Search results (305 entries covering 209 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
AURKA (AurA)AurOther8c1hAAadenosine-5'-diphosphateHuman15147
AURKA (AurA)AurOther4uzdAethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHuman2013
AURKA (AurA)AurOther2wtvAA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2056
AURKA (AurA)AurOther6c2tAB(2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acidHuman10863
Aurka (AurA)AUROther3d14AA1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouse5781
AURKA (AurA)AurOther3w2cE2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman1953
AURKA (AurA)AurOther3w10A1-(3-methoxyphenyl)-n-(5-methyl-1h-pyrazol-3-yl)isoquinolin-3-amineHuman2068
AURKA (AurA)AurOther4uynAethyl (9s)-9-[5-(1h-benzimidazol-2-ylsulfanyl)furan-2-yl]-8-hydroxy-5,6,7,9-tetrahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHuman2002
AURKA (AurA)AurOther2dwbAphosphoaminophosphonic acid-adenylate esterHuman2035
AURKA (AurA)AurOther5os5ABadenosine-5'-diphosphateHuman8629
AURKA (AurA)AurOther3w2cC2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman2021
AURKA (AurA)AurOther6vpmABadenosine monophosphateHuman12658
AURKA (AurA)AurOther2c6eAn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHuman1989
AURKA (AurA)AurOther5dn3ABadenosine-5'-triphosphateHuman6818
AURKA (AurA)AurOther6vplBBphosphoaminophosphonic acid-adenylate esterHuman12668
AURKA (AurA)AurOther2wtvBA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2037
AURKA (AurA)AurOther4dedA2-({2-[(4-carbamoylphenyl)amino]pyrimidin-4-yl}amino)benzamideHuman2043
AURKA (AurA)AurOther4j8nC-Human2007
AURKA (AurA)AurOther3w2cG2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman2026
AURKA (AurA)AurOther3m11A1-(4-{2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHuman2036
AURKA (AurA)AurOther3mygA2-{ethyl[(5-{[6-methyl-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-yl]amino}isothiazol-3-yl)methyl]amino}-2-methylpropan-1-olHuman2065
AURKA (AurA)AurOther3e5aAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman2006
Aurka (AurA)AUROther3dj7AA1-(5-{2-[(6-amino-5-bromopyrimidin-4-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouse5780
Aurka (AurA)AUROther3d14AB1-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}-3-[3-(trifluoromethyl)phenyl]ureaMouse5775
AURKA (AurA)AurOther3fdnAn-[3-(acetylamino)phenyl]-5-{(2e)-2-[(4-methoxyphenyl)methylidene]hydrazino}-3-methyl-1h-pyrazole-4-carboxamideHuman1973
AURKA (AurA)AurOther8c1iABadenosine-5'-diphosphateHuman15139
AURKA (AurA)AurOther8c1dABadenosine-5'-diphosphateHuman15138
AURKA (AurA)AurOther6z4yAB6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12307
AURKA (AurA)AurOther2xneA3-chloro-n-(4-morpholin-4-ylphenyl)-6-pyridin-3-ylimidazo[1,2-a]pyrazin-8-amineHuman7221
AURKA (AurA)AurOther6vpiABphosphoaminophosphonic acid-adenylate esterHuman12669
AURKA (AurA)AurOther5os5AAadenosine-5'-diphosphateHuman8647
AURKA (AurA)AurOther2bmcA(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2015
AURKA (AurA)AurOther6c83Aphosphomethylphosphonic acid adenylate esterHuman10934
AURKA (AurA)AurOther5l8jABadenosine-5'-diphosphateHuman6812
AURKA (AurA)AurOther3w16A4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-oneHuman2012
AURKA (AurA)AurOther3uohA4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2077
AURKA (AurA)AurOther4j8nB-Human2061
AURKA (AurA)AurOther8c14AAadenosine-5'-diphosphateHuman15143
AURKA (AurA)AurOther8c1gAadenosine-5'-diphosphateHuman15148
