| ABL1 | Abl | TK | 6xr6 | A | 18 | - | Human | 12912 | |
| ABL1 | Abl | TK | 8h7h | A | | 5-[3-(6-methoxyisoquinolin-7-yl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-~{n}-methyl-~{n}-prop-2-ynyl-pyridine-3-carboxamide | Human | 14666 | |
| ABL1 | Abl | TK | 6xr6 | A | 20 | - | Human | 12861 | |
| Abl1 (ABL1) | Abl | TK | 1m52 | A | | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Mouse | 5720 | |
| Abl1 (ABL1) | Abl | TK | 3oy3 | A | | 5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamide | Mouse | 5711 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | B | A | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5712 | |
| Abl1 (ABL1) | Abl | TK | 1fpu | B | | n-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamide | Mouse | 5705 | |
| Abl1 (ABL1) | Abl | TK | 1iep | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5703 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5723 | |
| Abl1 (ABL1) | Abl | TK | 3kf4 | A | | n-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amine | Mouse | 5717 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10610 | |
| Abl1 (ABL1) | Abl | TK | 3mss | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5730 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5734 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | A | B | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5729 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5722 | |
| Abl1 (ABL1) | Abl | TK | 3ik3 | B | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Mouse | 5739 | |
| Abl1 (ABL1) | Abl | TK | 3dk6 | A | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5725 | |
| Abl1 (ABL1) | Abl | TK | 1m52 | B | | 6-(2,6-dichloro-phenyl)-8-methyl-2-(3-methylsulfanyl-phenylamino)-8h-pyrido[2,3-d]pyrimidin-7-one | Mouse | 5715 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5733 | |
| ABL1 | Abl | TK | 6xr6 | A | 19 | - | Human | 12892 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10611 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10648 | |
| Abl1 (ABL1) | Abl | TK | 3oy3 | B | | 5-[(5-{[4-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}-3-(trifluoromethyl)phenyl]carbamoyl}-2-methylphenyl)ethynyl]-1-methyl-1h-imidazole-2-carboxamide | Mouse | 5738 | |
| ABL1 | Abl | TK | 6xrg | A | 1 | - | Human | 12890 | |
| ABL1 | Abl | TK | 6xrg | A | 9 | - | Human | 12891 | |
| ABL1 | Abl | TK | 6npu | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10942 | |
| ABL1 | Abl | TK | 6xrg | A | 4 | - | Human | 12899 | |
| Abl1 (ABL1) | Abl | TK | 3dk7 | B | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5714 | |
| Abl1 (ABL1) | Abl | TK | 2qoh | B | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5716 | |
| ABL1 | Abl | TK | 2g2f | B | | phosphothiophosphoric acid-adenylate ester | Human | 1079 | |
| ABL1 | Abl | TK | 4twp | A | | axitinib | Human | 1091 | |
| ABL1 | Abl | TK | 7cc2 | A | | [4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methyl-phenyl]boronic acid | Human | 13620 | |
| ABL1 | Abl | TK | 7dt2 | A | | [4-[5-[5-(dimethylcarbamoyl)pyridin-3-yl]-1h-pyrrolo[2,3-b]pyridin-3-yl]-2-methanoyl-5-methoxy-phenyl]boronic acid | Human | 13621 | |
| ABL1 | Abl | TK | 4zog | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 7043 | |
| ABL1 | Abl | TK | 5mo4 | A | B | nilotinib | Human | 7526 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5708 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10645 | |
| ABL1 | Abl | TK | 6xr6 | A | 11 | - | Human | 12872 | |
| ABL1 | Abl | TK | 6xr6 | A | 14 | - | Human | 12873 | |
| ABL1 | Abl | TK | 6bl8 | A | A | purvalanol b | Human | 9699 | |
| ABL1 | Abl | TK | 3pyy | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1049 | |
