3-chlorophenyl)pyrazol-3-yl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14917
CDK12 (CRK7)CDKCMGC6td3H(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12370
CDK12 (CRK7)CDKCMGC8bu2B~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-2-morpholin-4-yl-9-propan-2-yl-purin-6-amineHuman14918
CDK12 (CRK7)CDKCMGC5acbCn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman6701
CDK12 (CRK7)CDKCMGC6b3eA2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-olHuman9452
CDK12 (CRK7)CDKCMGC8bufB2-(6,7-dihydro-4~{h}-thieno[3,2-c]pyridin-5-ylmethyl)-6,7-dimethoxy-3~{h}-quinazolin-4-oneHuman14919
CDK12 (CRK7)CDKCMGC4un0C-Human4854
CDK12 (CRK7)CDKCMGC9jk1An-[5-[[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-[(phenylmethyl)carbamoyl]amino]-2-[4-(dimethylamino)piperidin-1-yl]phenyl]propanamideHuman15853
CDK12 (CRK7)CDKCMGC8burBB~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamideHuman14920
CDK12 (CRK7)CDKCMGC6td3B(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12371
CDK12 (CRK7)CDKCMGC8buhB6-[[[2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-9-propan-2-yl-purin-6-yl]amino]methyl]-3-pyridin-2-yl-1~{h}-pyridin-2-oneHuman14922
CDK12 (CRK7)CDKCMGC4cxaC-Human4853
CDK12 (CRK7)CDKCMGC8bupB(2~{r})-2-[[6-[3-(3-methylphenyl)propylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14923
CDK12 (CRK7)CDKCMGC8bumB(2r)-2-[[6-(5-naphthalen-1-ylpentylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14924
CDK12 (CRK7)CDKCMGC8buiB(2~{r})-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)amino]purin-2-yl]amino]butan-1-olHuman14925
CDK12 (CRK7)CDKCMGC8bu5B~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman14926
CDK12 (CRK7)CDKCMGC8bukB(2~{r})-2-[[6-(naphthalen-2-ylmethylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14927
CDK12 (CRK7)CDKCMGC8bubB~{n}-(5-methyl-2,3-dihydro-1,3-thiazol-2-yl)-3-(5-methylfuran-2-yl)carbonyl-1,3-thiazolidine-4-carboxamideHuman14928
CDK12 (CRK7)CDKCMGC9x26AB(2s)-n-[2-[4-(dimethylamino)piperidin-1-yl]-5-[[(1s)-1-(4-fluorophenyl)ethyl]carbamoyl-[4-(quinazolin-2-ylamino)cyclohexyl]amino]pyridin-3-yl]-2-fluoranyl-propanamideHuman15855
CDK12 (CRK7)CDKCMGC8budB~{n}-(5-bromanylpyridin-2-yl)-3-(4-oxidanylidenequinazolin-3-yl)propanamideHuman14929
CDK12 (CRK7)CDKCMGC9x26AA(2s)-n-[2-[4-(dimethylamino)piperidin-1-yl]-5-[[(1s)-1-(4-fluorophenyl)ethyl]carbamoyl-[4-(quinazolin-2-ylamino)cyclohexyl]amino]pyridin-3-yl]-2-fluoranyl-propanamideHuman15856
CDK12 (CRK7)CDKCMGC8p81AB~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman15061
CDK12 (CRK7)CDKCMGC4nstCadenosine-5'-diphosphateHuman4851
CDK12 (CRK7)CDKCMGC6ckxCn-[4-(1-methyl-1h-pyrazol-4-yl)phenyl]-n-{trans-4-[(quinazolin-2-yl)amino]cyclohexyl}acetamideHuman10579
CDK12 (CRK7)CDKCMGC8bu1B(2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-olHuman14930
CDK12 (CRK7)CDKCMGC6b3eC2-[(2s)-1-(6-{[(4,5-difluoro-1h-benzimidazol-2-yl)methyl]amino}-9-ethyl-9h-purin-2-yl)piperidin-2-yl]ethan-1-olHuman9453
CDK12 (CRK7)CDKCMGC4un0D-Human4855
CDK12 (CRK7)CDKCMGC8bu3B2-morpholin-4-yl-9-propan-2-yl-~{n}-[(4-pyridin-2-ylphenyl)methyl]purin-6-amineHuman14931
CDK12 (CRK7)CDKCMGC8buaB(2~{r})-~{n}-(1~{h}-benzimidazol-2-yl)-2-(3-oxidanylidene-1~{h}-isoindol-2-yl)propanamideHuman14932
CDK12 (CRK7)CDKCMGC8bujB(2~{r})-2-[[6-(octylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14933
CDK12 (CRK7)CDKCMGC8buoB(2~{r})-2-[[6-[(3-fluoranyl-4-pyridin-2-yl-phenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14934
CDK12 (CRK7)CDKCMGC4cxaAphosphoaminophosphonic acid-adenylate esterHuman4856
CDK12 (CRK7)CDKCMGC8bugB2-[2-[(6-methylpyridin-2-yl)amino]-1,3-thiazol-4-yl]-~{n}-(5-methyl-1,3-thiazol-2-yl)ethanamideHuman14935
CDK12 (CRK7)CDKCMGC8p81AA~{n}-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methyl]-9-(1-methylpyrazol-4-yl)-2-morpholin-4-yl-purin-6-amineHuman15062
CDK12 (CRK7)CDKCMGC8butB2-[[6-[[4-(2-hydroxyethyloxy)phenyl]methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14936
MAPK1 (Erk2)MAPKCMGC4qp4BAn-cyclohexyl-9h-purin-6-amineHuman6086
MAPK1 (Erk2)MAPKCMGC4fv0AAn-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amineHuman2562
MAPK1 (Erk2)MAPKCMGC8aohAA~{n}-(6,7-dihydro-4~{h}-pyrano[4,3-d][1,3]thiazol-2-yl)propanamideHuman14385
MAPK1 (Erk2)MAPKCMGC5nhpA5-(2-methoxyethyl)-1-methyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydropyrrolo[3,2-c]pyridin-4-oneHuman7998
MAPK1 (Erk2)MAPKCMGC4qp1Bn-benzyl-9h-purin-6-amineHuman6080
MAPK9 (JNK2)MAPKCMGC7cmlBB-Human12704
MAPK1 (Erk2)MAPKCMGC6ophA1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman11509
MAPK1 (Erk2)MAPKCMGC4h3qAphosphoaminophosphonic acid-adenylate esterHuman2611
MAPK1 (Erk2)MAPKCMGC2ojjA(s)-n-(1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl)-4-(4-(3-chlorophenyl)-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamideHuman2612
MAPK1 (Erk2)MAPKCMGC6g97AB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-(2-methoxyethyl)-3~{h}-isoindol-1-oneHuman9970
MAPK1 (Erk2)MAPKCMGC7nr5AA(2~{r})-2-[5-[5-chloranyl-2-[(2-methyl-1,2,3-triazol-4-yl)amino]pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-fluoranyl-5-methoxy-phenyl)-2-oxidanyl-ethyl]propanamideHuman13921
MAPK1 (Erk2)MAPKCMGC4iz7CA-Human2569
MAPK1 (Erk2)MAPKCMGC6q7sAA-Human11349
MAPK1 (Erk2)MAPKCMGC4iz5Aadenosine-5'-diphosphateHuman2554
MAPK1 (Erk2)MAPKCMGC4qpaA7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6077
MAPK1 (Erk2)MAPKCMGC4iz7CB-Human2597
MAPK1 (Erk2)MAPKCMGC4fuxAtrans-4-{[4-(5-methyl-3-phenyl-1,2-oxazol-4-yl)pyrimidin-2-yl]amino}cyclohexanolHuman2568
MAPK1 (Erk2)MAPKCMGC6g9mAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamideHuman9944
MAPK1 (Erk2)MAPKCMGC6qaqABthiophen-3-ylmethylazaniumHuman10989
MAPK1 (Erk2)MAPKCMGC7nr3AA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,2,4,5-tetrahydro-3-benzazepin-3-yl)ethyl]-3~{h}-isoindol-1-oneHuman13923
MAPK1 (Erk2)MAPKCMGC6g93AB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-oneHuman9959
MAPK1 (Erk2)MAPKCMGC4qp4AAn-cyclohexyl-9h-purin-6-amineHuman6088
MAPK1 (Erk2)MAPKCMGC5nguA2-[2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]pyrimidin-4-yl]-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-4-oneHuman7991
MAPK1 (Erk2)MAPKCMGC6qaqAAthiophen-3-ylmethylazaniumHuman10983
MAPK1 (Erk2)MAPKCMGC7nqwAB6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2-[2-oxidanylidene-2-(1,3,4,5-tetrahydro-2-benzazepin-2-yl)ethyl]-3~{h}-isoindol-1-oneHuman13924
MAPK1 (Erk2)MAPKCMGC6qa3ABpyrazoleHuman11345
MAPK1 (Erk2)MAPKCMGC4n0sAAcaffeic acidHuman2589
MAPK1 (Erk2)MAPKCMGC5nhhA5-(2-methoxyethyl)-2-[2-(oxan-4-ylamino)pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7996
MAPK1 (Erk2)MAPKCMGC4zznAB2-[[5-chloranyl-2-(oxan-4-ylamino)pyridin-4-yl]amino]-n-methyl-benzamideHuman2610
MAPK1 (Erk2)MAPKCMGC4o6eAAn-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamideHuman2559
MAPK1 (Erk2)MAPKCMGC4nifEAphosphoaminophosphonic acid-adenylate esterHuman2621
MAPK1 (Erk2)MAPKCMGC6g54ABn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10937
MAPK1 (Erk2)MAPKCMGC7e73A-Human14114
MAPK1 (Erk2)MAPKCMGC6gdmAA(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamideHuman9968
MAPK1 (Erk2)MAPKCMGC6g9mAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-(2-phenylpropan-2-yl)ethanamideHuman9964
MAPK1 (Erk2)MAPKCMGC4fv1AAn-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamideHuman2594
MAPK1 (Erk2)MAPKCMGC6g9dAB~{n}-~{tert}-butyl-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]ethanamideHuman9953
MAPK1 (Erk2)MAPKCMGC6qagAA1~{h}-1,2,3-triazoleHuman10988
MAPK1 (Erk2)MAPKCMGC6g9kAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamideHuman9966
MAPK1 (Erk2)MAPKCMGC4qp6A5h-pyrrolo[2,3-b]pyrazineHuman6089
MAPK1 (Erk2)MAPKCMGC4fmqAAphosphoaminophosphonic acid-adenylate esterHuman2604
MAPK1 (Erk2)MAPKCMGC2ojgAn,n-dimethyl-4-(4-phenyl-1h-pyrazol-3-yl)-1h-pyrrole-2-carboxamideHuman2603
MAPK1 (Erk2)MAPKCMGC6g8xAB4-chloranyl-1~{h}-indazol-3-amineHuman9954
MAPK1 (Erk2)MAPKCMGC6g9nAA(2~{r})-2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-1-(3-methylphenyl)-2-oxidanyl-ethyl]propanamideHuman11410
MAPK1 (Erk2)MAPKCMGC4fv3ABethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman2580
MAPK1 (Erk2)MAPKCMGC4xj0A1-[(1s)-1-(4-chloro-3-fluorophenyl)-2-hydroxyethyl]-4-[2-(tetrahydro-2h-pyran-4-ylamino)pyrimidin-4-yl]pyridin-2(1h)-oneHuman6048
MAPK1 (Erk2)MAPKCMGC1pmeA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman2583
MAPK1 (Erk2)MAPKCMGC4fv2AB4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHuman2571
MAPK1 (Erk2)MAPKCMGC4h3pAphosphoaminophosphonic acid-adenylate esterHuman2624
MAPK1 (Erk2)MAPKCMGC8aobAA~{n}-[(1-methylindazol-3-yl)methyl]propanamideHuman14402
MAPK1 (Erk2)MAPKCMGC4izaCA-Human2588
MAPK1 (Erk2)MAPKCMGC6qa4AA1~{h}-pyridin-2-oneHuman11344
MAPK1 (Erk2)MAPKCMGC8psrAAphosphoaminophosphonic acid-adenylate esterHuman15300
MAPK1 (Erk2)MAPKCMGC5bujAB4-[3-(pyridin-4-yl)-2,4,6,7-tetrahydro-5h-pyrazolo[4,3-c]pyridin-5-yl]pyridin-2(1h)-oneHuman2561
MAPK1 (Erk2)MAPKCMGC5ax3A(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman6398
MAPK1 (Erk2)MAPKCMGC6gdmAB(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]-~{n}-(3-pyridin-4-yl-1~{h}-indazol-5-yl)pyrrolidine-3-carboxamideHuman9946
MAPK1 (Erk2)MAPKCMGC6dmgABethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman10810
MAPK1 (Erk2)MAPKCMGC8aogAA~{n}-(5-methyl-1,2-oxazol-3-yl)propanamideHuman14403
MAPK1 (Erk2)MAPKCMGC4fv8AB6-({4-[(3-cyclopropyl-1h-pyrazol-5-yl)amino]-5-(phenylamino)pyrimidin-2-yl}amino)-1,2-dihydro-3h-indazol-3-oneHuman2601
MAPK1 (Erk2)MAPKCMGC3i60A4-{2-[(2-chlorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-2-hydroxy-1-phenylethyl]-1h-pyrrole-2-carboxamideHuman2584
MAPK1 (Erk2)MAPKCMGC4fv6An-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-4-(2-{[(2s)-1-hydroxybutan-2-yl]amino}-5-methylpyrimidin-4-yl)-1h-pyrrole-2-carboxamideHuman2551
MAPK1 (Erk2)MAPKCMGC5nhvA7-[2-(oxan-4-ylamino)pyrimidin-4-yl]-3,4-dihydro-2~{h}-pyrrolo[1,2-a]pyrazin-1-oneHuman7995
MAPK1 (Erk2)MAPKCMGC6qalAA1,1-bis(oxidanylidene)thietan-3-olHuman10987
MAPK1 (Erk2)MAPKCMGC4fv9AA3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman2582
MAPK1 (Erk2)MAPKCMGC4iz5Cadenosine-5'-diphosphateHuman2595
MAPK1 (Erk2)MAPKCMGC6g92AA~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amineHuman11409
MAPK1 (Erk2)MAPKCMGC3sa0ABnorathyriolHuman2557
MAPK1 (Erk2)MAPKCMGC5lcjAB[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman6834
MAPK1 (Erk2)MAPKCMGC5v60ABphosphomethylphosphonic acid adenylate esterHuman8263
MAPK1 (Erk2)MAPKCMGC6opiA(3r)-n-[3-(2-cyclopropylpyridin-4-yl)-1h-indazol-5-yl]-3-(methoxymethyl)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]-3,6-dihydropyridin-1(2h)-yl}ethyl)pyrrolidine-3-carboxamideHuman11511
MAPK1 (Erk2)MAPKCMGC6g9kAB2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{s})-2-oxidanyl-1-phenyl-ethyl]ethanamideHuman9947
MAPK1 (Erk2)MAPKCMGC2ojiAn-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamideHuman2570
MAPK1 (Erk2)MAPKCMGC6qawAB[1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazaniumHuman10986
MAPK1 (Erk2)MAPKCMGC5bvfAB2-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-8-(2-{[(1s,3r)-3-hydroxycyclopentyl]amino}pyrimidin-4-yl)-2,3,4,5-tetrahydro-1h-pyrrolo[1,2-a][1,4]diazepin-1-oneHuman6027
MAPK1 (Erk2)MAPKCMGC4qp4ABn-cyclohexyl-9h-purin-6-amineHuman6075
MAPK1 (Erk2)MAPKCMGC4qp8B2-(1h-pyrazol-4-yl)-7-(pyridin-3-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6076
MAPK1 (Erk2)MAPKCMGC4fv2AA4-[4-(3-chlorophenyl)-1h-pyrazol-5-yl]-n-(2,3-dihydro-1-benzofuran-5-ylmethyl)-1h-pyrrole-2-carboxamideHuman2592
MAPK1 (Erk2)MAPKCMGC8pt0ABphosphoaminophosphonic acid-adenylate esterHuman15307
MAPK1 (Erk2)MAPKCMGC8aofAB~{n}-(2-methylpyrimidin-5-yl)propanamideHuman14408
MAPK1 (Erk2)MAPKCMGC6g9jAA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-phenylethyl]ethanamideHuman9952
MAPK1 (Erk2)MAPKCMGC4qp3B(2s)-3-phenyl-2-(9h-purin-6-ylamino)propan-1-olHuman6079
MAPK1 (Erk2)MAPKCMGC4fv7AA4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrileHuman2572
MAPK1 (Erk2)MAPKCMGC4nifBBphosphoaminophosphonic acid-adenylate esterHuman2566
MAPK1 (Erk2)MAPKCMGC4fuyAB{4-[4-(3,5-dichlorophenyl)-1h-pyrazol-5-yl]-1h-pyrrol-2-yl}(morpholin-4-yl)methanoneHuman2587
MAPK1 (Erk2)MAPKCMGC4izaAA-Human2586
MAPK1 (Erk2)MAPKCMGC4qp9A7-(1-propyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6085
MAPK1 (Erk2)MAPKCMGC4qpaB7-(1-benzyl-1h-pyrazol-4-yl)-2-(pyridin-4-yl)-5h-pyrrolo[2,3-b]pyrazineHuman6090
MAPK1 (Erk2)MAPKCMGC4qteAA4-{2-[(2-chloro-4-fluorophenyl)amino]-5-methylpyrimidin-4-yl}-n-[(1s)-1-(3-chlorophenyl)-2-hydroxyethyl]-1h-pyrrole-2-carboxamideHuman2590
MAPK1 (Erk2)MAPKCMGC8pt1ABphosphoaminophosphonic acid-adenylate esterHuman15309
MAPK1 (Erk2)MAPKCMGC8pswAAamp phosphoramidateHuman15310
MAPK1 (Erk2)MAPKCMGC6dmgACethyl n-{2-chloro-4-[5-(5-{[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]carbamoyl}-1h-pyrrol-3-yl)-1h-pyrazol-4-yl]benzyl}glycinateHuman10809
MAPK1 (Erk2)MAPKCMGC6qa1ABpyridin-2-amineHuman11346
MAPK1 (Erk2)MAPKCMGC4fv9AB3-[4-(2,3-difluorophenyl)-1,2-oxazol-5-yl]-5-(pyridin-4-yl)-1h-pyrrolo[2,3-b]pyridineHuman2552
MAPK1 (Erk2)MAPKCMGC4qp4BBn-cyclohexyl-9h-purin-6-amineHuman6083
MAPK1 (Erk2)MAPKCMGC8ao4AA~{n}-(1~{h}-indazol-5-yl)ethanesulfonamideHuman14416
MAPK1 (Erk2)MAPKCMGC6g93AA6-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-2,3-dihydroisoindol-1-oneHuman9955
MAPK1 (Erk2)MAPKCMGC4qp6B5h-pyrrolo[2,3-b]pyrazineHuman6091
MAPK1 (Erk2)MAPKCMGC5nhlA(6~{r})-5-(2-methoxyethyl)-6-methyl-2-[5-methyl-2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7992
MAPK1 (Erk2)MAPKCMGC6d5yA-Human10939
MAPK1 (Erk2)MAPKCMGC4fv4AB9-(dimethylamino)-2-[(3-hydroxyphenyl)amino]-5,6-dihydrothieno[3,4-h]quinazoline-7-carbonitrileHuman2558
MAPK1 (Erk2)MAPKCMGC6q7sAB-Human11343
MAPK1 (Erk2)MAPKCMGC6g92AB~{n}-(1,5-dimethylpyrazol-4-yl)-5-methyl-pyrimidin-2-amineHuman11411
MAPK1 (Erk2)MAPKCMGC4qp1An-benzyl-9h-purin-6-amineHuman6092
MAPK1 (Erk2)MAPKCMGC6ge0AA2-[5-[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]-3-oxidanylidene-1~{h}-isoindol-2-yl]-~{n}-[(1~{r})-1-(3-methoxyphenyl)ethyl]ethanamideHuman9950
MAPK1 (Erk2)MAPKCMGC6rq4AB6,6-dimethyl-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-5-(2-morpholin-4-ylethyl)thieno[2,3-c]pyrrol-4-oneHuman11855
MAPK1 (Erk2)MAPKCMGC4fv7AB4-(3-chlorophenyl)-5-{2-[(3-hydroxyphenyl)amino]pyrimidin-4-yl}-2-{[2-(piperidin-1-yl)ethyl]amino}thiophene-3-carbonitrileHuman2614
MAPK1 (Erk2)MAPKCMGC6nbsAB-Human11508
MAPK1 (Erk2)MAPKCMGC6qagAB1~{h}-1,2,3-triazoleHuman10982
MAPK1 (Erk2)MAPKCMGC4qp2A5-chloro-1,3-benzoxazol-2-amineHuman6078
MAPK1 (Erk2)MAPKCMGC2y9qABphosphoaminophosphonic acid-adenylate esterHuman2556
MAPK1 (Erk2)MAPKCMGC4fv1ABn-[(1s)-2-hydroxy-1-phenylethyl]-4-{4-[3-(trifluoromethyl)phenyl]-1h-pyrazol-5-yl}-1h-pyrrole-2-carboxamideHuman2613
MAPK1 (Erk2)MAPKCMGC5lcjAA[(1~{r},4~{z})-cyclooct-4-en-1-yl] ~{n}-[4-[4-[[5-chloranyl-4-[[2-(propanoylamino)phenyl]amino]pyrimidin-2-yl]amino]pyridin-2-yl]but-3-ynyl]carbamateHuman6833
MAPK1 (Erk2)MAPKCMGC5nhjA5-(2-methoxyethyl)-2-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]-6,7-dihydro-1~{h}-pyrrolo[3,2-c]pyridin-4-oneHuman7994
MAPK1 (Erk2)MAPKCMGC4iz5Badenosine-5'-diphosphateHuman2600
MAPK1 (Erk2)MAPKCMGC3sa0AAnorathyriolHuman2596
MAPK1 (Erk2)MAPKCMGC6qahAA1-azanylpropylideneazaniumHuman11354
MAPK1 (Erk2)MAPKCMGC6qawAA[1-(7~{h}-pyrrolo[2,3-d]pyrimidin-4-yl)piperidin-4-yl]methylazaniumHuman10984