AURKA (AurA)AurOther5orvAadenosine-5'-diphosphateHuman8643
AURKA (AurA)AurOther5dpvAB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6826
AURKA (AurA)AurOther8c1kAadenosine-5'-diphosphateHuman15146
AURKA (AurA)AurOther9qvzABadenosine-5'-diphosphateHuman15482
AURKA (AurA)AurOther9rvkBAadenosine-5'-diphosphateHuman15483
AURKA (AurA)AurOther9kdsA-Human15484
AURKA (AurA)AurOther9qvzAAadenosine-5'-diphosphateHuman15485
AURKA (AurA)AurOther9s7tAadenosine-5'-diphosphateHuman15486
AURKA (AurA)AurOther5dt0AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6803
AURKA (AurA)AurOther9ks6A-Human15487
AURKA (AurA)AurOther5dnrAAadenosine-5'-triphosphateHuman6810
AURKA (AurA)AurOther4deeAadenosine-5'-diphosphateHuman1952
AURKA (AurA)AurOther5orrAadenosine-5'-diphosphateHuman8636
AURKA (AurA)AurOther6hjkA(~{e})-~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-but-2-enamideHuman10411
AURKA (AurA)AurOther4ztqA(2z,5z)-2-[(4-ethylphenyl)imino]-3-(2-methoxyethyl)-5-(pyridin-4-ylmethylidene)-1,3-thiazolidin-4-oneHuman6804
AURKA (AurA)AurOther1ol6Aadenosine-5'-triphosphateHuman2081
AURKA (AurA)AurOther5odtABadenosine-5'-diphosphateHuman9736
AURKA (AurA)AurOther5orwAadenosine-5'-diphosphateHuman8631
AURKA (AurA)AurOther2w1eA4-[(2-{4-[(phenylcarbamoyl)amino]-1h-pyrazol-3-yl}-1h-benzimidazol-5-yl)methyl]morpholin-4-iumHuman2038
AURKA (AurA)AurOther2j50An-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman2001
AURKA (AurA)AurOther8sspAAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14868
AURKA (AurA)AurOther5dr2Aadenosine-5'-triphosphateHuman6825
AURKA (AurA)AurOther3uo5A4-{[4-(phenylamino)pyrimidin-2-yl]amino}benzoic acidHuman2045
AURKA (AurA)AurOther2w1cA4-{[2-(4-{[(4-fluorophenyl)carbonyl]amino}-1h-pyrazol-3-yl)-1h-benzimidazol-6-yl]methyl}morpholin-4-iumHuman2027
AURKA (AurA)AurOther5os3Aadenosine-5'-diphosphateHuman8637
AURKA (AurA)AurOther5dr6AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6811
AURKA (AurA)AurOther3h0zC4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHuman2063
AURKA (AurA)AurOther2j4zB4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHuman1990
AURKA (AurA)AurOther3vapA3-(1-{2-[(3-fluoropyridinium-4-yl)amino]-2-oxoethyl}-1h-pyrazol-4-yl)-6-methyl-8-[(3-{[(1r,3r)-3-methylpiperidinium-1-yl]methyl}-1,2-thiazol-5-yl)amino]imidazo[1,2-a]pyrazin-1-iumHuman2029
AURKA (AurA)AurOther6vpmAAadenosine monophosphateHuman12661
AURKA (AurA)AurOther5osfAadenosine-5'-diphosphateHuman8640
AURKA (AurA)AurOther5oneAB4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamideHuman8370
AURKA (AurA)AurOther7o2vA1-[[3,4-bis(fluoranyl)phenyl]methyl]-~{n}-[(1~{r})-2-[[(3~{e})-3-(1~{h}-imidazol-5-ylmethylidene)-2-oxidanylidene-1~{h}-indol-5-yl]amino]-2-oxidanylidene-1-phenyl-ethyl]-6-methyl-2-oxidanylidene-pyridine-3-carboxamideHuman13947
AURKA (AurA)AurOther4dhfB7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman1982
AURKA (AurA)AurOther5drdAadenosine-5'-triphosphateHuman6823
AURKA (AurA)AurOther6hjjAA~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamideHuman10410
AURKA (AurA)AurOther1muoAadenosineHuman2062
AURKA (AurA)AurOther5l8lABadenosine-5'-diphosphateHuman6824
AURKA (AurA)AurOther3cohA8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-oneHuman1963
AURKA (AurA)AurOther6vpjABphosphoaminophosphonic acid-adenylate esterHuman12654
AURKA (AurA)AurOther5aadA7-(1-benzyl-1h-pyrazol-4-yl)-6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridineHuman6011