| ABL1 | Abl | TK | 2hz4 | A | | - | Human | 1059 | |
| ABL1 | Abl | TK | 4xey | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1094 | |
| ABL1 | Abl | TK | 6xrg | A | 3 | - | Human | 12893 | |
| ABL1 | Abl | TK | 6xr6 | A | 3 | - | Human | 12908 | |
| ABL1 | Abl | TK | 6xrg | A | 11 | - | Human | 12877 | |
| ABL1 | Abl | TK | 6xrg | A | 12 | - | Human | 12882 | |
| ABL1 | Abl | TK | 2hzi | A | A | 6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1102 | |
| ABL1 | Abl | TK | 4wa9 | A | | axitinib | Human | 1061 | |
| ABL1 | Abl | TK | 4yc8 | B | | 2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-n-(4-phenoxyphenyl)-1,3-thiazole-5-carboxamide | Human | 6420 | |
| ABL1 | Abl | TK | 6xr6 | A | 15 | - | Human | 12862 | |
| ABL1 | Abl | TK | 6xr6 | A | 1 | - | Human | 12905 | |
| ABL1 | Abl | TK | 2gqg | B | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1082 | |
| ABL1 | Abl | TK | 6xrg | A | 13 | - | Human | 12904 | |
| ABL1 | Abl | TK | 6xrg | A | 19 | - | Human | 12886 | |
| ABL1 | Abl | TK | 6xrg | A | 18 | - | Human | 12880 | |
| ABL1 | Abl | TK | 7w7x | A | | 5-[5-(dimethylcarbamoyl)pyridin-3-yl]-3-(5-fluorosulfonyloxy-2-methoxy-phenyl)-1h-pyrrolo[2,3-b]pyridine | Human | 14196 | |
| ABL1 | Abl | TK | 6xr7 | A | 15 | - | Human | 12913 | |
| ABL1 | Abl | TK | 6xr6 | A | 5 | - | Human | 12858 | |
| ABL1 | Abl | TK | 7w7y | A | | 5-[3-(5-methanoyl-2-methoxy-4-oxidanyl-phenyl)-1~{h}-pyrrolo[2,3-b]pyridin-5-yl]-~{n},~{n}-dimethyl-pyridine-3-carboxamide | Human | 14195 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5713 | |
| ABL1 | Abl | TK | 6xr7 | A | 5 | - | Human | 12857 | |
| ABL1 | Abl | TK | 2hz4 | B | | 1,2,3,4-tetrahydrogen-staurosporine | Human | 1058 | |
| ABL1 | Abl | TK | 2hz0 | B | B | 2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamide | Human | 1109 | |
| ABL1 | Abl | TK | 6xr7 | A | 16 | - | Human | 12859 | |
| ABL1 | Abl | TK | 3cs9 | B | B | nilotinib | Human | 1112 | |
| ABL1 | Abl | TK | 2hz0 | A | B | 2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamide | Human | 1083 | |
| ABL1 | Abl | TK | 6npv | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10949 | |
| ABL1 | Abl | TK | 2hyy | C | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1048 | |
| ABL1 | Abl | TK | 6npv | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10948 | |
| ABL1 | Abl | TK | 3pyy | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1098 | |
| ABL1 | Abl | TK | 3pyy | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1071 | |
| ABL1 | Abl | TK | 6bl8 | B | A | purvalanol b | Human | 9701 | |
| ABL1 | Abl | TK | 6xr7 | A | 8 | - | Human | 12863 | |
| ABL1 | Abl | TK | 6xrg | A | 8 | - | Human | 12864 | |
| ABL1 | Abl | TK | 3ue4 | B | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 1074 | |
| ABL1 | Abl | TK | 4wa9 | B | | axitinib | Human | 1063 | |
| ABL1 | Abl | TK | 3qrk | A | | (3s)-6-(3-tert-butyl-5-{[(2,3-dichlorophenyl)carbamoyl]amino}-1h-pyrazol-1-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid | Human | 1056 | |
| ABL1 | Abl | TK | 6xr7 | A | 14 | - | Human | 12865 | |
| ABL1 | Abl | TK | 6xr7 | A | 11 | - | Human | 12866 | |
| ABL1 | Abl | TK | 6xr7 | A | 1 | - | Human | 12867 | |
| ABL1 | Abl | TK | 6xrg | A | 7 | - | Human | 12868 | |
| ABL1 | Abl | TK | 6npe | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10947 | |
| ABL1 | Abl | TK | 2hzi | A | B | 6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1087 | |
| ABL1 | Abl | TK | 2g2f | A | | - | Human | 1097 | |
| ABL1 | Abl | TK | 6xr6 | A | 13 | - | Human | 12869 | |
| ABL1 | Abl | TK | 6xr7 | A | 17 | - | Human | 12870 | |
| ABL1 | Abl | TK | 4xey | B | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1100 | |
