Search results (26 entries covering 7 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
DAPK3DAPKCAMK5vjaCA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10345
DAPK3DAPKCAMK2j90AB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman382
DAPK3DAPKCAMK3bqrAB4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acidHuman386
DAPK3DAPKCAMK5a6nBB-Human6161
DAPK3DAPKCAMK1yrpA-Human384
DAPK3DAPKCAMK5a6oBB-Human6166
DAPK3DAPKCAMK5a6nAA5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ideHuman6164
DAPK3DAPKCAMK5vjaCB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10352
DAPK3DAPKCAMK2j90AA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman387
DAPK3DAPKCAMK5a6nBA-Human6162
DAPK3DAPKCAMK5vjaBA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10346
DAPK3DAPKCAMK5vjaAA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10351
DAPK3DAPKCAMK5vjaDB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10347
DAPK3DAPKCAMK3bqrAA4-(6-{[(1r)-1-(hydroxymethyl)propyl]amino}imidazo[1,2-b]pyridazin-3-yl)benzoic acidHuman380
DAPK3DAPKCAMK2j90BA2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman378
DAPK3DAPKCAMK2j90BB2-tert-butyl-9-fluoro-3,6-dihydro-7h-benz[h]-imidaz[4,5-f]isoquinoline-7-oneHuman379
DAPK3DAPKCAMK5vjaBB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10350
DAPK3DAPKCAMK5a6oAB-Human6163
DAPK3DAPKCAMK5a6nAB5-(3-sulfamoylphenyl)-1h-1,2,3,4-tetrazol-1-ideHuman6165
DAPK3DAPKCAMK3bhyAA(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman385
DAPK3DAPKCAMK5vjaAB(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10349
DAPK3DAPKCAMK3bhyAB(4r)-7,8-dichloro-1',9-dimethyl-1-oxo-1,2,4,9-tetrahydrospiro[beta-carboline-3,4'-piperidine]-4-carbonitrileHuman381
DAPK3DAPKCAMK5vjaDA(2r)-2-{[1-(3-chlorophenyl)-4-oxo-4,5-dihydro-1h-pyrazolo[3,4-d]pyrimidin-6-yl]sulfanyl}propanamideHuman10348
DAPK3DAPKCAMK5a6oBA-Human6168
DAPK3DAPKCAMK1yrpB-Human383
DAPK3DAPKCAMK5a6oAA-Human6167