| Btk (BTK) | Tec | TK | 8s93 | A | A | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | 14997 | |
| Abl1 (ABL1) | Abl | TK | 1m52 | A | | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Mouse | 5720 | |
| Abl1 (ABL1) | Abl | TK | 3oy3 | A | | 5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamide | Mouse | 5711 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | B | A | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5712 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10610 | |
| Abl1 (ABL1) | Abl | TK | 3mss | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5730 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5734 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | A | B | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5729 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5722 | |
| Abl1 (ABL1) | Abl | TK | 3dk6 | A | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5725 | |
| Abl1 (ABL1) | Abl | TK | 3ik3 | B | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Mouse | 5739 | |
| Abl1 (ABL1) | Abl | TK | 1m52 | B | | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Mouse | 5715 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5733 | |
| Jak2 (JAK2) | JakA | TK | 4gl9 | D | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6935 | |
| Jak2 (JAK2) | JakA | TK | 4gl9 | B | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6936 | |
| Jak2 (JAK2) | JakA | TK | 4gl9 | C | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6934 | |
| Jak2 (JAK2) | JakA | TK | 4gl9 | A | | 2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-one | Mouse | 6933 | |
| Src (SRC) | Src | TK | 6f3f | A | | adenosine-5'-diphosphate | Mouse | 9461 | |
| Tyk2 (TYK2) | JakA | TK | 4e1z | A | | n-[5-(4-{[(3-chlorophenyl)sulfonyl]amino}phenyl)-1h-indazol-3-yl]furan-2-carboxamide | Mouse | 5828 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10611 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10648 | |
| Abl1 (ABL1) | Abl | TK | 3oy3 | B | | 5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamide | Mouse | 5738 | |
| Tyk2 (TYK2) | JakA | TK | 4e20 | A | | n-[4-(3-amino-1h-indazol-5-yl)phenyl]-3-chlorobenzenesulfonamide | Mouse | 5827 | |
| Tyro3 (TYRO3) | Axl | TK | 3qup | A | | (5-fluoro-1h-indol-2-yl)[(3r)-1'-[(3r)-piperidin-3-yl]spiro[indole-3,3'-pyrrolidin]-1(2h)-yl]methanone | Mouse | 5799 | |
| Abl1 (ABL1) | Abl | TK | 3dk7 | B | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5714 | |
| Abl1 (ABL1) | Abl | TK | 2qoh | B | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5716 | |
| Insr (INSR) | InsR | TK | 8eyx | A | | - | Mouse | 14496 | |
| Insr (INSR) | InsR | TK | 8eyy | A | | - | Mouse | 14497 | |
| Epha4 (EphA4) | Eph | TK | 2hel | A | | - | Mouse | 5812 | |
| Epha4 (EphA4) | Eph | TK | 2y6m | A | A | - | Mouse | 5809 | |
| Epha4 (EphA4) | Eph | TK | 2xyu | A | | 5-(5-fluoro-2-methylphenyl)-6,7,8,9-tetrahydro-3h-pyrazolo[3,4-c]isoquinolin-1-amine | Mouse | 5810 | |
| Epha4 (EphA4) | Eph | TK | 2y6o | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5814 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5708 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10645 | |
| Btk (BTK) | Tec | TK | 8s93 | A | B | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | 14996 | |
| Btk (BTK) | Tec | TK | 8s9f | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 14998 | |
| Btk (BTK) | Tec | TK | 8gmb | A | | 2-[3'-(hydroxymethyl)-1-methyl-5-({5-[(2s)-2-methyl-4-(oxetan-3-yl)piperazin-1-yl]pyridin-2-yl}amino)-6-oxo[1,6-dihydro[3,4'-bipyridine]]-2'-yl]-7,7-dimethyl-3,4,7,8-tetrahydro-2h-cyclopenta[4,5]pyrrolo[1,2-a]pyrazin-1(6h)-one | Mouse | 14999 | |
