Search results (19 entries covering 12 PDB structures)
| # | Kinase | Family | Group | PDB | Chain | (Alternate) Model | Orthosteric ligand | Organism | Details | File |
|---|---|---|---|---|---|---|---|---|---|---|
| CDK7 | CDK | CMGC | 8p4z | A | A | 2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine | Human | 14796 | ||
| CDK7 | CDK | CMGC | 8p4z | A | B | 2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amine | Human | 14797 | ||
| CDK7 | CDK | CMGC | 8pyr | A | B | - | Human | 15253 | ||
| CDK7 | CDK | CMGC | 1ua2 | C | adenosine-5'-triphosphate | Human | 542 | |||
| CDK7 | CDK | CMGC | 7b5o | J | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13278 | ||
| CDK7 | CDK | CMGC | 7nvr | 8 | - | Human | 13543 | |||
| CDK7 | CDK | CMGC | 7b5q | J | A | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13277 | ||
| CDK7 | CDK | CMGC | 1ua2 | D | adenosine-5'-triphosphate | Human | 543 | |||
| CDK7 | CDK | CMGC | 6xd3 | J | n-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamide | Human | 12772 | |||
| CDK7 | CDK | CMGC | 8byq | I | - | Human | 14732 | |||
| CDK7 | CDK | CMGC | 6o9l | 8 | - | Human | 11055 | |||
| CDK7 | CDK | CMGC | 8pyr | A | A | - | Human | 15254 | ||
| CDK7 | CDK | CMGC | 6xbz | J | phosphothiophosphoric acid-adenylate ester | Human | 12773 | |||
| CDK7 | CDK | CMGC | 1ua2 | B | adenosine-5'-triphosphate | Human | 541 | |||
| CDK7 | CDK | CMGC | 1ua2 | A | adenosine-5'-triphosphate | Human | 540 | |||
| CDK7 | CDK | CMGC | 29wd | I | - | Human | 16031 | |||
| CDK7 | CDK | CMGC | 8bvw | I | - | Human | 14733 | |||
| CDK7 | CDK | CMGC | 7b5o | J | B | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13279 | ||
| CDK7 | CDK | CMGC | 7b5q | J | B | (3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-ol | Human | 13280 |