MAPK1 (Erk2)MAPKCMGC5buiA3-(4-fluorophenyl)-5-(pyridin-2-yl)-4,5,6,7-tetrahydro-2h-pyrazolo[4,3-c]pyridineHuman2563
MAPK1 (Erk2)MAPKCMGC6gjdABcyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamateHuman10830
MAPK1 (Erk2)MAPKCMGC4zzoAAn-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamideHuman2620
MAPK1 (Erk2)MAPKCMGC4o6eABn-[(1s)-1-(3-chloro-4-fluorophenyl)-2-hydroxyethyl]-2-(tetrahydro-2h-pyran-4-ylamino)-5,8-dihydropyrido[3,4-d]pyrimidine-7(6h)-carboxamideHuman2553
CSNK2A2 (CK2a2)CK2CMGC7a1bAB 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13144
CSNK2A2 (CK2a2)CK2CMGC7a1zAA6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13145
CSNK2A2 (CK2a2)CK2CMGC8qcdAB4,5,6,7-tetrabromobenzotriazoleHuman15019
CSNK2A2 (CK2a2)CK2CMGC5m4uAB4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7391
CSNK2A2 (CK2a2)CK2CMGC6tewAA4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12443
CSNK2A2 (CK2a2)CK2CMGC6hmcAA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman10996
CSNK2A2 (CK2a2)CK2CMGC6qy8CA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12115
CSNK2A2 (CK2a2)CK2CMGC5ywmXnicotinic acidHuman10759
CSNK2A2 (CK2a2)CK2CMGC8qcdAA4,5,6,7-tetrabromobenzotriazoleHuman15023
CSNK2A2 (CK2a2)CK2CMGC3ofmAA3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman2728
CSNK2A2 (CK2a2)CK2CMGC6l20J(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman11994
CSNK2A2 (CK2a2)CK2CMGC5yf9BBnicotinic acidHuman11416
CSNK2A2 (CK2a2)CK2CMGC6tewAB4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12447
CSNK2A2 (CK2a2)CK2CMGC7a22AA5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13148
CSNK2A2 (CK2a2)CK2CMGC5ooiAB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9446
CSNK2A2 (CK2a2)CK2CMGC5ooiBA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9445
CSNK2A2 (CK2a2)CK2CMGC7a1bAA 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13149
CSNK2A2 (CK2a2)CK2CMGC7a2hAA5,6,7-tris(bromanyl)-1~{h}-imidazo[4,5-b]pyridineHuman13150
CSNK2A2 (CK2a2)CK2CMGC7xyhA5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrileHuman14587
CSNK2A2 (CK2a2)CK2CMGC6tguAA4-[[4-(4-chlorophenyl)-1,3-thiazol-2-yl]amino]-2-oxidanyl-benzoic acidHuman12448
CSNK2A2 (CK2a2)CK2CMGC7at9AA3-(4,5,6,7-tetrabromo-1h-benzotriazol-1-yl)propan-1-olHuman13832
CSNK2A2 (CK2a2)CK2CMGC5y9mXnicotinic acidHuman9909
CSNK2A2 (CK2a2)CK2CMGC7a22AB5,6,7-tris(bromanyl)-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13151
MAPK13 (p38d)MAPKCMGC4mygA-Human2951
MAPK13 (p38d)MAPKCMGC4mygB-Human2950
MAPK13 (p38d)MAPKCMGC8x23AA-Human15129
MAPK13 (p38d)MAPKCMGC5ekoA3-(4-methyl-1h-imidazol-1-yl)-n-[4-(pyridin-4-yloxy)phenyl]benzamideHuman6746
MAPK13 (p38d)MAPKCMGC3coiAA-Human2948
MAPK13 (p38d)MAPKCMGC4eyjA1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-yloxy)phenyl]ureaHuman2949
MAPK13 (p38d)MAPKCMGC5eknA1-(3-tert-butyl-1-methyl-1h-pyrazol-5-yl)-3-[4-(pyridin-4-ylsulfanyl)phenyl]ureaHuman6745
MAPK13 (p38d)MAPKCMGC4eymA2-(morpholin-4-yl)-n-[4-(pyridin-4-yloxy)phenyl]pyridine-4-carboxamideHuman2945
MAPK13 (p38d)MAPKCMGC3coiAB-Human2946
CDK4CDKCMGC5fwmK-Human6749
CDK4CDKCMGC5fwkK-Human6747
CDK4CDKCMGC6p8fB-Human11892
CDK4CDKCMGC3g33C-Human3384
CDK4CDKCMGC6p8eB-Human11891
CDK4CDKCMGC2w9zBB-Human3383
DYRK1ADYRKCMGC3anrB7-methoxy-1-methyl-9h-beta-carbolineHuman3729
DYRK1ADYRKCMGC5a4eDBn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6733
DYRK1ADYRKCMGC6a1fAB8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10521
DYRK1ADYRKCMGC6s1jAA3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazineHuman11365
DYRK1ADYRKCMGC6s11BB6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11372
DYRK1ADYRKCMGC6t6aAA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11857
DYRK1ADYRKCMGC6eiqB[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10529
DYRK1ADYRKCMGC6eifD4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10532
DYRK1ADYRKCMGC7a53AB(3~{e})-3-[(5-methylfuran-2-yl)methylidene]-1~{h}-indol-2-oneHuman13741
DYRK1ADYRKCMGC7a5dAA4-azanyl-2-methyl-6-pyridin-3-yl-7~{h}-pyrrolo[2,3-d]pyrimidine-5-carbonitrileHuman13742
DYRK1ADYRKCMGC6ej4D3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10545
DYRK1ADYRKCMGC4nctApkc412Human3794
DYRK1ADYRKCMGC5a3xAn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6723
DYRK1ADYRKCMGC7zh8AB6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridineHuman14488
DYRK1ADYRKCMGC6yf8D~{n}-[5-(5-methoxy-1,3-benzothiazol-2-yl)pyridin-3-yl]ethanamideHuman13460
DYRK1ADYRKCMGC4mq1AAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3796
DYRK1ADYRKCMGC5a4tAn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6732
DYRK1ADYRKCMGC7zh8AA6-bromanyl-3h-[1,2,3]triazolo[4,5-b]pyridineHuman14489
DYRK1ADYRKCMGC4mq1DBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3763
DYRK1ADYRKCMGC6s1iCB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11373
DYRK1ADYRKCMGC7a4rAB2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-oneHuman13743
DYRK1ADYRKCMGC5a4eDAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6714
DYRK1ADYRKCMGC5aikD4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3742
DYRK1ADYRKCMGC7o7kABn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman13987
DYRK1ADYRKCMGC5a3xCn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6722
DYRK1ADYRKCMGC4yljBB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3785
DYRK1ADYRKCMGC6a1gB5,5-dimethyl-8-[1-(piperidin-4-yl)ethenyl]-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10539
DYRK1ADYRKCMGC5a4lBAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6719
DYRK1ADYRKCMGC4mq2CAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3730
DYRK1ADYRKCMGC4azeC5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3788
DYRK1ADYRKCMGC5aikA4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3732
DYRK1ADYRKCMGC6eisAA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10553
DYRK1ADYRKCMGC6eivA~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10540
DYRK1ADYRKCMGC4mq1DAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3744
DYRK1ADYRKCMGC6uwyDA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11988
DYRK1ADYRKCMGC5a4lDBn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6730
DYRK1ADYRKCMGC6uwyBB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11982
DYRK1ADYRKCMGC6s1jAB3-[2-[(3~{s})-3-fluoranylpyrrolidin-1-yl]pyrimidin-4-yl]pyrazolo[1,5-b]pyridazineHuman11360
DYRK1ADYRKCMGC6t6aCB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11859
DYRK1ADYRKCMGC6qu2DA8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12091
DYRK1ADYRKCMGC6uipB4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHuman12025
DYRK1ADYRKCMGC6eirC~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10528
DYRK1ADYRKCMGC6t6aCA4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11863
DYRK1ADYRKCMGC4mq1CBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3750
DYRK1ADYRKCMGC2vx3ABn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3762
DYRK1ADYRKCMGC7ajvA4-(2,3-dibutylimidazo[4,5-b]pyridin-5-yl)pyridine-2,6-diamineHuman13594
DYRK1ADYRKCMGC7a55A3-(1-methylpyrazol-4-yl)-1~{h}-pyrazole-5-carboxylic acidHuman13746
DYRK1ADYRKCMGC6eilA[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHuman10546
DYRK1ADYRKCMGC6eiqA[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]-phenyl-methanoneHuman10554
DYRK1ADYRKCMGC6eilC-Human10552
DYRK1ADYRKCMGC7a5lAA4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amineHuman13747
DYRK1ADYRKCMGC3anqD(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3795
DYRK1ADYRKCMGC3anrA7-methoxy-1-methyl-9h-beta-carbolineHuman3778
DYRK1ADYRKCMGC6eisAB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10526
DYRK1ADYRKCMGC6eilB[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHuman10557
DYRK1ADYRKCMGC5a54An-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6736
DYRK1ADYRKCMGC6uwyBA4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11983
DYRK1ADYRKCMGC5a4lABn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6728
DYRK1ADYRKCMGC5a4eBAn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6713
DYRK1ADYRKCMGC6eisCA1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10535
DYRK1ADYRKCMGC7akaAA4-[2-methyl-3-[(2~{r})-2-pyridin-2-yloxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13596
DYRK1ADYRKCMGC4ylkAB10-chloro-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3756
DYRK1ADYRKCMGC3anrD7-methoxy-1-methyl-9h-beta-carbolineHuman3755
DYRK1ADYRKCMGC6s11BA6-pyridin-4-yl-3-[3-(trifluoromethyloxy)phenyl]imidazo[1,2-b]pyridazineHuman11378
DYRK1ADYRKCMGC5a4qCn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6738
DYRK1ADYRKCMGC4nctCpkc412Human3779
DYRK1ADYRKCMGC6qu2AB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12092
DYRK1ADYRKCMGC4yllAA10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3747
DYRK1ADYRKCMGC4mq1BAn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3773
DYRK1ADYRKCMGC6s1iDA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11362
DYRK1ADYRKCMGC4yu2CA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3741
DYRK1ADYRKCMGC6ej4A3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10520
DYRK1ADYRKCMGC3anrC7-methoxy-1-methyl-9h-beta-carbolineHuman3783
DYRK1ADYRKCMGC6s1iDB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11379
DYRK1ADYRKCMGC6s17AB~{n},~{n}-dimethyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11375
DYRK1ADYRKCMGC6s1iCA~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11366
DYRK1ADYRKCMGC7a52AA3-phenyl-1h,4h,5h-pyrazolo[3,4-d]pyrimidin-4-oneHuman13748
DYRK1ADYRKCMGC2vx3AAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3776
DYRK1ADYRKCMGC6eilD[3-azanyl-6-(5-azanyl-2-methoxy-phenyl)pyrazin-2-yl]-pyridin-3-yl-methanoneHuman10551
DYRK1ADYRKCMGC7a4sA7-chlorothieno[3,2-c]pyridin-4-amineHuman13749
DYRK1ADYRKCMGC7aj7A4-(3-methylbenzimidazol-5-yl)pyridine-2,6-diamineHuman13600
DYRK1ADYRKCMGC6s1hAA~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman11419
DYRK1ADYRKCMGC6eirB~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10558
DYRK1ADYRKCMGC6eisBB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10537
DYRK1ADYRKCMGC5a4qBn-(5-chloranyl-1,3-benzothiazol-2-yl)ethanamideHuman6729
DYRK1ADYRKCMGC6t6aDB-Human11856
DYRK1ADYRKCMGC6eivD~{n}-[3-[[4-azanyl-2-[[4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10527
DYRK1ADYRKCMGC6eisDB1-[4-fluoranyl-2-(trifluoromethyl)phenyl]-9-(1~{h}-pyrazol-4-yl)benzo[h][1,6]naphthyridin-2-oneHuman10543
DYRK1ADYRKCMGC6eirA~{n}-[4-[[4-azanyl-2-[[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]amino]-1,3-thiazol-5-yl]carbonyl]phenyl]propanamideHuman10550
DYRK1ADYRKCMGC4yu2AA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3774
DYRK1ADYRKCMGC4yljAA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3782
DYRK1ADYRKCMGC7z5nA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman14667
DYRK1ADYRKCMGC4mq2ABmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3771
DYRK1ADYRKCMGC6uipC4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHuman12026
DYRK1ADYRKCMGC5a3xDn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6718
DYRK1ADYRKCMGC4mq2BAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3792
DYRK1ADYRKCMGC4mq1BBn-(5-{[(1r)-3-amino-1-(3-chlorophenyl)propyl]carbamoyl}-2-chlorophenyl)-2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidine-6-carboxamideHuman3770
DYRK1ADYRKCMGC2vx3DBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3790
DYRK1ADYRKCMGC4yljAB10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3746
DYRK1ADYRKCMGC2vx3BBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman3769
DYRK1ADYRKCMGC6eifA4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10534
DYRK1ADYRKCMGC6s1hAB~{n},~{n}-dimethyl-4-(1~{h}-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-amineHuman11420
DYRK1ADYRKCMGC7a4rAA2-amino-3h,4h,7h-pyrrolo[2,3-d]pyrimidin-4-oneHuman13751
DYRK1ADYRKCMGC5a4lCBn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6711
DYRK1ADYRKCMGC6qu2CB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12087
DYRK1ADYRKCMGC6uipA4-ethyl-n-{4-[1-(oxan-4-yl)-1h-pyrrolo[2,3-c]pyridin-3-yl]pyridin-2-yl}piperazine-1-carboxamideHuman12027
DYRK1ADYRKCMGC5a54Dn-(6-nitro-1,3-benzothiazol-2-yl)ethanamideHuman6710
DYRK1ADYRKCMGC5a4lAAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6731
DYRK1ADYRKCMGC4mq2DBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3734
DYRK1ADYRKCMGC4nctBpkc412Human3743
DYRK1ADYRKCMGC6eijC~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10538
DYRK1ADYRKCMGC6qu2BB8-cyclopropyl-2-pyridin-3-yl-[1,3]thiazolo[5,4-f]quinazolin-9-oneHuman12088
DYRK1ADYRKCMGC7ajyA4-[2-methyl-3-[(2~{r})-2-phenoxypropyl]imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13606
DYRK1ADYRKCMGC5a4tBn-(6-cyano-3h-1,3-benzothiazol-2-ylidene)ethanamideHuman6715
DYRK1ADYRKCMGC5a3xBn-(5-oxidanyl-1,3-benzothiazol-2-yl)ethanamideHuman6724
DYRK1ADYRKCMGC7akbAA4-[3-[2-(6-bromanylpyridin-2-yl)oxyethyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13608
DYRK1ADYRKCMGC6s1iBB~{n}-methyl-~{n}-phenyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11367
DYRK1ADYRKCMGC7a4zA3-(4-methoxyphenyl)-1~{h}-pyrazol-5-amineHuman13752
DYRK1ADYRKCMGC7a4wA6-(4-methoxyphenyl)pyrimidine-2,4-diamineHuman13754
DYRK1ADYRKCMGC4mq2BBmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3787
DYRK1ADYRKCMGC5aikC4-(7-methoxy-1-(trifluoromethyl)-9h-pyrido[3,4-b]indol-9-yl)butan-1-amineHuman3754
DYRK1ADYRKCMGC6t6aBB4-chloranyl-5~{h}-cyclohepta[b]indol-10-oneHuman11861
DYRK1ADYRKCMGC4yllAB10-bromo-2-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3772
DYRK1ADYRKCMGC4yu2DA(1-chloro-7-methoxy-9h-beta-carbolin-9-yl)acetonitrileHuman3760
DYRK1ADYRKCMGC6a1fAA8-methoxy-5,5-dimethyl-5,6-dihydrobenzo[h]quinazolin-4-amineHuman10522
DYRK1ADYRKCMGC6ej4B3-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)anilineHuman10523
DYRK1ADYRKCMGC5a4lDAn-(5-fluoranyl-1,3-benzothiazol-2-yl)ethanamideHuman6739
DYRK1ADYRKCMGC6uwyAB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11987
DYRK1ADYRKCMGC4mq2AAmethyl 4-chloro-3-{[(2-methoxy-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl)carbonyl]amino}benzoateHuman3752
DYRK1ADYRKCMGC7o7kAAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman13988
DYRK1ADYRKCMGC3anqB(1z)-1-(3-ethyl-5-hydroxy-1,3-benzothiazol-2(3h)-ylidene)propan-2-oneHuman3745
DYRK1ADYRKCMGC6eifC4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10525
DYRK1ADYRKCMGC6eijA~{n}-[5-[3-(2-morpholin-4-ylethylcarbamoylamino)phenyl]-[1,3]thiazolo[5,4-b]pyridin-2-yl]cyclopropanecarboxamideHuman10518
DYRK1ADYRKCMGC4yljDA10-iodo-11h-indolo[3,2-c]quinoline-6-carboxylic acidHuman3784
DYRK1ADYRKCMGC5a4eCBn-(5-methoxy-1,3-benzothiazol-2-yl)ethanamideHuman6727
DYRK1ADYRKCMGC6s14AB~{n}-cyclopropyl-~{n}-methyl-4-pyrazolo[1,5-b]pyridazin-3-yl-pyrimidin-2-amineHuman11421
DYRK1ADYRKCMGC7fhtAA(5~{z})-5-[(3-ethynyl-4-methoxy-phenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-oneHuman14161
DYRK1ADYRKCMGC6eifB4-(3-pyridin-3-yl-1~{h}-pyrrolo[2,3-b]pyridin-5-yl)benzenesulfonamideHuman10544
DYRK1ADYRKCMGC6uwyDB4-(7-methoxy-1-methyl-9h-beta-carbolin-9-yl)butanamideHuman11986
DYRK1ADYRKCMGC7a5lAB4-[2-methyl-4-(thiophen-3-ylmethoxy)-7~{h}-pyrrolo[2,3-d]pyrimidin-5-yl]pyridin-2-amineHuman13758
MAPK10 (JNK3)MAPKCMGC3v6rBA4-{[4-(dimethylamino)butanoyl]amino}-n-(3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}phenyl)benzamideHuman3427
MAPK10 (JNK3)MAPKCMGC2o2uAn-(3-cyano-4,5,6,7-tetrahydro-1-benzothien-2-yl)-2-fluorobenzamideHuman3457
MAPK10 (JNK3)MAPKCMGC3g90X(3e)-5-fluoro-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-1h-indole-2,3-dione 3-oximeHuman3477