| ABL1 | Abl | TK | 6xr6 | A | 12 | - | Human | 12871 | |
| ABL1 | Abl | TK | 3qri | B | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1103 | |
| ABL1 | Abl | TK | 2hyy | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1078 | |
| ABL1 | Abl | TK | 2hzi | B | A | 6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1108 | |
| ABL1 | Abl | TK | 6xr6 | A | 17 | - | Human | 12874 | |
| ABL1 | Abl | TK | 6npv | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10950 | |
| ABL1 | Abl | TK | 3qri | A | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1051 | |
| ABL1 | Abl | TK | 6xrg | A | 14 | - | Human | 12875 | |
| ABL1 | Abl | TK | 6bl8 | B | B | purvalanol b | Human | 9700 | |
| ABL1 | Abl | TK | 2v7a | A | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 1088 | |
| ABL1 | Abl | TK | 6xr6 | A | 2 | - | Human | 12878 | |
| ABL1 | Abl | TK | 2g2i | B | | adenosine-5'-diphosphate | Human | 1075 | |
| ABL1 | Abl | TK | 2hiw | A | | 7-amino-1-methyl-3-(2-methyl-5-{[3-(trifluoromethyl)benzoyl]amino}phenyl)-2-oxo-2,3-dihydropyrimido[4,5-d]pyrimidin-1-ium | Human | 1069 | |
| ABL1 | Abl | TK | 6xr7 | A | 19 | - | Human | 12879 | |
| ABL1 | Abl | TK | 6npe | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10945 | |
| ABL1 | Abl | TK | 6xr6 | A | 7 | - | Human | 12881 | |
| ABL1 | Abl | TK | 3qrj | B | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1101 | |
| ABL1 | Abl | TK | 2hz4 | C | | - | Human | 1067 | |
| ABL1 | Abl | TK | 3cs9 | C | A | nilotinib | Human | 1046 | |
| ABL1 | Abl | TK | 2g1t | C | | - | Human | 1064 | |
| ABL1 | Abl | TK | 6xr7 | A | 2 | - | Human | 12883 | |
| ABL1 | Abl | TK | 2hyy | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1092 | |
| ABL1 | Abl | TK | 6xrg | A | 5 | - | Human | 12884 | |
| ABL1 | Abl | TK | 3ue4 | A | | 4-[(2,4-dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methylpiperazin-1-yl)propoxy]quinoline-3-carbonitrile | Human | 1057 | |
| ABL1 | Abl | TK | 6xr6 | A | 9 | - | Human | 12885 | |
| ABL1 | Abl | TK | 2f4j | A | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 1090 | |
| ABL1 | Abl | TK | 3pyy | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1062 | |
| ABL1 | Abl | TK | 3cs9 | C | B | nilotinib | Human | 1093 | |
| ABL1 | Abl | TK | 2g2h | B | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1089 | |
| ABL1 | Abl | TK | 3cs9 | D | B | nilotinib | Human | 1066 | |
| ABL1 | Abl | TK | 6xrg | A | 16 | - | Human | 12887 | |
| ABL1 | Abl | TK | 6xrg | A | 20 | - | Human | 12888 | |
| ABL1 | Abl | TK | 6xrg | A | 10 | - | Human | 12889 | |
| ABL1 | Abl | TK | 4twp | B | | axitinib | Human | 1081 | |
| ABL1 | Abl | TK | 2g1t | B | | - | Human | 1105 | |
| ABL1 | Abl | TK | 5hu9 | A | B | 4-[(4-methylpiperazin-1-yl)methyl]-n-(4-methyl-3-{[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]oxy}phenyl)-3-(trifluoromethyl)benzamide | Human | 6755 | |
| ABL1 | Abl | TK | 2hz0 | A | A | 2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamide | Human | 1052 | |
| ABL1 | Abl | TK | 6xr7 | A | 4 | - | Human | 12894 | |
| ABL1 | Abl | TK | 6xrg | A | 2 | - | Human | 12895 | |
| ABL1 | Abl | TK | 4zog | B | | cyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amide | Human | 7042 | |
| ABL1 | Abl | TK | 6xr6 | A | 6 | - | Human | 12896 | |
| ABL1 | Abl | TK | 3cs9 | A | A | nilotinib | Human | 1080 | |
| ABL1 | Abl | TK | 6xr6 | A | 4 | - | Human | 12898 | |
| ABL1 | Abl | TK | 5hu9 | A | A | 4-[(4-methylpiperazin-1-yl)methyl]-n-(4-methyl-3-{[1-(pyridin-3-ylcarbonyl)piperidin-4-yl]oxy}phenyl)-3-(trifluoromethyl)benzamide | Human | 6754 | |
| ABL1 | Abl | TK | 2e2b | A | | n-[3-(4,5'-bipyrimidin-2-ylamino)-4-methylphenyl]-4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-3-(trifluoromethyl)benzamide | Human | 1054 | |
