Search results (21 entries covering 11 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
AAK1NAKOther5te0Amethyl (3z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1h-indole-6-carboxylateHuman7156
Aak1 (AAK1)NAKOther7rj6AB5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineMouse14131
Aak1 (AAK1)NAKOther7rj7AA2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrileMouse14128
Aak1 (AAK1)NAKOther7lviAB(2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamideMouse13821
Aak1 (AAK1)NAKOther7lviAA(2r,3r)-n-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-3-(propan-2-yl)piperidine-2-carboxamideMouse13822
Aak1 (AAK1)NAKOther7lvhAn-[3-methoxy-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse13820
AAK1NAKOther9qb5A~{n}-(phenylmethyl)-7,10-dioxa-13,17,18,21-tetrazatetracyclo[12.5.2.1^{2,6}.0^{17,20}]docosa-1(20),2(22),3,5,14(21),15,18-heptaene-5-carboxamideHuman16225
AAK1NAKOther5l4qBA~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6680
AAK1NAKOther5l4qAB~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6677
AAK1NAKOther8gmdA(5p)-3-({(8r)-5-[(4-aminopiperidin-1-yl)methyl]pyrrolo[2,1-f][1,2,4]triazin-4-yl}amino)-5-[2-(propan-2-yl)-2h-tetrazol-5-yl]phenolHuman14844
AAK1NAKOther8gmcA5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineHuman14843
AAK1NAKOther5l4qAA~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6679
AAK1NAKOther4wsqBBk-252aHuman3835
AAK1NAKOther4wsqAAk-252aHuman3834
AAK1NAKOther5l4qBB~{n}-[5-(4-cyanophenyl)-1~{h}-pyrrolo[2,3-b]pyridin-3-yl]pyridine-3-carboxamideHuman6678
AAK1NAKOther4wsqBAk-252aHuman3833
AAK1NAKOther4wsqABk-252aHuman3836
Aak1 (AAK1)NAKOther7rj8ABn-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse14127
Aak1 (AAK1)NAKOther7rj7AB2-[(1s)-1-amino-3-methylbutyl]-6-(pyridin-4-yl)quinoline-4-carbonitrileMouse14129
Aak1 (AAK1)NAKOther7rj8AAn-[3-(difluoromethoxy)-4-(1,3-oxazol-5-yl)phenyl]-d-leucinamideMouse14130
Aak1 (AAK1)NAKOther7rj6AA5-[(4-aminopiperidin-1-yl)methyl]-n-{3-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]phenyl}pyrrolo[2,1-f][1,2,4]triazin-4-amineMouse14132