MAPK10 (JNK3)MAPKCMGC6eq9ABphosphomethylphosphonic acid adenylate esterHuman10509
MAPK10 (JNK3)MAPKCMGC3fv8AB5-bromo-n-(3-chloro-2-(4-(prop-2-ynyl)piperazin-1-yl)phenyl)furan-2-carboxamideHuman3426
MAPK10 (JNK3)MAPKCMGC3da6An-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)naphthalen-1-yl]-1h-benzimidazol-2-amineHuman3476
MAPK10 (JNK3)MAPKCMGC6emhBB4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10501
MAPK10 (JNK3)MAPKCMGC8vs0A(4p)-4-[6-fluoro-5-(2-methoxyanilino)-1h-indazol-1-yl]-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamideHuman15635
MAPK10 (JNK3)MAPKCMGC2r9sAn-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamideHuman3450
MAPK10 (JNK3)MAPKCMGC4h39AA-Human3460
MAPK10 (JNK3)MAPKCMGC4kkgA-Human3443
MAPK10 (JNK3)MAPKCMGC3cgoA2-{4-[(4-imidazo[1,2-a]pyridin-3-ylpyrimidin-2-yl)amino]piperidin-1-yl}-n-methylacetamideHuman6771
MAPK10 (JNK3)MAPKCMGC8vtfA(4p)-4-[6-fluoro-5-(2-methoxyanilino)-1h-indazol-1-yl]-n-(oxetan-3-yl)thiophene-2-carboxamideHuman15636
MAPK10 (JNK3)MAPKCMGC3oy1A5-[2-(cyclohexylamino)pyridin-4-yl]-4-naphthalen-2-yl-2-(tetrahydro-2h-pyran-4-yl)-2,4-dihydro-3h-1,2,4-triazol-3-oneHuman3469
MAPK10 (JNK3)MAPKCMGC4h3bCA-Human3475
MAPK10 (JNK3)MAPKCMGC7oreAB4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamideHuman13810
MAPK10 (JNK3)MAPKCMGC6ekdAB4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10502
MAPK10 (JNK3)MAPKCMGC4y46A1-{trans-4-[(8-cyclopentyl-7-oxo-7,8-dihydropyrido[2,3-d]pyrimidin-2-yl)amino]cyclohexyl}-3-propan-2-ylureaHuman3414
MAPK10 (JNK3)MAPKCMGC7oreAA4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamideHuman13811
MAPK10 (JNK3)MAPKCMGC2b1pA3-{6-[(2-chlorophenyl)amino]-1h-indazol-3-yl}-5-{[4-(dimethylamino)butanoyl]amino}benzoic acidHuman3464
MAPK10 (JNK3)MAPKCMGC1pmuA9-(4-hydroxyphenyl)-2,7-phenanthrolineHuman3474
MAPK10 (JNK3)MAPKCMGC4h3bAA-Human3480
MAPK10 (JNK3)MAPKCMGC4z9lAAphosphoaminophosphonic acid-adenylate esterHuman3432
MAPK10 (JNK3)MAPKCMGC7orfAAn-[4-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]phenyl]-3-(propanoylamino)benzamideHuman13812
MAPK10 (JNK3)MAPKCMGC6emhAA4-(4-methyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10508
MAPK10 (JNK3)MAPKCMGC3ttjAB9-cyclopentyl-n~8~-(2-fluorophenyl)-n~2~-(4-methoxyphenyl)-9h-purine-2,8-diamineHuman3428
MAPK10 (JNK3)MAPKCMGC2r9sBn-(tert-butyl)-4-[5-(pyridin-2-ylamino)quinolin-3-yl]benzenesulfonamideHuman3420
MAPK10 (JNK3)MAPKCMGC7ksiA4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-5-methyl-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13387
MAPK10 (JNK3)MAPKCMGC1jnkAphosphoaminophosphonic acid-adenylate esterHuman3451
MAPK10 (JNK3)MAPKCMGC6eq9AAphosphomethylphosphonic acid adenylate esterHuman10500
MAPK10 (JNK3)MAPKCMGC3g9nA(3z)-1-[(6-fluoro-4h-1,3-benzodioxin-8-yl)methyl]-4-phenyl-1h-indole-2,3-dione 3-oximeHuman3416
MAPK10 (JNK3)MAPKCMGC7oreAC4-(dimethylamino)-n-[(5z)-9-[[4-[5-(4-fluorophenyl)-3-methyl-2-methylsulfanyl-imidazol-4-yl]pyridin-2-yl]amino]-11,12-dihydrobenzo[c][1,2]benzodiazocin-2-yl]butanamideHuman13813
MAPK10 (JNK3)MAPKCMGC4kkhAcyclopropyl[(3r)-3-({4-[6-hydroxy-2-(naphthalen-2-yl)-1h-benzimidazol-1-yl]pyrimidin-2-yl}amino)piperidin-1-yl]methanoneHuman3419
MAPK10 (JNK3)MAPKCMGC3ptgAn-[4-methyl-3-(1h-1,2,4-triazol-5-yl)thiophen-2-yl]-2-(2-oxo-3,4-dihydroquinolin-1(2h)-yl)acetamideHuman3470
MAPK10 (JNK3)MAPKCMGC7ksjA4-(4-{[(2-chloro-6-fluorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(oxetan-3-yl)thiophene-2-carboxamideHuman13388
MAPK10 (JNK3)MAPKCMGC2wajAB1-(3-bromophenyl)-7-chloro-6-methoxy-3,4-dihydroisoquinolineHuman3471
MAPK10 (JNK3)MAPKCMGC2ok1ABn-benzyl-4-[4-(3-chlorophenyl)-1h-pyrazol-3-yl]-1h-pyrrole-2-carboxamideHuman3473
MAPK10 (JNK3)MAPKCMGC4w4yA3-(4-{[(4-methylphenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-n-(2-methylpyridin-4-yl)benzamideHuman3447
MAPK10 (JNK3)MAPKCMGC6ekdAA4-(4-methyl-2-methylsulfanyl-1~{h}-imidazol-5-yl)-~{n}-(4-morpholin-4-ylphenyl)pyridin-2-amineHuman10498
SRPK1SRPKCMGC4wuaAAn-[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamideHuman9471
SRPK1SRPKCMGC6fadB-Human11640
SRPK1SRPKCMGC4wuaABn-[2-(1-piperidinyl)-5-(trifluoromethyl)phenyl]-4-pyridinecarboxamideHuman9469
SRPK1SRPKCMGC6fadC-Human11639
SRPK1SRPKCMGC5my8AAsphinx31Human9466
SRPK1SRPKCMGC5my8ABsphinx31Human9468
SRPK1SRPKCMGC7zksAAn-[3-[[[2-(6-chloranyl-5-fluoranyl-1h-benzimidazol-2-yl)pyrimidin-4-yl]amino]methyl]pyridin-2-yl]-n-methyl-methanesulfonamideHuman14619
SRPK1SRPKCMGC5mxxAA5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman9470
SRPK1SRPKCMGC7dd1A-Human13510
SRPK1SRPKCMGC5mxxAB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman9467
GSK3AGSKCMGC7sxfAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14780
GSK3AGSKCMGC7sxfAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14781
GSK3AGSKCMGC7sxgAB(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14782
GSK3AGSKCMGC7sxgAA(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14783
CDKL3CDKLCMGC3zduA[4-({4-[(3-cyclopentyl-1h-pyrazol-5-yl)amino]pyrimidin-2-yl}amino)phenyl]acetonitrileHuman4677
CDKL1CDKLCMGC4aguAn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman761
CDKL1CDKLCMGC4aguBn-(5-{[(2s)-4-amino-2-(3-chlorophenyl)butanoyl]amino}-1h-indazol-3-yl)benzamideHuman760
MAPK14 (p38a)MAPKCMGC4r3cAA6-(4-methylpiperazin-1-yl)-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazineHuman5198
MAPK14 (p38a)MAPKCMGC3ctqAn-benzyl-1-[5-({5-tert-butyl-2-methoxy-3-[(methylsulfonyl)amino]phenyl}carbamoyl)-2-methylphenyl]-1h-1,2,3-triazole-4-carboxamideHuman5220
MAPK14 (p38a)MAPKCMGC5tcoA3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulene-9-carboxamideHuman8031
MAPK14 (p38a)MAPKCMGC2gfsAB[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanoneHuman5050
MAPK14 (p38a)MAPKCMGC3hv5AA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5203
MAPK14 (p38a)MAPKCMGC3nnvAA1-{3-tert-butyl-1-[4-(hydroxymethyl)phenyl]-1h-pyrazol-5-yl}-3-naphthalen-1-ylureaHuman5037
MAPK14 (p38a)MAPKCMGC3ds6An-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5074
MAPK14 (p38a)MAPKCMGC4dliA-Human5092
MAPK14 (p38a)MAPKCMGC2y8oAA-Human5079
MAPK14 (p38a)MAPKCMGC3oefXB-Human5231
MAPK14 (p38a)MAPKCMGC5tbeA~{n}-[2,4-bis(fluoranyl)-5-[[9-(2-morpholin-4-ylethylcarbamoyl)-11-oxidanylidene-5,6-dihydrodibenzo[1,2-~{d}:1',2'-~{f}][7]annulen-3-yl]amino]phenyl]thiophene-2-carboxamideHuman8032
MAPK14 (p38a)MAPKCMGC3k3jA2-(4-fluorophenyl)-3-oxo-6-pyridin-4-yl-n-[2-(trifluoromethyl)benzyl]-2,3-dihydropyridazine-4-carboxamideHuman5047
MAPK14 (p38a)MAPKCMGC6sfjAC~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamideHuman11618
MAPK14 (p38a)MAPKCMGC5omgAA3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxideHuman11246
MAPK14 (p38a)MAPKCMGC3hrbA[3-amino-2-(2-methylphenyl)-1-oxidopyridin-4-yl](2,4-difluorophenyl)methanoneHuman5202
MAPK14 (p38a)MAPKCMGC1w84A3-(2-pyridin-4-ylethyl)-1h-indoleHuman5065
MAPK14 (p38a)MAPKCMGC2gfsAA[5-amino-1-(4-fluorophenyl)-1h-pyrazol-4-yl](3-{[(2r)-2,3-dihydroxypropyl]oxy}phenyl)methanoneHuman5227
MAPK14 (p38a)MAPKCMGC3u8wA3-[3-(2-chloro-6-fluorophenyl)-5-ethyl-6-oxo-5,6-dihydro[1,2,4]triazolo[4,3-b]pyridazin-7-yl]-n-cyclopropyl-4-methylbenzamideHuman5192
MAPK14 (p38a)MAPKCMGC3hucAAn-[2-phenyl-4-(1h-pyrazol-3-ylamino)quinazolin-7-yl]prop-2-enamideHuman5027
MAPK14 (p38a)MAPKCMGC4kiqAethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5141
MAPK14 (p38a)MAPKCMGC1wbtA3-fluoro-5-morpholin-4-yl-n-[1-(2-pyridin-4-ylethyl)-1h-indol-6-yl]benzamideHuman5082
MAPK14 (p38a)MAPKCMGC3k3iAB(3s)-3-[4-(4-bromophenyl)-1h-imidazol-2-yl]-1,2,3,4-tetrahydroisoquinolineHuman5022
MAPK14 (p38a)MAPKCMGC3nnwAB2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamideHuman5138
MAPK14 (p38a)MAPKCMGC5mtxAB3-[(3-benzamido-4-fluoranyl-phenyl)amino]-~{n}-(2-morpholin-4-ylethyl)-11-oxidanylidene-6~{h}-benzo[c][1]benzoxepine-9-carboxamideHuman8379
MAPK14 (p38a)MAPKCMGC6sfiAA~{n}-[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]-2-[[[1-(2-methylphenyl)pyrazol-4-yl]carbonylamino]methyl]-1,3-thiazole-5-carboxamideHuman11613
MAPK14 (p38a)MAPKCMGC6sfoAB5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman11621
MAPK14 (p38a)MAPKCMGC1w83An-[4-chloro-3-(pyridin-3-yloxymethyl)-phenyl]-3-fluoro-Human4986
MAPK14 (p38a)MAPKCMGC5mtyA~{n}-[2,4-bis(fluoranyl)-5-[[14-(2-hydroxyethylcarbamoyl)-2-oxidanylidene-6-tricyclo[9.4.0.0^{3,8}]pentadeca-1(15),3(8),4,6,11,13-hexaenyl]amino]phenyl]thiophene-2-carboxamideHuman8383
MAPK14 (p38a)MAPKCMGC5o8vA-Human8380
MAPK14 (p38a)MAPKCMGC3lfbAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-(1,3-thiazol-2-yl)ureaHuman5001
MAPK14 (p38a)MAPKCMGC5etfAA-Human7134
MAPK14 (p38a)MAPKCMGC3fsfA3-(2,6-dichlorophenyl)-7-({4-[(diethylamino)methoxy]phenyl}amino)-1-methyl-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1h)-oneHuman5097
MAPK14 (p38a)MAPKCMGC3fmkA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(2h-tetrazol-2-yl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5209
MAPK14 (p38a)MAPKCMGC3uvqAAn-{5-[(7-{[(2r)-2,3-dihydroxypropyl]oxy}-5-oxo-10,11-dihydro-5h-dibenzo[a,d][7]annulen-2-yl)amino]-2-fluorophenyl}benzamideHuman5183
MAPK14 (p38a)MAPKCMGC4eh9A-Human4982
MAPK14 (p38a)MAPKCMGC1bl6A4-(4-fluorophenyl)-1-cycloropropylmethyl-5-(4-pyridyl)-imidazoleHuman5243
MAPK14 (p38a)MAPKCMGC6tcaDAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12486
MAPK14 (p38a)MAPKCMGC6sfkAB~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-phenyl-5-(trifluoromethyl)pyrazole-4-carboxamideHuman11620
MAPK14 (p38a)MAPKCMGC3iphAB6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamideHuman5156
MAPK14 (p38a)MAPKCMGC3pg3AA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}ureaHuman5122
MAPK14 (p38a)MAPKCMGC3flsA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1r)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5119
MAPK14 (p38a)MAPKCMGC3queA2-[(2,4-difluorophenyl)amino]-7-{[(2r)-2,3-dihydroxypropyl]oxy}-10,11-dihydro-5h-dibenzo[a,d][7]annulen-5-oneHuman5095
MAPK14 (p38a)MAPKCMGC6hwtAB3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamideHuman11254
MAPK14 (p38a)MAPKCMGC3nnuAB2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamideHuman5059
MAPK14 (p38a)MAPKCMGC4kiqCethyl 6-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]carbamoyl}-1h-indole-1-carboxylateHuman5215
MAPK14 (p38a)MAPKCMGC3mh3A-Human5109
MAPK14 (p38a)MAPKCMGC3zsgABtak-715Human5098
MAPK14 (p38a)MAPKCMGC6sfjAB~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamideHuman11616
MAPK14 (p38a)MAPKCMGC6qyxA-Human12127
MAPK14 (p38a)MAPKCMGC3flzA8-methyl-6-phenoxy-2-(tetrahydro-2h-pyran-4-ylamino)pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5204
MAPK14 (p38a)MAPKCMGC3hubA2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamideHuman5029
MAPK14 (p38a)MAPKCMGC6hwvAA-Human11253
MAPK14 (p38a)MAPKCMGC2lgcA2-Human5093
MAPK14 (p38a)MAPKCMGC3newAA-Human5025
MAPK14 (p38a)MAPKCMGC3qudAB{4-[(2-aminophenyl)amino]phenyl}(phenyl)methanoneHuman5262
MAPK14 (p38a)MAPKCMGC3gc7AA5-(2-chloro-4-fluorophenyl)-1-(2,6-dichlorophenyl)-7-[1-(1-methylethyl)piperidin-4-yl]-3,4-dihydroquinazolin-2(1h)-oneHuman5061
MAPK14 (p38a)MAPKCMGC4eh3AnaringeninHuman5042
MAPK14 (p38a)MAPKCMGC3uvrAA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}ureaHuman6880
MAPK14 (p38a)MAPKCMGC6hwuAA-Human11247
MAPK14 (p38a)MAPKCMGC5mz3AA~{n}-[3-(2-acetamidoimidazo[1,2-a]pyridin-6-yl)-4-methyl-phenyl]-3-(trifluoromethyl)benzamideHuman8680
MAPK14 (p38a)MAPKCMGC4eh2A3-phenylquinazolin-4(3h)-oneHuman5244
MAPK14 (p38a)MAPKCMGC2fslX-Human5264
MAPK14 (p38a)MAPKCMGC2onlA-Human5177
MAPK14 (p38a)MAPKCMGC3ha8ABn~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamideHuman5187
MAPK14 (p38a)MAPKCMGC3mvmB4-{[5-(isoxazol-3-ylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5210
MAPK14 (p38a)MAPKCMGC3itzA4-chloro-n-cyclopropyl-3-{[1-(2,6-difluorophenyl)-1h-pyrazolo[3,4-d]pyridazin-4-yl]amino}benzamideHuman5135
MAPK14 (p38a)MAPKCMGC3kq7ABn-(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)-6-({2-[(2s)-1-methylpyrrolidin-2-yl]ethyl}amino)pyridine-3-carboxamideHuman5057
MAPK14 (p38a)MAPKCMGC6qe1A1-[5-~{tert}-butyl-2-(4-methylphenyl)pyrazol-3-yl]-3-[(1~{s},4~{r})-4-[(3-propan-2-yl-[1,2,4]triazolo[4,3-a]pyridin-6-yl)oxy]-1,2,3,4-tetrahydronaphthalen-1-yl]ureaHuman11957
MAPK14 (p38a)MAPKCMGC3uvpAAn-{2-fluoro-5-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}benzamideHuman5070
MAPK14 (p38a)MAPKCMGC3newAB-Human5248
MAPK14 (p38a)MAPKCMGC3hv4A1-{3-[(6-aminoquinolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5121
MAPK14 (p38a)MAPKCMGC3bx5An-[2-methyl-5-(methylcarbamoyl)phenyl]-2-{[(1r)-1-methylpropyl]amino}-1,3-thiazole-5-carboxamideHuman5000
MAPK14 (p38a)MAPKCMGC3nnwAA2-[3-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-2,5-dihydro-1h-pyrazol-1-yl)phenyl]acetamideHuman5139
MAPK14 (p38a)MAPKCMGC2fstXA-Human5080
MAPK14 (p38a)MAPKCMGC6tcaBBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12488
MAPK14 (p38a)MAPKCMGC1kv1A1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5252
MAPK14 (p38a)MAPKCMGC2i0hAB2-(3-{(2-chloro-4-fluorophenyl)[1-(2-chlorophenyl)-6-oxo-1,6-dihydropyridazin-3-yl]amino}propyl)-1h-isoindole-1,3(2h)-dioneHuman5009
MAPK14 (p38a)MAPKCMGC3pg3AB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{4-[2-(pyridin-3-ylmethoxy)ethyl]-1,3-thiazol-2-yl}ureaHuman5096
MAPK14 (p38a)MAPKCMGC4aa4An-[4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]phenyl]furan-3-carboxamideHuman5045
MAPK14 (p38a)MAPKCMGC1wbsA3-fluoro-5-morpholin-4-yl-n-[3-(2-pyridin-4-ylethyl)-1h-indol-5-yl]benzamideHuman5258
MAPK14 (p38a)MAPKCMGC1m7qA1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperazin-1-yl-3,4-dihydroquinazolin-2(1h)-oneHuman5128
MAPK14 (p38a)MAPKCMGC4e6aA-Human5238
MAPK14 (p38a)MAPKCMGC3bv3A5-methyl-4-[(2-methyl-5-{[(3-morpholin-4-ylphenyl)carbonyl]amino}phenyl)amino]-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5207
MAPK14 (p38a)MAPKCMGC6tcaFBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12490
MAPK14 (p38a)MAPKCMGC3hecAA4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamideHuman5166
MAPK14 (p38a)MAPKCMGC3lffAA(4-{3-tert-butyl-5-[(1,3-thiazol-2-ylcarbamoyl)amino]-1h-pyrazol-1-yl}phenyl)acetic acidHuman5140
MAPK14 (p38a)MAPKCMGC5etiA-Human6362
MAPK14 (p38a)MAPKCMGC6tcaBAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12491
MAPK14 (p38a)MAPKCMGC1w82An-[(3z)-5-tert-butyl-2-phenyl-1,2-dihydro-3h-pyrazol-3-ylidene]-n'-(4-chlorophenyl)ureaHuman5165
MAPK14 (p38a)MAPKCMGC4geoA-Human5190
MAPK14 (p38a)MAPKCMGC6tcaDBn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12492
MAPK14 (p38a)MAPKCMGC3gcsAA4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5077
MAPK14 (p38a)MAPKCMGC3iw7A2-({4-[(4-benzylpiperidin-1-yl)carbonyl]benzyl}sulfanyl)-3h-imidazo[4,5-c]pyridineHuman5084
MAPK14 (p38a)MAPKCMGC3d7zABn~3~-cyclopropyl-n~4~'-(cyclopropylmethyl)-6-methylbiphenyl-3,4'-dicarboxamideHuman5108
MAPK14 (p38a)MAPKCMGC6sfoAA5-azanyl-~{n}-[[4-(3-cyclohexylpropylcarbamoyl)phenyl]methyl]-1-phenyl-pyrazole-4-carboxamideHuman11615
MAPK14 (p38a)MAPKCMGC2zazAA4-{4-[(5-hydroxy-2-methylphenyl)amino]quinolin-7-yl}-1,3-thiazole-2-carbaldehydeHuman4980
MAPK14 (p38a)MAPKCMGC1r39A-Human5116
MAPK14 (p38a)MAPKCMGC5omgAB3-(4-fluorophenyl)-4-methyl-1~{h}-pyrazolo[4,3-c][1,2]benzothiazine 5,5-dioxideHuman11245
MAPK14 (p38a)MAPKCMGC1a9uA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5229
MAPK14 (p38a)MAPKCMGC3flqA6-(2,4-difluorophenoxy)-8-methyl-2-{[(1s)-1-methyl-2-(methylsulfonyl)ethyl]amino}pyrido[2,3-d]pyrimidin-7(8h)-oneHuman5168