AURKA (AurA)AurOther2bmcD(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman1984
AURKA (AurA)AurOther7ayhA7-[2-[(4-methoxyphenyl)amino]pyrimidin-4-yl]-1,3,4,5-tetrahydro-1-benzazepin-2-oneHuman13228
AURKA (AurA)AurOther2x6dAA6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridineHuman1978
AURKA (AurA)AurOther3h0zA4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHuman1970
AURKA (AurA)AurOther9s0wAadenosine-5'-diphosphateHuman15488
AURKA (AurA)AurOther6vphABdithiane diolHuman12655
AURKA (AurA)AurOther8jmxA5-(4-morpholin-4-yl-7h-pyrrolo[2,3-d]pyrimidin-5-yl)-2-oxidanyl-benzaldehydeHuman14864
AURKA (AurA)AurOther6vpiAAphosphoaminophosphonic acid-adenylate esterHuman12656
AURKA (AurA)AurOther5ew9AB4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHuman6360
AURKA (AurA)AurOther3uolBn~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamineHuman2051
AURKA (AurA)AurOther9suyAadenosine-5'-diphosphateHuman15489
AURKA (AurA)AurOther8sspABn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14865
AURKA (AurA)AurOther5odtAAadenosine-5'-diphosphateHuman9738
AURKA (AurA)AurOther2x6dAB6-bromo-7-[4-(4-chlorobenzyl)piperazin-1-yl]-2-[4-(morpholin-4-ylmethyl)phenyl]-3h-imidazo[4,5-b]pyridineHuman1975
AURKA (AurA)AurOther5l8kABadenosine-5'-diphosphateHuman6813
AURKA (AurA)AurOther3o50Bn-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHuman2067
AURKA (AurA)AurOther9s0kBadenosine-5'-diphosphateHuman15490
AURKA (AurA)AurOther7ztlABadenosine-5'-diphosphateHuman14581
AURKA (AurA)AurOther5orzAAadenosine-5'-diphosphateHuman8639
AURKA (AurA)AurOther3up7A2-({2-[(4-carboxyphenyl)amino]pyrimidin-4-yl}amino)benzoic acidHuman2025
AURKA (AurA)AurOther5aaeA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-5-methylisoxazoleHuman6012
AURKA (AurA)AurOther5orzABadenosine-5'-diphosphateHuman8650
AURKA (AurA)AurOther9rvkBBadenosine-5'-diphosphateHuman15491
AURKA (AurA)AurOther4jajAbenzo[c][1,8]naphthyridin-6(5h)-oneHuman2040
AURKA (AurA)AurOther4j8nA-Human2028
AURKA (AurA)AurOther5ew9AA4-(3-chloranyl-2-fluoranyl-phenoxy)-1-[[6-(1,3-thiazol-2-ylamino)pyridin-2-yl]methyl]cyclohexane-1-carboxylic acidHuman6359
AURKA (AurA)AurOther9sv0BAadenosine-5'-diphosphateHuman15492
AURKA (AurA)AurOther4deaA4,4'-(pyrimidine-2,4-diyldiimino)dibenzoic acidHuman2064
AURKA (AurA)AurOther3nrmAn-(3-methylisothiazol-5-yl)-3-(1h-pyrazol-4-yl)imidazo[1,2-a]pyrazin-8-amineHuman2052
AURKA (AurA)AurOther4uzdBethyl (9s)-9-[3-(1h-benzimidazol-2-yloxy)phenyl]-8-oxo-4,5,6,7,8,9-hexahydro-2h-pyrrolo[3,4-b]quinoline-3-carboxylateHuman1968
AURKA (AurA)AurOther6cpeAA-Human10036
AURKA (AurA)AurOther3unzA4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1972
AURKA (AurA)AurOther8c1hABadenosine-5'-diphosphateHuman15142
AURKA (AurA)AurOther9s1gBadenosine-5'-diphosphateHuman15494
AURKA (AurA)AurOther8c1eAadenosine-5'-triphosphateHuman15145
AURKA (AurA)AurOther3unzB4-({4-[(2-fluorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2049
AURKA (AurA)AurOther4b0gAA6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridineHuman2082
AURKA (AurA)AurOther4c3pAphosphomethylphosphonic acid adenylate esterHuman2018
AURKA (AurA)AurOther6vplAAphosphoaminophosphonic acid-adenylate esterHuman12662
AURKA (AurA)AurOther8of5Aadenosine-5'-diphosphateHuman15218
AURKA (AurA)AurOther9sv0BBadenosine-5'-diphosphateHuman15496
AURKA (AurA)AurOther3w18A2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamideHuman1961
AURKA (AurA)AurOther2wtvCB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2016
