Search results (19 entries covering 12 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
CDK7CDKCMGC8p4zAA2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHuman14796
CDK7CDKCMGC8p4zAB2-[(3r)-piperidin-3-yl]oxy-8-propan-2-yl-n-[(2-pyrazol-1-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazin-4-amineHuman14797
CDK7CDKCMGC8pyrAB-Human15253
CDK7CDKCMGC1ua2Cadenosine-5'-triphosphateHuman542
CDK7CDKCMGC7b5oJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13278
CDK7CDKCMGC7nvr8-Human13543
CDK7CDKCMGC7b5qJA(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13277
CDK7CDKCMGC1ua2Dadenosine-5'-triphosphateHuman543
CDK7CDKCMGC6xd3Jn-(3-{[5-chloro-4-(1h-indol-3-yl)pyrimidin-2-yl]amino}phenyl)-4-{[4-(dimethylamino)butanoyl]amino}benzamideHuman12772
CDK7CDKCMGC8byqI-Human14732
CDK7CDKCMGC6o9l8-Human11055
CDK7CDKCMGC8pyrAA-Human15254
CDK7CDKCMGC6xbzJphosphothiophosphoric acid-adenylate esterHuman12773
CDK7CDKCMGC1ua2Badenosine-5'-triphosphateHuman541
CDK7CDKCMGC1ua2Aadenosine-5'-triphosphateHuman540
CDK7CDKCMGC29wdI-Human16031
CDK7CDKCMGC8bvwI-Human14733
CDK7CDKCMGC7b5oJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13279
CDK7CDKCMGC7b5qJB(3r,4r)-4-[[[7-[(phenylmethyl)amino]-3-propan-2-yl-pyrazolo[1,5-a]pyrimidin-5-yl]amino]methyl]piperidin-3-olHuman13280