| Insr (INSR) | InsR | TK | 8dtl | B | | - | Mouse | 14362 | |
| Btk (BTK) | Tec | TK | 8ff0 | A | | 6-azanyl-9-[(3~{r})-1-[(~{e})-but-2-enoyl]pyrrolidin-3-yl]-7-(4-phenoxyphenyl)purin-8-one | Mouse | 14834 | |
| Btk (BTK) | Tec | TK | 8fd9 | A | A | acalabrutinib | Mouse | 14836 | |
| Btk (BTK) | Tec | TK | 8fd9 | A | B | acalabrutinib | Mouse | 14835 | |
| Ephb2 (EphB2) | Eph | TK | 2hen | B | | adenosine-5'-diphosphate | Mouse | 5804 | |
| Ephb2 (EphB2) | Eph | TK | 1jpa | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5806 | |
| Ephb2 (EphB2) | Eph | TK | 2hen | A | | adenosine-5'-diphosphate | Mouse | 5807 | |
| Ephb2 (EphB2) | Eph | TK | 2hen | D | | adenosine-5'-diphosphate | Mouse | 5803 | |
| Ephb2 (EphB2) | Eph | TK | 2hen | C | | adenosine-5'-diphosphate | Mouse | 5808 | |
| Jak1 (JAK1) | JakA | TK | 8ewy | A | | - | Mouse | 14664 | |
| Src (SRC) | Src | TK | 8xn8 | A | A | adenosine-5'-diphosphate | Mouse | 15182 | |
| Src (SRC) | Src | TK | 8xn8 | A | B | adenosine-5'-diphosphate | Mouse | 15183 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5713 | |
| Lyn (LYN) | Src | TK | 2zva | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5774 | |
| Lyn (LYN) | Src | TK | 2zv7 | A | | - | Mouse | 5771 | |
| Abl1 (ABL1) | Abl | TK | 1opj | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5736 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10609 | |
| Abl1 (ABL1) | Abl | TK | 1opk | A | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Mouse | 5709 | |
| Lyn (LYN) | Src | TK | 2zv8 | A | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5772 | |
| Lyn (LYN) | Src | TK | 2zv9 | A | | 1-tert-butyl-3-(4-chloro-phenyl)-1h-pyrazolo[3,4-d]pyrimidin-4-ylamine | Mouse | 5773 | |
| Abl1 (ABL1) | Abl | TK | 1opj | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5732 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | B | B | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5737 | |
| Abl1 (ABL1) | Abl | TK | 3kf4 | B | | n-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amine | Mouse | 5741 | |
| Abl1 (ABL1) | Abl | TK | 3mss | C | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5719 | |
| Abl1 (ABL1) | Abl | TK | 3ik3 | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Mouse | 5731 | |
| Abl1 (ABL1) | Abl | TK | 3kfa | A | | 3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamide | Mouse | 5742 | |
| Abl1 (ABL1) | Abl | TK | 1fpu | B | | n-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamide | Mouse | 5705 | |
| Abl1 (ABL1) | Abl | TK | 1iep | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5703 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5723 | |
| Abl1 (ABL1) | Abl | TK | 3kf4 | A | | n-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amine | Mouse | 5717 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10608 | |
| Abl1 (ABL1) | Abl | TK | 1iep | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5727 | |
| Abl1 (ABL1) | Abl | TK | 3dk6 | B | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5718 | |
| Abl1 (ABL1) | Abl | TK | 3dk7 | A | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5704 | |
| Abl1 (ABL1) | Abl | TK | 2z60 | A | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5735 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5706 | |
| Abl1 (ABL1) | Abl | TK | 3oxz | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Mouse | 5721 | |