AURKA (AurA)AurOther5dosAadenosine-5'-triphosphateHuman6807
AURKA (AurA)AurOther5os1ABadenosine-5'-diphosphateHuman8630
AURKA (AurA)AurOther3uo6A4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1985
AURKA (AurA)AurOther6z4yAA6-(2-methoxyethoxy)-11-methyl-8-oxa-2,11,15,19,21,23-hexazatetracyclo[15.6.1.13,7.020,24]pentacosa-1(23),3(25),4,6,17,20(24),21-heptaen-10-one Human12306
AURKA (AurA)AurOther5oneAA4-(propanoylamino)-~{n}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamideHuman8371
AURKA (AurA)AurOther2bmcF(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman1993
AURKA (AurA)AurOther3up2A4-[(4-{[2-(trifluoromethoxy)phenyl]amino}pyrimidin-2-yl)amino]benzoic acidHuman2005
AURKA (AurA)AurOther3w2cA2-{4-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-1-yl}-n-(3-methylbutyl)acetamideHuman2066
AURKA (AurA)AurOther5oryAadenosine-5'-diphosphateHuman8627
AURKA (AurA)AurOther2wtvAB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman1997
AURKA (AurA)AurOther3w18B2-{3-[3-(1h-benzimidazol-2-yl)-1h-indazol-6-yl]-1h-pyrazol-5-yl}-n-(3-fluorophenyl)acetamideHuman1967
AURKA (AurA)AurOther9bzgAA7-cyclopentyl-n,n-dimethyl-2-[4-(methylcarbamoyl)anilino]-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman15497
AURKA (AurA)AurOther7ficAA6-[(5-cyclopropyl-1~{h}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{n}-prop-2-ynyl-pyrimidine-4-carboxamideHuman14234
AURKA (AurA)AurOther4debA4-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzamideHuman1996
AURKA (AurA)AurOther5dnrABadenosine-5'-triphosphateHuman6809
AURKA (AurA)AurOther6c2tAA(2s,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-2-methyl-4-({3-[(1,3-thiazol-2-yl)amino]isoquinolin-1-yl}methyl)piperidine-4-carboxylic acidHuman10866
AURKA (AurA)AurOther5osdAadenosine-5'-diphosphateHuman8634
AURKA (AurA)AurOther6cpgD1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10034
AURKA (AurA)AurOther4j8mA1-[4-[[4-[(5-cyclopentyl-1h-pyrazol-3-yl)amino]pyrimidin-2-yl]amino]phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHuman2020
AURKA (AurA)AurOther5objAadenosine-5'-triphosphateHuman8305
AURKA (AurA)AurOther3o50An-{3-methyl-4-[(3-pyrimidin-4-ylpyridin-2-yl)oxy]phenyl}-3-(trifluoromethyl)benzamideHuman1958
AURKA (AurA)AurOther3uodA4-[(4-{[2-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]benzoic acidHuman1980
AURKA (AurA)AurOther2w1gA2-{4-[(cyclopropylcarbamoyl)amino]-1h-pyrazol-3-yl}-6-(morpholin-4-ium-4-ylmethyl)-1h-3,1-benzimidazol-3-iumHuman1962
AURKA (AurA)AurOther5orxAadenosine-5'-diphosphateHuman8644
AURKA (AurA)AurOther2x6eA6-bromo-7-{4-[(5-methylisoxazol-3-yl)methyl]piperazin-1-yl}-2-[4-(4-methylpiperazin-1-yl)phenyl]-1h-imidazo[4,5-b]pyridineHuman2079
AURKA (AurA)AurOther7ayiA7-(2-phenylazanylpyrimidin-4-yl)-1,3,4,5-tetrahydro-1-benzazepin-2-oneHuman13229
AURKA (AurA)AurOther2c6eBn-{5-[(7-{[(2s)-2-hydroxy-3-piperidin-1-ylpropyl]oxy}-6-methoxyquinazolin-4-yl)amino]pyrimidin-2-yl}benzamideHuman2046
AURKA (AurA)AurOther3uojB4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1979
AURKA (AurA)AurOther4c3pDphosphomethylphosphonic acid adenylate esterHuman2030
AURKA (AurA)AurOther8ssoACn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14863
AURKA (AurA)AurOther8ssoABn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14867
AURKA (AurA)AurOther4j8nD-Human1995
AURKA (AurA)AurOther3uo6B4-({4-[(2-chlorophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman1960