MAPK14 (p38a)MAPKCMGC3uvrAB1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5h-benzo[7]annulen-2-yl)amino]phenyl}ureaHuman6879
MAPK14 (p38a)MAPKCMGC3o8tA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5167
MAPK14 (p38a)MAPKCMGC3o8pA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5071
MAPK14 (p38a)MAPKCMGC2yisA1-[3-tert-butyl-1-(3-chloro-4-hydroxyphenyl)-1h-pyrazol-5-yl]-3-{2-[(3-{2-[(2-hydroxyethyl)sulfanyl]phenyl}[1,2,4]triazolo[4,3-a]pyridin-6-yl)sulfanyl]benzyl}ureaHuman5240
MAPK14 (p38a)MAPKCMGC3iw6ABethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylateHuman5154
MAPK14 (p38a)MAPKCMGC2qd9A1-[(3ar)-5-{[3-(2,4-difluorophenyl)-5,6-dihydroimidazo[1,5-a]pyrazin-7(8h)-yl]carbonyl}-6-methoxy-3ah-pyrrolo[2,3-b]pyridin-3-yl]-2-[(3r)-3-hydroxypyrrolidin-1-yl]-2-oxoethanoneHuman5197
MAPK14 (p38a)MAPKCMGC3mvlB4-{[5-(cyclopropylcarbamoyl)-2-methylphenyl]amino}-5-methyl-n-propylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5091
MAPK14 (p38a)MAPKCMGC1oveAA1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-oneHuman5178
MAPK14 (p38a)MAPKCMGC3iphAA6-[5-(cyclopropylcarbamoyl)-2-methylphenyl]-n-(cyclopropylmethyl)pyridine-3-carboxamideHuman4999
MAPK14 (p38a)MAPKCMGC6hwtAA3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-(2-phenylhydrazinyl)-1,3-thiazol-5-yl]pyridin-2-yl]propanamideHuman11248
MAPK14 (p38a)MAPKCMGC3l8sA3-[(4-bromo-2,6-difluorobenzyl)oxy]-5-{[(4-pyrrolidin-1-ylbutyl)carbamoyl]amino}isothiazole-4-carboxamideHuman5055
MAPK14 (p38a)MAPKCMGC4f9wABn,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5106
MAPK14 (p38a)MAPKCMGC6tcaHAn-[5-(dimethylsulfamoyl)-2-methylphenyl]-1-phenyl-5-propyl-1h-pyrazole-4-carboxamideHuman12493
MAPK14 (p38a)MAPKCMGC3fi4A(2s)-1-{[3-(2-chlorophenyl)-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propan-2-olHuman5051
MAPK14 (p38a)MAPKCMGC3o8uA1-(5-tert-butyl-2-methyl-2h-pyrazol-3-yl)-3-(4-chloro-phenyl)-ureaHuman5250
MAPK14 (p38a)MAPKCMGC3s3iA3-(3-tert-butyl[1,2,4]triazolo[4,3-a]pyridin-7-yl)-n-cyclopropyl-4-methylbenzamideHuman5169
MAPK14 (p38a)MAPKCMGC3dt1An-cyclopropyl-4-methyl-3-{2-[(2-morpholin-4-ylethyl)amino]quinazolin-6-yl}benzamideHuman5086
MAPK14 (p38a)MAPKCMGC3lfdA1-{4-[2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5102
MAPK14 (p38a)MAPKCMGC3gcvAB1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5174
MAPK14 (p38a)MAPKCMGC1ouyA1-(2,6-dichlorophenyl)-6-[(2,4-difluorophenyl)sulfanyl]-7-(1,2,3,6-tetrahydro-4-pyridinyl)-3,4-dihydropyrido[3,2-d]pyrimidin-2(1h)-oneHuman7258
MAPK14 (p38a)MAPKCMGC2zb1ABn-(cyclopropylmethyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)biphenyl-4-carboxamideHuman5103
MAPK14 (p38a)MAPKCMGC5etaA-Human7136
MAPK14 (p38a)MAPKCMGC2yixA1-ethyl-3-(2-{[3-(1-methylethyl)[1,2,4]triazolo[4,3-a]pyridin-6-yl]sulfanyl}benzyl)ureaHuman5143
MAPK14 (p38a)MAPKCMGC3zs5AA4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman4987
MAPK14 (p38a)MAPKCMGC8x3mAA-Human15701
MAPK14 (p38a)MAPKCMGC3rinAn-cyclopropyl-4-methyl-3-(2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indol]-6'-yl)benzamideHuman5239
MAPK14 (p38a)MAPKCMGC1wbvA3-fluoro-n-1h-indol-5-yl-5-morpholin-4-ylbenzamideHuman5148
MAPK14 (p38a)MAPKCMGC4f9yAAn,n-dimethyl-6-(naphthalen-1-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5225
MAPK14 (p38a)MAPKCMGC2zb0ABn-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamideHuman5147
MAPK14 (p38a)MAPKCMGC3nnuAA2-{3-[(5e)-5-{[(2,3-dichlorophenyl)carbamoyl]imino}-3-thiophen-2-yl-2,5-dihydro-1h-pyrazol-1-yl]phenyl}acetamideHuman5094
MAPK14 (p38a)MAPKCMGC3zyaAA2-amino-phenylamino-dibenzosuberoneHuman5105
MAPK14 (p38a)MAPKCMGC4eh7AB(3-phenoxyphenyl)methanolHuman5020
MAPK14 (p38a)MAPKCMGC3iw6AAethyl 4-[(4-benzylpiperazin-1-yl)carbonyl]-1-ethyl-3,5-dimethyl-1h-pyrrole-2-carboxylateHuman4990
MAPK14 (p38a)MAPKCMGC1w7hA3-(benzyloxy)pyridin-2-amineHuman5023
MAPK14 (p38a)MAPKCMGC2okrD-Human5100
MAPK14 (p38a)MAPKCMGC9cj2AB-Human15702
MAPK14 (p38a)MAPKCMGC4aa5An-cyclopropyl-4-methyl-3-[6-(4-methylpiperazin-1-yl)-4-oxidanylidene-quinazolin-3-yl]benzamideHuman5206
MAPK14 (p38a)MAPKCMGC4fa2ABtrans-4-[4-(4-fluorophenyl)-5-(2-methoxypyrimidin-4-yl)-1h-imidazol-1-yl]cyclohexanolHuman5145
MAPK14 (p38a)MAPKCMGC6hwvAB-Human11250
MAPK14 (p38a)MAPKCMGC5n66A1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman8524
MAPK14 (p38a)MAPKCMGC2lgcA1-Human5021
MAPK14 (p38a)MAPKCMGC3gcuAB1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5162
MAPK14 (p38a)MAPKCMGC6m95A(4-benzylpiperidin-1-yl)[2-methoxy-4-(methylsulfanyl)phenyl]methanoneHuman11252
MAPK14 (p38a)MAPKCMGC4eh8AB[3-(benzyloxy)phenyl]methanolHuman5014
MAPK14 (p38a)MAPKCMGC2lgcA10-Human5063
MAPK14 (p38a)MAPKCMGC2zb0AAn-(3-cyanophenyl)-2'-methyl-5'-(5-methyl-1,3,4-oxadiazol-2-yl)-4-biphenylcarboxamideHuman5099
MAPK14 (p38a)MAPKCMGC6anlABtak-715Human9518
MAPK14 (p38a)MAPKCMGC3ds6Dn-cyclopropyl-4-methyl-3-[1-(2-methylphenyl)phthalazin-6-yl]benzamideHuman5123
MAPK14 (p38a)MAPKCMGC5ml5A3-(2,5-dimethoxyphenyl)-~{n}-[4-[4-(4-fluorophenyl)-2-methylsulfanyl-1~{h}-imidazol-5-yl]pyridin-2-yl]propanamideHuman7544
MAPK14 (p38a)MAPKCMGC2rg6A4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methyl-n-[(1s)-1-phenylethyl]pyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5228
MAPK14 (p38a)MAPKCMGC9cj4AA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman15703
MAPK14 (p38a)MAPKCMGC3ha8AAn~2~-{4-[6-(3,4-dihydroquinolin-1(2h)-ylcarbonyl)-1h-benzimidazol-1-yl]-6-ethoxy-1,3,5-triazin-2-yl}-3-(2,2-dimethyl-4h-1,3-benzodioxin-6-yl)-n-methyl-l-alaninamideHuman5253
MAPK14 (p38a)MAPKCMGC2lgcA6-Human5219
MAPK14 (p38a)MAPKCMGC3e93AA4-methyl-n-(3-morpholin-4-ylphenyl)-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)benzamideHuman5241
MAPK14 (p38a)MAPKCMGC9cj4AB1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman15704
MAPK14 (p38a)MAPKCMGC3gcsAB4-{4-[({[4-chloro-3-(trifluoromethyl)phenyl]amino}carbonyl)amino]phenoxy}-n-methylpyridine-2-carboxamideHuman5052
MAPK14 (p38a)MAPKCMGC4eh6An-phenylpyridine-3-carboxamideHuman5083
MAPK14 (p38a)MAPKCMGC3bv2A5-methyl-4-[(2-methyl-5-{[(2-morpholin-4-ylpyridin-4-yl)carbonyl]amino}phenyl)amino]-n-(1-phenylethenyl)pyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5191
MAPK14 (p38a)MAPKCMGC8x3mAB-Human15705
MAPK14 (p38a)MAPKCMGC3hllAB3-{3-bromo-4-[(2,4-difluorobenzyl)oxy]-6-methyl-2-oxopyridin-1(2h)-yl}-n,4-dimethylbenzamideHuman5104
MAPK14 (p38a)MAPKCMGC3mptAAn-(furan-2-ylmethyl)-4-[(2-methylphenyl)carbonyl]-1h-pyrrole-2-carboxamideHuman5224
MAPK14 (p38a)MAPKCMGC4e5bA-Human5221
MAPK14 (p38a)MAPKCMGC2lgcA7-Human5161
MAPK14 (p38a)MAPKCMGC5xyxAAn-(2-chloro-6-fluorobenzyl)-5-(furan-2-yl)-2h-1,2,4-triazol-3-amineHuman9519
MAPK14 (p38a)MAPKCMGC4f9wAAn,n-dimethyl-6-(naphthalen-2-yl)-5-(pyridin-4-yl)pyridazin-3-amineHuman5130
MAPK14 (p38a)MAPKCMGC1zz2An-[3-(4-fluorophenoxy)phenyl]-4-[(2-hydroxybenzyl)amino]piperidine-1-sulfonamideHuman5164
MAPK14 (p38a)MAPKCMGC3gcuBB1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5126
MAPK14 (p38a)MAPKCMGC3iw8A1-{4-[(1s)-1-amino-2-(benzyloxy)ethyl]-1,3-thiazol-2-yl}-3-(3-chloro-4-fluorophenyl)ureaHuman5181
MAPK14 (p38a)MAPKCMGC4ewqAB3-phenyl-4-(pyridin-4-yl)-6-[4-(pyrimidin-2-yl)piperazin-1-yl]pyridazineHuman5245
MAPK14 (p38a)MAPKCMGC4eh4Aphenyl(piperidin-1-yl)methanoneHuman5043
MAPK14 (p38a)MAPKCMGC5etfAB-Human7135
MAPK14 (p38a)MAPKCMGC3fklAn-cyclopropyl-4-methyl-3-[8-methyl-7-oxo-2-(tetrahydro-2h-pyran-4-ylamino)-7,8-dihydropyrido[2,3-d]pyrimidin-6-yl]benzamideHuman5172
MAPK14 (p38a)MAPKCMGC4eh5Abenzyl pyridine-3-carboxylateHuman5185
MAPK14 (p38a)MAPKCMGC5n67AB-Human8521
MAPK14 (p38a)MAPKCMGC4zthAA6-chloro-3-phenyl-4-(pyridin-4-yl)pyridazineHuman6706
MAPK14 (p38a)MAPKCMGC1zyjA4-phenoxy-n-(pyridin-2-ylmethyl)benzamideHuman5058
MAPK14 (p38a)MAPKCMGC3fknA3-[2-chloro-5-(methylsulfonyl)phenyl]-6-(2,4-difluorophenoxy)-1h-pyrazolo[3,4-d]pyrimidineHuman5049
MAPK14 (p38a)MAPKCMGC6sfjAA~{n}-[5-[[(2~{s})-1-azanyl-4-cyclohexyl-1-oxidanylidene-butan-2-yl]carbamoyl]-2-methyl-phenyl]-1-(2-methylphenyl)pyrazole-4-carboxamideHuman11614
MAPK14 (p38a)MAPKCMGC1oveAB1-(2,6-dichlorophenyl)-5-(2,4-difluorophenyl)-7-piperidin-4-yl-3,4-dihydroquinolin-2(1h)-oneHuman5087
MAPK14 (p38a)MAPKCMGC2rg5An-ethyl-4-{[5-(methoxycarbamoyl)-2-methylphenyl]amino}-5-methylpyrrolo[2,1-f][1,2,4]triazine-6-carboxamideHuman5254
MAPK14 (p38a)MAPKCMGC5n65A2-phenyl-~{n}4-(2-thiophen-2-ylethyl)quinazoline-4,7-diamineHuman8525
MAPK14 (p38a)MAPKCMGC4dljA2-phenyl-n~4~-(2-phenylethyl)quinazoline-4,7-diamineHuman5242
MAPK14 (p38a)MAPKCMGC5n63A-Human8526
MAPK14 (p38a)MAPKCMGC3gcpAB4-[5-(4-fluoro-phenyl)-2-(4-methanesulfinyl-phenyl)-3h-imidazol-4-yl]-pyridineHuman5157
MAPK14 (p38a)MAPKCMGC3hv5BA1-[3-tert-butyl-1-(4-methylphenyl)-1h-pyrazol-5-yl]-3-{3-[(6-nitroquinolin-4-yl)amino]phenyl}ureaHuman5085
MAPK14 (p38a)MAPKCMGC1oz1AB3-(4-fluorophenyl)-2-pyridin-4-yl-1h-pyrrolo[3,2-b]pyridin-1-olHuman5261
MAPK14 (p38a)MAPKCMGC3zshAB2-(6-chloro-5-{[(2r,5s)-4-(4-fluorobenzyl)-2,5-dimethylpiperazin-1-yl]carbonyl}-1-methyl-1h-indol-3-yl)-n,n-dimethyl-2-oxoacetamideHuman5118
MAPK14 (p38a)MAPKCMGC6ohdAA3-(3-tert-butyl-2-oxo-2,3-dihydro-1h-imidazo[4,5-b]pyridin-6-yl)-4-methyl-n-(1,2-oxazol-3-yl)benzamideHuman11818
MAPK14 (p38a)MAPKCMGC3gcvAA1-{3-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5088
MAPK14 (p38a)MAPKCMGC5n64A-Human8527
MAPK14 (p38a)MAPKCMGC3gcqAA1-{4-[(6-aminoquinazolin-4-yl)amino]phenyl}-3-[3-tert-butyl-1-(3-methylphenyl)-1h-pyrazol-5-yl]ureaHuman5066
GSK3BGSKCMGC9x2qAB-Human15789
GSK3BGSKCMGC4acgA2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamideHuman681
GSK3BGSKCMGC9fr5A~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)furo[3,2-d]pyrimidine-2,4-diamineHuman15790
GSK3BGSKCMGC4ptgBB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman754
GSK3BGSKCMGC6hk4BB3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11427
GSK3BGSKCMGC1gngB-Human700
GSK3BGSKCMGC5f94BA2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6372
GSK3BGSKCMGC3sd0B3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dioneHuman673
GSK3BGSKCMGC4ptgAA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman735
GSK3BGSKCMGC8djdAB2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamideHuman14668
GSK3BGSKCMGC5kpkB(4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9731
GSK3BGSKCMGC3pupAruthenium octasporineHuman7207
GSK3BGSKCMGC6y9sAA~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12286
GSK3BGSKCMGC8djcAB(4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamideHuman14669
GSK3BGSKCMGC4achA3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamideHuman653
GSK3BGSKCMGC3gb2AB2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazoleHuman734
GSK3BGSKCMGC3zrlBA7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman718
GSK3BGSKCMGC3zrlBC7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman676
GSK3BGSKCMGC3f88AB5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman679
GSK3BGSKCMGC4j71AA(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman642
GSK3BGSKCMGC5hlpBA4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6646
GSK3BGSKCMGC1o9uA9-methyl-9h-purin-6-amineHuman708
GSK3BGSKCMGC4acdA3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamideHuman723
GSK3BGSKCMGC1q4lA2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acidHuman714
GSK3BGSKCMGC5hlpAB4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6648
GSK3BGSKCMGC4achB3-amino-n-(3-methoxypropyl)-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}pyrazine-2-carboxamideHuman702
GSK3BGSKCMGC9x2uAA-Human15791
GSK3BGSKCMGC7u33AA3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamideHuman14198
GSK3BGSKCMGC3i4bBn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHuman629
GSK3BGSKCMGC1j1cAadenosine-5'-diphosphateHuman696
GSK3BGSKCMGC3m1sBBruthenium pyridocarbazoleHuman7208
GSK3BGSKCMGC7z1gA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman14662
GSK3BGSKCMGC3f7zBC2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman686
GSK3BGSKCMGC1pyxBphosphoaminophosphonic acid-adenylate esterHuman663
GSK3BGSKCMGC3zrkAC2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman697
GSK3BGSKCMGC4pteAAn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman716
GSK3BGSKCMGC1r0eAB3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman672
GSK3BGSKCMGC3pupBruthenium octasporineHuman7211
GSK3BGSKCMGC5t31A(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9565
GSK3BGSKCMGC5k5nB5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamideHuman7410
GSK3BGSKCMGC6gjoA(3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-oneHuman10974
GSK3BGSKCMGC3l1sB(4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-oneHuman713
GSK3BGSKCMGC1q41A(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman628
GSK3BGSKCMGC6v6lAB1-(6-((2-((6-amino-5-nitropyridin-2-yl)amino)ethyl)amino)-2-(2,4-dichlorophenyl)pyridin-3-yl)-4-methylpiperazin-2-oneHuman11912
GSK3BGSKCMGC9fr8A~{n}4-(3-cyclobutyl-1~{h}-pyrazol-5-yl)-~{n}2-(pyridin-3-ylmethyl)thieno[3,2-d]pyrimidine-2,4-diamineHuman15793
GSK3BGSKCMGC4nm0ABadenosine-5'-diphosphateHuman671
GSK3BGSKCMGC4ptcAA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman664
GSK3BGSKCMGC7sxhAB(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14784
GSK3BGSKCMGC3gb2AA2-methyl-5-(3-{4-[(s)-methylsulfinyl]phenyl}-1-benzofuran-5-yl)-1,3,4-oxadiazoleHuman727
GSK3BGSKCMGC4nm3ABadenosine-5'-diphosphateHuman640
GSK3BGSKCMGC4accB3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman669
GSK3BGSKCMGC3zdiA3,6-diamino-4-(2-chlorophenyl)thieno[2,3-b]pyridine-2,5-dicarbonitrileHuman748
GSK3BGSKCMGC4nm5AAadenosine-5'-diphosphateHuman755
GSK3BGSKCMGC5hlnAchir99021Human6649
GSK3BGSKCMGC7b6fAA3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrileHuman13069
GSK3BGSKCMGC7sxjAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14785
GSK3BGSKCMGC3sayAB(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman661
GSK3BGSKCMGC6hk4AA3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11429
GSK3BGSKCMGC4j71BA(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman641
GSK3BGSKCMGC6y9rAA~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamideHuman12287
GSK3BGSKCMGC4pteBAn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman722
GSK3BGSKCMGC6hk4AB3-azanyl-6-(4-morpholin-4-ylsulfonylphenyl)-~{n}-pyridin-3-yl-pyrazine-2-carboxamideHuman11423
GSK3BGSKCMGC5k5nA5-(3-chloranyl-4-methoxy-phenyl)-~{n}-[3-(1,2,4-triazol-1-yl)propyl]-1,3-oxazole-4-carboxamideHuman7411
GSK3BGSKCMGC2jldBAruthenium pyridocarbazoleHuman7205
GSK3BGSKCMGC2jldABruthenium pyridocarbazoleHuman7214
GSK3BGSKCMGC6h0uA(2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamideHuman11049
GSK3BGSKCMGC3sayAA(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman738
GSK3BGSKCMGC3f88AA5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman741
GSK3BGSKCMGC8av1AA2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14706
GSK3BGSKCMGC8auzAA8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14707
GSK3BGSKCMGC3zrlAA7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman712
GSK3BGSKCMGC5hlpAA4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6647
GSK3BGSKCMGC5kplBA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9728
GSK3BGSKCMGC8djeAA(4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamideHuman14670
GSK3BGSKCMGC5oy4A~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamideHuman8621
GSK3BGSKCMGC3zrmBB7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman652
GSK3BGSKCMGC5f95A2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamideHuman6373
GSK3BGSKCMGC2jldAAruthenium pyridocarbazoleHuman7213
