Search results (37 entries covering 22 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
Aurka (AurA)AUROther3d14AA1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouse5781
Pomk (SGK196)Other-UniqueOther5gz8A-Mouse8033
Ern1 (IRE1)IREOther4pl3Aadenosine-5'-diphosphateMouse5769
Aurka (AurA)AUROther3dj7AA1-(5-{2-[(6-amino-5-bromopyrimidin-4-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouse5780
Aurka (AurA)AUROther3d14AB1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouse5775
Aak1 (AAK1)NAKOther7rj6AB5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineMouse14131
Aak1 (AAK1)NAKOther7rj7AA2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrileMouse14128
Aak1 (AAK1)NAKOther7lviAB(2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamideMouse13821
Aak1 (AAK1)NAKOther7lviAA(2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamideMouse13822
Aak1 (AAK1)NAKOther7lvhAn-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse13820
Ern1 (IRE1)IREOther4pl3Badenosine-5'-diphosphateMouse5768
Ern1 (IRE1)IREOther4pl4Cadenosine-5'-diphosphateMouse5761
Ern1 (IRE1)IREOther4pl5Badenosine-5'-diphosphateMouse5764
Ern1 (IRE1)IREOther4pl5Cadenosine-5'-diphosphateMouse5766
Ern1 (IRE1)IREOther4pl5Dadenosine-5'-diphosphateMouse5763
Ern1 (IRE1)IREOther4pl4Dadenosine-5'-diphosphateMouse5765
Ern1 (IRE1)IREOther4pl4Aadenosine-5'-diphosphateMouse5770
Ern1 (IRE1)IREOther4pl4Badenosine-5'-diphosphateMouse5767
Ern1 (IRE1)IREOther4pl5Aadenosine-5'-diphosphateMouse5762
Tbk1 (TBK1)IKKOther4jlcA3-{2,4-dimethyl-5-[(z)-(2-oxo-1,2-dihydro-3h-indol-3-ylidene)methyl]-1h-pyrrol-3-yl}propanoic acidMouse5698
Tbk1 (TBK1)IKKOther6o8cBBn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse11304
Tbk1 (TBK1)IKKOther6o8cABn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse11302
Tbk1 (TBK1)IKKOther6o8cAAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse11303
Tbk1 (TBK1)IKKOther4jl9An-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse5697
Tbk1 (TBK1)IKKOther6o8cBAn-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamideMouse11305
Aurka (AurA)AUROther3d2kA(7-{[2-(2-{[(3-chlorophenyl)carbamoyl]amino}-1,3-thiazol-5-yl)ethyl]amino}-1h-pyrazolo[4,3-d]pyrimidin-1-yl)acetic acidMouse5776
Aurka (AurA)AUROther3dajAn-butyl-3-{[6-(9h-purin-6-ylamino)hexanoyl]amino}benzamideMouse5779
Aurka (AurA)AUROther3dj5A3-({3-[(6-amino-5-bromopyrimidin-4-yl)sulfanyl]propanoyl}amino)-4-methoxy-n-phenylbenzamideMouse5783
Aurka (AurA)AUROther3d2iA1-(5-{2-[(1-methyl-1h-pyrazolo[4,3-d]pyrimidin-7-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouse5782
Aurka (AurA)AUROther3d15AA1-(3-chlorophenyl)-3-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}ureaMouse5777
Aurka (AurA)AUROther3dj6A4-methoxy-n-phenyl-3-({3-[(1h-pyrrolo[2,3-b]pyridin-5-ylmethyl)sulfanyl]propanoyl}amino)benzamideMouse5778
Pomk (SGK196)Other-UniqueOther5gz9Aphosphoaminophosphonic acid-adenylate esterMouse8034
Eif2ak3 (PEK)PEKOther3qd2B-Mouse5802
Aak1 (AAK1)NAKOther7rj8ABn-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse14127
Aak1 (AAK1)NAKOther7rj7AB2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrileMouse14129
Aak1 (AAK1)NAKOther7rj8AAn-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse14130
Aak1 (AAK1)NAKOther7rj6AA5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineMouse14132