AURKA (AurA)AurOther4byiA(s)-n-((1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)methyl)acetamideHuman1992
AURKA (AurA)AurOther5aafA3-((4-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)-1h-pyrazol-1-yl)methyl)-n,n-dimethylbenzamideHuman6013
AURKA (AurA)AurOther5l8lAAadenosine-5'-diphosphateHuman6822
AURKA (AurA)AurOther3r21ABn-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHuman2033
AURKA (AurA)AurOther5os4Aadenosine-5'-diphosphateHuman8652
AURKA (AurA)AurOther2wtvBB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2057
AURKA (AurA)AurOther5g1xAAadenosine-5'-diphosphateHuman7267
AURKA (AurA)AurOther5orpAadenosine-5'-diphosphateHuman8648
AURKA (AurA)AurOther5g15ABphosphomethylphosphonic acid adenylate esterHuman9739
AURKA (AurA)AurOther5os2ABadenosine-5'-diphosphateHuman8633
AURKA (AurA)AurOther3k5uA2-[(5,6-diphenylfuro[2,3-d]pyrimidin-4-yl)amino]ethanolHuman2031
AURKA (AurA)AurOther5dpvAA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6808
AURKA (AurA)AurOther6r4cAadenosine-5'-diphosphateHuman11135
AURKA (AurA)AurOther5dt0AA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6806
AURKA (AurA)AurOther3p9jA4-[(5-methyl-1h-pyrazol-3-yl)amino]-2-phenylphthalazin-1(2h)-oneHuman2003
AURKA (AurA)AurOther5dt4Aadenosine-5'-triphosphateHuman6815
AURKA (AurA)AurOther6vpmBAadenosine monophosphateHuman12660
AURKA (AurA)AurOther8c1mAadenosine-5'-diphosphateHuman15137
AURKA (AurA)AurOther8c1fAAadenosine-5'-diphosphateHuman15140
AURKA (AurA)AurOther8c14ABadenosine-5'-diphosphateHuman15150
AURKA (AurA)AurOther8c15ABadenosine-5'-diphosphateHuman15151
AURKA (AurA)AurOther8c1dAAadenosine-5'-diphosphateHuman15152
AURKA (AurA)AurOther3uojA4-({4-[(2-cyanophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2042
AURKA (AurA)AurOther8pr7Aadenosine-5'-diphosphateHuman15292
AURKA (AurA)AurOther5zanA7-(4-methylpiperazin-1-yl)-n-(5-methyl-1h-pyrazol-3-yl)-2-[(e)-2-phenylethenyl]quinazolin-4-amineHuman10898
AURKA (AurA)AurOther3qbnA5-chloro-n~4~-cyclopropyl-n~2~-[4-(2-methoxyethoxy)phenyl]pyrimidine-2,4-diamineHuman2032
AURKA (AurA)AurOther8c1fABadenosine-5'-diphosphateHuman15149
AURKA (AurA)AurOther4cegAadenosine-5'-diphosphateHuman2073
AURKA (AurA)AurOther4c3rAphosphomethylphosphonic acid adenylate esterHuman2058
AURKA (AurA)AurOther8c15AAadenosine-5'-diphosphateHuman15141
AURKA (AurA)AurOther1mq4Aadenosine-5'-diphosphateHuman1977
AURKA (AurA)AurOther4jaiAn-{4-[(6-oxo-5,6-dihydrobenzo[c][1,8]naphthyridin-1-yl)amino]phenyl}benzamideHuman1999
AURKA (AurA)AurOther5os2AAadenosine-5'-diphosphateHuman8635
AURKA (AurA)AurOther5orsAadenosine-5'-diphosphateHuman8646
AURKA (AurA)AurOther2c6dABphosphoaminophosphonic acid-adenylate esterHuman1981
AURKA (AurA)AurOther1ol5Aadenosine-5'-diphosphateHuman2080
AURKA (AurA)AurOther4jbqAcyclopropanecarboxylic acid {4-[4-(4-methyl-piperazin-1-yl)-6-(5-methyl-2h-pyrazol-3-ylamino)-pyrimidin-2-ylsulfanyl]-phenyl}-amideHuman1957
AURKA (AurA)AurOther4zs0A5-hydroxy-1'h-1,2'-bibenzimidazol-2(3h)-oneHuman6801
AURKA (AurA)AurOther2wtwA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman1956
AURKA (AurA)AurOther4jboA1-(4-{2-[(6-{4-[2-(dimethylamino)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHuman2072
AURKA (AurA)AurOther1ol7Aadenosine-5'-diphosphateHuman2014
AURKA (AurA)AurOther3lauAn-[6-(4-hydroxyphenyl)-1h-indazol-3-yl]butanamideHuman1971
AURKA (AurA)AurOther5dr6AB4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6805