GSK3BGSKCMGC4afjBA5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman678
GSK3BGSKCMGC3zrmAC7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman724
GSK3BGSKCMGC4b7tA(5z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-methyl-2-(propan-2-ylamino)imidazol-4-oneHuman732
GSK3BGSKCMGC3zrkAA2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman675
GSK3BGSKCMGC1uv5A6-bromoindirubin-3'-oximeHuman759
GSK3BGSKCMGC4j71AB(2r)-2-methyl-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman690
GSK3BGSKCMGC1q5kAn-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)ureaHuman680
GSK3BGSKCMGC8auzAB8-morpholin-4-yl-2-pyridin-3-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14708
GSK3BGSKCMGC5kpmB(4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9734
GSK3BGSKCMGC3zrlAB7-bromo-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman725
GSK3BGSKCMGC6hk3BA3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11422
GSK3BGSKCMGC7u31AA5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amineHuman14199
GSK3BGSKCMGC6hk7A3-azanyl-~{n}-(2-methoxyethyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11428
GSK3BGSKCMGC4ptcBA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman747
GSK3BGSKCMGC4pteABn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman717
GSK3BGSKCMGC3zrkBA2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman637
GSK3BGSKCMGC1r0eBA3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman687
GSK3BGSKCMGC1h8fA-Human745
GSK3BGSKCMGC6y9sBB~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12288
GSK3BGSKCMGC5f94BB2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6371
GSK3BGSKCMGC4ptgBA2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman740
GSK3BGSKCMGC3l1sA(4e)-4-[(4-chlorophenyl)hydrazono]-5-(3,4-dimethoxyphenyl)-2,4-dihydro-3h-pyrazol-3-oneHuman757
GSK3BGSKCMGC7u33AB3-[2-amino-5-(4-fluorophenyl)pyrimidin-4-yl]-n,n-dimethylazetidine-1-sulfonamideHuman14200
GSK3BGSKCMGC5f94AB2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6369
GSK3BGSKCMGC6y9rAB~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-5-(5-propan-2-yloxypyridin-3-yl)-1~{h}-indazole-3-carboxamideHuman12289
GSK3BGSKCMGC4afjAA5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman632
GSK3BGSKCMGC3f7zAC2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman685
GSK3BGSKCMGC4acdB3-amino-6-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-pyridin-3-ylpyrazine-2-carboxamideHuman692
GSK3BGSKCMGC3zrmAA7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman751
GSK3BGSKCMGC4afjAC5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman742
GSK3BGSKCMGC1q41B(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman658
GSK3BGSKCMGC1j1bBphosphoaminophosphonic acid-adenylate esterHuman657
GSK3BGSKCMGC1gngA-Human665
GSK3BGSKCMGC6hk3AA3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11425
GSK3BGSKCMGC4j1rC(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman688
GSK3BGSKCMGC4afjBC5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman711
GSK3BGSKCMGC4ditAn-(pyridin-3-yl)-2-(thiophen-3-yl)-3h-imidazo[4,5-b]pyridine-7-carboxamideHuman689
GSK3BGSKCMGC7u31AB5-(4-fluorophenyl)-4-[1-(methanesulfonyl)azetidin-3-yl]pyrimidin-2-amineHuman14201
GSK3BGSKCMGC3m1sBAruthenium pyridocarbazoleHuman7210
GSK3BGSKCMGC4afjAB5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman683
GSK3BGSKCMGC1h8fB-Human666
GSK3BGSKCMGC4acgB2-amino-5-{4-[(4-methylpiperazin-1-yl)sulfonyl]phenyl}-n-[4-(pyrrolidin-1-ylmethyl)pyridin-3-yl]pyridine-3-carboxamideHuman721
GSK3BGSKCMGC4ptcBB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman758
GSK3BGSKCMGC4nm7ABadenosine-5'-diphosphateHuman684
GSK3BGSKCMGC3zrmAB7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman648
GSK3BGSKCMGC1q3wA9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-oneHuman635
GSK3BGSKCMGC5f94AA2-[(cyclopropylcarbonyl)amino]-n-(4-methoxypyridin-3-yl)pyridine-4-carboxamideHuman6374
GSK3BGSKCMGC4nm5ABadenosine-5'-diphosphateHuman694
GSK3BGSKCMGC5hlpBB4-(2-methoxyphenyl)-3,7,7-trimethyl-1,6,7,8-tetrahydro-5h-pyrazolo[3,4-b]quinolin-5-oneHuman6645
GSK3BGSKCMGC3sayBB(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman710
GSK3BGSKCMGC8av1AB2-pyridin-3-yl-8-thiomorpholin-4-yl-[1,3]oxazolo[5,4-f]quinoxalineHuman14709
GSK3BGSKCMGC1q5kBn-(4-methoxybenzyl)-n'-(5-nitro-1,3-thiazol-2-yl)ureaHuman651
GSK3BGSKCMGC3zrkBC2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman731
GSK3BGSKCMGC5kpkA(4~{s})-3-cyclopropyl-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9735
GSK3BGSKCMGC6hk3AB3-azanyl-~{n}-(2-methoxyphenyl)-6-[4-(4-methylpiperazin-1-yl)sulfonylphenyl]pyrazine-2-carboxamideHuman11426
GSK3BGSKCMGC5oy4B~{n}-[6-[3,4-bis(oxidanyl)phenyl]-1~{h}-pyrazolo[3,4-b]pyridin-3-yl]ethanamideHuman8622
GSK3BGSKCMGC2ow3Abis-(indole)maleimide pyridinophaneHuman698
GSK3BGSKCMGC1pyxAphosphoaminophosphonic acid-adenylate esterHuman645
GSK3BGSKCMGC5kplAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9730
GSK3BGSKCMGC3sd0A3-(5-fluoro-6-iodo-1-methyl-1h-indol-3-yl)-4-(7-methoxy-1-benzofuran-3-yl)-1h-pyrrole-2,5-dioneHuman720
GSK3BGSKCMGC1q3wB9-nitro-5,12-dihydro-7h-benzo[2,3]azepino[4,5-b]indol-6-oneHuman693
GSK3BGSKCMGC3f7zAB2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman647
GSK3BGSKCMGC3f7zBA2-(1,3-benzodioxol-5-yl)-5-[(3-fluoro-4-methoxybenzyl)sulfanyl]-1,3,4-oxadiazoleHuman749
GSK3BGSKCMGC6gjoB(3~{z})-5-ethanoyl-3-[[(1-methylpiperidin-4-yl)amino]-phenyl-methylidene]-1~{h}-indol-2-oneHuman10973
GSK3BGSKCMGC4ptgAB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-methoxypyrimidine-5-carboxamideHuman634
GSK3BGSKCMGC3du8B(7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman737
GSK3BGSKCMGC1i09B-Human638
GSK3BGSKCMGC6b8jABchir99021Human8659
GSK3BGSKCMGC4iq6A6-chloro-n-cyclohexyl-4-(1h-pyrrolo[2,3-b]pyridin-3-yl)pyridin-2-amineHuman728
GSK3BGSKCMGC7u2zAB(3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHuman14202
GSK3BGSKCMGC4nm0AAadenosine-5'-diphosphateHuman715
GSK3BGSKCMGC4j1rB(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman656
GSK3BGSKCMGC3du8A(7s)-2-(2-aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4h-pyrrolo[3,2-c]pyridin-4-oneHuman701
GSK3BGSKCMGC7u2zAA(3r)-1-[3-(2-fluorophenyl)propanoyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHuman14203
GSK3BGSKCMGC5hlnBchir99021Human6650
GSK3BGSKCMGC4pteBBn-[4-(isoquinolin-7-yl)pyridin-2-yl]cyclopropanecarboxamideHuman667
GSK3BGSKCMGC2ow3Bbis-(indole)maleimide pyridinophaneHuman649
GSK3BGSKCMGC1q4lB2-chloro-5-[4-(3-chloro-phenyl)-2,5-dioxo-2,5-dihydro-1h-pyrrol-3-ylamino]-benzoic acidHuman655
GSK3BGSKCMGC8djeAB(4s)-3-[(cyclopropylmethyl)amino]-n-(4-phenylpyridin-3-yl)imidazo[1,2-b]pyridazine-8-carboxamideHuman14671
GSK3BGSKCMGC3sayBA(3z)-n,n-diethyl-3-[(3e)-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-ylidene]-2-oxo-2,3-dihydro-1h-indole-5-sulfonamideHuman682
GSK3BGSKCMGC1j1bAphosphoaminophosphonic acid-adenylate esterHuman707
GSK3BGSKCMGC6gn1A~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamideHuman9997
GSK3BGSKCMGC4nm7AAadenosine-5'-diphosphateHuman695
GSK3BGSKCMGC5kplBB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9733
GSK3BGSKCMGC4j1rA(2r)-2-(1h-indol-3-ylmethyl)-1,4-dihydropyrido[2,3-b]pyrazin-3(2h)-oneHuman709
GSK3BGSKCMGC2o5kA2-(2,4-dichloro-phenyl)-7-hydroxy-1h-benzoimidazole-4-carboxylic acid [2-(4-methanesulfonylamino-phenyl)-ethyl]-amideHuman633
GSK3BGSKCMGC7sxjAB(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman14786
GSK3BGSKCMGC6y9sAB~{n}-(oxan-4-ylmethyl)-6-(5-propan-2-yloxypyridin-3-yl)imidazo[1,5-a]pyridine-3-carboxamideHuman12290
GSK3BGSKCMGC3q3bA4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHuman660
GSK3BGSKCMGC6b8jAAchir99021Human8658
GSK3BGSKCMGC7z1fA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman14663
GSK3BGSKCMGC3zrmBC7-(4-hydroxyphenyl)-2-pyridin-4-yl-5h-thieno[3,2-c]pyridin-4-oneHuman706
GSK3BGSKCMGC6tcuAB5-[2,3-bis(fluoranyl)phenyl]-~{n}-[[1-(2-methoxyethyl)piperidin-4-yl]methyl]-1~{h}-indazole-3-carboxamideHuman12781
GSK3BGSKCMGC7u36A(3s)-1-[(2-fluorophenoxy)acetyl]-n-(pyridin-2-yl)pyrrolidine-3-carboxamideHuman14204
GSK3BGSKCMGC5kplAA(4~{s})-4-ethyl-7,7-dimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9729
GSK3BGSKCMGC5f95B2-[(cyclopropylcarbonyl)amino]-n-(4-phenylpyridin-3-yl)pyridine-4-carboxamideHuman6370
GSK3BGSKCMGC7sxhAA(4s,5r,8r)-4-ethyl-8-fluoro-4-[3-(3-fluoro-5-methoxypyridin-4-yl)phenyl]-7,7-dimethyl-4,5,6,7,8,9-hexahydro-2h-pyrazolo[3,4-b]quinolin-5-olHuman14787
GSK3BGSKCMGC8ff8A2-(4-cyanoanilino)-n-(4-phenylpyridin-3-yl)pyrimidine-4-carboxamideHuman14763
GSK3BGSKCMGC3zrkBB2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman662
GSK3BGSKCMGC3zrkAB2-(4-pyridinyl)furo[3,2-c]pyridin-4(5h)-oneHuman644
GSK3BGSKCMGC3f88BB5-[1-(4-methoxyphenyl)-1h-benzimidazol-6-yl]-1,3,4-oxadiazole-2(3h)-thioneHuman756
GSK3BGSKCMGC7b6fAB3-[(3~{s})-3-[(7-chloranyl-9~{h}-pyrimido[4,5-b]indol-4-yl)-methyl-amino]piperidin-1-yl]propanenitrileHuman13070
GSK3BGSKCMGC4accA3-amino-6-(4-{[2-(dimethylamino)ethyl]sulfamoyl}phenyl)-n-pyridin-3-ylpyrazine-2-carboxamideHuman704
GSK3BGSKCMGC6gn1B~{n}-[(~{e})-(6-bromanylimidazo[1,2-a]pyridin-3-yl)methylideneamino]-~{n},2-dimethyl-5-nitro-benzenesulfonamideHuman9996
GSK3BGSKCMGC2jldBBruthenium pyridocarbazoleHuman7209
GSK3BGSKCMGC8djcAA(4s)-n-{4-[(2s)-2-methylmorpholin-4-yl]pyridin-3-yl}-2-phenylimidazo[1,2-b]pyridazine-8-carboxamideHuman14672
GSK3BGSKCMGC3q3bB4-(4-hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(5h)-oneHuman674
GSK3BGSKCMGC3m1sAAruthenium pyridocarbazoleHuman7212
GSK3BGSKCMGC3i4bAn-[(1s)-2-hydroxy-1-phenylethyl]-4-[5-methyl-2-(phenylamino)pyrimidin-4-yl]-1h-pyrrole-2-carboxamideHuman646
GSK3BGSKCMGC4nm3AAadenosine-5'-diphosphateHuman730
GSK3BGSKCMGC3m1sABruthenium pyridocarbazoleHuman7206
GSK3BGSKCMGC4ptcAB2-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}-4-oxo-4h-1lambda~4~,3-thiazole-5-carboxamideHuman659
GSK3BGSKCMGC1i09A-Human630
GSK3BGSKCMGC5kpmA(4~{s})-3-(2,2-dimethylpropyl)-4,7,7-trimethyl-4-phenyl-2,6,8,9-tetrahydropyrazolo[3,4-b]quinolin-5-oneHuman9732
GSK3BGSKCMGC1r0eBB3-[3-(2,3-dihydroxy-propylamino)-phenyl]-4-(5-fluoro-1-methyl-1h-indol-3-yl)-pyrrole-2,5-dioneHuman639
GSK3BGSKCMGC8djdAA2-[(cyclopropanecarbonyl)amino]-n-(5-phenylpyridin-3-yl)pyridine-4-carboxamideHuman14673
SRPK2SRPKCMGC5myvAB5-methyl-~{n}-[2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)phenyl]furan-2-carboxamideHuman7575
CLK1CLKCMGC5j1vApyrido[3,4-g]quinazoline-2,10-diamineHuman6582
MAPK1 (Erk2)MAPKCMGC6qalAB1,1-bis(oxidanylidene)thietan-3-olHuman10981
MAPK1 (Erk2)MAPKCMGC6g91AA5-chloranyl-~{n}-(oxan-4-yl)pyrimidin-2-amineHuman9965
MAPK1 (Erk2)MAPKCMGC4fmqABphosphoaminophosphonic acid-adenylate esterHuman2619
MAPK1 (Erk2)MAPKCMGC4zzoABn-[2-[[5-chloranyl-2-(oxan-4-ylamino)pyrimidin-4-yl]amino]phenyl]propanamideHuman2606
MAPK1 (Erk2)MAPKCMGC6qa4AB1~{h}-pyridin-2-oneHuman11351
MAPK1 (Erk2)MAPKCMGC5v60AAphosphomethylphosphonic acid adenylate esterHuman8261
MAPK1 (Erk2)MAPKCMGC6gdqAB4-[5-chloranyl-2-(propan-2-ylamino)pyridin-4-yl]-~{n}-[(1~{s})-1-(3-chlorophenyl)-2-oxidanyl-ethyl]-1~{h}-pyrrole-2-carboxamideHuman9973
MAPK1 (Erk2)MAPKCMGC6gjdAAcyclooctyl ~{n}-[3-[[4-[5-[[(3~{r})-1-[2-oxidanylidene-2-[4-(4-pyrimidin-2-ylphenyl)piperazin-1-yl]ethyl]pyrrolidin-3-yl]carbonylamino]-1~{h}-indazol-3-yl]pyridin-2-yl]carbonylamino]propyl]carbamateHuman10829
MAPK1 (Erk2)MAPKCMGC4fv0ABn-cyclohexyl-4-[3-(4-fluorophenyl)-1h-pyrazol-4-yl]pyridin-2-amineHuman2599
CSNK2A2 (CK2a2)CK2CMGC8q77AB(2~{s})-2-[[(2~{s})-2-[[(2~{s})-2-[12-[[4-[[5-(4-carboxyphenyl)-1,3-thiazol-2-yl]amino]-4-oxidanylidene-butanoyl]-(2-hydroxy-2-oxoethyl)amino]dodecanoylamino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]-4-oxidanyl-4-oxidanylidene-butanoyl]amino]butanedioic acidHuman15022
CSNK2A2 (CK2a2)CK2CMGC5ooiBB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9444
SRPK1SRPKCMGC1wakA-Human120
MAPK14 (p38a)MAPKCMGC3od6X-Human5134
MAPK14 (p38a)MAPKCMGC5n68A-Human8522
MAPK14 (p38a)MAPKCMGC3zsiAA5-(2,6-dichlorophenyl)-2-[(2,4-difluorophenyl)sulfanyl]-6h-pyrimido[1,6-b]pyridazin-6-oneHuman5056
GSK3BGSKCMGC6h0uB(2~{r})-3-[7-azanyl-5-(cyclohexylamino)-[1,2,4]triazolo[1,5-a][1,3,5]triazin-2-yl]-2-cyano-propanamideHuman11050
GSK3BGSKCMGC4afjBB5-(4-methoxyphenyl)-n-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamideHuman726
CDK12 (CRK7)CDKCMGC8busB1,3-dimethyl-5-[[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]methyl]pyrazole-4-sulfonamideHuman14908
CDK12 (CRK7)CDKCMGC8bucB2-(1~{h}-benzimidazol-2-ylsulfanyl)-~{n}-(5-chloranylpyridin-2-yl)ethanamideHuman14909
CDK12 (CRK7)CDKCMGC8bu4B(2~{r})-2-[[6-[[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]methylamino]-9-(1-methylpyrazol-4-yl)purin-2-yl]amino]butan-1-olHuman14910
CDK12 (CRK7)CDKCMGC8bulB(2~{r})-2-[[6-(3-phenylpropylamino)-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14911
CDK12 (CRK7)CDKCMGC6td3E(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman12369
CDK12 (CRK7)CDKCMGC8bueB~{n}-(1~{h}-benzimidazol-2-yl)-1-(2-methoxy-5-methyl-phenyl)-5-oxidanylidene-pyrrolidine-3-carboxamideHuman14912
CDK12 (CRK7)CDKCMGC8bu7B-Human14913
CDK12 (CRK7)CDKCMGC8bu9Br-roscovitineHuman14914
CDK12 (CRK7)CDKCMGC5acbDn-[4-[(3r)-3-[[5-chloranyl-4-(1h-indol-3-yl)pyrimidin-2-yl]amino]piperidin-1-yl]carbonylphenyl]-4-(dimethylamino)butanamideHuman6702
CDK12 (CRK7)CDKCMGC8burBA~{n}-[2-(2-methoxyphenyl)ethyl]-2-[[9-propan-2-yl-6-[(4-pyridin-2-ylphenyl)methylamino]purin-2-yl]amino]ethanamideHuman14915
CDK12 (CRK7)CDKCMGC8bunB(2~{r})-2-[[6-[(4-phenylphenyl)methylamino]-9-propan-2-yl-purin-2-yl]amino]butan-1-olHuman14916
CDK12 (CRK7)CDKCMGC4nstAadenosine-5'-diphosphateHuman4852
CDK6CDKCMGC1g3nE-Human2805
CDK6CDKCMGC3nupA4-[3-(1-methylethyl)-1h-pyrazol-4-yl]-n-(1-methylpiperidin-4-yl)pyrimidin-2-amineHuman2797
CDK6CDKCMGC4tthB9-cyclopentyl-n-(5-piperazin-1-ylpyridin-2-yl)pyrido[4,5]pyrrolo[1,2-d]pyrimidin-2-amineHuman2803
CDK6CDKCMGC5l2iA6-acetyl-8-cyclopentyl-5-methyl-2-[(5-piperazin-1-ylpyridin-2-yl)amino]pyrido[2,3-d]pyrimidin-7(8h)-oneHuman6991
CDK2CDKCMGC2r3iAA5-(2-fluorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4135
CDK2CDKCMGC3r7uAB2-{[4-(aminomethyl)benzyl]amino}-5-nitrobenzamideHuman4023
CDK2CDKCMGC1h08AA(2r)-1-{4-[(4-anilino-5-bromopyrimidin-2-yl)amino]phenoxy}-3-(dimethylamino)propan-2-olHuman4220
CDK2CDKCMGC2whbCB-Human4352
CDK2CDKCMGC4eoiCA(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4522
CDK2CDKCMGC1ckpAApurvalanol bHuman4066
CDK2CDKCMGC2uzdC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}benzenesulfonamideHuman3900
CDK2CDKCMGC4fkjABn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-[4-(2-pyrrolidin-1-ylethoxy)phenyl]acetamideHuman4164
CDK2CDKCMGC1pxpAB-Human3943
CDK2CDKCMGC2wfyAB-Human4426
CDK2CDKCMGC2wevAC[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4007
CDK2CDKCMGC2b53A6-(3-aminophenyl)-n-(tert-butyl)-2-(trifluoromethyl)quinazolin-4-amineHuman3875
CDK2CDKCMGC4fkpAC3-{[4-([amino(imino)methyl]aminosulfonyl)anilino]methylene}-2-oxo-2,3-dihydro-1h-indoleHuman4468
CDK2CDKCMGC4d1zA(4s)-2-(8-hydroxyquinolin-2-yl)-4,5-dihydro-1,3-thiazole-4-carboxylic acidHuman4486
CDK2CDKCMGC1h0wAA1-amino-6-cyclohex-3-enylmethyloxypurineHuman3987
CDK2CDKCMGC1oirA1-(dimethylamino)-3-(4-{{4-(2-methylimidazo[1,2-a]pyridin-3-yl)pyrimidin-2-yl]amino}phenoxy)propan-2-olHuman4389
CDK2CDKCMGC3ezrA3-methoxy-4-{3-[4-(4-methylpiperazin-1-yl)-1h-benzimidazol-2-yl]-1h-indazol-6-yl}anilineHuman4475