| ABL1 | Abl | TK | 6npu | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10944 | |
| ABL1 | Abl | TK | 5mo4 | A | A | nilotinib | Human | 7527 | |
| ABL1 | Abl | TK | 6xr7 | A | 3 | - | Human | 12900 | |
| ABL1 | Abl | TK | 2hyy | D | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 1068 | |
| ABL1 | Abl | TK | 6xr6 | A | 10 | - | Human | 12901 | |
| ABL1 | Abl | TK | 7n9g | A | | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 14197 | |
| ABL1 | Abl | TK | 4yc8 | A | | 2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-n-(4-phenoxyphenyl)-1,3-thiazole-5-carboxamide | Human | 6419 | |
| ABL1 | Abl | TK | 3qrj | A | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1099 | |
| ABL1 | Abl | TK | 6xr6 | A | 16 | - | Human | 12902 | |
| ABL1 | Abl | TK | 6xr7 | A | 10 | - | Human | 12903 | |
| ABL1 | Abl | TK | 3qrj | A | A | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1085 | |
| ABL1 | Abl | TK | 6npe | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10943 | |
| ABL1 | Abl | TK | 2gqg | A | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1060 | |
| ABL1 | Abl | TK | 6bl8 | A | B | purvalanol b | Human | 9698 | |
| ABL1 | Abl | TK | 6xr6 | A | 8 | - | Human | 12906 | |
| ABL1 | Abl | TK | 6npv | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10951 | |
| ABL1 | Abl | TK | 6xr7 | A | 7 | - | Human | 12907 | |
| ABL1 | Abl | TK | 3qrj | B | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1070 | |
| ABL1 | Abl | TK | 6xr7 | A | 18 | - | Human | 12909 | |
| ABL1 | Abl | TK | 2g2i | A | | adenosine-5'-diphosphate | Human | 1111 | |
| ABL1 | Abl | TK | 2gqg | B | A | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1084 | |
| ABL1 | Abl | TK | 1opl | B | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1086 | |
| ABL1 | Abl | TK | 2g1t | A | | - | Human | 1045 | |
| ABL1 | Abl | TK | 2hzi | B | B | 6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1055 | |
| ABL1 | Abl | TK | 8h7f | A | | 1-[6-(6-methoxyisoquinolin-7-yl)-1,3-benzothiazol-2-yl]-3-(2-oxidanylideneethyl)urea | Human | 14632 | |
| ABL1 | Abl | TK | 6npe | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Human | 10946 | |
| ABL1 | Abl | TK | 6xr7 | A | 13 | - | Human | 12910 | |
| ABL1 | Abl | TK | 6xrg | A | 15 | - | Human | 12911 | |
| ABL1 | Abl | TK | 3cs9 | A | B | nilotinib | Human | 1107 | |
| ABL1 | Abl | TK | 1opl | A | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1104 | |
| ABL1 | Abl | TK | 2fo0 | A | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1073 | |
| ABL1 | Abl | TK | 6xr7 | A | 20 | - | Human | 12914 | |
| ABL1 | Abl | TK | 6xr7 | A | 9 | - | Human | 12915 | |
| ABL1 | Abl | TK | 3cs9 | B | A | nilotinib | Human | 1050 | |
| ABL1 | Abl | TK | 6xrg | A | 17 | - | Human | 12916 | |
| ABL1 | Abl | TK | 3qri | A | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1047 | |
| ABL1 | Abl | TK | 3qri | B | B | 4-[4-({[3-tert-butyl-1-(quinolin-6-yl)-1h-pyrazol-5-yl]carbamoyl}amino)-3-fluorophenoxy]-n-methylpyridine-2-carboxamide | Human | 1076 | |
| ABL1 | Abl | TK | 2hz0 | B | A | 2-{[(6-oxo-1,6-dihydropyridin-3-yl)methyl]amino}-n-[4-propyl-3-(trifluoromethyl)phenyl]benzamide | Human | 1095 | |
| ABL1 | Abl | TK | 8ssn | A | | 6,7-dimethoxy-n-(4-phenoxyphenyl)quinazolin-4-amine | Human | 14878 | |
| ABL1 | Abl | TK | 2gqg | A | B | n-(2-chloro-6-methylphenyl)-2-({6-[4-(2-hydroxyethyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}amino)-1,3-thiazole-5-carboxamide | Human | 1053 | |
| Abl1 (ABL1) | Abl | TK | 1opj | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5732 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | B | B | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5737 | |