AURKA (AurA)AurOther4jbpA1-(4-{2-[(6-{4-[2-(4-hydroxypiperidin-1-yl)ethoxy]phenyl}furo[2,3-d]pyrimidin-4-yl)amino]ethyl}phenyl)-3-phenylureaHuman2041
AURKA (AurA)AurOther4o0sAadenosineHuman2039
AURKA (AurA)AurOther5lxmAAadenosine-5'-diphosphateHuman7142
AURKA (AurA)AurOther6c2rAA(2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acidHuman10864
AURKA (AurA)AurOther6vpjAAphosphoaminophosphonic acid-adenylate esterHuman12657
AURKA (AurA)AurOther8ssoAAn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman14866
AURKA (AurA)AurOther5os0Aadenosine-5'-diphosphateHuman8632
AURKA (AurA)AurOther8jf4A2-[4-[4-[bis(oxidanylidene)-$l^5-sulfanyl]oxyphenyl]carbonylpiperazin-1-yl]-6-[(5-cyclopropyl-1h-pyrazol-3-yl)amino]-n-prop-2-ynyl-pyrimidine-4-carboxamideHuman15217
AURKA (AurA)AurOther5os6Aadenosine-5'-diphosphateHuman8651
AURKA (AurA)AurOther6hjjAB~{n}-[4-(4-azanyl-1-propan-2-yl-pyrazolo[3,4-d]pyrimidin-3-yl)-3-methyl-phenyl]-4-[4-fluoranyl-3-(trifluoromethyl)phenyl]-4-oxidanylidene-butanamideHuman10412
AURKA (AurA)AurOther2xngABn-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamideHuman2083
AURKA (AurA)AurOther5dn3AAadenosine-5'-triphosphateHuman6802
AURKA (AurA)AurOther2w1fAn-[3-(1h-benzimidazol-2-yl)-1h-pyrazol-4-yl]benzamideHuman2055
AURKA (AurA)AurOther4byjA(s)-n-(1-(6-chloro-2-(1,3-dimethyl-1h-pyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl)pyrrolidin-3-yl)acetamideHuman1969
AURKA (AurA)AurOther5l8kAAadenosine-5'-diphosphateHuman6819
AURKA (AurA)AurOther3o51An-[4-({3-[5-fluoro-2-(methylideneamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-2-(phenylamino)benzamideHuman1974
AURKA (AurA)AurOther5g15AAphosphomethylphosphonic acid adenylate esterHuman9737
AURKA (AurA)AurOther3uolAn~4~-(2-chlorophenyl)-n~2~-[4-(1h-tetrazol-5-yl)phenyl]pyrimidine-2,4-diamineHuman2004
AURKA (AurA)AurOther5os1AAadenosine-5'-diphosphateHuman8628
AURKA (AurA)AurOther3h10D9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHuman2059
AURKA (AurA)AurOther6r4dAadenosine-5'-diphosphateHuman11132
AURKA (AurA)AurOther4dhfA7-cyclopentyl-2-({1-methyl-5-[(4-methylpiperazin-1-yl)carbonyl]-1h-pyrrol-3-yl}amino)-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman1964
AURKA (AurA)AurOther5ortAadenosine-5'-diphosphateHuman8638
AURKA (AurA)AurOther3h0zB4-{[2-({4-[2-(4-acetylpiperazin-1-yl)-2-oxoethyl]phenyl}amino)-5-fluoropyrimidin-4-yl]amino}-n-(2-chlorophenyl)benzamideHuman1986
AURKA (AurA)AurOther6vpgAAphosphoaminophosphonic acid-adenylate esterHuman12659
AURKA (AurA)AurOther2bmcE(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2069
AURKA (AurA)AurOther2j50Bn-[(3e)-5-[(2r)-2-methoxy-2-phenylacetyl]pyrrolo[3,4-c]pyrazol-3(5h)-ylidene]-4-(4-methylpiperazin-1-yl)benzamideHuman2050
AURKA (AurA)AurOther4b0gAB6-bromo-2-(1-methyl-1h-imidazol-5-yl)-7-{4-[(5-methyl-1,2-oxazol-3-yl)methyl]piperazin-1-yl}-1h-imidazo[4,5-b]pyridineHuman2070
AURKA (AurA)AurOther4prjAn-[1-(3-cyanobenzyl)-1h-pyrazol-4-yl]-6-(1h-pyrazol-4-yl)-1h-indazole-3-carboxamideHuman2023
AURKA (AurA)AurOther5oroAadenosine-5'-diphosphateHuman8641
AURKA (AurA)AurOther3h10B9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHuman1988
AURKA (AurA)AurOther5ornAadenosine-5'-diphosphateHuman8649
AURKA (AurA)AurOther7ztlAAadenosine-5'-diphosphateHuman14582
AURKA (AurA)AurOther5g1xABadenosine-5'-diphosphateHuman7266
AURKA (AurA)AurOther5l8jAAadenosine-5'-diphosphateHuman6820
AURKA (AurA)AurOther2wtvDB4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2076
