Search results (22 entries covering 13 PDB structures)

#KinaseFamilyGroupPDBChain(Alternate) Model Orthosteric ligandOrganismDetails File
MAPK7 (Erk5)MAPKCMGC5byyAA2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman6591
MAPK7 (Erk5)MAPKCMGC5o7iAA4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamideHuman9995
MAPK7 (Erk5)MAPKCMGC7pusAB4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamideHuman14219
MAPK7 (Erk5)MAPKCMGC9ltaA4-[5-chloranyl-2-[[3-[(dimethylamino)methyl]phenyl]amino]pyrimidin-4-yl]-~{n}-morpholin-4-yl-thiophene-2-carboxamideHuman15439
MAPK7 (Erk5)MAPKCMGC7pusAA4-[3,6-bis(chloranyl)-2-fluoranyl-phenyl]carbonyl-~{n}-(1-methylpyrazol-4-yl)-1~{h}-pyrrole-2-carboxamideHuman14218
MAPK7 (Erk5)MAPKCMGC6hknAA[2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanoneHuman10918
MAPK7 (Erk5)MAPKCMGC4ic7Dphosphoaminophosphonic acid-adenylate esterHuman391
MAPK7 (Erk5)MAPKCMGC6hknAB[2-azanyl-4-(trifluoromethyloxy)phenyl]-[4-(7-methoxyquinazolin-4-yl)piperidin-1-yl]methanoneHuman10919
MAPK7 (Erk5)MAPKCMGC4zsjAB3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6585
MAPK7 (Erk5)MAPKCMGC4ic7Aphosphoaminophosphonic acid-adenylate esterHuman392
MAPK7 (Erk5)MAPKCMGC5o7iAB4-(2-bromanyl-6-fluoranyl-phenyl)carbonyl-~{n}-pyridin-3-yl-1~{h}-pyrrole-2-carboxamideHuman9994
MAPK7 (Erk5)MAPKCMGC5byyAB2-{[2-ethoxy-4-(4-hydroxypiperidin-1-yl)phenyl]amino}-5,11-dimethyl-5,11-dihydro-6h-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman6587
MAPK7 (Erk5)MAPKCMGC4zslA3-amino-5-[(4-chlorophenyl)amino]-n-[(1s)-1-phenylethyl]-1h-1,2,4-triazole-1-carboxamideHuman6586
MAPK7 (Erk5)MAPKCMGC4zsgAB3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6584
MAPK7 (Erk5)MAPKCMGC6hkmA[4-(6,7-dimethoxyquinazolin-4-yl)piperidin-1-yl]-[4-(trifluoromethyloxy)phenyl]methanoneHuman10917
MAPK7 (Erk5)MAPKCMGC4b99A11-cyclopentyl-2-[[2-methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]carbonyl-phenyl]amino]-5-methyl-pyrimido[4,5-b][1,4]benzodiazepin-6-oneHuman388
MAPK7 (Erk5)MAPKCMGC5byzAB4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamideHuman6592
MAPK7 (Erk5)MAPKCMGC4zsgAA3-amino-5-[(4-chlorophenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6589
MAPK7 (Erk5)MAPKCMGC5byzAA4-({5-fluoro-4-[2-methyl-1-(propan-2-yl)-1h-imidazol-5-yl]pyrimidin-2-yl}amino)-n-[2-(piperidin-1-yl)ethyl]benzamideHuman6590
MAPK7 (Erk5)MAPKCMGC4zsjAA3-amino-5-[(4-chloro-3-methylphenyl)amino]-n-(propan-2-yl)-1h-1,2,4-triazole-1-carboxamideHuman6588
MAPK7 (Erk5)MAPKCMGC4ic8B-Human389
MAPK7 (Erk5)MAPKCMGC4ic8A-Human390