| Abl1 (ABL1) | Abl | TK | 3kf4 | B | | n-[4-(dimethylphosphoryl)phenyl]-9-[(e)-2-(5-methyl-1h-indazol-4-yl)ethenyl]-9h-purin-6-amine | Mouse | 5741 | |
| Abl1 (ABL1) | Abl | TK | 3mss | C | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5719 | |
| Abl1 (ABL1) | Abl | TK | 3ik3 | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Mouse | 5731 | |
| Abl1 (ABL1) | Abl | TK | 3kfa | A | | 3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamide | Mouse | 5742 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10608 | |
| Abl1 (ABL1) | Abl | TK | 1iep | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5727 | |
| Abl1 (ABL1) | Abl | TK | 3dk6 | B | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5718 | |
| Abl1 (ABL1) | Abl | TK | 1opj | B | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5736 | |
| Abl1 (ABL1) | Abl | TK | 6hd6 | A | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10609 | |
| Abl1 (ABL1) | Abl | TK | 1opk | A | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Mouse | 5709 | |
| Abl1 (ABL1) | Abl | TK | 3dk7 | A | | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5704 | |
| Abl1 (ABL1) | Abl | TK | 2z60 | A | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5735 | |
| Abl1 (ABL1) | Abl | TK | 3ms9 | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5706 | |
| Abl1 (ABL1) | Abl | TK | 3oxz | A | | 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide | Mouse | 5721 | |
| Abl1 (ABL1) | Abl | TK | 3mss | D | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5702 | |
| Abl1 (ABL1) | Abl | TK | 3dk3 | A | A | 2-amino-5-[3-(1-ethyl-1h-pyrazol-5-yl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylbenzamide | Mouse | 5726 | |
| Abl1 (ABL1) | Abl | TK | 2qoh | A | | 5-[3-(2-methoxyphenyl)-1h-pyrrolo[2,3-b]pyridin-5-yl]-n,n-dimethylpyridine-3-carboxamide | Mouse | 5707 | |
| Abl1 (ABL1) | Abl | TK | 1fpu | A | | n-[4-methyl-3-[[4-(3-pyridinyl)-2-pyrimidinyl]amino]phenyl]-3-pyridinecarboxamide | Mouse | 5728 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | B | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10646 | |
| Abl1 (ABL1) | Abl | TK | 2hzn | A | | 1-[4-(pyridin-4-yloxy)phenyl]-3-[3-(trifluoromethyl)phenyl]urea | Mouse | 5701 | |
| Abl1 (ABL1) | Abl | TK | 6hd4 | A | B | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 10647 | |
| Abl1 (ABL1) | Abl | TK | 3k5v | B | A | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5710 | |
| Abl1 (ABL1) | Abl | TK | 3kfa | B | | 3-{(e)-2-[6-(cyclopropylamino)-9h-purin-9-yl]ethenyl}-4-methyl-n-[3-(4-methyl-1h-imidazol-1-yl)-5-(trifluoromethyl)phenyl]benzamide | Mouse | 5740 | |
| Abl1 (ABL1) | Abl | TK | 3mss | A | | 4-(4-methyl-piperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl-pyrimidin-2-ylamino)-phenyl]-benzamide | Mouse | 5724 | |
| ABL1 | Abl | TK | 6xr7 | A | 12 | - | Human | 12860 | |
| ABL1 | Abl | TK | 2e2b | B | | n-[3-(4,5'-bipyrimidin-2-ylamino)-4-methylphenyl]-4-{[(3s)-3-(dimethylamino)pyrrolidin-1-yl]methyl}-3-(trifluoromethyl)benzamide | Human | 1065 | |
| ABL1 | Abl | TK | 3cs9 | D | A | nilotinib | Human | 1077 | |
| ABL1 | Abl | TK | 6xrg | A | 6 | - | Human | 12876 | |
| ABL1 | Abl | TK | 2g2h | A | | 6-(2,6-dichlorophenyl)-2-{[3-(hydroxymethyl)phenyl]amino}-8-methylpyrido[2,3-d]pyrimidin-7(8h)-one | Human | 1106 | |
| ABL1 | Abl | TK | 2g1t | D | | - | Human | 1096 | |
| ABL1 | Abl | TK | 6xr7 | A | 6 | - | Human | 12897 | |
| ABL1 | Abl | TK | 2hiw | B | | 7-amino-1-methyl-3-(2-methyl-5-{[3-(trifluoromethyl)benzoyl]amino}phenyl)-2-oxo-2,3-dihydropyrimido[4,5-d]pyrimidin-1-ium | Human | 1110 | |
| ABL1 | Abl | TK | 2v7a | B | | n-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamide | Human | 1072 | |