AURKA (AurA)AurOther4ztrA6-({4-[(z)-{(2z)-2-[(4-ethylphenyl)imino]-3-methyl-4-oxo-1,3-thiazolidin-5-ylidene}methyl]pyridin-2-yl}amino)pyridine-3-carboxylic acidHuman6817
AURKA (AurA)AurOther5orlAadenosine-5'-diphosphateHuman8642
AURKA (AurA)AurOther3cohB8-ethyl-3,10,10-trimethyl-4,5,6,8,10,12-hexahydropyrazolo[4',3':6,7]cyclohepta[1,2-b]pyrrolo[2,3-f]indol-9(1h)-oneHuman2024
AURKA (AurA)AurOther6r4aAadenosine-5'-diphosphateHuman11134
AURKA (AurA)AurOther9s14Badenosine-5'-diphosphateHuman15493
AURKA (AurA)AurOther3uo4A4-{[4-(biphenyl-2-ylamino)pyrimidin-2-yl]amino}benzoic acidHuman1976
AURKA (AurA)AurOther6cpeAB-Human10035
AURKA (AurA)AurOther3uohB4-({4-[(2-bromophenyl)amino]pyrimidin-2-yl}amino)benzoic acidHuman2000
AURKA (AurA)AurOther2np8An-{3-[(4-{[3-(trifluoromethyl)phenyl]amino}pyrimidin-2-yl)amino]phenyl}cyclopropanecarboxamideHuman2075
AURKA (AurA)AurOther2wtvCA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2017
AURKA (AurA)AurOther3h10A9-chloro-7-(2,6-difluorophenyl)-n-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-5h-pyrimido[5,4-d][2]benzazepin-2-amineHuman2009
AURKA (AurA)AurOther3uokB4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acidHuman2047
AURKA (AurA)AurOther6c2rAB(2r,4r)-1-[(3-chloro-2-fluorophenyl)methyl]-4-({3-fluoro-6-[(5-methyl-1h-pyrazol-3-yl)amino]pyridin-2-yl}methyl)-2-methylpiperidine-4-carboxylic acidHuman10865
AURKA (AurA)AurOther2xruA3-({[4-(4-methylpiperazin-1-yl)phenyl]carbonyl}amino)-n-[(1r)-1-phenylpropyl]-1h-thieno[3,2-c]pyrazole-5-carboxamideHuman1954
AURKA (AurA)AurOther9gucABadenosine-5'-diphosphateHuman15495
AURKA (AurA)AurOther3ha6An~2~-(3,4-dimethoxyphenyl)-n~4~-[2-(2-fluorophenyl)ethyl]-n~6~-quinolin-6-yl-1,3,5-triazine-2,4,6-triamineHuman2048
AURKA (AurA)AurOther6graA1-[(2~{r},3~{s})-2-[[1,3-benzodioxol-5-ylmethyl(methyl)amino]methyl]-3-methyl-6-oxidanylidene-5-[(2~{s})-1-oxidanylpropan-2-yl]-3,4-dihydro-2~{h}-1,5-benzoxazocin-8-yl]-3-(4-methoxyphenyl)ureaHuman11130
AURKA (AurA)AurOther6r4bABadenosine-5'-diphosphateHuman11133
AURKA (AurA)AurOther5dt3Aadenosine-5'-triphosphateHuman6816
AURKA (AurA)AurOther7ficAB6-[(5-cyclopropyl-1~{h}-pyrazol-3-yl)amino]-2-[4-[(3-methyl-4-oxidanyl-phenyl)methyl]piperazin-1-yl]-~{n}-prop-2-ynyl-pyrimidine-4-carboxamideHuman14233
AURKA (AurA)AurOther6cpfAphosphomethylphosphonic acid adenylate esterHuman10033
AURKA (AurA)AurOther2wqeAadenosine-5'-diphosphateHuman2071
AURKA (AurA)AurOther8c1iAAadenosine-5'-diphosphateHuman15144
AURKA (AurA)AurOther5aagA[3-[[4-[6-chloranyl-2-(1,3-dimethylpyrazol-4-yl)-3h-imidazo[4,5-b]pyridin-7-yl]pyrazol-1-yl]methyl]phenyl]-(4-methylpiperazin-1-yl)methanoneHuman6010
AURKA (AurA)AurOther6r49Aadenosine-5'-diphosphateHuman11131
AURKA (AurA)AurOther6vpmBBadenosine monophosphateHuman12663
AURKA (AurA)AurOther2bmcB(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2008
AURKA (AurA)AurOther3efwA1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHuman2010
AURKA (AurA)AurOther6cpgA1-cyclopropyl-3-{3-[5-(morpholin-4-ylmethyl)-1h-benzimidazol-2-yl]-1h-pyrazol-4-yl}ureaHuman10032
AURKA (AurA)AurOther2x81A4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman1966
AURKA (AurA)AurOther3efwB1-[3-methyl-4-({3-[2-(methylamino)pyrimidin-4-yl]pyridin-2-yl}oxy)phenyl]-3-[3-(trifluoromethyl)phenyl]ureaHuman2074
AURKA (AurA)AurOther2bmcC(3e)-n-(2,6-diethylphenyl)-3-{[4-(4-methylpiperazin-1-yl)benzoyl]imino}pyrrolo[3,4-c]pyrazole-5(3h)-carboxamideHuman2060
AURKA (AurA)AurOther6vplBAphosphoaminophosphonic acid-adenylate esterHuman12664