CDK2CDKCMGC5l2wA3-[({3-ethyl-5-[(2s)-2-(2-hydroxyethyl)piperidin-1-yl]pyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1-hydroxypyridiniumHuman6993
CDK2CDKCMGC1h1rCA6-cyclohexylmethoxy-2-(3'-chloroanilino) purineHuman3920
CDK2CDKCMGC3qqfAB5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4287
CDK2CDKCMGC6q3cAB4-bromo-1h-pyrazoleHuman11203
CDK2CDKCMGC5ieyAB4-[(4-{[(2r,3r)-3-hydroxybutan-2-yl]amino}pyrimidin-2-yl)amino]benzene-1-sulfonamideHuman6573
CDK2CDKCMGC4nj3AB6-(3-chlorophenyl)-2-{[(2s)-3-(4-hydroxyphenyl)-1-methoxy-1-oxopropan-2-yl]carbamoyl}quinoline-4-carboxylic acidHuman4366
CDK2CDKCMGC9glaAB7-dimethylphosphoryl-3-[2-[[(3~{s})-6,6-dimethylpiperidin-3-yl]amino]-5-(trifluoromethyl)pyrimidin-4-yl]-1~{h}-indole-6-carbonitrileHuman15921
CDK2CDKCMGC2iw8CAo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman4294
CDK2CDKCMGC6sg4CB-Human13245
CDK2CDKCMGC2vtlAn-phenyl-1h-pyrazole-3-carboxamideHuman3870
CDK2CDKCMGC4cfwCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylbenzenesulfonamideHuman4508
CDK2CDKCMGC1w98A-Human4013
CDK2CDKCMGC7vduAA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14136
CDK2CDKCMGC9esnAA4-bromo-1-(2-hydroxyethyl)pyridin-2(1h)-oneHuman15922
CDK2CDKCMGC2r3oAB(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4354
CDK2CDKCMGC2vtaA1h-indazoleHuman4118
CDK2CDKCMGC4fkoAA2-chloro-n~4~-[4-(2,4-dimethyl-1,3-thiazol-5-yl)pyrimidin-2-yl]-n~1~,n~1~-dimethylbenzene-1,4-diamineHuman4449
CDK2CDKCMGC3qtrAA[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman3874
CDK2CDKCMGC4bckCA3-[[5-cyano-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidin-2-yl]amino]benzenesulfonamideHuman4268
CDK2CDKCMGC3ej1An-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amineHuman4168
CDK2CDKCMGC6q4gAA2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHuman11214
CDK2CDKCMGC2uzlC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]furan-2-yl}-2-(trifluoromethyl)benzenesulfonamideHuman4106
CDK2CDKCMGC1dm2AA4-(5-amino-4-oxo-4h-pyrazol-3-yl)-2-bromo-4,5,6,7-tetrahydro-3ah-pyrrolo[2,3-c]azepin-8-oneHuman4104
CDK2CDKCMGC3rpyAA4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4261
CDK2CDKCMGC3royAB4-(hexylamino)-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4239
CDK2CDKCMGC3py0AB(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman3869
CDK2CDKCMGC3ddqCBr-roscovitineHuman4289
CDK2CDKCMGC4cfnAA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4285
CDK2CDKCMGC4eoqABadenosine-5'-triphosphateHuman4230
CDK2CDKCMGC6q4bAA5-bromanylpyrimidineHuman11198
CDK2CDKCMGC2a0cXB2-{[(2-{[(1r)-1-(hydroxymethyl)propyl]amino}-9-isopropyl-9h-purin-6-yl)amino]methyl}phenolHuman3868
CDK2CDKCMGC9esoAA-Human15926
CDK2CDKCMGC4lynA(2s)-n-(5-{[(5-tert-butyl-1,3-oxazol-2-yl)methyl]sulfanyl}-1,3-thiazol-2-yl)-2-phenylpropanamideHuman4550
CDK2CDKCMGC3qtrAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](phenyl)methanoneHuman4243
CDK2CDKCMGC2r3fAA5-(2,3-dichlorophenyl)-n-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amineHuman4175
CDK2CDKCMGC1oiuAA3-(6-cyclohexylmethoxy-9h-purin-2-ylamino)-benzenesulfonamideHuman4110
CDK2CDKCMGC6rijAB4-[[[5-nitroso-2-[[(2~{r})-1-oxidanylbutan-2-yl]amino]-6-(propan-2-ylamino)pyrimidin-4-yl]amino]methyl]phenolHuman12624
CDK2CDKCMGC4ek4AA4-bromo-n-(5-methyl-1h-pyrazol-3-yl)benzamideHuman4212
CDK2CDKCMGC3rpyAB4-amino-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4519
CDK2CDKCMGC5osjAA-Human9743
CDK2CDKCMGC5cyiAB6-(cyclohexylmethoxy)-n-[4-(ethylsulfonyl)phenyl]-9h-purin-2-amineHuman6054
CDK2CDKCMGC1jstAadenosine-5'-triphosphateHuman4455
CDK2CDKCMGC4fkgAA4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acidHuman4020
CDK2CDKCMGC2w17AAn-(4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]carbonyl}phenyl)-5-fluoro-4-[2-methyl-1-(1-methylethyl)-1h-imidazol-5-yl]pyrimidin-2-amineHuman3968
CDK2CDKCMGC2r64An-[5-(1,1-dioxidoisothiazolidin-2-yl)-1h-indazol-3-yl]-2-(4-piperidin-1-ylphenyl)acetamideHuman4425
CDK2CDKCMGC6gufAn2-[(1r,2s)-2-aminocyclohexyl]-n6-(3-chlorophenyl)-9-ethyl-9h-purine-2,6-diamineHuman10770
CDK2CDKCMGC2r3oAA(5-phenyl-7-(pyridin-3-ylmethylamino)pyrazolo[1,5-a]pyrimidin-3-yl)methanolHuman4147
CDK2CDKCMGC13gkAA4-[(1m)-1-{4-[(azetidin-1-yl)methyl]-2-chlorophenyl}-1h-imidazol-4-yl]-n-[1-(methanesulfonyl)piperidin-4-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman15927
CDK2CDKCMGC1aq1AstaurosporineHuman4267
CDK2CDKCMGC2vtrAB5-chloro-7-[(1-methylethyl)amino]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman3907
CDK2CDKCMGC8ypwAmethyl 3-[4-[3-[[3-[(1-ethylsulfonylpiperidin-4-yl)carbamoyl]-1~{h}-pyrazol-4-yl]carbamoyl]-2,4-bis(fluoranyl)phenyl]piperidin-1-yl]-3-oxidanylidene-propanoateHuman15928
CDK2CDKCMGC3my5CB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman4003
CDK2CDKCMGC2uzbCC4-{5-[(z)-(2-imino-4-oxo-1,3-thiazolidin-5-ylidene)methyl]-2-furyl}-n-methylbenzenesulfonamideHuman4045
CDK2CDKCMGC1urwAA2-[4-(n-(3-dimethylaminopropyl)sulphamoyl)anilino]-Human4054
CDK2CDKCMGC1h28A-Human4169
CDK2CDKCMGC9espAA4-bromo-1-(2-methoxyethyl)-1h-pyrazoleHuman15929
CDK2CDKCMGC5if1AB-Human6569
CDK2CDKCMGC2bkzC1-[4-(aminosulfonyl)phenyl]-1,6-dihydropyrazolo[3,4-e]indazole-3-carboxamideHuman4555
CDK2CDKCMGC1r78AB4-((3r,4s,5r)-4-amino-3,5-dihydroxy-hex-1-ynyl)-5-fluoro-3-[1-(3-methoxy-1h-pyrrol-2-yl)-meth-(z)-ylidene]-1,3-dihydro-indol-2-oneHuman4249
CDK2CDKCMGC2wevAA[4-(2-amino-4-methyl-thiazol-5-yl)-pyrimidin-2-yl]-(3-nitro-phenyl)-amineHuman4067
CDK2CDKCMGC3rkbAA[4-amino-2-(cyclohexylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4460
CDK2CDKCMGC4fkgAB4-[(5-cyclopropyl-1h-pyrazol-3-yl)carbamoyl]benzoic acidHuman4559
CDK2CDKCMGC3unjA4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acidHuman4498
CDK2CDKCMGC4ez3A4-[(e)-(6-hydroxy-2-oxo-1,2-dihydropyridin-3-yl)diazenyl]benzenesulfonamideHuman4551
CDK2CDKCMGC4bcmCA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman4227
CDK2CDKCMGC6q49AA-Human11185
CDK2CDKCMGC5k4jAB1-[(1~{s})-1-(4-chloranyl-3-fluoranyl-phenyl)-2-oxidanyl-ethyl]-4-[2-[(2-methylpyrazol-3-yl)amino]pyrimidin-4-yl]pyridin-2-oneHuman6750
CDK2CDKCMGC1ykrA4-{[6-(2,6-dichlorobenzoyl)imidazo[1,2-a]pyridin-2-yl]amino}benzenesulfonamideHuman4578
CDK2CDKCMGC6q4kAB-Human11186
CDK2CDKCMGC2i40CB5-[5,6-bis(methyloxy)-1h-benzimidazol-1-yl]-3-{[1-(2-chlorophenyl)ethyl]oxy}-2-thiophenecarboxamideHuman4043
CDK2CDKCMGC1ke8A4-{[(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}-n-(1,3-thiazol-2-yl)benzenesulfonamideHuman4048
CDK2CDKCMGC2cchCBadenosine-5'-triphosphateHuman4000
CDK2CDKCMGC2wihCn,1,4,4-tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1h-pyrazolo[4,3-h]quinazoline-3-carboxamideHuman4119
CDK2CDKCMGC2c5vCB4-(2,4-dimethyl-1,3-thiazol-5-yl)-n-[4-(trifluoromethyl)phenyl]pyrimidin-2-amineHuman4209
CDK2CDKCMGC2r3qAC3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman3976
CDK2CDKCMGC3r83AB4-(4-aminopiperidin-1-yl)-2-{[(2-aminopyrimidin-5-yl)methyl]amino}-5-nitrobenzamideHuman4543
CDK2CDKCMGC3r7vAB5-nitro-2-[(pyridin-2-ylmethyl)amino]benzamideHuman4183
CDK2CDKCMGC4cfxCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]benzenesulfonamideHuman4257
CDK2CDKCMGC3r73AA4-[(3-aminopropyl)amino]-5-nitro-2-[(pyridin-3-ylmethyl)amino]benzamideHuman4187
CDK2CDKCMGC5mhqAA(2~{r},3~{s})-3-[[9-propan-2-yl-6-(pyridin-3-ylmethylamino)purin-2-yl]amino]pentan-2-olHuman9409
CDK2CDKCMGC9eszAA-Human15944
CDK2CDKCMGC4cfnCA6-(cyclohexylmethoxy)-8-(trifluoromethyl)-9h-purin-2-amineHuman4355
CDK2CDKCMGC3qzgAB2-(4,6-diamino-1,3,5-triazin-2-yl)-4-fluorophenolHuman4347
CDK2CDKCMGC2jgzA-Human4117
CDK2CDKCMGC7ackCB8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13452
CDK2CDKCMGC6jgmA4-{[6-(cyclohexylmethoxy)-7h-purin-2-yl]amino}-n,n-diethylbenzamideHuman12008
CDK2CDKCMGC4fx3AA(3z)-2-oxo-3-[2-(4-sulfamoylphenyl)hydrazinylidene]-2,3-dihydro-1h-indole-5-carboxylic acidHuman4518
CDK2CDKCMGC1gz8AA1-[(2-amino-6,9-dihydro-1h-purin-6-yl)oxy]-3-methyl-2-butanolHuman3981
CDK2CDKCMGC3qtqAA[4-amino-2-(prop-2-en-1-ylamino)-1,3-thiazol-5-yl](pyridin-3-yl)methanoneHuman4210
CDK2CDKCMGC2iw9ABo6-cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineHuman3955
CDK2CDKCMGC1oguCA4-{[4-amino-6-(cyclohexylmethoxy)-5-nitrosopyrimidin-2-yl]amino}benzamideHuman3964
CDK2CDKCMGC3qu0AB4-{[4-amino-5-(pyridin-3-ylcarbonyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4558
CDK2CDKCMGC7rweA5-nitro-2-[(3-phenylpropyl)amino]benzoic acidHuman14345
CDK2CDKCMGC9eszAB5-iodanylpyrimidineHuman15946
CDK2CDKCMGC1p5eA4,5,6,7-tetrabromobenzotriazoleHuman4090
CDK2CDKCMGC2r3qAB3-((3-bromo-5-o-tolylpyrazolo[1,5-a]pyrimidin-7-ylamino)methyl)pyridine 1-oxideHuman4459
CDK2CDKCMGC3rpvAB4-{[4-amino-5-(3-aminobenzoyl)-1,3-thiazol-2-yl]amino}benzenesulfonamideHuman4372
CDK2CDKCMGC4fktAAn-[2-(dimethylamino)ethyl]-4-{[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]amino}benzenesulfonamideHuman4548
CDK2CDKCMGC1finAadenosine-5'-triphosphateHuman4367
CDK2CDKCMGC3dogAB(2r)-2-{[4-(benzylamino)-8-(1-methylethyl)pyrazolo[1,5-a][1,3,5]triazin-2-yl]amino}butan-1-olHuman4365
CDK2CDKCMGC3ddpAA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6781
CDK2CDKCMGC1wccAA2-amino-6-chloropyrazineHuman4394
CDK2CDKCMGC6q48AB4-iodanyl-3~{h}-pyridin-2-oneHuman11218
CDK2CDKCMGC1oi9CB6-cyclohexylmethyloxy-2-(4'-hydroxyanilino)purineHuman4036
CDK2CDKCMGC7ackAB8-cyclohexyl-6~{h}-imidazo[1,2-c]pyrimidin-5-oneHuman13453
CDK2CDKCMGC13gkAB4-[(1m)-1-{4-[(azetidin-1-yl)methyl]-2-chlorophenyl}-1h-imidazol-4-yl]-n-[1-(methanesulfonyl)piperidin-4-yl]-5-(trifluoromethyl)pyrimidin-2-amineHuman15947
CDK2CDKCMGC1jvpP23-pyridin-4-yl-2,4-dihydroindeno[1,2-c]pyrazoleHuman4097
CDK2CDKCMGC4eooABadenosine-5'-triphosphateHuman4278
CDK2CDKCMGC3ddpCA(2r)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman6784
CDK2CDKCMGC11gvAB(1r,3s)-3-{3-[(1-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]-1h-pyrazol-5-yl}cyclopentyl bicyclo[1.1.1]pentan-1-ylcarbamateHuman15948
CDK2CDKCMGC6gueA4-(2-methyl-3-propan-2-yl-imidazol-4-yl)-~{n}-(4-methylsulfonylphenyl)pyrimidin-2-amineHuman10771
CDK2CDKCMGC6sg4AB-Human13247
CDK2CDKCMGC6gucC(3z)-3-(1h-imidazol-5-ylmethylene)-5-methoxy-1h-indol-2(3h)-oneHuman10766
CDK2CDKCMGC7e34A-Human13497
CDK2CDKCMGC2wpaAn-{6,6-dimethyl-5-[(1-methylpiperidin-4-yl)carbonyl]-1,4,5,6-tetrahydropyrrolo[3,4-c]pyrazol-3-yl}-3-methylbutanamideHuman4399
CDK2CDKCMGC1okvA-Human3921
CDK2CDKCMGC3qtsAB[4-amino-2-(phenylamino)-1,3-thiazol-5-yl](3-methoxyphenyl)methanoneHuman4564
CDK2CDKCMGC1hckAAadenosine-5'-triphosphateHuman3878
CDK2CDKCMGC6q4gAB2-[3-(2-azanyl-9~{h}-purin-6-yl)phenyl]ethanoic acidHuman11217
CDK2CDKCMGC3my5AC5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman3910
CDK2CDKCMGC6sg4CA-Human13248
CDK2CDKCMGC9eslAA4-bromanyl-1-(2-methoxyethyl)pyridin-2-oneHuman15950
CDK2CDKCMGC6q3cAC-Human11178
CDK2CDKCMGC4ii5CBadenosine-5'-diphosphateHuman4462
CDK2CDKCMGC6q4aAC5-iodanylpyrimidineHuman11216
CDK2CDKCMGC3qwjAA2-{[(2-aminopyrimidin-5-yl)methyl]amino}-4-chloro-5-nitrobenzamideHuman4265
CDK2CDKCMGC3r9oA4-amino-n-(3,5-difluorophenyl)-2-[(4-sulfamoylphenyl)amino]-1,3-thiazole-5-carboxamideHuman4279
CDK2CDKCMGC3qruAA(5s)-n-methyl-5-(2-methylbutan-2-yl)-4,5,6,7-tetrahydro-2h-indazole-3-carboxamideHuman4237
CDK2CDKCMGC1h0vAA5-{[(2-amino-9h-purin-6-yl)oxy]methyl}-2-pyrrolidinoneHuman4368
CDK2CDKCMGC4eonCB(5e)-5-(quinolin-6-ylmethylidene)-2-[(thiophen-2-ylmethyl)amino]-1,3-thiazol-4(5h)-oneHuman4192
CDK2CDKCMGC4ek3AB-Human4202
CDK2CDKCMGC4cfvCB3-[2-amino-6-(cyclohexylmethoxy)-7h-purin-8-yl]-2-methylphenolHuman3979
CDK2CDKCMGC1oiyCB4-(6-cyclohexylmethoxy-9h-purin-2-ylamino)--benzamideHuman4245
CDK2CDKCMGC6q48AA4-iodanyl-3~{h}-pyridin-2-oneHuman11192
CDK2CDKCMGC4bzdAA6-(benzimidazol-1-yl)-n-[5-[3-(dimethylamino)propoxy]pyridin-2-yl]pyrimidin-4-amineHuman3865
CDK2CDKCMGC1vywAn-(3-cyclopropyl-1h-pyrazol-5-yl)-2-(2-naphthyl)acetamideHuman3992
CDK2CDKCMGC1y91A4-[5-(trans-4-aminocyclohexylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-7-ylamino]-n,n-dimethylbenzenesulfonamideHuman4505
CDK2CDKCMGC7b5lL-Human13266
CDK8CDKCMGC4f7sAAn-(2-phenylethyl)quinazolin-4-amineHuman3850
CDK8CDKCMGC5hbeAB8-[3-chloranyl-5-[1-methyl-2,2-bis(oxidanylidene)-3~{h}-2,1-benzothiazol-5-yl]pyridin-4-yl]-1-oxa-3,8-diazaspiro[4.5]decan-2-oneHuman6386
CDKL2CDKLCMGC4bbmB4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diolHuman965
CDKL2CDKLCMGC4aaaAA5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman964
CDKL2CDKLCMGC4aaaAB5-amino-3-{[4-(aminosulfonyl)phenyl]amino}-n-(2,6-difluorophenyl)-1h-1,2,4-triazole-1-carbothioamideHuman962
CDKL2CDKLCMGC4bbmA4'-[5-[[3-[(cyclopropylamino)methyl]phenyl]amino]-1h-pyrazol-3-yl]-[1,1'-biphenyl]-2,4-diolHuman963
MAPK9 (JNK2)MAPKCMGC7n8tAAadenosine monophosphateHuman14241
MAPK9 (JNK2)MAPKCMGC3npcA1-(5-tert-butyl-2-p-tolyl-2h-pyrazol-3-yl)-3-[4-(2-morpholin-4-yl-ethoxy)-naphthalen-1-yl]-ureaHuman1235
MAPK9 (JNK2)MAPKCMGC3e7oBn-{3-[5-(1h-1,2,4-triazol-3-yl)-1h-indazol-3-yl]phenyl}furan-2-carboxamideHuman1236
MAPK9 (JNK2)MAPKCMGC7cmlAA-Human12707
CDK9CDKCMGC3tniA-Human2250
CDK9CDKCMGC4imyEAadenosine monophosphateHuman2258
CDK9CDKCMGC4imyCBadenosine monophosphateHuman2245
CDK9CDKCMGC4bchA4-(4-methyl-2-methylimino-3h-1,3-thiazol-5-yl)-2-[(4-methyl-3-morpholin-4-ylsulfonyl-phenyl)amino]pyrimidine-5-carbonitrileHuman2246
CDK9CDKCMGC4bcgA2-[[3-(1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman2255
CDK9CDKCMGC4ogrAadenosineHuman2254
CDK9CDKCMGC4bcjA2-[(3-hydroxyphenyl)amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman2247
CDK9CDKCMGC6w9eAB(4-amino-2-{[(1s,2s,4r)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13858
CDK9CDKCMGC4or5A-Human2233
CDK9CDKCMGC6w9eAD(4-amino-2-{[(1r,2r,4s)-bicyclo[2.2.1]heptan-2-yl]amino}-1,3-thiazol-5-yl)(2-nitrophenyl)methanoneHuman13860
CDK9CDKCMGC3blhA-Human2251
CDK9CDKCMGC3my1A5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman2249
CDK9CDKCMGC3lq5A(2s)-2-({9-(1-methylethyl)-6-[(4-pyridin-2-ylbenzyl)amino]-9h-purin-2-yl}amino)butan-1-olHuman2253
CDK9CDKCMGC4or5F-Human2231
CDK9CDKCMGC3tnhA4-[(e)-(3,5-diamino-1h-pyrazol-4-yl)diazenyl]phenolHuman2232
CDK9CDKCMGC4bcfA2-[[3-(4-ethanoyl-1,4-diazepan-1-yl)phenyl]amino]-4-[4-methyl-2-(methylamino)-1,3-thiazol-5-yl]pyrimidine-5-carbonitrileHuman2257
MAPK6 (Erk3)MAPKCMGC6ykyCB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12784
MAPK6 (Erk3)MAPKCMGC6yllB-Human12785
MAPK6 (Erk3)MAPKCMGC6ykyBB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12786
MAPK6 (Erk3)MAPKCMGC6ykyCA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12787
MAPK6 (Erk3)MAPKCMGC6ykyAA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12788
MAPK6 (Erk3)MAPKCMGC6ykyDB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12789
MAPK6 (Erk3)MAPKCMGC6ykyAB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12790
MAPK6 (Erk3)MAPKCMGC7aqbBA-Human12980
MAPK6 (Erk3)MAPKCMGC7aqbAB-Human12981
CDK7CDKCMGC6xd3Jn-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamideHuman12772
CDK7CDKCMGC8byqI-Human14732
CDK7CDKCMGC6o9l8-Human11055
CDK7CDKCMGC8pyrAA-Human15254
CDK7CDKCMGC6xbzJphosphothiophosphoric acid-adenylate esterHuman12773
CDK7CDKCMGC1ua2Badenosine-5'-triphosphateHuman541
CDK7CDKCMGC1ua2Aadenosine-5'-triphosphateHuman540
CDK7CDKCMGC29wdI-Human16031
CDK7CDKCMGC8bvwI-Human14733
CDK7CDKCMGC7b5oJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13279
CDK7CDKCMGC7b5qJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13280
HIPK2DYRKCMGC6p5sAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11512
HIPK2DYRKCMGC6p5sAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman11513
