| AAK1 | NAK | Other | 5te0 | A | | methyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylate | Human | 7156 | |
| Aak1 (AAK1) | NAK | Other | 7rj6 | A | B | 5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Mouse | 14131 | |
| Aak1 (AAK1) | NAK | Other | 7rj7 | A | A | 2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrile | Mouse | 14128 | |
| Aak1 (AAK1) | NAK | Other | 7lvi | A | B | (2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamide | Mouse | 13821 | |
| Aak1 (AAK1) | NAK | Other | 7lvi | A | A | (2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamide | Mouse | 13822 | |
| Aak1 (AAK1) | NAK | Other | 7lvh | A | | n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamide | Mouse | 13820 | |
| AAK1 | NAK | Other | 9qb5 | A | | ~{n}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamide | Human | 16225 | |
| AAK1 | NAK | Other | 5l4q | B | A | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6680 | |
| AAK1 | NAK | Other | 5l4q | A | B | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6677 | |
| AAK1 | NAK | Other | 8gmd | A | | (5p)-3-({(8r)-5-[(4-aminopiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-[2-(propan-2-yl)-2h-tetrazol-5-yl]phenol | Human | 14844 | |
| AAK1 | NAK | Other | 8gmc | A | | 5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Human | 14843 | |
| AAK1 | NAK | Other | 5l4q | A | A | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6679 | |
| AAK1 | NAK | Other | 4wsq | B | B | k-252a | Human | 3835 | |
| AAK1 | NAK | Other | 4wsq | A | A | k-252a | Human | 3834 | |
| AAK1 | NAK | Other | 5l4q | B | B | ~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamide | Human | 6678 | |
| AAK1 | NAK | Other | 4wsq | B | A | k-252a | Human | 3833 | |
| AAK1 | NAK | Other | 4wsq | A | B | k-252a | Human | 3836 | |
| Aak1 (AAK1) | NAK | Other | 7rj8 | A | B | n-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamide | Mouse | 14127 | |
| Aak1 (AAK1) | NAK | Other | 7rj7 | A | B | 2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrile | Mouse | 14129 | |
| Aak1 (AAK1) | NAK | Other | 7rj8 | A | A | n-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamide | Mouse | 14130 | |
| Aak1 (AAK1) | NAK | Other | 7rj6 | A | A | 5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amine | Mouse | 14132 | |