AURKA (AurA)AurOther5dr9A4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman6821
AURKA (AurA)AurOther4bn1ABadenosine-5'-diphosphateHuman1983
AURKA (AurA)AurOther8guwAadenosine-5'-diphosphateHuman14753
AURKA (AurA)AurOther5oseAadenosine-5'-diphosphateHuman8645
AURKA (AurA)AurOther2xngAAn-(3-{3-chloro-8-[(4-morpholin-4-ylphenyl)amino]imidazo[1,2-a]pyrazin-6-yl}benzyl)methanesulfonamideHuman1994
AURKA (AurA)AurOther3r22An-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHuman2034
AURKA (AurA)AurOther5lxmABadenosine-5'-diphosphateHuman7141
AURKA (AurA)AurOther6xkaA-Human12665
AURKA (AurA)AurOther2j4zA4-(4-methylpiperazin-1-yl)-n-[5-(2-thienylacetyl)-1,5-dihydropyrrolo[3,4-c]pyrazol-3-yl]benzamideHuman2053
AURKA (AurA)AurOther6vphAAdithiane diolHuman12666
AURKA (AurA)AurOther5obrA4-({5-amino-1-[(2,6-difluorophenyl)carbonyl]-1h-1,2,4-triazol-3-yl}amino)benzenesulfonamideHuman8304
AURKA (AurA)AurOther4o0wAadenosineHuman1959
AURKA (AurA)AurOther3r21AAn-(2-aminoethyl)-n-{5-[(1-cycloheptyl-1h-pyrazolo[3,4-d]pyrimidin-6-yl)amino]pyridin-2-yl}methanesulfonamideHuman1991
AURKA (AurA)AurOther4ztsA(2z,5z)-2-[(4-ethylphenyl)imino]-3-methyl-5-[(2-{[4-(1h-tetrazol-5-yl)phenyl]amino}pyridin-4-yl)methylidene]-1,3-thiazolidin-4-oneHuman6814
AURKA (AurA)AurOther6i2uA-Human11652
AURKA (AurA)AurOther9sq7Badenosine-5'-diphosphateHuman15498
AURKA (AurA)AurOther3h0yA2-chloro-n-[4-({5-fluoro-2-[(4-hydroxyphenyl)amino]pyrimidin-4-yl}amino)phenyl]benzamideHuman1965
AURKA (AurA)AurOther4uzhA(4s)-4-(2-fluorophenyl)-2,4,6,7,8,9-hexahydro-5h-pyrazolo[3,4-b][1,7]naphthyridin-5-oneHuman1998
AURKA (AurA)AurOther6c83Bphosphomethylphosphonic acid adenylate esterHuman10935
AURKA (AurA)AurOther6vpgABphosphoaminophosphonic acid-adenylate esterHuman12667
AURKA (AurA)AurOther8jg8A4-[5-[3-[bis(oxidanylidene)-$l^5-sulfanyl]oxyphenyl]-7h-pyrrolo[2,3-d]pyrimidin-4-yl]morpholineHuman15272
AURKA (AurA)AurOther9s61Badenosine-5'-diphosphateHuman15499
AURKA (AurA)AurOther4o0uAadenosineHuman2022
AURKA (AurA)AurOther3uokA4-({4-[(2-chlorophenyl)amino]-5-fluoropyrimidin-2-yl}amino)benzoic acidHuman2054
AURKA (AurA)AurOther2w1dA2-(1h-pyrazol-3-yl)-1h-benzimidazoleHuman2011
AURKA (AurA)AurOther2wtvDA4-{[9-chloro-7-(2,6-difluorophenyl)-5h-pyrimido[5,4-d][2]benzazepin-2-yl]amino}benzoic acidHuman2078
AURKA (AurA)AurOther9gucAAadenosine-5'-diphosphateHuman15500
AURKA (AurA)AurOther9bzgAB7-cyclopentyl-n,n-dimethyl-2-[4-(methylcarbamoyl)anilino]-7h-pyrrolo[2,3-d]pyrimidine-6-carboxamideHuman15501
AURKA (AurA)AurOther2c6dAAphosphoaminophosphonic acid-adenylate esterHuman2019
AURKA (AurA)AurOther4bn1AAadenosine-5'-diphosphateHuman1955
AURKA (AurA)AurOther6vplABphosphoaminophosphonic acid-adenylate esterHuman12670
Aurka (AurA)AUROther3d2kA(7-{[2-(2-{[(3-chlorophenyl)carbamoyl]amino}-1,3-thiazol-5-yl)ethyl]amino}-1h-pyrazolo[4,3-d]pyrimidin-1-yl)acetic acidMouse5776
Aurka (AurA)AUROther3dajAn-butyl-3-{[6-(9h-purin-6-ylamino)hexanoyl]amino}benzamideMouse5779
Aurka (AurA)AUROther3dj5A3-({3-[(6-amino-5-bromopyrimidin-4-yl)sulfanyl]propanoyl}amino)-4-methoxy-n-phenylbenzamideMouse5783
Aurka (AurA)AUROther3d2iA1-(5-{2-[(1-methyl-1h-pyrazolo[4,3-d]pyrimidin-7-yl)amino]ethyl}-1,3-thiazol-2-yl)-3-[3-(trifluoromethyl)phenyl]ureaMouse5782
Aurka (AurA)AUROther3d15AA1-(3-chlorophenyl)-3-{5-[2-(thieno[3,2-d]pyrimidin-4-ylamino)ethyl]-1,3-thiazol-2-yl}ureaMouse5777
Aurka (AurA)AUROther3dj6A4-methoxy-n-phenyl-3-({3-[(1h-pyrrolo[2,3-b]pyridin-5-ylmethyl)sulfanyl]propanoyl}amino)benzamideMouse5778