MAPK3 (Erk1)MAPKCMGC6gesABn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10926
MAPK3 (Erk1)MAPKCMGC4qtbBB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman1715
MAPK3 (Erk1)MAPKCMGC6gesAAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10923
MAPK3 (Erk1)MAPKCMGC2zoqB(2r,3r,4s,5r)-2-(4-amino-5-iodo-7h-pyrrolo[2,3-d]pyrimidin-7-yl)-5-(hydroxymethyl)tetrahydrofuran-3,4-diolHuman1712
MAPK3 (Erk1)MAPKCMGC9uw3Bphosphoaminophosphonic acid-adenylate esterHuman16037
MAPK3 (Erk1)MAPKCMGC9uw4Aphosphoaminophosphonic acid-adenylate esterHuman16038
MAPK3 (Erk1)MAPKCMGC4qtbAB(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman1713
MAPK3 (Erk1)MAPKCMGC4qtbAA(3r)-1-(2-oxo-2-{4-[4-(pyrimidin-2-yl)phenyl]piperazin-1-yl}ethyl)-n-[3-(pyridin-4-yl)-2h-indazol-5-yl]pyrrolidine-3-carboxamideHuman1714
MAPK3 (Erk1)MAPKCMGC6gesBAn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10925
MAPK3 (Erk1)MAPKCMGC6gesBBn-{2-[(5-chloro-2-{[4-(4-methylpiperazin-1-yl)phenyl]amino}pyrimidin-4-yl)amino]phenyl}propanamideHuman10924
CDK4CDKCMGC5fwpK-Human7132
CDK4CDKCMGC6p8hB-Human11894
CDK4CDKCMGC2w9zBA-Human3388
CDK4CDKCMGC2w9fB-Human3386
CDK4CDKCMGC6p8gB-Human11893
CDK4CDKCMGC2w96BA-Human3390
CDK4CDKCMGC2w96BB-Human3389
CDK4CDKCMGC5fwlK-Human6748
CDK4CDKCMGC2w99B-Human3385
CSNK2A1 (CK2a1)CK2CMGC4ubaB4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acidHuman5525
CSNK2A1 (CK2a1)CK2CMGC3w8lA-Human5427
CSNK2A1 (CK2a1)CK2CMGC6eiiAB(3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azaniumHuman9647
CSNK2A1 (CK2a1)CK2CMGC5motAA4-hydroxybenzamideHuman7660
CSNK2A1 (CK2a1)CK2CMGC5cu4ABn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6895
CSNK2A1 (CK2a1)CK2CMGC4ib5BA-Human5532
CSNK2A1 (CK2a1)CK2CMGC5t1hBB7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman8684
CSNK2A1 (CK2a1)CK2CMGC5otqAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methoxy-phenyl]methyl]ethanamineHuman9638
CSNK2A1 (CK2a1)CK2CMGC3owlAA11-chloro-8-methyl-7h-benzo[e]pyrido[4,3-b]indol-3-olHuman5502
CSNK2A1 (CK2a1)CK2CMGC5oulAB[3-chloranyl-4-(3-fluorophenyl)phenyl]methanamineHuman9675
CSNK2A1 (CK2a1)CK2CMGC5cvhBBadenosine-5'-diphosphateHuman6917
CSNK2A1 (CK2a1)CK2CMGC7psuAA-Human14163
CSNK2A1 (CK2a1)CK2CMGC3q9zAA1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5510
CSNK2A1 (CK2a1)CK2CMGC6l21A(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12011
CSNK2A1 (CK2a1)CK2CMGC5t1hBA7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman8683
CSNK2A1 (CK2a1)CK2CMGC5oniAA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9455
CSNK2A1 (CK2a1)CK2CMGC3juhAAphosphoaminophosphonic acid-adenylate esterHuman5471
CSNK2A1 (CK2a1)CK2CMGC3q9xAB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5488
CSNK2A1 (CK2a1)CK2CMGC5othAA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9612
CSNK2A1 (CK2a1)CK2CMGC5mmrBA-Human7651
CSNK2A1 (CK2a1)CK2CMGC6ehuAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamineHuman9691
CSNK2A1 (CK2a1)CK2CMGC5mowAA5-bromopyridine-2,3-diamineHuman7670
CSNK2A1 (CK2a1)CK2CMGC7ayaAA~{n}-[2-[(1~{r},2~{r})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman13991
CSNK2A1 (CK2a1)CK2CMGC4kwpAB4,5,6,7-tetrabromo-1-(2-deoxy-beta-d-erythro-pentofuranosyl)-1h-benzimidazoleHuman5482
CSNK2A1 (CK2a1)CK2CMGC5othBB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9670
CSNK2A1 (CK2a1)CK2CMGC3q9xAA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5446
CSNK2A1 (CK2a1)CK2CMGC5ouuBB2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman9636
CSNK2A1 (CK2a1)CK2CMGC6qy7AA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12122
CSNK2A1 (CK2a1)CK2CMGC5m4cAA3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acidHuman7402
CSNK2A1 (CK2a1)CK2CMGC5ctpABn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7289
CSNK2A1 (CK2a1)CK2CMGC4rllAA4-[(e)-(9h-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acidHuman5418
CSNK2A1 (CK2a1)CK2CMGC6fvgAAadenosine-5'-triphosphateHuman11340
CSNK2A1 (CK2a1)CK2CMGC4dglC-Human5474
CSNK2A1 (CK2a1)CK2CMGC6ypgAA4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12425
CSNK2A1 (CK2a1)CK2CMGC1jwhAphosphoaminophosphonic acid-adenylate esterHuman5485
CSNK2A1 (CK2a1)CK2CMGC3h30BA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman5484
CSNK2A1 (CK2a1)CK2CMGC5cu3AAn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6902
CSNK2A1 (CK2a1)CK2CMGC6tloAB5,6,7-tris(bromanyl)-1~{h}-benzotriazoleHuman13074
CSNK2A1 (CK2a1)CK2CMGC5zn3AA-Human10703
CSNK2A1 (CK2a1)CK2CMGC4ub7A4-(6,8-dibromo-3-hydroxy-4-oxo-4h-chromen-2-yl)benzoic acidHuman5462
CSNK2A1 (CK2a1)CK2CMGC5cquAB4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6038
CSNK2A1 (CK2a1)CK2CMGC6ypkAB-Human12426
CSNK2A1 (CK2a1)CK2CMGC6teiBB3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12457
CSNK2A1 (CK2a1)CK2CMGC6tloAC-Human13075
CSNK2A1 (CK2a1)CK2CMGC5mo5AB~{n}-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propyl]methanesulfonamideHuman7661
CSNK2A1 (CK2a1)CK2CMGC5cshBBadenosine-5'-triphosphateHuman6907
CSNK2A1 (CK2a1)CK2CMGC5mo5AA~{n}-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propyl]methanesulfonamideHuman7676
CSNK2A1 (CK2a1)CK2CMGC5ot5AB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9676
CSNK2A1 (CK2a1)CK2CMGC5oquAAadenosine-5'-diphosphateHuman9615
CSNK2A1 (CK2a1)CK2CMGC3q9xBA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5516
CSNK2A1 (CK2a1)CK2CMGC6tllAC4,5,6,7-tetrabromobenzotriazoleHuman13076
CSNK2A1 (CK2a1)CK2CMGC3nszABphosphoaminophosphonic acid-adenylate esterHuman5503
CSNK2A1 (CK2a1)CK2CMGC3amyA5,7-dihydroxy-2-(4-hydroxyphenyl)-4h-chromen-4-oneHuman5506
CSNK2A1 (CK2a1)CK2CMGC5otdAA[2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azaniumHuman9697
CSNK2A1 (CK2a1)CK2CMGC5os8AAadenosine-5'-triphosphateHuman9608
CSNK2A1 (CK2a1)CK2CMGC5oulAA[3-chloranyl-4-(3-fluorophenyl)phenyl]methanamineHuman9622
CSNK2A1 (CK2a1)CK2CMGC4md8F-Human5475
CSNK2A1 (CK2a1)CK2CMGC6ypnBAadenosine-5'-diphosphateHuman12427
CSNK2A1 (CK2a1)CK2CMGC5ct0AA3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-olHuman7296
CSNK2A1 (CK2a1)CK2CMGC5ot6AB(3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-pyrrol-2-yl)ethyl]azaniumHuman9643
CSNK2A1 (CK2a1)CK2CMGC3ngaBB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5511
CSNK2A1 (CK2a1)CK2CMGC5cu4ACn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6916
CSNK2A1 (CK2a1)CK2CMGC5mo8AB3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acidHuman7673
CSNK2A1 (CK2a1)CK2CMGC5orhAB-Human9671
CSNK2A1 (CK2a1)CK2CMGC5otlAB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9633
CSNK2A1 (CK2a1)CK2CMGC6tlsAA5,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13077
CSNK2A1 (CK2a1)CK2CMGC5cu4AAn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6924
CSNK2A1 (CK2a1)CK2CMGC6yphBA4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12428
CSNK2A1 (CK2a1)CK2CMGC5orhAA-Human9620
CSNK2A1 (CK2a1)CK2CMGC6hopAB4-hydroxy-3-methoxybenzaldehydeHuman11660
CSNK2A1 (CK2a1)CK2CMGC6tlpAB5,6-dibromobenzotriazoleHuman13078
CSNK2A1 (CK2a1)CK2CMGC3mb7ABnaphtho[2,1-b:7,8-b']difuran-2,9-dicarboxylic acidHuman5455
CSNK2A1 (CK2a1)CK2CMGC6l24AA(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12013
CSNK2A1 (CK2a1)CK2CMGC6rffAB(~{e})-~{n}-(5-bromanyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-nitro-4-oxidanyl-phenyl)prop-2-enamideHuman12149
CSNK2A1 (CK2a1)CK2CMGC5otdAB[2-[2-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methylamino]ethyl]-3~{h}-benzimidazol-4-yl]-oxidanyl-oxidanylidene-azaniumHuman9696
CSNK2A1 (CK2a1)CK2CMGC6hbnAA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11287
CSNK2A1 (CK2a1)CK2CMGC5oquABadenosine-5'-diphosphateHuman9627
CSNK2A1 (CK2a1)CK2CMGC2zjwA2,3,7,8-tetrahydroxychromeno[5,4,3-cde]chromene-5,10-dioneHuman5423
CSNK2A1 (CK2a1)CK2CMGC6yphBB4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12429
CSNK2A1 (CK2a1)CK2CMGC5oyfAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methyl-phenyl]methyl]ethanamineHuman9658
CSNK2A1 (CK2a1)CK2CMGC7at5AB~{n}'-[2-(3,4-dichlorophenyl)ethyl]-~{n}-[4-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]butyl]butanediamideHuman13839
CSNK2A1 (CK2a1)CK2CMGC6gmdAAadenosine-5'-triphosphateHuman9993
CSNK2A1 (CK2a1)CK2CMGC5h8bA~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman6408
CSNK2A1 (CK2a1)CK2CMGC3w8lB-Human5469
CSNK2A1 (CK2a1)CK2CMGC5cvfAAadenosine-5'-triphosphateHuman6927
CSNK2A1 (CK2a1)CK2CMGC5oszAB2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azaniumHuman9685
CSNK2A1 (CK2a1)CK2CMGC5orkAAadenosine-5'-diphosphateHuman9693
CSNK2A1 (CK2a1)CK2CMGC5modBA-Human7679
CSNK2A1 (CK2a1)CK2CMGC3bqcAA3-methyl-1,6,8-trihydroxyanthraquinoneHuman5486
CSNK2A1 (CK2a1)CK2CMGC5zn4AB-Human10708
CSNK2A1 (CK2a1)CK2CMGC5ot5AA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9656
CSNK2A1 (CK2a1)CK2CMGC5mo7BB-Human7685
CSNK2A1 (CK2a1)CK2CMGC5zn4AA-Human10700
CSNK2A1 (CK2a1)CK2CMGC5oumAB~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]-2-(1~{h}-imidazol-2-yl)ethanamineHuman9677
CSNK2A1 (CK2a1)CK2CMGC7zweAB7-(1~{h}-indol-2-yl)-5-methyl-~{n}-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman14771
CSNK2A1 (CK2a1)CK2CMGC6gmdABadenosine-5'-triphosphateHuman9990
CSNK2A1 (CK2a1)CK2CMGC5cu2BAmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7292
CSNK2A1 (CK2a1)CK2CMGC7qgeAB4,5,6,7-tetrabromobenzotriazoleHuman14467
CSNK2A1 (CK2a1)CK2CMGC7a4bBB 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13166
CSNK2A1 (CK2a1)CK2CMGC5mpjBA-Human7675
CSNK2A1 (CK2a1)CK2CMGC6hbnBB5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11272
CSNK2A1 (CK2a1)CK2CMGC5cvhBAadenosine-5'-diphosphateHuman6914
CSNK2A1 (CK2a1)CK2CMGC5cs6AB-Human6901
CSNK2A1 (CK2a1)CK2CMGC6yulA7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.12,6.017,20]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxylic acidHuman12458
CSNK2A1 (CK2a1)CK2CMGC5cu0BAn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7295
CSNK2A1 (CK2a1)CK2CMGC5h8gA~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-[2-(dimethylamino)ethyl-methyl-amino]phenyl]ethanamideHuman6405
CSNK2A1 (CK2a1)CK2CMGC5mowBB-Human7686
CSNK2A1 (CK2a1)CK2CMGC5cu2BBmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7286
CSNK2A1 (CK2a1)CK2CMGC4md8H-Human5518
CSNK2A1 (CK2a1)CK2CMGC6hmeBA5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11279
CSNK2A1 (CK2a1)CK2CMGC2pvrAAphosphoaminophosphonic acid-adenylate esterHuman5509
CSNK2A1 (CK2a1)CK2CMGC4md8G-Human5478
CSNK2A1 (CK2a1)CK2CMGC6tlvAA6-bromanyl-1~{h}-benzotriazoleHuman13079
CSNK2A1 (CK2a1)CK2CMGC5os7BBadenosine-5'-triphosphateHuman9645
CSNK2A1 (CK2a1)CK2CMGC6yphAB4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12431
CSNK2A1 (CK2a1)CK2CMGC5csvAA3-aminobenzoic acidHuman6898
CSNK2A1 (CK2a1)CK2CMGC6z84B~{n}-[1-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]ethanamideHuman12649
CSNK2A1 (CK2a1)CK2CMGC5zn1AA-Human10696
CSNK2A1 (CK2a1)CK2CMGC3u9cA7-hydroxy-3h-phenoxazin-3-oneHuman5461
CSNK2A1 (CK2a1)CK2CMGC4nh1Aphosphomethylphosphonic acid adenylate esterHuman5412
CSNK2A1 (CK2a1)CK2CMGC5otsAA2-(1~{h}-benzimidazol-2-yl)ethyl-[[3,5-bis(chloranyl)-4-phenyl-phenyl]methyl]azaniumHuman10589
CSNK2A1 (CK2a1)CK2CMGC5othAB~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(4-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9659
CSNK2A1 (CK2a1)CK2CMGC4md7E-Human5435
CSNK2A1 (CK2a1)CK2CMGC3nszAAphosphoaminophosphonic acid-adenylate esterHuman5512
CSNK2A1 (CK2a1)CK2CMGC6gihAA-Human9941
CSNK2A1 (CK2a1)CK2CMGC3c13AB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5472
CSNK2A1 (CK2a1)CK2CMGC5m4fAA4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7405
CSNK2A1 (CK2a1)CK2CMGC6ypgAB4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12432
CSNK2A1 (CK2a1)CK2CMGC3owlAB11-chloro-8-methyl-7h-benzo[e]pyrido[4,3-b]indol-3-olHuman5416
CSNK2A1 (CK2a1)CK2CMGC9qsvA5-(methylamino)benzo[c][2,6]naphthyridine-8-carboxylic acidHuman16074
CSNK2A1 (CK2a1)CK2CMGC9qrjA5-[6-[(3-chloranyl-4-phenyl-phenyl)methylamino]hexylamino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman16075
CSNK2A1 (CK2a1)CK2CMGC6yphAA4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)amino]-2-oxidanyl-benzoic acidHuman12433
CSNK2A1 (CK2a1)CK2CMGC7a4bAA 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13167
CSNK2A1 (CK2a1)CK2CMGC5mo7AB3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanamideHuman7697
CSNK2A1 (CK2a1)CK2CMGC9s76AAphosphoaminophosphonic acid-adenylate esterHuman16076
CSNK2A1 (CK2a1)CK2CMGC7a49B6-bromanyl-5-chloranyl-1~{h}-[1,2,3]triazolo[4,5-b]pyridineHuman13168
CSNK2A1 (CK2a1)CK2CMGC5nqcAB(3e)-6,7-dichloro-3-(hydroxyimino)-1,3-dihydro-2h-indol-2-oneHuman8111
CSNK2A1 (CK2a1)CK2CMGC5b0xA4-[2-[(4-methoxyphenyl)carbonylamino]-1,3-thiazol-5-yl]benzoic acidHuman6475
CSNK2A1 (CK2a1)CK2CMGC9hyhAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman16077
CSNK2A1 (CK2a1)CK2CMGC5zn2AB-Human10702
CSNK2A1 (CK2a1)CK2CMGC7i8nAC-Human16078
CSNK2A1 (CK2a1)CK2CMGC5otlAA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9681
CSNK2A1 (CK2a1)CK2CMGC7zy8AA-Human14441
CSNK2A1 (CK2a1)CK2CMGC5m4fAB4-[6,8-bis(chloranyl)-3-oxidanyl-4-oxidanylidene-chromen-2-yl]benzoic acidHuman7401
CSNK2A1 (CK2a1)CK2CMGC7b8hAAnicotinic acidHuman13260
CSNK2A1 (CK2a1)CK2CMGC5clpBB2-(3,4-dichlorophenyl)ethanamineHuman6911
CSNK2A1 (CK2a1)CK2CMGC5oumAA~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]-2-(1~{h}-imidazol-2-yl)ethanamineHuman9668
CSNK2A1 (CK2a1)CK2CMGC5os7AAadenosine-5'-triphosphateHuman9644
CSNK2A1 (CK2a1)CK2CMGC5omyAA4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9457
CSNK2A1 (CK2a1)CK2CMGC3pe1AB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5500
CSNK2A1 (CK2a1)CK2CMGC3juhBAphosphoaminophosphonic acid-adenylate esterHuman5431
CSNK2A1 (CK2a1)CK2CMGC3wilA{[(2z)-2-(3,4-dimethoxybenzylidene)-3-oxo-2,3-dihydro-1-benzofuran-6-yl]oxy}acetic acidHuman5468
CSNK2A1 (CK2a1)CK2CMGC5ku8A~{n}-[2-[(1~{s},2~{s})-2-(aminomethyl)cyclopropyl]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman8664
CSNK2A1 (CK2a1)CK2CMGC3q9zBB1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5430
CSNK2A1 (CK2a1)CK2CMGC9qriA5-[4-[[4-[2-(3,4-dichlorophenyl)ethylamino]-4-oxidanylidene-butanoyl]amino]butylamino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman16079
CSNK2A1 (CK2a1)CK2CMGC5mmfBB-Human7657
CSNK2A1 (CK2a1)CK2CMGC6gmdBAadenosine-5'-triphosphateHuman9991
CSNK2A1 (CK2a1)CK2CMGC5cx9BAmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7285
CSNK2A1 (CK2a1)CK2CMGC5zn0AB-Human10699
CSNK2A1 (CK2a1)CK2CMGC5owlBA3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10590
CSNK2A1 (CK2a1)CK2CMGC5moeABadenosine-5'-diphosphateHuman7662
CSNK2A1 (CK2a1)CK2CMGC5zn1AB-Human10707
CSNK2A1 (CK2a1)CK2CMGC5ospAAadenosine-5'-triphosphateHuman10587
CSNK2A1 (CK2a1)CK2CMGC5oueBB(3-chloranyl-4-phenyl-phenyl)methyl-[2-(1~{h}-imidazol-4-yl)ethyl]azaniumHuman9631
CSNK2A1 (CK2a1)CK2CMGC6hnwAAcoumestrolHuman11523
CSNK2A1 (CK2a1)CK2CMGC6tlrAB4,7-bis(bromanyl)-1~{h}-benzotriazoleHuman13083
CSNK2A1 (CK2a1)CK2CMGC5orkBBadenosine-5'-diphosphateHuman9646
CSNK2A1 (CK2a1)CK2CMGC3h30AB5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman5460
CSNK2A1 (CK2a1)CK2CMGC7i85AB5-(ethylamino)benzo[c][2,6]naphthyridine-8-carboxamideHuman16080
CSNK2A1 (CK2a1)CK2CMGC6l24AB(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12012
CSNK2A1 (CK2a1)CK2CMGC9s7iAAphosphoaminophosphonic acid-adenylate esterHuman16081
CSNK2A1 (CK2a1)CK2CMGC5orkBAadenosine-5'-diphosphateHuman9674
CSNK2A1 (CK2a1)CK2CMGC9s8jACphosphoaminophosphonic acid-adenylate esterHuman16082
