Search results (18 entries covering 4 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
MAPK6 (Erk3)MAPKCMGC6ylcC5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12794
MAPK6 (Erk3)MAPKCMGC6ylcA5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12791
MAPK6 (Erk3)MAPKCMGC6ykyBA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12792
MAPK6 (Erk3)MAPKCMGC6yllA~{n}4-[3-(4-methoxyphenyl)-[1,2,3]triazolo[4,5-d]pyrimidin-5-yl]cyclohexane-1,4-diamineHuman12793
MAPK6 (Erk3)MAPKCMGC7aqbAA-Human12982
MAPK6 (Erk3)MAPKCMGC6ylcD5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12795
MAPK6 (Erk3)MAPKCMGC7aqbBB-Human12983
MAPK6 (Erk3)MAPKCMGC6ykyDA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12796
MAPK6 (Erk3)MAPKCMGC6ylcB5-fluoranyl-2-[5-[[1-(1-methylpiperidin-4-yl)pyrazol-4-yl]amino]-[1,2,3]triazolo[4,5-d]pyrimidin-3-yl]benzenecarbonitrileHuman12797
MAPK6 (Erk3)MAPKCMGC6ykyCB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12784
MAPK6 (Erk3)MAPKCMGC6yllB-Human12785
MAPK6 (Erk3)MAPKCMGC6ykyBB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12786
MAPK6 (Erk3)MAPKCMGC6ykyCA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12787
MAPK6 (Erk3)MAPKCMGC6ykyAA3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12788
MAPK6 (Erk3)MAPKCMGC6ykyDB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12789
MAPK6 (Erk3)MAPKCMGC6ykyAB3-(4-methoxyphenyl)-~{n}-[(3~{r})-1-pyridin-4-ylpyrrolidin-3-yl]-[1,2,3]triazolo[4,5-d]pyrimidin-5-amineHuman12790
MAPK6 (Erk3)MAPKCMGC7aqbBA-Human12980
MAPK6 (Erk3)MAPKCMGC7aqbAB-Human12981