Search results (19 entries covering 10 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
CDK5CDKCMGC4au8AB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2786
CDK5CDKCMGC1h4lA-Human2788
CDK5CDKCMGC7vdrA(1r)-1-[7-[(2-fluoranyl-4-pyrazol-1-yl-phenyl)amino]-1,6-naphthyridin-2-yl]-1-(1-methylpiperidin-4-yl)ethanolHuman14146
CDK5CDKCMGC7vdqA2-[[7-[[2-fluoranyl-4-[3-(hydroxymethyl)pyrazol-1-yl]phenyl]amino]-1,6-naphthyridin-2-yl]-(1-methylpiperidin-4-yl)amino]ethanoic acidHuman14144
CDK5CDKCMGC7vdsAA5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHuman14148
CDK5CDKCMGC1unhA(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2780
CDK5CDKCMGC3o0gA-Human2782
CDK5CDKCMGC1unlB-Human2790
CDK5CDKCMGC1unhB(z)-1h,1'h-[2,3']biindolylidene-3,2'-dione-3-oximeHuman2787
CDK5CDKCMGC3o0gB{4-amino-2-[(4-chlorophenyl)amino]-1,3-thiazol-5-yl}(3-nitrophenyl)methanoneHuman2783
CDK5CDKCMGC7vdsAB5-fluoranyl-4-[[2-[(1r)-1-(1-methylpiperidin-4-yl)-1-oxidanyl-ethyl]-1,6-naphthyridin-7-yl]amino]-2-morpholin-4-yl-benzenecarbonitrileHuman14147
CDK5CDKCMGC1ungB6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2789
CDK5CDKCMGC1ungA6-phenyl[5h]pyrrolo[2,3-b]pyrazineHuman2792
CDK5CDKCMGC1h4lB-Human2779
CDK5CDKCMGC4au8BB4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2781
CDK5CDKCMGC7vdpA[1-[3-fluoranyl-4-[(2-piperidin-4-yloxy-1,6-naphthyridin-7-yl)amino]phenyl]pyrazol-3-yl]methanolHuman14145
CDK5CDKCMGC4au8AA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2784
CDK5CDKCMGC1unlAr-roscovitineHuman2785
CDK5CDKCMGC4au8BA4-(1,3-benzothiazol-2-yl)thiophene-2-sulfonamideHuman2791