CSNK2A1 (CK2a1)CK2CMGC5t1hAB7-(cyclopropylamino)-5-[3-(6-oxo-1,6-dihydropyridin-3-yl)thiophen-2-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman8682
CSNK2A1 (CK2a1)CK2CMGC5zn3AB-Human10706
CSNK2A1 (CK2a1)CK2CMGC3r0tAB3-(cyclopropylamino)-5-{[3-(trifluoromethyl)phenyl]amino}pyrimido[4,5-c]quinoline-8-carboxylic acidHuman5517
CSNK2A1 (CK2a1)CK2CMGC6ypjAB4-[(4-phenyl-1,3-thiazol-2-yl)amino]benzoic acidHuman12434
CSNK2A1 (CK2a1)CK2CMGC1na7A-Human5533
CSNK2A1 (CK2a1)CK2CMGC5otpAB2-[5,6-bis(chloranyl)-1~{h}-benzimidazol-2-yl]-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman10586
CSNK2A1 (CK2a1)CK2CMGC6qy7BB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12124
CSNK2A1 (CK2a1)CK2CMGC5mmrAB~{n}'-[(3-chloranyl-4-phenyl-phenyl)methyl]butane-1,4-diamineHuman7659
CSNK2A1 (CK2a1)CK2CMGC5oueAA3-methyl-5-oxidanyl-benzoic acidHuman9686
CSNK2A1 (CK2a1)CK2CMGC6l23AA(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman13455
CSNK2A1 (CK2a1)CK2CMGC5omyAB4-(3-methylbut-2-enoxy)-5-propan-2-yl-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman9456
CSNK2A1 (CK2a1)CK2CMGC5orjBAadenosine-5'-diphosphateHuman9607
CSNK2A1 (CK2a1)CK2CMGC5mpjABadenosine-5'-diphosphateHuman7663
CSNK2A1 (CK2a1)CK2CMGC6q38AAbenzoic acidHuman11271
CSNK2A1 (CK2a1)CK2CMGC5owlAB3-[4,5,6,7-tetrakis(bromanyl)benzimidazol-1-yl]propan-1-amineHuman10596
CSNK2A1 (CK2a1)CK2CMGC4ib5CA-Human5498
CSNK2A1 (CK2a1)CK2CMGC8aemABadenosine-5'-triphosphateHuman14683
CSNK2A1 (CK2a1)CK2CMGC5oquBAadenosine-5'-diphosphateHuman9623
CSNK2A1 (CK2a1)CK2CMGC5cs6BA-Human6919
CSNK2A1 (CK2a1)CK2CMGC5cs6BB-Human6926
CSNK2A1 (CK2a1)CK2CMGC1pjkAAphosphoaminophosphonic acid-adenylate esterHuman5494
CSNK2A1 (CK2a1)CK2CMGC5ouuAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[(3-chloranyl-4-phenyl-phenyl)methyl]ethanamineHuman9662
CSNK2A1 (CK2a1)CK2CMGC3fwqA-Human5507
CSNK2A1 (CK2a1)CK2CMGC5oszAC2-(1~{h}-benzimidazol-2-yl)ethyl-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]azaniumHuman9683
CSNK2A1 (CK2a1)CK2CMGC3h30AA5,6-dichloro-1-beta-d-ribofuranosyl-1h-benzimidazoleHuman5496
CSNK2A1 (CK2a1)CK2CMGC3juhBBphosphoaminophosphonic acid-adenylate esterHuman5421
CSNK2A1 (CK2a1)CK2CMGC5mohAB2-(3-methoxy-4-oxidanyl-phenyl)ethanoic acidHuman7681
CSNK2A1 (CK2a1)CK2CMGC5mo8AA3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acidHuman7653
CSNK2A1 (CK2a1)CK2CMGC5cvgAA-Human6913
CSNK2A1 (CK2a1)CK2CMGC5oyfAA2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-methyl-phenyl]methyl]ethanamineHuman9617
CSNK2A1 (CK2a1)CK2CMGC5mo8BA3-[[3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoyl]amino]benzoic acidHuman7654
CSNK2A1 (CK2a1)CK2CMGC6rcmAB(~{e})-~{n}-(5-~{tert}-butyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12143
CSNK2A1 (CK2a1)CK2CMGC5orjABadenosine-5'-diphosphateHuman9624
CSNK2A1 (CK2a1)CK2CMGC3axwA4-(5-amino-1,3,4-thiadiazol-2-yl)benzoic acidHuman5440
CSNK2A1 (CK2a1)CK2CMGC7b8iAB-Human13261
CSNK2A1 (CK2a1)CK2CMGC7z39AB2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamideHuman14445
CSNK2A1 (CK2a1)CK2CMGC5otoAB2-(5-chloranyl-1~{h}-benzimidazol-2-yl)-~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9637
CSNK2A1 (CK2a1)CK2CMGC6z84A~{n}-[1-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]ethanamideHuman12650
CSNK2A1 (CK2a1)CK2CMGC5n1vBApyrazolo-pyrimidine macrocycleHuman7587
CSNK2A1 (CK2a1)CK2CMGC5orjBBadenosine-5'-diphosphateHuman9665
CSNK2A1 (CK2a1)CK2CMGC9fyfA~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-4-fluoranyl-2-[(3~{s})-3-(methylamino)piperidin-1-yl]phenyl]propanamideHuman16083
CSNK2A1 (CK2a1)CK2CMGC6spxA-Human11960
CSNK2A1 (CK2a1)CK2CMGC5zn0AD-Human10709
CSNK2A1 (CK2a1)CK2CMGC5ot5BA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(7-methyl-1~{h}-benzimidazol-2-yl)ethanamineHuman9689
CSNK2A1 (CK2a1)CK2CMGC3q04AA-Human5514
CSNK2A1 (CK2a1)CK2CMGC5motAB4-hydroxybenzamideHuman7691
CSNK2A1 (CK2a1)CK2CMGC3fwqB-Human5479
CSNK2A1 (CK2a1)CK2CMGC6l22AB(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12014
CSNK2A1 (CK2a1)CK2CMGC5cqwBA4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6039
CSNK2A1 (CK2a1)CK2CMGC6q4qBCbenzoic acidHuman11280
CSNK2A1 (CK2a1)CK2CMGC5oumBB-Human9606
CSNK2A1 (CK2a1)CK2CMGC9rfnAB-Human16084
CSNK2A1 (CK2a1)CK2CMGC5m44A3-[5-(4-methylphenyl)thieno[2,3-d]pyrimidin-4-yl]sulfanylpropanoic acidHuman7404
CSNK2A1 (CK2a1)CK2CMGC5cvfABadenosine-5'-triphosphateHuman6910
CSNK2A1 (CK2a1)CK2CMGC6qy7AB2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12123
CSNK2A1 (CK2a1)CK2CMGC8ae7ABadenosine-5'-diphosphateHuman14684
CSNK2A1 (CK2a1)CK2CMGC6tllAD4,5,6,7-tetrabromobenzotriazoleHuman13087
CSNK2A1 (CK2a1)CK2CMGC5mo6AA3-[3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propylamino]-3-oxidanylidene-propanoic acidHuman7672
CSNK2A1 (CK2a1)CK2CMGC6spwAB-Human11959
CSNK2A1 (CK2a1)CK2CMGC6fvfAA-Human11342
CSNK2A1 (CK2a1)CK2CMGC6ypjAA4-[(4-phenyl-1,3-thiazol-2-yl)amino]benzoic acidHuman12435
CSNK2A1 (CK2a1)CK2CMGC9s8jAAphosphoaminophosphonic acid-adenylate esterHuman16085
CSNK2A1 (CK2a1)CK2CMGC5oslAAadenosine-5'-diphosphateHuman9673
CSNK2A1 (CK2a1)CK2CMGC5mo7AA3-[(3-chloranyl-4-phenyl-phenyl)methylamino]propanamideHuman7669
CSNK2A1 (CK2a1)CK2CMGC6hnyAAboldineHuman11520
CSNK2A1 (CK2a1)CK2CMGC5otlBA~{n}-[[3-chloranyl-4-(2-ethylphenyl)phenyl]methyl]-2-(5-methoxy-1~{h}-benzimidazol-2-yl)ethanamineHuman9660
CSNK2A1 (CK2a1)CK2CMGC5cu2AAmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7303
CSNK2A1 (CK2a1)CK2CMGC6l22AA(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12009
CSNK2A1 (CK2a1)CK2CMGC7zwgAB(5~{z})-5-(quinolin-6-ylmethylidene)-1,3-thiazolidine-2,4-dioneHuman14774
CSNK2A1 (CK2a1)CK2CMGC8aemAAadenosine-5'-triphosphateHuman14685
CSNK2A1 (CK2a1)CK2CMGC4md9M-Human5520
CSNK2A1 (CK2a1)CK2CMGC6z83B~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamideHuman12651
CSNK2A1 (CK2a1)CK2CMGC5oueAB3-methyl-5-oxidanyl-benzoic acidHuman9614
CSNK2A1 (CK2a1)CK2CMGC6spwAA-Human11961
CSNK2A1 (CK2a1)CK2CMGC3at3A(1-{6-[6-(cyclopentylamino)-1h-indazol-1-yl]pyrazin-2-yl}-1h-pyrrol-3-yl)acetic acidHuman5504
CSNK2A1 (CK2a1)CK2CMGC9s6gAAphosphoaminophosphonic acid-adenylate esterHuman16086
CSNK2A1 (CK2a1)CK2CMGC3q04AB-Human5419
CSNK2A1 (CK2a1)CK2CMGC6hoqAB3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acidHuman11665
CSNK2A1 (CK2a1)CK2CMGC5cspAC2-hydroxy-5-methylbenzoic acidHuman6928
CSNK2A1 (CK2a1)CK2CMGC7x4hAB5-azanyl-3-[(~{z})-1-cyano-2-(1~{h}-indol-3-yl)ethenyl]-1~{h}-pyrazole-4-carbonitrileHuman14596
CSNK2A1 (CK2a1)CK2CMGC7z39AA2-[3-[4-(1~{h}-indazol-5-ylamino)quinazolin-2-yl]phenoxy]-~{n}-propan-2-yl-ethanamideHuman14449
CSNK2A1 (CK2a1)CK2CMGC5zn0AC-Human10704
CSNK2A1 (CK2a1)CK2CMGC6gihAB-Human9942
CSNK2A1 (CK2a1)CK2CMGC5n9lAB(4~{z})-6,7-bis(chloranyl)-4-[[(4-methylphenyl)amino]methylidene]-8-oxidanyl-1,2-dihydrodibenzofuran-3-oneHuman9621
CSNK2A1 (CK2a1)CK2CMGC8c5qAA2-methylpropyl 5-fluoranyl-3-[1-[[1-[2-[[4-(2-methylpropyl)phenyl]sulfonylamino]ethyl]piperidin-4-yl]methyl]-1,2,3-triazol-4-yl]-1~{h}-indole-2-carboxylateHuman15177
CSNK2A1 (CK2a1)CK2CMGC6rcmAA(~{e})-~{n}-(5-~{tert}-butyl-1,3,4-thiadiazol-2-yl)-2-cyano-3-(3-methoxy-4-oxidanyl-phenyl)prop-2-enamideHuman12150
CSNK2A1 (CK2a1)CK2CMGC3ngaAA5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman5422
CSNK2A1 (CK2a1)CK2CMGC4md9P-Human5434
CSNK2A1 (CK2a1)CK2CMGC5cu2ABmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7302
CSNK2A1 (CK2a1)CK2CMGC6hmeAB5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11283
CSNK2A1 (CK2a1)CK2CMGC5cqwAB4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6037
CSNK2A1 (CK2a1)CK2CMGC5ct0AB3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-olHuman7300
CSNK2A1 (CK2a1)CK2CMGC7bu4AB4-(6-aminocarbonyl-8-oxidanylidene-9-phenyl-7h-purin-2-yl)benzoic acidHuman13485
CSNK2A1 (CK2a1)CK2CMGC4md7F-Human5457
CSNK2A1 (CK2a1)CK2CMGC5otyABtrifluoroacetic acidHuman9680
CSNK2A1 (CK2a1)CK2CMGC9s8jABphosphoaminophosphonic acid-adenylate esterHuman16091
CSNK2A1 (CK2a1)CK2CMGC9fblAAnicotinic acidHuman16092
CSNK2A1 (CK2a1)CK2CMGC3mb6ABnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman5499
CSNK2A1 (CK2a1)CK2CMGC5orjAAadenosine-5'-diphosphateHuman9653
CSNK2A1 (CK2a1)CK2CMGC9s77ABnicotinic acidHuman16093
CSNK2A1 (CK2a1)CK2CMGC5mo7BA-Human7698
CSNK2A1 (CK2a1)CK2CMGC3r0tAA3-(cyclopropylamino)-5-{[3-(trifluoromethyl)phenyl]amino}pyrimido[4,5-c]quinoline-8-carboxylic acidHuman5497
CSNK2A1 (CK2a1)CK2CMGC7a4bBA 5,6-dibromo-1h-triazolo[4,5-b]pyridineHuman13172
CSNK2A1 (CK2a1)CK2CMGC9s7hAAphosphoaminophosphonic acid-adenylate esterHuman16094
CSNK2A1 (CK2a1)CK2CMGC5cqwAA4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6034
CSNK2A1 (CK2a1)CK2CMGC5mp8ABadenosine-5'-diphosphateHuman7649
CSNK2A1 (CK2a1)CK2CMGC5cshABadenosine-5'-triphosphateHuman6925
CSNK2A1 (CK2a1)CK2CMGC5h8bB~{n}-[5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman6406
CSNK2A1 (CK2a1)CK2CMGC6yzhABadenosine-5'-diphosphateHuman13560
CSNK2A1 (CK2a1)CK2CMGC6ehuBB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[4-(2-ethylphenyl)-3-(trifluoromethyl)phenyl]methyl]ethanamineHuman9664
CSNK2A1 (CK2a1)CK2CMGC5n9nAB1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diolHuman9628
CSNK2A1 (CK2a1)CK2CMGC4md9H-Human5466
CSNK2A1 (CK2a1)CK2CMGC5kwhAA~{n}-[5-[[7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]ethanamideHuman8617
CSNK2A1 (CK2a1)CK2CMGC5oumBA-Human9679
CSNK2A1 (CK2a1)CK2CMGC5osrABadenosine-5'-triphosphateHuman10594
CSNK2A1 (CK2a1)CK2CMGC6teiAA3-[(4-pyridin-2-yl-1,3-thiazol-2-yl)amino]benzoic acidHuman12461
CSNK2A1 (CK2a1)CK2CMGC6a1cAA5-bromanyl-2-methoxy-4-[(e)-(3-methylsulfanyl-5-phenyl-1,2,4-triazol-4-yl)iminomethyl]phenolHuman11273
CSNK2A1 (CK2a1)CK2CMGC5ospABadenosine-5'-triphosphateHuman10600
CSNK2A1 (CK2a1)CK2CMGC9s76ABphosphoaminophosphonic acid-adenylate esterHuman16095
CSNK2A1 (CK2a1)CK2CMGC9rcxAA-Human16096
CSNK2A1 (CK2a1)CK2CMGC5cu3BBn-[(2-chlorobiphenyl-4-yl)methyl]-beta-alanyl-n-(3-carboxyphenyl)-beta-alaninamideHuman6897
CSNK2A1 (CK2a1)CK2CMGC9fbmABnicotinic acidHuman16098
CSNK2A1 (CK2a1)CK2CMGC6hopAA3-(4-hydroxy-3-methoxyphenyl)-2-propenoic acidHuman11661
CSNK2A1 (CK2a1)CK2CMGC5h8eB~{n}-[2-[2-azanylethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]ethanamideHuman6407
CSNK2A1 (CK2a1)CK2CMGC6hopAD(2e)-3-(4-hydroxy-3-methoxyphenyl)prop-2-enalHuman11666
CSNK2A1 (CK2a1)CK2CMGC3at2AB-Human5492
CSNK2A1 (CK2a1)CK2CMGC5ctpBAn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7297
CSNK2A1 (CK2a1)CK2CMGC4ib5AA-Human5501
CSNK2A1 (CK2a1)CK2CMGC5n9nAA1,3-bis(chloranyl)-6-[(~{e})-(4-methoxyphenyl)iminomethyl]dibenzofuran-2,7-diolHuman9661
CSNK2A1 (CK2a1)CK2CMGC6z83A~{n}-[5-[[3-cyano-7-(cyclopropylamino)-3~{h}-pyrazolo[1,5-a]pyrimidin-5-yl]amino]-2-methyl-phenyl]propanamideHuman12652
CSNK2A1 (CK2a1)CK2CMGC5mo5BA-Human7689
CSNK2A1 (CK2a1)CK2CMGC5zn5AB-Human10701
CSNK2A1 (CK2a1)CK2CMGC6hnyABboldineHuman11522
CSNK2A1 (CK2a1)CK2CMGC5cu0AAn-(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)acetamideHuman7299
CSNK2A1 (CK2a1)CK2CMGC5ot6BB-Human9649
CSNK2A1 (CK2a1)CK2CMGC7zy5AB-Human14453
CSNK2A1 (CK2a1)CK2CMGC4kwpAA4,5,6,7-tetrabromo-1-(2-deoxy-beta-d-erythro-pentofuranosyl)-1h-benzimidazoleHuman5465
CSNK2A1 (CK2a1)CK2CMGC5orhBA-Human9694
CSNK2A1 (CK2a1)CK2CMGC7zy8AB-Human14454
CSNK2A1 (CK2a1)CK2CMGC3q9wAB3-methyl-1,6,8-trihydroxyanthraquinoneHuman5420
CSNK2A1 (CK2a1)CK2CMGC5otrAAadenosine-5'-triphosphateHuman9640
CSNK2A1 (CK2a1)CK2CMGC6eiiBB(3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azaniumHuman9642
CSNK2A1 (CK2a1)CK2CMGC4rllAB4-[(e)-(9h-fluoren-9-ylidenehydrazinylidene)methyl]benzoic acidHuman5449
CSNK2A1 (CK2a1)CK2CMGC5ct0BB3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propan-1-olHuman7298
CSNK2A1 (CK2a1)CK2CMGC9rcyAA-Human16099
CSNK2A1 (CK2a1)CK2CMGC9s9yAAphosphoaminophosphonic acid-adenylate esterHuman16100
CSNK2A1 (CK2a1)CK2CMGC7zweAA7-(1~{h}-indol-2-yl)-5-methyl-~{n}-(3,4,5-trimethoxyphenyl)imidazo[5,1-f][1,2,4]triazin-2-amineHuman14775
CSNK2A1 (CK2a1)CK2CMGC5os8ABadenosine-5'-triphosphateHuman9666
CSNK2A1 (CK2a1)CK2CMGC5cx9BBmethyl 3-[(3-{[(2-chlorobiphenyl-4-yl)methyl]amino}propyl)amino]-3-oxopropanoateHuman7294
CSNK2A1 (CK2a1)CK2CMGC3qa0AB-Human5451
CSNK2A1 (CK2a1)CK2CMGC5orhBB-Human9639
CSNK2A1 (CK2a1)CK2CMGC6l1zA(6ar)-3,4,6a,10-tetrakis(oxidanyl)-6,7-dihydroindeno[2,1-c]chromen-9-oneHuman12010
CSNK2A1 (CK2a1)CK2CMGC6houAB4-hydroxy-3-methoxybenzaldehydeHuman11664
CSNK2A1 (CK2a1)CK2CMGC5mmfBA-Human7696
CSNK2A1 (CK2a1)CK2CMGC3mb6AAnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman5424
CSNK2A1 (CK2a1)CK2CMGC6tloAA5,6,7-tris(bromanyl)-1~{h}-benzotriazoleHuman13092
CSNK2A1 (CK2a1)CK2CMGC6hmeBB5-propan-2-yl-4-prop-2-enoxy-7,8-dihydro-6~{h}-indeno[1,2-b]indole-9,10-dioneHuman11282
CSNK2A1 (CK2a1)CK2CMGC7zy5AA-Human14457
CSNK2A1 (CK2a1)CK2CMGC4nh1Bphosphomethylphosphonic acid adenylate esterHuman5531
CSNK2A1 (CK2a1)CK2CMGC5cvhABadenosine-5'-diphosphateHuman6912
CSNK2A1 (CK2a1)CK2CMGC3mb6ACnaphtho[2,1-b:7,6-b']difuran-2,8-dicarboxylic acidHuman5529
CSNK2A1 (CK2a1)CK2CMGC5mp8AAadenosine-5'-diphosphateHuman7690
CSNK2A1 (CK2a1)CK2CMGC5cqwBB4-[4-[2-[4,5,6,7-tetrakis(bromanyl)benzotriazol-2-yl]ethyl]-1,2,3-triazol-1-yl]butan-1-amineHuman6036
CSNK2A1 (CK2a1)CK2CMGC5csvAB3-aminobenzoic acidHuman6900
CSNK2A1 (CK2a1)CK2CMGC3q9zBA1,2,5,8-tetrahydroxyanthracene-9,10-dioneHuman5426
CSNK2A1 (CK2a1)CK2CMGC6qy7BA2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-olHuman12125
CSNK2A1 (CK2a1)CK2CMGC6eiiBA(3-chloranyl-4-phenyl-phenyl)methyl-(3-phenylpropyl)azaniumHuman9654
CSNK2A1 (CK2a1)CK2CMGC7zy2ABadenosine-5'-triphosphateHuman14458
CSNK2A1 (CK2a1)CK2CMGC7ay9A7-(cyclopropylamino)-5-(5-(6-oxo-1,6-dihydropyridin-3-yl)-1-(2-(piperidin-1-yl)ethyl)-1h-1,2,3-triazol-4-yl)pyrazolo[1,5-a]pyrimidine-3-carbonitrileHuman13993
CSNK2A1 (CK2a1)CK2CMGC6ehkAB2-(1~{h}-benzimidazol-2-yl)-~{n}-[[3,5-bis(chloranyl)-4-(2-ethylphenyl)phenyl]methyl]ethanamineHuman9663
CDK5CDKCMGC1ungA6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2792
CDK5CDKCMGC1h4lB-Human2779
CDK5CDKCMGC4au8BB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2781
CDK5CDKCMGC7vdpA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14145
CDK5CDKCMGC4au8AA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2784
CDK5CDKCMGC1unlAr-roscovitineHuman2785
CDK5CDKCMGC4au8BA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2791
HIPK3DYRKCMGC7o7jAn-{5-[(4-ethylpiperazin-1-yl)methyl]pyridin-2-yl}-5-fluoro-4-[4-fluoro-2-methyl-1-(propan-2-yl)-1h-benzimidazol-6-yl]pyrimidin-2-amineHuman13997
CLK2CLKCMGC6fykAB(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10408
CLK2CLKCMGC6fykAA(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10406
CLK2CLKCMGC6fykBB(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10401
CLK2CLKCMGC6fykBA(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10407
CLK2CLKCMGC6fylAB5-[(3-chlorophenyl)amino]benzo[c][2,6]naphthyridine-8-carboxylic acidHuman10404
CLK2CLKCMGC5unpBn~2~-methyl-n~4~-[(pyrimidin-2-yl)methyl]-5-(quinolin-6-yl)-7h-pyrrolo[2,3-d]pyrimidine-2,4-diamineHuman9888
CLK2CLKCMGC6fyiA(1~{z})-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-oneHuman10405
CLK2CLKCMGC6fykCB(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10409
CLK2CLKCMGC6fykCA(2~{s})-4-methyl-1-[5-(3-methyl-2~{h}-indazol-5-yl)pyridin-3-yl]oxy-pentan-2-amineHuman10402
MAPK12 (p38g)MAPKCMGC1cm8Aphosphoaminophosphonic acid-adenylate esterHuman4625
MAPK12 (p38g)MAPKCMGC6unaAA-Human11898
MAPK12 (p38g)MAPKCMGC6unaBB-Human11899
MAPK12 (p38g)MAPKCMGC1cm8Bphosphoaminophosphonic acid-adenylate esterHuman4626