Search results (42 entries covering 26 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
DYRK2DYRKCMGC5lxdBAmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7123
DYRK2DYRKCMGC6hdrAAcurcuminHuman11570
DYRK2DYRKCMGC5lxcBAmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7125
DYRK2DYRKCMGC3kvwAB(2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acidHuman3149
DYRK2DYRKCMGC7dh3A2,7-dimethoxy-9-piperidin-4-ylsulfanyl-acridineHuman13978
DYRK2DYRKCMGC5ztnB(1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneHuman10483
DYRK2DYRKCMGC7ejvBB[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14182
DYRK2DYRKCMGC7ejvBA[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14183
DYRK2DYRKCMGC7dhkA2-methoxy-7-phenylmethoxy-9-(piperidin-4-ylmethylsulfanyl)acridineHuman13977
DYRK2DYRKCMGC7akhA4-[3-[(2~{s})-2-(6-bromanylpyridin-2-yl)oxypropyl]-2-methyl-imidazo[4,5-b]pyridin-5-yl]pyridine-2,6-diamineHuman13615
DYRK2DYRKCMGC6hdpABscorzodihydrostilbene aHuman11573
DYRK2DYRKCMGC7dhvA2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridine-4-carboxylic acidHuman13974
DYRK2DYRKCMGC7dhhA[9-(azetidin-3-ylmethylsulfanyl)-2,7-dimethoxy-acridin-4-yl]methanolHuman13975
DYRK2DYRKCMGC9kqyA-Human16123
DYRK2DYRKCMGC9mc0A[2-[[4-(1,3-benzothiazol-5-yl)-5-fluoranyl-pyrimidin-2-yl]amino]-1,3-thiazol-5-yl]-piperazin-1-yl-methanoneHuman16124
DYRK2DYRKCMGC7dh9A[2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridin-4-yl]methanolHuman13976
DYRK2DYRKCMGC5ztnA(1z,4z,6e)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-oneHuman10482
DYRK2DYRKCMGC7dhnA7-methoxy-2-methylsulfanyl-9-(piperidin-4-ylmethylsulfanyl)-[1,3]thiazolo[5,4-b]quinolineHuman13971
DYRK2DYRKCMGC5lxdABmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7128
DYRK2DYRKCMGC4azfAB5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3146
DYRK2DYRKCMGC3k2lAB-Human3145
DYRK2DYRKCMGC3k2lAA-Human3147
DYRK2DYRKCMGC7dhoA2-methoxy-9-(piperidin-4-ylmethylsulfanyl)-7-propan-2-yloxy-acridineHuman13972
DYRK2DYRKCMGC7ejvAB[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14181
DYRK2DYRKCMGC7ejvAA[6-[[4-[2-(dimethylamino)-1,3-benzothiazol-6-yl]-5-fluoranyl-pyrimidin-2-yl]amino]pyridin-3-yl]-(4-ethylpiperazin-1-yl)methanoneHuman14180
DYRK2DYRKCMGC4azfAA5-(1,3-benzodioxol-5-ylmethyl)-2-(phenylamino)-4h-imidazol-4-oneHuman3144
DYRK2DYRKCMGC7dg4A2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridineHuman13967
DYRK2DYRKCMGC6hdrABcurcuminHuman11571
DYRK2DYRKCMGC5lxdAAmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7124
DYRK2DYRKCMGC7akfAB4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13614
DYRK2DYRKCMGC5lxcAAmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7122
DYRK2DYRKCMGC7akfAA4-(2,3-dimethyl-1-benzofuran-5-yl)pyridine-2,6-diamineHuman13613
DYRK2DYRKCMGC5lxcABmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7129
DYRK2DYRKCMGC6k0jA3-(2,7-dimethoxyacridin-9-yl)sulfanylpropan-1-amineHuman11817
DYRK2DYRKCMGC8hltA(6-{[(4p)-4-(1,3-benzothiazol-5-yl)-5-fluoropyrimidin-2-yl]amino}pyridin-3-yl)(piperazin-1-yl)methanoneHuman15091
DYRK2DYRKCMGC5lxcBBmethyl 9-[(2,4-dichlorophenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7126
DYRK2DYRKCMGC7dl6A[2,7-dimethoxy-9-[[(3r)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanolHuman14013
DYRK2DYRKCMGC5lxdBBmethyl 9-[(2-fluoranyl-4-methoxy-phenyl)amino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateHuman7127
DYRK2DYRKCMGC7dhcA4-[bis(fluoranyl)methyl]-2,7-dimethoxy-9-(piperidin-4-ylmethylsulfanyl)acridineHuman13973
DYRK2DYRKCMGC7djoA[2,7-dimethoxy-9-[[(3s)-pyrrolidin-3-yl]methylsulfanyl]acridin-4-yl]methanolHuman13994
DYRK2DYRKCMGC6hdpAAscorzodihydrostilbene aHuman11572
DYRK2DYRKCMGC3kvwAA(2z,3e)-7'-bromo-3-(hydroxyimino)-2'-oxo-1,1',2',3-tetrahydro-2,3'-biindole-5-carboxylic acidHuman3148