| Abl1 (ABL1) | Abl | TK | 3mss | D | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5702 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | A | A | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5726 | |
| Abl1 (ABL1) | Abl | TK | 2qoh | A | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5707 | |
| Abl1 (ABL1) | Abl | TK | 1fpu | A | | n-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamide | Mouse | 5728 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10646 | |
| Abl1 (ABL1) | Abl | TK | 2hzn | A | | 1-[4-(pyridin-4-yloxy)phenyl]-3-[3-(trifluoromethyl)phenyl]urea | Mouse | 5701 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10647 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5710 | |
| Abl1 (ABL1) | Abl | TK | 3kfa | B | | 3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamide | Mouse | 5740 | |
| Abl1 (ABL1) | Abl | TK | 3mss | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5724 | |
| Abl2 (ABL2) | Abl | TK | 4xli | B | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5690 | |
| Abl2 (ABL2) | Abl | TK | 4xli | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5689 | |
| Igf1r (IGF1R) | InsR | TK | 6pyh | A | | - | Mouse | 11777 | |
| Igf1r (IGF1R) | InsR | TK | 6pyh | D | | - | Mouse | 11776 | |
| Ephb2 (EphB2) | Eph | TK | 1jpa | B | | phosphoaminophosphonic acid-adenylate ester | Mouse | 5805 | |
| Insr (INSR) | InsR | TK | 7sl7 | A | | - | Mouse | 14169 | |
| Insr (INSR) | InsR | TK | 7stj | A | | - | Mouse | 14170 | |
| Insr (INSR) | InsR | TK | 7sl6 | A | | - | Mouse | 14171 | |
| Insr (INSR) | InsR | TK | 7sl4 | A | | - | Mouse | 14172 | |
| Btk (BTK) | Tec | TK | 9xyv | A | A | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Mouse | 16246 | |
| Btk (BTK) | Tec | TK | 9xz2 | A | B | 6-amino-7-(4-phenoxyphenyl)-9-[(3r)-1-propanoylpyrrolidin-3-yl]-7,9-dihydro-8h-purin-8-one | Mouse | 16247 | |
| Btk (BTK) | Tec | TK | 6mny | B | A | - | Mouse | 11306 | |
| Btk (BTK) | Tec | TK | 9xyv | A | C | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Mouse | 16248 | |
| Btk (BTK) | Tec | TK | 9xz2 | A | A | 6-amino-7-(4-phenoxyphenyl)-9-[(3r)-1-propanoylpyrrolidin-3-yl]-7,9-dihydro-8h-purin-8-one | Mouse | 16249 | |
| Btk (BTK) | Tec | TK | 4xi2 | A | | - | Mouse | 5815 | |
| Btk (BTK) | Tec | TK | 9xyy | A | | (2e)-1-{(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}but-2-en-1-one | Mouse | 16250 | |
| Btk (BTK) | Tec | TK | 6mny | B | B | - | Mouse | 11309 | |
| Btk (BTK) | Tec | TK | 9xyv | A | B | 1-[(3~{r})-3-[4-azanyl-3-(4-phenoxyphenyl)pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl]propan-1-one | Mouse | 16251 | |
| Btk (BTK) | Tec | TK | 6mny | A | B | 5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamide | Mouse | 11308 | |
| Btk (BTK) | Tec | TK | 6mny | A | A | 5-amino-1-[(3r)-1-cyanopiperidin-3-yl]-3-[4-(2,4-difluorophenoxy)phenyl]-1h-pyrazole-4-carboxamide | Mouse | 11307 | |
| Btk (BTK) | Tec | TK | 9ejx | A | | {(3r)-3-[4-amino-3-(4-phenoxyphenyl)-1h-pyrazolo[3,4-d]pyrimidin-1-yl]piperidin-1-yl}(cyclopropyl)methanone | Mouse | 16252 | |
| Tyro3 (TYRO3) | Axl | TK | 4feq | A | | 4-(cyclopentylamino)-n-[3-(2-oxopyrrolidin-1-yl)propyl]-2-{[2-(pyridin-4-yl)ethyl]amino}pyrimidine-5-carboxamide | Mouse | 5801 | |
| Tyro3 (TYRO3) | Axl | TK | 4ff8 | A | | 4-(cyclopentylamino)-2-[(2-methoxybenzyl)amino]-n-[3-(2-oxopyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide | Mouse | 5800 | |
| Epha4 (EphA4) | Eph | TK | 2y6m | A | B | - | Mouse | 5813 | |
| Epha4 (EphA4) | Eph | TK | 2y6o | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Mouse | 5811 | |